AR114134A2 - Sal de maleato de 11-(2-pirrolidin-1-il-etoxi)-14,19-dioxa-5,7,26-triaza-tetraciclo[19.3.1.1(2,6).1(8,12)]heptacosa-1(25),2(26),3,5,8,10,12(27),16,21,23-decaeno - Google Patents
Sal de maleato de 11-(2-pirrolidin-1-il-etoxi)-14,19-dioxa-5,7,26-triaza-tetraciclo[19.3.1.1(2,6).1(8,12)]heptacosa-1(25),2(26),3,5,8,10,12(27),16,21,23-decaenoInfo
- Publication number
- AR114134A2 AR114134A2 ARP190100702A ARP190100702A AR114134A2 AR 114134 A2 AR114134 A2 AR 114134A2 AR P190100702 A ARP190100702 A AR P190100702A AR P190100702 A ARP190100702 A AR P190100702A AR 114134 A2 AR114134 A2 AR 114134A2
- Authority
- AR
- Argentina
- Prior art keywords
- heptacose
- triaza
- dioxa
- pyrrolidin
- tetraciclo
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Sales maleato de 11-(2-pirrolidin-1-il-etoxi)-14,19-dioxa-5,7,26-triaza-tetraciclo[19.3.1.1(2,6),1(8,12)]heptacosa-1(25),2(26),3,5,8,10,12(27),16,21,23-decaeno (Compuesto I), de fórmula (1), del cual se descubrió que tiene propiedades mejoradas. También composiciones farmacéuticas que contienen esta sal.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US12167608P | 2008-12-11 | 2008-12-11 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR114134A2 true AR114134A2 (es) | 2020-07-22 |
Family
ID=42103945
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP090104835A AR074725A1 (es) | 2008-12-11 | 2009-12-11 | Sal de maleato de 11-(2-pirrolidin-1-il-etoxi)-14,19- dioxa-5,7,26-triaza-tetraciclo(19.3.1.1 (2,6).1 (8,12) heptacosa-1(25),2 (26),3,5,8,10,12 (27),16,21,23-decaeno |
ARP190100702A AR114134A2 (es) | 2008-12-11 | 2019-03-20 | Sal de maleato de 11-(2-pirrolidin-1-il-etoxi)-14,19-dioxa-5,7,26-triaza-tetraciclo[19.3.1.1(2,6).1(8,12)]heptacosa-1(25),2(26),3,5,8,10,12(27),16,21,23-decaeno |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP090104835A AR074725A1 (es) | 2008-12-11 | 2009-12-11 | Sal de maleato de 11-(2-pirrolidin-1-il-etoxi)-14,19- dioxa-5,7,26-triaza-tetraciclo(19.3.1.1 (2,6).1 (8,12) heptacosa-1(25),2 (26),3,5,8,10,12 (27),16,21,23-decaeno |
Country Status (10)
Country | Link |
---|---|
US (1) | US8987243B2 (es) |
EP (1) | EP2376500B1 (es) |
AR (2) | AR074725A1 (es) |
DK (1) | DK2376500T3 (es) |
ES (1) | ES2536276T3 (es) |
HR (1) | HRP20150413T8 (es) |
PL (1) | PL2376500T3 (es) |
PT (1) | PT2376500E (es) |
TW (1) | TWI457342B (es) |
WO (1) | WO2010068182A1 (es) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN103626742B (zh) | 2005-11-01 | 2017-04-26 | 塔格根公司 | 激酶的联-芳基间-嘧啶抑制剂 |
US8604042B2 (en) | 2005-11-01 | 2013-12-10 | Targegen, Inc. | Bi-aryl meta-pyrimidine inhibitors of kinases |
US8133900B2 (en) | 2005-11-01 | 2012-03-13 | Targegen, Inc. | Use of bi-aryl meta-pyrimidine inhibitors of kinases |
WO2012060847A1 (en) | 2010-11-07 | 2012-05-10 | Targegen, Inc. | Compositions and methods for treating myelofibrosis |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR20080090390A (ko) * | 2005-11-16 | 2008-10-08 | 에스*바이오 피티이 리미티드 | 헤테로알킬이 결합된 피리미딘 유도체 |
ES2536558T3 (es) * | 2008-12-11 | 2015-05-26 | Cti Biopharma Corp. | Sal citrato de 11-(2-pirrolidin-1-il-etoxi)-14,19-dioxa-5,7,26-triaza-tetraciclo[19.3.1.1(2,6).1(8,12)]heptacosa-1(25),2(26),3,5,8,10,12(27),16,21,23-deceno |
-
2009
- 2009-12-09 DK DK09793626T patent/DK2376500T3/en active
- 2009-12-09 PT PT97936264T patent/PT2376500E/pt unknown
- 2009-12-09 US US13/133,288 patent/US8987243B2/en active Active
- 2009-12-09 PL PL09793626T patent/PL2376500T3/pl unknown
- 2009-12-09 EP EP09793626.4A patent/EP2376500B1/en active Active
- 2009-12-09 ES ES09793626.4T patent/ES2536276T3/es active Active
- 2009-12-09 WO PCT/SG2009/000474 patent/WO2010068182A1/en active Application Filing
- 2009-12-11 TW TW098142603A patent/TWI457342B/zh active
- 2009-12-11 AR ARP090104835A patent/AR074725A1/es not_active Application Discontinuation
-
2015
- 2015-04-13 HR HRP20150413TT patent/HRP20150413T8/hr unknown
-
2019
- 2019-03-20 AR ARP190100702A patent/AR114134A2/es unknown
Also Published As
Publication number | Publication date |
---|---|
HRP20150413T1 (hr) | 2015-07-03 |
US20110263616A1 (en) | 2011-10-27 |
PL2376500T3 (pl) | 2015-07-31 |
US8987243B2 (en) | 2015-03-24 |
PT2376500E (pt) | 2015-06-02 |
ES2536276T3 (es) | 2015-05-22 |
AR074725A1 (es) | 2011-02-09 |
EP2376500B1 (en) | 2015-02-25 |
HRP20150413T8 (en) | 2015-08-14 |
TW201028425A (en) | 2010-08-01 |
TWI457342B (zh) | 2014-10-21 |
EP2376500A1 (en) | 2011-10-19 |
DK2376500T3 (en) | 2015-05-04 |
WO2010068182A1 (en) | 2010-06-17 |
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