AR123228A1 - Formas en estado sólido de un compuesto orgánico - Google Patents
Formas en estado sólido de un compuesto orgánicoInfo
- Publication number
- AR123228A1 AR123228A1 ARP210102263A ARP210102263A AR123228A1 AR 123228 A1 AR123228 A1 AR 123228A1 AR P210102263 A ARP210102263 A AR P210102263A AR P210102263 A ARP210102263 A AR P210102263A AR 123228 A1 AR123228 A1 AR 123228A1
- Authority
- AR
- Argentina
- Prior art keywords
- solid state
- state forms
- organic compound
- conditions
- forms
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1635—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Abstract
En el presente documento se proporcionan varias formas en estado sólido, que incluyen sales, así como varias formas cristalinas y amorfas, del Compuesto I, que está representado por la fórmula estructural: de fórmula (1). También se proporcionan composiciones farmacéuticas que comprenden estos materiales, métodos para su fabricación, usos de los mismos para tratar afecciones, incluidas, entre otras, afecciones que se beneficiarían de la inhibición de la metionina adenosiltransferasa 2a (MAT2A).
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US202063064866P | 2020-08-12 | 2020-08-12 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR123228A1 true AR123228A1 (es) | 2022-11-09 |
Family
ID=77693586
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP210102263A AR123228A1 (es) | 2020-08-12 | 2021-08-12 | Formas en estado sólido de un compuesto orgánico |
Country Status (3)
Country | Link |
---|---|
AR (1) | AR123228A1 (es) |
TW (1) | TW202227446A (es) |
WO (1) | WO2022036033A2 (es) |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE69637441T2 (de) * | 1995-10-17 | 2009-03-05 | Jagotec Ag | Verabreichung unlöslicher arzneistoffe |
PL3116491T3 (pl) | 2014-03-14 | 2022-02-07 | Les Laboratoires Servier | Kompozycje farmaceutyczne związków terapeutycznie aktywnych |
AU2017319500C1 (en) | 2016-08-31 | 2022-10-20 | Les Laboratoires Servier | Inhibitors of cellular metabolic processes |
WO2018039972A1 (en) * | 2016-08-31 | 2018-03-08 | Agios Pharmaceuticals, Inc. | Inhibitors of cellular metabolic processes |
KR20200095480A (ko) | 2017-11-02 | 2020-08-10 | 아지오스 파마슈티컬스 아이엔씨. | 공결정, 그의 제약 조성물, 및 그를 포함하는 치료 방법 |
-
2021
- 2021-08-12 WO PCT/US2021/045656 patent/WO2022036033A2/en active Application Filing
- 2021-08-12 AR ARP210102263A patent/AR123228A1/es unknown
- 2021-08-12 TW TW110129859A patent/TW202227446A/zh unknown
Also Published As
Publication number | Publication date |
---|---|
WO2022036033A4 (en) | 2022-06-23 |
WO2022036033A3 (en) | 2022-04-21 |
WO2022036033A2 (en) | 2022-02-17 |
TW202227446A (zh) | 2022-07-16 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
UY38076A (es) | Derivados de tetrahidroquinazolina útiles como agentes anticáncer | |
PE20191474A1 (es) | Compuestos de amino-triazolopiridina y su uso en el tratamiento del cancer | |
DOP2021000234A (es) | Pirroles triciclicos condensados como moduladores de alfa-1 antitripsina | |
CL2019000986A1 (es) | 1,3 di sustituto ciclobutano o derivados de azetidina como inhibidores de prostaglandina d sintasa hematopoyética(h-pgds). | |
ECSP20033467A (es) | Compuestos macrocíclicos para tratar enfermedades | |
CO6341623A2 (es) | Compuestos organicos | |
CO2019000932A2 (es) | Nuevos compuestos sulfonimidoilpurinona 7-sustituidos y derivados para el tratamiento y la profilaxis de la infección vírica. | |
CU20190101A7 (es) | Imidazopirimidinas diazabicíclicas sustituidas | |
UY37774A (es) | Compuestos 5-cianoindol sustituidos y usos de los mismos | |
CL2021000844A1 (es) | Compuestos de indolinona para uso como inhibidores de map4k1 | |
DOP2016000308A (es) | Compuestos de 1, 3, 4-tiadiazol y uso de los mismos para el tratamiento del cáncer | |
UY37378A (es) | Compuestos tricíclicos fusionados de piridazinona útiles para tratar infecciones de orthomyxovirus | |
CL2017002745A1 (es) | Nuevos compuestos y derivados de sulfonimidoilpurinona para el tratamiento y profilaxis de infecciones víricas | |
PE20171348A1 (es) | Compuestos de benzoxaborol 4-sustituidos y uso de los mismos | |
CO2022010547A2 (es) | Compuestos y usos de los mismos | |
CL2017000827A1 (es) | Inhibidores de aldosterona sintasa | |
CL2021002946A1 (es) | Un derivado de tetrahidroisoquinolina sustituido como modulador alostérico positivo de d1 | |
DOP2020000100A (es) | Novedosos derivados de pirazolo-pirrolo-pirimidina como inhibidores de p2x3 | |
CL2023002633A1 (es) | Derivados de uracilo como inhibidores de trpa1 | |
AR121483A1 (es) | Hidrato cristalino de un compuesto inhibidor de jak | |
AR117844A1 (es) | Derivados de tiazolopiridina como antagonistas del receptor de adenosina | |
AR127470A1 (es) | Inhibidores de lrrk2 | |
CL2021001640A1 (es) | Formas de sal y cristalinas de un compuesto orgánico y composiciones farmacéuticas del mismo | |
CL2020003248A1 (es) | Derivados de tetrahidrotienopiridina n-sustituidos y sus usos | |
AR123228A1 (es) | Formas en estado sólido de un compuesto orgánico |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FB | Suspension of granting procedure |