AR102995A1 - Uso de ligandos del receptor sigma en la osteoartritis - Google Patents
Uso de ligandos del receptor sigma en la osteoartritisInfo
- Publication number
- AR102995A1 AR102995A1 ARP150104064A ARP150104064A AR102995A1 AR 102995 A1 AR102995 A1 AR 102995A1 AR P150104064 A ARP150104064 A AR P150104064A AR P150104064 A ARP150104064 A AR P150104064A AR 102995 A1 AR102995 A1 AR 102995A1
- Authority
- AR
- Argentina
- Prior art keywords
- osteoartritis
- sigma receiver
- ligands
- sigma
- receiver ligands
- Prior art date
Links
- 239000003446 ligand Substances 0.000 title 1
- 201000008482 osteoarthritis Diseases 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 1
- 230000000144 pharmacologic effect Effects 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 108010085082 sigma receptors Proteins 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente se refiere a compuestos de fórmula (1) o fórmula (2) con actividad farmacológica contra el receptor sigma, para su uso en el tratamiento o la prevención de la osteoartritis y el dolor debido a la osteoartritis.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP14382519 | 2014-12-15 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR102995A1 true AR102995A1 (es) | 2017-04-05 |
Family
ID=52146389
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP150104064A AR102995A1 (es) | 2014-12-15 | 2015-12-14 | Uso de ligandos del receptor sigma en la osteoartritis |
Country Status (1)
Country | Link |
---|---|
AR (1) | AR102995A1 (es) |
-
2015
- 2015-12-14 AR ARP150104064A patent/AR102995A1/es unknown
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FB | Suspension of granting procedure |