AR083435A1 - Formas polimorficas de 4-trifluorometil-n-(3,3a,4,4a,5,5a,6,6a-octahidro-1,3-dioxo-4,6-etencicloprop[f]isoindol-2(1h)-il)-benzamida - Google Patents

Formas polimorficas de 4-trifluorometil-n-(3,3a,4,4a,5,5a,6,6a-octahidro-1,3-dioxo-4,6-etencicloprop[f]isoindol-2(1h)-il)-benzamida

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Publication number
AR083435A1
AR083435A1 ARP110102672A ARP110102672A AR083435A1 AR 083435 A1 AR083435 A1 AR 083435A1 AR P110102672 A ARP110102672 A AR P110102672A AR P110102672 A ARP110102672 A AR P110102672A AR 083435 A1 AR083435 A1 AR 083435A1
Authority
AR
Argentina
Prior art keywords
dioxo
benzamide
etencicloprop
trifluorometile
octahidro
Prior art date
Application number
ARP110102672A
Other languages
English (en)
Inventor
Dylan Nelson
Shanthakumar R Tyavanagimatt
William C Weimers
Melialani A C L Stone
Tove C Bolken
Dennis E Hruby
Michael H Oneill
Gary Sweet-Apple
Kelley A Mcloughan
Original Assignee
Siga Technologies Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/US2011/029576 external-priority patent/WO2011119698A1/en
Application filed by Siga Technologies Inc filed Critical Siga Technologies Inc
Publication of AR083435A1 publication Critical patent/AR083435A1/es

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Abstract

Formas polimórficas de 4-trifluorometil-N-(3,3a,4,4a,5,5a,6,6a-octahidro-1,3-dioxo-4,6-ethenocicloprop[f]isoindol-2(1H)-il)-benzamida de fórmula (1). Métodos para sintetizarlas. Composiciones farmacéuticas que las contienen. Antiviral útil para tratar infecciones de Orthopoxvirus y Eczema vaccinatum.
ARP110102672A 2010-08-12 2011-07-22 Formas polimorficas de 4-trifluorometil-n-(3,3a,4,4a,5,5a,6,6a-octahidro-1,3-dioxo-4,6-etencicloprop[f]isoindol-2(1h)-il)-benzamida AR083435A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US37303110P 2010-08-12 2010-08-12
PCT/US2011/029576 WO2011119698A1 (en) 2010-03-23 2011-03-23 Polymorphic forms st-246 and methods of preparation

Publications (1)

Publication Number Publication Date
AR083435A1 true AR083435A1 (es) 2013-02-27

Family

ID=48485620

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP110102672A AR083435A1 (es) 2010-08-12 2011-07-22 Formas polimorficas de 4-trifluorometil-n-(3,3a,4,4a,5,5a,6,6a-octahidro-1,3-dioxo-4,6-etencicloprop[f]isoindol-2(1h)-il)-benzamida

Country Status (1)

Country Link
AR (1) AR083435A1 (es)

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AR083435A1 (es) Formas polimorficas de 4-trifluorometil-n-(3,3a,4,4a,5,5a,6,6a-octahidro-1,3-dioxo-4,6-etencicloprop[f]isoindol-2(1h)-il)-benzamida

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