JP2015147757A - Heterocyclic derivative and pest control agent - Google Patents

Heterocyclic derivative and pest control agent Download PDF

Info

Publication number
JP2015147757A
JP2015147757A JP2014048820A JP2014048820A JP2015147757A JP 2015147757 A JP2015147757 A JP 2015147757A JP 2014048820 A JP2014048820 A JP 2014048820A JP 2014048820 A JP2014048820 A JP 2014048820A JP 2015147757 A JP2015147757 A JP 2015147757A
Authority
JP
Japan
Prior art keywords
optionally substituted
alkyl
group
substituted
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2014048820A
Other languages
Japanese (ja)
Inventor
沼田 昭
Akira Numata
昭 沼田
裕二 岩脇
Yuji Iwawaki
裕二 岩脇
公則 安藤
Kiminori Ando
公則 安藤
裕貴 古川
Hirotaka Furukawa
裕貴 古川
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Nissan Chemical Corp
Original Assignee
Nissan Chemical Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nissan Chemical Corp filed Critical Nissan Chemical Corp
Priority to JP2014048820A priority Critical patent/JP2015147757A/en
Publication of JP2015147757A publication Critical patent/JP2015147757A/en
Pending legal-status Critical Current

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

PROBLEM TO BE SOLVED: To provide a novel pest control agent, especially an insecticide or an acaricide.SOLUTION: There are provided: a heterocyclic derivative represented by the formula (1) [wherein, Arepresents -N(O)or -CR; Rrepresents a hydrogen atom, a halogen atom, an alkyl group having 1 to 6 carbon atoms or the like; Rrepresents a hydrogen atom, a cyano or an alkyl group having 1 to 12 carbon atoms or the like; Rrepresents -C(O)Ror the like; Rrepresents a halogen atom, an alkyl group having 1 to 6 carbon atoms or the like; B represents a heterocycle of B-1 to B-34; n represents an integer of 0 to 3.]; and a pest control agent.

Description

本発明は、新規な複素環誘導体及びそれらの塩、並びに該化合物を有効成分として含有することを特徴とする有害生物防除剤に関するものである。本発明における有害生物防除剤とは、農園芸分野又は畜産・衛生分野(家畜や愛玩動物としての哺乳動物又は鳥類に対する内部寄生虫・外部寄生虫や家庭用及び業務用の衛生害虫・不快害虫)等における有害な節足動物を対象とした害虫防除剤を意味する。また、本発明における農薬とは、農園芸分野における殺虫・殺ダニ剤、殺線虫剤、除草剤及び殺菌剤等を意味する。   The present invention relates to a novel heterocyclic derivative and a salt thereof, and a pest control agent comprising the compound as an active ingredient. The pest control agent in the present invention is the field of agriculture and horticulture or the field of livestock and hygiene (internal parasites / external parasites for domestic animals and pets, hygiene pests and unpleasant pests for domestic and commercial use) It means a pest control agent for harmful arthropods such as The agrochemical in the present invention means an insecticide / acaricide, nematicide, herbicide, fungicide, etc. in the field of agriculture and horticulture.

また特許文献1〜7には、複素環誘導体が殺虫剤として有用であることが開示されているが、本発明に係る複素環誘導体については何ら開示されていない。   Patent Documents 1 to 7 disclose that heterocyclic derivatives are useful as insecticides, but do not disclose any heterocyclic derivatives according to the present invention.

国際公開第2011/049150号International Publication No. 2011/049150 国際公開第2011/128304号International Publication No. 2011/128304 国際公開第2012/030681号International Publication No. 2012/030881 国際公開第2012/061288号International Publication No. 2012/061288 国際公開第2012/061290号International Publication No. 2012/061290 国際公開第2010/129497号International Publication No. 2010/129497 国際公開第2012/007500号International Publication No. 2012/007500

農園芸病害虫、森林病害虫、或いは衛生病害虫等、各種病害虫の防除を目的とする有害生物防除剤の開発が進み、多種多様な薬剤が今日まで実用に供されてきた。   The development of pest control agents for the purpose of controlling various pests such as agricultural and horticultural pests, forest pests, and hygiene pests has progressed, and a wide variety of drugs have been put to practical use to date.

しかしながら、こうした薬剤の長年にわたる使用により、近年、病害虫が薬剤抵抗性を獲得し、従来用いられてきた既存の殺虫剤や殺菌剤による防除が困難となる場面が増えてきている。また、既存の有害生物防除剤の一部のものは毒性が高く、或いはあるものは環境中に長期間残留することにより、生態系を攪乱するという問題も顕在化しつつある。このような状況下、高度な有害生物防除活性を有するのみならず、低毒性且つ低残留性の新規な有害生物防除剤の開発が常に期待されている。   However, due to the long-term use of such drugs, in recent years, pests have acquired drug resistance, making it difficult to control with existing insecticides and fungicides that have been used. In addition, some existing pest control agents are highly toxic, or some of them remain in the environment for a long time, and the problem of disturbing the ecosystem is becoming apparent. Under such circumstances, development of a novel pest control agent having not only high pest control activity but also low toxicity and low persistence is always expected.

本発明者らは、上記の課題解決を目標に鋭意研究を重ねた結果、本発明に係る下記式(1)で表される新規な複素環誘導体が優れた有害生物防除活性、特に殺虫・殺ダニ活性を示し、且つ、ホ乳動物、魚類及び益虫等の非標的生物に対してほとんど悪影響の無い、極めて有用な化合物であることを見い出し、本発明を完成した。   As a result of intensive research aimed at solving the above problems, the present inventors have found that the novel heterocyclic derivative represented by the following formula (1) according to the present invention has excellent pest control activity, particularly insecticidal / killing. The present invention was completed by discovering that it is a very useful compound that exhibits mite activity and has almost no adverse effect on non-target organisms such as mammals, fish and beneficial insects.

すなわち、本発明は下記〔1〕〜〔9〕に関するものである。   That is, the present invention relates to the following [1] to [9].

〔1〕
式(1):
[1]
Formula (1):

Figure 2015147757
Figure 2015147757

[式中、Aは、−N(−O)m2又は−CRを表し、
、R、R、R4a及びR4bは、各々独立して水素原子、ハロゲン原子、シアノ、ニトロ、−OH、−SH、−NH、C〜Cアルキル、R28aによって任意に置換された(C〜C)アルキル、C〜Cシクロアルキル、R28aによって任意に置換された(C〜C)シクロアルキル、C〜Cアルケニル、R28aによって任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R28aによって任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R28aによって任意に置換された(C〜C)アルキニル、C〜Cアルコキシ、C〜Cハロアルコキシ、C〜Cアルケニルオキシ、C〜Cアルキルチオ、C〜Cアルキルスルフィニル、C〜Cアルキルスルホニル、C〜Cハロアルキルチオ、C〜Cハロアルキルスルフィニル、C〜Cハロアルキルスルホニル、C〜Cアルキルカルボニル、C〜Cシクロアルキルカルボニル、C〜Cハロアルキルカルボニル、C〜Cハロシクロアルキルカルボニル、C〜Cアルコキシカルボニル、C〜Cハロアルコキシカルボニル、C〜Cアルキルチオカルボニル、C〜Cアルコキシチオカルボニル、C〜Cアルキルジチオカルボニル、C〜Cアルキルアミノカルボニル、C〜Cハロアルキルアミノカルボニル、ジ(C〜Cアルキル)アミノカルボニル、トリ(C〜Cアルキル)シリル、C〜Cアルキルアミノスルホニル、ジ(C〜Cアルキル)アミノスルホニル、C〜Cアルキルカルボニルオキシ、C〜Cアルキルスルホニルオキシ、C〜Cハロアルキルスルホニルオキシ、C〜Cアルキルアミノ、ジ(C〜Cアルキル)アミノ、フェニル、ナフチル、(Z)で置換されたフェニル、(Z)で置換されたナフチル又はD1−1〜D1−99を表し、
は、ハロゲン原子、シアノ、ニトロ、−OH、−SH、−NH、C〜Cアルキル、R28aによって任意に置換された(C〜C)アルキル、C〜Cシクロアルキル、R28aによって任意に置換された(C〜C)シクロアルキル、C〜Cアルケニル、R28aによって任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R28aによって任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R28aによって任意に置換された(C〜C)アルキニル、C〜Cアルコキシ、C〜Cハロアルコキシ、C〜Cアルケニルオキシ、C〜Cアルキルチオ、C〜Cアルキルスルフィニル、C〜Cアルキルスルホニル、C〜Cハロアルキルチオ、C〜Cハロアルキルスルフィニル、C〜Cハロアルキルスルホニル、C〜Cアルキルカルボニル、C〜Cシクロアルキルカルボニル、C〜Cハロアルキルカルボニル、C〜Cハロシクロアルキルカルボニル、C〜Cアルコキシカルボニル、C〜Cハロアルコキシカルボニル、C〜Cアルキルチオカルボニル、C〜Cアルコキシチオカルボニル、C〜Cアルキルジチオカルボニル、C〜Cアルキルアミノカルボニル、C〜Cハロアルキルアミノカルボニル、ジ(C〜Cアルキル)アミノカルボニル、トリ(C〜Cアルキル)シリル、C〜Cアルキルアミノスルホニル、ジ(C〜Cアルキル)アミノスルホニル、C〜Cアルキルカルボニルオキシ、C〜Cアルキルスルホニルオキシ、C〜Cハロアルキルスルホニルオキシ、C〜Cアルキルアミノ、ジ(C〜Cアルキル)アミノ、フェニル、ナフチル、(Z)で置換されたフェニル、(Z)で置換されたナフチル又はD1−1〜D1−99を表し、nが2以上の整数を表すとき、各々のRは互いに同一であっても又は互いに相異なってもよく、
3aは、水素原子、シアノ、ニトロ、−OH、−SH、−NH、C〜Cアルキル、R28aによって任意に置換された(C〜C)アルキル、C〜Cシクロアルキル、R28aによって任意に置換された(C〜C)シクロアルキル、C〜Cアルケニル、R28aによって任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R28aによって任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R28aによって任意に置換された(C〜C)アルキニル、C〜Cアルコキシ、C〜Cハロアルコキシ、C〜Cアルケニルオキシ、C〜Cアルキルチオ、C〜Cアルキルスルフィニル、C〜Cアルキルスルホニル、C〜Cハロアルキルチオ、C〜Cハロアルキルスルフィニル、C〜Cハロアルキルスルホニル、C〜Cアルキルカルボニル、C〜Cシクロアルキルカルボニル、C〜Cハロアルキルカルボニル、C〜Cハロシクロアルキルカルボニル、C〜Cアルコキシカルボニル、C〜Cハロアルコキシカルボニル、C〜Cアルキルチオカルボニル、C〜Cアルコキシチオカルボニル、C〜Cアルキルジチオカルボニル、C〜Cアルキルアミノカルボニル、C〜Cハロアルキルアミノカルボニル、ジ(C〜Cアルキル)アミノカルボニル、トリ(C〜Cアルキル)シリル、C〜Cアルキルアミノスルホニル、ジ(C〜Cアルキル)アミノスルホニル、C〜Cアルキルカルボニルオキシ、C〜Cアルキルスルホニルオキシ、C〜Cハロアルキルスルホニルオキシ、C〜Cアルキルアミノ、ジ(C〜Cアルキル)アミノ、フェニル、ナフチル、(Z)で置換されたフェニル、(Z)で置換されたナフチル又はD1−1〜D1−99を表し、
Bは、B−1〜B−34を表し、
B−1〜B−34は、以下の構造を表し、
Wherein, A 1 is, -N (-O) m2 or represents -CR 1,
R 1 , R 3 , R 4 , R 4a and R 4b are each independently a hydrogen atom, halogen atom, cyano, nitro, —OH, —SH, —NH 2 , C 1 -C 6 alkyl, R 28a . optionally substituted (C 1 ~C 6) alkyl, C 3 -C 8 cycloalkyl, optionally substituted by R 28a (C 3 ~C 8) cycloalkyl, C 2 -C 6 alkenyl, by R 28a optionally substituted (C 2 ~C 6) alkenyl, C 3 -C 8 cycloalkenyl, optionally substituted by R 28a (C 3 ~C 8) cycloalkenyl, C 2 -C 6 alkynyl, by R 28a optionally substituted (C 2 ~C 6) alkynyl, C 1 -C 6 alkoxy, C 1 -C 6 haloalkoxy, C 2 -C 6 alkenyloxy, C 1 -C 6 alkyl Thio, C 1 -C 6 alkylsulfinyl, C 1 -C 6 alkylsulfonyl, C 1 -C 6 haloalkylthio, C 1 -C 6 haloalkylsulfinyl, C 1 -C 6 haloalkylsulfonyl, C 1 -C 6 alkylcarbonyl, C 3 -C 8 cycloalkylcarbonyl, C 1 -C 6 haloalkylcarbonyl, C 3 -C 8 halocycloalkyl carbonyl, C 1 -C 6 alkoxycarbonyl, C 1 -C 6 haloalkoxycarbonyl, C 1 -C 6 alkylthio carbonyl, C 1 -C 6 alkoxythiocarbonyl, C 1 -C 6 alkyl dithio carbonyl, C 1 -C 6 alkylaminocarbonyl, C 1 -C 6 haloalkylcarbonyl aminocarbonyl, di (C 1 -C 6 alkyl) aminocarbonyl, tri (C 1 -C 6 alkyl) silyl , C 1 -C 6 alkylaminosulfonyl, di (C 1 -C 6 alkyl) aminosulfonyl, C 1 -C 6 alkylcarbonyloxy, C 1 -C 6 alkylsulfonyloxy, C 1 -C 6 haloalkylsulfonyloxy, C 1 -C 6 alkylamino, di (C 1 -C 6 alkyl) amino, phenyl, naphthyl, (Z) phenyl substituted with q, naphthyl or D1-1~D1-99 substituted with (Z) q Represent,
R 2 is a halogen atom, cyano, nitro, —OH, —SH, —NH 2 , C 1 -C 6 alkyl, (C 1 -C 6 ) alkyl optionally substituted by R 28a , C 3 -C 8. cycloalkyl, optionally substituted by an optionally substituted (C 3 ~C 8) cycloalkyl, C 2 -C 6 alkenyl, R 28a by R 28a (C 2 ~C 6) alkenyl, C 3 -C 8 cycloalkenyl, optionally substituted by R 28a (C 3 ~C 8) cycloalkenyl, C 2 -C 6 alkynyl, optionally substituted by R 28a (C 2 ~C 6) alkynyl, C 1 -C 6 alkoxy, C 1 -C 6 haloalkoxy, C 2 -C 6 alkenyloxy, C 1 -C 6 alkylthio, C 1 -C 6 alkylsulfinyl, C 1 -C 6 al Alkylsulfonyl, C 1 -C 6 haloalkylthio, C 1 -C 6 haloalkylsulfinyl, C 1 -C 6 haloalkylsulfonyl, C 1 -C 6 alkylcarbonyl, C 3 -C 8 cycloalkylcarbonyl, C 1 -C 6 haloalkyl carbonyl, C 3 -C 8 halocycloalkyl carbonyl, C 1 -C 6 alkoxycarbonyl, C 1 -C 6 haloalkoxycarbonyl, C 1 -C 6 alkylthiocarbonyl, C 1 -C 6 alkoxythiocarbonyl, C 1 -C 6 alkyl dithio carbonyl, C 1 -C 6 alkylaminocarbonyl, C 1 -C 6 haloalkylcarbonyl aminocarbonyl, di (C 1 -C 6 alkyl) aminocarbonyl, tri (C 1 -C 6 alkyl) silyl, C 1 -C 6 alkylaminosulfonyl, di (C 1 -C 6 Alkyl) aminosulfonyl, C 1 -C 6 alkylcarbonyloxy, C 1 -C 6 alkylsulfonyloxy, C 1 -C 6 haloalkylsulfonyloxy, C 1 -C 6 alkylamino, di (C 1 -C 6 alkyl) amino , phenyl, naphthyl, (Z) phenyl substituted with q, it represents naphthyl or D1-1~D1-99 substituted with (Z) q, when n represents an integer of 2 or more, each R 2 is They may be the same or different from each other,
R 3a is a hydrogen atom, cyano, nitro, —OH, —SH, —NH 2 , C 1 -C 6 alkyl, (C 1 -C 6 ) alkyl optionally substituted with R 28a , C 3 -C 8. cycloalkyl, optionally substituted by an optionally substituted (C 3 ~C 8) cycloalkyl, C 2 -C 6 alkenyl, R 28a by R 28a (C 2 ~C 6) alkenyl, C 3 -C 8 cycloalkenyl, optionally substituted by R 28a (C 3 ~C 8) cycloalkenyl, C 2 -C 6 alkynyl, optionally substituted by R 28a (C 2 ~C 6) alkynyl, C 1 -C 6 alkoxy, C 1 -C 6 haloalkoxy, C 2 -C 6 alkenyloxy, C 1 -C 6 alkylthio, C 1 -C 6 alkylsulfinyl, C 1 -C 6 alkyl Rusuruhoniru, C 1 -C 6 haloalkylthio, C 1 -C 6 haloalkylsulfinyl, C 1 -C 6 haloalkylsulfonyl, C 1 -C 6 alkylcarbonyl, C 3 -C 8 cycloalkylcarbonyl, C 1 -C 6 haloalkyl carbonyl, C 3 -C 8 halocycloalkyl carbonyl, C 1 -C 6 alkoxycarbonyl, C 1 -C 6 haloalkoxycarbonyl, C 1 -C 6 alkylthiocarbonyl, C 1 -C 6 alkoxythiocarbonyl, C 1 -C 6 alkyl dithio carbonyl, C 1 -C 6 alkylaminocarbonyl, C 1 -C 6 haloalkylcarbonyl aminocarbonyl, di (C 1 -C 6 alkyl) aminocarbonyl, tri (C 1 -C 6 alkyl) silyl, C 1 -C 6 alkylaminosulfonyl, di (C 1 -C 6 A Kill) aminosulfonyl, C 1 -C 6 alkylcarbonyloxy, C 1 -C 6 alkylsulfonyloxy, C 1 -C 6 haloalkylsulfonyloxy, C 1 -C 6 alkylamino, di (C 1 -C 6 alkyl) amino represents phenyl, naphthyl, phenyl substituted with (Z) q, a naphthyl or D1-1~D1-99 substituted with (Z) q,
B represents B-1 to B-34;
B-1 to B-34 represent the following structures:

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

明細書中
環Bの記載において、「*」は置換基「−N(R)R」との結合位置を表し、「**」は置換基「=NR」との結合位置を表し、「***」は下記に示した置換基との結合位置を表す。
In the description of ring B in the specification, “*” represents a bonding position with the substituent “—N (R a ) R b ”, “**” represents a bonding position with the substituent “═NR b ”, “***” represents a bonding position with the substituent shown below.

Figure 2015147757
Figure 2015147757

は、酸素原子又は硫黄原子を表し、
は、水素原子、シアノ、C〜C12アルキル、R5aによって任意に置換された(C〜C12)アルキル、C〜C12シクロアルキル、R5aによって任意に置換された(C〜C12)シクロアルキル、C〜C12アルケニル、R5aによって任意に置換された(C〜C12)アルケニル、C〜C12シクロアルケニル、R5aによって任意に置換された(C〜C12)シクロアルケニル、C〜C12アルキニル、R5aによって任意に置換された(C〜C12)アルキニル、、−OH、−OR6a、−SH、−S(O)r26a、−C(O)OR6a、−C(O)SR6a、−C(S)OR6a、−C(S)SR6a、−C(O)R7a、−C(S)R7a、−N(R8a)R9a、−C(O)N(R8a)R9a、−C(S)N(R8a)R9a又は−S(O)r2N(R8a)R9aを表すか、或いは、RはRと一緒になってC〜Cのアルキレン鎖又はC〜Cアルケニレン鎖を形成することにより、Rが結合する炭素原子及びRが結合する炭素原子と共に5〜8員環を形成してもよく、このときこのアルキレン鎖又はアルケニレン鎖は酸素原子、硫黄原子又は窒素原子を1又は2個含んでもよく、且つハロゲン原子、シアノ、ニトロ、C〜Cアルキル、−OH、−OR11a、−SH、−S(O)11a、オキソ基又はチオキソ基によって任意に置換されてもよく、
は、−C(O)R7b又は−C(S)R7bを表すか、或いは、RはRと一緒になって=C(Rb2)Rb3を形成してもよく、
b2は、−OR6a又は−S(O)6aを表し、
b3は、−C(=NOH)R12b、−C(=NOR11b)R12b又は−C{=NN(R13b)R14b}R12bを表し、
5aは、シアノ、C〜Cシクロアルキル、R10aによって任意に置換された(C〜C)シクロアルキル、−OR11a、−S(O)r211a、−N(R13a)R14a、−C(O)OH、−C(O)OR11a、−C(O)SR11a、−C(S)OR11a、−C(S)SR11a、−C(O)R12a、−C(S)R12a、−C(O)N(R13a)R14a、−C(S)N(R13a)R14a、−S(O)r2N(R13a)R14a、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル又はD1−1〜D1−99を表し、
6aは、水素原子、C〜Cアルキル、R10aによって任意に置換された(C〜C)アルキル、C〜Cアルケニル、R10aによって任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R10aによって任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R10aによって任意に置換された(C〜C)アルキニル、C〜Cシクロアルキル、R10aによって任意に置換された(C〜C)シクロアルキル、−S(O)r211a、−C(O)OR11a、−C(O)SR11a、−C(S)OR11a、−C(S)SR11a、−C(O)R12a、−C(S)R12a、−C(O)N(R13a)R14a、−C(S)N(R13a)R14a、−S(O)r2N(R13a)R14a、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチルを表し、
7aは、水素原子、C〜Cアルキル、R10aによって任意に置換された(C〜C)アルキル、C〜Cアルケニル、R10aによって任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R10aによって任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R10aによって任意に置換された(C〜C)アルキニル、C〜Cシクロアルキル、R10aによって任意に置換された(C〜C)シクロアルキル、−C(O)OH、−C(O)OR11a、−C(O)SR11a、−C(S)OR11a、−C(S)SR11a、−C(O)R12a、−C(S)R12a、−C(O)N(R13a)R14a、−C(S)N(R13a)R14a、−S(O)r2N(R13a)R14a、−C(=NR13a)R12a、−C(=NOH)R12a、−C(=NOR11a)R12a又は−C{=NN(R13a)R14a}R12aを表し、
7bは、−C(=NOH)R12b、−C(=NOR11b)R12b又は−C{=NN(R13b)R14b}R12bを表し、
8a及びR9aは、各々独立して水素原子、C〜Cアルキル、R10aによって任意に置換された(C〜C)アルキル、C〜Cアルケニル、R10aによって任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R10aによって任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R10aによって任意に置換された(C〜C)アルキニル、C〜Cシクロアルキル、R10aによって任意に置換された(C〜C)シクロアルキル、−OR11a、−S(O)r211a、−C(O)OR11a、−C(O)SR11a、−C(S)OR11a、−C(S)SR11a、−C(O)R12a、−C(S)R12a、−C(O)N(R13a)R14a、−C(S)N(R13a)R14a、−S(O)r2N(R13a)R14a、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル、D1−32、D1−33、D1−34又はD1−37を表すか、或いは、R8aはR9aと一緒になってC〜Cのアルキレン鎖又はC〜Cのアルケニレン鎖を形成することにより、R8a及びR9aが結合する窒素原子と共に3〜8員環を形成してもよく、このときこのアルキレン鎖又はアルケニレン鎖は酸素原子、硫黄原子又は窒素原子を1個含んでもよく、且つハロゲン原子、シアノ、C〜Cアルキル、R10aによって任意に置換された(C〜C)アルキル、C〜Cアルコキシ、C〜Cハロアルコキシ、C〜Cアルキルチオ、C〜Cハロアルキルチオ、C〜Cアルキルスルフィニル、C〜Cハロアルキルスルフィニル、C〜Cアルキルスルホニル、C〜Cハロアルキルスルホニル、フェニル、(Z)によって置換されたフェニル、オキソ基又はチオキソ基によって任意に置換されてもよく、
10aは、ハロゲン原子、シアノ、ニトロ、C〜Cシクロアルキル、C〜Cハロシクロアルキル、−OH、−OR11a、−SH、−S(O)11a又は−Si(R40a)(R40b)R40を表し、
11aは、C〜Cアルキル、R15aによって任意に置換された(C〜C)アルキル、C〜Cアルケニル、R15aによって任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R15aによって任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R15aによって任意に置換された(C〜C)アルキニル、C〜Cシクロアルキル、R15aによって任意に置換された(C〜C)シクロアルキル、−C(O)OR16a、−C(O)SR16a、−C(S)OR16a、−C(S)SR16a、−C(O)R17a、−C(S)R17a、−C(O)N(R18a)R19a、−C(S)N(R18a)R19a、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル又はD1−1〜D1−99を表し、
11bは、C〜Cアルキル、R15bによって任意に置換された(C〜C)アルキル、C〜Cアルケニル、R15bによって任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R15bによって任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R15bによって任意に置換された(C〜C)アルキニル、C〜Cシクロアルキル、R15bによって任意に置換された(C〜C)シクロアルキル、−C(O)OR16b、−C(O)SR16b、−C(S)OR16b、−C(S)SR16b、−C(O)R17b、−C(S)R17b、−C(O)N(R18b)R19b、−C(S)N(R18b)R19b、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル又はD1−1〜D1−99を表し、
12aは、水素原子、ハロゲン原子、シアノ、C〜Cアルキル、R15aによって任意に置換された(C〜C)アルキル、C〜Cアルケニル、R15aによって任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R15aによって任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R15aによって任意に置換された(C〜C)アルキニル、C〜Cシクロアルキル、R15aによって任意に置換された(C〜C)シクロアルキル、−OR16a、−S(O)r216a、−C(O)R17a、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル又はD1−1〜D1−99を表し、
12bは、水素原子、C〜Cアルキル、R15cによって任意に置換された(C〜C)アルキル、C〜Cアルケニル、R15cによって任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R15cによって任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R15cによって任意に置換された(C〜C)アルキニル、C〜Cシクロアルキル、R15cによって任意に置換された(C〜C)シクロアルキル、−OR16c、−S(O)16c、−C(O)OR16c、−C(O)SR16c、−C(S)OR16c、−C(S)SR16c、−C(O)R17c、−C(S)R17c、−C(O)N(R18c)R19c、−C(S)N(R18c)R19c、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル又はD1−1〜D1−99を表し、
13a及びR14aは、各々独立して水素原子又はC〜Cアルキルを表すか、或いは、R13aはR14aと一緒になってC〜Cのアルキレン鎖又はC〜Cのアルケニレン鎖を形成することにより、R13a及びR14aが結合する窒素原子と共に3〜8員環を形成してもよく、このときこのアルキレン鎖又はアルケニレン鎖は酸素原子、硫黄原子又は窒素原子を1個含んでもよく、且つハロゲン原子、シアノ、C〜Cアルキル、R15aによって任意に置換された(C〜C)アルキル、C〜Cアルコキシ、C〜Cハロアルコキシ、C〜Cアルキルチオ、C〜Cハロアルキルチオ、C〜Cアルキルスルフィニル、C〜Cハロアルキルスルフィニル、C〜Cアルキルスルホニル、C〜Cハロアルキルスルホニル、フェニル、(Z)によって置換されたフェニル、オキソ基又はチオキソ基によって任意に置換されてもよく、
13b及びR14bは、各々独立して水素原子、C〜Cアルキル、R15bによって任意に置換された(C〜C)アルキル、C〜Cアルケニル、R15bによって任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R15bによって任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R15bによって任意に置換された(C〜C)アルキニル、C〜Cシクロアルキル、R15bによって任意に置換された(C〜C)シクロアルキル、−S(O)16b、−C(O)OR16b、−C(O)SR16b、−C(S)OR16b、−C(S)SR16b、−C(O)R17b、−C(S)R17b、−C(O)N(R18b)R19b、−C(S)N(R18b)R19b、、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル又はD1−1〜D1−99を表すか、或いは、R13bはR14bと一緒になってC〜Cのアルキレン鎖又はC〜Cのアルケニレン鎖を形成することにより、R13b及びR14bが結合する窒素原子と共に3〜8員環を形成してもよく、このときこのアルキレン鎖又はアルケニレン鎖は酸素原子、硫黄原子又は窒素原子を1個含んでもよく、且つハロゲン原子、シアノ、C〜Cアルキル、R15bによって任意に置換された(C〜C)アルキル、C〜Cアルコキシ、C〜Cハロアルコキシ、C〜Cアルキルチオ、C〜Cハロアルキルチオ、C〜Cアルキルスルフィニル、C〜Cハロアルキルスルフィニル、C〜Cアルキルスルホニル、C〜Cハロアルキルスルホニル、フェニル、(Z)によって置換されたフェニル、オキソ基又はチオキソ基によって任意に置換されてもよく、
15aは、ハロゲン原子、シアノ、ニトロ、C〜Cシクロアルキル、C〜Cハロシクロアルキル、−OH、−OR16a、−SH、−S(O)r216a、−S(=NR18a)R16a、−S(O)(=NR18a)R16a、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル、D1−1〜D1−99又は−Si(R40a)(R40b)R40を表し、
15bは、ハロゲン原子、シアノ、ニトロ、C〜Cシクロアルキル、C〜Cハロシクロアルキル、−OH、−OR16b、−SH、−S(O)16b、−S(=NR18b)R16b、−S(O)(=NR18b)R16b、−C(O)OH、−C(O)OR16b、−C(O)R17b、−C(O)N(R18b)R19b、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル、D1−1〜D1−99又は−Si(R40a)(R40b)R40を表し、
15cは、ハロゲン原子、シアノ、ニトロ、C〜Cシクロアルキル、C〜Cハロシクロアルキル、−OH、−OR16c、−SH、−S(O)16c、−S(=NR18c)R16c、−S(O)(=NR18c)R16c、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル、D1−1〜D1−99又は−Si(R40a)(R40b)R40を表し、
16a、R16b及びR16cは、各々独立してC〜Cアルキル、C〜Cアルケニル、C〜Cアルキニル、C〜Cシクロアルキル、C〜Cシクロアルケニル、R20によって任意に置換された(C〜C)アルキル、R20によって任意に置換された(C〜C)アルケニル、R20によって任意に置換された(C〜C)アルキニル、R20によって任意に置換された(C〜C)シクロアルキル又はR20によって任意に置換された(C〜C)シクロアルケニルを表し、
17a、R17b及びR17cは、各々独立して水素原子、C〜Cアルキル又はR20によって任意に置換された(C〜C)アルキルを表し、
18a、R18b及びR18cは、各々独立して水素原子、シアノ、C〜Cアルキルを表し、
19a、R19b及びR19cは各々独立して、水素原子、C〜Cアルキル又はR20によって任意に置換された(C〜C)アルキルを表し、
20は、ハロゲン原子、シアノ、ニトロ、−OH、−SH、−NH、C〜Cシクロアルキル、C〜Cシクロアルケニル、C〜Cアルコキシ、C〜Cハロアルコキシ、C〜Cアルケニルオキシ、C〜Cアルキルチオ、C〜Cアルキルスルフィニル、C〜Cアルキルスルホニル、C〜Cハロアルキルチオ、C〜Cハロアルキルスルフィニル、C〜Cハロアルキルスルホニル、C〜Cアルキルカルボニル、C〜Cシクロアルキルカルボニル、C〜Cハロアルキルカルボニル、C〜Cハロシクロアルキルカルボニル、C〜Cアルコキシカルボニル、C〜Cハロアルコキシカルボニル、C〜Cアルキルチオカルボニル、C〜Cアルコキシチオカルボニル、C〜Cアルキルジチオカルボニル、C〜Cアルキルアミノカルボニル、C〜Cハロアルキルアミノカルボニル、ジ(C〜Cアルキル)アミノカルボニル、トリ(C〜Cアルキル)シリル、C〜Cアルキルアミノスルホニル、ジ(C〜Cアルキル)アミノスルホニル、C〜Cアルキルカルボニルオキシ、C〜Cアルキルスルホニルオキシ、C〜Cハロアルキルスルホニルオキシ、C〜Cアルキルアミノ、ジ(C〜Cアルキル)アミノ、C〜Cアルキルイミノ、C〜Cアルコキシイミノ、フェニル、ナフチル、(Z)で置換されたフェニル、(Z)で置換されたナフチル又はD1−1〜D1−99を表し、
D1−1〜D1−99は、それぞれ下記の構造で表される環を表し、
Q 1 represents an oxygen atom or a sulfur atom,
R a is a hydrogen atom, cyano, optionally substituted by C 1 -C 12 alkyl, optionally substituted by R 5a (C 1 ~C 12) alkyl, C 3 -C 12 cycloalkyl, R 5a ( C 3 -C 12) cycloalkyl, C 2 -C 12 alkenyl, optionally substituted by R 5a (C 2 ~C 12) alkenyl, C 3 -C 12 cycloalkenyl, optionally substituted by R 5a ( C 3 -C 12) cycloalkenyl, optionally substituted by C 2 -C 12 alkynyl, R 5a (C 2 ~C 12 ) alkynyl ,, - OH, -OR 6a, -SH , -S (O) r2 R6a , -C (O) OR6a , -C (O) SR6a , -C (S) OR6a , -C (S) SR6a , -C (O) R7a , -C (S) R7a , -N ( 8a) R 9a, -C (O ) N (R 8a) R 9a, or represents -C (S) N (R 8a ) R 9a or -S (O) r2 N (R 8a) R 9a, or, R a is by forming an alkylene chain or C 2 -C 5 alkenylene chain of C 2 -C 5 taken together with R 3,. 5 to together with the carbon atoms to carbon atoms and R 3 R a is attached is bound An 8-membered ring may be formed, in which case the alkylene chain or alkenylene chain may contain one or two oxygen atoms, sulfur atoms or nitrogen atoms, and is a halogen atom, cyano, nitro, C 1 -C 6 alkyl , —OH, —OR 11a , —SH, —S (O) r R 11a , an oxo group or a thioxo group,
R b represents —C (O) R 7b or —C (S) R 7b , or R b together with R a may form ═C (R b2 ) R b3 ,
R b2 represents —OR 6a or —S (O) r R 6a ,
R b3 represents -C (= NOH) R 12b , -C (= NOR 11b ) R 12b or -C {= NN (R 13b ) R 14b } R 12b ,
R 5a is cyano, C 3 -C 8 cycloalkyl, (C 3 -C 8 ) cycloalkyl optionally substituted by R 10a , —OR 11a , —S (O) r 2 R 11a , —N (R 13a ) R 14a , —C (O) OH, —C (O) OR 11a , —C (O) SR 11a , —C (S) OR 11a , —C (S) SR 11a , —C (O) R 12a , -C (S) R12a , -C (O) N ( R13a ) R14a , -C (S) N ( R13a ) R14a , -S (O) r2N ( R13a ) R14a , phenyl represents naphthyl or D1-1~D1-99 substituted phenyl which is substituted, naphthyl, the (Z) q by (Z) q,
R 6a is a hydrogen atom, C 1 -C 6 alkyl, optionally substituted by R 10a (C 1 ~C 6) alkyl, C 2 -C 6 alkenyl, optionally substituted by R 10a (C 2 ~ C 6) alkenyl, C 3 -C 8 cycloalkenyl, optionally substituted by R 10a (C 3 ~C 8) cycloalkenyl, C 2 -C 6 alkynyl, optionally substituted by R 10a (C 2 ~ C 6 ) alkynyl, C 3 -C 8 cycloalkyl, (C 3 -C 8 ) cycloalkyl optionally substituted by R 10a , —S (O) r 2 R 11a , —C (O) OR 11a , —C (O) SR 11a , -C (S) OR 11a , -C (S) SR 11a , -C (O) R 12a , -C (S) R 12a , -C (O) N (R 13a ) R 14a , -C (S) N (R 13a) R 14a, -S (O) r2 N (R 13a) R 14a, represents phenyl, phenyl, naphthyl, naphthyl substituted by (Z) q substituted by (Z) q ,
R 7a is hydrogen, C 1 -C 6 alkyl, optionally substituted by R 10a (C 1 ~C 6) alkyl, C 2 -C 6 alkenyl, optionally substituted by R 10a (C 2 ~ C 6) alkenyl, C 3 -C 8 cycloalkenyl, optionally substituted by R 10a (C 3 ~C 8) cycloalkenyl, C 2 -C 6 alkynyl, optionally substituted by R 10a (C 2 ~ C 6 ) alkynyl, C 3 -C 8 cycloalkyl, (C 3 -C 8 ) cycloalkyl optionally substituted by R 10a , —C (O) OH, —C (O) OR 11a , —C (O ) SR 11a , -C (S) OR 11a , -C (S) SR 11a , -C (O) R 12a , -C (S) R 12a , -C (O) N (R 13a ) R 14a ,- C (S) N ( 13a) R 14a, -S (O ) r2 N (R 13a) R 14a, -C (= NR 13a) R 12a, -C (= NOH) R 12a, -C (= NOR 11a) R 12a or -C {= NN (R 13a ) R 14a } R 12a
R 7b represents -C (= NOH) R 12b, -C (= NOR 11b ) R 12b or -C {= NN (R 13b ) R 14b } R 12b ,
R 8a and R 9a are each independently a hydrogen atom, C 1 -C 6 alkyl, (C 1 -C 6 ) alkyl optionally substituted with R 10a , C 2 -C 6 alkenyl, optionally with R 10a substituted (C 2 ~C 6) alkenyl, C 3 -C 8 cycloalkenyl, optionally substituted by R 10a (C 3 ~C 8) cycloalkenyl, C 2 -C 6 alkynyl, optionally by R 10a substituted (C 2 ~C 6) alkynyl, C 3 -C 8 cycloalkyl, optionally substituted by R 10a (C 3 ~C 8) cycloalkyl, -OR 11a, -S (O) r2 R 11a , -C (O) OR 11a, -C (O) SR 11a, -C (S) OR 11a, -C (S) SR 11a, -C (O) R 12a, -C (S) R 12a, - (O) N (R 13a) R 14a, -C (S) N (R 13a) R 14a, -S (O) r2 N (R 13a) R 14a, phenyl, phenyl substituted by (Z) q, Naphthyl, naphthyl substituted by (Z) q , D1-32, D1-33, D1-34 or D1-37, or R 8a together with R 9a is a C 2 -C 7 alkylene by forming a chain or alkenylene chain of C 2 -C 7, they may form a 3-8 membered ring together with the nitrogen atom to which R 8a and R 9a are bonded, the alkylene chain or alkenylene chain this time oxygen atom may contain one sulfur atom or a nitrogen atom, and a halogen atom, cyano, C 1 -C 6 alkyl, optionally substituted by R 10a (C 1 ~C 6) alkyl, C 1 -C 6 a Kokishi, C 1 -C 6 haloalkoxy, C 1 -C 6 alkylthio, C 1 -C 6 haloalkylthio, C 1 -C 6 alkylsulfinyl, C 1 -C 6 haloalkylsulfinyl, C 1 -C 6 alkylsulfonyl, C 1- C 6 haloalkylsulfonyl, phenyl, optionally substituted by phenyl, oxo group or thioxo group substituted by (Z) q ,
R 10a is a halogen atom, cyano, nitro, C 3 -C 8 cycloalkyl, C 3 -C 8 halocycloalkyl, —OH, —OR 11a , —SH, —S (O) r R 11a or —Si ( R 40a ) (R 40b ) R 40
R 11a is, C 1 -C 6 alkyl, optionally substituted by R 15a (C 1 ~C 6) alkyl, optionally substituted by C 2 -C 6 alkenyl, R 15a (C 2 ~C 6 ) alkenyl, optionally substituted by C 3 -C 8 cycloalkenyl, optionally substituted by R 15a (C 3 ~C 8) cycloalkenyl, C 2 -C 6 alkynyl, R 15a (C 2 ~C 6 ) Alkynyl, C 3 -C 8 cycloalkyl, (C 3 -C 8 ) cycloalkyl optionally substituted by R 15a , —C (O) OR 16a , —C (O) SR 16a , —C (S) OR 16a , -C (S) SR16a , -C (O) R17a , -C (S) R17a , -C (O) N ( R18a ) R19a , -C (S) N ( R18a ) R 19a Represents phenyl, naphthyl substituted by (Z) q , naphthyl substituted by (Z) q , or D1-1 to D1-99;
R 11b is, C 1 -C 6 alkyl, optionally substituted by R 15b (C 1 ~C 6) alkyl, optionally substituted by C 2 -C 6 alkenyl, R 15b (C 2 ~C 6 ) alkenyl, optionally substituted by C 3 -C 8 cycloalkenyl, optionally substituted by R 15b (C 3 ~C 8) cycloalkenyl, C 2 -C 6 alkynyl, R 15b (C 2 ~C 6 ) Alkynyl, C 3 -C 8 cycloalkyl, (C 3 -C 8 ) cycloalkyl optionally substituted by R 15b , —C (O) OR 16b , —C (O) SR 16b , —C (S) OR 16b , -C (S) SR16b , -C (O) R17b , -C (S) R17b , -C (O) N ( R18b ) R19b , -C (S) N ( R18b ) R 19b Represents phenyl, naphthyl substituted by (Z) q , naphthyl substituted by (Z) q , or D1-1 to D1-99;
R 12a represents a hydrogen atom, a halogen atom, cyano, substituted C 1 -C 6 alkyl, optionally substituted by R 15a (C 1 ~C 6) alkyl, C 2 -C 6 alkenyl, optionally by R 15a (C 2 -C 6 ) alkenyl, C 3 -C 8 cycloalkenyl, optionally substituted by R 15a (C 3 -C 8 ) cycloalkenyl, C 2 -C 6 alkynyl, optionally substituted by R 15a and (C 2 ~C 6) alkynyl, C 3 -C 8 cycloalkyl, optionally substituted by R 15a (C 3 ~C 8) cycloalkyl, -OR 16a, -S (O) r2 R 16a, - C (O) R 17a, phenyl, phenyl substituted by (Z) q, naphthyl, naphthyl, or substituted by (Z) q D1-1~D1-99 It represents,
R 12b is a hydrogen atom, C 1 -C 6 alkyl, optionally substituted by R 15c (C 1 ~C 6) alkyl, C 2 -C 6 alkenyl, optionally substituted by R 15c (C 2 ~ C 6 ) alkenyl, C 3 -C 8 cycloalkenyl, optionally substituted by R 15c (C 3 -C 8 ) cycloalkenyl, C 2 -C 6 alkynyl, optionally substituted by R 15c (C 2- C 6 ) alkynyl, C 3 -C 8 cycloalkyl, (C 3 -C 8 ) cycloalkyl optionally substituted by R 15c , —OR 16c , —S (O) r R 16c , —C (O) OR 16c , -C (O) SR16c , -C (S) OR16c , -C (S) SR16c , -C (O) R17c , -C (S) R17c , -C (O) N (R) 18c ) Represents R 19c, -C (S) N (R 18c) R 19c, phenyl, phenyl substituted by (Z) q, naphthyl, naphthyl or D1-1~D1-99 substituted by (Z) q,
R 13a and R 14a each independently represent a hydrogen atom or C 1 to C 6 alkyl, or R 13a together with R 14a is a C 2 to C 7 alkylene chain or C 2 to C 7. To form a 3- to 8-membered ring together with the nitrogen atom to which R 13a and R 14a are bonded. In this case, the alkylene chain or alkenylene chain contains an oxygen atom, a sulfur atom or a nitrogen atom. One (C 1 -C 6 ) alkyl optionally substituted by a halogen atom, cyano, C 1 -C 6 alkyl, R 15a , C 1 -C 6 alkoxy, C 1 -C 6 haloalkoxy , C 1 -C 6 alkylthio, C 1 -C 6 haloalkylthio, C 1 -C 6 alkylsulfinyl, C 1 -C 6 haloalkylsulfinyl, C 1 -C Alkylsulfonyl, C 1 -C 6 haloalkylsulfonyl, phenyl, may be optionally substituted by phenyl, oxo or thioxo group substituted by (Z) q,
R 13b and R 14b are each independently a hydrogen atom, C 1 -C 6 alkyl, (C 1 -C 6 ) alkyl optionally substituted with R 15b , C 2 -C 6 alkenyl, optionally with R 15b substituted (C 2 ~C 6) alkenyl, C 3 -C 8 cycloalkenyl, optionally substituted by R 15b (C 3 ~C 8) cycloalkenyl, C 2 -C 6 alkynyl, optionally by R 15b substituted (C 2 ~C 6) alkynyl, C 3 -C 8 cycloalkyl, optionally substituted by R 15b (C 3 ~C 8) cycloalkyl, -S (O) r R 16b , -C ( O) OR16b , -C (O) SR16b , -C (S) OR16b , -C (S) SR16b , -C (O) R17b , -C (S) R17b , -C (O) N (R 18b) R 19b, -C (S ) N (R 18b) R 19b ,, phenyl, (phenyl substituted by Z) q, naphthyl, naphthyl, or substituted by (Z) q D1-1~D1-99 or it represents, or, R 13b is by forming alkenylene chain alkylene chain or C 2 -C 7 of C 2 -C 7 together with R 14b, together with the nitrogen atom to which R 13b and R 14b are bonded A 3- to 8-membered ring may be formed, in which case the alkylene chain or alkenylene chain may contain one oxygen atom, sulfur atom or nitrogen atom, and is a halogen atom, cyano, C 1 -C 6 alkyl, R optionally substituted by 15b (C 1 ~C 6) alkyl, C 1 -C 6 alkoxy, C 1 -C 6 haloalkoxy, C 1 -C 6 alkylthio, C 1 ~ 6 haloalkylthio, C 1 -C 6 alkylsulfinyl, C 1 -C 6 haloalkylsulfinyl, C 1 -C 6 alkylsulfonyl, C 1 -C 6 haloalkylsulfonyl, phenyl, phenyl substituted by (Z) q, oxo group Or optionally substituted by a thioxo group,
R 15a is a halogen atom, cyano, nitro, C 3 -C 8 cycloalkyl, C 3 -C 8 halocycloalkyl, —OH, —OR 16a , —SH, —S (O) r 2 R 16a , —S ( = NR 18a) R 16a, -S (O) (= NR 18a) R 16a, phenyl, phenyl substituted by (Z) q, naphthyl, naphthyl substituted by (Z) q, D1-1~D1- 99 or -Si (R 40a ) (R 40b ) R 40 ,
R 15b is a halogen atom, cyano, nitro, C 3 to C 8 cycloalkyl, C 3 to C 8 halocycloalkyl, —OH, —OR 16b , —SH, —S (O) r R 16b , —S ( = NR18b ) R16b , -S (O) (= NR18b ) R16b , -C (O) OH, -C (O) OR16b , -C (O) R17b , -C (O) N ( R 18b ) R 19b , phenyl, phenyl substituted by (Z) q , naphthyl, naphthyl substituted by (Z) q , D1-1 to D1-99 or —Si (R 40a ) (R 40b ) R 40 Represents
R 15c is a halogen atom, cyano, nitro, C 3 to C 8 cycloalkyl, C 3 to C 8 halocycloalkyl, —OH, —OR 16c , —SH, —S (O) r R 16c , —S ( = NR 18c) R 16c, -S (O) (= NR 18c) R 16c, phenyl, phenyl substituted by (Z) q, naphthyl, naphthyl substituted by (Z) q, D1-1~D1- 99 or -Si (R 40a ) (R 40b ) R 40 ,
R 16a , R 16b and R 16c are each independently C 1 -C 6 alkyl, C 2 -C 6 alkenyl, C 2 -C 6 alkynyl, C 3 -C 8 cycloalkyl, C 3 -C 8 cycloalkenyl. , optionally substituted by R 20 (C 1 ~C 6) alkyl, optionally substituted by R 20 (C 2 ~C 6) alkenyl, optionally substituted by R 20 (C 2 ~C 6) It represents alkynyl, optionally substituted by R 20 (C 3 ~C 8) optionally substituted by cycloalkyl or R 20 a (C 3 ~C 8) cycloalkenyl,
R 17a , R 17b and R 17c each independently represent a hydrogen atom, C 1 -C 6 alkyl or (C 1 -C 6 ) alkyl optionally substituted with R 20 ,
R 18a , R 18b and R 18c each independently represent a hydrogen atom, cyano, C 1 -C 6 alkyl,
R 19a , R 19b and R 19c each independently represent a hydrogen atom, C 1 -C 6 alkyl or (C 1 -C 6 ) alkyl optionally substituted with R 20 ;
R 20 is a halogen atom, cyano, nitro, —OH, —SH, —NH 2 , C 3 to C 8 cycloalkyl, C 3 to C 8 cycloalkenyl, C 1 to C 6 alkoxy, C 1 to C 6 halo. alkoxy, C 2 -C 6 alkenyloxy, C 1 -C 6 alkylthio, C 1 -C 6 alkylsulfinyl, C 1 -C 6 alkylsulfonyl, C 1 -C 6 haloalkylthio, C 1 -C 6 haloalkylsulfinyl, C 1 -C 6 haloalkylsulfonyl, C 1 -C 6 alkylcarbonyl, C 3 -C 8 cycloalkylcarbonyl, C 1 -C 6 haloalkylcarbonyl, C 3 -C 8 halocycloalkyl carbonyl, C 1 -C 6 alkoxycarbonyl, C 1 -C 6 haloalkoxycarbonyl, C 1 -C 6 alkylthiocarbonyl, C 1 C 6 alkoxythiocarbonyl, C 1 -C 6 alkyl dithio carbonyl, C 1 -C 6 alkylaminocarbonyl, C 1 -C 6 haloalkylcarbonyl aminocarbonyl, di (C 1 -C 6 alkyl) aminocarbonyl, tri (C 1 ~ C 6 alkyl) silyl, C 1 -C 6 alkylaminosulfonyl, di (C 1 -C 6 alkyl) aminosulfonyl, C 1 -C 6 alkylcarbonyloxy, C 1 -C 6 alkylsulfonyloxy, C 1 -C 6 haloalkylsulfonyloxy, C 1 -C 6 alkylamino, di (C 1 -C 6 alkyl) amino, C 1 -C 6 alkylimino, C 1 -C 6 alkoxyimino, phenyl, naphthyl, substituted with (Z) q Phenyl, naphthyl substituted with (Z) q or D1-1 to D1-99,
D1-1 to D1-99 each represent a ring represented by the following structure:

