AR028970A1 - USE OF CILANSETRON OR ITS SALTS BY ADDITION OF CIDOS AND / OR PHARMACOLOGICALLY COMPATIBLE SOLVATES FOR THE OBTAINING OF PHARMACEUTICAL PREPARATIONS FOR THE TREATMENT AND / OR PROFILAXIS OF THE IRRITABLE INTESTINE SYNDROME - Google Patents
USE OF CILANSETRON OR ITS SALTS BY ADDITION OF CIDOS AND / OR PHARMACOLOGICALLY COMPATIBLE SOLVATES FOR THE OBTAINING OF PHARMACEUTICAL PREPARATIONS FOR THE TREATMENT AND / OR PROFILAXIS OF THE IRRITABLE INTESTINE SYNDROMEInfo
- Publication number
- AR028970A1 AR028970A1 ARP010102958A ARP010102958A AR028970A1 AR 028970 A1 AR028970 A1 AR 028970A1 AR P010102958 A ARP010102958 A AR P010102958A AR P010102958 A ARP010102958 A AR P010102958A AR 028970 A1 AR028970 A1 AR 028970A1
- Authority
- AR
- Argentina
- Prior art keywords
- cilansetron
- treatment
- cidos
- profilaxis
- salts
- Prior art date
Links
- NCNFDKWULDWJDS-OAHLLOKOSA-N cilansetron Chemical compound CC1=NC=CN1C[C@@H]1C(=O)C(C=2C=3N4CCCC=3C=CC=2)=C4CC1 NCNFDKWULDWJDS-OAHLLOKOSA-N 0.000 title abstract 2
- 229960002099 cilansetron Drugs 0.000 title abstract 2
- 210000000936 intestine Anatomy 0.000 title 1
- 239000000825 pharmaceutical preparation Substances 0.000 title 1
- 239000012453 solvate Substances 0.000 title 1
- 208000011580 syndromic disease Diseases 0.000 title 1
- 208000002551 irritable bowel syndrome Diseases 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/538—1,4-Oxazines, e.g. morpholine ortho- or peri-condensed with carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Uso de Cilansetron para el tratamiento de pacientes de IBS masculinos no estrenidos.Use of Cilansetron for the treatment of unstretched male IBS patients.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10036645 | 2000-07-26 | ||
DE10123447A DE10123447A1 (en) | 2000-07-26 | 2001-05-14 | Cilansetron-containing medicines for the treatment of non-obstipative male IBS patients |
Publications (1)
Publication Number | Publication Date |
---|---|
AR028970A1 true AR028970A1 (en) | 2003-05-28 |
Family
ID=26006529
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP010102958A AR028970A1 (en) | 2000-07-26 | 2001-06-21 | USE OF CILANSETRON OR ITS SALTS BY ADDITION OF CIDOS AND / OR PHARMACOLOGICALLY COMPATIBLE SOLVATES FOR THE OBTAINING OF PHARMACEUTICAL PREPARATIONS FOR THE TREATMENT AND / OR PROFILAXIS OF THE IRRITABLE INTESTINE SYNDROME |
Country Status (16)
Country | Link |
---|---|
EP (1) | EP1307195A2 (en) |
JP (1) | JP2004504343A (en) |
CN (1) | CN1444479A (en) |
AR (1) | AR028970A1 (en) |
AU (1) | AU2001276409A1 (en) |
BR (1) | BR0112690A (en) |
CA (1) | CA2417677A1 (en) |
CZ (1) | CZ2003158A3 (en) |
HU (1) | HUP0301479A2 (en) |
IL (1) | IL153972A0 (en) |
MX (1) | MXPA02012917A (en) |
NO (1) | NO20030373L (en) |
PL (1) | PL363517A1 (en) |
RU (1) | RU2003104798A (en) |
SK (1) | SK1272003A3 (en) |
WO (1) | WO2002007713A2 (en) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0216027D0 (en) | 2002-07-10 | 2002-08-21 | Arachnova Therapeutics Ltd | New therapeutic use |
RU2314808C2 (en) * | 2004-01-30 | 2008-01-20 | Астеллас Фарма Инк. | Means for treating irritated intestine syndrome cases with diarrhea predominance |
WO2005073220A1 (en) * | 2004-01-30 | 2005-08-11 | Yamanouchi Pharmaceutical Co., Ltd. | Remedy for irritable bowel syndrome with diarrhea |
JP4632204B2 (en) * | 2005-09-21 | 2011-02-16 | アステラス製薬株式会社 | Antidiarrheal irritable bowel syndrome treatment |
US7601856B2 (en) | 2006-07-27 | 2009-10-13 | Wyeth | Benzofurans as potassium ion channel modulators |
US7662831B2 (en) | 2006-07-27 | 2010-02-16 | Wyeth Llc | Tetracyclic indoles as potassium channel modulators |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9721139D0 (en) * | 1997-10-07 | 1997-12-03 | Glaxo Group Ltd | Medicaments |
GB9930077D0 (en) * | 1999-12-20 | 2000-02-09 | Glaxo Group Ltd | Medicaments |
-
2001
- 2001-06-21 AR ARP010102958A patent/AR028970A1/en unknown
- 2001-07-18 IL IL15397201A patent/IL153972A0/en unknown
- 2001-07-18 BR BR0112690-3A patent/BR0112690A/en not_active Application Discontinuation
- 2001-07-18 EP EP01954044A patent/EP1307195A2/en not_active Withdrawn
- 2001-07-18 CN CN01813307A patent/CN1444479A/en active Pending
- 2001-07-18 PL PL01363517A patent/PL363517A1/en not_active Application Discontinuation
- 2001-07-18 CZ CZ2003158A patent/CZ2003158A3/en unknown
- 2001-07-18 JP JP2002513449A patent/JP2004504343A/en active Pending
- 2001-07-18 SK SK127-2003A patent/SK1272003A3/en unknown
- 2001-07-18 AU AU2001276409A patent/AU2001276409A1/en not_active Abandoned
- 2001-07-18 WO PCT/EP2001/008260 patent/WO2002007713A2/en not_active Application Discontinuation
- 2001-07-18 HU HU0301479A patent/HUP0301479A2/en unknown
- 2001-07-18 CA CA002417677A patent/CA2417677A1/en not_active Abandoned
- 2001-07-18 RU RU2003104798/15A patent/RU2003104798A/en not_active Application Discontinuation
- 2001-07-18 MX MXPA02012917A patent/MXPA02012917A/en unknown
-
2003
- 2003-01-24 NO NO20030373A patent/NO20030373L/en not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
IL153972A0 (en) | 2003-07-31 |
PL363517A1 (en) | 2004-11-29 |
CN1444479A (en) | 2003-09-24 |
WO2002007713A3 (en) | 2002-11-14 |
CA2417677A1 (en) | 2003-01-27 |
BR0112690A (en) | 2003-06-24 |
CZ2003158A3 (en) | 2003-08-13 |
JP2004504343A (en) | 2004-02-12 |
RU2003104798A (en) | 2004-06-27 |
NO20030373D0 (en) | 2003-01-24 |
EP1307195A2 (en) | 2003-05-07 |
NO20030373L (en) | 2003-01-24 |
MXPA02012917A (en) | 2003-05-14 |
SK1272003A3 (en) | 2003-07-01 |
AU2001276409A1 (en) | 2002-02-05 |
WO2002007713A2 (en) | 2002-01-31 |
HUP0301479A2 (en) | 2003-09-29 |
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Legal Events
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FB | Suspension of granting procedure |