AR002258A1 -
DERIVATIVES OF PHENOXYPYRIMIDINYL, PHARMACEUTICAL PREPARATIONS CONTAINING THEM, A PROCEDURE FOR THEIR PREPARATION AND THEIR USE TO PREPARE MEDICINES
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DERIVATIVES OF PHENOXYPYRIMIDINYL, PHARMACEUTICAL PREPARATIONS CONTAINING THEM, A PROCEDURE FOR THEIR PREPARATION AND THEIR USE TO PREPARE MEDICINES
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Derivados fenoxipirimidinilo de fórmula (I) en donde R1 - R8, A y B tienen el significado dado en la descripción,son inhibidores de la endotelina y puedenemplearse para el tratamiento de trastornos asociados con actividades de la endotelina,tal es como la hipertensión arterial, se describe ademáspreparaciones farmacéuticas que los contienen y un procedimiento para su preparación.Phenoxypyrimidinyl derivatives of formula (I) where R1-R8, A and B have the meaning given in the description, are endothelin inhibitors and can be used for the treatment of disorders associated with endothelin activities, such as high blood pressure, It also describes pharmaceutical preparations containing them and a procedure for their preparation.
ARP950100612A1994-12-201995-12-18
DERIVATIVES OF PHENOXYPYRIMIDINYL, PHARMACEUTICAL PREPARATIONS CONTAINING THEM, A PROCEDURE FOR THEIR PREPARATION AND THEIR USE TO PREPARE MEDICINES
AR002258A1
(en)
AMIDAS OF ANTRANILIC ACIDS WITH SIDE CHAIN OF HETEROARILSULFONILO, PROCEDURE FOR THEIR PREPARATION, ITS EMPLOYMENT AS A MEDICINAL OR DIAGNOSTIC AGENT, AS WELL AS PHARMACEUTICAL PREPARATIONS CONTAINING THEM
DERIVATIVES OF PURIN-6-ONA, PROCEDURES FOR THEIR PREPARATION, THE USE OF THE SAME IN THE PREPARATION OF MEDICINES, MEDICINES THAT CONTAIN THEM AND A PROCEDURE FOR PREPARING SUCH MEDICINES
PIRROLOPYROLONE COMPOUNDS, A PHARMACEUTICAL COMPOSITION THAT CONTAINS THEM, ITS USE IN THE MANUFACTURE OF A MEDICINAL PRODUCT AND IN THERAPY, PROCESSES FOR ITS PREPARATION AND INTERMEDIARY COMPOUNDS FOR SUCH PROCESSES.