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

は、ハロゲン原子、シアノ、ニトロ、−OH、−SH又はR24を表し、g1、g2又はg4が2以上の整数を表すとき、各々のXは互いに同一であっても又は互いに相異なってもよく、更に2つのXが隣接する場合には、隣接する2つのXは、−CHCHCH−、−CHCHO−、−CHOCH−、−OCHO−、−CHCHS−、−CHSCH−、−CHCHCHCH−、−CHCHCHO−、−CHCHOCH−、−CHOCHO−、−OCHCHO−、−CHCHCHS−又は−OCHCHS−を形成することにより、それぞれのXが結合する炭素原子と共に5員環又は6員環を形成してもよく、このとき環を形成する各々の炭素原子に結合した水素原子は、ハロゲン原子、C〜Cアルキル基、C〜Cハロアルキル基、C〜Cアルコキシ基、C〜Cアルキルチオ基、C〜Cアルキルスルフィニル基又はC〜Cアルキルスルホニル基によって任意に置換されてもよく、
1aは、水素原子、シアノ、−OH又はR24を表し、
1bは、ハロゲン原子、シアノ、ニトロ、−OH、−SH又はR24を表し、f1、f2、f4、f5、f6、f7、f8又はf9が2以上の整数を表すとき、各々のX1bは互いに同一であっても又は互いに相異なってもよく、さらに、2つのX1bが同一の炭素上に置換している場合、2つのX1bは一緒になってオキソ、チオキソ、イミノ、C〜Cアルキルイミノ、C〜Cアルコキシイミノ又はC〜Cアルキリデンを形成してもよく、
Zは、ハロゲン原子、シアノ、ニトロ、−OH、−SH又はR24を表し、qが2以上の整数を表すとき、各々のZは互いに同一であっても又は互いに相異なってもよく、更に2つのZが隣接する場合には、隣接する2つのZは、−CHCHCH−、−CHCHO−、−CHOCH−、−OCHO−、−CHCHS−、−CHSCH−、−CHCHCHCH−、−CHCHCHO−、−CHCHOCH−、−CHOCHO−、−OCHCHO−、−CHCHCHS−又は−OCHCHS−を形成することにより、それぞれのZが結合する炭素原子と共に5員環又は6員環を形成してもよく、このとき環を形成する各々の炭素原子に結合した水素原子は、ハロゲン原子、C〜Cアルキル基、C〜Cハロアルキル基、C〜Cアルコキシ基、C〜Cアルキルチオ基、C〜Cアルキルスルフィニル基又はC〜Cアルキルスルホニル基によって任意に置換されてもよく、
24は、C〜Cアルキル、R28によって任意に置換された(C〜C)アルキル、C〜Cシクロアルキル、R28によって任意に置換された(C〜C)シクロアルキル、C〜Cアルケニル、R28によって任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R28によって任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R28によって任意に置換された(C〜C)アルキニル、C〜Cアルコキシ、C〜Cハロアルコキシ、C〜Cアルケニルオキシ、C〜Cアルキルチオ、C〜Cアルキルスルフィニル、C〜Cアルキルスルホニル、C〜Cハロアルキルチオ、C〜Cハロアルキルスルフィニル、C〜Cハロアルキルスルホニル、C〜Cアルキルカルボニル、C〜Cシクロアルキルカルボニル、C〜Cハロアルキルカルボニル、C〜Cハロシクロアルキルカルボニル、C〜Cアルコキシカルボニル、C〜Cハロアルコキシカルボニル、C〜Cアルキルチオカルボニル、C〜Cアルコキシチオカルボニル、C〜Cアルキルジチオカルボニル、C〜Cアルキルアミノカルボニル、C〜Cハロアルキルアミノカルボニル、ジ(C〜Cアルキル)アミノカルボニル、トリ(C〜Cアルキル)シリル、C〜Cアルキルアミノスルホニル、ジ(C〜Cアルキル)アミノスルホニル、C〜Cアルキルカルボニルオキシ、C〜Cアルキルスルホニルオキシ、C〜Cハロアルキルスルホニルオキシ、C〜Cアルキルアミノ、ジ(C〜Cアルキル)アミノ、フェニル、ナフチルを表し、
28及びR28aは、各々独立してハロゲン原子、シアノ、−OH、−SH、C〜Cアルコキシ、C〜Cハロアルコキシ、C〜Cアルケニルオキシ、C〜Cアルキルチオ、C〜Cアルキルスルフィニル、C〜Cアルキルスルホニル、C〜Cハロアルキルチオ、C〜Cハロアルキルスルフィニル又はC〜Cハロアルキルスルホニルを表し、
40、R40a及びR40bは、各々独立してC〜Cアルキル、C〜Cアルコキシ又はフェニルを表し、
n、g1及びf1は、各々独立して0、1、2又は3の整数を表し、
g2及びf2は、各々独立して0、1又は2の整数を表し、
g3は、0又は1の整数を表し、
g4及びf4は、各々独立して0、1、2、3又は4の整数を表し、
f5は、0、1、2、3、4又は5の整数を表し、
f6は、0、1、2、3、4、5又は6の整数を表し、
f7は、0、1、2、3、4、5、6又は7の整数を表し、
f8は、0、1、2、3、4、5、6、7又は8の整数を表し、
f9は、0、1、2、3、4、5、6、7、8又は9の整数を表し、
qは、1、2、3、4又は5の整数を表し、
m1、m2及びm3は、各々独立して0又は1の整数を表し、
r及びr2は、各々独立して0、1又は2の整数を表す。〕で表される複素環誘導体又はその塩。
X 1 represents a halogen atom, cyano, nitro, —OH, —SH, or R 24, and when g 1, g 2, or g 4 represents an integer of 2 or more, each X 1 may be the same as or different from each other. When two X 1 are adjacent to each other, the two adjacent X 1 are —CH 2 CH 2 CH 2 —, —CH 2 CH 2 O—, —CH 2 OCH 2 —, — OCH 2 O -, - CH 2 CH 2 S -, - CH 2 SCH 2 -, - CH 2 CH 2 CH 2 CH 2 -, - CH 2 CH 2 CH 2 O -, - CH 2 CH 2 OCH 2 -, By forming —CH 2 OCH 2 O—, —OCH 2 CH 2 O—, —CH 2 CH 2 CH 2 S— or —OCH 2 CH 2 S—, together with the carbon atom to which each X 1 is attached, A member ring or a six-member ring may be formed. Hydrogen atoms bonded to each carbon atom forming the ring time, a halogen atom, C 1 -C 6 alkyl group, C 1 -C 6 haloalkyl group, C 1 -C 6 alkoxy group, C 1 -C 6 alkylthio group may be optionally substituted by C 1 -C 6 alkylsulfinyl group or a C 1 -C 6 alkylsulfonyl group,
X 1a represents a hydrogen atom, cyano, —OH or R 24 ,
X 1b represents a halogen atom, cyano, nitro, —OH, —SH or R 24, and when f1, f2, f4, f5, f6, f7, f8 or f9 represents an integer of 2 or more, each X 1b May be the same or different from each other, and when two X 1b are substituted on the same carbon, the two X 1b together are oxo, thioxo, imino, C 1 -C 6 alkylimino, may form a C 1 -C 6 alkoxyimino or C 1 -C 6 alkylidene,
Z represents a halogen atom, cyano, nitro, —OH, —SH or R 24, and when q represents an integer of 2 or more, each Z may be the same as or different from each other; If the two Z are adjacent, the two adjacent Z is, -CH 2 CH 2 CH 2 - , - CH 2 CH 2 O -, - CH 2 OCH 2 -, - OCH 2 O -, - CH 2 CH 2 S -, - CH 2 SCH 2 -, - CH 2 CH 2 CH 2 CH 2 -, - CH 2 CH 2 CH 2 O -, - CH 2 CH 2 OCH 2 -, - CH 2 OCH 2 O-, By forming —OCH 2 CH 2 O—, —CH 2 CH 2 CH 2 S— or —OCH 2 CH 2 S—, a 5-membered or 6-membered ring is formed with the carbon atom to which each Z is bonded. Each of the carbon atoms forming the ring The hydrogen atom bonded to the halogen atom, C 1 -C 6 alkyl group, C 1 -C 6 haloalkyl group, C 1 -C 6 alkoxy group, C 1 -C 6 alkylthio group, C 1 -C 6 alkylsulfinyl group Or optionally substituted by a C 1 -C 6 alkylsulfonyl group,
R 24 is optionally substituted by C 1 -C 6 alkyl, optionally substituted by R 28 (C 1 ~C 6) alkyl, C 3 -C 8 cycloalkyl, R 28 (C 3 ~C 8 ) cycloalkyl, C 2 -C 6 alkenyl, optionally substituted by R 28 (C 2 ~C 6) alkenyl, C 3 -C 8 cycloalkenyl, optionally substituted by R 28 (C 3 ~C 8 ) cycloalkenyl, C 2 -C 6 alkynyl, optionally substituted by R 28 (C 2 ~C 6) alkynyl, C 1 -C 6 alkoxy, C 1 -C 6 haloalkoxy, C 2 -C 6 alkenyloxy , C 1 -C 6 alkylthio, C 1 -C 6 alkylsulfinyl, C 1 -C 6 alkylsulfonyl, C 1 -C 6 haloalkylthio, C 1 -C 6 Haroa Kirusurufiniru, C 1 -C 6 haloalkylsulfonyl, C 1 -C 6 alkylcarbonyl, C 3 -C 8 cycloalkylcarbonyl, C 1 -C 6 haloalkylcarbonyl, C 3 -C 8 halocycloalkyl carbonyl, C 1 -C 6 alkoxycarbonyl, C 1 -C 6 haloalkoxycarbonyl, C 1 -C 6 alkylthiocarbonyl, C 1 -C 6 alkoxythiocarbonyl, C 1 -C 6 alkyldithiocarbonyl, C 1 -C 6 alkylaminocarbonyl, C 1 -C 6 haloalkylaminocarbonyl, di (C 1 -C 6 alkyl) aminocarbonyl, tri (C 1 -C 6 alkyl) silyl, C 1 -C 6 alkylaminosulfonyl, di (C 1 -C 6 alkyl) aminosulfonyl , C 1 -C 6 alkylcarbonyloxy, C 1 -C 6 alkylsulfonyloxy, C 1 -C 6 haloalkylsulfonyloxy, C 1 -C 6 alkylamino, di (C 1 -C 6 alkyl) amino, represents phenyl, naphthyl,
R 28 and R 28a are each independently a halogen atom, cyano, —OH, —SH, C 1 -C 6 alkoxy, C 1 -C 6 haloalkoxy, C 2 -C 6 alkenyloxy, C 1 -C 6. represents alkylthio, C 1 -C 6 alkylsulfinyl, C 1 -C 6 alkylsulfonyl, C 1 -C 6 haloalkylthio, a C 1 -C 6 haloalkylsulfinyl or C 1 -C 6 haloalkylsulfonyl,
R 40 , R 40a and R 40b each independently represent C 1 -C 6 alkyl, C 1 -C 6 alkoxy or phenyl;
n, g1 and f1 each independently represent an integer of 0, 1, 2 or 3;
g2 and f2 each independently represent an integer of 0, 1 or 2;
g3 represents an integer of 0 or 1,
g4 and f4 each independently represent an integer of 0, 1, 2, 3 or 4;
f5 represents an integer of 0, 1, 2, 3, 4 or 5,
f6 represents an integer of 0, 1, 2, 3, 4, 5 or 6,
f7 represents an integer of 0, 1, 2, 3, 4, 5, 6 or 7,
f8 represents an integer of 0, 1, 2, 3, 4, 5, 6, 7 or 8;
f9 represents an integer of 0, 1, 2, 3, 4, 5, 6, 7, 8 or 9,
q represents an integer of 1, 2, 3, 4 or 5;
m1, m2 and m3 each independently represent an integer of 0 or 1,
r and r2 each independently represents an integer of 0, 1 or 2. Or a salt thereof.

〔2〕
は、−CRを表し、
は、水素原子、ハロゲン原子又はC〜Cアルキル表し、
は、ハロゲン原子又はC〜Cアルキルを表す上記〔1〕記載の複素環誘導体又はその塩。
[2]
A 1 represents -CR 1
R 1 represents a hydrogen atom, a halogen atom or C 1 -C 6 alkyl,
R 2 represents a heterocyclic derivative or a salt thereof according to the above [1], wherein R 2 represents a halogen atom or C 1 -C 6 alkyl.

〔3〕
は、水素原子を表し、
は、ハロゲン原子又はC〜Cアルキルを表し、
3aは、C〜Cアルキルを表し、
、R4a及びR4bは、水素原子を表し
Bは、B−1、B−2、B−3、B−5、B−7、B−9、B−17又はB−32を表し、
は、酸素原子を表し、
は、水素原子又はC〜Cアルキルを表し、
は、−C(O)R7bを表し、
7bは、−C(=NOR11b)R12bを表し、
11bは、C〜Cアルキルを表し、
12bは、C〜Cアルキル又はR15cによって任意に置換された(C〜C)アルキルを表し、
15cは、−S(O)16cを表し、
16cは、C〜Cアルキル又はC〜Cアルケニルを表し、
nは、0を表す上記〔2〕記載の複素環誘導体又はその塩。
[3]
R 1 represents a hydrogen atom,
R 3 represents a halogen atom or C 1 -C 6 alkyl,
R 3a represents C 1 -C 6 alkyl;
R 4 , R 4a and R 4b represent a hydrogen atom. B represents B-1, B-2, B-3, B-5, B-7, B-9, B-17, or B-32. ,
Q 1 represents an oxygen atom,
R a represents a hydrogen atom or C 1 -C 6 alkyl;
R b represents -C (O) R 7b ;
R 7b represents -C (= NOR 11b ) R 12b ,
R 11b represents C 1 -C 6 alkyl,
R 12b represents C 1 -C 6 alkyl or (C 1 -C 6 ) alkyl optionally substituted with R 15c ,
R 15c represents -S (O) r R 16c ,
R 16c represents C 1 -C 6 alkyl or C 1 -C 6 alkenyl,
n is the heterocyclic derivative or a salt thereof according to the above [2], wherein n represents 0.

〔4〕
上記〔1〕〜〔3〕記載の複素環誘導体及びその塩から選ばれる1種又は2種以上を有効成分として含有する有害生物防除剤。
[4]
A pest control agent comprising one or more selected from the heterocyclic derivatives described in [1] to [3] above and salts thereof as an active ingredient.

〔5〕
上記〔1〕〜〔3〕記載の複素環誘導体及びその塩から選ばれる1種又は2種以上を有効成分として含有する農薬。
[5]
An agrochemical containing one or more selected from the heterocyclic derivatives according to the above [1] to [3] and salts thereof as an active ingredient.

〔6〕
上記〔1〕〜〔3〕記載の複素環誘導体及びその塩から選ばれる1種又は2種以上を有効成分として含有する哺乳動物又は鳥類の内部もしくは外部寄生虫防除剤。
[6]
A mammal or bird internal or ectoparasite control agent comprising one or more selected from the heterocyclic derivatives according to the above [1] to [3] and salts thereof as an active ingredient.

〔7〕
上記〔1〕〜〔3〕記載の複素環誘導体及びその塩から選ばれる1種又は2種以上を有効成分として含有する殺虫剤又は殺ダニ剤。
[7]
An insecticide or acaricide containing as an active ingredient one or more selected from the heterocyclic derivatives described in [1] to [3] above and salts thereof.

〔8〕
上記〔1〕〜〔3〕記載の複素環誘導体及びその塩から選ばれる1種又は2種以上を有効成分として含有する土壌処理剤。
[8]
The soil treatment agent which contains 1 type, or 2 or more types chosen from the heterocyclic derivative and its salt as described in said [1]-[3] as an active ingredient.

〔9〕
土壌処理方法が土壌潅注処理である上記〔8〕記載の土壌処理剤。
[9]
The soil treatment agent according to the above [8], wherein the soil treatment method is soil irrigation treatment.

本発明化合物は多くの農業害虫、ハダニ類、哺乳動物又は鳥類の内部もしくは外部寄生虫に対して優れた殺虫・殺ダニ活性を有し、既存の殺虫剤に対して抵抗性を獲得した害虫に対しても十分な防除効果を発揮する。さらに、ホ乳類、魚類及び益虫に対してほとんど悪影響を及ぼさず、低残留性で環境に対する負荷も軽い。   The compound of the present invention has excellent insecticidal / miticidal activity against many agricultural pests, spider mites, mammals or birds, or against insects that have acquired resistance to existing insecticides. Even against this, it exhibits a sufficient control effect. Furthermore, it has little adverse effect on mammals, fish and beneficial insects, has low persistence, and has a light environmental impact.

従って、本発明は有用な新規有害生物防除剤を提供することができる。   Therefore, the present invention can provide a useful novel pest control agent.

本発明に包含される化合物には、置換基の種類によってはE−体及びZ−体の幾何異性体が存在する場合があるが、本発明はこれらE−体、Z−体又はE−体及びZ−体を任意の割合で含む混合物を包含するものである。また、本発明に包含される化合物は、1個又は2個以上の不斉炭素原子の存在に起因する光学活性体が存在するが、本発明は全ての光学活性体又はラセミ体を包含する。   The compounds included in the present invention may have geometrical isomers of E-form and Z-form depending on the type of substituent, and the present invention is not limited to these E-form, Z-form or E-form. And a mixture containing the Z-form in an arbitrary ratio. In addition, the compounds included in the present invention include optically active substances resulting from the presence of one or more asymmetric carbon atoms, but the present invention includes all optically active substances or racemates.

本発明に包含される化合物のうちで、常法に従って酸付加塩にすることができるものは、例えば、フッ化水素酸、塩酸、臭化水素酸、ヨウ化水素酸等のハロゲン化水素酸の塩、硝酸、硫酸、燐酸、塩素酸、過塩素酸等の無機酸の塩、メタンスルホン酸、エタンスルホン酸、トリフルオロメタンスルホン酸、ベンゼンスルホン酸、p−トルエンスルホン酸等のスルホン酸の塩、ギ酸、酢酸、プロピオン酸、トリフルオロ酢酸、フマール酸、酒石酸、蓚酸、マレイン酸、リンゴ酸、コハク酸、安息香酸、マンデル酸、アスコルビン酸、乳酸、グルコン酸、クエン酸等のカルボン酸の塩又はグルタミン酸、アスパラギン酸等のアミノ酸の塩とすることができる。   Among the compounds included in the present invention, those that can be converted into acid addition salts according to a conventional method include, for example, hydrohalic acids such as hydrofluoric acid, hydrochloric acid, hydrobromic acid, hydroiodic acid, and the like. Salts of inorganic acids such as salts, nitric acid, sulfuric acid, phosphoric acid, chloric acid, perchloric acid, salts of sulfonic acids such as methanesulfonic acid, ethanesulfonic acid, trifluoromethanesulfonic acid, benzenesulfonic acid, p-toluenesulfonic acid, Salts of carboxylic acids such as formic acid, acetic acid, propionic acid, trifluoroacetic acid, fumaric acid, tartaric acid, succinic acid, maleic acid, malic acid, succinic acid, benzoic acid, mandelic acid, ascorbic acid, lactic acid, gluconic acid, citric acid, etc. A salt of an amino acid such as glutamic acid or aspartic acid can be used.

或いは、本発明に包含される化合物のうちで、常法に従って金属塩にすることができるものは、例えば、リチウム、ナトリウム、カリウムといったアルカリ金属の塩、カルシウム、バリウム、マグネシウムといったアルカリ土類金属の塩又はアルミニウムの塩とすることができる。   Alternatively, among the compounds included in the present invention, those that can be converted into metal salts according to conventional methods include, for example, alkali metal salts such as lithium, sodium, and potassium, and alkaline earth metals such as calcium, barium, and magnesium. It can be a salt or a salt of aluminum.

次に、本明細書において示した各置換基の具体例を以下に示す。ここで、n−はノルマル、i−はイソ、s−はセカンダリー及びtert−はターシャリーを各々意味し、Phはフェニルを意味する。   Next, specific examples of each substituent shown in the present specification are shown below. Here, n- represents normal, i- represents iso, s- represents secondary, and tert- represents tertiary, and Ph represents phenyl.

本明細書におけるハロゲン原子としては、フッ素原子、塩素原子、臭素原子及びヨウ素原子が挙げられる。尚、本明細書中「ハロ」の表記もこれらのハロゲン原子を表す。   Examples of the halogen atom in the present specification include a fluorine atom, a chlorine atom, a bromine atom and an iodine atom. In the present specification, the notation “halo” also represents these halogen atoms.

本明細書におけるC〜Cアルキルの表記は、炭素原子数がa〜b個よりなる直鎖状又は分岐鎖状の炭化水素基を表し、例えばメチル基、エチル基、n−プロピル基、i−プロピル基、n−ブチル基、i−ブチル基、s−ブチル基、tert−ブチル基、n−ペンチル基、1,1−ジメチルプロピル基、n−ヘキシル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b alkyl in the present specification represents a linear or branched hydrocarbon group having a carbon number of a to b , for example, methyl group, ethyl group, n-propyl group, Specific examples include i-propyl group, n-butyl group, i-butyl group, s-butyl group, tert-butyl group, n-pentyl group, 1,1-dimethylpropyl group, n-hexyl group, and the like. Each selected range of carbon atoms is selected.

本明細書におけるC〜Cハロアルキルの表記は、炭素原子に結合した水素原子が、ハロゲン原子によって任意に置換された、炭素原子数がa〜b個よりなる直鎖状又は分岐鎖状の炭化水素基を表し、このとき、2個以上のハロゲン原子によって置換されている場合、それらのハロゲン原子は互いに同一でも、又は互いに相異なっていてもよい。例えばフルオロメチル基、クロロメチル基、ブロモメチル基、ヨードメチル基、ジフルオロメチル基、ジクロロメチル基、トリフルオロメチル基、クロロジフルオロメチル基、トリクロロメチル基、ブロモジフルオロメチル基、2−フルオロエチル基、2−クロロエチル基、2−ブロモエチル基、2,2−ジフルオロエチル基、2,2,2−トリフルオロエチル基、2−クロロ−2,2−ジフルオロエチル基、2,2,2−トリクロロエチル基、1,1,2,2−テトラフルオロエチル基、2−クロロ−1,1,2−トリフルオロエチル基、ペンタフルオロエチル基、3,3,3−トリフルオロプロピル基、2,2,3,3,3−ペンタフルオロプロピル基、1,1,2,3,3,3−ヘキサフルオロプロピル基、ヘプタフルオロプロピル基、2,2,2−トリフルオロ−1−(トリフルオロメチル)エチル基、1,2,2,2−テトラフルオロ−1−(トリフルオロメチル)エチル基、2,2,3,3,4,4,4−ヘプタフルオロブチル基、ノナフルオロブチル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, C a -C b haloalkyl is represented by a linear or branched chain having a to b carbon atoms in which a hydrogen atom bonded to a carbon atom is optionally substituted with a halogen atom. Represents a hydrocarbon group, and when substituted by two or more halogen atoms, the halogen atoms may be the same as or different from each other. For example, fluoromethyl group, chloromethyl group, bromomethyl group, iodomethyl group, difluoromethyl group, dichloromethyl group, trifluoromethyl group, chlorodifluoromethyl group, trichloromethyl group, bromodifluoromethyl group, 2-fluoroethyl group, 2- Chloroethyl group, 2-bromoethyl group, 2,2-difluoroethyl group, 2,2,2-trifluoroethyl group, 2-chloro-2,2-difluoroethyl group, 2,2,2-trichloroethyl group, 1 , 1,2,2-tetrafluoroethyl group, 2-chloro-1,1,2-trifluoroethyl group, pentafluoroethyl group, 3,3,3-trifluoropropyl group, 2,2,3,3 , 3-pentafluoropropyl group, 1,1,2,3,3,3-hexafluoropropyl group, heptafluoropropyl group 2,2,2-trifluoro-1- (trifluoromethyl) ethyl group, 1,2,2,2-tetrafluoro-1- (trifluoromethyl) ethyl group, 2,2,3,3,4, Specific examples include 4,4-heptafluorobutyl group, nonafluorobutyl group and the like, and each is selected within the range of the number of carbon atoms designated.

本明細書におけるC〜Cシクロアルキルの表記は、炭素原子数がa〜b個よりなる環状の炭化水素基を表し、3員環から6員環までの単環又は複合環構造を形成することが出来る。また、各々の環は指定の炭素原子数の範囲でアルキル基によって任意に置換されていてもよい。例えばシクロプロピル基、1−メチルシクロプロピル基、2−メチルシクロプロピル基、2,2−ジメチルシクロプロピル基、シクロブチル基、シクロペンチル基、シクロヘキシル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, C a -C b cycloalkyl represents a cyclic hydrocarbon group having a carbon number of a to b , and forms a monocyclic or complex ring structure having 3 to 6 members. I can do it. Each ring may be optionally substituted with an alkyl group within the range of the specified number of carbon atoms. Specific examples include, for example, cyclopropyl group, 1-methylcyclopropyl group, 2-methylcyclopropyl group, 2,2-dimethylcyclopropyl group, cyclobutyl group, cyclopentyl group, cyclohexyl group and the like. Selected in a range of numbers.

本明細書におけるC〜Cハロシクロアルキルの表記は、炭素原子に結合した水素原子が、ハロゲン原子によって任意に置換された、炭素原子数がa〜b個よりなる環状の炭化水素基を表し、3員環から6員環までの単環又は複合環構造を形成することが出来る。また、各々の環は指定の炭素原子数の範囲でアルキル基によって任意に置換されていてもよく、ハロゲン原子による置換は環構造部分であっても、側鎖部分であっても、或いはそれらの両方であってもよく、さらに、2個以上のハロゲン原子によって置換されている場合、それらのハロゲン原子は互いに同一でも、又は互いに相異なっていてもよい。例えば2,2−ジフルオロシクロプロピル基、2,2−ジクロロシクロプロピル基、2,2−ジブロモシクロプロピル基、2,2−ジフルオロ−1−メチルシクロプロピル基、2,2−ジクロロ−1−メチルシクロプロピル基、2,2−ジブロモ−1−メチルシクロプロピル基、2,2,3,3−テトラフルオロシクロブチル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, C a -C b halocycloalkyl is a cyclic hydrocarbon group having a carbon number of a to b in which a hydrogen atom bonded to a carbon atom is optionally substituted with a halogen atom. And can form monocyclic or complex ring structures from 3 to 6-membered rings. Each ring may be optionally substituted with an alkyl group within the range of the specified number of carbon atoms, and the substitution with a halogen atom may be a ring structure part, a side chain part, They may be both, and when they are substituted by two or more halogen atoms, the halogen atoms may be the same as or different from each other. For example, 2,2-difluorocyclopropyl group, 2,2-dichlorocyclopropyl group, 2,2-dibromocyclopropyl group, 2,2-difluoro-1-methylcyclopropyl group, 2,2-dichloro-1-methyl Specific examples include cyclopropyl group, 2,2-dibromo-1-methylcyclopropyl group, 2,2,3,3-tetrafluorocyclobutyl group, and the like, and each is selected within the range of the designated number of carbon atoms. The

本明細書におけるC〜Cアルケニルの表記は、炭素原子数がa〜b個よりなる直鎖状又は分岐鎖状で、且つ分子内に1個又は2個以上の二重結合を有する不飽和炭化水素基を表し、例えばビニル基、1−プロペニル基、2−プロペニル基、1−メチルエテニル基、2−ブテニル基、2−メチル−2−プロペニル基、3−メチル−2−ブテニル基、1,1−ジメチル−2−プロペニル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, C a -C b alkenyl is a linear or branched chain composed of a to b carbon atoms and has one or more double bonds in the molecule. Represents a saturated hydrocarbon group, for example, vinyl group, 1-propenyl group, 2-propenyl group, 1-methylethenyl group, 2-butenyl group, 2-methyl-2-propenyl group, 3-methyl-2-butenyl group, 1 , 1-dimethyl-2-propenyl group and the like are listed as specific examples, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるC〜Cハロアルケニルの表記は、炭素原子に結合した水素原子が、ハロゲン原子によって任意に置換された、炭素原子数がa〜b個よりなる直鎖状又は分岐鎖状で、且つ分子内に1個又は2個以上の二重結合を有する不飽和炭化水素基を表す。このとき、2個以上のハロゲン原子によって置換されている場合、それらのハロゲン原子は互いに同一でも、又は互いに相異なっていてもよい。例えば2,2−ジクロロビニル基、2−フルオロ−2−プロペニル基、2−クロロ−2−プロペニル基、3−クロロ−2−プロペニル基、2−ブロモ−2−プロペニル基、3,3−ジフルオロ−2−プロペニル基、2,3−ジクロロ−2−プロペニル基、3,3−ジクロロ−2−プロペニル基、2,3,3−トリフルオロ−2−プロペニル基、2,3,3−トリクロロ−2−プロペニル基、1−(トリフルオロメチル)エテニル基、4,4−ジフルオロ−3−ブテニル基、3,4,4−トリフルオロ−3−ブテニル基、3−クロロ−4,4,4−トリフルオロ−2−ブテニル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, C a -C b haloalkenyl is a linear or branched chain in which a hydrogen atom bonded to a carbon atom is optionally substituted with a halogen atom, and the number of carbon atoms is ab. And an unsaturated hydrocarbon group having one or more double bonds in the molecule. At this time, when substituted by two or more halogen atoms, these halogen atoms may be the same as or different from each other. For example, 2,2-dichlorovinyl group, 2-fluoro-2-propenyl group, 2-chloro-2-propenyl group, 3-chloro-2-propenyl group, 2-bromo-2-propenyl group, 3,3-difluoro -2-propenyl group, 2,3-dichloro-2-propenyl group, 3,3-dichloro-2-propenyl group, 2,3,3-trifluoro-2-propenyl group, 2,3,3-trichloro- 2-propenyl group, 1- (trifluoromethyl) ethenyl group, 4,4-difluoro-3-butenyl group, 3,4,4-trifluoro-3-butenyl group, 3-chloro-4,4,4- Specific examples include a trifluoro-2-butenyl group and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるC〜Cシクロアルケニルの表記は、炭素原子数がa〜b個よりなる環状の、且つ1個又は2個以上の二重結合を有する不飽和炭化水素基を表し、3員環から6員環までの単環又は複合環構造を形成することが出来る。また、各々の環は指定の炭素原子数の範囲でアルキル基によって任意に置換されていてもよく、さらに、二重結合はendo−又はexo−のどちらの形式であってもよい。例えば1−シクロペンテン−1−イル基、2−シクロペンテン−1−イル基、1−シクロヘキセン−1−イル基、2−シクロヘキセン−1−イル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b cycloalkenyl in the present specification represents a cyclic unsaturated hydrocarbon group having 1 to 2 carbon atoms and having 1 or 2 or more double bonds. A monocyclic or complex ring structure from a member ring to a 6-member ring can be formed. Each ring may be optionally substituted with an alkyl group within the range of the specified number of carbon atoms, and the double bond may be either endo- or exo-. Specific examples include 1-cyclopenten-1-yl group, 2-cyclopenten-1-yl group, 1-cyclohexen-1-yl group, 2-cyclohexen-1-yl group, and the like. Selected in a range of numbers.

本明細書におけるC〜Cアルキリデンの表記は、炭素原子数がa〜b個よりなる直鎖状又は分岐鎖状で、二重結合によって結合した炭化水素基を表し、例えばメチリデン基、エチリデン基、プロピリデン基、1−メチルエチリデン基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, C a -C b alkylidene represents a linear or branched hydrocarbon group having a carbon number of a to b and bonded by a double bond, such as a methylidene group or an ethylidene group. Specific examples include a group, a propylidene group, a 1-methylethylidene group, and the like, and each group is selected within the range of the designated number of carbon atoms.

本明細書におけるC〜Cアルキニルの表記は、炭素原子数がa〜b個よりなる直鎖状又は分岐鎖状で、且つ分子内に1個又は2個以上の三重結合を有する不飽和炭化水素基を表し、例えばエチニル基、1−プロピニル基、2−プロピニル基、1−ブチニル基、2−ブチニル基、3−ブチニル基、1,1−ジメチル−2−プロピニル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, C a -C b alkynyl is a linear or branched chain composed of a to b carbon atoms and has one or more triple bonds in the molecule. Represents a hydrocarbon group, for example, ethynyl group, 1-propynyl group, 2-propynyl group, 1-butynyl group, 2-butynyl group, 3-butynyl group, 1,1-dimethyl-2-propynyl group, etc. Each of which is selected for each specified number of carbon atoms.

本明細書におけるC〜Cハロアルキニルの表記は、炭素原子に結合した水素原子が、ハロゲン原子によって任意に置換された、炭素原子数がa〜b個よりなる直鎖状又は分岐鎖状で、且つ分子内に1個又は2個以上の三重結合を有する不飽和炭化水素基を表す。このとき、2個以上のハロゲン原子によって置換されている場合、それらのハロゲン原子は互いに同一でも、又は互いに相異なっていてもよい。例えば2−クロロエチニル基、2−ブロモエチニル基、2−ヨードエチニル基、3−クロロ−2−プロピニル基、3−ブロモ−2−プロピニル基、3−ヨード−2−プロピニル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, C a -C b haloalkynyl represents a linear or branched chain in which a hydrogen atom bonded to a carbon atom is optionally substituted with a halogen atom, and the number of carbon atoms is a to b. And an unsaturated hydrocarbon group having one or more triple bonds in the molecule. At this time, when substituted by two or more halogen atoms, these halogen atoms may be the same as or different from each other. Specific examples include 2-chloroethynyl group, 2-bromoethynyl group, 2-iodoethynyl group, 3-chloro-2-propynyl group, 3-bromo-2-propynyl group, 3-iodo-2-propynyl group and the like. Each of which is selected for each specified number of carbon atoms.

