AR002258A1 - DERIVATIVES OF PHENOXYPYRIMIDINYL, PHARMACEUTICAL PREPARATIONS CONTAINING THEM, A PROCEDURE FOR THEIR PREPARATION AND THEIR USE TO PREPARE MEDICINES - Google Patents

DERIVATIVES OF PHENOXYPYRIMIDINYL, PHARMACEUTICAL PREPARATIONS CONTAINING THEM, A PROCEDURE FOR THEIR PREPARATION AND THEIR USE TO PREPARE MEDICINES

Info

Publication number
AR002258A1
AR002258A1 ARP950100612A AR10061295A AR002258A1 AR 002258 A1 AR002258 A1 AR 002258A1 AR P950100612 A ARP950100612 A AR P950100612A AR 10061295 A AR10061295 A AR 10061295A AR 002258 A1 AR002258 A1 AR 002258A1
Authority
AR
Argentina
Prior art keywords
phenoxypyrimidinyl
derivatives
procedure
preparation
pharmaceutical preparations
Prior art date
Application number
ARP950100612A
Other languages
Spanish (es)
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of AR002258A1 publication Critical patent/AR002258A1/en

Links

Abstract

Derivados fenoxipirimidinilo de fórmula (I) en donde R1 - R8, A y B tienen el significado dado en la descripción,son inhibidores de la endotelina y puedenemplearse para el tratamiento de trastornos asociados con actividades de la endotelina,tal es como la hipertensión arterial, se describe ademáspreparaciones farmacéuticas que los contienen y un procedimiento para su preparación.Phenoxypyrimidinyl derivatives of formula (I) where R1-R8, A and B have the meaning given in the description, are endothelin inhibitors and can be used for the treatment of disorders associated with endothelin activities, such as high blood pressure, It also describes pharmaceutical preparations containing them and a procedure for their preparation.

ARP950100612A 1994-12-20 1995-12-18 DERIVATIVES OF PHENOXYPYRIMIDINYL, PHARMACEUTICAL PREPARATIONS CONTAINING THEM, A PROCEDURE FOR THEIR PREPARATION AND THEIR USE TO PREPARE MEDICINES AR002258A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH383794 1994-12-20

Publications (1)

Publication Number Publication Date
AR002258A1 true AR002258A1 (en) 1998-03-11

Family

ID=4264545

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP950100612A AR002258A1 (en) 1994-12-20 1995-12-18 DERIVATIVES OF PHENOXYPYRIMIDINYL, PHARMACEUTICAL PREPARATIONS CONTAINING THEM, A PROCEDURE FOR THEIR PREPARATION AND THEIR USE TO PREPARE MEDICINES

Country Status (8)

Country Link
AR (1) AR002258A1 (en)
CO (1) CO4700288A1 (en)
PE (1) PE60196A1 (en)
PL (1) PL188801B1 (en)
RU (1) RU2151767C1 (en)
TR (1) TR199501608A2 (en)
UY (1) UY24121A1 (en)
ZA (1) ZA9510622B (en)

Also Published As

Publication number Publication date
ZA9510622B (en) 1996-06-20
RU2151767C1 (en) 2000-06-27
PL188801B1 (en) 2005-04-29
CO4700288A1 (en) 1998-12-29
PE60196A1 (en) 1996-12-28
PL320941A1 (en) 1997-11-24
TR199501608A2 (en) 1996-07-21
UY24121A1 (en) 2000-12-29

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AR002258A1 (en) DERIVATIVES OF PHENOXYPYRIMIDINYL, PHARMACEUTICAL PREPARATIONS CONTAINING THEM, A PROCEDURE FOR THEIR PREPARATION AND THEIR USE TO PREPARE MEDICINES