AR012114A1 - SUBSTITUTED CYAN AND ALKAN CYCLOALCANS, INTERMEDIATE COMPOUND, PROCESSES TO PREPARE THEM, AND COMPOSITION AND METHOD TO COMBAT INSECT PESTS, MITTINGS AND NEMATODES - Google Patents

SUBSTITUTED CYAN AND ALKAN CYCLOALCANS, INTERMEDIATE COMPOUND, PROCESSES TO PREPARE THEM, AND COMPOSITION AND METHOD TO COMBAT INSECT PESTS, MITTINGS AND NEMATODES

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Publication number
AR012114A1
AR012114A1 ARP980101244A ARP980101244A AR012114A1 AR 012114 A1 AR012114 A1 AR 012114A1 AR P980101244 A ARP980101244 A AR P980101244A AR P980101244 A ARP980101244 A AR P980101244A AR 012114 A1 AR012114 A1 AR 012114A1
Authority
AR
Argentina
Prior art keywords
carbamyl
alkoxycarbonyl
groups
formyl
alkynyl
Prior art date
Application number
ARP980101244A
Other languages
Spanish (es)
Original Assignee
Zeneca Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zeneca Ltd filed Critical Zeneca Ltd
Publication of AR012114A1 publication Critical patent/AR012114A1/en

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/45—Carboxylic acid nitriles having cyano groups bound to carbon atoms of rings other than six-membered aromatic rings
    • C07C255/46—Carboxylic acid nitriles having cyano groups bound to carbon atoms of rings other than six-membered aromatic rings to carbon atoms of non-condensed rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/60—1,4-Diazines; Hydrogenated 1,4-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/76—1,3-Oxazoles; Hydrogenated 1,3-oxazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/78—1,3-Thiazoles; Hydrogenated 1,3-thiazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/18—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof containing a —O—CO—N< group, or a thio analogue thereof, directly attached to a heterocyclic or cycloaliphatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/61—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/26—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D241/14—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D241/16—Halogen atoms; Nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/56—Benzoxazoles; Hydrogenated benzoxazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/64—Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
    • C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated

Abstract

Un compuesto de la formula (I), en la cual R1 es Ar-(CH2)n- donde n es cero o uno y Ar es un fenilo opcionalmente sustituido o un sistema de anillosheterocíclicos de 5 o 6 miembros opcionalmente sustituido que contiene entre 1 y 3 heteroátomos independientemente seleccionados entre nitrogeno, oxígeno yazufre, y al menos una insaturacion (doble enlace) entre átomos adyacentes en el anillo, donde los sustituyentes, si los hay, se seleccionan entre átomos dehalogeno, grupos alquilo, alquenilo, alquinilo, alcoxilo, haloalquilo, haloalquenilo, haloalcoxilo, alquitiol y alquilamino, teniendo dichos gruposhasta seis átomos de carbono; R2 y R3 son independientemente hidrogeno o un grupo seleccionado entre grupos alquilo, arilo, heteroarilo, aralquilo,formilo, alquilcarbonilo, arilcarbonilo, heteroarilalquilo, alquenilo, aralquenilo, alquinilo, alcoxicarbonilo, alcanosulfonilo, fenilsulfonilo,alqueniloxicarbonilo, aralquiloxicarbonilo, ariloxicarbonilo,heterociclilalquilo, carbamilo o ditiocarboxilo; las porciones alquilo de R2 yR3 comprenden de 1 a 15 átomos de carbono, y están opcionalmente sustituidas con uno o más sustituyentes seleccionados entre grupos halogeno, ciano,carboxilo, acilo carboxílico, formilo, carbamilo, alcoxicarbonilo, alcoxilo, alquilendioxilo, hidroxilo, nitro, amino, alquilamino, imidato y fosfonato;los miembros arilo, heteroarilo, aralquilo, heteroarilalquilo, alquenilo, aralquenilo, alquinilo, alcoxicarbonilo, alcanosulfonilo, fenilsulfonilo,alqueniloxicarbonilo, aralquiloxicarbonilo, ariloxicarbonilo, heterociclilalquilo, carbamilo y ditiocarboxilo de R2 y R3 están opcionalmentesustituidos con uno o más sustituyentes elegidos entre los grupos halogeno, ciano, carboxilo, arilo carboxílico, formilo, carbamilo, alcoxicarbonilo,A compound of formula (I), in which R1 is Ar- (CH2) n- where n is zero or one and Ar is an optionally substituted phenyl or an optionally substituted 5 or 6 membered heterocyclic ring system containing between 1 and 3 heteroatoms independently selected from nitrogen, oxygen, and sulfur, and at least one unsaturation (double bond) between adjacent ring atoms, where substituents, if any, are selected from halogen atoms, alkyl, alkenyl, alkynyl, alkoxy groups, haloalkyl, haloalkenyl, haloalkoxy, alkythiol and alkylamino, said groups having up to six carbon atoms; R2 and R3 are independently hydrogen or a group selected from alkyl, aryl, heteroaryl, aralkyl, formyl, alkylcarbonyl, arylcarbonyl, heteroarylalkyl, alkenyl, aralkenyl, alkynyl, alkoxycarbonyl, alkanesulfonyl, phenylsulfonyl, alkenyloxycarbonyl, aralkyloxycarbonyl, aryloxycarbonyl, heterocyclylalkyl, carbamyl or dithiocarboxyl; the alkyl portions of R2 and R3 comprise from 1 to 15 carbon atoms, and are optionally substituted with one or more substituents selected from halogen, cyano, carboxyl, carboxylic acyl, formyl, carbamyl, alkoxycarbonyl, alkoxy, alkylenedioxy, hydroxyl, nitro groups, amino, alkylamino, imidate and phosphonate; aryl members, heteroaryl, aralkyl, heteroarylalkyl, alkenyl, aralkenyl, alkynyl, alkoxycarbonyl, alkanesulfonyl, phenylsulfonyl, alkenyloxycarbonyl, aralkyloxycarbonyl, aryloxycarbonyl, heterocyclylalkyl, carbamyl and dithiocarboxyl R2 and R3 are opcionalmentesustituidos with one or more substituents chosen from the groups halogen, cyano, carboxyl, aryl carboxylic, formyl, carbamyl, alkoxycarbonyl,