本明細書におけるC〜Cアルコキシの表記は、炭素原子数がa〜b個よりなる前記の意味であるアルキル−O−基を表し、例えばメトキシ基、エトキシ基、n−プロピルオキシ基、i−プロピルオキシ基、n−ブチルオキシ基、i−ブチルオキシ基、s−ブチルオキシ基、tert−ブチルオキシ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b alkoxy in the present specification represents an alkyl-O— group having the above-mentioned meaning consisting of a to b carbon atoms, for example, methoxy group, ethoxy group, n-propyloxy group, Specific examples include an i-propyloxy group, an n-butyloxy group, an i-butyloxy group, an s-butyloxy group, a tert-butyloxy group, and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるC〜Cハロアルコキシの表記は、炭素原子数がa〜b個よりなる前記の意味であるハロアルキル−O−基を表し、例えばジフルオロメトキシ基、トリフルオロメトキシ基、クロロジフルオロメトキシ基、ブロモジフルオロメトキシ基、2−フルオロエトキシ基、2−クロロエトキシ基、2,2,2−トリフルオロエトキシ基、1,1,2,2,−テトラフルオロエトキシ基、2−クロロ−1,1,2−トリフルオロエトキシ基、1,1,2,3,3,3−ヘキサフルオロプロピルオキシ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b haloalkoxy in the present specification represents a haloalkyl-O— group having the above-mentioned meaning consisting of a to b carbon atoms, for example, difluoromethoxy group, trifluoromethoxy group, chlorodifluoro Methoxy group, bromodifluoromethoxy group, 2-fluoroethoxy group, 2-chloroethoxy group, 2,2,2-trifluoroethoxy group, 1,1,2,2, -tetrafluoroethoxy group, 2-chloro-1 Specific examples include 1,2,2-trifluoroethoxy group, 1,1,2,3,3,3-hexafluoropropyloxy group and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるC〜Cアルケニルオキシの表記は、炭素原子数がa〜b個よりなる前記の意味であるアルケニル−O−基を表し、例えば2−プロペニルオキシ基、2−ブテニルオキシ基、2−メチル−2−プロペニルオキシ基、3−メチル−2−ブテニルオキシ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b alkenyloxy in the present specification represents an alkenyl-O— group having the above-mentioned meaning consisting of a to b carbon atoms, for example, 2-propenyloxy group, 2-butenyloxy group, Specific examples include 2-methyl-2-propenyloxy group, 3-methyl-2-butenyloxy group and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるC〜Cアルキルチオの表記は、炭素原子数がa〜b個よりなる前記の意味であるアルキル−S−基を表し、例えばメチルチオ基、エチルチオ基、n−プロピルチオ基、i−プロピルチオ基、n−ブチルチオ基、i−ブチルチオ基、s−ブチルチオ基、tert−ブチルチオ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b alkylthio in the present specification represents an alkyl-S-group having the above-mentioned meaning consisting of a to b carbon atoms, for example, methylthio group, ethylthio group, n-propylthio group, i Specific examples include -propylthio group, n-butylthio group, i-butylthio group, s-butylthio group, tert-butylthio group and the like, which are selected within the range of the number of carbon atoms specified.

本明細書におけるC〜Cハロアルキルチオの表記は、炭素原子数がa〜b個よりなる前記の意味であるハロアルキル−S−基を表し、例えばジフルオロメチルチオ基、トリフルオロメチルチオ基、クロロジフルオロメチルチオ基、ブロモジフルオロメチルチオ基、2,2,2−トリフルオロエチルチオ基、1,1,2,2−テトラフルオロエチルチオ基、2−クロロ−1,1,2−トリフルオロエチルチオ基、ペンタフルオロエチルチオ基、1,1,2,3,3,3−ヘキサフルオロプロピルチオ基、ヘプタフルオロプロピルチオ基、1,2,2,2−テトラフルオロ−1−(トリフルオロメチル)エチルチオ基、ノナフルオロブチルチオ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b haloalkylthio in the present specification represents a haloalkyl-S— group having the above-mentioned meaning consisting of a to b carbon atoms, for example, difluoromethylthio group, trifluoromethylthio group, chlorodifluoro Methylthio group, bromodifluoromethylthio group, 2,2,2-trifluoroethylthio group, 1,1,2,2-tetrafluoroethylthio group, 2-chloro-1,1,2-trifluoroethylthio group, Pentafluoroethylthio group, 1,1,2,3,3,3-hexafluoropropylthio group, heptafluoropropylthio group, 1,2,2,2-tetrafluoro-1- (trifluoromethyl) ethylthio group , Nonafluorobutylthio group and the like are given as specific examples, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるC〜Cアルキルスルフィニルの表記は、炭素原子数がa〜b個よりなる前記の意味であるアルキル−S(O)−基を表し、例えばメチルスルフィニル基、エチルスルフィニル基、n−プロピルスルフィニル基、i−プロピルスルフィニル基、n−ブチルスルフィニル基、i−ブチルスルフィニル基、s−ブチルスルフィニル基、tert−ブチルスルフィニル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b alkylsulfinyl in the present specification represents an alkyl-S (O) -group having the above-mentioned meaning consisting of a to b carbon atoms, for example, methylsulfinyl group, ethylsulfinyl group, Specific examples include n-propylsulfinyl group, i-propylsulfinyl group, n-butylsulfinyl group, i-butylsulfinyl group, s-butylsulfinyl group, tert-butylsulfinyl group and the like. The range is selected.

本明細書におけるC〜Cハロアルキルスルフィニルの表記は、炭素原子数がa〜b個よりなる前記の意味であるハロアルキル−S(O)−基を表し、例えばジフルオロメチルスルフィニル基、トリフルオロメチルスルフィニル基、クロロジフルオロメチルスルフィニル基、ブロモジフルオロメチルスルフィニル基、2,2,2−トリフルオロエチルスルフィニル基、1,2,2,2−テトラフルオロ−1−(トリフルオロメチル)エチルスルフィニル基、ノナフルオロブチルスルフィニル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, the expression C a -C b haloalkylsulfinyl represents a haloalkyl-S (O) -group having the above-mentioned meaning consisting of a to b carbon atoms, for example, difluoromethylsulfinyl group, trifluoromethyl Sulfinyl group, chlorodifluoromethylsulfinyl group, bromodifluoromethylsulfinyl group, 2,2,2-trifluoroethylsulfinyl group, 1,2,2,2-tetrafluoro-1- (trifluoromethyl) ethylsulfinyl group, nona Specific examples include a fluorobutylsulfinyl group and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるC〜Cアルキルスルホニルの表記は、炭素原子数がa〜b個よりなる前記の意味であるアルキル−SO−基を表し、例えばメチルスルホニル基、エチルスルホニル基、n−プロピルスルホニル基、i−プロピルスルホニル基、n−ブチルスルホニル基、i−ブチルスルホニル基、s−ブチルスルホニル基、tert−ブチルスルホニル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b alkylsulfonyl in the present specification represents an alkyl-SO 2 -group having the above-mentioned meaning consisting of a to b carbon atoms, for example, methylsulfonyl group, ethylsulfonyl group, n- Specific examples include a propylsulfonyl group, an i-propylsulfonyl group, an n-butylsulfonyl group, an i-butylsulfonyl group, an s-butylsulfonyl group, a tert-butylsulfonyl group, and the range of each designated number of carbon atoms. Selected.

本明細書におけるC〜Cハロアルキルスルホニルの表記は、炭素原子数がa〜b個よりなる前記の意味であるハロアルキル−SO−基を表し、例えばジフルオロメチルスルホニル基、トリフルオロメチルスルホニル基、クロロジフルオロメチルスルホニル基、ブロモジフルオロメチルスルホニル基、2,2,2−トリフルオロエチルスルホニル基、1,1,2,2−テトラフルオロエチルスルホニル基、2−クロロ−1,1,2−トリフルオロエチルスルホニル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b haloalkylsulfonyl in the present specification represents a haloalkyl-SO 2 -group having the above-mentioned meaning consisting of a to b carbon atoms, such as a difluoromethylsulfonyl group or a trifluoromethylsulfonyl group. Chlorodifluoromethylsulfonyl group, bromodifluoromethylsulfonyl group, 2,2,2-trifluoroethylsulfonyl group, 1,1,2,2-tetrafluoroethylsulfonyl group, 2-chloro-1,1,2-trimethyl Specific examples include a fluoroethylsulfonyl group and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるC〜Cアルキルアミノの表記は、水素原子の一方が炭素原子数がa〜b個よりなる前記の意味であるアルキル基によって置換されたアミノ基を表し、例えばメチルアミノ基、エチルアミノ基、n−プロピルアミノ基、i−プロピルアミノ基、n−ブチルアミノ基、i−ブチルアミノ基、tert−ブチルアミノ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b alkylamino in the present specification represents an amino group in which one of the hydrogen atoms is substituted with an alkyl group having the above-mentioned meaning consisting of a to b carbon atoms, for example, a methylamino group , Ethylamino group, n-propylamino group, i-propylamino group, n-butylamino group, i-butylamino group, tert-butylamino group and the like. Selected by range.

本明細書におけるジ(C〜Cアルキル)アミノの表記は、水素原子が両方とも、それぞれ同一でも又は互いに相異なっていてもよい炭素原子数がa〜b個よりなる前記の意味であるアルキル基によって置換されたアミノ基を表し、例えばジメチルアミノ基、エチル(メチル)アミノ基、ジエチルアミノ基、n−プロピル(メチル)アミノ基、i−プロピル(メチル)アミノ基、ジ(n−プロピル)アミノ基、ジ(n−ブチル)アミノ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, the notation of di (C a -C b alkyl) amino has the above-mentioned meaning that the number of carbon atoms which may be the same or different from each other is ab. Represents an amino group substituted by an alkyl group, such as dimethylamino group, ethyl (methyl) amino group, diethylamino group, n-propyl (methyl) amino group, i-propyl (methyl) amino group, di (n-propyl) Specific examples include an amino group, a di (n-butyl) amino group, and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるC〜Cアルキルイミノの表記は、炭素原子数がa〜b個よりなる前記の意味であるアルキル−N=基を表し、例えばメチルイミノ基、エチルイミノ基、n−プロピルイミノ基、i−プロピルイミノ基、n−ブチルイミノ基、i−ブチルイミノ基、s−ブチルイミノ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b alkylimino in the present specification represents an alkyl-N = group having the above-mentioned meaning consisting of a to b carbon atoms, for example, methylimino group, ethylimino group, n-propylimino group. Specific examples include i-propylimino group, n-butylimino group, i-butylimino group, s-butylimino group, and the like, and each is selected within the range of the number of carbon atoms designated.

本明細書におけるC〜Cアルコキシイミノの表記は、炭素原子数がa〜b個よりなる前記の意味であるアルコキシ−N=基を表し、例えばメトキシイミノ基、エトキシイミノ基、n−プロピルオキシイミノ基、i−プロピルオキシイミノ基、n−ブチルオキシイミノ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b alkoxyimino in the present specification represents an alkoxy-N = group having the above-mentioned meaning consisting of a to b carbon atoms, for example, methoxyimino group, ethoxyimino group, n-propyl. Specific examples include an oxyimino group, an i-propyloxyimino group, an n-butyloxyimino group, and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるC〜Cアルキルカルボニルの表記は、炭素原子数がa〜b個よりなる前記の意味であるアルキル−C(O)−基を表し、例えばアセチル基、プロピオニル基、ブチリル基、イソブチリル基、バレリル基、イソバレリル基、2−メチルブタノイル基、ピバロイル基、ヘキサノイル基、ヘプタノイル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b alkylcarbonyl in the present specification represents an alkyl-C (O) -group having the above-mentioned meaning consisting of a to b carbon atoms, for example, acetyl group, propionyl group, butyryl group. , Isobutyryl group, valeryl group, isovaleryl group, 2-methylbutanoyl group, pivaloyl group, hexanoyl group, heptanoyl group, and the like, and specific examples thereof are selected within the range of the number of carbon atoms designated.

本明細書におけるC〜Cハロアルキルカルボニルの表記は、炭素原子数がa〜b個よりなる前記の意味であるハロアルキル−C(O)−基を表し、例えばフルオロアセチル基、クロロアセチル基、ジフルオロアセチル基、ジクロロアセチル基、トリフルオロアセチル基、クロロジフルオロアセチル基、ブロモジフルオロアセチル基、トリクロロアセチル基、ペンタフルオロプロピオニル基、ヘプタフルオロブタノイル基、3−クロロ−2,2−ジメチルプロパノイル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b haloalkylcarbonyl in the present specification represents a haloalkyl-C (O) -group having the above-mentioned meaning consisting of a to b carbon atoms, such as a fluoroacetyl group, a chloroacetyl group, Difluoroacetyl group, dichloroacetyl group, trifluoroacetyl group, chlorodifluoroacetyl group, bromodifluoroacetyl group, trichloroacetyl group, pentafluoropropionyl group, heptafluorobutanoyl group, 3-chloro-2,2-dimethylpropanoyl group Etc. are given as specific examples, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるC〜Cシクロアルキルカルボニルの表記は、炭素原子数がa〜b個よりなる前記の意味であるシクロアルキル−C(O)−基を表し、例えばシクロプロピルカルボニル基、2−メチルシクロプロピルカルボニル基、シクロブチルカルボニル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b cycloalkylcarbonyl in the present specification represents a cycloalkyl-C (O) -group having the above-mentioned meaning consisting of a to b carbon atoms, such as cyclopropylcarbonyl group, 2 Specific examples include -methylcyclopropylcarbonyl group, cyclobutylcarbonyl group, etc., and each is selected within the range of the designated number of carbon atoms.

本明細書におけるC〜Cハロシクロアルキルカルボニルの表記は、炭素原子数がa〜b個よりなる前記の意味であるハロシクロアルキル−C(O)−基を表し、例えば2,2−ジクロロシクロプロピルカルボニル基、2,2−ジクロロ−1−メチルシクロプロピルカルボニル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, the expression C a -C b halocycloalkylcarbonyl represents a halocycloalkyl-C (O) — group having the above-mentioned meaning consisting of a to b carbon atoms. Specific examples include a dichlorocyclopropylcarbonyl group, a 2,2-dichloro-1-methylcyclopropylcarbonyl group, and the like, which are selected in the range of the designated number of carbon atoms.

本明細書におけるC〜Cアルコキシカルボニルの表記は、炭素原子数がa〜b個よりなる前記の意味であるアルキル−O−C(O)−基を表し、例えばメトキシカルボニル基、エトキシカルボニル基、n−プロピルオキシカルボニル基、i−プロピルオキシカルボニル基、n−ブトキシカルボニル基、i−ブトキシカルボニル基、tert−ブトキシカルボニル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b alkoxycarbonyl in the present specification represents an alkyl-O—C (O) — group having the above-mentioned meaning consisting of a to b carbon atoms, for example, methoxycarbonyl group, ethoxycarbonyl Group, n-propyloxycarbonyl group, i-propyloxycarbonyl group, n-butoxycarbonyl group, i-butoxycarbonyl group, tert-butoxycarbonyl group and the like, and specific ranges of the number of carbon atoms are designated. Selected.

本明細書におけるC〜Cハロアルコキシカルボニルの表記は、炭素原子数がa〜b個よりなる前記の意味であるハロアルキル−O−C(O)−基を表し、例えばクロロメトキシカルボニル基、2−クロロエトキシカルボニル基、2,2−ジフルオロエトキシカルボニル基、2,2,2−トリフルオロエトキシカルボニル基、2,2,2−トリクロロエトキシカルボニル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b haloalkoxycarbonyl in the present specification represents a haloalkyl-O—C (O) — group having the above-mentioned meaning consisting of a to b carbon atoms, such as a chloromethoxycarbonyl group, Specific examples include 2-chloroethoxycarbonyl group, 2,2-difluoroethoxycarbonyl group, 2,2,2-trifluoroethoxycarbonyl group, 2,2,2-trichloroethoxycarbonyl group, and the like. Selected in the range of the number of carbon atoms.

本明細書におけるC〜Cアルキルチオカルボニルの表記は、炭素原子数がa〜b個よりなる前記の意味であるアルキル−S−C(O)−基を表し、例えばメチルチオ−C(O)−基、エチルチオ−C(O)−基、n−プロピルチオ−C(O)−基、i−プロピルチオ−C(O)−基、n−ブチルチオ−C(O)−基、i−ブチルチオ−C(O)−基、tert−ブチルチオ−C(O)−基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b alkylthiocarbonyl in the present specification represents an alkyl-S—C (O) — group having the above meaning consisting of a to b carbon atoms, for example, methylthio-C (O) -Group, ethylthio-C (O)-group, n-propylthio-C (O)-group, i-propylthio-C (O)-group, n-butylthio-C (O)-group, i-butylthio-C Specific examples include (O) -group, tert-butylthio-C (O) -group, etc., and each is selected within the range of the designated number of carbon atoms.

本明細書におけるC〜Cアルコキシチオカルボニルの表記は、炭素原子数がa〜b個よりなる前記の意味であるアルキル−O−C(S)−基を表し、例えばメトキシ−C(S)−基、エトキシ−C(S)−基、n−プロピルオキシ−C(S)−基、i−プロピルオキシ−C(S)−基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, the expression C a -C b alkoxythiocarbonyl represents an alkyl-O—C (S) — group having the above-mentioned meaning consisting of a to b carbon atoms, for example, methoxy-C (S ) -Group, ethoxy-C (S) -group, n-propyloxy-C (S) -group, i-propyloxy-C (S) -group, etc. Selected in a range of numbers.

本明細書におけるC〜Cアルキルジチオカルボニルの表記は、炭素原子数がa〜b個よりなる前記の意味であるアルキル−S−C(S)−基を表し、例えばメチルチオ−C(S)−基、エチルチオ−C(S)−基、n−プロピルチオ−C(S)−基、i−プロピルチオ−C(S)−基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b alkyldithiocarbonyl in the present specification represents an alkyl-S—C (S) — group having the above-mentioned meaning consisting of a to b carbon atoms, for example, methylthio-C (S ) -Group, ethylthio-C (S) -group, n-propylthio-C (S) -group, i-propylthio-C (S) -group and the like. Selected by range.

本明細書におけるC〜Cアルキルアミノスルホニルの表記は、水素原子の一方が炭素原子数がa〜b個よりなる前記の意味であるアルキル基によって置換されたスルファモイル基を表し、例えばメチルスルファモイル基、エチルスルファモイル基、n−プロピルスルファモイル基、i−プロピルスルファモイル基、n−ブチルスルファモイル基、i−ブチルスルファモイル基、s−ブチルスルファモイル基、tert−ブチルスルファモイル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, C a -C b alkylaminosulfonyl represents a sulfamoyl group in which one of the hydrogen atoms is substituted with an alkyl group having the above-mentioned meaning consisting of a to b carbon atoms. Famoyl group, ethylsulfamoyl group, n-propylsulfamoyl group, i-propylsulfamoyl group, n-butylsulfamoyl group, i-butylsulfamoyl group, s-butylsulfamoyl group, Specific examples include a tert-butylsulfamoyl group and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるジ(C〜Cアルキル)アミノスルホニルの表記は、水素原子が両方とも、それぞれ同一でも又は互いに相異なっていてもよい炭素原子数がa〜b個よりなる前記の意味であるアルキル基によって置換されたスルファモイル基を表し、例えばN,N−ジメチルスルファモイル基、N−エチル−N−メチルスルファモイル基、N,N−ジエチルスルファモイル基、N,N−ジ(n−プロピル)スルファモイル基、N,N−ジ(n−ブチル)スルファモイル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, the notation of di (C a -C b alkyl) aminosulfonyl means in the above meaning that the number of carbon atoms which may be the same or different from each other is a to b. Represents a sulfamoyl group substituted by an alkyl group, such as N, N-dimethylsulfamoyl group, N-ethyl-N-methylsulfamoyl group, N, N-diethylsulfamoyl group, N, N-di- Specific examples include (n-propyl) sulfamoyl group, N, N-di (n-butyl) sulfamoyl group and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるC〜Cアルキルアミノカルボニルの表記は、水素原子の一方が炭素原子数がa〜b個よりなる前記の意味であるアルキル基によって置換されたカルバモイル基を表し、例えばメチルカルバモイル基、エチルカルバモイル基、n−プロピルカルバモイル基、i−プロピルカルバモイル基、n−ブチルカルバモイル基、i−ブチルカルバモイル基、s−ブチルカルバモイル基、tert−ブチルカルバモイル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b alkylaminocarbonyl in the present specification represents a carbamoyl group in which one of the hydrogen atoms is substituted with an alkyl group having the above-mentioned meaning consisting of a to b carbon atoms, for example, methylcarbamoyl Group, ethylcarbamoyl group, n-propylcarbamoyl group, i-propylcarbamoyl group, n-butylcarbamoyl group, i-butylcarbamoyl group, s-butylcarbamoyl group, tert-butylcarbamoyl group, etc. Is selected within the range of the specified number of carbon atoms.

本明細書におけるジ(C〜Cアルキル)アミノカルボニルの表記は、水素原子が両方とも、それぞれ同一でも又は互いに相異なっていてもよい炭素原子数がa〜b個よりなる前記の意味であるアルキル基によって置換されたカルバモイル基を表し、例えばN,N−ジメチルカルバモイル基、N−エチル−N−メチルカルバモイル基、N,N−ジエチルカルバモイル基、N,N−ジ(n−プロピル)カルバモイル基、N,N−ジ(n−ブチル)カルバモイル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, the notation of di (C a -C b alkyl) aminocarbonyl means in the above meaning that the number of carbon atoms which may be the same or different from each other is a to b. Represents a carbamoyl group substituted by an alkyl group, such as N, N-dimethylcarbamoyl group, N-ethyl-N-methylcarbamoyl group, N, N-diethylcarbamoyl group, N, N-di (n-propyl) carbamoyl Specific examples include a group, an N, N-di (n-butyl) carbamoyl group, and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるC〜Cハロアルキルアミノカルボニルの表記は、水素原子の一方が炭素原子数a〜b個よりなる前記の意味であるハロアルキル基によって置換されたカルバモイル基を表し、例えば2−フルオロエチルカルバモイル基、2−クロロエチルカルバモイル基、2,2−ジフルオロエチルカルバモイル基、2,2,2−トリフルオロエチルカルバモイル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, the expression C a -C b haloalkylaminocarbonyl represents a carbamoyl group in which one of the hydrogen atoms is substituted with a haloalkyl group having the above-described meaning consisting of a to b carbon atoms, for example, 2-fluoro Specific examples include ethylcarbamoyl group, 2-chloroethylcarbamoyl group, 2,2-difluoroethylcarbamoyl group, 2,2,2-trifluoroethylcarbamoyl group, etc. Is done.

本明細書におけるトリ(C〜Cアルキル)シリルの表記は、それぞれ同一でも又は互いに相異なっていてもよい炭素原子数がa〜b個よりなる前記の意味であるアルキル基によって置換されたシリル基を表し、例えばトリメチルシリル基、トリエチルシリル基、トリ(n−プロピル)シリル基、エチルジメチルシリル基、n−プロピルジメチルシリル基、n−ブチルジメチルシリル基、i−ブチルジメチルシリル基、tert−ブチルジメチルシリル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, the notation of tri (C a -C b alkyl) silyl is substituted by an alkyl group having the above-mentioned meanings, each having the same or different number of carbon atoms. Represents a silyl group, for example, trimethylsilyl group, triethylsilyl group, tri (n-propyl) silyl group, ethyldimethylsilyl group, n-propyldimethylsilyl group, n-butyldimethylsilyl group, i-butyldimethylsilyl group, tert- Specific examples include a butyldimethylsilyl group and the like, and each butyldimethylsilyl group is selected within a range of each designated number of carbon atoms.

本明細書におけるC〜Cアルキルカルボニルオキシの表記は、炭素原子数がa〜b個よりなる前記の意味であるアルキルカルボニル−O−基を表し、例えばアセトキシ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b alkylcarbonyloxy in the present specification represents an alkylcarbonyl-O-group having the above-mentioned meaning consisting of a to b carbon atoms, and examples thereof include an acetoxy group and the like. , Each selected range of carbon atoms.

本明細書におけるC〜Cアルキルスルホニルオキシの表記は、炭素原子数がa〜b個よりなる前記の意味であるアルキルスルホニル−O−基を表し、例えばメチルスルホニルオキシ基、エチルスルホニルオキシ基、n−プロピルスルホニルオキシ基、i−プロピルスルホニルオキシ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b alkylsulfonyloxy in the present specification represents an alkylsulfonyl-O— group having the above-mentioned meaning consisting of a to b carbon atoms, for example, methylsulfonyloxy group, ethylsulfonyloxy group Specific examples include an n-propylsulfonyloxy group, an i-propylsulfonyloxy group, and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるC〜Cハロアルキルスルホニルオキシの表記は、炭素原子数がa〜b個よりなる前記の意味であるハロアルキルスルホニル−O−基を表し、例えばジフルオロメチルスルホニルオキシ基、トリフルオロメチルスルホニルオキシ基、クロロジフルオロメチルスルホニルオキシ基、ブロモジフルオロメチルスルホニルオキシ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C a -C b haloalkylsulfonyloxy in the present specification represents a haloalkylsulfonyl-O— group having the above-mentioned meaning consisting of a to b carbon atoms, for example, difluoromethylsulfonyloxy group, trifluoromethyl Specific examples include a sulfonyloxy group, a chlorodifluoromethylsulfonyloxy group, a bromodifluoromethylsulfonyloxy group, and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるR5aによって任意に置換された(C〜C)アルキル、R10aによって任意に置換された(C〜C)アルキル、R15aによって任意に置換された(C〜C)アルキル、R15bによって任意に置換された(C〜C)アルキル、R15cによって任意に置換された(C〜C)アルキル、R20によって任意に置換された(C〜C)アルキル、R28によって任意に置換された(C〜C)アルキル又はR28aによって任意に置換された(C〜C)アルキル等の表記は、任意のR5a、R10a、R15a、R15b、R15c、R20、R28又はR28aによって、炭素原子に結合した水素原子が任意に置換された炭素原子数がa〜b個よりなる前記の意味であるアルキル基を表し、各々の指定の炭素原子数の範囲で選択される。このとき、それぞれの(C〜C)アルキル基上の置換基R5a、R10a、R15a、R15b、R15c、R20、R28又はR28aが2個以上存在するとき、それぞれのR5a、R10a、R15a、R15b、R15c、R20、R28又はR28aは互いに同一でも異なってもよい。 Optionally substituted by R 5a herein (C a ~C b) alkyl, optionally substituted by R 10a (C a ~C b) alkyl, optionally substituted by R 15a (C a ~ C b) alkyl, optionally substituted by R 15b (C a ~C b) alkyl, optionally substituted by R 15c (C a ~C b) alkyl, optionally substituted by R 20 (C a -C b) alkyl, optionally substituted by R 28 (C a ~C b) alkyl or optionally substituted by R 28a (C a ~C b) notation alkyl or the like, any of R 5a, R 10a, R 15a, R 15b, R 15c, the R 20, R 28 or R 28a, it than a~b number carbon atoms bonded to hydrogen atoms are optionally substituted carbon atoms It represents an alkyl group wherein the meaning of, is selected from the range of the specified number of carbon atoms. At this time, when two or more substituents R 5a , R 10a , R 15a , R 15b , R 15c , R 20 , R 28 or R 28a on each (C a -C b ) alkyl group are present, R 5a , R 10a , R 15a , R 15b , R 15c , R 20 , R 28 or R 28a may be the same or different from each other.

本明細書におけるR5aによって任意に置換された(C〜C)シクロアルキル、R10aによって任意に置換された(C〜C)シクロアルキル、R15aによって任意に置換された(C〜C)シクロアルキル、R15bによって任意に置換された(C〜C)シクロアルキル、R15cによって任意に置換された(C〜C)シクロアルキル、R20によって任意に置換された(C〜C)シクロアルキル、R28によって任意に置換された(C〜C)シクロアルキル又はR28aによって任意に置換された(C〜C)シクロアルキル等の表記は、任意のR5a、R10a、R15a、R15b、R15c、R20、R28又はR28aによって任意に置換された(C〜C)シクロアルキルによって、炭素原子に結合した水素原子が任意に置換された炭素原子数がa〜b個よりなる前記の意味であるシクロアルキル基を表し、各々の指定の炭素原子数の範囲で選択される。このとき、それぞれの(C〜C)シクロアルキル基上の置換基R5a、R10a、R15a、R15b、R15c、R20、R28又はR28aが2個以上存在するとき、それぞれのR5a、R10a、R15a、R15b、R15c、R20、R28又はR28aは互いに同一でも異なってもよく、さらに置換位置は環構造部分であっても、側鎖部分であっても、或いはそれらの両方にあってもよい。 Optionally substituted by R 5a herein (C a ~C b) cycloalkyl, optionally substituted by R 10a (C a ~C b) cycloalkyl, optionally substituted by R 15a (C a -C b) cycloalkyl, substituted optionally substituted by R 15b (C a ~C b) cycloalkyl, optionally substituted by R 15c (C a ~C b) cycloalkyl, optionally by R 20 been (C a ~C b) cycloalkyl, notation (C a ~C b) cycloalkyl such as optionally substituted by optionally substituted (C a ~C b) cycloalkyl or R 28a by R 28 It can be any R 5a, R 10a, R 15a , R 15b, R 15c, R 20, optionally substituted by R 28 or R 28a (C a C b) by cycloalkyl, a cycloalkyl group is defined above which number of carbon atoms in which the hydrogen atoms bonded to carbon atom is optionally substituted is more a~b number, the range of the specified number of carbon atoms Selected. At this time, when two or more substituents R 5a , R 10a , R 15a , R 15b , R 15c , R 20 , R 28 or R 28a on each (C a -C b ) cycloalkyl group are present, Each R 5a , R 10a , R 15a , R 15b , R 15c , R 20 , R 28 or R 28a may be the same as or different from each other, and the substitution position may be a ring structure part or a side chain part. Or both.

本明細書におけるR5aによって任意に置換された(C〜C)アルケニル、R10aによって任意に置換された(C〜C)アルケニル、R15aによって任意に置換された(C〜C)アルケニル、R15bによって任意に置換された(C〜C)アルケニル、R15cによって任意に置換された(C〜C)アルケニル、R20によって任意に置換された(C〜C)アルケニル、R28によって任意に置換された(C〜C)アルケニル又はR28aによって任意に置換された(C〜C)アルケニル等の表記は、任意のR5a、R10a、R15a、R15b、R15c、R20、R28又はR28aによって、炭素原子に結合した水素原子が任意に置換された炭素原子数がa〜b個よりなる前記の意味であるアルケニル基を表し、各々の指定の炭素原子数の範囲で選択される。このとき、それぞれの(C〜C)アルケニル基上の置換基R5a、R10a、R15a、R15b、R15c、R20、R28又はR28aが2個以上存在するとき、それぞれのR5a、R10a、R15a、R15b、R15c、R20、R28又はR28aは互いに同一でも異なってもよい。 Optionally substituted by R 5a herein (C a ~C b) alkenyl, optionally substituted by R 10a (C a ~C b) alkenyl, optionally substituted by R 15a (C a ~ C b) alkenyl, optionally substituted by R 15b (C a ~C b) alkenyl, optionally substituted by R 15c (C a ~C b) alkenyl, optionally substituted by R 20 (C a -C b) alkenyl, optionally substituted by R 28 (C a ~C b) optionally substituted by alkenyl or R 28a (C a ~C b) notation alkenyl or the like, any of R 5a, R 10a, R 15a, R 15b, R 15c, R 20, by R 28 or R 28a, the number of carbon atoms bonded to hydrogen atoms are optionally substituted carbon atoms An alkenyl group wherein the meaning of a~b pieces made of is selected from the range of the specified number of carbon atoms. At this time, when two or more substituents R 5a , R 10a , R 15a , R 15b , R 15c , R 20 , R 28 or R 28a on each (C a -C b ) alkenyl group are present, R 5a , R 10a , R 15a , R 15b , R 15c , R 20 , R 28 or R 28a may be the same or different from each other.

本明細書におけるR5aによって任意に置換された(C〜C)シクロアルケニル、R10aによって任意に置換された(C〜C)シクロアルケニル、R15aによって任意に置換された(C〜C)シクロアルケニル、R15bによって任意に置換された(C〜C)シクロアルケニル、R15cによって任意に置換された(C〜C)シクロアルケニル、R20によって任意に置換された(C〜C)シクロアルケニル、R28によって任意に置換された(C〜C)シクロアルケニル又はR28aによって任意に置換された(C〜C)シクロアルケニル等の表記は、任意のR5a、R10a、R15a、R15b、R15c、R20又はR28aによって、炭素原子に結合した水素原子が任意に置換された炭素原子数がa〜b個よりなる前記の意味であるシクロアルケニル基を表し、各々の指定の炭素原子数の範囲で選択される。このとき、それぞれの(C〜C)シクロアルケニル基上の置換基R5a、R10a、R15a、R15b、R15c、R20、R28又はR28aが2個以上存在するとき、それぞれのR5a、R10a、R15a、R15b、R15c、R20、R28又はR28aは互いに同一でも異なってもよく、さらに置換位置は環構造部分であっても、側鎖部分であっても、或いはそれらの両方にあってもよい。 Optionally substituted by R 5a herein (C a ~C b) cycloalkenyl, optionally substituted by R 10a (C a ~C b) cycloalkenyl, optionally substituted by R 15a (C a- C b ) cycloalkenyl, optionally substituted by R 15b (C a -C b ) cycloalkenyl, optionally substituted by R 15c (C a -C b ) cycloalkenyl, optionally substituted by R 20 been (C a ~C b) cycloalkenyl, notation such as (C a ~C b) cycloalkenyl optionally substituted by optionally substituted (C a ~C b) cycloalkenyl or R 28a by R 28 Are bonded to the carbon atom by any R 5a , R 10a , R 15a , R 15b , R 15c , R 20 or R 28a . And a cycloalkenyl group having the above-mentioned meanings consisting of a to b carbon atoms in which hydrogen atoms are optionally substituted, each being selected in the range of the designated number of carbon atoms. At this time, when there are two or more substituents R 5a , R 10a , R 15a , R 15b , R 15c , R 20 , R 28 or R 28a on each (C a -C b ) cycloalkenyl group, Each R 5a , R 10a , R 15a , R 15b , R 15c , R 20 , R 28 or R 28a may be the same or different from each other, and the substitution position may be a ring structure part or a side chain part. Or both.

本明細書におけるR5aによって任意に置換された(C〜C)アルキニル、R10aによって任意に置換された(C〜C)アルキニル、R15aによって任意に置換された(C〜C)アルキニル、R15bによって任意に置換された(C〜C)アルキニル、R15cによって任意に置換された(C〜C)アルキニル、R20によって任意に置換された(C〜C)アルキニル、R28によって任意に置換された(C〜C)アルキニル又はR28aによって任意に置換された(C〜C)アルキニル等の表記は、任意のR5a、R10a、R15a、R15b、R15c、R20、R28又はR28aによって、炭素原子に結合した水素原子が任意に置換された炭素原子数がa〜b個よりなる前記の意味であるアルキニル基を表し、各々の指定の炭素原子数の範囲で選択される。このとき、それぞれの(C〜C)アルキニル基上の置換基R5a、R10a、R15a、R15b、R15c、R20、R28又はR28aが2個以上存在するとき、それぞれのR5a、R10a、R15a、R15b、R15c、R20、R28又はR28aは互いに同一でも異なってもよい。 Optionally substituted by R 5a herein (C a ~C b) alkynyl, optionally substituted by R 10a (C a ~C b) alkynyl, optionally substituted by R 15a (C a ~ C b) alkynyl, optionally substituted by R 15b (C a ~C b) alkynyl, optionally substituted by R 15c (C a ~C b) alkynyl, optionally substituted by R 20 (C a -C b) alkynyl, optionally substituted by R 28 (C a ~C b) optionally substituted by alkynyl, or R 28a (C a ~C b) notation alkynyl or the like, any of R 5a, R 10a, R 15a, R 15b, R 15c, R 20, by R 28 or R 28a, the number of carbon atoms bonded to hydrogen atoms are optionally substituted carbon atoms It represents the meaning a is an alkynyl group which a~b pieces made of is selected from the range of the specified number of carbon atoms. At this time, when two or more substituents R 5a , R 10a , R 15a , R 15b , R 15c , R 20 , R 28 or R 28a on each (C a -C b ) alkynyl group are present, R 5a , R 10a , R 15a , R 15b , R 15c , R 20 , R 28 or R 28a may be the same as or different from each other.

本明細書における
〔R8aはR9aと一緒になってC〜Cのアルキレン鎖又はC〜Cのアルケニレン鎖を形成することにより、R8a及びR9aが結合する窒素原子と共に3〜8員環を形成してもよく、このときこのアルキレン鎖又はアルケニレン鎖は酸素原子、硫黄原子又は窒素原子を1個含んでもよく、〕
〔R13aはR14aと一緒になってC〜Cのアルキレン鎖又はC〜Cのアルケニレン鎖を形成することにより、R13a及びR14aが結合する窒素原子と共に3〜8員環を形成してもよく、このときこのアルキレン鎖又はアルケニレン鎖は酸素原子、硫黄原子又は窒素原子を1個含んでもよく、〕
等の表記の具体例として、例えばアジリジン、アゼチジン、アゼチジン−2−オン、ピロリジン、ピロリジン−2−オン、オキサゾリジン、オキサゾリジン−2−オン、オキサゾリジン−2−チオン、チアゾリジン、チアゾリジン−2−オン、チアゾリジン−2−チオン、イミダゾリジン、イミダゾリジン−2−オン、イミダゾリジン−2−チオン、ピペリジン、ピペリジン−2−オン、ピペリジン−2−チオン、2H−3,4,5,6−テトラヒドロ−1,3−オキサジン−2−オン、2H−3,4,5,6−テトラヒドロ−1,3−オキサジン−2−チオン、モルホリン、2H−3,4,5,6−テトラヒドロ−1,3−チアジン−2−オン、2H−3,4,5,6−テトラヒドロ−1,3−チアジン−2−チオン、チオモルホリン、ペルヒドロピリミジン−2−オン、ピペラジン、ホモピペリジン、ホモピペリジン−2−オン、ヘプタメチレンイミン等が挙げられ、各々の指定の原子数の範囲で選択される。
[R 8a herein by forming the alkenylene chain alkylene chain or C 2 -C 7 of C 2 -C 7 together with R 9a, 3 together with the nitrogen atom to which R 8a and R 9a are bonded An 8-membered ring may be formed, in which case the alkylene chain or alkenylene chain may contain one oxygen atom, sulfur atom or nitrogen atom.]
[R 13a is by forming alkenylene chain alkylene chain or C 2 -C 7 of C 2 -C 7 together with R 14a, 3 to 8-membered ring together with the nitrogen atom to which R 13a and R 14a are attached Wherein the alkylene chain or alkenylene chain may contain one oxygen atom, sulfur atom or nitrogen atom,
Specific examples of the notation such as aziridine, azetidine, azetidin-2-one, pyrrolidine, pyrrolidin-2-one, oxazolidine, oxazolidine-2-one, oxazolidine-2-thione, thiazolidine, thiazolidine-2-one, thiazolidine -2-thione, imidazolidine, imidazolidine-2-one, imidazolidine-2-thione, piperidine, piperidin-2-one, piperidine-2-thione, 2H-3,4,5,6-tetrahydro-1, 3-Oxazin-2-one, 2H-3,4,5,6-tetrahydro-1,3-oxazine-2-thione, morpholine, 2H-3,4,5,6-tetrahydro-1,3-thiazine- 2-one, 2H-3,4,5,6-tetrahydro-1,3-thiazine-2-thione, thiomorpholine, pe Tetrahydropyrimidine-2-one, piperazine, homopiperidine, homopiperidine-2-one, heptamethyleneimine, and the like, may be selected from the range of the number of each of the specified atoms.

本発明化合物は、以下の方法で製造することができる。   The compound of the present invention can be produced by the following method.

製造法A   Manufacturing method A

Figure 2015147757
Figure 2015147757

式(7)[式中A、B、R、R及びnは前記と同じ意味を表す。]で表される化合物を、式(8−1)[式中R7bは前記と同じ意味を表す。]で表される化合物と反応させるか、若しくは式(8−2)[式中R7bは前記と同じ意味を表す。]で表される化合物と縮合剤の存在下で反応させることにより、式(9)[式中A、B、R、R、R及びnは前記と同じ意味を表す。]で表される本発明化合物を合成することができる。 Formula (7) [wherein A 1 , B, R 2 , R a and n represent the same meaning as described above. ] The compound represented by formula (8-1) [wherein R 7b represents the same meaning as described above. Or a compound represented by formula (8-2) [wherein R 7b represents the same meaning as described above. The compound represented by formula (9) [wherein A 1 , B, R 2 , R a , R b and n represent the same meaning as described above]. This invention compound represented by this can be synthesize | combined.

本反応では式(7)で表される化合物1当量に対して、式(8−1)で表される化合物は、0.5〜50当量の範囲で用いることができる。   In this reaction, the compound represented by the formula (8-1) can be used in the range of 0.5 to 50 equivalents with respect to 1 equivalent of the compound represented by the formula (7).

また、本反応では、式(8−2)で表される化合物1当量に対して1〜4当量の縮合剤を用いることができる。用いる縮合剤としては、WSC{1−エチル−3−(3−ジメチルアミノプロピル)カルボジイミド塩酸塩}、CDI(カルボニルジイミダゾール)等が挙げられる。さらに、式(7)で表される化合物1当量に対して、式(8−2)で表される化合物を、0.5〜50当量の範囲で用いることができる。   In this reaction, 1 to 4 equivalents of a condensing agent can be used with respect to 1 equivalent of the compound represented by Formula (8-2). Examples of the condensing agent to be used include WSC {1-ethyl-3- (3-dimethylaminopropyl) carbodiimide hydrochloride}, CDI (carbonyldiimidazole) and the like. Furthermore, the compound represented by Formula (8-2) can be used in the range of 0.5-50 equivalent with respect to 1 equivalent of compound represented by Formula (7).

必要ならば、炭酸カリウム、トリエチルアミン、ピリジン、4−(ジメチルアミノ)ピリジン等の塩基を使用することができる。   If necessary, a base such as potassium carbonate, triethylamine, pyridine, 4- (dimethylamino) pyridine can be used.

