AR057888A1 - Polimorfos de 5-ciclopropil-2-(4-fluorofenil)-6-[(2- hidroxi etil) (metilsulfonil) amino]-n-metil-1-bezofuran-3-carboxamida y metodos para prepararlos - Google Patents

Polimorfos de 5-ciclopropil-2-(4-fluorofenil)-6-[(2- hidroxi etil) (metilsulfonil) amino]-n-metil-1-bezofuran-3-carboxamida y metodos para prepararlos

Info

Publication number
AR057888A1
AR057888A1 ARP060104944A ARP060104944A AR057888A1 AR 057888 A1 AR057888 A1 AR 057888A1 AR P060104944 A ARP060104944 A AR P060104944A AR P060104944 A ARP060104944 A AR P060104944A AR 057888 A1 AR057888 A1 AR 057888A1
Authority
AR
Argentina
Prior art keywords
carboxamide
fluorophenyl
amino
methyl
metilsulfonil
Prior art date
Application number
ARP060104944A
Other languages
English (en)
Original Assignee
Wyeth Corp
Viropharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp, Viropharma Inc filed Critical Wyeth Corp
Publication of AR057888A1 publication Critical patent/AR057888A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/82—Benzo [b] furans; Hydrogenated benzo [b] furans with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D307/84—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Furan Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Reivindicacion 1: Una forma cristalina sustancialmente pura A de la 5-ciclopropil-2-(4-fluorofenil)-6-[(2-hidroxietil)(metilsulfonil)amino]-N-metil-1-benzofuran-3-carboxamida.
ARP060104944A 2005-11-10 2006-11-10 Polimorfos de 5-ciclopropil-2-(4-fluorofenil)-6-[(2- hidroxi etil) (metilsulfonil) amino]-n-metil-1-bezofuran-3-carboxamida y metodos para prepararlos AR057888A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US73519005P 2005-11-10 2005-11-10

Publications (1)

Publication Number Publication Date
AR057888A1 true AR057888A1 (es) 2007-12-26

Family

ID=37951864

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP060104944A AR057888A1 (es) 2005-11-10 2006-11-10 Polimorfos de 5-ciclopropil-2-(4-fluorofenil)-6-[(2- hidroxi etil) (metilsulfonil) amino]-n-metil-1-bezofuran-3-carboxamida y metodos para prepararlos

Country Status (5)

Country Link
US (1) US20070265335A1 (es)
EP (1) EP1945623A2 (es)
AR (1) AR057888A1 (es)
TW (1) TW200804328A (es)
WO (1) WO2007059421A2 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2511774T3 (es) * 2000-05-15 2014-10-23 Takeda Pharmaceutical Company Limited Formas cristalinas de (R)-lansoprazol
US20080182895A1 (en) * 2006-08-25 2008-07-31 Howe Anita Y M Identification and characterization of hcv replicon variants with reduced susceptibility to hcv-796, and methods related thereto
MX2013004655A (es) 2010-10-26 2013-08-27 Presidio Pharmaceuticals Inc Inhibidores del virus de la hepatitis c.

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EA009943B1 (ru) * 2002-11-01 2008-04-28 Вирофарма Инкорпорейтед Соединения бензофурана, композиции и способы лечения и профилактики инфекций, вызванных вирусом гепатита с, и связанных с ним заболеваний

Also Published As

Publication number Publication date
US20070265335A1 (en) 2007-11-15
EP1945623A2 (en) 2008-07-23
WO2007059421A2 (en) 2007-05-24
WO2007059421A3 (en) 2007-07-26
TW200804328A (en) 2008-01-16

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