AR080504A1 - SALTS OF AN INDAZOLILIPIRROLOTRIAZINA - Google Patents

SALTS OF AN INDAZOLILIPIRROLOTRIAZINA

Info

Publication number
AR080504A1
AR080504A1 ARP110100780A ARP110100780A AR080504A1 AR 080504 A1 AR080504 A1 AR 080504A1 AR P110100780 A ARP110100780 A AR P110100780A AR P110100780 A ARP110100780 A AR P110100780A AR 080504 A1 AR080504 A1 AR 080504A1
Authority
AR
Argentina
Prior art keywords
salts
sulfonic acid
crystalline forms
acid
indazolilipirrolotriazina
Prior art date
Application number
ARP110100780A
Other languages
Spanish (es)
Original Assignee
Ambit Biosciences Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ambit Biosciences Corp filed Critical Ambit Biosciences Corp
Publication of AR080504A1 publication Critical patent/AR080504A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Abstract

Sales de una indazoliIpirrolotriazina, sus procesos de preparacion y sus composiciones farmacéuticas. También métodos de uso para tratar, prevenir o mejorar uno enfermedad proliferativa. Sales de ácido sulfonico de 4-(1-(3-flurobencil)-1H-indazol-5-ilamino)-5-metilpirrolo[1,2-F][1,2,4]triazin-6-il-carbamato de (5)-morfolin-3-ilmetilo. El ácido sulfonico es alquil C1-6 o aril C6-14-sulfonico, formas morfa y cristalinas. Sales de ácido acético, maleico, formas amorfa y cristalina, sales de ácidos nítrico, fosforico.Salts of an indazoliIpyrrolotriazine, its preparation processes and its pharmaceutical compositions. Also methods of use to treat, prevent or improve a proliferative disease. Sulfonic acid salts of 4- (1- (3-flurobenzyl) -1H-indazol-5-ylamino) -5-methylpyrrolo [1,2-F] [1,2,4] triazin-6-yl-carbamate (5) -morpholin-3-ylmethyl. The sulfonic acid is C1-6 alkyl or C6-14-sulfonic acid, morphic and crystalline forms. Salts of acetic acid, maleic, amorphous and crystalline forms, salts of nitric acid, phosphoric.

ARP110100780A 2010-03-11 2011-03-11 SALTS OF AN INDAZOLILIPIRROLOTRIAZINA AR080504A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US31303810P 2010-03-11 2010-03-11

Publications (1)

Publication Number Publication Date
AR080504A1 true AR080504A1 (en) 2012-04-11

Family

ID=43919890

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP110100780A AR080504A1 (en) 2010-03-11 2011-03-11 SALTS OF AN INDAZOLILIPIRROLOTRIAZINA

Country Status (3)

Country Link
AR (1) AR080504A1 (en)
TW (1) TW201136935A (en)
WO (1) WO2011112689A2 (en)

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Also Published As

Publication number Publication date
WO2011112689A3 (en) 2011-11-03
WO2011112689A9 (en) 2011-12-22
TW201136935A (en) 2011-11-01
WO2011112689A2 (en) 2011-09-15

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Legal Events

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