AR067502A1 - Pelets de administracion oral y liberacion retardada de clorhidrato de duloxetina - Google Patents

Pelets de administracion oral y liberacion retardada de clorhidrato de duloxetina

Info

Publication number
AR067502A1
AR067502A1 ARP080102970A ARP080102970A AR067502A1 AR 067502 A1 AR067502 A1 AR 067502A1 AR P080102970 A ARP080102970 A AR P080102970A AR P080102970 A ARP080102970 A AR P080102970A AR 067502 A1 AR067502 A1 AR 067502A1
Authority
AR
Argentina
Prior art keywords
pelets
chlorhydrate
duloxetine
oral administration
delayed delay
Prior art date
Application number
ARP080102970A
Other languages
English (en)
Inventor
Perez Sergio Lloret
Pena Agnes Fernandez
Original Assignee
Combino Pharm Sl
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Combino Pharm Sl filed Critical Combino Pharm Sl
Publication of AR067502A1 publication Critical patent/AR067502A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/38Heterocyclic compounds having sulfur as a ring hetero atom
    • A61K31/381Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Procesos para la elaboracion y el uso de los mismos. Reivindicacion 1: Un pélet de clorhidrato de duloxetina de liberacion retardada caracterizado porque comprende: i) un nucleo inerte; (ii) una primera capa que contiene clorhidrato de duloxetina y opcionalmente uno o más excipientes aceptables para uso farmacéutico; (iii) una capa intermedia que comprende un polímero derivado de celulosa y opcionalmente uno o más excipientes aceptables para uso farmacéutico; y (iv) una capa entérica que comprende un polímero entérico y opcionalmente uno o más excipientes aceptables para uso farmacéutico.
ARP080102970A 2007-07-09 2008-07-10 Pelets de administracion oral y liberacion retardada de clorhidrato de duloxetina AR067502A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US92969707P 2007-07-09 2007-07-09

Publications (1)

Publication Number Publication Date
AR067502A1 true AR067502A1 (es) 2009-10-14

Family

ID=40667910

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP080102970A AR067502A1 (es) 2007-07-09 2008-07-10 Pelets de administracion oral y liberacion retardada de clorhidrato de duloxetina

Country Status (2)

Country Link
AR (1) AR067502A1 (es)
WO (1) WO2009066181A2 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2376095B1 (es) * 2008-10-02 2013-01-24 Laboratorios Del Dr. Esteve, S.A. Pellets entéricos de duloxetina.
MX2012003082A (es) * 2009-09-17 2012-04-19 Cadila Healthcare Ltd Composiciones farmaceuticas para reducir la absorcion rapida de la dosis inducida por el alcohol.
PL224543B1 (pl) 2013-08-21 2017-01-31 Pabianickie Zakłady Farm Polfa Spółka Akcyjna Dojelitowa tabletka duloksetyny

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5508276A (en) * 1994-07-18 1996-04-16 Eli Lilly And Company Duloxetine enteric pellets
DE69721747T2 (de) * 1996-03-11 2004-04-01 Eli Lilly And Co., Indianapolis Methode zur behandlung oder verhütung von interstitieller blasenentzundung
EP1424079A1 (en) * 2002-11-27 2004-06-02 Boehringer Ingelheim International GmbH Combination of a beta-3-receptor agonist and of a reuptake inhibitor of serotonin and/or norepinephrine
JP2008543929A (ja) * 2005-06-20 2008-12-04 カディラ・ヘルスケア・リミテッド デュロキセチンの調節放出型の投与製剤
WO2007139886A2 (en) * 2006-05-22 2007-12-06 Teva Pharmaceutical Industries Ltd. Duloxetine hydrochloride delayed release formulations
EP1938840A1 (en) * 2006-12-27 2008-07-02 LEK Pharmaceuticals D.D. Duloxetine composition
WO2008129501A2 (en) * 2007-04-20 2008-10-30 Wockhardt Research Centre Pharmaceutical compositions of duloxetine

Also Published As

Publication number Publication date
WO2009066181A2 (en) 2009-05-28
WO2009066181A3 (en) 2009-08-20

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