AR020559A1 - Compuestos n-oxidos de piridina triciclicos, agonistas de la vasopresina, composicion farmaceutica que los comprende y el uso de los mismos para lamanufactura de un medicamento. - Google Patents

Compuestos n-oxidos de piridina triciclicos, agonistas de la vasopresina, composicion farmaceutica que los comprende y el uso de los mismos para lamanufactura de un medicamento.

Info

Publication number
AR020559A1
AR020559A1 ARP000100464A ARP000100464A AR020559A1 AR 020559 A1 AR020559 A1 AR 020559A1 AR P000100464 A ARP000100464 A AR P000100464A AR P000100464 A ARP000100464 A AR P000100464A AR 020559 A1 AR020559 A1 AR 020559A1
Authority
AR
Argentina
Prior art keywords
vasopresine
lamanufacture
piridine
agonists
pharmaceutical composition
Prior art date
Application number
ARP000100464A
Other languages
English (en)
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of AR020559A1 publication Critical patent/AR020559A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/04—Antihaemorrhagics; Procoagulants; Haemostatic agents; Antifibrinolytic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/12—Antidiuretics, e.g. drugs for diabetes insipidus

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

Compuestos N-oxidos de piridina tricíclicos de la siguiente formula general 1 en las cuales se utilizan dichos compuestos y el uso de los mismos para lamanufactura de un medicamento para inducir el retardo temporal de la miccion o para eltratamiento de trastornos que pueden ser remediados o aliviados mediantela actividad agonista de la vasopresina, los cuales incluyen la diabetes insipidus, enuresis nocturna, nocturia, incontinencia urinaria, trastornos de lahemorragia y de lacoagulacion.
ARP000100464A 1999-02-04 2000-02-03 Compuestos n-oxidos de piridina triciclicos, agonistas de la vasopresina, composicion farmaceutica que los comprende y el uso de los mismos para lamanufactura de un medicamento. AR020559A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US24468099A 1999-02-04 1999-02-04

Publications (1)

Publication Number Publication Date
AR020559A1 true AR020559A1 (es) 2002-05-15

Family

ID=22923704

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP000100464A AR020559A1 (es) 1999-02-04 2000-02-03 Compuestos n-oxidos de piridina triciclicos, agonistas de la vasopresina, composicion farmaceutica que los comprende y el uso de los mismos para lamanufactura de un medicamento.

Country Status (12)

Country Link
EP (1) EP1149096B1 (es)
JP (1) JP2002536374A (es)
CN (1) CN1347415A (es)
AR (1) AR020559A1 (es)
AT (1) ATE229956T1 (es)
AU (1) AU2849500A (es)
CA (1) CA2358894A1 (es)
DE (1) DE60001054T2 (es)
DK (1) DK1149096T3 (es)
ES (1) ES2188509T3 (es)
PT (1) PT1149096E (es)
WO (1) WO2000046224A2 (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6455554B1 (en) 1999-06-07 2002-09-24 Targacept, Inc. Oxopyridinyl pharmaceutical compositions and methods for use
GB0115515D0 (en) * 2001-06-25 2001-08-15 Ferring Bv Oxytocin agonisys
WO2004096775A1 (ja) 2003-04-28 2004-11-11 Astellas Pharma Inc. ４，４－ジフルオロ－１，２，３，４－テトラヒドロ－５ｈ－１－ベンゾアゼピン誘導体又はその塩
TWI436988B (zh) * 2007-03-05 2014-05-11 Transform Pharmaceuticals Inc ７-〔（３-氯-６，１１-二氫-６-甲基二苯并〔ｃ，ｆ〕〔１，２〕噻氮呯-１１-基）胺〕庚酸ｓ，ｓ二氧化物之多晶型及其製造與使用方法
GB201005623D0 (en) 2010-04-01 2010-05-19 Vantia Ltd New polymorph
AR094929A1 (es) 2013-02-28 2015-09-09 Bristol Myers Squibb Co Derivados de fenilpirazol como inhibidores potentes de rock1 y rock2
JP6423372B2 (ja) 2013-02-28 2018-11-14 ブリストル−マイヤーズ スクイブ カンパニーＢｒｉｓｔｏｌ−Ｍｙｅｒｓ Ｓｑｕｉｂｂ Ｃｏｍｐａｎｙ 強力なｒｏｃｋ１およびｒｏｃｋ２阻害剤としてのフェニルピラゾール誘導体

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5849735A (en) * 1995-01-17 1998-12-15 American Cyanamid Company Tricyclic benzazepine vasopressin antagonists
AU8592598A (en) * 1997-07-30 1999-02-22 Wyeth Tricyclic vasopressin agonists

Also Published As

Publication number Publication date
CA2358894A1 (en) 2000-08-10
AU2849500A (en) 2000-08-25
EP1149096B1 (en) 2002-12-18
DE60001054D1 (de) 2003-01-30
JP2002536374A (ja) 2002-10-29
ATE229956T1 (de) 2003-01-15
EP1149096A2 (en) 2001-10-31
CN1347415A (zh) 2002-05-01
ES2188509T3 (es) 2003-07-01
DK1149096T3 (da) 2003-04-07
DE60001054T2 (de) 2003-07-24
PT1149096E (pt) 2003-03-31
WO2000046224A3 (en) 2000-12-07
WO2000046224A2 (en) 2000-08-10

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