本反応は、無溶媒で実施してもよいが、溶媒を用いてもよく、例えば、N,N−ジメチルホルムアミド、N,N−ジメチルアセトアミド、アセトニトリル、ジメチルスルホキシド、1,3−ジメチル−2−イミダゾリノン等の極性溶媒、メタノール、エタノール、プロパノール、2−プロパノール、エチレングリコール等のアルコール類、ジエチルエーテル、テトラヒドロフラン、ジフェニルエーテル等のエーテル類、ベンゼン、トルエン、キシレン等の芳香族炭化水素類、塩化メチレン、クロロホルム、四塩化炭素等のハロゲン化炭化水素類、ペンタン、n−ヘキサン等の脂肪族炭化水素類が挙げられる。これらの溶媒は単独で用いても、これらの内の2種類以上を混合して用いてもよい。   This reaction may be carried out without solvent, but a solvent may be used, for example, N, N-dimethylformamide, N, N-dimethylacetamide, acetonitrile, dimethyl sulfoxide, 1,3-dimethyl-2- Polar solvents such as imidazolinone, alcohols such as methanol, ethanol, propanol, 2-propanol and ethylene glycol, ethers such as diethyl ether, tetrahydrofuran and diphenyl ether, aromatic hydrocarbons such as benzene, toluene and xylene, methylene chloride , Halogenated hydrocarbons such as chloroform and carbon tetrachloride, and aliphatic hydrocarbons such as pentane and n-hexane. These solvents may be used alone or as a mixture of two or more thereof.

反応温度は、−60℃から反応混合物の還流温度までの任意の温度を設定することができ、反応時間は、反応基質の濃度、反応温度によって変化するが、通常5分から100時間の範囲で任意に設定できる。   The reaction temperature can be set to any temperature from −60 ° C. to the reflux temperature of the reaction mixture, and the reaction time varies depending on the concentration of the reaction substrate and the reaction temperature, but is usually arbitrary in the range of 5 minutes to 100 hours. Can be set.

式(8−1)で表される化合物の或るものは公知化合物であり、一部は市販品として入手できる。また、それ以外のものも文献記載の公知の方法に準じて合成することができる。   Some of the compounds represented by formula (8-1) are known compounds, and some of them are commercially available. Others can be synthesized according to known methods described in the literature.

式(8−2)で表される化合物の或るものは公知化合物であり、一部は市販品として入手できる。また、それ以外のものも文献記載の公知の方法に準じて合成することができる。   Some of the compounds represented by formula (8-2) are known compounds, and some of them are commercially available. Others can be synthesized according to known methods described in the literature.

式(7)で表される化合物の或るものは、例えば、BがB−1、B−4、B−5、B−6、B−7、B−17、B−18、B−30、B−32、B−33又はB−34で表される化合物は、以下の文献記載の公知の方法により製造することが出来る。
B−1;バイオオーガニック アンド メディシナル ケミストリー レターズ 2000年,10巻,1211頁等
B−4;ヘテロサイクルス 2007年,7巻,2249頁等
B−5;バイオオーガニック メディシナル ケミストリー 2012年,10巻,1785ページ等
B−6;ジャーナル メディシナル ケミストリー 2012年,55巻,1817頁等
B−7;ジャーナル ヘテロサイクリック ケミストリー 1981年,18巻,1379頁等
B−17;国際公開第2011/049150号等
B−18;ジャーナル オブ ザ ケミカル ソサエティー パーキン トランスアクション1 オーガニック アンド バイオオーガニックケミストリー 1977年,2536頁等
B−30;テトラへドロン レタース 2005年,46巻,2075頁等
B−32ジャーナル オブ オーガニック ケミストリー 1980年,45巻,1473頁等
B−33;アルヒーフ デア ファーマツィー 1980年,313巻,867頁
B−34;バイオオーガニック アンド メディシナル ケミストリー レターズ 2000年,10巻,1211頁等
また、それ以外のものも文献記載の公知の方法に準じて合成することができる。
Some of the compounds represented by formula (7) include, for example, B is B-1, B-4, B-5, B-6, B-7, B-17, B-18, B-30. , B-32, B-33 or B-34 can be produced by known methods described in the following literature.
B-1; Bioorganic and Medicinal Chemistry Letters 2000, 10, 1211 etc. B-4; Heterocycles 2007, 7, 2249 etc. B-5; Bioorganic Medicinal Chemistry 2012, 10, 1785 Journal Medicinal Chemistry 2012, 55, 1817 etc. B-7; Journal Heterocyclic Chemistry 1981, 18, 1379 etc. B-17; International Publication No. 2011-049150 etc. B- 18; Journal of the Chemical Society Parkin Transaction 1 Organic and Bioorganic Chemistry 1977, 2536, etc. B-30; Tetrahedron Letters 2005, 46, 2075, etc. B 32 Journal of Organic Chemistry 1980, 45, 1473 etc. B-33; Alphee Der Pharmacy 1980, 313, 867 B-34; Bioorganic and Medicinal Chemistry Letters 2000, 10, 1211 etc. Others can be synthesized according to known methods described in the literature.

製造法B   Manufacturing method B

Figure 2015147757
Figure 2015147757

式(9)で表される化合物と、五硫化二燐、五硫化二燐−HMDO(ヘキサメチルジシロキサン)、ローソン試薬(Lawesson’s Reagent;2,4−ビス(4−メトキシフェニル)−1,3,2,4−ジチアジホスフェタン−2,4−ジスルフィド)等の硫化剤を反応させることにより、式(35)[式中A、B、R、R、R及びnは前記と同じ意味を表す。]で表される本発明化合物を得ることができる。 A compound represented by the formula (9), diphosphorus pentasulfide, diphosphorus pentasulfide-HMDO (hexamethyldisiloxane), Lawesson's Reagent; 2,4-bis (4-methoxyphenyl) -1 , 3,2,4-dithiadiphosphetane-2,4-disulfide) and the like to react with the compound represented by formula (35) [wherein A 1 , B, R 2 , R a , R b and n represents the same meaning as described above. This invention compound represented by this can be obtained.

本反応で用いる硫化剤は、式(9)で表される化合物1当量に対して0.5〜50当量の範囲で用いることができる。   The sulfurizing agent used in this reaction can be used in the range of 0.5 to 50 equivalents relative to 1 equivalent of the compound represented by formula (9).

必要ならば、炭酸カリウム、トリエチルアミン、ピリジン、4−(ジメチルアミノ)ピリジン等の塩基を使用することができる。   If necessary, a base such as potassium carbonate, triethylamine, pyridine, 4- (dimethylamino) pyridine can be used.

本反応は、無溶媒でも実施することができるが、溶媒を用いてもよい。例えば、N,N−ジメチルホルムアミド、N,N−ジメチルアセトアミド、アセトニトリル、ジメチルスルホキシド、1,3−ジメチル−2−イミダゾリノン、水等の極性溶媒、メタノール、エタノール、プロパノール、2−プロパノール、エチレングリコール等のアルコール類、ジエチルエーテル、テトラヒドロフラン、ジフェニルエーテル等のエーテル類、ベンゼン、トルエン、キシレン等の芳香族炭化水素類、塩化メチレン、クロロホルム、四塩化炭素等のハロゲン化炭化水素類、ペンタン、n−ヘキサン等の脂肪族炭化水素類が挙げられる。これらの溶媒は単独で用いても、これらの内の2種類以上を混合して用いてもよい。   This reaction can be carried out without solvent, but a solvent may be used. For example, polar solvent such as N, N-dimethylformamide, N, N-dimethylacetamide, acetonitrile, dimethyl sulfoxide, 1,3-dimethyl-2-imidazolinone, water, methanol, ethanol, propanol, 2-propanol, ethylene glycol Alcohols such as diethyl ether, tetrahydrofuran and diphenyl ether, aromatic hydrocarbons such as benzene, toluene and xylene, halogenated hydrocarbons such as methylene chloride, chloroform and carbon tetrachloride, pentane and n-hexane And aliphatic hydrocarbons. These solvents may be used alone or as a mixture of two or more thereof.

反応温度は、−60℃から反応混合物の還流温度までの任意の温度を設定することができ、反応時間は、反応基質の濃度、反応温度によって変化するが、通常5分から100時間の範囲で任意に設定できる。   The reaction temperature can be set to any temperature from −60 ° C. to the reflux temperature of the reaction mixture, and the reaction time varies depending on the concentration of the reaction substrate and the reaction temperature, but is usually arbitrary in the range of 5 minutes to 100 hours. Can be set.

製造法C   Manufacturing method C

Figure 2015147757
Figure 2015147757

式(13)[式中A、B、R及びnは前記と同じ意味を表す。]で表される化合物を、製造法Aと同様の方法を用いて、式(8−1)で表される化合物又は式(8−2)で表される化合物と反応させることにより、式(41)[式中A、B、R、R7b及びnは前記と同じ意味を表す。]で表される本発明化合物を得ることができる。 Formula (13) [wherein A 1 , B, R 2 and n represent the same meaning as described above. The compound represented by formula (8-1) or the compound represented by formula (8-2) is reacted with the compound represented by formula (8-1) using the same method as in Production Method A. 41) [wherein A 1 , B, R 2 , R 7b and n represent the same meaning as described above. This invention compound represented by this can be obtained.

次いで、式(41)で表される化合物を、式(5)[式中Rは前記と同じ意味を表し、Jはハロゲン原子、−OH、−OSOCH、−OSOCF等の脱離基を表す。]で表される化合物と反応させて、式(9)で表される化合物を得ることができる。 Subsequently, the compound represented by formula (41) is represented by formula (5) [wherein R a represents the same meaning as described above, and J b represents a halogen atom, —OH, —OSO 2 CH 3 , —OSO 2 CF 3. Represents a leaving group. And a compound represented by the formula (9) can be obtained.

本反応は、式(41)で表される化合物1当量に対して、式(5)で表される化合物を、0.5〜50当量の範囲で用いることができる。必要ならば塩酸、硫酸、p−トルエンスルホン酸等の酸、炭酸カリウム、トリエチルアミン、ピリジン、4−(ジメチルアミノ)ピリジン、水素化ナトリウム、水酸化ナトリウム、水酸化カリウム等の塩基を使用することができる。   In this reaction, the compound represented by the formula (5) can be used in the range of 0.5 to 50 equivalents with respect to 1 equivalent of the compound represented by the formula (41). If necessary, an acid such as hydrochloric acid, sulfuric acid, p-toluenesulfonic acid, a base such as potassium carbonate, triethylamine, pyridine, 4- (dimethylamino) pyridine, sodium hydride, sodium hydroxide, potassium hydroxide may be used. it can.

本反応は、ジエチルアゾジカルボキシレートとトリフェニルホスフィン等を使用する光延反応を使用することができる。   In this reaction, Mitsunobu reaction using diethyl azodicarboxylate and triphenylphosphine can be used.

本反応は、無溶媒でも実施することができるが、溶媒を用いてもよい。例えば、N,N−ジメチルホルムアミド、N,N−ジメチルアセトアミド、アセトニトリル、ジメチルスルホキシド、1,3−ジメチル−2−イミダゾリノン、水等の極性溶媒、メタノール、エタノール、プロパノール、2−プロパノール、エチレングリコール等のアルコール類、ジエチルエーテル、テトラヒドロフラン、ジフェニルエーテル等のエーテル類、ベンゼン、トルエン、キシレン等の芳香族炭化水素類、塩化メチレン、クロロホルム、四塩化炭素等のハロゲン化炭化水素類、ペンタン、n−ヘキサン等の脂肪族炭化水素類が挙げられる。これらの溶媒は単独で用いても、これらの内の2種類以上を混合して用いてもよい。   This reaction can be carried out without solvent, but a solvent may be used. For example, polar solvent such as N, N-dimethylformamide, N, N-dimethylacetamide, acetonitrile, dimethyl sulfoxide, 1,3-dimethyl-2-imidazolinone, water, methanol, ethanol, propanol, 2-propanol, ethylene glycol Alcohols such as diethyl ether, tetrahydrofuran and diphenyl ether, aromatic hydrocarbons such as benzene, toluene and xylene, halogenated hydrocarbons such as methylene chloride, chloroform and carbon tetrachloride, pentane and n-hexane And aliphatic hydrocarbons. These solvents may be used alone or as a mixture of two or more thereof.

反応温度は、−60℃から反応混合物の還流温度までの任意の温度を設定することができ、反応時間は、反応基質の濃度、反応温度によって変化するが、通常5分から100時間の範囲で任意に設定できる。   The reaction temperature can be set to any temperature from −60 ° C. to the reflux temperature of the reaction mixture, and the reaction time varies depending on the concentration of the reaction substrate and the reaction temperature, but is usually arbitrary in the range of 5 minutes to 100 hours. Can be set.

式(5)で表される化合物の或るものは公知化合物であり、一部は市販品として入手できる。また、それ以外のものも文献記載の公知の方法に準じて合成することができる。   Some of the compounds represented by formula (5) are known compounds, and some of them are commercially available. Others can be synthesized according to known methods described in the literature.

製造法Aから製造法Cの反応は、必要であれば窒素、アルゴン等の不活性ガス雰囲気下で実施しても良い。   The reaction from production method A to production method C may be carried out in an inert gas atmosphere such as nitrogen or argon if necessary.

製造法Aから製造法Cの反応において、反応終了後の反応混合物は、直接濃縮、又は有機溶媒に溶解し、水洗後濃縮、又は氷水に投入、有機溶媒抽出後濃縮といった通常の後処理を行ない、目的の本発明化合物を得ることができる。また、精製の必要が生じたときには、再結晶、カラムクロマトグラフ、薄層クロマトグラフ、液体クロマトグラフ分取等の任意の精製方法によって分離、精製することができる。   In the reaction from production method A to production method C, the reaction mixture after completion of the reaction is directly concentrated, or dissolved in an organic solvent, concentrated after washing with water, or poured into ice water, followed by normal post-treatment such as concentration after extraction with an organic solvent. The objective compound of the present invention can be obtained. Moreover, when the necessity for purification arises, it can be separated and purified by any purification method such as recrystallization, column chromatograph, thin layer chromatograph, liquid chromatographic fractionation and the like.

製造法Aで用いられる式(7)で表される化合物のうち、BがB−9〜B−16、B−28又はB−31を表すとき、例えば以下のようにして合成することが出来る。   Of the compounds represented by formula (7) used in production method A, when B represents B-9 to B-16, B-28 or B-31, for example, the compound can be synthesized as follows. .

反応式1   Reaction formula 1

Figure 2015147757
Figure 2015147757

式(7−1)[式中R及びBは前記と同じ意味を表し、Jはハロゲン原子、−OH、−OSOCH、−OSOCF等の脱離基を表す。]で表される化合物と式(2−2)[式中A、R及びnは前記と同じ意味を表し、Lはフッ素原子、塩素原子、臭素原子、ヨウ素原子、−B(OH)基又は−B(OR51基(式中R51は、水素原子又は、同一又は異なってもよいC〜Cアルキルを表し、或いは、2つのR51が一緒になって−CHCH−又は−C(CHC(CH−を形成してもよい)を表す。]で表される化合物を、触媒及び塩基の存在下で反応させることにより、式(7)で表される化合物を得ることができる。 Formula (7-1) [wherein R a and B represent the same meaning as described above, and J b represents a leaving group such as a halogen atom, —OH, —OSO 2 CH 3 , —OSO 2 CF 3, etc. And a compound represented by formula (2-2) [wherein A 1 , R 2 and n represent the same meaning as described above, and L 1 represents a fluorine atom, a chlorine atom, a bromine atom, an iodine atom, —B (OH ) 2 groups or -B (OR 51 ) 2 groups (wherein R 51 represents a hydrogen atom or C 1 to C 6 alkyl which may be the same or different, or two R 51 together represent- CH 2 CH 2 — or —C (CH 3 ) 2 C (CH 3 ) 2 — may be formed). The compound represented by the formula (7) can be obtained by reacting the compound represented by formula (7) in the presence of a catalyst and a base.

式(2−2)で表される化合物の量は、式(7−1)で表される化合物1当量に対して0.8〜5当量の範囲で、用いることができる。   The amount of the compound represented by Formula (2-2) can be used in the range of 0.8 to 5 equivalents relative to 1 equivalent of the compound represented by Formula (7-1).

ここで用いられる式(2−2)で表される化合物の或るものは公知化合物であり、一部は市販品として入手できる。また、それ以外のものも文献記載の方法に準じて合成することができる。   Some of the compounds represented by the formula (2-2) used here are known compounds, and some of them are available as commercial products. Others can be synthesized according to the methods described in the literature.

本反応で使用できる触媒としては、例えば、パラジウム−炭素、塩化パラジウム、酢酸パラジウム、ビス(トリフェニルホスフィン)パラジウムジクロリド、テトラキス(トリフェニルホスフィン)パラジウム等のパラジウム触媒又は金属銅、酢酸銅(I)、酢酸銅(II)、酸化銅(I)、酸化銅(II)、ヨウ化銅等の銅触媒が挙げられる。触媒の使用量は、式(2−2)で表される化合物1当量に対して0.001〜1.0当量、好ましくは、0.01〜0.5当量、さらに好ましくは0.05〜0.2当量の範囲で、用いることができる。   Examples of the catalyst that can be used in this reaction include palladium catalysts such as palladium-carbon, palladium chloride, palladium acetate, bis (triphenylphosphine) palladium dichloride, tetrakis (triphenylphosphine) palladium, or copper metal, copper acetate (I). And copper catalysts such as copper (II) acetate, copper (I) oxide, copper (II) oxide and copper iodide. The catalyst is used in an amount of 0.001 to 1.0 equivalent, preferably 0.01 to 0.5 equivalent, more preferably 0.05 to 1 equivalent to 1 equivalent of the compound represented by formula (2-2). It can be used in the range of 0.2 equivalents.

使用する塩基としては、例えば、ピリジン、ジイソプロピルエチルアミン、トリエチルアミン等の三級アミン化合物、例えば水酸化ナトリウム、水酸化カリウム、炭酸ナトリウム、炭酸カリウム、炭酸セシウム、炭酸水素ナトリウム等の無機塩基等が挙げられる。塩基の使用量は、式(7−1)で表される化合物1当量に対して0.1〜10.0当量の範囲で用いることができる。   Examples of the base used include tertiary amine compounds such as pyridine, diisopropylethylamine, and triethylamine, and inorganic bases such as sodium hydroxide, potassium hydroxide, sodium carbonate, potassium carbonate, cesium carbonate, and sodium bicarbonate. . The usage-amount of a base can be used in the range of 0.1-10.0 equivalent with respect to 1 equivalent of compounds represented by Formula (7-1).

本反応は、無溶媒でも実施することができるが、溶媒を用いてもよい。例えば、N,N−ジメチルホルムアミド、N,N−ジメチルアセトアミド、アセトニトリル、ジメチルスルホキシド、1,3−ジメチル−2−イミダゾリノン、水等の極性溶媒、メタノール、エタノール、プロパノール、2−プロパノール、エチレングリコール等のアルコール類、ジエチルエーテル、テトラヒドロフラン、ジフェニルエーテル等のエーテル類、ベンゼン、トルエン、キシレン等の芳香族炭化水素類、塩化メチレン、クロロホルム、四塩化炭素等のハロゲン化炭化水素類、ペンタン、n−ヘキサン等の脂肪族炭化水素類が挙げられる。これらの溶媒は単独で用いても、これらの内の2種類以上を混合して用いてもよい。   This reaction can be carried out without solvent, but a solvent may be used. For example, polar solvent such as N, N-dimethylformamide, N, N-dimethylacetamide, acetonitrile, dimethyl sulfoxide, 1,3-dimethyl-2-imidazolinone, water, methanol, ethanol, propanol, 2-propanol, ethylene glycol Alcohols such as diethyl ether, tetrahydrofuran and diphenyl ether, aromatic hydrocarbons such as benzene, toluene and xylene, halogenated hydrocarbons such as methylene chloride, chloroform and carbon tetrachloride, pentane and n-hexane And aliphatic hydrocarbons. These solvents may be used alone or as a mixture of two or more thereof.

反応温度は、−60℃から反応混合物の還流温度までの任意の温度を設定することができ、反応時間は、反応基質の濃度、反応温度によって変化するが、通常5分から100時間の範囲で任意に設定できる。   The reaction temperature can be set to any temperature from −60 ° C. to the reflux temperature of the reaction mixture, and the reaction time varies depending on the concentration of the reaction substrate and the reaction temperature, but is usually arbitrary in the range of 5 minutes to 100 hours. Can be set.

式(7−1)で表される化合物の或るものは、例えば、BがB−9、B−10、B−11、B−12、B−13、B−14、B−16又はB−27で表される化合物の或るものは公知化合物であり、一部は市販品として入手できる。また、それ以外のものも文献記載の公知の方法に準じて合成することができる。   Some of the compounds represented by formula (7-1) are, for example, wherein B is B-9, B-10, B-11, B-12, B-13, B-14, B-16 or B Some of the compounds represented by −27 are known compounds, and some of them are commercially available. Others can be synthesized according to known methods described in the literature.

また、BがB−15、B−19、B−20、B−21、B−22、B−23、B−24、B−25、B−28又はB−31で表される化合物は、以下の文献記載の公知の方法により製造することが出来る。
B−15;日本国特許出願公開第55/160768号等
B−19;テトラへドロン 2003年,59巻,7695頁等
B−20;国際公開第2010/080864号等
B−21;国際公開第2010/135650号等
B−22;ケミカル ファーマシューティカル ブルチン 1976年,24巻,26頁等
B−23;テトラへドロン レタース 2003年,44巻,3355頁等
B−24;テトラへドロン 2004年,60巻,3311頁等
B−25;テトラへドロン レタース 2011年,52巻,5224頁等
B−28;ヘテロサイクルス 1984年,22巻,1195頁等
B−31;ケミッシェ ベリヒテ 1970年,103巻,272頁等
また、それ以外のものも文献記載の公知の方法に準じて合成することができる。
In addition, the compound in which B is represented by B-15, B-19, B-20, B-21, B-22, B-23, B-24, B-25, B-28 or B-31, It can be produced by a known method described in the following literature.
B-15; Japanese Patent Application Publication No. 55/160768 etc. B-19; Tetrahedron 2003, 59, p. 7695 etc. B-20; International Publication No. 2010/080864 etc. B-21; No. 2010/135650 etc. B-22; Chemical Pharmaceutical Bulletin 1976, 24, 26 etc. B-23; Tetrahedron Letters 2003, 44, 3355 etc. B-24; Tetrahedron 2004, 60, 3311, etc. B-25; Tetrahedron Letters 2011, 52, 5224, etc. B-28; Heterocycles 1984, 22, 1195, etc. B-31; Chemichet Berichte 1970, 103 , P.272, etc. Others can also be synthesized according to known methods described in the literature.

製造法Aで用いられる式(7)で表される化合物のうち、BがB−2又はB−3を表す化合物は、例えば反応式2〜3を用いて合成することが出来る。   Among the compounds represented by Formula (7) used in Production Method A, the compound in which B represents B-2 or B-3 can be synthesized using, for example, Reaction Formulas 2-3.

反応式2   Reaction formula 2

Figure 2015147757
Figure 2015147757

式(7−2)[式中A、R、B及びnは前記と同じ意味を表す。]で表される化合物は、文献既知の方法、例えば、BがB−2を表す化合物の場合バイオオーガニック アンド メディシナル ケミストリー レターズ 2008年,18巻,1195頁等の公知の方法により製造することができる。また、BがB−3を表す化合物の場合、ジャーナル オブ ヘテロサイクリック ケミストリー 1987年,24巻,973頁等の公知の方法により製造することができる。 Formula (7-2) [wherein A 1, R 2, B and n are as defined above. ] Can be produced by known methods such as Bioorganic and Medicinal Chemistry Letters 2008, Vol. 18, p. 1195, etc. in the literature. . In the case where B is a compound representing B-3, it can be produced by a known method such as Journal of Heterocyclic Chemistry 1987, Vol. 24, page 973.

式(7−2)で表される化合物を、テトラへドロン レタース 2003年,44巻,7629頁等に記載の方法に準じて、反応させることにより式(7−3)[式中A、R、B及びnは前記と同じ意味を表す。]で表される化合物を合成することができる。 By reacting the compound represented by the formula (7-2) according to the method described in Tetrahedron Letters 2003, 44, 7629, etc., the compound represented by the formula (7-3) [wherein A 1 , R 2 , B, and n represent the same meaning as described above. ] Can be synthesized.

続いて、式(7−3)で表される化合物を文献既知の方法、例えば、実験科学講座 第5版(日本化学会編) 2005年,14巻,374頁等に記載の方法に準じて式(2−18)[式中Mはナトリウム、カリウム等のアルカリ金属を表す。]で表される化合物又は式(2−19)[式中Mは前記と同じ意味を表す。]で表される化合物と式(3−2)[式中R6aは前記と同じ意味を表す。]で表される化合物とともに反応させることにより、式(7−4)[式中A、R、R6a、B及びnは前記と同じ意味を表す。]で表される化合物を合成することができる。 Subsequently, the compound represented by the formula (7-3) is converted into a method known in the literature, for example, according to the method described in Experimental Science Course 5th Edition (Edited by The Chemical Society of Japan) 2005, Vol. Formula (2-18) [In formula, M represents alkali metals, such as sodium and potassium. Or a compound represented by formula (2-19): wherein M represents the same meaning as described above. And a compound represented by formula (3-2) [wherein R 6a represents the same meaning as described above. ] Is reacted with the compound represented by the formula (7-4) [wherein A 1 , R 2 , R 6a , B and n represent the same meaning as described above. ] Can be synthesized.

式(3−2)で表される化合物の或るものは公知化合物であり、一部は市販品として入手できる。また、それ以外のものも文献記載の公知の方法に準じて容易に合成することができる。   Some of the compounds represented by formula (3-2) are known compounds, and some of them are commercially available. Others can be easily synthesized according to known methods described in the literature.

一方、式(7−2)で表される化合物を、ジフェニルホスホリルアジド(DPPA)及び式(3−2)で表される化合物と反応させることにより、式(7−4)で表される化合物を得ることができる。   On the other hand, a compound represented by the formula (7-4) is reacted with a compound represented by the formula (7-2) and a compound represented by the formula (3-2). Can be obtained.

本反応では、式(7−2)で表される化合物1当量に対して、DPPAは0.5〜50当量の範囲で用いることができ、式(3−2)で表される化合物は、式(7−2)で表される化合物1当量に対して、1当量から溶媒量の範囲で用いることができる。必要ならば炭酸カリウム、トリエチルアミン、ピリジン、4−(ジメチルアミノ)ピリジン等の塩基を使用することができる。   In this reaction, DPPA can be used in the range of 0.5 to 50 equivalents relative to 1 equivalent of the compound represented by formula (7-2), and the compound represented by formula (3-2) It can be used in the range of 1 equivalent to the amount of solvent with respect to 1 equivalent of the compound represented by formula (7-2). If necessary, a base such as potassium carbonate, triethylamine, pyridine, 4- (dimethylamino) pyridine can be used.

本反応は、無溶媒でも実施することができるが、溶媒を用いてもよい。例えば、N,N−ジメチルホルムアミド、N,N−ジメチルアセトアミド、アセトニトリル、ジメチルスルホキシド、1,3−ジメチル−2−イミダゾリノン、水等の極性溶媒、メタノール、エタノール、プロパノール、2−プロパノール、エチレングリコール等のアルコール類、ジエチルエーテル、テトラヒドロフラン、ジフェニルエーテル等のエーテル類、ベンゼン、トルエン、キシレン等の芳香族炭化水素類、塩化メチレン、クロロホルム、四塩化炭素等のハロゲン化炭化水素類、ペンタン、n−ヘキサン等の脂肪族炭化水素類が挙げられる。これらの溶媒は単独で用いても、これらの内の2種類以上を混合して用いてもよい。   This reaction can be carried out without solvent, but a solvent may be used. For example, polar solvent such as N, N-dimethylformamide, N, N-dimethylacetamide, acetonitrile, dimethyl sulfoxide, 1,3-dimethyl-2-imidazolinone, water, methanol, ethanol, propanol, 2-propanol, ethylene glycol Alcohols such as diethyl ether, tetrahydrofuran and diphenyl ether, aromatic hydrocarbons such as benzene, toluene and xylene, halogenated hydrocarbons such as methylene chloride, chloroform and carbon tetrachloride, pentane and n-hexane And aliphatic hydrocarbons. These solvents may be used alone or as a mixture of two or more thereof.

反応温度は、−60℃から反応混合物の還流温度までの任意の温度を設定することができ、反応時間は、反応基質の濃度、反応温度によって変化するが、通常5分から100時間の範囲で任意に設定できる。   The reaction temperature can be set to any temperature from −60 ° C. to the reflux temperature of the reaction mixture, and the reaction time varies depending on the concentration of the reaction substrate and the reaction temperature, but is usually arbitrary in the range of 5 minutes to 100 hours. Can be set.

反応式3   Reaction formula 3

Figure 2015147757
Figure 2015147757

反応式2に従って合成することのできる式(7−4)で表される化合物を、式(5)[式中Rは前記と同じ意味を表し、Jはハロゲン原子、−OH、−OSOCH、−OSOCF等の脱離基を表す。]で表される化合物と反応させて、式(7−5)[式中A、R、R6a、R、B及びnは前記と同じ意味を表す。]で表される化合物を得ることができる。 A compound represented by the formula (7-4) that can be synthesized according to the reaction formula 2 is represented by the formula (5) [wherein R a represents the same meaning as described above, J b represents a halogen atom, —OH, —OSO. 2 represents a leaving group such as CH 3 and —OSO 2 CF 3 . The compound represented by formula (7-5) [wherein A 1 , R 2 , R 6a , R a , B and n represent the same meaning as described above]. The compound represented by this can be obtained.

本反応は、式(7−4)で表される化合物1当量に対して、式(5)で表される化合物を、0.5〜50当量の範囲で用いることができる。必要ならば塩酸、硫酸、p−トルエンスルホン酸等の酸、炭酸カリウム、トリエチルアミン、ピリジン、4−(ジメチルアミノ)ピリジン、水素化ナトリウム、水酸化ナトリウム、水酸化カリウム等の塩基を使用することができる。   In this reaction, the compound represented by the formula (5) can be used in the range of 0.5 to 50 equivalents with respect to 1 equivalent of the compound represented by the formula (7-4). If necessary, an acid such as hydrochloric acid, sulfuric acid, p-toluenesulfonic acid, a base such as potassium carbonate, triethylamine, pyridine, 4- (dimethylamino) pyridine, sodium hydride, sodium hydroxide, potassium hydroxide may be used. it can.

本反応は、ジエチルアゾジカルボキシレートとトリフェニルホスフィン等を使用する光延反応を使用することができる。   In this reaction, Mitsunobu reaction using diethyl azodicarboxylate and triphenylphosphine can be used.

本反応は、無溶媒でも実施することができるが、溶媒を用いてもよい。例えば、N,N−ジメチルホルムアミド、N,N−ジメチルアセトアミド、アセトニトリル、ジメチルスルホキシド、1,3−ジメチル−2−イミダゾリノン、水等の極性溶媒、メタノール、エタノール、プロパノール、2−プロパノール、エチレングリコール等のアルコール類、ジエチルエーテル、テトラヒドロフラン、ジフェニルエーテル等のエーテル類、ベンゼン、トルエン、キシレン等の芳香族炭化水素類、塩化メチレン、クロロホルム、四塩化炭素等のハロゲン化炭化水素類、ペンタン、n−ヘキサン等の脂肪族炭化水素類が挙げられる。これらの溶媒は単独で用いても、これらの内の2種類以上を混合して用いてもよい。   This reaction can be carried out without solvent, but a solvent may be used. For example, polar solvent such as N, N-dimethylformamide, N, N-dimethylacetamide, acetonitrile, dimethyl sulfoxide, 1,3-dimethyl-2-imidazolinone, water, methanol, ethanol, propanol, 2-propanol, ethylene glycol Alcohols such as diethyl ether, tetrahydrofuran and diphenyl ether, aromatic hydrocarbons such as benzene, toluene and xylene, halogenated hydrocarbons such as methylene chloride, chloroform and carbon tetrachloride, pentane and n-hexane And aliphatic hydrocarbons. These solvents may be used alone or as a mixture of two or more thereof.

反応温度は、−60℃から反応混合物の還流温度までの任意の温度を設定することができ、反応時間は、反応基質の濃度、反応温度によって変化するが、通常5分から100時間の範囲で任意に設定できる。   The reaction temperature can be set to any temperature from −60 ° C. to the reflux temperature of the reaction mixture, and the reaction time varies depending on the concentration of the reaction substrate and the reaction temperature, but is usually arbitrary in the range of 5 minutes to 100 hours. Can be set.

式(5)で表される化合物の或るものは公知化合物であり、一部は市販品として入手できる。また、それ以外のものも文献記載の公知の方法に準じて合成することができる。   Some of the compounds represented by formula (5) are known compounds, and some of them are commercially available. Others can be synthesized according to known methods described in the literature.

引き続き、式(7−5)で表される化合物を、酸又は塩基と反応させて、式(7)で表される化合物を得ることができる。   Subsequently, the compound represented by the formula (7-5) can be reacted with an acid or a base to obtain the compound represented by the formula (7).

酸としては、塩酸、硫酸、p−トルエンスルホン酸、トリフルオロ酢酸等を用いることができる。塩基としては、炭酸カリウム、水酸化ナトリウム等を用いることができる。   As the acid, hydrochloric acid, sulfuric acid, p-toluenesulfonic acid, trifluoroacetic acid and the like can be used. As the base, potassium carbonate, sodium hydroxide or the like can be used.

製造法Cで用いられる式(13)で表される化合物のうち、BがB−8を表す化合物は、例えば以下のようにして合成することが出来る。   Of the compounds represented by formula (13) used in production method C, the compound in which B represents B-8 can be synthesized, for example, as follows.

反応式4   Reaction formula 4

Figure 2015147757
Figure 2015147757

式(7−7)[式中A、R、B及びnは前記と同じ意味を表す。]で表される化合物は、文献既知の方法、例えば、ジャーナル オブ メディシナル ケミストリー 1977年,7巻,2249頁等の公知の方法により製造することができる。 Formula (7-7) [wherein A 1 , R 2 , B and n represent the same meaning as described above. ] Can be produced by a known method in the literature, for example, a known method such as Journal of Medicinal Chemistry 1977, Vol. 7, page 2249.

式(7−7)で表される化合物を、公知のニトロ基の還元法により式(13)で表される化合物を合成することが出来る。   The compound represented by the formula (7-7) can be synthesized from the compound represented by the formula (13) by a known nitro group reduction method.

本発明に包含される活性化合物としては、具体的に例えば第1表に示す化合物が挙げられる。但し、第1表の化合物は例示のためのものであって、本発明はこれらのみに限定されるものではない。尚、表中、Meと記載される置換基はメチル基を表し、以下、Etとの記載はエチル基を表し、n−Pr及びPr−nはノルマルプロピル基を、i−Pr及びPr−iはイソプロピル基を、c−Pr及びPr−cはシクロプロピル基を、n−Bu及びBu−nノルマルブチル基を、s−Bu及びBu−sはセカンダリーブチル基を、i−Bu及びBu−iはイソブチル基を、t−Bu及びBu−tはターシャリーブチル基を、c−Bu及びBu−cはシクロブチル基を、n−Pen及びPen−nはノルマルペンチル基を、c−Pen及びPen−cはシクロペンチル基を、n−Hex及びHex−nはノルマルヘキシル基を、c−Hex及びHex−cはシクロヘキシル基を、Heptはヘプチル基を、Octはオクチル基を、Phはフェニル基をそれぞれ表す。   Specific examples of the active compound included in the present invention include compounds shown in Table 1. However, the compounds in Table 1 are for illustrative purposes, and the present invention is not limited thereto. In the table, the substituent described as Me represents a methyl group, hereinafter, Et represents an ethyl group, n-Pr and Pr-n represent normal propyl groups, i-Pr and Pr-i. Is an isopropyl group, c-Pr and Pr-c are cyclopropyl groups, n-Bu and Bu-n normal butyl groups, s-Bu and Bu-s are secondary butyl groups, i-Bu and Bu-i. Is an isobutyl group, t-Bu and Bu-t are tertiary butyl groups, c-Bu and Bu-c are cyclobutyl groups, n-Pen and Pen-n are normal pentyl groups, c-Pen and Pen- c is a cyclopentyl group, n-Hex and Hex-n are normal hexyl groups, c-Hex and Hex-c are cyclohexyl groups, Hept is a heptyl group, Oct is an octyl group, and Ph is a fethyl group. It represents Le group, respectively.

表中、D1−32a、D1−32b、D1−33a、D1−34a、D1−37a、D1−81a、D1−82a、D1−84a、D1−85a、D1−87a、D1−92a、D1−93a、D1−95a、D1−96a、D1−98a、D1−103b、D1−108a及びD1−108bで表される構造は下記の構造を表し、D1−32bの構造式に記された番号は、Xの置換位置を表し、D1−108bの構造式に記された番号は、Zの置換位置を表す。 In the table, D1-32a, D1-32b, D1-33a, D1-34a, D1-37a, D1-81a, D1-82a, D1-84a, D1-85a, D1-87a, D1-92a, D1-93a , D1-95a, D1-96a, D1-98a, D1-103b, D1-108a, and D1-108b represent the following structures, and the number written in the structural formula of D1-32b is X 1 represents the substitution position, and the number written in the structural formula of D1-108b represents the substitution position of Z.

