AR054874A1 - METHOD TO PRODUCE A DERIVATIVE OF 5- HIDROXI -1-ALQUILPIRAZOL - Google Patents
METHOD TO PRODUCE A DERIVATIVE OF 5- HIDROXI -1-ALQUILPIRAZOLInfo
- Publication number
- AR054874A1 AR054874A1 ARP060103247A ARP060103247A AR054874A1 AR 054874 A1 AR054874 A1 AR 054874A1 AR P060103247 A ARP060103247 A AR P060103247A AR P060103247 A ARP060103247 A AR P060103247A AR 054874 A1 AR054874 A1 AR 054874A1
- Authority
- AR
- Argentina
- Prior art keywords
- alquilpirazol
- hidroxi
- derivative
- produce
- alkyl group
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
- C07D231/20—One oxygen atom attached in position 3 or 5
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
Un método para producir un derivado de 5-hidroxi-1-alquilpirazol representado por la formula general (3); donde R2 representa un grupo extractor de electrones, y R3 representa un grupo alquilo C1-6, caracterizado porque un compuesto beta-cetoéster representado por la formula (1) donde R1 representa un grupo alquilo C1-6, y R2 tiene el mismo significado dado anteriormente, se hace reaccionar con una alquilhidrazina representada por la siguiente formula (2) donde R3 tiene el significado ya indicado, bajo una condicion ácida.A method for producing a 5-hydroxy-1-alkylpyrazole derivative represented by the general formula (3); where R2 represents an electron extractor group, and R3 represents a C1-6 alkyl group, characterized in that a beta-ketoester compound represented by formula (1) where R1 represents a C1-6 alkyl group, and R2 has the same given meaning above, it is reacted with an alkylhydrazine represented by the following formula (2) where R3 has the meaning already indicated, under an acidic condition.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2005217098A JP2007031342A (en) | 2005-07-27 | 2005-07-27 | Method for producing 5-hydroxy-1-alkylpyrazole derivative |
Publications (1)
Publication Number | Publication Date |
---|---|
AR054874A1 true AR054874A1 (en) | 2007-07-25 |
Family
ID=37683427
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP060103247A AR054874A1 (en) | 2005-07-27 | 2006-07-27 | METHOD TO PRODUCE A DERIVATIVE OF 5- HIDROXI -1-ALQUILPIRAZOL |
Country Status (4)
Country | Link |
---|---|
JP (1) | JP2007031342A (en) |
AR (1) | AR054874A1 (en) |
TW (1) | TW200740763A (en) |
WO (1) | WO2007013536A1 (en) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20120238760A1 (en) | 2009-11-26 | 2012-09-20 | Basf Se | Method for Producing 5,5-Disubstituted 2-Isoxazolines |
JP5763179B2 (en) | 2010-05-20 | 2015-08-12 | バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングBayer Intellectual Property GmbH | Process for producing 1-alkyl-3-difluoromethyl-5-hydroxypyrazoles |
CN108026051A (en) * | 2015-11-16 | 2018-05-11 | 隆萨有限公司 | Prepare 1- methyl -3-(Trifluoromethyl)The method of -1H- pyrazoles -5- alcohol |
WO2019230831A1 (en) * | 2018-05-31 | 2019-12-05 | クミアイ化学工業株式会社 | Production method for fluorinated pyrazole derivative and intermediate thereof |
CN115385792B (en) * | 2021-05-21 | 2024-02-02 | 帕潘纳(北京)科技有限公司 | Process for the preparation of pyrazole herbicide intermediates |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPH06199804A (en) * | 1992-09-29 | 1994-07-19 | Nippon Nohyaku Co Ltd | Production of 3-substituted phenyl-5-hydroxypyrazole derivative |
JP2000500448A (en) * | 1995-11-15 | 2000-01-18 | ゼネカ リミテッド | Herbicidal substituted pyrazole compounds |
JPH10287654A (en) * | 1997-04-11 | 1998-10-27 | Nissan Chem Ind Ltd | Pyrazolone derivative, and herbicide |
DE10020665A1 (en) * | 2000-04-27 | 2001-10-31 | Schlafhorst & Co W | Method for operating a textile machine producing cross-wound bobbins |
CA2494130C (en) * | 2002-08-01 | 2011-08-23 | Ihara Chemical Industry Co., Ltd. | Pyrazole derivatives and process for the production thereof |
JP4621939B2 (en) * | 2004-03-31 | 2011-02-02 | イハラケミカル工業株式会社 | Process for producing 5-hydroxy-4-thiomethylpyrazole compound |
-
2005
- 2005-07-27 JP JP2005217098A patent/JP2007031342A/en active Pending
-
2006
- 2006-07-20 WO PCT/JP2006/314819 patent/WO2007013536A1/en active Application Filing
- 2006-07-26 TW TW095127200A patent/TW200740763A/en unknown
- 2006-07-27 AR ARP060103247A patent/AR054874A1/en not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
TW200740763A (en) | 2007-11-01 |
WO2007013536A1 (en) | 2007-02-01 |
JP2007031342A (en) | 2007-02-08 |
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