AR011094A1 - MEDICINAL PRODUCT CONTAINING TRIPLE COMBINATION QUINOXALINS AND THE USE OF QUINOXALINES IN TRIPLE COMBINATION WITH PROTEASE INHIBITORS AND TRANSCRIPTASE INHIBITORS AS A MEDICATION FOR THE TREATMENT OF AIDS AND / OR HIV INFECTIONS - Google Patents
MEDICINAL PRODUCT CONTAINING TRIPLE COMBINATION QUINOXALINS AND THE USE OF QUINOXALINES IN TRIPLE COMBINATION WITH PROTEASE INHIBITORS AND TRANSCRIPTASE INHIBITORS AS A MEDICATION FOR THE TREATMENT OF AIDS AND / OR HIV INFECTIONSInfo
- Publication number
- AR011094A1 AR011094A1 ARP980100377A ARP980100377A AR011094A1 AR 011094 A1 AR011094 A1 AR 011094A1 AR P980100377 A ARP980100377 A AR P980100377A AR P980100377 A ARP980100377 A AR P980100377A AR 011094 A1 AR011094 A1 AR 011094A1
- Authority
- AR
- Argentina
- Prior art keywords
- triple combination
- quinoxalines
- inhibitors
- aids
- treatment
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/04—Immunostimulants
Abstract
Medicamento que contiene quinoxalinas en triple combinacion con inhibidores de proteasas e inhibidores de transcriptasa inversa, de formula(I), así como sus formas tautomeras de formula general (Ia), en donde R1, R2, R3, R4 y R5 tienenlos significados dados en las descripcion, son utiles, comomedicamento para el tratamiento del SIDA y/o de infecciones por HIV. También se refiere al uso de las quinoxalinas, de los inhibidores de proteasas y de losinhibidores de transcriptasa inversa, para la produccion de medicamentos para la terapia de infecciones por HIV.A drug containing quinoxalines in triple combination with protease inhibitors and reverse transcriptase inhibitors, of formula (I), as well as their tautomeric forms of general formula (Ia), where R1, R2, R3, R4 and R5 have the meanings given in The descriptions are useful as a medicine for the treatment of AIDS and / or HIV infections. It also refers to the use of quinoxalines, protease inhibitors, and reverse transcriptase inhibitors, for the production of drugs for the therapy of HIV infections.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19703131A DE19703131A1 (en) | 1997-01-29 | 1997-01-29 | Use of quinoxaline in a combination of three with protease inhibitors and reverse transcriptase inhibitors as medicaments for the treatment of AIDS and / or HIV infections |
Publications (1)
Publication Number | Publication Date |
---|---|
AR011094A1 true AR011094A1 (en) | 2000-08-02 |
Family
ID=7818634
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP980100377A AR011094A1 (en) | 1997-01-29 | 1998-01-28 | MEDICINAL PRODUCT CONTAINING TRIPLE COMBINATION QUINOXALINS AND THE USE OF QUINOXALINES IN TRIPLE COMBINATION WITH PROTEASE INHIBITORS AND TRANSCRIPTASE INHIBITORS AS A MEDICATION FOR THE TREATMENT OF AIDS AND / OR HIV INFECTIONS |
Country Status (16)
Country | Link |
---|---|
EP (1) | EP0977570A1 (en) |
JP (1) | JP2001511124A (en) |
KR (1) | KR20000070543A (en) |
CN (1) | CN1251525A (en) |
AR (1) | AR011094A1 (en) |
AU (1) | AU6094098A (en) |
BR (1) | BR9807523A (en) |
CA (1) | CA2278773A1 (en) |
DE (1) | DE19703131A1 (en) |
ID (1) | ID22414A (en) |
IL (1) | IL130877A0 (en) |
NO (1) | NO993670L (en) |
PL (1) | PL334770A1 (en) |
SK (1) | SK99899A3 (en) |
WO (1) | WO1998032442A1 (en) |
ZA (1) | ZA98679B (en) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU4219799A (en) * | 1998-05-29 | 1999-12-13 | University Of Florida | Combination therapy for treatment of fiv infection |
US6875773B1 (en) | 1998-05-29 | 2005-04-05 | Ben M. Dunn | Combination therapy for treatment of FIV infection |
AU6329599A (en) * | 1998-09-28 | 2000-04-17 | Glaxo Group Limited | Antiviral combinations comprising (s)-2-ethyl -7-fluoro -3-oxo-3, 4-dihydro -2h-quinoxaline -1-carboxylic acid isopropyl ester |