Figure 2015147757
Figure 2015147757

〔第1表〕 [Table 1]

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

Figure 2015147757
Figure 2015147757

-----------------------------------------------------
R12b R11b
-----------------------------------------------------
H Me
H Et
H Pr-n
H Pr-i
H Pr-c
H Bu-n
H Bu-i
H Bu-c
H Bu-s
H Bu-t
H Pen-n
H Pen-c
H Hex-n
H Hex-c
H CH2Pr-c
H CH2Bu-c
H CH2Pen-c
H CH2Hex-c
H CH2CH=CH2
H CH2CH=C(Cl)2
H CH2C≡CH
H CH2CN
H CH2CF3
H CH2OMe
H CH2OCF3
H CH2SMe
H CH2S(O)Me
H CH2S(O)2Me
H CH2SCF3
H CH2S(O)CF3
H CH2S(O)2CF3
H CH2CH(OMe)2
H CH2CH(SMe)2
H CH2C(O)Me
H CH2C(O)CF3
H CH2C(O)OMe
H CH2(D1-32a)
H CH2(D1-33a)
H CH2(D1-34a)
H CH2(D1-37a)
H CH2(D1-81a)
H CH2(D1-82a)
H CH2(D1-84a)
H CH2(D1-85a)
H CH2(D1-87a)
H CH2(D1-92a)
H CH2(D1-93a)
H CH2(D1-95a)
H CH2(D1-96a)
H CH2(D1-98a)
H CH2(D1-108a)
H CH2(D1-108b,Z=2-Cl)
H CH2(D1-108b,Z=3-Me)
H CH2(D1-108b,Z=4-OMe)
H CH2(D1-108b,Z=2-SMe)
H CH2(D1-108b,Z=3-CF3)
H CH2(D1-108b,Z=4-OCF3)
H CH2(D1-108b,Z=2-SCF3)
H CH2CH2CN
H CH2CH2CF3
H CH2CH2OMe
H CH2CH2SMe
H CH2CH2S(O)Me
H CH2CH2S(O)2Me
H D1-32a
H D1-33a
H D1-34a
H D1-37a
H D1-81a
H D1-82a
H D1-84a
H D1-85a
H D1-87a
H D1-92a
H D1-93a
H D1-95a
H D1-96a
H D1-98a
H D1-108a
H D1-108b(Z=2-Cl)
H D1-108b(Z=3-Me)
H D1-108b(Z=4-OMe)
H D1-108b(Z=2-SMe)
H D1-108b(Z=3-CF3)
H D1-108b(Z=4-OCF3)
H D1-108b(Z=2-SCF3)
H C(O)Me
H C(O)CF3
H C(O)OMe
CF3 Me
CF3 Et
CF3 Pr-n
CF3 Pr-i
CF3 Pr-c
CF3 Bu-n
CF3 Bu-i
CF3 Bu-c
CF3 Bu-s
CF3 Bu-t
CF3 Pen-n
CF3 Pen-c
CF3 Hex-n
CF3 Hex-c
CF3 CH2Pr-c
CF3 CH2Bu-c
CF3 CH2Pen-c
CF3 CH2Hex-c
CF3 CH2CH=CH2
CF3 CH2CH=C(Cl)2
CF3 CH2C≡CH
CF3 CH2CN
CF3 CH2CF3
CF3 CH2OMe
CF3 CH2OCF3
CF3 CH2SMe
CF3 CH2S(O)Me
CF3 CH2S(O)2Me
CF3 CH2SCF3
CF3 CH2S(O)CF3
CF3 CH2S(O)2CF3
CF3 CH2CH(OMe)2
CF3 CH2CH(SMe)2
CF3 CH2C(O)Me
CF3 CH2C(O)CF3
CF3 CH2C(O)OMe
CF3 CH2(D1-32a)
CF3 CH2(D1-33a)
CF3 CH2(D1-34a)
CF3 CH2(D1-37a)
CF3 CH2(D1-81a)
CF3 CH2(D1-82a)
CF3 CH2(D1-84a)
CF3 CH2(D1-85a)
CF3 CH2(D1-87a)
CF3 CH2(D1-92a)
CF3 CH2(D1-93a)
CF3 CH2(D1-95a)
CF3 CH2(D1-96a)
CF3 CH2(D1-98a)
CF3 CH2(D1-108a)
CF3 CH2(D1-108b,Z=2-Cl)
CF3 CH2(D1-108b,Z=3-Me)
CF3 CH2(D1-108b,Z=4-OMe)
CF3 CH2(D1-108b,Z=2-SMe)
CF3 CH2(D1-108b,Z=3-CF3)
CF3 CH2(D1-108b,Z=4-OCF3)
CF3 CH2(D1-108b,Z=2-SCF3)
CF3 CH2CH2CN
CF3 CH2CH2CF3
CF3 CH2CH2OMe
CF3 CH2CH2SMe
CF3 CH2CH2S(O)Me
CF3 CH2CH2S(O)2Me
CF3 D1-32a
CF3 D1-33a
CF3 D1-34a
CF3 D1-37a
CF3 D1-81a
CF3 D1-82a
CF3 D1-84a
CF3 D1-85a
CF3 D1-87a
CF3 D1-92a
CF3 D1-93a
CF3 D1-95a
CF3 D1-96a
CF3 D1-98a
CF3 D1-108a
CF3 D1-108b(Z=2-Cl)
CF3 D1-108b(Z=3-Me)
CF3 D1-108b(Z=4-OMe)
CF3 D1-108b(Z=2-SMe)
CF3 D1-108b(Z=3-CF3)
CF3 D1-108b(Z=4-OCF3)
CF3 D1-108b(Z=2-SCF3)
CF3 C(O)Me
CF3 C(O)CF3
CF3 C(O)OMe
Me Me
Me Et
Me Pr-n
Me Pr-i
Me Pr-c
Me Bu-n
Me Bu-i
Me Bu-c
Me Bu-s
Me Bu-t
Me Pen-n
Me Pen-c
Me Hex-n
Me Hex-c
Me CH2Pr-c
Me CH2Bu-c
Me CH2Pen-c
Me CH2Hex-c
Me CH2CH=CH2
Me CH2CH=C(Cl)2
Me CH2C≡CH
Me CH2CN
Me CH2CF3
Me CH2OMe
Me CH2OCF3
Me CH2SMe
Me CH2S(O)Me
Me CH2S(O)2Me
Me CH2SCF3
Me CH2S(O)CF3
Me CH2S(O)2CF3
Me CH2CH(OMe)2
Me CH2CH(SMe)2
Me CH2C(O)Me
Me CH2C(O)CF3
Me CH2C(O)OMe
Me CH2(D1-32a)
Me CH2(D1-33a)
Me CH2(D1-34a)
Me CH2(D1-37a)
Me CH2(D1-81a)
Me CH2(D1-82a)
Me CH2(D1-84a)
Me CH2(D1-85a)
Me CH2(D1-87a)
Me CH2(D1-92a)
Me CH2(D1-93a)
Me CH2(D1-95a)
Me CH2(D1-96a)
Me CH2(D1-98a)
Me CH2(D1-108a)
Me CH2(D1-108b,Z=2-Cl)
Me CH2(D1-108b,Z=3-Me)
Me CH2(D1-108b,Z=4-OMe)
Me CH2(D1-108b,Z=2-SMe)
Me CH2(D1-108b,Z=3-CF3)
Me CH2(D1-108b,Z=4-OCF3)
Me CH2(D1-108b,Z=2-SCF3)
Me CH2CH2CN
Me CH2CH2CF3
Me CH2CH2OMe
Me CH2CH2SMe
Me CH2CH2S(O)Me
Me CH2CH2S(O)2Me
Me D1-32a
Me D1-33a
Me D1-34a
Me D1-37a
Me D1-81a
Me D1-82a
Me D1-84a
Me D1-85a
Me D1-87a
Me D1-92a
Me D1-93a
Me D1-95a
Me D1-96a
Me D1-98a
Me D1-108a
Me D1-108b(Z=2-Cl)
Me D1-108b(Z=3-Me)
Me D1-108b(Z=4-OMe)
Me D1-108b(Z=2-SMe)
Me D1-108b(Z=3-CF3)
Me D1-108b(Z=4-OCF3)
Me D1-108b(Z=2-SCF3)
Me C(O)Me
Me C(O)CF3
Me C(O)OMe
OMe Me
OMe Et
OMe Pr-n
OMe Pr-i
OMe Pr-c
OMe Bu-n
OMe Bu-i
OMe Bu-c
OMe Bu-s
OMe Bu-t
OMe Pen-n
OMe Pen-c
OMe Hex-n
OMe Hex-c
OMe CH2Pr-c
OMe CH2Bu-c
OMe CH2Pen-c
OMe CH2Hex-c
OMe CH2CH=CH2
OMe CH2CH=C(Cl)2
OMe CH2C≡CH
OMe CH2CN
OMe CH2CF3
OMe CH2OMe
OMe CH2OCF3
OMe CH2SMe
OMe CH2S(O)Me
OMe CH2S(O)2Me
OMe CH2SCF3
OMe CH2S(O)CF3
OMe CH2S(O)2CF3
OMe CH2CH(OMe)2
OMe CH2CH(SMe)2
OMe CH2C(O)Me
OMe CH2C(O)CF3
OMe CH2C(O)OMe
OMe CH2(D1-32a)
OMe CH2(D1-33a)
OMe CH2(D1-34a)
OMe CH2(D1-37a)
OMe CH2(D1-81a)
OMe CH2(D1-82a)
OMe CH2(D1-84a)
OMe CH2(D1-85a)
OMe CH2(D1-87a)
OMe CH2(D1-92a)
OMe CH2(D1-93a)
OMe CH2(D1-95a)
OMe CH2(D1-96a)
OMe CH2(D1-98a)
OMe CH2(D1-108a)
OMe CH2(D1-108b,Z=2-Cl)
OMe CH2(D1-108b,Z=3-Me)
OMe CH2(D1-108b,Z=4-OMe)
OMe CH2(D1-108b,Z=2-SMe)
OMe CH2(D1-108b,Z=3-CF3)
OMe CH2(D1-108b,Z=4-OCF3)
OMe CH2(D1-108b,Z=2-SCF3)
OMe CH2CH2CN
OMe CH2CH2CF3
OMe CH2CH2OMe
OMe CH2CH2SMe
OMe CH2CH2S(O)Me
OMe CH2CH2S(O)2Me
OMe D1-32a
OMe D1-33a
OMe D1-34a
OMe D1-37a
OMe D1-81a
OMe D1-82a
OMe D1-84a
OMe D1-85a
OMe D1-87a
OMe D1-92a
OMe D1-93a
OMe D1-95a
OMe D1-96a
OMe D1-98a
OMe D1-108a
OMe D1-108b(Z=2-Cl)
OMe D1-108b(Z=3-Me)
OMe D1-108b(Z=4-OMe)
OMe D1-108b(Z=2-SMe)
OMe D1-108b(Z=3-CF3)
OMe D1-108b(Z=4-OCF3)
OMe D1-108b(Z=2-SCF3)
OMe C(O)Me
OMe C(O)CF3
OMe C(O)OMe
SMe Me
SMe Et
SMe Pr-n
SMe Pr-i
SMe Pr-c
SMe Bu-n
SMe Bu-i
SMe Bu-c
SMe Bu-s
SMe Bu-t
SMe Pen-n
SMe Pen-c
SMe Hex-n
SMe Hex-c
SMe CH2Pr-c
SMe CH2Bu-c
SMe CH2Pen-c
SMe CH2Hex-c
SMe CH2CH=CH2
SMe CH2CH=C(Cl)2
SMe CH2C≡CH
SMe CH2CN
SMe CH2CF3
SMe CH2OMe
SMe CH2OCF3
SMe CH2SMe
SMe CH2S(O)Me
SMe CH2S(O)2Me
SMe CH2SCF3
SMe CH2S(O)CF3
SMe CH2S(O)2CF3
SMe CH2CH(OMe)2
SMe CH2CH(SMe)2
SMe CH2C(O)Me
SMe CH2C(O)CF3
SMe CH2C(O)OMe
SMe CH2(D1-32a)
SMe CH2(D1-33a)
SMe CH2(D1-34a)
SMe CH2(D1-37a)
SMe CH2(D1-81a)
SMe CH2(D1-82a)
SMe CH2(D1-84a)
SMe CH2(D1-85a)
SMe CH2(D1-87a)
SMe CH2(D1-92a)
SMe CH2(D1-93a)
SMe CH2(D1-95a)
SMe CH2(D1-96a)
SMe CH2(D1-98a)
SMe CH2(D1-108a)
SMe CH2(D1-108b,Z=2-Cl)
SMe CH2(D1-108b,Z=3-Me)
SMe CH2(D1-108b,Z=4-OMe)
SMe CH2(D1-108b,Z=2-SMe)
SMe CH2(D1-108b,Z=3-CF3)
SMe CH2(D1-108b,Z=4-OCF3)
SMe CH2(D1-108b,Z=2-SCF3)
SMe CH2CH2CN
SMe CH2CH2CF3
SMe CH2CH2OMe
SMe CH2CH2SMe
SMe CH2CH2S(O)Me
SMe CH2CH2S(O)2Me
SMe D1-32a
SMe D1-33a
SMe D1-34a
SMe D1-37a
SMe D1-81a
SMe D1-82a
SMe D1-84a
SMe D1-85a
SMe D1-87a
SMe D1-92a
SMe D1-93a
SMe D1-95a
SMe D1-96a
SMe D1-98a
SMe D1-108a
SMe D1-108b(Z=2-Cl)
SMe D1-108b(Z=3-Me)
SMe D1-108b(Z=4-OMe)
SMe D1-108b(Z=2-SMe)
SMe D1-108b(Z=3-CF3)
SMe D1-108b(Z=4-OCF3)
SMe D1-108b(Z=2-SCF3)
SMe C(O)Me
SMe C(O)CF3
SMe C(O)OMe
CH2OMe Me
CH2OMe Et
CH2OMe Pr-n
CH2OMe Pr-i
CH2OMe Pr-c
CH2OMe Bu-n
CH2OMe Bu-i
CH2OMe Bu-c
CH2OMe Bu-s
CH2OMe Bu-t
CH2OMe Pen-n
CH2OMe Pen-c
CH2OMe Hex-n
CH2OMe Hex-c
CH2OMe CH2Pr-c
CH2OMe CH2Bu-c
CH2OMe CH2Pen-c
CH2OMe CH2Hex-c
CH2OMe CH2CH=CH2
CH2OMe CH2CH=C(Cl)2
CH2OMe CH2C≡CH
CH2OMe CH2CN
CH2OMe CH2CF3
CH2OMe CH2OMe
CH2OMe CH2OCF3
CH2OMe CH2SMe
CH2OMe CH2S(O)Me
CH2OMe CH2S(O)2Me
CH2OMe CH2SCF3
CH2OMe CH2S(O)CF3
CH2OMe CH2S(O)2CF3
CH2OMe CH2CH(OMe)2
CH2OMe CH2CH(SMe)2
CH2OMe CH2C(O)Me
CH2OMe CH2C(O)CF3
CH2OMe CH2C(O)OMe
CH2OMe CH2(D1-32a)
CH2OMe CH2(D1-33a)
CH2OMe CH2(D1-34a)
CH2OMe CH2(D1-37a)
CH2OMe CH2(D1-81a)
CH2OMe CH2(D1-82a)
CH2OMe CH2(D1-84a)
CH2OMe CH2(D1-85a)
CH2OMe CH2(D1-87a)
CH2OMe CH2(D1-92a)
CH2OMe CH2(D1-93a)
CH2OMe CH2(D1-95a)
CH2OMe CH2(D1-96a)
CH2OMe CH2(D1-98a)
CH2OMe CH2(D1-108a)
CH2OMe CH2(D1-108b,Z=2-Cl)
CH2OMe CH2(D1-108b,Z=3-Me)
CH2OMe CH2(D1-108b,Z=4-OMe)
CH2OMe CH2(D1-108b,Z=2-SMe)
CH2OMe CH2(D1-108b,Z=3-CF3)
CH2OMe CH2(D1-108b,Z=4-OCF3)
CH2OMe CH2(D1-108b,Z=2-SCF3)
CH2OMe CH2CH2CN
CH2OMe CH2CH2CF3
CH2OMe CH2CH2OMe
CH2OMe CH2CH2SMe
CH2OMe CH2CH2S(O)Me
CH2OMe CH2CH2S(O)2Me
CH2OMe D1-32a
CH2OMe D1-33a
CH2OMe D1-34a
CH2OMe D1-37a
CH2OMe D1-81a
CH2OMe D1-82a
CH2OMe D1-84a
CH2OMe D1-85a
CH2OMe D1-87a
CH2OMe D1-92a
CH2OMe D1-93a
CH2OMe D1-95a
CH2OMe D1-96a
CH2OMe D1-98a
CH2OMe D1-108a
CH2OMe D1-108b(Z=2-Cl)
CH2OMe D1-108b(Z=3-Me)
CH2OMe D1-108b(Z=4-OMe)
CH2OMe D1-108b(Z=2-SMe)
CH2OMe D1-108b(Z=3-CF3)
CH2OMe D1-108b(Z=4-OCF3)
CH2OMe D1-108b(Z=2-SCF3)
CH2OMe C(O)Me
CH2OMe C(O)CF3
CH2OMe C(O)OMe
CH2SMe Me
CH2SMe Et
CH2SMe Pr-n
CH2SMe Pr-i
CH2SMe Pr-c
CH2SMe Bu-n
CH2SMe Bu-i
CH2SMe Bu-c
CH2SMe Bu-s
CH2SMe Bu-t
CH2SMe Pen-n
CH2SMe Pen-c
CH2SMe Hex-n
CH2SMe Hex-c
CH2SMe CH2Pr-c
CH2SMe CH2Bu-c
CH2SMe CH2Pen-c
CH2SMe CH2Hex-c
CH2SMe CH2CH=CH2
CH2SMe CH2CH=C(Cl)2
CH2SMe CH2C≡CH
CH2SMe CH2CN
CH2SMe CH2CF3
CH2SMe CH2OMe
CH2SMe CH2OCF3
CH2SMe CH2SMe
CH2SMe CH2S(O)Me
CH2SMe CH2S(O)2Me
CH2SMe CH2SCF3
CH2SMe CH2S(O)CF3
CH2SMe CH2S(O)2CF3
CH2SMe CH2CH(OMe)2
CH2SMe CH2CH(SMe)2
CH2SMe CH2C(O)Me
CH2SMe CH2C(O)CF3
CH2SMe CH2C(O)OMe
CH2SMe CH2(D1-32a)
CH2SMe CH2(D1-33a)
CH2SMe CH2(D1-34a)
CH2SMe CH2(D1-37a)
CH2SMe CH2(D1-81a)
CH2SMe CH2(D1-82a)
CH2SMe CH2(D1-84a)
CH2SMe CH2(D1-85a)
CH2SMe CH2(D1-87a)
CH2SMe CH2(D1-92a)
CH2SMe CH2(D1-93a)
CH2SMe CH2(D1-95a)
CH2SMe CH2(D1-96a)
CH2SMe CH2(D1-98a)
CH2SMe CH2(D1-108a)
CH2SMe CH2(D1-108b,Z=2-Cl)
CH2SMe CH2(D1-108b,Z=3-Me)
CH2SMe CH2(D1-108b,Z=4-OMe)
CH2SMe CH2(D1-108b,Z=2-SMe)
CH2SMe CH2(D1-108b,Z=3-CF3)
CH2SMe CH2(D1-108b,Z=4-OCF3)
CH2SMe CH2(D1-108b,Z=2-SCF3)
CH2SMe CH2CH2CN
CH2SMe CH2CH2CF3
CH2SMe CH2CH2OMe
CH2SMe CH2CH2SMe
CH2SMe CH2CH2S(O)Me
CH2SMe CH2CH2S(O)2Me
CH2SMe D1-32a
CH2SMe D1-33a
CH2SMe D1-34a
CH2SMe D1-37a
CH2SMe D1-81a
CH2SMe D1-82a
CH2SMe D1-84a
CH2SMe D1-85a
CH2SMe D1-87a
CH2SMe D1-92a
CH2SMe D1-93a
CH2SMe D1-95a
CH2SMe D1-96a
CH2SMe D1-98a
CH2SMe D1-108a
CH2SMe D1-108b(Z=2-Cl)
CH2SMe D1-108b(Z=3-Me)
CH2SMe D1-108b(Z=4-OMe)
CH2SMe D1-108b(Z=2-SMe)
CH2SMe D1-108b(Z=3-CF3)
CH2SMe D1-108b(Z=4-OCF3)
CH2SMe D1-108b(Z=2-SCF3)
CH2SMe C(O)Me
CH2SMe C(O)CF3
CH2SMe C(O)OMe
CH2S(O)Me Me
CH2S(O)Me Et
CH2S(O)Me Pr-n
CH2S(O)Me Pr-i
CH2S(O)Me Pr-c
CH2S(O)Me Bu-n
CH2S(O)Me Bu-i
CH2S(O)Me Bu-c
CH2S(O)Me Bu-s
CH2S(O)Me Bu-t
CH2S(O)Me Pen-n
CH2S(O)Me Pen-c
CH2S(O)Me Hex-n
CH2S(O)Me Hex-c
CH2S(O)Me CH2Pr-c
CH2S(O)Me CH2Bu-c
CH2S(O)Me CH2Pen-c
CH2S(O)Me CH2Hex-c
CH2S(O)Me CH2CH=CH2
CH2S(O)Me CH2CH=C(Cl)2
CH2S(O)Me CH2C≡CH
CH2S(O)Me CH2CN
CH2S(O)Me CH2CF3
CH2S(O)Me CH2OMe
CH2S(O)Me CH2OCF3
CH2S(O)Me CH2SMe
CH2S(O)Me CH2S(O)Me
CH2S(O)Me CH2S(O)2Me
CH2S(O)Me CH2SCF3
CH2S(O)Me CH2S(O)CF3
CH2S(O)Me CH2S(O)2CF3
CH2S(O)Me CH2CH(OMe)2
CH2S(O)Me CH2CH(SMe)2
CH2S(O)Me CH2C(O)Me
CH2S(O)Me CH2C(O)CF3
CH2S(O)Me CH2C(O)OMe
CH2S(O)Me CH2(D1-32a)
CH2S(O)Me CH2(D1-33a)
CH2S(O)Me CH2(D1-34a)
CH2S(O)Me CH2(D1-37a)
CH2S(O)Me CH2(D1-81a)
CH2S(O)Me CH2(D1-82a)
CH2S(O)Me CH2(D1-84a)
CH2S(O)Me CH2(D1-85a)
CH2S(O)Me CH2(D1-87a)
CH2S(O)Me CH2(D1-92a)
CH2S(O)Me CH2(D1-93a)
CH2S(O)Me CH2(D1-95a)
CH2S(O)Me CH2(D1-96a)
CH2S(O)Me CH2(D1-98a)
CH2S(O)Me CH2(D1-108a)
CH2S(O)Me CH2(D1-108b,Z=2-Cl)
CH2S(O)Me CH2(D1-108b,Z=3-Me)
CH2S(O)Me CH2(D1-108b,Z=4-OMe)
CH2S(O)Me CH2(D1-108b,Z=2-SMe)
CH2S(O)Me CH2(D1-108b,Z=3-CF3)
CH2S(O)Me CH2(D1-108b,Z=4-OCF3)
CH2S(O)Me CH2(D1-108b,Z=2-SCF3)
CH2S(O)Me CH2CH2CN
CH2S(O)Me CH2CH2CF3
CH2S(O)Me CH2CH2OMe
CH2S(O)Me CH2CH2SMe
CH2S(O)Me CH2CH2S(O)Me
CH2S(O)Me CH2CH2S(O)2Me
CH2S(O)Me D1-32a
CH2S(O)Me D1-33a
CH2S(O)Me D1-34a
CH2S(O)Me D1-37a
CH2S(O)Me D1-81a
CH2S(O)Me D1-82a
CH2S(O)Me D1-84a
CH2S(O)Me D1-85a
CH2S(O)Me D1-87a
CH2S(O)Me D1-92a
CH2S(O)Me D1-93a
CH2S(O)Me D1-95a
CH2S(O)Me D1-96a
CH2S(O)Me D1-98a
CH2S(O)Me D1-108a
CH2S(O)Me D1-108b(Z=2-Cl)
CH2S(O)Me D1-108b(Z=3-Me)
CH2S(O)Me D1-108b(Z=4-OMe)
CH2S(O)Me D1-108b(Z=2-SMe)
CH2S(O)Me D1-108b(Z=3-CF3)
CH2S(O)Me D1-108b(Z=4-OCF3)
CH2S(O)Me D1-108b(Z=2-SCF3)
CH2S(O)Me C(O)Me
CH2S(O)Me C(O)CF3
CH2S(O)Me C(O)OMe
CH2S(O)2Me Me
CH2S(O)2Me Et
CH2S(O)2Me Pr-n
CH2S(O)2Me Pr-i
CH2S(O)2Me Pr-c
CH2S(O)2Me Bu-n
CH2S(O)2Me Bu-i
CH2S(O)2Me Bu-c
CH2S(O)2Me Bu-s
CH2S(O)2Me Bu-t
CH2S(O)2Me Pen-n
CH2S(O)2Me Pen-c
CH2S(O)2Me Hex-n
CH2S(O)2Me Hex-c
CH2S(O)2Me CH2Pr-c
CH2S(O)2Me CH2Bu-c
CH2S(O)2Me CH2Pen-c
CH2S(O)2Me CH2Hex-c
CH2S(O)2Me CH2CH=CH2
CH2S(O)2Me CH2CH=C(Cl)2
CH2S(O)2Me CH2C≡CH
CH2S(O)2Me CH2CN
CH2S(O)2Me CH2CF3
CH2S(O)2Me CH2OMe
CH2S(O)2Me CH2OCF3
CH2S(O)2Me CH2SMe
CH2S(O)2Me CH2S(O)Me
CH2S(O)2Me CH2S(O)2Me
CH2S(O)2Me CH2SCF3
CH2S(O)2Me CH2S(O)CF3
CH2S(O)2Me CH2S(O)2CF3
CH2S(O)2Me CH2CH(OMe)2
CH2S(O)2Me CH2CH(SMe)2
CH2S(O)2Me CH2C(O)Me
CH2S(O)2Me CH2C(O)CF3
CH2S(O)2Me CH2C(O)OMe
CH2S(O)2Me CH2(D1-32a)
CH2S(O)2Me CH2(D1-33a)
CH2S(O)2Me CH2(D1-34a)
CH2S(O)2Me CH2(D1-37a)
CH2S(O)2Me CH2(D1-81a)
CH2S(O)2Me CH2(D1-82a)
CH2S(O)2Me CH2(D1-84a)
CH2S(O)2Me CH2(D1-85a)
CH2S(O)2Me CH2(D1-87a)
CH2S(O)2Me CH2(D1-92a)
CH2S(O)2Me CH2(D1-93a)
CH2S(O)2Me CH2(D1-95a)
CH2S(O)2Me CH2(D1-96a)
CH2S(O)2Me CH2(D1-98a)
CH2S(O)2Me CH2(D1-108a)
CH2S(O)2Me CH2(D1-108b,Z=2-Cl)
CH2S(O)2Me CH2(D1-108b,Z=3-Me)
CH2S(O)2Me CH2(D1-108b,Z=4-OMe)
CH2S(O)2Me CH2(D1-108b,Z=2-SMe)
CH2S(O)2Me CH2(D1-108b,Z=3-CF3)
CH2S(O)2Me CH2(D1-108b,Z=4-OCF3)
CH2S(O)2Me CH2(D1-108b,Z=2-SCF3)
CH2S(O)2Me CH2CH2CN
CH2S(O)2Me CH2CH2CF3
CH2S(O)2Me CH2CH2OMe
CH2S(O)2Me CH2CH2SMe
CH2S(O)2Me CH2CH2S(O)Me
CH2S(O)2Me CH2CH2S(O)2Me
CH2S(O)2Me D1-32a
CH2S(O)2Me D1-33a
CH2S(O)2Me D1-34a
CH2S(O)2Me D1-37a
CH2S(O)2Me D1-81a
CH2S(O)2Me D1-82a
CH2S(O)2Me D1-84a
CH2S(O)2Me D1-85a
CH2S(O)2Me D1-87a
CH2S(O)2Me D1-92a
CH2S(O)2Me D1-93a
CH2S(O)2Me D1-95a
CH2S(O)2Me D1-96a
CH2S(O)2Me D1-98a
CH2S(O)2Me D1-108a
CH2S(O)2Me D1-108b(Z=2-Cl)
CH2S(O)2Me D1-108b(Z=3-Me)
CH2S(O)2Me D1-108b(Z=4-OMe)
CH2S(O)2Me D1-108b(Z=2-SMe)
CH2S(O)2Me D1-108b(Z=3-CF3)
CH2S(O)2Me D1-108b(Z=4-OCF3)
CH2S(O)2Me D1-108b(Z=2-SCF3)
CH2S(O)2Me C(O)Me
CH2S(O)2Me C(O)CF3
CH2S(O)2Me C(O)OMe
CH(Me)SMe Me
CH(Me)SMe Et
CH(Me)SMe Pr-n
CH(Me)SMe Pr-i
CH(Me)SMe Pr-c
CH(Me)SMe Bu-n
CH(Me)SMe Bu-i
CH(Me)SMe Bu-c
CH(Me)SMe Bu-s
CH(Me)SMe Bu-t
CH(Me)SMe Pen-n
CH(Me)SMe Pen-c
CH(Me)SMe Hex-n
CH(Me)S(O)Me Me
CH(Me)S(O)Me Et
CH(Me)S(O)Me Pr-n
CH(Me)S(O)Me Pr-i
CH(Me)S(O)Me Pr-c
CH(Me)S(O)Me Bu-n
CH(Me)S(O)Me Bu-i
CH(Me)S(O)Me Bu-c
CH(Me)S(O)Me Bu-s
CH(Me)S(O)Me Bu-t
CH(Me)S(O)Me Pen-n
CH(Me)S(O)Me Pen-c
CH(Me)S(O)Me Hex-n
CH(Me)S(O)2Me Me
CH(Me)S(O)2Me Et
CH(Me)S(O)2Me Pr-n
CH(Me)S(O)2Me Pr-i
CH(Me)S(O)2Me Pr-c
CH(Me)S(O)2Me Bu-n
CH(Me)S(O)2Me Bu-i
CH(Me)S(O)2Me Bu-c
CH(Me)S(O)2Me Bu-s
CH(Me)S(O)2Me Bu-t
CH(Me)S(O)2Me Pen-n
CH(Me)S(O)2Me Pen-c
CH(Me)S(O)2Me Hex-n
CH(Et)SMe Me
CH(Et)SMe Et
CH(Et)SMe Pr-n
CH(Et)SMe Pr-i
CH(Et)SMe Pr-c
CH(Et)SMe Bu-n
CH(Et)SMe Bu-i
CH(Et)SMe Bu-c
CH(Et)SMe Bu-s
CH(Et)SMe Bu-t
CH(Et)SMe Pen-n
CH(Et)SMe Pen-c
CH(Et)SMe Hex-n
CH(Et)S(O)Me Me
CH(Et)S(O)Me Et
CH(Et)S(O)Me Pr-n
CH(Et)S(O)Me Pr-i
CH(Et)S(O)Me Pr-c
CH(Et)S(O)Me Bu-n
CH(Et)S(O)Me Bu-i
CH(Et)S(O)Me Bu-c
CH(Et)S(O)Me Bu-s
CH(Et)S(O)Me Bu-t
CH(Et)S(O)Me Pen-n
CH(Et)S(O)Me Pen-c
CH(Et)S(O)Me Hex-n
CH(Et)S(O)2Me Me
CH(Et)S(O)2Me Et
CH(Et)S(O)2Me Pr-n
CH(Et)S(O)2Me Pr-i
CH(Et)S(O)2Me Pr-c
CH(Et)S(O)2Me Bu-n
CH(Et)S(O)2Me Bu-i
CH(Et)S(O)2Me Bu-c
CH(Et)S(O)2Me Bu-s
CH(Et)S(O)2Me Bu-t
CH(Et)S(O)2Me Pen-n
CH(Et)S(O)2Me Pen-c
CH(Et)S(O)2Me Hex-n
CH(Me)SEt Me
CH(Me)SEt Et
CH(Me)SEt Pr-n
CH(Me)SEt Pr-i
CH(Me)SEt Pr-c
CH(Me)SEt Bu-n
CH(Me)SEt Bu-i
CH(Me)SEt Bu-c
CH(Me)SEt Bu-s
CH(Me)SEt Bu-t
CH(Me)SEt Pen-n
CH(Me)SEt Pen-c
CH(Me)SEt Hex-n
CH(Me)S(O)Et Me
CH(Me)S(O)Et Et
CH(Me)S(O)Et Pr-n
CH(Me)S(O)Et Pr-i
CH(Me)S(O)Et Pr-c
CH(Me)S(O)Et Bu-n
CH(Me)S(O)Et Bu-i
CH(Me)S(O)Et Bu-c
CH(Me)S(O)Et Bu-s
CH(Me)S(O)Et Bu-t
CH(Me)S(O)Et Pen-n
CH(Me)S(O)Et Pen-c
CH(Me)S(O)Et Hex-n
CH(Me)S(O)2Et Me
CH(Me)S(O)2Et Et
CH(Me)S(O)2Et Pr-n
CH(Me)S(O)2Et Pr-i
CH(Me)S(O)2Et Pr-c
CH(Me)S(O)2Et Bu-n
CH(Me)S(O)2Et Bu-i
CH(Me)S(O)2Et Bu-c
CH(Me)S(O)2Et Bu-s
CH(Me)S(O)2Et Bu-t
CH(Me)S(O)2Et Pen-n
CH(Me)S(O)2Et Pen-c
CH(Me)S(O)2Et Hex-n
CH(Et)SEt Me
CH(Et)SEt Et
CH(Et)SEt Pr-n
CH(Et)SEt Pr-i
CH(Et)SEt Pr-c
CH(Et)SEt Bu-n
CH(Et)SEt Bu-i
CH(Et)SEt Bu-c
CH(Et)SEt Bu-s
CH(Et)SEt Bu-t
CH(Et)SEt Pen-n
CH(Et)SEt Pen-c
CH(Et)SEt Hex-n
CH(Et)S(O)Et Me
CH(Et)S(O)Et Et
CH(Et)S(O)Et Pr-n
CH(Et)S(O)Et Pr-i
CH(Et)S(O)Et Pr-c
CH(Et)S(O)Et Bu-n
CH(Et)S(O)Et Bu-i
CH(Et)S(O)Et Bu-c
CH(Et)S(O)Et Bu-s
CH(Et)S(O)Et Bu-t
CH(Et)S(O)Et Pen-n
CH(Et)S(O)Et Pen-c
CH(Et)S(O)Et Hex-n
CH(Et)S(O)2Et Me
CH(Et)S(O)2Et Et
CH(Et)S(O)2Et Pr-n
CH(Et)S(O)2Et Pr-i
CH(Et)S(O)2Et Pr-c
CH(Et)S(O)2Et Bu-n
CH(Et)S(O)2Et Bu-i
CH(Et)S(O)2Et Bu-c
CH(Et)S(O)2Et Bu-s
CH(Et)S(O)2Et Bu-t
CH(Et)S(O)2Et Pen-n
CH(Et)S(O)2Et Pen-c
CH(Et)S(O)2Et Hex-n
CH2SCH2CH2CN Me
CH2SCH2CH2CN Et
CH2SCH2CH2CN Pr-n
CH2SCH2CH2CN Pr-i
CH2SCH2CH2CN Pr-c
CH2SCH2CH2CN Bu-n
CH2SCH2CH2CN Bu-i
CH2SCH2CH2CN Bu-c
CH2SCH2CH2CN Bu-s
CH2SCH2CH2CN Bu-t
CH2SCH2CH2CN Pen-n
CH2SCH2CH2CN Pen-c
CH2SCH2CH2CN Hex-n
CH2S(O)CH2CH2CN Me
CH2S(O)CH2CH2CN Et
CH2S(O)CH2CH2CN Pr-n
CH2S(O)CH2CH2CN Pr-i
CH2S(O)CH2CH2CN Pr-c
CH2S(O)CH2CH2CN Bu-n
CH2S(O)CH2CH2CN Bu-i
CH2S(O)CH2CH2CN Bu-c
CH2S(O)CH2CH2CN Bu-s
CH2S(O)CH2CH2CN Bu-t
CH2S(O)CH2CH2CN Pen-n
CH2S(O)CH2CH2CN Pen-c
CH2S(O)CH2CH2CN Hex-n
CH2S(O)2CH2CH2CN Me
CH2S(O)2CH2CH2CN Et
CH2S(O)2CH2CH2CN Pr-n
CH2S(O)2CH2CH2CN Pr-i
CH2S(O)2CH2CH2CN Pr-c
CH2S(O)2CH2CH2CN Bu-n
CH2S(O)2CH2CH2CN Bu-i
CH2S(O)2CH2CH2CN Bu-c
CH2S(O)2CH2CH2CN Bu-s
CH2S(O)2CH2CH2CN Bu-t
CH2S(O)2CH2CH2CN Pen-n
CH2S(O)2CH2CH2CN Pen-c
CH2S(O)2CH2CH2CN Hex-n
CH(Me)SCH2CH2CN Me
CH(Me)SCH2CH2CN Et
CH(Me)SCH2CH2CN Pr-n
CH(Me)SCH2CH2CN Pr-i
CH(Me)SCH2CH2CN Pr-c
CH(Me)SCH2CH2CN Bu-n
CH(Me)SCH2CH2CN Bu-i
CH(Me)SCH2CH2CN Bu-c
CH(Me)SCH2CH2CN Bu-s
CH(Me)SCH2CH2CN Bu-t
CH(Me)SCH2CH2CN Pen-n
CH(Me)SCH2CH2CN Pen-c
CH(Me)SCH2CH2CN Hex-n
CH(Me)S(O)CH2CH2CN Me
CH(Me)S(O)CH2CH2CN Et
CH(Me)S(O)CH2CH2CN Pr-n
CH(Me)S(O)CH2CH2CN Pr-i
CH(Me)S(O)CH2CH2CN Pr-c
CH(Me)S(O)CH2CH2CN Bu-n
CH(Me)S(O)CH2CH2CN Bu-i
CH(Me)S(O)CH2CH2CN Bu-c
CH(Me)S(O)CH2CH2CN Bu-s
CH(Me)S(O)CH2CH2CN Bu-t
CH(Me)S(O)CH2CH2CN Pen-n
CH(Me)S(O)CH2CH2CN Pen-c
CH(Me)S(O)CH2CH2CN Hex-n
CH(Me)S(O)2CH2CH2CN Me
CH(Me)S(O)2CH2CH2CN Et
CH(Me)S(O)2CH2CH2CN Pr-n
CH(Me)S(O)2CH2CH2CN Pr-i
CH(Me)S(O)2CH2CH2CN Pr-c
CH(Me)S(O)2CH2CH2CN Bu-n
CH(Me)S(O)2CH2CH2CN Bu-i
CH(Me)S(O)2CH2CH2CN Bu-c
CH(Me)S(O)2CH2CH2CN Bu-s
CH(Me)S(O)2CH2CH2CN Bu-t
CH(Me)S(O)2CH2CH2CN Pen-n
CH(Me)S(O)2CH2CH2CN Pen-c
CH(Me)S(O)2CH2CH2CN Hex-n
CH(Et)SCH2CH2CN Me
CH(Et)SCH2CH2CN Et
CH(Et)SCH2CH2CN Pr-n
CH(Et)SCH2CH2CN Pr-i
CH(Et)SCH2CH2CN Pr-c
CH(Et)SCH2CH2CN Bu-n
CH(Et)SCH2CH2CN Bu-i
CH(Et)SCH2CH2CN Bu-c
CH(Et)SCH2CH2CN Bu-s
CH(Et)SCH2CH2CN Bu-t
CH(Et)SCH2CH2CN Pen-n
CH(Et)SCH2CH2CN Pen-c
CH(Et)SCH2CH2CN Hex-n
CH(Et)S(O)CH2CH2CN Me
CH(Et)S(O)CH2CH2CN Et
CH(Et)S(O)CH2CH2CN Pr-n
CH(Et)S(O)CH2CH2CN Pr-i
CH(Et)S(O)CH2CH2CN Pr-c
CH(Et)S(O)CH2CH2CN Bu-n
CH(Et)S(O)CH2CH2CN Bu-i
CH(Et)S(O)CH2CH2CN Bu-c
CH(Et)S(O)CH2CH2CN Bu-s
CH(Et)S(O)CH2CH2CN Bu-t
CH(Et)S(O)CH2CH2CN Pen-n
CH(Et)S(O)CH2CH2CN Pen-c
CH(Et)S(O)CH2CH2CN Hex-n
CH(Et)S(O)2CH2CH2CN Me
CH(Et)S(O)2CH2CH2CN Et
CH(Et)S(O)2CH2CH2CN Pr-n
CH(Et)S(O)2CH2CH2CN Pr-i
CH(Et)S(O)2CH2CH2CN Pr-c
CH(Et)S(O)2CH2CH2CN Bu-n
CH(Et)S(O)2CH2CH2CN Bu-i
CH(Et)S(O)2CH2CH2CN Bu-c
CH(Et)S(O)2CH2CH2CN Bu-s
CH(Et)S(O)2CH2CH2CN Bu-t
CH(Et)S(O)2CH2CH2CN Pen-n
CH(Et)S(O)2CH2CH2CN Pen-c
CH(Et)S(O)2CH2CH2CN Hex-n
CH2SC(O)Me Me
CH2CH2SC(O)Me Me
CH(Me)SC(O)Me Me
CH(Me)CH2SC(O)Me Me
CH(Et)SC(O)Me Me
CH(Et)CH2SC(O)Me Me
CH2SCF3 Me
CH2SCF3 Et
CH2SCF3 Pr-n
CH2SCF3 Pr-i
CH2SCF3 Pr-c
CH2SCF3 Bu-n
CH2SCF3 Bu-i
CH2SCF3 Bu-c
CH2SCF3 Bu-s
CH2SCF3 Bu-t
CH2SCF3 Pen-n
CH2SCF3 Pen-c
CH2SCF3 Hex-n
CH2SCF3 Hex-c
CH2SCF3 CH2Pr-c
CH2SCF3 CH2Bu-c
CH2SCF3 CH2Pen-c
CH2SCF3 CH2Hex-c
CH2SCF3 CH2CH=CH2
CH2SCF3 CH2CH=C(Cl)2
CH2SCF3 CH2C≡CH
CH2SCF3 CH2CN
CH2SCF3 CH2CF3
CH2SCF3 CH2OMe
CH2SCF3 CH2OCF3
CH2SCF3 CH2SMe
CH2SCF3 CH2S(O)Me
CH2SCF3 CH2S(O)2Me
CH2SCF3 CH2SCF3
CH2SCF3 CH2S(O)CF3
CH2SCF3 CH2S(O)2CF3
CH2SCF3 CH2CH(OMe)2
CH2SCF3 CH2CH(SMe)2
CH2SCF3 CH2C(O)Me
CH2SCF3 CH2C(O)CF3
CH2SCF3 CH2C(O)OMe
CH2SCF3 CH2(D1-32a)
CH2SCF3 CH2(D1-33a)
CH2SCF3 CH2(D1-34a)
CH2SCF3 CH2(D1-37a)
CH2SCF3 CH2(D1-81a)
CH2SCF3 CH2(D1-82a)
CH2SCF3 CH2(D1-84a)
CH2SCF3 CH2(D1-85a)
CH2SCF3 CH2(D1-87a)
CH2SCF3 CH2(D1-92a)
CH2SCF3 CH2(D1-93a)
CH2SCF3 CH2(D1-95a)
CH2SCF3 CH2(D1-96a)
CH2SCF3 CH2(D1-98a)
CH2SCF3 CH2(D1-108a)
CH2SCF3 CH2(D1-108b,Z=2-Cl)
CH2SCF3 CH2(D1-108b,Z=3-Me)
CH2SCF3 CH2(D1-108b,Z=4-OMe)
