AR077297A1 - Medicamento para uso prolongado de nsaid - Google Patents

Medicamento para uso prolongado de nsaid

Info

Publication number
AR077297A1
AR077297A1 ARP100102334A ARP100102334A AR077297A1 AR 077297 A1 AR077297 A1 AR 077297A1 AR P100102334 A ARP100102334 A AR P100102334A AR P100102334 A ARP100102334 A AR P100102334A AR 077297 A1 AR077297 A1 AR 077297A1
Authority
AR
Argentina
Prior art keywords
nsaid
cobisprotone
pharmaceutically acceptable
acid
patient
Prior art date
Application number
ARP100102334A
Other languages
English (en)
Inventor
Ryuji Ueno
Original Assignee
Sucampo Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sucampo Ag filed Critical Sucampo Ag
Publication of AR077297A1 publication Critical patent/AR077297A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/192Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/557Eicosanoids, e.g. leukotrienes or prostaglandins
    • A61K31/5575Eicosanoids, e.g. leukotrienes or prostaglandins having a cyclopentane, e.g. prostaglandin E2, prostaglandin F2-alpha
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P39/00General protective or antinoxious agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Toxicology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Se provee un medicamento que comprende cobisprotona o su sal, éster, éter o amida farmacéuticamente aceptable para el tratamiento prolongado de una enfermedad o condicion patologica que es una de las indicaciones para el uso de NSAID en un paciente humano, en donde la cobisprotona se administra en al menos 36 mcg por día al paciente que recibe un NSAID. Al administrar cobisprotona o su sal, éster, éter o amida farmacéuticamente aceptable en combinacion con un NSAID, el paciente puede recibir el NSAID durante un período prolongado. Reivindicacion 5: El uso de acuerdo con la reivindicacion 1, en donde la NSAID está seleccionada del grupo que consiste en salicilatos, indometacina, flurbiprofeno, diclofenac, ketorolac, naproxeno, piroxicam, tebufelona, ibuprofeno, etodolac, nabumetona, tenidap, alcofenac, antipirina, aminopirina, dipirona, aminopirona, fenilbutazona, clofezona, oxifenbutazona, prenazona, apazona, benzidamina, bucolome, cincofeno, clonixina, ditrazol, epirizol, fenoprofeno, floctafenina, ácido flufenámico, glafenina, indoprofeno, ketoprofeno, loxoprofeno, ácido meclofenámico, ácido mefenámico, ácido niflumico, fenacetina, salidifamidas, sulindac, suprofeno, tolmetina, una de sus sales farmacéuticamente aceptables y una mezcla de ellos.
ARP100102334A 2009-06-30 2010-06-30 Medicamento para uso prolongado de nsaid AR077297A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US22169809P 2009-06-30 2009-06-30

Publications (1)

Publication Number Publication Date
AR077297A1 true AR077297A1 (es) 2011-08-17

Family

ID=43411168

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP100102334A AR077297A1 (es) 2009-06-30 2010-06-30 Medicamento para uso prolongado de nsaid

Country Status (15)

Country Link
US (1) US20110034424A1 (es)
EP (1) EP2448573A4 (es)
KR (1) KR20120099366A (es)
CN (1) CN102470122A (es)
AR (1) AR077297A1 (es)
AU (1) AU2010267000A1 (es)
BR (1) BRPI1015919A2 (es)
CA (1) CA2765453A1 (es)
IL (1) IL216858A0 (es)
MX (1) MX2012000058A (es)
NZ (1) NZ597675A (es)
RU (1) RU2012102980A (es)
TW (1) TW201105329A (es)
WO (1) WO2011002100A1 (es)
ZA (1) ZA201200656B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN108685929A (zh) * 2012-04-23 2018-10-23 苏坎波公司 用于治疗具有腹泻的肠易激综合征的方法
WO2014159679A1 (en) 2013-03-12 2014-10-02 The United States Of America, As Represented By The Secretary, Department Of Health & Human Services Methods for using lubiprostone to absorb fluid from the subretinal space
US20150057351A1 (en) * 2013-08-22 2015-02-26 Sucampo Ag Method for treating neuropathic pain

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1041012A (en) * 1973-07-10 1978-10-24 American Home Products Corporation Method of reducing the incidence of gastrointestinal side effects during the treatment of inflammatory conditions with antiinflammotory drugs and compositions therefor
US3917828A (en) * 1974-01-28 1975-11-04 Upjohn Co Method of reducing the undesirable gastraintestinal effects of prostaglandin synthetase inhibitors
US5380709A (en) * 1987-01-28 1995-01-10 K.K. Ueno Seiyaku Oyo Kenkyujo Prostaglandins E and anti ulcers containing same
US5225439A (en) * 1987-01-28 1993-07-06 K.K. Ueno Seiyaku Oyo Kenkyujo Prostaglandins E and anti ulcers containing same
US5166174A (en) * 1987-01-28 1992-11-24 K.K. Ueno Seiyaku Oyo Kenkyujo Prostaglandins E and anti-ulcers containing same
US5602184A (en) * 1993-03-03 1997-02-11 The United States Of America As Represented By Department Of Health And Human Services Monoterpenes, sesquiterpenes and diterpenes as cancer therapy
CA2150287C (en) * 1994-06-03 2004-08-10 Ryuji Ueno Agent for treating hepato-biliary diseases
AR026046A1 (es) * 1999-10-15 2002-12-26 R Tech Ueno Ltd NUEVA COMPOSICIoN Y MÉTODO PARA ESTABILIZAR LA MISMA
MXPA04002006A (es) * 2001-08-31 2004-06-07 Sucampo Ag Analogos de prostagladina como abridor del canal de cloruro.
US8337891B2 (en) * 2003-07-03 2012-12-25 Sucampo Ag Enteric coated composition comprising prostaglandin analogs as chloride channel opener
CA2602812C (en) * 2005-04-12 2014-11-18 Sucampo Ag Combined use of prostaglandin compound and proton pump inhibitor for the treatment of gastrointestinal disorders
US20090012165A1 (en) * 2007-07-03 2009-01-08 Sucampo Ag Pharmaceutical combination of nsaid and prostaglandin compound

Also Published As

Publication number Publication date
RU2012102980A (ru) 2013-08-10
CA2765453A1 (en) 2011-01-06
AU2010267000A1 (en) 2012-02-09
EP2448573A1 (en) 2012-05-09
KR20120099366A (ko) 2012-09-10
US20110034424A1 (en) 2011-02-10
EP2448573A4 (en) 2012-11-28
MX2012000058A (es) 2012-01-27
CN102470122A (zh) 2012-05-23
BRPI1015919A2 (pt) 2016-04-26
WO2011002100A1 (en) 2011-01-06
IL216858A0 (en) 2012-02-29
NZ597675A (en) 2014-07-25
TW201105329A (en) 2011-02-16
ZA201200656B (en) 2012-10-31

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