AR099035A1 - Derivado de 6-oxo-1,6-dihidro-piridazina para usar en el tratamiento de carcinoma de células renales (rcc) - Google Patents

Derivado de 6-oxo-1,6-dihidro-piridazina para usar en el tratamiento de carcinoma de células renales (rcc)

Info

Publication number
AR099035A1
AR099035A1 ARP150100023A ARP150100023A AR099035A1 AR 099035 A1 AR099035 A1 AR 099035A1 AR P150100023 A ARP150100023 A AR P150100023A AR P150100023 A ARP150100023 A AR P150100023A AR 099035 A1 AR099035 A1 AR 099035A1
Authority
AR
Argentina
Prior art keywords
rcc
oxo
treatment
carcinoma
piridazina
Prior art date
Application number
ARP150100023A
Other languages
English (en)
Inventor
Dr Bladt Friedhelm
Dr Friese-Hamim Manja
Original Assignee
Merck Patent Ges Mit Beschränkter Haftung
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Ges Mit Beschränkter Haftung filed Critical Merck Patent Ges Mit Beschränkter Haftung
Publication of AR099035A1 publication Critical patent/AR099035A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0031—Rectum, anus
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/02—Suppositories; Bougies; Bases therefor; Ovules
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Abstract

3-(1-{3-[5-(1-metil-piperidin-4-ilmetoxi)-pirimidin-2-il]-bencil}-6-oxo-1,6-dihidro-piridazin-3-il)-benzonitrilo o una sal farmacéuticamente aceptable y/o solvato del mismo para usar Para el tratamiento de carcinoma de células renales (RCC).
ARP150100023A 2014-01-07 2015-01-07 Derivado de 6-oxo-1,6-dihidro-piridazina para usar en el tratamiento de carcinoma de células renales (rcc) AR099035A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP14000036 2014-01-07

Publications (1)

Publication Number Publication Date
AR099035A1 true AR099035A1 (es) 2016-06-22

Family

ID=49916969

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP150100023A AR099035A1 (es) 2014-01-07 2015-01-07 Derivado de 6-oxo-1,6-dihidro-piridazina para usar en el tratamiento de carcinoma de células renales (rcc)

Country Status (17)

Country Link
US (1) US20160331748A1 (es)
EP (1) EP3091980A1 (es)
JP (1) JP2017502978A (es)
KR (1) KR20160099724A (es)
CN (1) CN105873591A (es)
AR (1) AR099035A1 (es)
AU (1) AU2014377079A1 (es)
CA (1) CA2935889C (es)
CL (1) CL2016001726A1 (es)
IL (1) IL246628A0 (es)
MX (1) MX2016008815A (es)
MY (1) MY191613A (es)
PH (1) PH12016500964A1 (es)
RU (1) RU2016132401A (es)
SG (1) SG11201605501RA (es)
TW (1) TW201609103A (es)
WO (1) WO2015104042A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LT3996688T (lt) * 2019-07-10 2023-12-27 Merck Patent Gmbh Farmacinis preparatas

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102007032507A1 (de) * 2007-07-12 2009-04-02 Merck Patent Gmbh Pyridazinonderivate
CA2949515C (en) * 2009-01-08 2018-10-23 Axel Becker Polymorphic forms of 3-(1-{3-[5-(1-methyl-piperidin-4-ylmethoxy)-pyrimidin-2-yl]-benzyl}-6-oxo-1,6-dihydro-pyridazin-3-yl)-benzonitrile hydrochloride salt and processes of manufacturing thereof

Also Published As

Publication number Publication date
TW201609103A (zh) 2016-03-16
EP3091980A1 (en) 2016-11-16
IL246628A0 (en) 2016-08-31
RU2016132401A (ru) 2018-02-13
CN105873591A (zh) 2016-08-17
MY191613A (en) 2022-07-03
CA2935889A1 (en) 2015-07-16
JP2017502978A (ja) 2017-01-26
NZ722879A (en) 2021-08-27
SG11201605501RA (en) 2016-08-30
MX2016008815A (es) 2016-09-08
CA2935889C (en) 2022-08-16
US20160331748A1 (en) 2016-11-17
KR20160099724A (ko) 2016-08-22
AU2014377079A1 (en) 2016-08-18
RU2016132401A3 (es) 2018-08-29
CL2016001726A1 (es) 2016-12-16
PH12016500964A1 (en) 2016-06-20
WO2015104042A1 (en) 2015-07-16

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