CH2SCF3 CH2(D1-108b,Z=2-SMe)
CH2SCF3 CH2(D1-108b,Z=3-CF3)
CH2SCF3 CH2(D1-108b,Z=4-OCF3)
CH2SCF3 CH2(D1-108b,Z=2-SCF3)
CH2SCF3 CH2CH2CN
CH2SCF3 CH2CH2CF3
CH2SCF3 CH2CH2OMe
CH2SCF3 CH2CH2SMe
CH2SCF3 CH2CH2S(O)Me
CH2SCF3 CH2CH2S(O)2Me
CH2SCF3 D1-32a
CH2SCF3 D1-33a
CH2SCF3 D1-34a
CH2SCF3 D1-37a
CH2SCF3 D1-81a
CH2SCF3 D1-82a
CH2SCF3 D1-84a
CH2SCF3 D1-85a
CH2SCF3 D1-87a
CH2SCF3 D1-92a
CH2SCF3 D1-93a
CH2SCF3 D1-95a
CH2SCF3 D1-96a
CH2SCF3 D1-98a
CH2SCF3 D1-108a
CH2SCF3 D1-108b(Z=2-Cl)
CH2SCF3 D1-108b(Z=3-Me)
CH2SCF3 D1-108b(Z=4-OMe)
CH2SCF3 D1-108b(Z=2-SMe)
CH2SCF3 D1-108b(Z=3-CF3)
CH2SCF3 D1-108b(Z=4-OCF3)
CH2SCF3 D1-108b(Z=2-SCF3)
CH2SCF3 C(O)Me
CH2SCF3 C(O)CF3
CH2SCF3 C(O)OMe
CH2S(O)CF3 Me
CH2S(O)CF3 Et
CH2S(O)CF3 Pr-n
CH2S(O)CF3 Pr-i
CH2S(O)CF3 Pr-c
CH2S(O)CF3 Bu-n
CH2S(O)CF3 Bu-i
CH2S(O)CF3 Bu-c
CH2S(O)CF3 Bu-s
CH2S(O)CF3 Bu-t
CH2S(O)CF3 Pen-n
CH2S(O)CF3 Pen-c
CH2S(O)CF3 Hex-n
CH2S(O)CF3 Hex-c
CH2S(O)CF3 CH2Pr-c
CH2S(O)CF3 CH2Bu-c
CH2S(O)CF3 CH2Pen-c
CH2S(O)CF3 CH2Hex-c
CH2S(O)CF3 CH2CH=CH2
CH2S(O)CF3 CH2CH=C(Cl)2
CH2S(O)CF3 CH2C≡CH
CH2S(O)CF3 CH2CN
CH2S(O)CF3 CH2CF3
CH2S(O)CF3 CH2OMe
CH2S(O)CF3 CH2OCF3
CH2S(O)CF3 CH2SMe
CH2S(O)CF3 CH2S(O)Me
CH2S(O)CF3 CH2S(O)2Me
CH2S(O)CF3 CH2SCF3
CH2S(O)CF3 CH2S(O)CF3
CH2S(O)CF3 CH2S(O)2CF3
CH2S(O)CF3 CH2CH(OMe)2
CH2S(O)CF3 CH2CH(SMe)2
CH2S(O)CF3 CH2C(O)Me
CH2S(O)CF3 CH2C(O)CF3
CH2S(O)CF3 CH2C(O)OMe
CH2S(O)CF3 CH2(D1-32a)
CH2S(O)CF3 CH2(D1-33a)
CH2S(O)CF3 CH2(D1-34a)
CH2S(O)CF3 CH2(D1-37a)
CH2S(O)CF3 CH2(D1-81a)
CH2S(O)CF3 CH2(D1-82a)
CH2S(O)CF3 CH2(D1-84a)
CH2S(O)CF3 CH2(D1-85a)
CH2S(O)CF3 CH2(D1-87a)
CH2S(O)CF3 CH2(D1-92a)
CH2S(O)CF3 CH2(D1-93a)
CH2S(O)CF3 CH2(D1-95a)
CH2S(O)CF3 CH2(D1-96a)
CH2S(O)CF3 CH2(D1-98a)
CH2S(O)CF3 CH2(D1-108a)
CH2S(O)CF3 CH2(D1-108b,Z=2-Cl)
CH2S(O)CF3 CH2(D1-108b,Z=3-Me)
CH2S(O)CF3 CH2(D1-108b,Z=4-OMe)
CH2S(O)CF3 CH2(D1-108b,Z=2-SMe)
CH2S(O)CF3 CH2(D1-108b,Z=3-CF3)
CH2S(O)CF3 CH2(D1-108b,Z=4-OCF3)
CH2S(O)CF3 CH2(D1-108b,Z=2-SCF3)
CH2S(O)CF3 CH2CH2CN
CH2S(O)CF3 CH2CH2CF3
CH2S(O)CF3 CH2CH2OMe
CH2S(O)CF3 CH2CH2SMe
CH2S(O)CF3 CH2CH2S(O)Me
CH2S(O)CF3 CH2CH2S(O)2Me
CH2S(O)CF3 D1-32a
CH2S(O)CF3 D1-33a
CH2S(O)CF3 D1-34a
CH2S(O)CF3 D1-37a
CH2S(O)CF3 D1-81a
CH2S(O)CF3 D1-82a
CH2S(O)CF3 D1-84a
CH2S(O)CF3 D1-85a
CH2S(O)CF3 D1-87a
CH2S(O)CF3 D1-92a
CH2S(O)CF3 D1-93a
CH2S(O)CF3 D1-95a
CH2S(O)CF3 D1-96a
CH2S(O)CF3 D1-98a
CH2S(O)CF3 D1-108a
CH2S(O)CF3 D1-108b(Z=2-Cl)
CH2S(O)CF3 D1-108b(Z=3-Me)
CH2S(O)CF3 D1-108b(Z=4-OMe)
CH2S(O)CF3 D1-108b(Z=2-SMe)
CH2S(O)CF3 D1-108b(Z=3-CF3)
CH2S(O)CF3 D1-108b(Z=4-OCF3)
CH2S(O)CF3 D1-108b(Z=2-SCF3)
CH2S(O)CF3 C(O)Me
CH2S(O)CF3 C(O)CF3
CH2S(O)CF3 C(O)OMe
CH2S(O)2CF3 Me
CH2S(O)2CF3 Et
CH2S(O)2CF3 Pr-n
CH2S(O)2CF3 Pr-i
CH2S(O)2CF3 Pr-c
CH2S(O)2CF3 Bu-n
CH2S(O)2CF3 Bu-i
CH2S(O)2CF3 Bu-c
CH2S(O)2CF3 Bu-s
CH2S(O)2CF3 Bu-t
CH2S(O)2CF3 Pen-n
CH2S(O)2CF3 Pen-c
CH2S(O)2CF3 Hex-n
CH2S(O)2CF3 Hex-c
CH2S(O)2CF3 CH2Pr-c
CH2S(O)2CF3 CH2Bu-c
CH2S(O)2CF3 CH2Pen-c
CH2S(O)2CF3 CH2Hex-c
CH2S(O)2CF3 CH2CH=CH2
CH2S(O)2CF3 CH2CH=C(Cl)2
CH2S(O)2CF3 CH2C≡CH
CH2S(O)2CF3 CH2CN
CH2S(O)2CF3 CH2CF3
CH2S(O)2CF3 CH2OMe
CH2S(O)2CF3 CH2OCF3
CH2S(O)2CF3 CH2SMe
CH2S(O)2CF3 CH2S(O)Me
CH2S(O)2CF3 CH2S(O)2Me
CH2S(O)2CF3 CH2SCF3
CH2S(O)2CF3 CH2S(O)CF3
CH2S(O)2CF3 CH2S(O)2CF3
CH2S(O)2CF3 CH2CH(OMe)2
CH2S(O)2CF3 CH2CH(SMe)2
CH2S(O)2CF3 CH2C(O)Me
CH2S(O)2CF3 CH2C(O)CF3
CH2S(O)2CF3 CH2C(O)OMe
CH2S(O)2CF3 CH2(D1-32a)
CH2S(O)2CF3 CH2(D1-33a)
CH2S(O)2CF3 CH2(D1-34a)
CH2S(O)2CF3 CH2(D1-37a)
CH2S(O)2CF3 CH2(D1-81a)
CH2S(O)2CF3 CH2(D1-82a)
CH2S(O)2CF3 CH2(D1-84a)
CH2S(O)2CF3 CH2(D1-85a)
CH2S(O)2CF3 CH2(D1-87a)
CH2S(O)2CF3 CH2(D1-92a)
CH2S(O)2CF3 CH2(D1-93a)
CH2S(O)2CF3 CH2(D1-95a)
CH2S(O)2CF3 CH2(D1-96a)
CH2S(O)2CF3 CH2(D1-98a)
CH2S(O)2CF3 CH2(D1-108a)
CH2S(O)2CF3 CH2(D1-108b,Z=2-Cl)
CH2S(O)2CF3 CH2(D1-108b,Z=3-Me)
CH2S(O)2CF3 CH2(D1-108b,Z=4-OMe)
CH2S(O)2CF3 CH2(D1-108b,Z=2-SMe)
CH2S(O)2CF3 CH2(D1-108b,Z=3-CF3)
CH2S(O)2CF3 CH2(D1-108b,Z=4-OCF3)
CH2S(O)2CF3 CH2(D1-108b,Z=2-SCF3)
CH2S(O)2CF3 CH2CH2CN
CH2S(O)2CF3 CH2CH2CF3
CH2S(O)2CF3 CH2CH2OMe
CH2S(O)2CF3 CH2CH2SMe
CH2S(O)2CF3 CH2CH2S(O)Me
CH2S(O)2CF3 CH2CH2S(O)2Me
CH2S(O)2CF3 D1-32a
CH2S(O)2CF3 D1-33a
CH2S(O)2CF3 D1-34a
CH2S(O)2CF3 D1-37a
CH2S(O)2CF3 D1-81a
CH2S(O)2CF3 D1-82a
CH2S(O)2CF3 D1-84a
CH2S(O)2CF3 D1-85a
CH2S(O)2CF3 D1-87a
CH2S(O)2CF3 D1-92a
CH2S(O)2CF3 D1-93a
CH2S(O)2CF3 D1-95a
CH2S(O)2CF3 D1-96a
CH2S(O)2CF3 D1-98a
CH2S(O)2CF3 D1-108a
CH2S(O)2CF3 D1-108b(Z=2-Cl)
CH2S(O)2CF3 D1-108b(Z=3-Me)
CH2S(O)2CF3 D1-108b(Z=4-OMe)
CH2S(O)2CF3 D1-108b(Z=2-SMe)
CH2S(O)2CF3 D1-108b(Z=3-CF3)
CH2S(O)2CF3 D1-108b(Z=4-OCF3)
CH2S(O)2CF3 D1-108b(Z=2-SCF3)
CH2S(O)2CF3 C(O)Me
CH2S(O)2CF3 C(O)CF3
CH2S(O)2CF3 C(O)OMe
CH2CH2SCF3 Me
CH2CH2SCF3 Et
CH2CH2SCF3 Pr-n
CH2CH2SCF3 Pr-i
CH2CH2SCF3 Pr-c
CH2CH2SCF3 Bu-n
CH2CH2SCF3 Bu-i
CH2CH2SCF3 Bu-c
CH2CH2SCF3 Bu-s
CH2CH2SCF3 Bu-t
CH2CH2SCF3 Pen-n
CH2CH2SCF3 Pen-c
CH2CH2SCF3 Hex-n
CH2CH2SCF3 Hex-c
CH2CH2SCF3 CH2Pr-c
CH2CH2SCF3 CH2Bu-c
CH2CH2SCF3 CH2Pen-c
CH2CH2SCF3 CH2Hex-c
CH2CH2SCF3 CH2CH=CH2
CH2CH2SCF3 CH2CH=C(Cl)2
CH2CH2SCF3 CH2C≡CH
CH2CH2SCF3 CH2CN
CH2CH2SCF3 CH2CF3
CH2CH2SCF3 CH2OMe
CH2CH2SCF3 CH2OCF3
CH2CH2SCF3 CH2SMe
CH2CH2SCF3 CH2S(O)Me
CH2CH2SCF3 CH2S(O)2Me
CH2CH2SCF3 CH2SCF3
CH2CH2SCF3 CH2S(O)CF3
CH2CH2SCF3 CH2S(O)2CF3
CH2CH2SCF3 CH2CH(OMe)2
CH2CH2SCF3 CH2CH(SMe)2
CH2CH2SCF3 CH2C(O)Me
CH2CH2SCF3 CH2C(O)CF3
CH2CH2SCF3 CH2C(O)OMe
CH2CH2SCF3 CH2(D1-32a)
CH2CH2SCF3 CH2(D1-33a)
CH2CH2SCF3 CH2(D1-34a)
CH2CH2SCF3 CH2(D1-37a)
CH2CH2SCF3 CH2(D1-81a)
CH2CH2SCF3 CH2(D1-82a)
CH2CH2SCF3 CH2(D1-84a)
CH2CH2SCF3 CH2(D1-85a)
CH2CH2SCF3 CH2(D1-87a)
CH2CH2SCF3 CH2(D1-92a)
CH2CH2SCF3 CH2(D1-93a)
CH2CH2SCF3 CH2(D1-95a)
CH2CH2SCF3 CH2(D1-96a)
CH2CH2SCF3 CH2(D1-98a)
CH2CH2SCF3 CH2(D1-108a)
CH2CH2SCF3 CH2(D1-108b,Z=2-Cl)
CH2CH2SCF3 CH2(D1-108b,Z=3-Me)
CH2CH2SCF3 CH2(D1-108b,Z=4-OMe)
CH2CH2SCF3 CH2(D1-108b,Z=2-SMe)
CH2CH2SCF3 CH2(D1-108b,Z=3-CF3)
CH2CH2SCF3 CH2(D1-108b,Z=4-OCF3)
CH2CH2SCF3 CH2(D1-108b,Z=2-SCF3)
CH2CH2SCF3 CH2CH2CN
CH2CH2SCF3 CH2CH2CF3
CH2CH2SCF3 CH2CH2OMe
CH2CH2SCF3 CH2CH2SMe
CH2CH2SCF3 CH2CH2S(O)Me
CH2CH2SCF3 CH2CH2S(O)2Me
CH2CH2SCF3 D1-32a
CH2CH2SCF3 D1-33a
CH2CH2SCF3 D1-34a
CH2CH2SCF3 D1-37a
CH2CH2H2SCF3 D1-81a
CH2CH2SCF3 D1-82a
CH2CH2SCF3 D1-84a
CH2CH2SCF3 D1-85a
CH2CH2SCF3 D1-87a
CH2CH2SCF3 D1-92a
CH2CH2SCF3 D1-93a
CH2CH2SCF3 D1-95a
CH2CH2SCF3 D1-96a
CH2CH2SCF3 D1-98a
CH2CH2SCF3 D1-108a
CH2CH2SCF3 D1-108b(Z=2-Cl)
CH2CH2SCF3 D1-108b(Z=3-Me)
CH2CH2SCF3 D1-108b(Z=4-OMe)
CH2CH2SCF3 D1-108b(Z=2-SMe)
CH2CH2SCF3 D1-108b(Z=3-CF3)
CH2CH2SCF3 D1-108b(Z=4-OCF3)
CH2CH2SCF3 D1-108b(Z=2-SCF3)
CH2CH2SCF3 C(O)Me
CH2CH2SCF3 C(O)CF3
CH2CH2SCF3 C(O)OMe
CH2CH2S(O)CF3 Me
CH2CH2S(O)CF3 Et
CH2CH2S(O)CF3 Pr-n
CH2CH2S(O)CF3 Pr-i
CH2CH2S(O)CF3 Pr-c
CH2CH2S(O)CF3 Bu-n
CH2CH2S(O)CF3 Bu-i
CH2CH2S(O)CF3 Bu-c
CH2CH2S(O)CF3 Bu-s
CH2CH2S(O)CF3 Bu-t
CH2CH2S(O)CF3 Pen-n
CH2CH2S(O)CF3 Pen-c
CH2CH2S(O)CF3 Hex-n
CH2CH2S(O)CF3 Hex-c
CH2CH2S(O)CF3 CH2Pr-c
CH2CH2S(O)CF3 CH2Bu-c
CH2CH2S(O)CF3 CH2Pen-c
CH2CH2S(O)CF3 CH2Hex-c
CH2CH2S(O)CF3 CH2CH=CH2
CH2CH2S(O)CF3 CH2CH=C(Cl)2
CH2CH2S(O)CF3 CH2C≡CH
CH2CH2S(O)CF3 CH2CN
CH2CH2S(O)CF3 CH2CF3
CH2CH2S(O)CF3 CH2OMe
CH2CH2S(O)CF3 CH2OCF3
CH2CH2S(O)CF3 CH2SMe
CH2CH2S(O)CF3 CH2S(O)Me
CH2CH2S(O)CF3 CH2S(O)2Me
CH2CH2S(O)CF3 CH2SCF3
CH2CH2S(O)CF3 CH2S(O)CF3
CH2CH2S(O)CF3 CH2S(O)2CF3
CH2CH2S(O)CF3 CH2CH(OMe)2
CH2CH2S(O)CF3 CH2CH(SMe)2
CH2CH2S(O)CF3 CH2C(O)Me
CH2CH2S(O)CF3 CH2C(O)CF3
CH2CH2S(O)CF3 CH2C(O)OMe
CH2CH2S(O)CF3 CH2(D1-32a)
CH2CH2S(O)CF3 CH2(D1-33a)
CH2CH2S(O)CF3 CH2(D1-34a)
CH2CH2S(O)CF3 CH2(D1-37a)
CH2CH2S(O)CF3 CH2(D1-81a)
CH2CH2S(O)CF3 CH2(D1-82a)
CH2CH2S(O)CF3 CH2(D1-84a)
CH2CH2S(O)CF3 CH2(D1-85a)
CH2CH2S(O)CF3 CH2(D1-87a)
CH2CH2S(O)CF3 CH2(D1-92a)
CH2CH2S(O)CF3 CH2(D1-93a)
CH2CH2S(O)CF3 CH2(D1-95a)
CH2CH2S(O)CF3 CH2(D1-96a)
CH2CH2S(O)CF3 CH2(D1-98a)
CH2CH2S(O)CF3 CH2(D1-108a)
CH2CH2S(O)CF3 CH2(D1-108b,Z=2-Cl)
CH2CH2S(O)CF3 CH2(D1-108b,Z=3-Me)
CH2CH2S(O)CF3 CH2(D1-108b,Z=4-OMe)
CH2CH2S(O)CF3 CH2(D1-108b,Z=2-SMe)
CH2CH2S(O)CF3 CH2(D1-108b,Z=3-CF3)
CH2CH2S(O)CF3 CH2(D1-108b,Z=4-OCF3)
CH2CH2S(O)CF3 CH2(D1-108b,Z=2-SCF3)
CH2CH2S(O)CF3 CH2CH2CN
CH2CH2S(O)CF3 CH2CH2CF3
CH2CH2S(O)CF3 CH2CH2OMe
CH2CH2S(O)CF3 CH2CH2SMe
CH2CH2S(O)CF3 CH2CH2S(O)Me
CH2CH2S(O)CF3 CH2CH2S(O)2Me
CH2CH2S(O)CF3 D1-32a
CH2CH2S(O)CF3 D1-33a
CH2CH2S(O)CF3 D1-34a
CH2CH2S(O)CF3 D1-37a
CH2CH2S(O)CF3 D1-81a
CH2CH2S(O)CF3 D1-82a
CH2CH2S(O)CF3 D1-84a
CH2CH2S(O)CF3 D1-85a
CH2CH2S(O)CF3 D1-87a
CH2CH2S(O)CF3 D1-92a
CH2CH2S(O)CF3 D1-93a
CH2CH2S(O)CF3 D1-95a
CH2CH2S(O)CF3 D1-96a
CH2CH2S(O)CF3 D1-98a
CH2CH2S(O)CF3 D1-108a
CH2CH2S(O)CF3 D1-108b(Z=2-Cl)
CH2CH2S(O)CF3 D1-108b(Z=3-Me)
CH2CH2S(O)CF3 D1-108b(Z=4-OMe)
CH2CH2S(O)CF3 D1-108b(Z=2-SMe)
CH2CH2S(O)CF3 D1-108b(Z=3-CF3)
CH2CH2S(O)CF3 D1-108b(Z=4-OCF3)
CH2CH2S(O)CF3 D1-108b(Z=2-SCF3)
CH2CH2S(O)CF3 C(O)Me
CH2CH2S(O)CF3 C(O)CF3
CH2CH2S(O)CF3 C(O)OMe
CH2CH2S(O)2CF3 Me
CH2CH2S(O)2CF3 Et
CH2CH2S(O)2CF3 Pr-n
CH2CH2S(O)2CF3 Pr-i
CH2CH2S(O)2CF3 Pr-c
CH2CH2S(O)2CF3 Bu-n
CH2CH2S(O)2CF3 Bu-i
CH2CH2S(O)2CF3 Bu-c
CH2CH2S(O)2CF3 Bu-s
CH2CH2S(O)2CF3 Bu-t
CH2CH2S(O)2CF3 Pen-n
CH2CH2S(O)2CF3 Pen-c
CH2CH2S(O)2CF3 Hex-n
CH2CH2S(O)2CF3 Hex-c
CH2CH2S(O)2CF3 CH2Pr-c
CH2CH2S(O)2CF3 CH2Bu-c
CH2CH2S(O)2CF3 CH2Pen-c
CH2CH2S(O)2CF3 CH2Hex-c
CH2CH2S(O)2CF3 CH2CH=CH2
CH2CH2S(O)2CF3 CH2CH=C(Cl)2
CH2CH2S(O)2CF3 CH2C≡CH
CH2CH2S(O)2CF3 CH2CN
CH2CH2S(O)2CF3 CH2CF3
CH2CH2S(O)2CF3 CH2OMe
CH2CH2S(O)2CF3 CH2OCF3
CH2CH2S(O)2CF3 CH2SMe
CH2CH2S(O)2CF3 CH2S(O)Me
CH2CH2S(O)2CF3 CH2S(O)2Me
CH2CH2S(O)2CF3 CH2SCF3
CH2CH2S(O)2CF3 CH2S(O)CF3
CH2CH2S(O)2CF3 CH2S(O)2CF3
CH2CH2S(O)2CF3 CH2CH(OMe)2
CH2CH2S(O)2CF3 CH2CH(SMe)2
CH2CH2S(O)2CF3 CH2C(O)Me
CH2CH2S(O)2CF3 CH2C(O)CF3
CH2CH2S(O)2CF3 CH2C(O)OMe
CH2CH2S(O)2CF3 CH2(D1-32a)
CH2CH2S(O)2CF3 CH2(D1-33a)
CH2CH2S(O)2CF3 CH2(D1-34a)
CH2CH2S(O)2CF3 CH2(D1-37a)
CH2CH2S(O)2CF3 CH2(D1-81a)
CH2CH2S(O)2CF3 CH2(D1-82a)
CH2CH2S(O)2CF3 CH2(D1-84a)
CH2CH2S(O)2CF3 CH2(D1-85a)
CH2CH2S(O)2CF3 CH2(D1-87a)
CH2CH2S(O)2CF3 CH2(D1-92a)
CH2CH2S(O)2CF3 CH2(D1-93a)
CH2CH2S(O)2CF3 CH2(D1-95a)
CH2CH2S(O)2CF3 CH2(D1-96a)
CH2CH2S(O)2CF3 CH2(D1-98a)
CH2CH2S(O)2CF3 CH2(D1-108a)
CH2CH2S(O)2CF3 CH2(D1-108b,Z=2-Cl)
CH2CH2S(O)2CF3 CH2(D1-108b,Z=3-Me)
CH2CH2S(O)2CF3 CH2(D1-108b,Z=4-OMe)
CH2CH2S(O)2CF3 CH2(D1-108b,Z=2-SMe)
CH2CH2S(O)2CF3 CH2(D1-108b,Z=3-CF3)
CH2CH2S(O)2CF3 CH2(D1-108b,Z=4-OCF3)
CH2CH2S(O)2CF3 CH2(D1-108b,Z=2-SCF3)
CH2CH2S(O)2CF3 CH2CH2CN
CH2CH2S(O)2CF3 CH2CH2CF3
CH2CH2S(O)2CF3 CH2CH2OMe
CH2CH2S(O)2CF3 CH2CH2SMe
CH2CH2S(O)2CF3 CH2CH2S(O)Me
CH2CH2S(O)2CF3 CH2CH2S(O)2Me
CH2CH2S(O)2CF3 D1-32a
CH2CH2S(O)2CF3 D1-33a
CH2CH2S(O)2CF3 D1-34a
CH2CH2S(O)2CF3 D1-37a
CH2CH2S(O)2CF3 D1-81a
CH2CH2S(O)2CF3 D1-82a
CH2CH2S(O)2CF3 D1-84a
CH2CH2S(O)2CF3 D1-85a
CH2CH2S(O)2CF3 D1-87a
CH2CH2S(O)2CF3 D1-92a
CH2CH2S(O)2CF3 D1-93a
CH2CH2S(O)2CF3 D1-95a
CH2CH2S(O)2CF3 D1-96a
CH2CH2S(O)2CF3 D1-98a
CH2CH2S(O)2CF3 D1-108a
CH2CH2S(O)2CF3 D1-108b(Z=2-Cl)
CH2CH2S(O)2CF3 D1-108b(Z=3-Me)
CH2CH2S(O)2CF3 D1-108b(Z=4-OMe)
CH2CH2S(O)2CF3 D1-108b(Z=2-SMe)
CH2CH2S(O)2CF3 D1-108b(Z=3-CF3)
CH2CH2S(O)2CF3 D1-108b(Z=4-OCF3)
CH2CH2S(O)2CF3 D1-108b(Z=2-SCF3)
CH2CH2S(O)2CF3 C(O)Me
CH2CH2S(O)2CF3 C(O)CF3
CH2CH2S(O)2CF3 C(O)OMe
D1-32a Me
D1-32a Et
D1-32a Pr-n
D1-32a Pr-i
D1-32a Pr-c
D1-32a Bu-n
D1-32a Bu-i
D1-32a Bu-c
D1-32a Bu-s
D1-32a Bu-t
D1-32a Pen-n
D1-32a Pen-c
D1-32a Hex-n
D1-32a Hex-c
D1-32a CH2Pr-c
D1-32a CH2Bu-c
D1-32a CH2Pen-c
D1-32a CH2Hex-c
D1-32a CH2CH=CH2
D1-32a CH2CH=C(Cl)2
D1-32a CH2C≡CH
D1-32a CH2CN
D1-32a CH2CF3
D1-32a CH2OMe
D1-32a CH2OCF3
D1-32a CH2SMe
D1-32a CH2S(O)Me
D1-32a CH2S(O)2Me
D1-32a CH2SCF3
D1-32a CH2S(O)CF3
D1-32a CH2S(O)2CF3
D1-32a CH2CH(OMe)2
D1-32a CH2CH(SMe)2
D1-32a CH2C(O)Me
D1-32a CH2C(O)CF3
D1-32a CH2C(O)OMe
D1-32a CH2(D1-32a)
D1-32a CH2(D1-33a)
D1-32a CH2(D1-34a)
D1-32a CH2(D1-37a)
D1-32a CH2(D1-81a)
D1-32a CH2(D1-82a)
D1-32a CH2(D1-84a)
D1-32a CH2(D1-85a)
D1-32a CH2(D1-87a)
D1-32a CH2(D1-92a)
D1-32a CH2(D1-93a)
D1-32a CH2(D1-95a)
D1-32a CH2(D1-96a)
D1-32a CH2(D1-98a)
D1-32a CH2(D1-108a)
D1-32a CH2(D1-108b,Z=2-Cl)
D1-32a CH2(D1-108b,Z=3-Me)
D1-32a CH2(D1-108b,Z=4-OMe)
D1-32a CH2(D1-108b,Z=2-SMe)
D1-32a CH2(D1-108b,Z=3-CF3)
D1-32a CH2(D1-108b,Z=4-OCF3)
D1-32a CH2(D1-108b,Z=2-SCF3)
D1-32a CH2CH2CN
D1-32a CH2CH2CF3
D1-32a CH2CH2OMe
D1-32a CH2CH2SMe
D1-32a CH2CH2S(O)Me
D1-32a CH2CH2S(O)2Me
D1-32a D1-32a
D1-32a D1-33a
D1-32a D1-34a
D1-32a D1-37a
D1-32a D1-81a
D1-32a D1-82a
D1-32a D1-84a
D1-32a D1-85a
D1-32a D1-87a
D1-32a D1-92a
D1-32a D1-93a
D1-32a D1-95a
D1-32a D1-96a
D1-32a D1-98a
D1-32a D1-108a
D1-32a D1-108b(Z=2-Cl)
D1-32a D1-108b(Z=3-Me)
D1-32a D1-108b(Z=4-OMe)
D1-32a D1-108b(Z=2-SMe)
D1-32a D1-108b(Z=3-CF3)
D1-32a D1-108b(Z=4-OCF3)
D1-32a D1-108b(Z=2-SCF3)
D1-32a C(O)Me
D1-32a C(O)CF3
D1-32a C(O)OMe
D1-33a Me
D1-33a Et
D1-33a Pr-n
D1-33a Pr-i
D1-33a Pr-c
D1-33a Bu-n
D1-33a Bu-i
D1-33a Bu-c
D1-33a Bu-s
D1-33a Bu-t
D1-33a Pen-n
D1-33a Pen-c
D1-33a Hex-n
D1-33a Hex-c
D1-33a CH2Pr-c
D1-33a CH2Bu-c
D1-33a CH2Pen-c
D1-33a CH2Hex-c
D1-33a CH2CH=CH2
D1-33a CH2CH=C(Cl)2
D1-33a CH2C≡CH
D1-33a CH2CN
D1-33a CH2CF3
D1-33a CH2OMe
D1-33a CH2OCF3
D1-33a CH2SMe
D1-33a CH2S(O)Me
D1-33a CH2S(O)2Me
D1-33a CH2SCF3
D1-33a CH2S(O)CF3
D1-33a CH2S(O)2CF3
D1-33a CH2CH(OMe)2
D1-33a CH2CH(SMe)2
D1-33a CH2C(O)Me
D1-33a CH2C(O)CF3
D1-33a CH2C(O)OMe
D1-33a CH2(D1-32a)
D1-33a CH2(D1-33a)
D1-33a CH2(D1-34a)
D1-33a CH2(D1-37a)
D1-33a CH2(D1-81a)
D1-33a CH2(D1-82a)
D1-33a CH2(D1-84a)
D1-33a CH2(D1-85a)
D1-33a CH2(D1-87a)
D1-33a CH2(D1-92a)
D1-33a CH2(D1-93a)
D1-33a CH2(D1-95a)
D1-33a CH2(D1-96a)
D1-33a CH2(D1-98a)
D1-33a CH2(D1-108a)
D1-33a CH2(D1-108b,Z=2-Cl)
D1-33a CH2(D1-108b,Z=3-Me)
D1-33a CH2(D1-108b,Z=4-OMe)
D1-33a CH2(D1-108b,Z=2-SMe)
D1-33a CH2(D1-108b,Z=3-CF3)
D1-33a CH2(D1-108b,Z=4-OCF3)
D1-33a CH2(D1-108b,Z=2-SCF3)
D1-33a CH2CH2CN
D1-33a CH2CH2CF3
D1-33a CH2CH2OMe
D1-33a CH2CH2SMe
D1-33a CH2CH2S(O)Me
D1-33a CH2CH2S(O)2Me
D1-33a D1-32a
D1-33a D1-33a
D1-33a D1-34a
D1-33a D1-37a
D1-33a D1-81a
D1-33a D1-82a
D1-33a D1-84a
D1-33a D1-85a
D1-33a D1-87a
D1-33a D1-92a
D1-33a D1-93a
D1-33a D1-95a
D1-33a D1-96a
D1-33a D1-98a
D1-33a D1-108a
D1-33a D1-108b(Z=2-Cl)
D1-33a D1-108b(Z=3-Me)
D1-33a D1-108b(Z=4-OMe)
D1-33a D1-108b(Z=2-SMe)
D1-33a D1-108b(Z=3-CF3)
D1-33a D1-108b(Z=4-OCF3)
D1-33a D1-108b(Z=2-SCF3)
D1-33a C(O)Me
D1-33a C(O)CF3
D1-33a C(O)OMe
D1-34a Me
D1-34a Et
D1-34a Pr-n
D1-34a Pr-i
D1-34a Pr-c
D1-34a Bu-n
D1-34a Bu-i
D1-34a Bu-c
D1-34a Bu-s
D1-34a Bu-t
D1-34a Pen-n
D1-34a Pen-c
D1-34a Hex-n
D1-34a Hex-c
D1-34a CH2Pr-c
D1-34a CH2Bu-c
D1-34a CH2Pen-c
D1-34a CH2Hex-c
D1-34a CH2CH=CH2
D1-34a CH2CH=C(Cl)2
D1-34a CH2C≡CH
D1-34a CH2CN
D1-34a CH2CF3
D1-34a CH2OMe
D1-34a CH2OCF3
D1-34a CH2SMe
D1-34a CH2S(O)Me
D1-34a CH2S(O)2Me
D1-34a CH2SCF3
D1-34a CH2S(O)CF3
D1-34a CH2S(O)2CF3
D1-34a CH2CH(OMe)2
D1-34a CH2CH(SMe)2
D1-34a CH2C(O)Me
D1-34a CH2C(O)CF3
D1-34a CH2C(O)OMe
D1-34a CH2(D1-32a)
D1-34a CH2(D1-33a)
D1-34a CH2(D1-34a)
D1-34a CH2(D1-37a)
D1-34a CH2(D1-81a)
D1-34a CH2(D1-82a)
D1-34a CH2(D1-84a)
D1-34a CH2(D1-85a)
D1-34a CH2(D1-87a)
D1-34a CH2(D1-92a)
D1-34a CH2(D1-93a)
D1-34a CH2(D1-95a)
D1-34a CH2(D1-96a)
D1-34a CH2(D1-98a)
D1-34a CH2(D1-108a)
D1-34a CH2(D1-108b,Z=2-Cl)
D1-34a CH2(D1-108b,Z=3-Me)
D1-34a CH2(D1-108b,Z=4-OMe)
D1-34a CH2(D1-108b,Z=2-SMe)
D1-34a CH2(D1-108b,Z=3-CF3)
D1-34a CH2(D1-108b,Z=4-OCF3)
D1-34a CH2(D1-108b,Z=2-SCF3)
D1-34a CH2CH2CN
D1-34a CH2CH2CF3
D1-34a CH2CH2OMe
D1-34a CH2CH2SMe
D1-34a CH2CH2S(O)Me
D1-34a CH2CH2S(O)2Me
D1-34a D1-32a
D1-34a D1-33a
D1-34a D1-34a
D1-34a D1-37a
D1-34a D1-81a
D1-34a D1-82a
D1-34a D1-84a
D1-34a D1-85a
D1-34a D1-87a
D1-34a D1-92a
D1-34a D1-93a
D1-34a D1-95a
D1-34a D1-96a
D1-34a D1-98a
D1-34a D1-108a
D1-34a D1-108b(Z=2-Cl)
D1-34a D1-108b(Z=3-Me)
D1-34a D1-108b(Z=4-OMe)
D1-34a D1-108b(Z=2-SMe)
D1-34a D1-108b(Z=3-CF3)
D1-34a D1-108b(Z=4-OCF3)
D1-34a D1-108b(Z=2-SCF3)
D1-34a C(O)Me
D1-34a C(O)CF3
D1-34a C(O)OMe
D1-37a Me
D1-37a Et
D1-37a Pr-n
D1-37a Pr-i
D1-37a Pr-c
D1-37a Bu-n
D1-37a Bu-i
D1-37a Bu-c
D1-37a Bu-s
D1-37a Bu-t
D1-37a Pen-n
D1-37a Pen-c
D1-37a Hex-n
D1-37a Hex-c
D1-37a CH2Pr-c
D1-37a CH2Bu-c
D1-37a CH2Pen-c
D1-37a CH2Hex-c
D1-37a CH2CH=CH2
D1-37a CH2CH=C(Cl)2
D1-37a CH2C≡CH
D1-37a CH2CN
D1-37a CH2CF3
D1-37a CH2OMe
D1-37a CH2OCF3
D1-37a CH2SMe
D1-37a CH2S(O)Me
D1-37a CH2S(O)2Me
D1-37a CH2SCF3
D1-37a CH2S(O)CF3
D1-37a CH2S(O)2CF3
D1-37a CH2CH(OMe)2
D1-37a CH2CH(SMe)2
D1-37a CH2C(O)Me
D1-37a CH2C(O)CF3
D1-37a CH2C(O)OMe
D1-37a CH2(D1-32a)
D1-37a CH2(D1-33a)
D1-37a CH2(D1-34a)
D1-37a CH2(D1-37a)
D1-37a CH2(D1-81a)
D1-37a CH2(D1-82a)
D1-37a CH2(D1-84a)
D1-37a CH2(D1-85a)
D1-37a CH2(D1-87a)
D1-37a CH2(D1-92a)
D1-37a CH2(D1-93a)
D1-37a CH2(D1-95a)
D1-37a CH2(D1-96a)
D1-37a CH2(D1-98a)
D1-37a CH2(D1-108a)
D1-37a CH2(D1-108b,Z=2-Cl)
D1-37a CH2(D1-108b,Z=3-Me)
D1-37a CH2(D1-108b,Z=4-OMe)
D1-37a CH2(D1-108b,Z=2-SMe)
D1-37a CH2(D1-108b,Z=3-CF3)
D1-37a CH2(D1-108b,Z=4-OCF3)
D1-37a CH2(D1-108b,Z=2-SCF3)
D1-37a CH2CH2CN
D1-37a CH2CH2CF3
D1-37a CH2CH2OMe
D1-37a CH2CH2SMe
D1-37a CH2CH2S(O)Me
D1-37a CH2CH2S(O)2Me
D1-37a D1-32a
D1-37a D1-33a
D1-37a D1-34a
D1-37a D1-37a
D1-37a D1-81a
D1-37a D1-82a
D1-37a D1-84a
D1-37a D1-85a
D1-37a D1-87a
D1-37a D1-92a
D1-37a D1-93a
D1-37a D1-95a
D1-37a D1-96a
D1-37a D1-98a
D1-37a D1-108a
D1-37a D1-108b(Z=2-Cl)
D1-37a D1-108b(Z=3-Me)
D1-37a D1-108b(Z=4-OMe)
D1-37a D1-108b(Z=2-SMe)
D1-37a D1-108b(Z=3-CF3)
D1-37a D1-108b(Z=4-OCF3)
D1-37a D1-108b(Z=2-SCF3)
D1-37a C(O)Me
D1-37a C(O)CF3
D1-37a C(O)OMe
D1-81a Me
D1-81a Et
D1-81a Pr-n
D1-81a Pr-i
D1-81a Pr-c
D1-81a Bu-n
D1-81a Bu-i
D1-81a Bu-c
D1-81a Bu-s
D1-81a Bu-t
D1-81a Pen-n
D1-81a Pen-c
D1-81a Hex-n
D1-81a Hex-c
D1-81a CH2Pr-c
D1-81a CH2Bu-c
D1-81a CH2Pen-c
D1-81a CH2Hex-c
D1-81a CH2CH=CH2
D1-81a CH2CH=C(Cl)2
D1-81a CH2C≡CH
D1-81a CH2CN
D1-81a CH2CF3
D1-81a CH2OMe
D1-81a CH2OCF3
D1-81a CH2SMe
D1-81a CH2S(O)Me
D1-81a CH2S(O)2Me
D1-81a CH2SCF3
D1-81a CH2S(O)CF3
D1-81a CH2S(O)2CF3
D1-81a CH2CH(OMe)2
D1-81a CH2CH(SMe)2
D1-81a CH2C(O)Me
D1-81a CH2C(O)CF3
D1-81a CH2C(O)OMe
D1-81a CH2(D1-32a)
D1-81a CH2(D1-33a)
D1-81a CH2(D1-34a)
D1-81a CH2(D1-37a)
D1-81a CH2(D1-81a)
D1-81a CH2(D1-82a)
D1-81a CH2(D1-84a)
D1-81a CH2(D1-85a)
D1-81a CH2(D1-87a)
D1-81a CH2(D1-92a)
D1-81a CH2(D1-93a)
D1-81a CH2(D1-95a)
D1-81a CH2(D1-96a)
D1-81a CH2(D1-98a)
D1-81a CH2(D1-108a)
D1-81a CH2(D1-108b,Z=2-Cl)
D1-81a CH2(D1-108b,Z=3-Me)
D1-81a CH2(D1-108b,Z=4-OMe)
D1-81a CH2(D1-108b,Z=2-SMe)
D1-81a CH2(D1-108b,Z=3-CF3)
D1-81a CH2(D1-108b,Z=4-OCF3)
D1-81a CH2(D1-108b,Z=2-SCF3)
D1-81a CH2CH2CN
D1-81a CH2CH2CF3
D1-81a CH2CH2OMe
D1-81a CH2CH2SMe
D1-81a CH2CH2S(O)Me
D1-81a CH2CH2S(O)2Me
D1-81a D1-32a
D1-81a D1-33a
D1-81a D1-34a
D1-81a D1-37a
D1-81a D1-81a
D1-81a D1-82a
D1-81a D1-84a
D1-81a D1-85a
D1-81a D1-87a
D1-81a D1-92a
D1-81a D1-93a
D1-81a D1-95a
D1-81a D1-96a
D1-81a D1-98a
D1-81a D1-108a
D1-81a D1-108b(Z=2-Cl)
D1-81a D1-108b(Z=3-Me)
D1-81a D1-108b(Z=4-OMe)
D1-81a D1-108b(Z=2-SMe)
D1-81a D1-108b(Z=3-CF3)
D1-81a D1-108b(Z=4-OCF3)
D1-81a D1-108b(Z=2-SCF3)
D1-81a C(O)Me
D1-81a C(O)CF3
D1-81a C(O)OMe
D1-82a Me
D1-82a Et
D1-82a Pr-n
D1-82a Pr-i
D1-82a Pr-c
D1-82a Bu-n
D1-82a Bu-i
D1-82a Bu-c
D1-82a Bu-s
D1-82a Bu-t
D1-82a Pen-n
D1-82a Pen-c
D1-82a Hex-n
D1-82a Hex-c
D1-82a CH2Pr-c
D1-82a CH2Bu-c
D1-82a CH2Pen-c
D1-82a CH2Hex-c
D1-82a CH2CH=CH2
D1-82a CH2CH=C(Cl)2
D1-82a CH2C≡CH
D1-82a CH2CN
D1-82a CH2CF3
D1-82a CH2OMe
D1-82a CH2OCF3
D1-82a CH2SMe
D1-82a CH2S(O)Me
D1-82a CH2S(O)2Me
D1-82a CH2SCF3
D1-82a CH2S(O)CF3
D1-82a CH2S(O)2CF3
D1-82a CH2CH(OMe)2
D1-82a CH2CH(SMe)2
D1-82a CH2C(O)Me
D1-82a CH2C(O)CF3
D1-82a CH2C(O)OMe
D1-82a CH2(D1-32a)
D1-82a CH2(D1-33a)
D1-82a CH2(D1-34a)
D1-82a CH2(D1-37a)
D1-82a CH2(D1-81a)
D1-82a CH2(D1-82a)
D1-82a CH2(D1-84a)
D1-82a CH2(D1-85a)
D1-82a CH2(D1-87a)
D1-82a CH2(D1-92a)
D1-82a CH2(D1-93a)
D1-82a CH2(D1-95a)
D1-82a CH2(D1-96a)
D1-82a CH2(D1-98a)
D1-82a CH2(D1-108a)
D1-82a CH2(D1-108b,Z=2-Cl)
D1-82a CH2(D1-108b,Z=3-Me)
D1-82a CH2(D1-108b,Z=4-OMe)