ARP980101244A 1997-04-01 1998-03-19 SUBSTITUTED CYAN AND ALKAN CYCLOALCANS, INTERMEDIATE COMPOUND, PROCESSES TO PREPARE THEM, AND COMPOSITION AND METHOD TO COMBAT INSECT PESTS, MITTINGS AND NEMATODES AR012114A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9706574.2A GB9706574D0 (en) 1997-04-01 1997-04-01 Cyano substituted cycloalkanes

Publications (1)

Publication Number Publication Date
AR012114A1 true AR012114A1 (en) 2000-09-27

Family

ID=10810089

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP980101244A AR012114A1 (en) 1997-04-01 1998-03-19 SUBSTITUTED CYAN AND ALKAN CYCLOALCANS, INTERMEDIATE COMPOUND, PROCESSES TO PREPARE THEM, AND COMPOSITION AND METHOD TO COMBAT INSECT PESTS, MITTINGS AND NEMATODES

Country Status (8)

Country Link
EP (1) EP0971893A1 (en)
JP (1) JP2002504092A (en)
KR (1) KR20010005811A (en)
AR (1) AR012114A1 (en)
AU (1) AU6508598A (en)
GB (1) GB9706574D0 (en)
WO (1) WO1998043957A1 (en)
ZA (1) ZA982408B (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR101283930B1 (en) 2005-03-28 2013-07-16 토야마 케미칼 컴퍼니 리미티드 Process for production of 1-(3-(2-(1-benzothiophen-5-yl)-ethoxy)propyl)azetidin-3-ol or salts thereof

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1793383C3 (en) * 1968-09-10 1979-03-01 Knoll Ag, 6700 Ludwigshafen 4-Cyano-4-phenyl-aminocyclohexanes and their water-soluble salts, processes for their preparation and pharmaceuticals containing them
US4323388A (en) * 1980-03-10 1982-04-06 Ciba-Geigy Corporation Cyanoalkyl-phenylureas having selective herbicidal activity
GB9510459D0 (en) * 1995-05-24 1995-07-19 Zeneca Ltd Bicyclic amines

Also Published As

Publication number Publication date
JP2002504092A (en) 2002-02-05
GB9706574D0 (en) 1997-05-21
EP0971893A1 (en) 2000-01-19
AU6508598A (en) 1998-10-22
KR20010005811A (en) 2001-01-15
ZA982408B (en) 1998-10-01
WO1998043957A1 (en) 1998-10-08

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