AR100619A1 - PHARMACEUTICAL COMPOSITION THAT COMBINES 3-QUINASA D PHOSFOINOSITE INHIBITORS AND CORTICOESTEROIDS FOR THE TREATMENT OF IMMUNOAMPOLOUS CUTANEOUS DISEASES - Google Patents

PHARMACEUTICAL COMPOSITION THAT COMBINES 3-QUINASA D PHOSFOINOSITE INHIBITORS AND CORTICOESTEROIDS FOR THE TREATMENT OF IMMUNOAMPOLOUS CUTANEOUS DISEASES

Info

Publication number
AR100619A1
AR100619A1 ARP150101655A ARP150101655A AR100619A1 AR 100619 A1 AR100619 A1 AR 100619A1 AR P150101655 A ARP150101655 A AR P150101655A AR P150101655 A ARP150101655 A AR P150101655A AR 100619 A1 AR100619 A1 AR 100619A1
Authority
AR
Argentina
Prior art keywords
hydrocortisone
propionate
dexamethasone
compound
treatment
Prior art date
Application number
ARP150101655A
Other languages
Spanish (es)
Inventor
Balague Pelaez Cristina
Godessart Marina Nuria
Original Assignee
Almirall Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Almirall Sa filed Critical Almirall Sa
Publication of AR100619A1 publication Critical patent/AR100619A1/en

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Composición farmacéutica que comprende (a) un compuesto que es un inhibidor de la fosfoinosítido 3-quinasa d o una sal farmacéuticamente aceptable y/o un solvato de los mismos, y (b) un corticosteroide. Reivindicación 2: La composición según la reivindicación 1, en donde el compuesto se selecciona de LAS191954, idelalisib, duvelisib, enzastaurina, rigosertib, buparlisib, taselisib, dactolisib, copanlisib, pictrelisib, apitolisib, sonolisib, voxtalisib, ZSTK-474, GSK-2269557, UCB-5857, RV-1729, RP-6530, omipalisib, SB-2343, WX-037, CAL-120, PWT-33597, CUDC-907, AMG-319, puquitinib, pilaralisib, RP-5264, GDC-0084 o GDC-7666), LY-3023414, PQR-309, DS-7423, XL-499, KAR-4141, RP-5090, PWT-143, IPI-443, RP-6503, ONO-146040, SPR-965, LOR-220, SF-2626, X-339, X-480, PQR-401, INCB-050465, LS-008, CLR-457, PCN-5603, 7-hidroxi-estaurosporina, PF-04691502, TG-100115, BGT-226, SF-1126, PKI-179, panulisib, o una sal farmacéuticamente aceptable y/o un solvato de los mismos. Reivindicación 3: La composición según una cualquiera de las reivindicaciones 1 y 2, en donde el corticoesteroide es uno seleccionado de prednisolona, metilprednisolona, dexametasona, cipecilato de dexametasona, naflocort, deflazacort, acetato de halopredona, budesonida, dipropionato de beclometasona, hidrocortisona, acetonido de triamcinolona, acetonido de fluocinolona, fluocinonida, pivalato de clocortolona, aceponato de metilprednisolona, palmitoato de dexametasona, tipredano, aceponato de hidrocortisona, prednicarbato, dipropionato de alclometasona, halometasona, suleptanato de metilprednisolona, furoato de mometasona, rimexolona, farnesilato de prednisolona, ciclesonida, propionato de butixocort, propionato de deprodona, propionato de fluticasona, propionato de halobetasol, etabonato de loteprednol, butirato-propionato de betametasona, flunisolida, prednisona, fosfato de dexametasona y sodio, triamcinolona, 17-valerato de betametasona, betametasona, dipropionato de betametasona, acetato de hidrocortisona, succinato de hidrocortisona y sodio, fosfato de prednisolona y sodio y probutato de hidrocortisona. Reivindicación 6: Una composición de acuerdo con una cualquiera de las reivindicaciones 1 a 4 para uso en el tratamiento de una enfermedad cutánea. Reivindicación 11: Un compuesto que es un inhibidor de la fosfoinositido 3-quinasa d o una sal y/o un solvato de los mismos farmacéuticamente aceptable tal como se define en la reivindicación 1 ó 2 para uso en el tratamiento del cuerpo humano o animal, por administración simultanea, concurrente, separada o secuencial en combinación con un corticosteroide tal como se define en la reivindicación 1 ó 3 y, opcionalmente, al menos otro compuesto activo, tal como se define en la reivindicación 4.Pharmaceutical composition comprising (a) a compound that is a phosphoinositide 3-kinase d inhibitor or a pharmaceutically acceptable salt and / or a solvate thereof, and (b) a corticosteroid. Claim 2: The composition according to claim 1, wherein the compound is selected from LAS191954, idelalisib, duvelisib, enzastaurin, rigosertib, buparlisib, taselisib, dactolisib, copanlisib, pictrelisib, apitolisib, sonolisib, voxtalisib, ZSTK-47697, GSK-22697 , UCB-5857, RV-1729, RP-6530, omipalisib, SB-2343, WX-037, CAL-120, PWT-33597, CUDC-907, AMG-319, puquitinib, pilaralisib, RP-5264, GDC-0084 or GDC-7666), LY-3023414, PQR-309, DS-7423, XL-499, KAR-4141, RP-5090, PWT-143, IPI-443, RP-6503, ONO-146040, SPR-965, LOR-220, SF-2626, X-339, X-480, PQR-401, INCB-050465, LS-008, CLR-457, PCN-5603, 7-hydroxy-staurosporine, PF-04691502, TG-100115, BGT-226, SF-1126, PKI-179, panulisib, or a pharmaceutically acceptable salt and / or solvate thereof. Claim 3: The composition according to any one of claims 1 and 2, wherein the corticosteroid is one selected from prednisolone, methylprednisolone, dexamethasone, dexamethasone cipecylate, naflocort, deflazacort, halopredone acetate, budesonide, beclomethasone dipropionate, hydrocortisone acetone triamcinolone, fluocinolone acetonide, fluocinonide, clocortolone pivalate, methylprednisolone aceponate, dexamethasone palmitoate, tipredane, hydrocortisone aceponate, prednicarbate, alclometasone dipropionate, halometasone, methylprednisolone suleptanate, mometasone furoate, rimexolone, farnesylate prednisolone, ciclesonide , butixocort propionate, deprodone propionate, fluticasone propionate, halobetasol propionate, loteprednol ethabonate, betamethasone butyrate-propionate, flunisolide, prednisone, dexamethasone sodium phosphate, triamcinolone, betamettasonate betamethasone betamethasone, betamettasonate , hydrocortisone acetate, hydrocortisone and sodium succinate, prednisolone and sodium phosphate and hydrocortisone probutate. Claim 6: A composition according to any one of claims 1 to 4 for use in the treatment of a skin disease. Claim 11: A compound that is a 3-kinase phosphoinositide inhibitor of a pharmaceutically acceptable salt and / or solvate thereof as defined in claim 1 or 2 for use in the treatment of the human or animal body, by simultaneous, concurrent, separate or sequential administration in combination with a corticosteroid as defined in claim 1 or 3 and, optionally, at least one other active compound, as defined in claim 4.