GB9821000D0 (en) * | 1998-09-28 | 1998-11-18 | Glaxo Group Ltd | Antiviral combinations |
GB9911887D0 (en) * | 1999-05-21 | 1999-07-21 | Glaxo Group Ltd | Methods and medicaments for post exposure prophylaxis of an hiv infection |
SE9902987D0 (en) | 1999-08-24 | 1999-08-24 | Astra Pharma Prod | Novel compounds |
CO5300399A1 (en) | 2000-02-25 | 2003-07-31 | Astrazeneca Ab | HETEROCICLIOCS CONTAINING NITROGEN, PROCESS FOR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
AR028948A1 (en) | 2000-06-20 | 2003-05-28 | Astrazeneca Ab | NEW COMPOUNDS |
US7005439B2 (en) | 2000-06-20 | 2006-02-28 | Astrazeneca Ab | Compounds |
GB0104050D0 (en) | 2001-02-19 | 2001-04-04 | Astrazeneca Ab | Chemical compounds |
AR035230A1 (en) | 2001-03-19 | 2004-05-05 | Astrazeneca Ab | BENCIMIDAZOL COMPOUNDS, PROCESS FOR PREPARATION, PHARMACEUTICAL COMPOSITION, PROCESS FOR THE PREPARATION OF SUCH PHARMACEUTICAL COMPOSITION, AND USES OF THESE COMPOUNDS FOR THE PREPARATION OF MEDICINES |
GB0107228D0 (en) | 2001-03-22 | 2001-05-16 | Astrazeneca Ab | Chemical compounds |
SE0101038D0 (en) | 2001-03-23 | 2001-03-23 | Astrazeneca Ab | Novel compounds |
SE0103818D0 (en) | 2001-11-15 | 2001-11-15 | Astrazeneca Ab | Chemical compounds |
SE0301369D0 (en) | 2003-05-09 | 2003-05-09 | Astrazeneca Ab | Chemical compounds |
US7351709B2 (en) | 2004-06-09 | 2008-04-01 | Wyeth | Estrogen receptor ligands |
TW200738634A (en) | 2005-08-02 | 2007-10-16 | Astrazeneca Ab | New salt |
CA2633400A1 (en) * | 2005-12-15 | 2007-06-21 | Bayer Healthcare Ag | Diaryl urea for treating virus infections |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK0509398T3 (en) * | 1991-04-15 | 2002-01-14 | Aventis Pharma Gmbh | Quinoxalins, processes for their preparation and their use |
DE4342024A1 (en) * | 1993-12-09 | 1995-06-14 | Hoechst Ag | Combination preparations containing a quinoxaline and a nucleoside |
DE19506742A1 (en) * | 1995-02-27 | 1996-08-29 | Bayer Ag | Use of quinoxalines in combination with protease inhibitors as medicaments for the treatment of AIDS and / or HIV infections |
-
1997
- 1997-01-29 DE DE19703131A patent/DE19703131A1/en not_active Withdrawn
-
1998
- 1998-01-15 JP JP53154098A patent/JP2001511124A/en active Pending
- 1998-01-15 BR BR9807523A patent/BR9807523A/en not_active Application Discontinuation
- 1998-01-15 WO PCT/EP1998/000197 patent/WO1998032442A1/en not_active Application Discontinuation
- 1998-01-15 SK SK998-99A patent/SK99899A3/en unknown
- 1998-01-15 KR KR1019997006788A patent/KR20000070543A/en not_active Application Discontinuation
- 1998-01-15 CN CN98803782A patent/CN1251525A/en active Pending
- 1998-01-15 CA CA002278773A patent/CA2278773A1/en not_active Abandoned
- 1998-01-15 PL PL98334770A patent/PL334770A1/en unknown
- 1998-01-15 IL IL13087798A patent/IL130877A0/en unknown
- 1998-01-15 AU AU60940/98A patent/AU6094098A/en not_active Abandoned
- 1998-01-15 ID IDW990759A patent/ID22414A/en unknown
- 1998-01-15 EP EP98905297A patent/EP0977570A1/en not_active Withdrawn
- 1998-01-28 ZA ZA98679A patent/ZA98679B/en unknown
- 1998-01-28 AR ARP980100377A patent/AR011094A1/en unknown
-
1999
- 1999-07-28 NO NO993670A patent/NO993670L/en not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
BR9807523A (en) | 2000-03-21 |
JP2001511124A (en) | 2001-08-07 |
CN1251525A (en) | 2000-04-26 |
PL334770A1 (en) | 2000-03-13 |
ZA98679B (en) | 1998-08-05 |
CA2278773A1 (en) | 1998-07-30 |
WO1998032442A1 (en) | 1998-07-30 |
EP0977570A1 (en) | 2000-02-09 |
DE19703131A1 (en) | 1998-07-30 |
NO993670L (en) | 1999-09-10 |
IL130877A0 (en) | 2001-01-28 |
ID22414A (en) | 1999-10-14 |
SK99899A3 (en) | 2000-03-13 |
KR20000070543A (en) | 2000-11-25 |
NO993670D0 (en) | 1999-07-28 |
AU6094098A (en) | 1998-08-18 |
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