AR051314A1 - METHODS OF TREATMENT OF EPILEPTOGENESIS AND EPILIPSY. PHARMACEUTICAL COMPOSITION AND KIT. - Google Patents

METHODS OF TREATMENT OF EPILEPTOGENESIS AND EPILIPSY. PHARMACEUTICAL COMPOSITION AND KIT.

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Publication number
AR051314A1
AR051314A1 ARP050104150A AR051314A1 AR 051314 A1 AR051314 A1 AR 051314A1 AR P050104150 A ARP050104150 A AR P050104150A AR 051314 A1 AR051314 A1 AR 051314A1
Authority
AR
Argentina
Prior art keywords
epileptogenesis
group
methods
phenyl
alkyl
Prior art date
Application number
Other languages
Spanish (es)
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37600951&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR051314(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of AR051314A1 publication Critical patent/AR051314A1/en

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  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Métodos para prevenir, tratar, revertir, inhibir o detener la epilepsia y la epileptogénesis en un sujeto, que comprenden administrar al sujeto que lo necesita una cantidad terapéuticamente efectiva e un compuesto seleccionado el grupo formado por la formula (1) y la formula (2), o una de sus sales o ésteres aceptables desde el punto de vista farmacéutico, en las cuales fenilo está sustituido en X con uno a cinco átomos de halogeno seleccionados del grupo formado por F, Cl, Br, e I; y R1, R2, R3, R4, R5 y R6 se seleccionan en forma independiente del grupo formado por H y alquilo C1-4; donde el alquilo C1-4 está sustituido en forma opcional con fenilo (donde fenilo está sustituido en forma opcional con sustituyentes seleccionados en forma independiente del grupo formado por halogeno, alquilo C1-4, alcoxi C1-4, amino, nitro y ciano).Methods for preventing, treating, reversing, inhibiting or stopping epilepsy and epileptogenesis in a subject, comprising administering to the subject in need a therapeutically effective amount and a compound selected from the group formed by the formula (1) and the formula (2 ), or one of its pharmaceutically acceptable salts or esters, in which phenyl is substituted on X with one to five halogen atoms selected from the group consisting of F, Cl, Br, and I; and R1, R2, R3, R4, R5 and R6 are independently selected from the group consisting of H and C1-4 alkyl; wherein C1-4 alkyl is optionally substituted with phenyl (where phenyl is optionally substituted with substituents independently selected from the group consisting of halogen, C1-4 alkyl, C1-4 alkoxy, amino, nitro and cyano).

ARP050104150 2005-07-12 2005-09-30 METHODS OF TREATMENT OF EPILEPTOGENESIS AND EPILIPSY. PHARMACEUTICAL COMPOSITION AND KIT. AR051314A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US69862505P 2005-07-12 2005-07-12
US70724205P 2005-08-11 2005-08-11

Publications (1)

Publication Number Publication Date
AR051314A1 true AR051314A1 (en) 2007-01-03

Family

ID=37600951

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP050104150 AR051314A1 (en) 2005-07-12 2005-09-30 METHODS OF TREATMENT OF EPILEPTOGENESIS AND EPILIPSY. PHARMACEUTICAL COMPOSITION AND KIT.

Country Status (4)

Country Link
AR (1) AR051314A1 (en)
PE (1) PE20061039A1 (en)
TW (1) TW200701978A (en)
UY (1) UY29158A1 (en)

Also Published As

Publication number Publication date
TW200701978A (en) 2007-01-16
PE20061039A1 (en) 2006-11-08
UY29158A1 (en) 2005-11-30

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