AR022469A1 - USE OF SUBSTITUTED AND DERIVATIVE ISOXAZOLCARBOXILIC ACIDS AND NEW SUBSTANCES - Google Patents
USE OF SUBSTITUTED AND DERIVATIVE ISOXAZOLCARBOXILIC ACIDS AND NEW SUBSTANCESInfo
- Publication number
- AR022469A1 AR022469A1 ARP000100427A ARP000100427A AR022469A1 AR 022469 A1 AR022469 A1 AR 022469A1 AR P000100427 A ARP000100427 A AR P000100427A AR P000100427 A ARP000100427 A AR P000100427A AR 022469 A1 AR022469 A1 AR 022469A1
- Authority
- AR
- Argentina
- Prior art keywords
- acids
- substituted
- isoxazolcarboxilic
- derivative
- new substances
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/06—Antianaemics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
- C07D261/08—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
Abstract
La presente invencion se refiere al uso de ácidos isoxazolcarboxílicos sustituidos y derivados de formula general (1) para el tratamiento y profilaxis deenfermedades de anemias, así como de nuevas sustancias de formula general (2) y a nuevos procedimientos para su obtencion.The present invention relates to the use of substituted isoxazolcarboxylic acids and derivatives of the general formula (1) for the treatment and prophylaxis of anemia diseases, as well as new substances of the general formula (2) and to new methods for obtaining them.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19904389A DE19904389A1 (en) | 1999-02-04 | 1999-02-04 | Use of substituted isoxazolecarboxylic acids and derivatives and new substances |
Publications (1)
Publication Number | Publication Date |
---|---|
AR022469A1 true AR022469A1 (en) | 2002-09-04 |
Family
ID=7896332
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP000100427A AR022469A1 (en) | 1999-02-04 | 2000-02-01 | USE OF SUBSTITUTED AND DERIVATIVE ISOXAZOLCARBOXILIC ACIDS AND NEW SUBSTANCES |
Country Status (5)
Country | Link |
---|---|
AR (1) | AR022469A1 (en) |
AU (1) | AU2110000A (en) |
DE (1) | DE19904389A1 (en) |
GT (1) | GT200000011A (en) |
WO (1) | WO2000045799A2 (en) |
Families Citing this family (31)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU6320998A (en) | 1997-02-21 | 1998-09-09 | Bristol-Myers Squibb Company | Benzoic acid derivatives and related compounds as antiarrhythmic agents |
MY151199A (en) | 2001-11-02 | 2014-04-30 | Rigel Pharmaceuticals Inc | Substituted diphenyl heterocycles useful for treating hcv infection |
AU2003262831A1 (en) | 2002-08-23 | 2004-03-11 | Rigel Pharmaceuticals, Inc. | Pyridyl substituted heterocycles useful for treating or preventing hcv infection |
WO2004099165A2 (en) | 2003-05-02 | 2004-11-18 | Rigel Pharmaceuticals, Inc. | Heterocyclic compounds and hydro isomers thereof |
US7115642B2 (en) | 2003-05-02 | 2006-10-03 | Rigel Pharmaceuticals, Inc. | Substituted diphenyl isoxazoles, pyrazoles and oxadiazoles useful for treating HCV infection |
US7220745B2 (en) | 2003-05-15 | 2007-05-22 | Rigel Pharmaceuticals | Heterocyclic compounds useful to treat HCV |
US8580842B2 (en) | 2003-09-30 | 2013-11-12 | Abbott Gmbh & Co. Kg | Heteroaryl-substituted 1,3-dihydroindol-2-one derivatives and medicaments containing them |
WO2005049065A2 (en) | 2003-11-19 | 2005-06-02 | Rigel Pharmaceuticals, Inc. | Synergistic combinations of dihaloacetamide with interferon or ribavirin for treatment hcv infections |
US7514434B2 (en) | 2004-02-23 | 2009-04-07 | Rigel Pharmaceuticals, Inc. | Heterocyclic compounds having an oxadiazole moiety and hydro isomers thereof |
JP2008515992A (en) | 2004-10-13 | 2008-05-15 | ピーティーシー セラピューティクス,インコーポレーテッド | Use of prescribed compounds for the manufacture of medicaments for the prevention / treatment of diseases caused by somatic mutations |
EP1883633A2 (en) | 2005-05-02 | 2008-02-06 | Rigel Pharmaceuticals, Inc. | Heterocyclic anti-viral compounds comprising metabolizable moieties and their uses |
WO2006131336A1 (en) * | 2005-06-08 | 2006-12-14 | Novartis Ag | POLYCYCLIC OXADIAZOLES OR I SOXAZOLES AND THEIR USE AS SlP RECEPTOR LIGANDS |
GB0601744D0 (en) * | 2006-01-27 | 2006-03-08 | Novartis Ag | Organic compounds |
SI2069336T1 (en) | 2006-09-07 | 2013-03-29 | Actelion Pharmaceuticals Ltd. | Pyridin-4-yl derivatives as immunomodulating agents |
