AP9300596A0 - Azole derivatives. - Google Patents

Azole derivatives.

Info

Publication number
AP9300596A0
AP9300596A0 APAP/P/1993/000596A AP9300596A AP9300596A0 AP 9300596 A0 AP9300596 A0 AP 9300596A0 AP 9300596 A AP9300596 A AP 9300596A AP 9300596 A0 AP9300596 A0 AP 9300596A0
Authority
AP
ARIPO
Prior art keywords
azole derivatives
triazolo
ethylamino
morpholino
furyl
Prior art date
Application number
APAP/P/1993/000596A
Inventor
Geraint Jones
Original Assignee
Zeneca Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zeneca Ltd filed Critical Zeneca Ltd
Publication of AP9300596A0 publication Critical patent/AP9300596A0/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

2-(2-furyl)-5-[2-(morpholino)ethylamino][1,2,4]triazolo[1,5-a][1,3,5]triazine-7-amine and the pharmaceutically acceptable salts thereof, which are selective a2a adenosine antagonists. Also disclosed are pharmaceutical compositions comprising the compounds and processes for their preparation.
APAP/P/1993/000596A 1992-12-22 1993-12-02 Azole derivatives. AP9300596A0 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB929226735A GB9226735D0 (en) 1992-12-22 1992-12-22 Azole derivatives

Publications (1)

Publication Number Publication Date
AP9300596A0 true AP9300596A0 (en) 1994-01-31

Family

ID=10727043

Family Applications (1)

Application Number Title Priority Date Filing Date
APAP/P/1993/000596A AP9300596A0 (en) 1992-12-22 1993-12-02 Azole derivatives.

Country Status (9)

Country Link
CN (1) CN1093708A (en)
AP (1) AP9300596A0 (en)
AU (1) AU5656494A (en)
GB (2) GB9226735D0 (en)
HR (1) HRP931512A2 (en)
IL (1) IL107876A0 (en)
SI (1) SI9300674A (en)
WO (1) WO1994014812A1 (en)
ZA (1) ZA939045B (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2639299A (en) * 1998-02-24 1999-09-15 Kyowa Hakko Kogyo Co. Ltd. Remedies/preventives for parkinson's disease
US6355653B1 (en) 1999-09-06 2002-03-12 Hoffmann-La Roche Inc. Amino-triazolopyridine derivatives
US6506772B1 (en) * 2000-12-15 2003-01-14 Hoffmann-La Roche Inc. Substituted [1,2,4]triazolo[1,5a]pyridine derivatives with activity as adenosine receptor ligands
US6514989B1 (en) * 2001-07-20 2003-02-04 Hoffmann-La Roche Inc. Aromatic and heteroaromatic substituted 1,2,4-triazolo pyridine derivatives
BR0304925A (en) * 2002-05-30 2004-09-28 Solvay Pharm Bv Compounds, pharmaceutical compositions, and use of compounds
CN112608316B (en) * 2019-07-30 2022-10-21 厦门宝太生物科技股份有限公司 Pyrazolotriazine adenosine receptor antagonist

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2244487B (en) * 1990-05-29 1994-02-02 Ici Plc Azole derivatives

Also Published As

Publication number Publication date
GB9324349D0 (en) 1994-01-12
WO1994014812A1 (en) 1994-07-07
SI9300674A (en) 1994-06-30
GB9226735D0 (en) 1993-02-17
HRP931512A2 (en) 1994-12-31
ZA939045B (en) 1994-06-22
CN1093708A (en) 1994-10-19
IL107876A0 (en) 1994-04-12
AU5656494A (en) 1994-07-19

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