D1-82a CH2(D1-108b,Z=2-SMe)
D1-82a CH2(D1-108b,Z=3-CF3)
D1-82a CH2(D1-108b,Z=4-OCF3)
D1-82a CH2(D1-108b,Z=2-SCF3)
D1-82a CH2CH2CN
D1-82a CH2CH2CF3
D1-82a CH2CH2OMe
D1-82a CH2CH2SMe
D1-82a CH2CH2S(O)Me
D1-82a CH2CH2S(O)2Me
D1-82a D1-32a
D1-82a D1-33a
D1-82a D1-34a
D1-82a D1-37a
D1-82a D1-81a
D1-82a D1-82a
D1-82a D1-84a
D1-82a D1-85a
D1-82a D1-87a
D1-82a D1-92a
D1-82a D1-93a
D1-82a D1-95a
D1-82a D1-96a
D1-82a D1-98a
D1-82a D1-108a
D1-82a D1-108b(Z=2-Cl)
D1-82a D1-108b(Z=3-Me)
D1-82a D1-108b(Z=4-OMe)
D1-82a D1-108b(Z=2-SMe)
D1-82a D1-108b(Z=3-CF3)
D1-82a D1-108b(Z=4-OCF3)
D1-82a D1-108b(Z=2-SCF3)
D1-82a C(O)Me
D1-82a C(O)CF3
D1-82a C(O)OMe
D1-84a Me
D1-84a Et
D1-84a Pr-n
D1-84a Pr-i
D1-84a Pr-c
D1-84a Bu-n
D1-84a Bu-i
D1-84a Bu-c
D1-84a Bu-s
D1-84a Bu-t
D1-84a Pen-n
D1-84a Pen-c
D1-84a Hex-n
D1-84a Hex-c
D1-84a CH2Pr-c
D1-84a CH2Bu-c
D1-84a CH2Pen-c
D1-84a CH2Hex-c
D1-84a CH2CH=CH2
D1-84a CH2CH=C(Cl)2
D1-84a CH2C≡CH
D1-84a CH2CN
D1-84a CH2CF3
D1-84a CH2OMe
D1-84a CH2OCF3
D1-84a CH2SMe
D1-84a CH2S(O)Me
D1-84a CH2S(O)2Me
D1-84a CH2SCF3
D1-84a CH2S(O)CF3
D1-84a CH2S(O)2CF3
D1-84a CH2CH(OMe)2
D1-84a CH2CH(SMe)2
D1-84a CH2C(O)Me
D1-84a CH2C(O)CF3
D1-84a CH2C(O)OMe
D1-84a CH2(D1-32a)
D1-84a CH2(D1-33a)
D1-84a CH2(D1-34a)
D1-84a CH2(D1-37a)
D1-84a CH2(D1-81a)
D1-84a CH2(D1-82a)
D1-84a CH2(D1-84a)
D1-84a CH2(D1-85a)
D1-84a CH2(D1-87a)
D1-84a CH2(D1-92a)
D1-84a CH2(D1-93a)
D1-84a CH2(D1-95a)
D1-84a CH2(D1-96a)
D1-84a CH2(D1-98a)
D1-84a CH2(D1-108a)
D1-84a CH2(D1-108b,Z=2-Cl)
D1-84a CH2(D1-108b,Z=3-Me)
D1-84a CH2(D1-108b,Z=4-OMe)
D1-84a CH2(D1-108b,Z=2-SMe)
D1-84a CH2(D1-108b,Z=3-CF3)
D1-84a CH2(D1-108b,Z=4-OCF3)
D1-84a CH2(D1-108b,Z=2-SCF3)
D1-84a CH2CH2CN
D1-84a CH2CH2CF3
D1-84a CH2CH2OMe
D1-84a CH2CH2SMe
D1-84a CH2CH2S(O)Me
D1-84a CH2CH2S(O)2Me
D1-84a D1-32a
D1-84a D1-33a
D1-84a D1-34a
D1-84a D1-37a
D1-84a D1-81a
D1-84a D1-82a
D1-84a D1-84a
D1-84a D1-85a
D1-84a D1-87a
D1-84a D1-92a
D1-84a D1-93a
D1-84a D1-95a
D1-84a D1-96a
D1-84a D1-98a
D1-84a D1-108a
D1-84a D1-108b(Z=2-Cl)
D1-84a D1-108b(Z=3-Me)
D1-84a D1-108b(Z=4-OMe)
D1-84a D1-108b(Z=2-SMe)
D1-84a D1-108b(Z=3-CF3)
D1-84a D1-108b(Z=4-OCF3)
D1-84a D1-108b(Z=2-SCF3)
D1-84a C(O)Me
D1-84a C(O)CF3
D1-84a C(O)OMe
D1-85a Me
D1-85a Et
D1-85a Pr-n
D1-85a Pr-i
D1-85a Pr-c
D1-85a Bu-n
D1-85a Bu-i
D1-85a Bu-c
D1-85a Bu-s
D1-85a Bu-t
D1-85a Pen-n
D1-85a Pen-c
D1-85a Hex-n
D1-85a Hex-c
D1-85a CH2Pr-c
D1-85a CH2Bu-c
D1-85a CH2Pen-c
D1-85a CH2Hex-c
D1-85a CH2CH=CH2
D1-85a CH2CH=C(Cl)2
D1-85a CH2C≡CH
D1-85a CH2CN
D1-85a CH2CF3
D1-85a CH2OMe
D1-85a CH2OCF3
D1-85a CH2SMe
D1-85a CH2S(O)Me
D1-85a CH2S(O)2Me
D1-85a CH2SCF3
D1-85a CH2S(O)CF3
D1-85a CH2S(O)2CF3
D1-85a CH2CH(OMe)2
D1-85a CH2CH(SMe)2
D1-85a CH2C(O)Me
D1-85a CH2C(O)CF3
D1-85a CH2C(O)OMe
D1-85a CH2(D1-32a)
D1-85a CH2(D1-33a)
D1-85a CH2(D1-34a)
D1-85a CH2(D1-37a)
D1-85a CH2(D1-81a)
D1-85a CH2(D1-82a)
D1-85a CH2(D1-84a)
D1-85a CH2(D1-85a)
D1-85a CH2(D1-87a)
D1-85a CH2(D1-92a)
D1-85a CH2(D1-93a)
D1-85a CH2(D1-95a)
D1-85a CH2(D1-96a)
D1-85a CH2(D1-98a)
D1-85a CH2(D1-108a)
D1-85a CH2(D1-108b,Z=2-Cl)
D1-85a CH2(D1-108b,Z=3-Me)
D1-85a CH2(D1-108b,Z=4-OMe)
D1-85a CH2(D1-108b,Z=2-SMe)
D1-85a CH2(D1-108b,Z=3-CF3)
D1-85a CH2(D1-108b,Z=4-OCF3)
D1-85a CH2(D1-108b,Z=2-SCF3)
D1-85a CH2CH2CN
D1-85a CH2CH2CF3
D1-85a CH2CH2OMe
D1-85a CH2CH2SMe
D1-85a CH2CH2S(O)Me
D1-85a CH2CH2S(O)2Me
D1-85a D1-32a
D1-85a D1-33a
D1-85a D1-34a
D1-85a D1-37a
D1-85a D1-81a
D1-85a D1-82a
D1-85a D1-84a
D1-85a D1-85a
D1-85a D1-87a
D1-85a D1-92a
D1-85a D1-93a
D1-85a D1-95a
D1-85a D1-96a
D1-85a D1-98a
D1-85a D1-108a
D1-85a D1-108b(Z=2-Cl)
D1-85a D1-108b(Z=3-Me)
D1-85a D1-108b(Z=4-OMe)
D1-85a D1-108b(Z=2-SMe)
D1-85a D1-108b(Z=3-CF3)
D1-85a D1-108b(Z=4-OCF3)
D1-85a D1-108b(Z=2-SCF3)
D1-85a C(O)Me
D1-85a C(O)CF3
D1-85a C(O)OMe
D1-87a Me
D1-87a Et
D1-87a Pr-n
D1-87a Pr-i
D1-87a Pr-c
D1-87a Bu-n
D1-87a Bu-i
D1-87a Bu-c
D1-87a Bu-s
D1-87a Bu-t
D1-87a Pen-n
D1-87a Pen-c
D1-87a Hex-n
D1-87a Hex-c
D1-87a CH2Pr-c
D1-87a CH2Bu-c
D1-87a CH2Pen-c
D1-87a CH2Hex-c
D1-87a CH2CH=CH2
D1-87a CH2CH=C(Cl)2
D1-87a CH2C≡CH
D1-87a CH2CN
D1-87a CH2CF3
D1-87a CH2OMe
D1-87a CH2OCF3
D1-87a CH2SMe
D1-87a CH2S(O)Me
D1-87a CH2S(O)2Me
D1-87a CH2SCF3
D1-87a CH2S(O)CF3
D1-87a CH2S(O)2CF3
D1-87a CH2CH(OMe)2
D1-87a CH2CH(SMe)2
D1-87a CH2C(O)Me
D1-87a CH2C(O)CF3
D1-87a CH2C(O)OMe
D1-87a CH2(D1-32a)
D1-87a CH2(D1-33a)
D1-87a CH2(D1-34a)
D1-87a CH2(D1-37a)
D1-87a CH2(D1-81a)
D1-87a CH2(D1-82a)
D1-87a CH2(D1-84a)
D1-87a CH2(D1-85a)
D1-87a CH2(D1-87a)
D1-87a CH2(D1-92a)
D1-87a CH2(D1-93a)
D1-87a CH2(D1-95a)
D1-87a CH2(D1-96a)
D1-87a CH2(D1-98a)
D1-87a CH2(D1-108a)
D1-87a CH2(D1-108b,Z=2-Cl)
D1-87a CH2(D1-108b,Z=3-Me)
D1-87a CH2(D1-108b,Z=4-OMe)
D1-87a CH2(D1-108b,Z=2-SMe)
D1-87a CH2(D1-108b,Z=3-CF3)
D1-87a CH2(D1-108b,Z=4-OCF3)
D1-87a CH2(D1-108b,Z=2-SCF3)
D1-87a CH2CH2CN
D1-87a CH2CH2CF3
D1-87a CH2CH2OMe
D1-87a CH2CH2SMe
D1-87a CH2CH2S(O)Me
D1-87a CH2CH2S(O)2Me
D1-87a D1-32a
D1-87a D1-33a
D1-87a D1-34a
D1-87a D1-37a
D1-87a D1-81a
D1-87a D1-82a
D1-87a D1-84a
D1-87a D1-85a
D1-87a D1-87a
D1-87a D1-92a
D1-87a D1-93a
D1-87a D1-95a
D1-87a D1-96a
D1-87a D1-98a
D1-87a D1-108a
D1-87a D1-108b(Z=2-Cl)
D1-87a D1-108b(Z=3-Me)
D1-87a D1-108b(Z=4-OMe)
D1-87a D1-108b(Z=2-SMe)
D1-87a D1-108b(Z=3-CF3)
D1-87a D1-108b(Z=4-OCF3)
D1-87a D1-108b(Z=2-SCF3)
D1-87a C(O)Me
D1-87a C(O)CF3
D1-87a C(O)OMe
D1-92a Me
D1-92a Et
D1-92a Pr-n
D1-92a Pr-i
D1-92a Pr-c
D1-92a Bu-n
D1-92a Bu-i
D1-92a Bu-c
D1-92a Bu-s
D1-92a Bu-t
D1-92a Pen-n
D1-92a Pen-c
D1-92a Hex-n
D1-92a Hex-c
D1-92a CH2Pr-c
D1-92a CH2Bu-c
D1-92a CH2Pen-c
D1-92a CH2Hex-c
D1-92a CH2CH=CH2
D1-92a CH2CH=C(Cl)2
D1-92a CH2C≡CH
D1-92a CH2CN
D1-92a CH2CF3
D1-92a CH2OMe
D1-92a CH2OCF3
D1-92a CH2SMe
D1-92a CH2S(O)Me
D1-92a CH2S(O)2Me
D1-92a CH2SCF3
D1-92a CH2S(O)CF3
D1-92a CH2S(O)2CF3
D1-92a CH2CH(OMe)2
D1-92a CH2CH(SMe)2
D1-92a CH2C(O)Me
D1-92a CH2C(O)CF3
D1-92a CH2C(O)OMe
D1-92a CH2(D1-32a)
D1-92a CH2(D1-33a)
D1-92a CH2(D1-34a)
D1-92a CH2(D1-37a)
D1-92a CH2(D1-81a)
D1-92a CH2(D1-82a)
D1-92a CH2(D1-84a)
D1-92a CH2(D1-85a)
D1-92a CH2(D1-87a)
D1-92a CH2(D1-92a)
D1-92a CH2(D1-93a)
D1-92a CH2(D1-95a)
D1-92a CH2(D1-96a)
D1-92a CH2(D1-98a)
D1-92a CH2(D1-108a)
D1-92a CH2(D1-108b,Z=2-Cl)
D1-92a CH2(D1-108b,Z=3-Me)
D1-92a CH2(D1-108b,Z=4-OMe)
D1-92a CH2(D1-108b,Z=2-SMe)
D1-92a CH2(D1-108b,Z=3-CF3)
D1-92a CH2(D1-108b,Z=4-OCF3)
D1-92a CH2(D1-108b,Z=2-SCF3)
D1-92a CH2CH2CN
D1-92a CH2CH2CF3
D1-92a CH2CH2OMe
D1-92a CH2CH2SMe
D1-92a CH2CH2S(O)Me
D1-92a CH2CH2S(O)2Me
D1-92a D1-32a
D1-92a D1-33a
D1-92a D1-34a
D1-92a D1-37a
D1-92a D1-81a
D1-92a D1-82a
D1-92a D1-84a
D1-92a D1-85a
D1-92a D1-87a
D1-92a D1-92a
D1-92a D1-93a
D1-92a D1-95a
D1-92a D1-96a
D1-92a D1-98a
D1-92a D1-108a
D1-92a D1-108b(Z=2-Cl)
D1-92a D1-108b(Z=3-Me)
D1-92a D1-108b(Z=4-OMe)
D1-92a D1-108b(Z=2-SMe)
D1-92a D1-108b(Z=3-CF3)
D1-92a D1-108b(Z=4-OCF3)
D1-92a D1-108b(Z=2-SCF3)
D1-92a C(O)Me
D1-92a C(O)CF3
D1-92a C(O)OMe
D1-93a Me
D1-93a Et
D1-93a Pr-n
D1-93a Pr-i
D1-93a Pr-c
D1-93a Bu-n
D1-93a Bu-i
D1-93a Bu-c
D1-93a Bu-s
D1-93a Bu-t
D1-93a Pen-n
D1-93a Pen-c
D1-93a Hex-n
D1-93a Hex-c
D1-93a CH2Pr-c
D1-93a CH2Bu-c
D1-93a CH2Pen-c
D1-93a CH2Hex-c
D1-93a CH2CH=CH2
D1-93a CH2CH=C(Cl)2
D1-93a CH2C≡CH
D1-93a CH2CN
D1-93a CH2CF3
D1-93a CH2OMe
D1-93a CH2OCF3
D1-93a CH2SMe
D1-93a CH2S(O)Me
D1-93a CH2S(O)2Me
D1-93a CH2SCF3
D1-93a CH2S(O)CF3
D1-93a CH2S(O)2CF3
D1-93a CH2CH(OMe)2
D1-93a CH2CH(SMe)2
D1-93a CH2C(O)Me
D1-93a CH2C(O)CF3
D1-93a CH2C(O)OMe
D1-93a CH2(D1-32a)
D1-93a CH2(D1-33a)
D1-93a CH2(D1-34a)
D1-93a CH2(D1-37a)
D1-93a CH2(D1-81a)
D1-93a CH2(D1-82a)
D1-93a CH2(D1-84a)
D1-93a CH2(D1-85a)
D1-93a CH2(D1-87a)
D1-93a CH2(D1-92a)
D1-93a CH2(D1-93a)
D1-93a CH2(D1-95a)
D1-93a CH2(D1-96a)
D1-93a CH2(D1-98a)
D1-93a CH2(D1-108a)
D1-93a CH2(D1-108b,Z=2-Cl)
D1-93a CH2(D1-108b,Z=3-Me)
D1-93a CH2(D1-108b,Z=4-OMe)
D1-93a CH2(D1-108b,Z=2-SMe)
D1-93a CH2(D1-108b,Z=3-CF3)
D1-93a CH2(D1-108b,Z=4-OCF3)
D1-93a CH2(D1-108b,Z=2-SCF3)
D1-93a CH2CH2CN
D1-93a CH2CH2CF3
D1-93a CH2CH2OMe
D1-93a CH2CH2SMe
D1-93a CH2CH2S(O)Me
D1-93a CH2CH2S(O)2Me
D1-93a D1-32a
D1-93a D1-33a
D1-93a D1-34a
D1-93a D1-37a
D1-93a D1-81a
D1-93a D1-82a
D1-93a D1-84a
D1-93a D1-85a
D1-93a D1-87a
D1-93a D1-92a
D1-93a D1-93a
D1-93a D1-95a
D1-93a D1-96a
D1-93a D1-98a
D1-93a D1-108a
D1-93a D1-108b(Z=2-Cl)
D1-93a D1-108b(Z=3-Me)
D1-93a D1-108b(Z=4-OMe)
D1-93a D1-108b(Z=2-SMe)
D1-93a D1-108b(Z=3-CF3)
D1-93a D1-108b(Z=4-OCF3)
D1-93a D1-108b(Z=2-SCF3)
D1-93a C(O)Me
D1-93a C(O)CF3
D1-93a C(O)OMe
D1-95a Me
D1-95a Et
D1-95a Pr-n
D1-95a Pr-i
D1-95a Pr-c
D1-95a Bu-n
D1-95a Bu-i
D1-95a Bu-c
D1-95a Bu-s
D1-95a Bu-t
D1-95a Pen-n
D1-95a Pen-c
D1-95a Hex-n
D1-95a Hex-c
D1-95a CH2Pr-c
D1-95a CH2Bu-c
D1-95a CH2Pen-c
D1-95a CH2Hex-c
D1-95a CH2CH=CH2
D1-95a CH2CH=C(Cl)2
D1-95a CH2C≡CH
D1-95a CH2CN
D1-95a CH2CF3
D1-95a CH2OMe
D1-95a CH2OCF3
D1-95a CH2SMe
D1-95a CH2S(O)Me
D1-95a CH2S(O)2Me
D1-95a CH2SCF3
D1-95a CH2S(O)CF3
D1-95a CH2S(O)2CF3
D1-95a CH2CH(OMe)2
D1-95a CH2CH(SMe)2
D1-95a CH2C(O)Me
D1-95a CH2C(O)CF3
D1-95a CH2C(O)OMe
D1-95a CH2(D1-32a)
D1-95a CH2(D1-33a)
D1-95a CH2(D1-34a)
D1-95a CH2(D1-37a)
D1-95a CH2(D1-81a)
D1-95a CH2(D1-82a)
D1-95a CH2(D1-84a)
D1-95a CH2(D1-85a)
D1-95a CH2(D1-87a)
D1-95a CH2(D1-92a)
D1-95a CH2(D1-93a)
D1-95a CH2(D1-95a)
D1-95a CH2(D1-96a)
D1-95a CH2(D1-98a)
D1-95a CH2(D1-108a)
D1-95a CH2(D1-108b,Z=2-Cl)
D1-95a CH2(D1-108b,Z=3-Me)
D1-95a CH2(D1-108b,Z=4-OMe)
D1-95a CH2(D1-108b,Z=2-SMe)
D1-95a CH2(D1-108b,Z=3-CF3)
D1-95a CH2(D1-108b,Z=4-OCF3)
D1-95a CH2(D1-108b,Z=2-SCF3)
D1-95a CH2CH2CN
D1-95a CH2CH2CF3
D1-95a CH2CH2OMe
D1-95a CH2CH2SMe
D1-95a CH2CH2S(O)Me
D1-95a CH2CH2S(O)2Me
D1-95a D1-32a
D1-95a D1-33a
D1-95a D1-34a
D1-95a D1-37a
D1-95a D1-81a
D1-95a D1-82a
D1-95a D1-84a
D1-95a D1-85a
D1-95a D1-87a
D1-95a D1-92a
D1-95a D1-93a
D1-95a D1-95a
D1-95a D1-96a
D1-95a D1-98a
D1-95a D1-108a
D1-95a D1-108b(Z=2-Cl)
D1-95a D1-108b(Z=3-Me)
D1-95a D1-108b(Z=4-OMe)
D1-95a D1-108b(Z=2-SMe)
D1-95a D1-108b(Z=3-CF3)
D1-95a D1-108b(Z=4-OCF3)
D1-95a D1-108b(Z=2-SCF3)
D1-95a C(O)Me
D1-95a C(O)CF3
D1-95a C(O)OMe
D1-96a Me
D1-96a Et
D1-96a Pr-n
D1-96a Pr-i
D1-96a Pr-c
D1-96a Bu-n
D1-96a Bu-i
D1-96a Bu-c
D1-96a Bu-s
D1-96a Bu-t
D1-96a Pen-n
D1-96a Pen-c
D1-96a Hex-n
D1-96a Hex-c
D1-96a CH2Pr-c
D1-96a CH2Bu-c
D1-96a CH2Pen-c
D1-96a CH2Hex-c
D1-96a CH2CH=CH2
D1-96a CH2CH=C(Cl)2
D1-96a CH2C≡CH
D1-96a CH2CN
D1-96a CH2CF3
D1-96a CH2OMe
D1-96a CH2OCF3
D1-96a CH2SMe
D1-96a CH2S(O)Me
D1-96a CH2S(O)2Me
D1-96a CH2SCF3
D1-96a CH2S(O)CF3
D1-96a CH2S(O)2CF3
D1-96a CH2CH(OMe)2
D1-96a CH2CH(SMe)2
D1-96a CH2C(O)Me
D1-96a CH2C(O)CF3
D1-96a CH2C(O)OMe
D1-96a CH2(D1-32a)
D1-96a CH2(D1-33a)
D1-96a CH2(D1-34a)
D1-96a CH2(D1-37a)
D1-96a CH2(D1-81a)
D1-96a CH2(D1-82a)
D1-96a CH2(D1-84a)
D1-96a CH2(D1-85a)
D1-96a CH2(D1-87a)
D1-96a CH2(D1-92a)
D1-96a CH2(D1-93a)
D1-96a CH2(D1-95a)
D1-96a CH2(D1-96a)
D1-96a CH2(D1-98a)
D1-96a CH2(D1-108a)
D1-96a CH2(D1-108b,Z=2-Cl)
D1-96a CH2(D1-108b,Z=3-Me)
D1-96a CH2(D1-108b,Z=4-OMe)
D1-96a CH2(D1-108b,Z=2-SMe)
D1-96a CH2(D1-108b,Z=3-CF3)
D1-96a CH2(D1-108b,Z=4-OCF3)
D1-96a CH2(D1-108b,Z=2-SCF3)
D1-96a CH2CH2CN
D1-96a CH2CH2CF3
D1-96a CH2CH2OMe
D1-96a CH2CH2SMe
D1-96a CH2CH2S(O)Me
D1-96a CH2CH2S(O)2Me
D1-96a D1-32a
D1-96a D1-33a
D1-96a D1-34a
D1-96a D1-37a
D1-96a D1-81a
D1-96a D1-82a
D1-96a D1-84a
D1-96a D1-85a
D1-96a D1-87a
D1-96a D1-92a
D1-96a D1-93a
D1-96a D1-95a
D1-96a D1-96a
D1-96a D1-98a
D1-96a D1-108a
D1-96a D1-108b(Z=2-Cl)
D1-96a D1-108b(Z=3-Me)
D1-96a D1-108b(Z=4-OMe)
D1-96a D1-108b(Z=2-SMe)
D1-96a D1-108b(Z=3-CF3)
D1-96a D1-108b(Z=4-OCF3)
D1-96a D1-108b(Z=2-SCF3)
D1-96a C(O)Me
D1-96a C(O)CF3
D1-96a C(O)OMe
D1-98a Me
D1-98a Et
D1-98a Pr-n
D1-98a Pr-i
D1-98a Pr-c
D1-98a Bu-n
D1-98a Bu-i
D1-98a Bu-c
D1-98a Bu-s
D1-98a Bu-t
D1-98a Pen-n
D1-98a Pen-c
D1-98a Hex-n
D1-98a Hex-c
D1-98a CH2Pr-c
D1-98a CH2Bu-c
D1-98a CH2Pen-c
D1-98a CH2Hex-c
D1-98a CH2CH=CH2
D1-98a CH2CH=C(Cl)2
D1-98a CH2C≡CH
D1-98a CH2CN
D1-98a CH2CF3
D1-98a CH2OMe
D1-98a CH2OCF3
D1-98a CH2SMe
D1-98a CH2S(O)Me
D1-98a CH2S(O)2Me
D1-98a CH2SCF3
D1-98a CH2S(O)CF3
D1-98a CH2S(O)2CF3
D1-98a CH2CH(OMe)2
D1-98a CH2CH(SMe)2
D1-98a CH2C(O)Me
D1-98a CH2C(O)CF3
D1-98a CH2C(O)OMe
D1-98a CH2(D1-32a)
D1-98a CH2(D1-33a)
D1-98a CH2(D1-34a)
D1-98a CH2(D1-37a)
D1-98a CH2(D1-81a)
D1-98a CH2(D1-82a)
D1-98a CH2(D1-84a)
D1-98a CH2(D1-85a)
D1-98a CH2(D1-87a)
D1-98a CH2(D1-92a)
D1-98a CH2(D1-93a)
D1-98a CH2(D1-95a)
D1-98a CH2(D1-96a)
D1-98a CH2(D1-98a)
D1-98a CH2(D1-108a)
D1-98a CH2(D1-108b,Z=2-Cl)
D1-98a CH2(D1-108b,Z=3-Me)
D1-98a CH2(D1-108b,Z=4-OMe)
D1-98a CH2(D1-108b,Z=2-SMe)
D1-98a CH2(D1-108b,Z=3-CF3)
D1-98a CH2(D1-108b,Z=4-OCF3)
D1-98a CH2(D1-108b,Z=2-SCF3)
D1-98a CH2CH2CN
D1-98a CH2CH2CF3
D1-98a CH2CH2OMe
D1-98a CH2CH2SMe
D1-98a CH2CH2S(O)Me
D1-98a CH2CH2S(O)2Me
D1-98a D1-32a
D1-98a D1-33a
D1-98a D1-34a
D1-98a D1-37a
D1-98a D1-81a
D1-98a D1-82a
D1-98a D1-84a
D1-98a D1-85a
D1-98a D1-87a
D1-98a D1-92a
D1-98a D1-93a
D1-98a D1-95a
D1-98a D1-96a
D1-98a D1-98a
D1-98a D1-108a
D1-98a D1-108b(Z=2-Cl)
D1-98a D1-108b(Z=3-Me)
D1-98a D1-108b(Z=4-OMe)
D1-98a D1-108b(Z=2-SMe)
D1-98a D1-108b(Z=3-CF3)
D1-98a D1-108b(Z=4-OCF3)
D1-98a D1-108b(Z=2-SCF3)
D1-98a C(O)Me
D1-98a C(O)CF3
D1-98a C(O)OMe
D1-108a Me
D1-108a Et
D1-108a Pr-n
D1-108a Pr-i
D1-108a Pr-c
D1-108a Bu-n
D1-108a Bu-i
D1-108a Bu-c
D1-108a Bu-s
D1-108a Bu-t
D1-108a Pen-n
D1-108a Pen-c
D1-108a Hex-n
D1-108a Hex-c
D1-108a CH2Pr-c
D1-108a CH2Bu-c
D1-108a CH2Pen-c
D1-108a CH2Hex-c
D1-108a CH2CH=CH2
D1-108a CH2CH=C(Cl)2
D1-108a CH2C≡CH
D1-108a CH2CN
D1-108a CH2CF3
D1-108a CH2OMe
D1-108a CH2OCF3
D1-108a CH2SMe
D1-108a CH2S(O)Me
D1-108a CH2S(O)2Me
D1-108a CH2SCF3
D1-108a CH2S(O)CF3
D1-108a CH2S(O)2CF3
D1-108a CH2CH(OMe)2
D1-108a CH2CH(SMe)2
D1-108a CH2C(O)Me
D1-108a CH2C(O)CF3
D1-108a CH2C(O)OMe
D1-108a CH2(D1-32a)
D1-108a CH2(D1-33a)
D1-108a CH2(D1-34a)
D1-108a CH2(D1-37a)
D1-108a CH2(D1-81a)
D1-108a CH2(D1-82a)
D1-108a CH2(D1-84a)
D1-108a CH2(D1-85a)
D1-108a CH2(D1-87a)
D1-108a CH2(D1-92a)
D1-108a CH2(D1-93a)
D1-108a CH2(D1-95a)
D1-108a CH2(D1-96a)
D1-108a CH2(D1-98a)
D1-108a CH2(D1-108a)
D1-108a CH2(D1-108b,Z=2-Cl)
D1-108a CH2(D1-108b,Z=3-Me)
D1-108a CH2(D1-108b,Z=4-OMe)
D1-108a CH2(D1-108b,Z=2-SMe)
D1-108a CH2(D1-108b,Z=3-CF3)
D1-108a CH2(D1-108b,Z=4-OCF3)
D1-108a CH2(D1-108b,Z=2-SCF3)
D1-108a CH2CH2CN
D1-108a CH2CH2CF3
D1-108a CH2CH2OMe
D1-108a CH2CH2SMe
D1-108a CH2CH2S(O)Me
D1-108a CH2CH2S(O)2Me
D1-108a D1-32a
D1-108a D1-33a
D1-108a D1-34a
D1-108a D1-37a
D1-108a D1-81a
D1-108a D1-82a
D1-108a D1-84a
D1-108a D1-85a
D1-108a D1-87a
D1-108a D1-92a
D1-108a D1-93a
D1-108a D1-95a
D1-108a D1-96a
D1-108a D1-98a
D1-108a D1-108a
D1-108a D1-108b(Z=2-Cl)
D1-108a D1-108b(Z=3-Me)
D1-108a D1-108b(Z=4-OMe)
D1-108a D1-108b(Z=2-SMe)
D1-108a D1-108b(Z=3-CF3)
D1-108a D1-108b(Z=4-OCF3)
D1-108a D1-108b(Z=2-SCF3)
D1-108a C(O)Me
D1-108a C(O)CF3
D1-108a C(O)OMe
CH2SCH2CH2CF3 Me
CH2SCH2CH2CF3 Et
CH2SCH2CH2CF3 Pr-n
CH2SCH2CH2CF3 Pr-i
CH2SCH2CH2CF3 Pr-c
CH2SCH2CH2CF3 Bu-n
CH2SCH2CH2CF3 Bu-i
CH2SCH2CH2CF3 Bu-c
CH2SCH2CH2CF3 Bu-s
CH2SCH2CH2CF3 Bu-t
CH2SCH2CH2CF3 Pen-n
CH2SCH2CH2CF3 Pen-c
CH2SCH2CH2CF3 Hex-n
CH2SCH2CH2CF3 Hex-c
CH2SCH2CH2CF3 CH2Pr-c
CH2SCH2CH2CF3 CH2Bu-c
CH2SCH2CH2CF3 CH2Pen-c
CH2SCH2CH2CF3 CH2Hex-c
CH2SCH2CH2CF3 CH2CH=CH2
CH2SCH2CH2CF3 CH2CH=C(Cl)2
CH2SCH2CH2CF3 CH2C≡CH
CH2SCH2CH2CF3 CH2CN
CH2SCH2CH2CF3 CH2CF3
CH2SCH2CH2CF3 CH2OMe
CH2SCH2CH2CF3 CH2OCF3
CH2SCH2CH2CF3 CH2SMe
CH2SCH2CH2CF3 CH2S(O)Me
CH2SCH2CH2CF3 CH2S(O)2Me
CH2SCH2CH2CF3 CH2SCF3
CH2SCH2CH2CF3 CH2S(O)CF3
CH2SCH2CH2CF3 CH2S(O)2CF3
CH2SCH2CH2CF3 CH2CH(OMe)2
CH2SCH2CH2CF3 CH2CH(SMe)2
CH2SCH2CH2CF3 CH2C(O)Me
CH2SCH2CH2CF3 CH2C(O)CF3
CH2SCH2CH2CF3 CH2C(O)OMe
CH2SCH2CH2CF3 CH2(D1-32a)
CH2SCH2CH2CF3 CH2(D1-33a)
CH2SCH2CH2CF3 CH2(D1-34a)
CH2SCH2CH2CF3 CH2(D1-37a)
CH2SCH2CH2CF3 CH2(D1-81a)
CH2SCH2CH2CF3 CH2(D1-82a)
CH2SCH2CH2CF3 CH2(D1-84a)
CH2SCH2CH2CF3 CH2(D1-85a)
CH2SCH2CH2CF3 CH2(D1-87a)
CH2SCH2CH2CF3 CH2(D1-92a)
CH2SCH2CH2CF3 CH2(D1-93a)
CH2SCH2CH2CF3 CH2(D1-95a)
CH2SCH2CH2CF3 CH2(D1-96a)
CH2SCH2CH2CF3 CH2(D1-98a)
CH2SCH2CH2CF3 CH2(D1-108a)
CH2SCH2CH2CF3 CH2(D1-108b,Z=2-Cl)
CH2SCH2CH2CF3 CH2(D1-108b,Z=3-Me)
CH2SCH2CH2CF3 CH2(D1-108b,Z=4-OMe)
CH2SCH2CH2CF3 CH2(D1-108b,Z=2-SMe)
CH2SCH2CH2CF3 CH2(D1-108b,Z=3-CF3)
CH2SCH2CH2CF3 CH2(D1-108b,Z=4-OCF3)
CH2SCH2CH2CF3 CH2(D1-108b,Z=2-SCF3)
CH2SCH2CH2CF3 CH2CH2CN
CH2SCH2CH2CF3 CH2CH2CF3
CH2SCH2CH2CF3 CH2CH2OMe
CH2SCH2CH2CF3 CH2CH2SMe
CH2SCH2CH2CF3 CH2CH2S(O)Me
CH2SCH2CH2CF3 CH2CH2S(O)2Me
CH2SCH2CH2CF3 D1-32a
CH2SCH2CH2CF3 D1-33a
CH2SCH2CH2CF3 D1-34a
CH2SCH2CH2CF3 D1-37a
CH2SCH2CH2CF3 D1-81a
CH2SCH2CH2CF3 D1-82a
CH2SCH2CH2CF3 D1-84a
CH2SCH2CH2CF3 D1-85a
CH2SCH2CH2CF3 D1-87a
CH2SCH2CH2CF3 D1-92a
CH2SCH2CH2CF3 D1-93a
CH2SCH2CH2CF3 D1-95a
CH2SCH2CH2CF3 D1-96a
CH2SCH2CH2CF3 D1-98a
CH2SCH2CH2CF3 D1-108a
CH2SCH2CH2CF3 D1-108b(Z=2-Cl)
CH2SCH2CH2CF3 D1-108b(Z=3-Me)
CH2SCH2CH2CF3 D1-108b(Z=4-OMe)
CH2SCH2CH2CF3 D1-108b(Z=2-SMe)
CH2SCH2CH2CF3 D1-108b(Z=3-CF3)
CH2SCH2CH2CF3 D1-108b(Z=4-OCF3)
CH2SCH2CH2CF3 D1-108b(Z=2-SCF3)
CH2SCH2CH2CF3 C(O)Me
CH2SCH2CH2CF3 C(O)CF3
CH2SCH2CH2CF3 C(O)OMe
CH2S(O)CH2CH2CF3 Me
CH2S(O)CH2CH2CF3 Et
CH2S(O)CH2CH2CF3 Pr-n
CH2S(O)CH2CH2CF3 Pr-i
CH2S(O)CH2CH2CF3 Pr-c
CH2S(O)CH2CH2CF3 Bu-n
CH2S(O)CH2CH2CF3 Bu-i
CH2S(O)CH2CH2CF3 Bu-c
CH2S(O)CH2CH2CF3 Bu-s
CH2S(O)CH2CH2CF3 Bu-t
CH2S(O)CH2CH2CF3 Pen-n
CH2S(O)CH2CH2CF3 Pen-c
CH2S(O)CH2CH2CF3 Hex-n
CH2S(O)CH2CH2CF3 Hex-c
CH2S(O)CH2CH2CF3 CH2Pr-c
CH2S(O)CH2CH2CF3 CH2Bu-c
CH2S(O)CH2CH2CF3 CH2Pen-c
CH2S(O)CH2CH2CF3 CH2Hex-c
CH2S(O)CH2CH2CF3 CH2CH=CH2
CH2S(O)CH2CH2CF3 CH2CH=C(Cl)2
CH2S(O)CH2CH2CF3 CH2C≡CH
CH2S(O)CH2CH2CF3 CH2CN
CH2S(O)CH2CH2CF3 CH2CF3
CH2S(O)CH2CH2CF3 CH2OMe
CH2S(O)CH2CH2CF3 CH2OCF3
CH2S(O)CH2CH2CF3 CH2SMe
CH2S(O)CH2CH2CF3 CH2S(O)Me
CH2S(O)CH2CH2CF3 CH2S(O)2Me
CH2S(O)CH2CH2CF3 CH2SCF3
CH2S(O)CH2CH2CF3 CH2S(O)CF3
CH2S(O)CH2CH2CF3 CH2S(O)2CF3
CH2S(O)CH2CH2CF3 CH2CH(OMe)2
CH2S(O)CH2CH2CF3 CH2CH(SMe)2
CH2S(O)CH2CH2CF3 CH2C(O)Me
CH2S(O)CH2CH2CF3 CH2C(O)CF3
CH2S(O)CH2CH2CF3 CH2C(O)OMe
CH2S(O)CH2CH2CF3 CH2(D1-32a)
CH2S(O)CH2CH2CF3 CH2(D1-33a)
CH2S(O)CH2CH2CF3 CH2(D1-34a)
CH2S(O)CH2CH2CF3 CH2(D1-37a)
CH2S(O)CH2CH2CF3 CH2(D1-81a)
CH2S(O)CH2CH2CF3 CH2(D1-82a)
CH2S(O)CH2CH2CF3 CH2(D1-84a)
CH2S(O)CH2CH2CF3 CH2(D1-85a)
CH2S(O)CH2CH2CF3 CH2(D1-87a)
CH2S(O)CH2CH2CF3 CH2(D1-92a)
CH2S(O)CH2CH2CF3 CH2(D1-93a)
CH2S(O)CH2CH2CF3 CH2(D1-95a)
CH2S(O)CH2CH2CF3 CH2(D1-96a)
CH2S(O)CH2CH2CF3 CH2(D1-98a)
CH2S(O)CH2CH2CF3 CH2(D1-108a)
CH2S(O)CH2CH2CF3 CH2(D1-108b,Z=2-Cl)
CH2S(O)CH2CH2CF3 CH2(D1-108b,Z=3-Me)
CH2S(O)CH2CH2CF3 CH2(D1-108b,Z=4-OMe)
CH2S(O)CH2CH2CF3 CH2(D1-108b,Z=2-SMe)
CH2S(O)CH2CH2CF3 CH2(D1-108b,Z=3-CF3)
CH2S(O)CH2CH2CF3 CH2(D1-108b,Z=4-OCF3)
CH2S(O)CH2CH2CF3 CH2(D1-108b,Z=2-SCF3)
CH2S(O)CH2CH2CF3 CH2CH2CN
CH2S(O)CH2CH2CF3 CH2CH2CF3
CH2S(O)CH2CH2CF3 CH2CH2OMe
CH2S(O)CH2CH2CF3 CH2CH2SMe
CH2S(O)CH2CH2CF3 CH2CH2S(O)Me
CH2S(O)CH2CH2CF3 CH2CH2S(O)2Me
CH2S(O)CH2CH2CF3 D1-32a
CH2S(O)CH2CH2CF3 D1-33a
CH2S(O)CH2CH2CF3 D1-34a
CH2S(O)CH2CH2CF3 D1-37a
CH2S(O)CH2CH2CF3 D1-81a
CH2S(O)CH2CH2CF3 D1-82a
CH2S(O)CH2CH2CF3 D1-84a
CH2S(O)CH2CH2CF3 D1-85a
CH2S(O)CH2CH2CF3 D1-87a
CH2S(O)CH2CH2CF3 D1-92a
CH2S(O)CH2CH2CF3 D1-93a
CH2S(O)CH2CH2CF3 D1-95a
CH2S(O)CH2CH2CF3 D1-96a
CH2S(O)CH2CH2CF3 D1-98a
CH2S(O)CH2CH2CF3 D1-108a
CH2S(O)CH2CH2CF3 D1-108b(Z=2-Cl)
CH2S(O)CH2CH2CF3 D1-108b(Z=3-Me)
CH2S(O)CH2CH2CF3 D1-108b(Z=4-OMe)
CH2S(O)CH2CH2CF3 D1-108b(Z=2-SMe)
CH2S(O)CH2CH2CF3 D1-108b(Z=3-CF3)
CH2S(O)CH2CH2CF3 D1-108b(Z=4-OCF3)
CH2S(O)CH2CH2CF3 D1-108b(Z=2-SCF3)
CH2S(O)CH2CH2CF3 C(O)Me
CH2S(O)CH2CH2CF3 C(O)CF3
CH2S(O)CH2CH2CF3 C(O)OMe
CH2S(O)2CH2CH2CF3 Me
CH2S(O)2CH2CH2CF3 Et
CH2S(O)2CH2CH2CF3 Pr-n
CH2S(O)2CH2CH2CF3 Pr-i
CH2S(O)2CH2CH2CF3 Pr-c
CH2S(O)2CH2CH2CF3 Bu-n
CH2S(O)2CH2CH2CF3 Bu-i
CH2S(O)2CH2CH2CF3 Bu-c
CH2S(O)2CH2CH2CF3 Bu-s
CH2S(O)2CH2CH2CF3 Bu-t
CH2S(O)2CH2CH2CF3 Pen-n
CH2S(O)2CH2CH2CF3 Pen-c
CH2S(O)2CH2CH2CF3 Hex-n