PL2069335T3 (en) * | 2006-09-08 | 2013-05-31 | Actelion Pharmaceuticals Ltd | Pyridin-3-yl derivatives as immunomodulating agents |
US20080167286A1 (en) | 2006-12-12 | 2008-07-10 | Abbott Laboratories | Pharmaceutical compositions and their methods of use |
US8486979B2 (en) | 2006-12-12 | 2013-07-16 | Abbvie Inc. | 1,2,4 oxadiazole compounds and methods of use thereof |
UY30846A1 (en) | 2006-12-30 | 2008-07-31 | Abbott Gmbh & Amp | OXINDOL DERIVATIVES REPLACED, MEDICINES THAT UNDERSTAND AND USE THEMSELVES |
WO2008114157A1 (en) | 2007-03-16 | 2008-09-25 | Actelion Pharmaceuticals Ltd | Amino- pyridine derivatives as s1p1 /edg1 receptor agonists |
EP3311813B1 (en) | 2007-08-27 | 2019-08-07 | Dart Neuroscience (Cayman) Ltd | Therapeutic isoxazole compounds |
MX2010006202A (en) | 2007-12-07 | 2011-03-04 | Abbott Gmbh & Co Kg | Amidomethyl-substituted oxindole derivatives and the use thereof for the treatment of vasopressin-dependent illnesses. |
BRPI0820668A2 (en) | 2007-12-07 | 2017-08-22 | Abbott Gmbh & Co Kg | 5-HALOGEN SUBSTITUTED OXINDOL DERIVATIVES AND THEIR USE TO TREAT VASOPRESSIN DEPENDENT DISEASES |
CA2707671C (en) | 2007-12-07 | 2016-02-02 | Abbott Gmbh & Co. Kg | 5,6-disubstituted oxindole-derivatives and use thereof for treating vasopressine-dependent diseases |
WO2010009775A1 (en) | 2007-12-07 | 2010-01-28 | Abbott Gmbh & Co. Kg | Carbamate-substituted oxindole derivatives and use thereof for the treatment of vasopressin-dependent diseases |
WO2010138600A2 (en) | 2009-05-29 | 2010-12-02 | Abbott Laboratories | Pharmaceutical compositions for the treatment of pain |
MX2012000435A (en) | 2009-07-08 | 2012-06-01 | Dermira Canada Inc | Tofa analogs useful in treating dermatological disorders or conditions. |
JP5036923B1 (en) | 2009-07-16 | 2012-09-26 | アクテリオン ファーマシューティカルズ リミテッド | Pyridin-4-yl derivative |
US9133179B2 (en) | 2011-01-19 | 2015-09-15 | Actelion Pharmaceuticals Ltd. | 2-methoxy-pyridin-4-yl-derivatives |
CN102329277B (en) * | 2011-10-24 | 2013-08-07 | 海南霞迪药业有限公司 | Method for preparing Parecoxib |
BR112017024785B1 (en) | 2015-05-20 | 2022-05-17 | Idorsia Pharmaceuticals Ltd | CRYSTALLINE FORM OF COMPOUND (S)-3-{4-[5-(2-CYCLOPENTYL-6-METOXY-PYRIDIN-4-YL)-[1,2,4]OXADIAZOLE-3-YL]-2-ETHYL- 6-METHYLPHENOXY}-PROPANE-1,2-DIOL, PHARMACEUTICAL COMPOSITION, AND USE |
CN116535399B (en) * | 2022-01-25 | 2024-02-27 | 中国药科大学 | 3-hydroxy-5- (isoxazol-5-yl) pyridine formyl glycine compound, preparation method, pharmaceutical composition and application |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB149877A (en) * | 1919-11-22 | 1920-08-26 | Arthur William Wells | Improvements in and in connection with safety razors |
DE3065860D1 (en) * | 1979-02-22 | 1984-01-19 | Monsanto Co | Thermolysis of 2-(3-aryl-isoxazol-5-yl)benzoic acids, salts and halides from 3'-(aryl)-spiro(isobenzofuran-1(3h),5'(4'h)isoxazol)-3-ones |
US5330994A (en) * | 1992-03-24 | 1994-07-19 | Warner-Lambert Company | Tetrahydropyridine isoxazoline derivatives |
DE4314966A1 (en) * | 1993-05-06 | 1994-11-10 | Fahlberg List Pharma Gmbh | 2-Hydroxyphenyl-substituted isoxazoles, the use thereof as pharmaceutical agents and pharmaceutical compositions containing them |
WO1997019039A1 (en) * | 1995-11-17 | 1997-05-29 | Novartis Ag | Solid phase synthesis of heterocyclic compounds and combinatorial compound library |
DE19640370C1 (en) * | 1996-09-30 | 1998-02-12 | Dornier Gmbh Lindauer | Assemblies to hold and guide loom shaft rods |
WO1998057923A1 (en) * | 1997-06-18 | 1998-12-23 | Fujisawa Pharmaceutical Co., Ltd. | New production process |
-
1999
- 1999-02-04 DE DE19904389A patent/DE19904389A1/en not_active Withdrawn
-
2000
- 2000-01-24 WO PCT/EP2000/000517 patent/WO2000045799A2/en active Application Filing
- 2000-01-24 AU AU21100/00A patent/AU2110000A/en not_active Abandoned
- 2000-02-01 AR ARP000100427A patent/AR022469A1/en unknown
- 2000-02-03 GT GT200000011A patent/GT200000011A/en unknown
Also Published As
Publication number | Publication date |
---|---|
WO2000045799A3 (en) | 2002-01-24 |
WO2000045799A2 (en) | 2000-08-10 |
GT200000011A (en) | 2001-07-27 |
DE19904389A1 (en) | 2000-08-10 |
AU2110000A (en) | 2000-08-25 |
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