AR037427A1 - Compuesto de quinolina, uso del mismo para preparar un medicamento, composicion farmaceutica que lo comprende, procedimiento para prepararlo y compuestos de quinolina de utilidad como intermediarios en dicho procedimiento - Google Patents
Compuesto de quinolina, uso del mismo para preparar un medicamento, composicion farmaceutica que lo comprende, procedimiento para prepararlo y compuestos de quinolina de utilidad como intermediarios en dicho procedimientoInfo
- Publication number
- AR037427A1 AR037427A1 ARP020104526A ARP020104526A AR037427A1 AR 037427 A1 AR037427 A1 AR 037427A1 AR P020104526 A ARP020104526 A AR P020104526A AR P020104526 A ARP020104526 A AR P020104526A AR 037427 A1 AR037427 A1 AR 037427A1
- Authority
- AR
- Argentina
- Prior art keywords
- prepare
- procedure
- quinoline
- compound
- pharmaceutical composition
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Immunology (AREA)
- Pulmonology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Un compuesto de quinolina inhibidor de la formación de sCD23 soluble humano que es N-[2-(3-quinolilmetanosulfonil)-1-tetrahidrofuran-2-iletil]-N-hidroxiformamida de fórmula (1). Uso de dicho compuesto para preparar un medicamento para el tratamiento o profilaxis de trastornos en los que está implicada la sobreproducción de sCD23, y composición farmacéutica que lo comprende junto con, opcionalmente, un vehículo farmacéuticamente aceptable. Procedimiento para preparar dicho compuesto y compuestos de quinolina útiles como intermediarios de síntesis.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0128378.7A GB0128378D0 (en) | 2001-11-27 | 2001-11-27 | Novel Compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
AR037427A1 true AR037427A1 (es) | 2004-11-10 |
Family
ID=9926525
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP020104526A AR037427A1 (es) | 2001-11-27 | 2002-11-25 | Compuesto de quinolina, uso del mismo para preparar un medicamento, composicion farmaceutica que lo comprende, procedimiento para prepararlo y compuestos de quinolina de utilidad como intermediarios en dicho procedimiento |
Country Status (11)
Country | Link |
---|---|
US (1) | US7045626B2 (es) |
EP (1) | EP1448552B1 (es) |
JP (1) | JP2005513036A (es) |
AR (1) | AR037427A1 (es) |
AT (1) | ATE334124T1 (es) |
AU (1) | AU2002365511A1 (es) |
DE (1) | DE60213450T2 (es) |
ES (1) | ES2268133T3 (es) |
GB (1) | GB0128378D0 (es) |
TW (1) | TW200303745A (es) |
WO (1) | WO2003045938A1 (es) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR100882156B1 (ko) | 2003-08-08 | 2009-02-06 | 아지노모토 가부시키가이샤 | 나테글리니드 함유 제제 |
PL2780015T3 (pl) | 2011-11-18 | 2017-06-30 | Heptares Therapeutics Limited | Agonisty receptora muskarynowego M1 |
WO2014122474A1 (en) | 2013-02-07 | 2014-08-14 | Takeda Pharmaceutical Company Limited | Piperidin-1 -yl and azepin-1 -yl carboxylates as muscarinic m4 receptor agonists |
GB201617454D0 (en) | 2016-10-14 | 2016-11-30 | Heptares Therapeutics Limited | Pharmaceutical compounds |
GB201810239D0 (en) | 2018-06-22 | 2018-08-08 | Heptares Therapeutics Ltd | Pharmaceutical compounds |
GB201819960D0 (en) | 2018-12-07 | 2019-01-23 | Heptares Therapeutics Ltd | Pharmaceutical compounds |
GB202020191D0 (en) | 2020-12-18 | 2021-02-03 | Heptares Therapeutics Ltd | Pharmaceutical compounds |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NZ501166A (en) | 1997-07-31 | 2001-12-21 | Abbott Lab | Reverse hydroxamate-containing compounds and their use as inhibitors of matrix metalloproteinases |
US6100266A (en) * | 1998-01-30 | 2000-08-08 | Darwin Discovery Limited | Hydroxamic and carboxylic acid derivatives |
-
2001
- 2001-11-27 GB GBGB0128378.7A patent/GB0128378D0/en not_active Ceased
-
2002
- 2002-11-25 WO PCT/EP2002/013264 patent/WO2003045938A1/en active IP Right Grant
- 2002-11-25 DE DE60213450T patent/DE60213450T2/de not_active Expired - Lifetime
- 2002-11-25 ES ES02790436T patent/ES2268133T3/es not_active Expired - Lifetime
- 2002-11-25 AR ARP020104526A patent/AR037427A1/es not_active Application Discontinuation
- 2002-11-25 JP JP2003547388A patent/JP2005513036A/ja active Pending
- 2002-11-25 AU AU2002365511A patent/AU2002365511A1/en not_active Abandoned
- 2002-11-25 TW TW091134147A patent/TW200303745A/zh unknown
- 2002-11-25 US US10/496,193 patent/US7045626B2/en not_active Expired - Fee Related
- 2002-11-25 AT AT02790436T patent/ATE334124T1/de not_active IP Right Cessation
- 2002-11-25 EP EP02790436A patent/EP1448552B1/en not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
DE60213450D1 (de) | 2006-09-07 |
US7045626B2 (en) | 2006-05-16 |
AU2002365511A1 (en) | 2003-06-10 |
EP1448552B1 (en) | 2006-07-26 |
US20050085505A1 (en) | 2005-04-21 |
ES2268133T3 (es) | 2007-03-16 |
EP1448552A1 (en) | 2004-08-25 |
DE60213450T2 (de) | 2007-09-20 |
WO2003045938A1 (en) | 2003-06-05 |
TW200303745A (en) | 2003-09-16 |
ATE334124T1 (de) | 2006-08-15 |
GB0128378D0 (en) | 2002-01-16 |
JP2005513036A (ja) | 2005-05-12 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FA | Abandonment or withdrawal |