ARP150101655A 2014-05-27 2015-05-27 PHARMACEUTICAL COMPOSITION THAT COMBINES 3-QUINASA D PHOSFOINOSITE INHIBITORS AND CORTICOESTEROIDS FOR THE TREATMENT OF IMMUNOAMPOLOUS CUTANEOUS DISEASES AR100619A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP14382192 2014-05-27

Publications (1)

Publication Number Publication Date
AR100619A1 true AR100619A1 (en) 2016-10-19

Family

ID=50828850

Family Applications (2)

Application Number Title Priority Date Filing Date
ARP150101656A AR100620A1 (en) 2014-05-27 2015-05-27 ADDITION SALTS OF (S) -2- (1- (6-AMINO-5-CYANOPIRIMIDIN-4-ILAMINO) ETIL) -4-OXO-3-PHENYL-3,4-DIHYDROPIRROLO [1,2-F] [ 1,2,4] TRIAZINE-5-CARBONITRILE
ARP150101655A AR100619A1 (en) 2014-05-27 2015-05-27 PHARMACEUTICAL COMPOSITION THAT COMBINES 3-QUINASA D PHOSFOINOSITE INHIBITORS AND CORTICOESTEROIDS FOR THE TREATMENT OF IMMUNOAMPOLOUS CUTANEOUS DISEASES

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ARP150101656A AR100620A1 (en) 2014-05-27 2015-05-27 ADDITION SALTS OF (S) -2- (1- (6-AMINO-5-CYANOPIRIMIDIN-4-ILAMINO) ETIL) -4-OXO-3-PHENYL-3,4-DIHYDROPIRROLO [1,2-F] [ 1,2,4] TRIAZINE-5-CARBONITRILE

Country Status (1)

Country Link
AR (2) AR100620A1 (en)

Also Published As

Publication number Publication date
AR100620A1 (en) 2016-10-19

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