CH2S(O)2CH2CH2CF3 Hex-c
CH2S(O)2CH2CH2CF3 CH2Pr-c
CH2S(O)2CH2CH2CF3 CH2Bu-c
CH2S(O)2CH2CH2CF3 CH2Pen-c
CH2S(O)2CH2CH2CF3 CH2Hex-c
CH2S(O)2CH2CH2CF3 CH2CH=CH2
CH2S(O)2CH2CH2CF3 CH2CH=C(Cl)2
CH2S(O)2CH2CH2CF3 CH2C≡CH
CH2S(O)2CH2CH2CF3 CH2CN
CH2S(O)2CH2CH2CF3 CH2CF3
CH2S(O)2CH2CH2CF3 CH2OMe
CH2S(O)2CH2CH2CF3 CH2OCF3
CH2S(O)2CH2CH2CF3 CH2SMe
CH2S(O)2CH2CH2CF3 CH2S(O)Me
CH2S(O)2CH2CH2CF3 CH2S(O)2Me
CH2S(O)2CH2CH2CF3 CH2SCF3
CH2S(O)2CH2CH2CF3 CH2S(O)CF3
CH2S(O)2CH2CH2CF3 CH2S(O)2CF3
CH2S(O)2CH2CH2CF3 CH2CH(OMe)2
CH2S(O)2CH2CH2CF3 CH2CH(SMe)2
CH2S(O)2CH2CH2CF3 CH2C(O)Me
CH2S(O)2CH2CH2CF3 CH2C(O)CF3
CH2S(O)2CH2CH2CF3 CH2C(O)OMe
CH2S(O)2CH2CH2CF3 CH2(D1-32a)
CH2S(O)2CH2CH2CF3 CH2(D1-33a)
CH2S(O)2CH2CH2CF3 CH2(D1-34a)
CH2S(O)2CH2CH2CF3 CH2(D1-37a)
CH2S(O)2CH2CH2CF3 CH2(D1-81a)
CH2S(O)2CH2CH2CF3 CH2(D1-82a)
CH2S(O)2CH2CH2CF3 CH2(D1-84a)
CH2S(O)2CH2CH2CF3 CH2(D1-85a)
CH2S(O)2CH2CH2CF3 CH2(D1-87a)
CH2S(O)2CH2CH2CF3 CH2(D1-92a)
CH2S(O)2CH2CH2CF3 CH2(D1-93a)
CH2S(O)2CH2CH2CF3 CH2(D1-95a)
CH2S(O)2CH2CH2CF3 CH2(D1-96a)
CH2S(O)2CH2CH2CF3 CH2(D1-98a)
CH2S(O)2CH2CH2CF3 CH2(D1-108a)
CH2S(O)2CH2CH2CF3 CH2(D1-108b,Z=2-Cl)
CH2S(O)2CH2CH2CF3 CH2(D1-108b,Z=3-Me)
CH2S(O)2CH2CH2CF3 CH2(D1-108b,Z=4-OMe)
CH2S(O)2CH2CH2CF3 CH2(D1-108b,Z=2-SMe)
CH2S(O)2CH2CH2CF3 CH2(D1-108b,Z=3-CF3)
CH2S(O)2CH2CH2CF3 CH2(D1-108b,Z=4-OCF3)
CH2S(O)2CH2CH2CF3 CH2(D1-108b,Z=2-SCF3)
CH2S(O)2CH2CH2CF3 CH2CH2CN
CH2S(O)2CH2CH2CF3 CH2CH2CF3
CH2S(O)2CH2CH2CF3 CH2CH2OMe
CH2S(O)2CH2CH2CF3 CH2CH2SMe
CH2S(O)2CH2CH2CF3 CH2CH2S(O)Me
CH2S(O)2CH2CH2CF3 CH2CH2S(O)2Me
CH2S(O)2CH2CH2CF3 D1-32a
CH2S(O)2CH2CH2CF3 D1-33a
CH2S(O)2CH2CH2CF3 D1-34a
CH2S(O)2CH2CH2CF3 D1-37a
CH2S(O)2CH2CH2CF3 D1-81a
CH2S(O)2CH2CH2CF3 D1-82a
CH2S(O)2CH2CH2CF3 D1-84a
CH2S(O)2CH2CH2CF3 D1-85a
CH2S(O)2CH2CH2CF3 D1-87a
CH2S(O)2CH2CH2CF3 D1-92a
CH2S(O)2CH2CH2CF3 D1-93a
CH2S(O)2CH2CH2CF3 D1-95a
CH2S(O)2CH2CH2CF3 D1-96a
CH2S(O)2CH2CH2CF3 D1-98a
CH2S(O)2CH2CH2CF3 D1-108a
CH2S(O)2CH2CH2CF3 D1-108b(Z=2-Cl)
CH2S(O)2CH2CH2CF3 D1-108b(Z=3-Me)
CH2S(O)2CH2CH2CF3 D1-108b(Z=4-OMe)
CH2S(O)2CH2CH2CF3 D1-108b(Z=2-SMe)
CH2S(O)2CH2CH2CF3 D1-108b(Z=3-CF3)
CH2S(O)2CH2CH2CF3 D1-108b(Z=4-OCF3)
CH2S(O)2CH2CH2CF3 D1-108b(Z=2-SCF3)
CH2S(O)2CH2CH2CF3 C(O)Me
CH2S(O)2CH2CH2CF3 C(O)CF3
CH2S(O)2CH2CH2CF3 C(O)OMe
CH(Me)SCH2CH2CF3 Me
CH(Me)SCH2CH2CF3 Et
CH(Me)SCH2CH2CF3 Pr-n
CH(Me)SCH2CH2CF3 Pr-i
CH(Me)SCH2CH2CF3 Pr-c
CH(Me)SCH2CH2CF3 Bu-n
CH(Me)SCH2CH2CF3 Bu-i
CH(Me)SCH2CH2CF3 Bu-c
CH(Me)SCH2CH2CF3 Bu-s
CH(Me)SCH2CH2CF3 Bu-t
CH(Me)SCH2CH2CF3 Pen-n
CH(Me)SCH2CH2CF3 Pen-c
CH(Me)SCH2CH2CF3 Hex-n
CH(Me)SCH2CH2CF3 Hex-c
CH(Me)SCH2CH2CF3 CH2Pr-c
CH(Me)SCH2CH2CF3 CH2Bu-c
CH(Me)SCH2CH2CF3 CH2Pen-c
CH(Me)SCH2CH2CF3 CH2Hex-c
CH(Me)SCH2CH2CF3 CH2CH=CH2
CH(Me)SCH2CH2CF3 CH2CH=C(Cl)2
CH(Me)SCH2CH2CF3 CH2C≡CH
CH(Me)SCH2CH2CF3 CH2CN
CH(Me)SCH2CH2CF3 CH2CF3
CH(Me)SCH2CH2CF3 CH2OMe
CH(Me)SCH2CH2CF3 CH2OCF3
CH(Me)SCH2CH2CF3 CH2SMe
CH(Me)SCH2CH2CF3 CH2S(O)Me
CH(Me)SCH2CH2CF3 CH2S(O)2Me
CH(Me)SCH2CH2CF3 CH2SCF3
CH(Me)SCH2CH2CF3 CH2S(O)CF3
CH(Me)SCH2CH2CF3 CH2S(O)2CF3
CH(Me)SCH2CH2CF3 CH2CH(OMe)2
CH(Me)SCH2CH2CF3 CH2CH(SMe)2
CH(Me)SCH2CH2CF3 CH2C(O)Me
CH(Me)SCH2CH2CF3 CH2C(O)CF3
CH(Me)SCH2CH2CF3 CH2C(O)OMe
CH(Me)SCH2CH2CF3 CH2(D1-32a)
CH(Me)SCH2CH2CF3 CH2(D1-33a)
CH(Me)SCH2CH2CF3 CH2(D1-34a)
CH(Me)SCH2CH2CF3 CH2(D1-37a)
CH(Me)SCH2CH2CF3 CH2(D1-81a)
CH(Me)SCH2CH2CF3 CH2(D1-82a)
CH(Me)SCH2CH2CF3 CH2(D1-84a)
CH(Me)SCH2CH2CF3 CH2(D1-85a)
CH(Me)SCH2CH2CF3 CH2(D1-87a)
CH(Me)SCH2CH2CF3 CH2(D1-92a)
CH(Me)SCH2CH2CF3 CH2(D1-93a)
CH(Me)SCH2CH2CF3 CH2(D1-95a)
CH(Me)SCH2CH2CF3 CH2(D1-96a)
CH(Me)SCH2CH2CF3 CH2(D1-98a)
CH(Me)SCH2CH2CF3 CH2(D1-108a)
CH(Me)SCH2CH2CF3 CH2(D1-108b,Z=2-Cl)
CH(Me)SCH2CH2CF3 CH2(D1-108b,Z=3-Me)
CH(Me)SCH2CH2CF3 CH2(D1-108b,Z=4-OMe)
CH(Me)SCH2CH2CF3 CH2(D1-108b,Z=2-SMe)
CH(Me)SCH2CH2CF3 CH2(D1-108b,Z=3-CF3)
CH(Me)SCH2CH2CF3 CH2(D1-108b,Z=4-OCF3)
CH(Me)SCH2CH2CF3 CH2(D1-108b,Z=2-SCF3)
CH(Me)SCH2CH2CF3 CH2CH2CN
CH(Me)SCH2CH2CF3 CH2CH2CF3
CH(Me)SCH2CH2CF3 CH2CH2OMe
CH(Me)SCH2CH2CF3 CH2CH2SMe
CH(Me)SCH2CH2CF3 CH2CH2S(O)Me
CH(Me)SCH2CH2CF3 CH2CH2S(O)2Me
CH(Me)SCH2CH2CF3 D1-32a
CH(Me)SCH2CH2CF3 D1-33a
CH(Me)SCH2CH2CF3 D1-34a
CH(Me)SCH2CH2CF3 D1-37a
CH(Me)SCH2CH2CF3 D1-81a
CH(Me)SCH2CH2CF3 D1-82a
CH(Me)SCH2CH2CF3 D1-84a
CH(Me)SCH2CH2CF3 D1-85a
CH(Me)SCH2CH2CF3 D1-87a
CH(Me)SCH2CH2CF3 D1-92a
CH(Me)SCH2CH2CF3 D1-93a
CH(Me)SCH2CH2CF3 D1-95a
CH(Me)SCH2CH2CF3 D1-96a
CH(Me)SCH2CH2CF3 D1-98a
CH(Me)SCH2CH2CF3 D1-108a
CH(Me)SCH2CH2CF3 D1-108b(Z=2-Cl)
CH(Me)SCH2CH2CF3 D1-108b(Z=3-Me)
CH(Me)SCH2CH2CF3 D1-108b(Z=4-OMe)
CH(Me)SCH2CH2CF3 D1-108b(Z=2-SMe)
CH(Me)SCH2CH2CF3 D1-108b(Z=3-CF3)
CH(Me)SCH2CH2CF3 D1-108b(Z=4-OCF3)
CH(Me)SCH2CH2CF3 D1-108b(Z=2-SCF3)
CH(Me)SCH2CH2CF3 C(O)Me
CH(Me)SCH2CH2CF3 C(O)CF3
CH(Me)SCH2CH2CF3 C(O)OMe
CH(Me)S(O)CH2CH2CF3 Me
CH(Me)S(O)CH2CH2CF3 Et
CH(Me)S(O)CH2CH2CF3 Pr-n
CH(Me)S(O)CH2CH2CF3 Pr-i
CH(Me)S(O)CH2CH2CF3 Pr-c
CH(Me)S(O)CH2CH2CF3 Bu-n
CH(Me)S(O)CH2CH2CF3 Bu-i
CH(Me)S(O)CH2CH2CF3 Bu-c
CH(Me)S(O)CH2CH2CF3 Bu-s
CH(Me)S(O)CH2CH2CF3 Bu-t
CH(Me)S(O)CH2CH2CF3 Pen-n
CH(Me)S(O)CH2CH2CF3 Pen-c
CH(Me)S(O)CH2CH2CF3 Hex-n
CH(Me)S(O)CH2CH2CF3 Hex-c
CH(Me)S(O)CH2CH2CF3 CH2Pr-c
CH(Me)S(O)CH2CH2CF3 CH2Bu-c
CH(Me)S(O)CH2CH2CF3 CH2Pen-c
CH(Me)S(O)CH2CH2CF3 CH2Hex-c
CH(Me)S(O)CH2CH2CF3 CH2CH=CH2
CH(Me)S(O)CH2CH2CF3 CH2CH=C(Cl)2
CH(Me)S(O)CH2CH2CF3 CH2C≡CH
CH(Me)S(O)CH2CH2CF3 CH2CN
CH(Me)S(O)CH2CH2CF3 CH2CF3
CH(Me)S(O)CH2CH2CF3 CH2OMe
CH(Me)S(O)CH2CH2CF3 CH2OCF3
CH(Me)S(O)CH2CH2CF3 CH2SMe
CH(Me)S(O)CH2CH2CF3 CH2S(O)Me
CH(Me)S(O)CH2CH2CF3 CH2S(O)2Me
CH(Me)S(O)CH2CH2CF3 CH2SCF3
CH(Me)S(O)CH2CH2CF3 CH2S(O)CF3
CH(Me)S(O)CH2CH2CF3 CH2S(O)2CF3
CH(Me)S(O)CH2CH2CF3 CH2CH(OMe)2
CH(Me)S(O)CH2CH2CF3 CH2CH(SMe)2
CH(Me)S(O)CH2CH2CF3 CH2C(O)Me
CH(Me)S(O)CH2CH2CF3 CH2C(O)CF3
CH(Me)S(O)CH2CH2CF3 CH2C(O)OMe
CH(Me)S(O)CH2CH2CF3 CH2(D1-32a)
CH(Me)S(O)CH2CH2CF3 CH2(D1-33a)
CH(Me)S(O)CH2CH2CF3 CH2(D1-34a)
CH(Me)S(O)CH2CH2CF3 CH2(D1-37a)
CH(Me)S(O)CH2CH2CF3 CH2(D1-81a)
CH(Me)S(O)CH2CH2CF3 CH2(D1-82a)
CH(Me)S(O)CH2CH2CF3 CH2(D1-84a)
CH(Me)S(O)CH2CH2CF3 CH2(D1-85a)
CH(Me)S(O)CH2CH2CF3 CH2(D1-87a)
CH(Me)S(O)CH2CH2CF3 CH2(D1-92a)
CH(Me)S(O)CH2CH2CF3 CH2(D1-93a)
CH(Me)S(O)CH2CH2CF3 CH2(D1-95a)
CH(Me)S(O)CH2CH2CF3 CH2(D1-96a)
CH(Me)S(O)CH2CH2CF3 CH2(D1-98a)
CH(Me)S(O)CH2CH2CF3 CH2(D1-108a)
CH(Me)S(O)CH2CH2CF3 CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)CH2CH2CF3 CH2(D1-108b,Z=3-Me)
CH(Me)S(O)CH2CH2CF3 CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)CH2CH2CF3 CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)CH2CH2CF3 CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)CH2CH2CF3 CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)CH2CH2CF3 CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)CH2CH2CF3 CH2CH2CN
CH(Me)S(O)CH2CH2CF3 CH2CH2CF3
CH(Me)S(O)CH2CH2CF3 CH2CH2OMe
CH(Me)S(O)CH2CH2CF3 CH2CH2SMe
CH(Me)S(O)CH2CH2CF3 CH2CH2S(O)Me
CH(Me)S(O)CH2CH2CF3 CH2CH2S(O)2Me
CH(Me)S(O)CH2CH2CF3 D1-32a
CH(Me)S(O)CH2CH2CF3 D1-33a
CH(Me)S(O)CH2CH2CF3 D1-34a
CH(Me)S(O)CH2CH2CF3 D1-37a
CH(Me)S(O)CH2CH2CF3 D1-81a
CH(Me)S(O)CH2CH2CF3 D1-82a
CH(Me)S(O)CH2CH2CF3 D1-84a
CH(Me)S(O)CH2CH2CF3 D1-85a
CH(Me)S(O)CH2CH2CF3 D1-87a
CH(Me)S(O)CH2CH2CF3 D1-92a
CH(Me)S(O)CH2CH2CF3 D1-93a
CH(Me)S(O)CH2CH2CF3 D1-95a
CH(Me)S(O)CH2CH2CF3 D1-96a
CH(Me)S(O)CH2CH2CF3 D1-98a
CH(Me)S(O)CH2CH2CF3 D1-108a
CH(Me)S(O)CH2CH2CF3 D1-108b(Z=2-Cl)
CH(Me)S(O)CH2CH2CF3 D1-108b(Z=3-Me)
CH(Me)S(O)CH2CH2CF3 D1-108b(Z=4-OMe)
CH(Me)S(O)CH2CH2CF3 D1-108b(Z=2-SMe)
CH(Me)S(O)CH2CH2CF3 D1-108b(Z=3-CF3)
CH(Me)S(O)CH2CH2CF3 D1-108b(Z=4-OCF3)
CH(Me)S(O)CH2CH2CF3 D1-108b(Z=2-SCF3)
CH(Me)S(O)CH2CH2CF3 C(O)Me
CH(Me)S(O)CH2CH2CF3 C(O)CF3
CH(Me)S(O)CH2CH2CF3 C(O)OMe
CH(Me)S(O)2CH2CH2CF3 Me
CH(Me)S(O)2CH2CH2CF3 Et
CH(Me)S(O)2CH2CH2CF3 Pr-n
CH(Me)S(O)2CH2CH2CF3 Pr-i
CH(Me)S(O)2CH2CH2CF3 Pr-c
CH(Me)S(O)2CH2CH2CF3 Bu-n
CH(Me)S(O)2CH2CH2CF3 Bu-i
CH(Me)S(O)2CH2CH2CF3 Bu-c
CH(Me)S(O)2CH2CH2CF3 Bu-s
CH(Me)S(O)2CH2CH2CF3 Bu-t
CH(Me)S(O)2CH2CH2CF3 Pen-n
CH(Me)S(O)2CH2CH2CF3 Pen-c
CH(Me)S(O)2CH2CH2CF3 Hex-n
CH(Me)S(O)2CH2CH2CF3 Hex-c
CH(Me)S(O)2CH2CH2CF3 CH2Pr-c
CH(Me)S(O)2CH2CH2CF3 CH2Bu-c
CH(Me)S(O)2CH2CH2CF3 CH2Pen-c
CH(Me)S(O)2CH2CH2CF3 CH2Hex-c
CH(Me)S(O)2CH2CH2CF3 CH2CH=CH2
CH(Me)S(O)2CH2CH2CF3 CH2CH=C(Cl)2
CH(Me)S(O)2CH2CH2CF3 CH2C≡CH
CH(Me)S(O)2CH2CH2CF3 CH2CN
CH(Me)S(O)2CH2CH2CF3 CH2CF3
CH(Me)S(O)2CH2CH2CF3 CH2OMe
CH(Me)S(O)2CH2CH2CF3 CH2OCF3
CH(Me)S(O)2CH2CH2CF3 CH2SMe
CH(Me)S(O)2CH2CH2CF3 CH2S(O)Me
CH(Me)S(O)2CH2CH2CF3 CH2S(O)2Me
CH(Me)S(O)2CH2CH2CF3 CH2SCF3
CH(Me)S(O)2CH2CH2CF3 CH2S(O)CF3
CH(Me)S(O)2CH2CH2CF3 CH2S(O)2CF3
CH(Me)S(O)2CH2CH2CF3 CH2CH(OMe)2
CH(Me)S(O)2CH2CH2CF3 CH2CH(SMe)2
CH(Me)S(O)2CH2CH2CF3 CH2C(O)Me
CH(Me)S(O)2CH2CH2CF3 CH2C(O)CF3
CH(Me)S(O)2CH2CH2CF3 CH2C(O)OMe
CH(Me)S(O)2CH2CH2CF3 CH2(D1-32a)
CH(Me)S(O)2CH2CH2CF3 CH2(D1-33a)
CH(Me)S(O)2CH2CH2CF3 CH2(D1-34a)
CH(Me)S(O)2CH2CH2CF3 CH2(D1-37a)
CH(Me)S(O)2CH2CH2CF3 CH2(D1-81a)
CH(Me)S(O)2CH2CH2CF3 CH2(D1-82a)
CH(Me)S(O)2CH2CH2CF3 CH2(D1-84a)
CH(Me)S(O)2CH2CH2CF3 CH2(D1-85a)
CH(Me)S(O)2CH2CH2CF3 CH2(D1-87a)
CH(Me)S(O)2CH2CH2CF3 CH2(D1-92a)
CH(Me)S(O)2CH2CH2CF3 CH2(D1-93a)
CH(Me)S(O)2CH2CH2CF3 CH2(D1-95a)
CH(Me)S(O)2CH2CH2CF3 CH2(D1-96a)
CH(Me)S(O)2CH2CH2CF3 CH2(D1-98a)
CH(Me)S(O)2CH2CH2CF3 CH2(D1-108a)
CH(Me)S(O)2CH2CH2CF3 CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)2CH2CH2CF3 CH2(D1-108b,Z=3-Me)
CH(Me)S(O)2CH2CH2CF3 CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)2CH2CH2CF3 CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)2CH2CH2CF3 CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)2CH2CH2CF3 CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)2CH2CH2CF3 CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)2CH2CH2CF3 CH2CH2CN
CH(Me)S(O)2CH2CH2CF3 CH2CH2CF3
CH(Me)S(O)2CH2CH2CF3 CH2CH2OMe
CH(Me)S(O)2CH2CH2CF3 CH2CH2SMe
CH(Me)S(O)2CH2CH2CF3 CH2CH2S(O)Me
CH(Me)S(O)2CH2CH2CF3 CH2CH2S(O)2Me
CH(Me)S(O)2CH2CH2CF3 D1-32a
CH(Me)S(O)2CH2CH2CF3 D1-33a
CH(Me)S(O)2CH2CH2CF3 D1-34a
CH(Me)S(O)2CH2CH2CF3 D1-37a
CH(Me)S(O)2CH2CH2CF3 D1-81a
CH(Me)S(O)2CH2CH2CF3 D1-82a
CH(Me)S(O)2CH2CH2CF3 D1-84a
CH(Me)S(O)2CH2CH2CF3 D1-85a
CH(Me)S(O)2CH2CH2CF3 D1-87a
CH(Me)S(O)2CH2CH2CF3 D1-92a
CH(Me)S(O)2CH2CH2CF3 D1-93a
CH(Me)S(O)2CH2CH2CF3 D1-95a
CH(Me)S(O)2CH2CH2CF3 D1-96a
CH(Me)S(O)2CH2CH2CF3 D1-98a
CH(Me)S(O)2CH2CH2CF3 D1-108a
CH(Me)S(O)2CH2CH2CF3 D1-108b(Z=2-Cl)
CH(Me)S(O)2CH2CH2CF3 D1-108b(Z=3-Me)
CH(Me)S(O)2CH2CH2CF3 D1-108b(Z=4-OMe)
CH(Me)S(O)2CH2CH2CF3 D1-108b(Z=2-SMe)
CH(Me)S(O)2CH2CH2CF3 D1-108b(Z=3-CF3)
CH(Me)S(O)2CH2CH2CF3 D1-108b(Z=4-OCF3)
CH(Me)S(O)2CH2CH2CF3 D1-108b(Z=2-SCF3)
CH(Me)S(O)2CH2CH2CF3 C(O)Me
CH(Me)S(O)2CH2CH2CF3 C(O)CF3
CH(Me)S(O)2CH2CH2CF3 C(O)OMe
CH(Et)SCH2CH2CF3 Me
CH(Et)SCH2CH2CF3 Et
CH(Et)SCH2CH2CF3 Pr-n
CH(Et)SCH2CH2CF3 Pr-i
CH(Et)SCH2CH2CF3 Pr-c
CH(Et)SCH2CH2CF3 Bu-n
CH(Et)SCH2CH2CF3 Bu-i
CH(Et)SCH2CH2CF3 Bu-c
CH(Et)SCH2CH2CF3 Bu-s
CH(Et)SCH2CH2CF3 Bu-t
CH(Et)SCH2CH2CF3 Pen-n
CH(Et)SCH2CH2CF3 Pen-c
CH(Et)SCH2CH2CF3 Hex-n
CH(Et)SCH2CH2CF3 Hex-c
CH(Et)SCH2CH2CF3 CH2Pr-c
CH(Et)SCH2CH2CF3 CH2Bu-c
CH(Et)SCH2CH2CF3 CH2Pen-c
CH(Et)SCH2CH2CF3 CH2Hex-c
CH(Et)SCH2CH2CF3 CH2CH=CH2
CH(Et)SCH2CH2CF3 CH2CH=C(Cl)2
CH(Et)SCH2CH2CF3 CH2C≡CH
CH(Et)SCH2CH2CF3 CH2CN
CH(Et)SCH2CH2CF3 CH2CF3
CH(Et)SCH2CH2CF3 CH2OMe
CH(Et)SCH2CH2CF3 CH2OCF3
CH(Et)SCH2CH2CF3 CH2SMe
CH(Et)SCH2CH2CF3 CH2S(O)Me
CH(Et)SCH2CH2CF3 CH2S(O)2Me
CH(Et)SCH2CH2CF3 CH2SCF3
CH(Et)SCH2CH2CF3 CH2S(O)CF3
CH(Et)SCH2CH2CF3 CH2S(O)2CF3
CH(Et)SCH2CH2CF3 CH2CH(OMe)2
CH(Et)SCH2CH2CF3 CH2CH(SMe)2
CH(Et)SCH2CH2CF3 CH2C(O)Me
CH(Et)SCH2CH2CF3 CH2C(O)CF3
CH(Et)SCH2CH2CF3 CH2C(O)OMe
CH(Et)SCH2CH2CF3 CH2(D1-32a)
CH(Et)SCH2CH2CF3 CH2(D1-33a)
CH(Et)SCH2CH2CF3 CH2(D1-34a)
CH(Et)SCH2CH2CF3 CH2(D1-37a)
CH(Et)SCH2CH2CF3 CH2(D1-81a)
CH(Et)SCH2CH2CF3 CH2(D1-82a)
CH(Et)SCH2CH2CF3 CH2(D1-84a)
CH(Et)SCH2CH2CF3 CH2(D1-85a)
CH(Et)SCH2CH2CF3 CH2(D1-87a)
CH(Et)SCH2CH2CF3 CH2(D1-92a)
CH(Et)SCH2CH2CF3 CH2(D1-93a)
CH(Et)SCH2CH2CF3 CH2(D1-95a)
CH(Et)SCH2CH2CF3 CH2(D1-96a)
CH(Et)SCH2CH2CF3 CH2(D1-98a)
CH(Et)SCH2CH2CF3 CH2(D1-108a)
CH(Et)SCH2CH2CF3 CH2(D1-108b,Z=2-Cl)
CH(Et)SCH2CH2CF3 CH2(D1-108b,Z=3-Me)
CH(Et)SCH2CH2CF3 CH2(D1-108b,Z=4-OMe)
CH(Et)SCH2CH2CF3 CH2(D1-108b,Z=2-SMe)
CH(Et)SCH2CH2CF3 CH2(D1-108b,Z=3-CF3)
CH(Et)SCH2CH2CF3 CH2(D1-108b,Z=4-OCF3)
CH(Et)SCH2CH2CF3 CH2(D1-108b,Z=2-SCF3)
CH(Et)SCH2CH2CF3 CH2CH2CN
CH(Et)SCH2CH2CF3 CH2CH2CF3
CH(Et)SCH2CH2CF3 CH2CH2OMe
CH(Et)SCH2CH2CF3 CH2CH2SMe
CH(Et)SCH2CH2CF3 CH2CH2S(O)Me
CH(Et)SCH2CH2CF3 CH2CH2S(O)2Me
CH(Et)SCH2CH2CF3 D1-32a
CH(Et)SCH2CH2CF3 D1-33a
CH(Et)SCH2CH2CF3 D1-34a
CH(Et)SCH2CH2CF3 D1-37a
CH(Et)SCH2CH2CF3 D1-81a
CH(Et)SCH2CH2CF3 D1-82a
CH(Et)SCH2CH2CF3 D1-84a
CH(Et)SCH2CH2CF3 D1-85a
CH(Et)SCH2CH2CF3 D1-87a
CH(Et)SCH2CH2CF3 D1-92a
CH(Et)SCH2CH2CF3 D1-93a
CH(Et)SCH2CH2CF3 D1-95a
CH(Et)SCH2CH2CF3 D1-96a
CH(Et)SCH2CH2CF3 D1-98a
CH(Et)SCH2CH2CF3 D1-108a
CH(Et)SCH2CH2CF3 D1-108b(Z=2-Cl)
CH(Et)SCH2CH2CF3 D1-108b(Z=3-Me)
CH(Et)SCH2CH2CF3 D1-108b(Z=4-OMe)
CH(Et)SCH2CH2CF3 D1-108b(Z=2-SMe)
CH(Et)SCH2CH2CF3 D1-108b(Z=3-CF3)
CH(Et)SCH2CH2CF3 D1-108b(Z=4-OCF3)
CH(Et)SCH2CH2CF3 D1-108b(Z=2-SCF3)
CH(Et)SCH2CH2CF3 C(O)Me
CH(Et)SCH2CH2CF3 C(O)CF3
CH(Et)SCH2CH2CF3 C(O)OMe
CH(Et)S(O)CH2CH2CF3 Me
CH(Et)S(O)CH2CH2CF3 Et
CH(Et)S(O)CH2CH2CF3 Pr-n
CH(Et)S(O)CH2CH2CF3 Pr-i
CH(Et)S(O)CH2CH2CF3 Pr-c
CH(Et)S(O)CH2CH2CF3 Bu-n
CH(Et)S(O)CH2CH2CF3 Bu-i
CH(Et)S(O)CH2CH2CF3 Bu-c
CH(Et)S(O)CH2CH2CF3 Bu-s
CH(Et)S(O)CH2CH2CF3 Bu-t
CH(Et)S(O)CH2CH2CF3 Pen-n
CH(Et)S(O)CH2CH2CF3 Pen-c
CH(Et)S(O)CH2CH2CF3 Hex-n
CH(Et)S(O)CH2CH2CF3 Hex-c
CH(Et)S(O)CH2CH2CF3 CH2Pr-c
CH(Et)S(O)CH2CH2CF3 CH2Bu-c
CH(Et)S(O)CH2CH2CF3 CH2Pen-c
CH(Et)S(O)CH2CH2CF3 CH2Hex-c
CH(Et)S(O)CH2CH2CF3 CH2CH=CH2
CH(Et)S(O)CH2CH2CF3 CH2CH=C(Cl)2
CH(Et)S(O)CH2CH2CF3 CH2C≡CH
CH(Et)S(O)CH2CH2CF3 CH2CN
CH(Et)S(O)CH2CH2CF3 CH2CF3
CH(Et)S(O)CH2CH2CF3 CH2OMe
CH(Et)S(O)CH2CH2CF3 CH2OCF3
CH(Et)S(O)CH2CH2CF3 CH2SMe
CH(Et)S(O)CH2CH2CF3 CH2S(O)Me
CH(Et)S(O)CH2CH2CF3 CH2S(O)2Me
CH(Et)S(O)CH2CH2CF3 CH2SCF3
CH(Et)S(O)CH2CH2CF3 CH2S(O)CF3
CH(Et)S(O)CH2CH2CF3 CH2S(O)2CF3
CH(Et)S(O)CH2CH2CF3 CH2CH(OMe)2
CH(Et)S(O)CH2CH2CF3 CH2CH(SMe)2
CH(Et)S(O)CH2CH2CF3 CH2C(O)Me
CH(Et)S(O)CH2CH2CF3 CH2C(O)CF3
CH(Et)S(O)CH2CH2CF3 CH2C(O)OMe
CH(Et)S(O)CH2CH2CF3 CH2(D1-32a)
CH(Et)S(O)CH2CH2CF3 CH2(D1-33a)
CH(Et)S(O)CH2CH2CF3 CH2(D1-34a)
CH(Et)S(O)CH2CH2CF3 CH2(D1-37a)
CH(Et)S(O)CH2CH2CF3 CH2(D1-81a)
CH(Et)S(O)CH2CH2CF3 CH2(D1-82a)
CH(Et)S(O)CH2CH2CF3 CH2(D1-84a)
CH(Et)S(O)CH2CH2CF3 CH2(D1-85a)
CH(Et)S(O)CH2CH2CF3 CH2(D1-87a)
CH(Et)S(O)CH2CH2CF3 CH2(D1-92a)
CH(Et)S(O)CH2CH2CF3 CH2(D1-93a)
CH(Et)S(O)CH2CH2CF3 CH2(D1-95a)
CH(Et)S(O)CH2CH2CF3 CH2(D1-96a)
CH(Et)S(O)CH2CH2CF3 CH2(D1-98a)
CH(Et)S(O)CH2CH2CF3 CH2(D1-108a)
CH(Et)S(O)CH2CH2CF3 CH2(D1-108b,Z=2-Cl)
CH(Et)S(O)CH2CH2CF3 CH2(D1-108b,Z=3-Me)
CH(Et)S(O)CH2CH2CF3 CH2(D1-108b,Z=4-OMe)
CH(Et)S(O)CH2CH2CF3 CH2(D1-108b,Z=2-SMe)
CH(Et)S(O)CH2CH2CF3 CH2(D1-108b,Z=3-CF3)
CH(Et)S(O)CH2CH2CF3 CH2(D1-108b,Z=4-OCF3)
CH(Et)S(O)CH2CH2CF3 CH2(D1-108b,Z=2-SCF3)
CH(Et)S(O)CH2CH2CF3 CH2CH2CN
CH(Et)S(O)CH2CH2CF3 CH2CH2CF3
CH(Et)S(O)CH2CH2CF3 CH2CH2OMe
CH(Et)S(O)CH2CH2CF3 CH2CH2SMe
CH(Et)S(O)CH2CH2CF3 CH2CH2S(O)Me
CH(Et)S(O)CH2CH2CF3 CH2CH2S(O)2Me
CH(Et)S(O)CH2CH2CF3 D1-32a
CH(Et)S(O)CH2CH2CF3 D1-33a
CH(Et)S(O)CH2CH2CF3 D1-34a
CH(Et)S(O)CH2CH2CF3 D1-37a
CH(Et)S(O)CH2CH2CF3 D1-81a
CH(Et)S(O)CH2CH2CF3 D1-82a
CH(Et)S(O)CH2CH2CF3 D1-84a
CH(Et)S(O)CH2CH2CF3 D1-85a
CH(Et)S(O)CH2CH2CF3 D1-87a
CH(Et)S(O)CH2CH2CF3 D1-92a
CH(Et)S(O)CH2CH2CF3 D1-93a
CH(Et)S(O)CH2CH2CF3 D1-95a
CH(Et)S(O)CH2CH2CF3 D1-96a
CH(Et)S(O)CH2CH2CF3 D1-98a
CH(Et)S(O)CH2CH2CF3 D1-108a
CH(Et)S(O)CH2CH2CF3 D1-108b(Z=2-Cl)
CH(Et)S(O)CH2CH2CF3 D1-108b(Z=3-Me)
CH(Et)S(O)CH2CH2CF3 D1-108b(Z=4-OMe)
CH(Et)S(O)CH2CH2CF3 D1-108b(Z=2-SMe)
CH(Et)S(O)CH2CH2CF3 D1-108b(Z=3-CF3)
CH(Et)S(O)CH2CH2CF3 D1-108b(Z=4-OCF3)
CH(Et)S(O)CH2CH2CF3 D1-108b(Z=2-SCF3)
CH(Et)S(O)CH2CH2CF3 C(O)Me
CH(Et)S(O)CH2CH2CF3 C(O)CF3
CH(Et)S(O)CH2CH2CF3 C(O)OMe
CH(Et)S(O)2CH2CH2CF3 Me
CH(Et)S(O)2CH2CH2CF3 Et
CH(Et)S(O)2CH2CH2CF3 Pr-n
CH(Et)S(O)2CH2CH2CF3 Pr-i
CH(Et)S(O)2CH2CH2CF3 Pr-c
CH(Et)S(O)2CH2CH2CF3 Bu-n
CH(Et)S(O)2CH2CH2CF3 Bu-i
CH(Et)S(O)2CH2CH2CF3 Bu-c
CH(Et)S(O)2CH2CH2CF3 Bu-s
CH(Et)S(O)2CH2CH2CF3 Bu-t
CH(Et)S(O)2CH2CH2CF3 Pen-n
CH(Et)S(O)2CH2CH2CF3 Pen-c
CH(Et)S(O)2CH2CH2CF3 Hex-n
CH(Et)S(O)2CH2CH2CF3 Hex-c
CH(Et)S(O)2CH2CH2CF3 CH2Pr-c
CH(Et)S(O)2CH2CH2CF3 CH2Bu-c
CH(Et)S(O)2CH2CH2CF3 CH2Pen-c
CH(Et)S(O)2CH2CH2CF3 CH2Hex-c
CH(Et)S(O)2CH2CH2CF3 CH2CH=CH2
CH(Et)S(O)2CH2CH2CF3 CH2CH=C(Cl)2
CH(Et)S(O)2CH2CH2CF3 CH2C≡CH
CH(Et)S(O)2CH2CH2CF3 CH2CN
CH(Et)S(O)2CH2CH2CF3 CH2CF3
CH(Et)S(O)2CH2CH2CF3 CH2OMe
CH(Et)S(O)2CH2CH2CF3 CH2OCF3
CH(Et)S(O)2CH2CH2CF3 CH2SMe
CH(Et)S(O)2CH2CH2CF3 CH2S(O)Me
CH(Et)S(O)2CH2CH2CF3 CH2S(O)2Me
CH(Et)S(O)2CH2CH2CF3 CH2SCF3
CH(Et)S(O)2CH2CH2CF3 CH2S(O)CF3
CH(Et)S(O)2CH2CH2CF3 CH2S(O)2CF3
CH(Et)S(O)2CH2CH2CF3 CH2CH(OMe)2
CH(Et)S(O)2CH2CH2CF3 CH2CH(SMe)2
CH(Et)S(O)2CH2CH2CF3 CH2C(O)Me
CH(Et)S(O)2CH2CH2CF3 CH2C(O)CF3
CH(Et)S(O)2CH2CH2CF3 CH2C(O)OMe
CH(Et)S(O)2CH2CH2CF3 CH2(D1-32a)
CH(Et)S(O)2CH2CH2CF3 CH2(D1-33a)
CH(Et)S(O)2CH2CH2CF3 CH2(D1-34a)
CH(Et)S(O)2CH2CH2CF3 CH2(D1-37a)
CH(Et)S(O)2CH2CH2CF3 CH2(D1-81a)
CH(Et)S(O)2CH2CH2CF3 CH2(D1-82a)
CH(Et)S(O)2CH2CH2CF3 CH2(D1-84a)
CH(Et)S(O)2CH2CH2CF3 CH2(D1-85a)
CH(Et)S(O)2CH2CH2CF3 CH2(D1-87a)
CH(Et)S(O)2CH2CH2CF3 CH2(D1-92a)
CH(Et)S(O)2CH2CH2CF3 CH2(D1-93a)
CH(Et)S(O)2CH2CH2CF3 CH2(D1-95a)
CH(Et)S(O)2CH2CH2CF3 CH2(D1-96a)
CH(Et)S(O)2CH2CH2CF3 CH2(D1-98a)
CH(Et)S(O)2CH2CH2CF3 CH2(D1-108a)
CH(Et)S(O)2CH2CH2CF3 CH2(D1-108b,Z=2-Cl)
CH(Et)S(O)2CH2CH2CF3 CH2(D1-108b,Z=3-Me)
CH(Et)S(O)2CH2CH2CF3 CH2(D1-108b,Z=4-OMe)
CH(Et)S(O)2CH2CH2CF3 CH2(D1-108b,Z=2-SMe)
CH(Et)S(O)2CH2CH2CF3 CH2(D1-108b,Z=3-CF3)
CH(Et)S(O)2CH2CH2CF3 CH2(D1-108b,Z=4-OCF3)
CH(Et)S(O)2CH2CH2CF3 CH2(D1-108b,Z=2-SCF3)
CH(Et)S(O)2CH2CH2CF3 CH2CH2CN
CH(Et)S(O)2CH2CH2CF3 CH2CH2CF3
CH(Et)S(O)2CH2CH2CF3 CH2CH2OMe
CH(Et)S(O)2CH2CH2CF3 CH2CH2SMe
CH(Et)S(O)2CH2CH2CF3 CH2CH2S(O)Me
CH(Et)S(O)2CH2CH2CF3 CH2CH2S(O)2Me
CH(Et)S(O)2CH2CH2CF3 D1-32a
CH(Et)S(O)2CH2CH2CF3 D1-33a
CH(Et)S(O)2CH2CH2CF3 D1-34a
CH(Et)S(O)2CH2CH2CF3 D1-37a
CH(Et)S(O)2CH2CH2CF3 D1-81a
CH(Et)S(O)2CH2CH2CF3 D1-82a
CH(Et)S(O)2CH2CH2CF3 D1-84a
CH(Et)S(O)2CH2CH2CF3 D1-85a
CH(Et)S(O)2CH2CH2CF3 D1-87a
CH(Et)S(O)2CH2CH2CF3 D1-92a
CH(Et)S(O)2CH2CH2CF3 D1-93a
CH(Et)S(O)2CH2CH2CF3 D1-95a
CH(Et)S(O)2CH2CH2CF3 D1-96a
CH(Et)S(O)2CH2CH2CF3 D1-98a
CH(Et)S(O)2CH2CH2CF3 D1-108a
CH(Et)S(O)2CH2CH2CF3 D1-108b(Z=2-Cl)
CH(Et)S(O)2CH2CH2CF3 D1-108b(Z=3-Me)
CH(Et)S(O)2CH2CH2CF3 D1-108b(Z=4-OMe)
CH(Et)S(O)2CH2CH2CF3 D1-108b(Z=2-SMe)
CH(Et)S(O)2CH2CH2CF3 D1-108b(Z=3-CF3)
CH(Et)S(O)2CH2CH2CF3 D1-108b(Z=4-OCF3)
CH(Et)S(O)2CH2CH2CF3 D1-108b(Z=2-SCF3)
CH(Et)S(O)2CH2CH2CF3 C(O)Me
CH(Et)S(O)2CH2CH2CF3 C(O)CF3
CH(Et)S(O)2CH2CH2CF3 C(O)OMe
CH2SCH2(D1-103a) Me
CH2SCH2(D1-103a) Et
CH2SCH2(D1-103a) Pr-n
CH2SCH2(D1-103a) Pr-i
CH2SCH2(D1-103a) Pr-c
CH2SCH2(D1-103a) Bu-n
CH2SCH2(D1-103a) Bu-i
CH2SCH2(D1-103a) Bu-c
CH2SCH2(D1-103a) Bu-s
CH2SCH2(D1-103a) Bu-t
CH2SCH2(D1-103a) Pen-n
CH2SCH2(D1-103a) Pen-c
CH2SCH2(D1-103a) Hex-n
CH2SCH2(D1-103a) Hex-c
CH2SCH2(D1-103a) CH2Pr-c
CH2SCH2(D1-103a) CH2Bu-c
CH2SCH2(D1-103a) CH2Pen-c
CH2SCH2(D1-103a) CH2Hex-c
CH2SCH2(D1-103a) CH2CH=CH2
CH2SCH2(D1-103a) CH2CH=C(Cl)2
CH2SCH2(D1-103a) CH2C≡CH
CH2SCH2(D1-103a) CH2CN
CH2SCH2(D1-103a) CH2CF3
CH2SCH2(D1-103a) CH2OMe
CH2SCH2(D1-103a) CH2OCF3
CH2SCH2(D1-103a) CH2SMe
CH2SCH2(D1-103a) CH2S(O)Me
CH2SCH2(D1-103a) CH2S(O)2Me
CH2SCH2(D1-103a) CH2SCF3
CH2SCH2(D1-103a) CH2S(O)CF3
CH2SCH2(D1-103a) CH2S(O)2CF3
CH2SCH2(D1-103a) CH2CH(OMe)2
CH2SCH2(D1-103a) CH2CH(SMe)2
CH2SCH2(D1-103a) CH2C(O)Me
CH2SCH2(D1-103a) CH2C(O)CF3
CH2SCH2(D1-103a) CH2C(O)OMe
CH2SCH2(D1-103a) CH2(D1-32a)
CH2SCH2(D1-103a) CH2(D1-33a)
CH2SCH2(D1-103a) CH2(D1-34a)
CH2SCH2(D1-103a) CH2(D1-37a)
CH2SCH2(D1-103a) CH2(D1-81a)
CH2SCH2(D1-103a) CH2(D1-82a)
CH2SCH2(D1-103a) CH2(D1-84a)
CH2SCH2(D1-103a) CH2(D1-85a)
CH2SCH2(D1-103a) CH2(D1-87a)
CH2SCH2(D1-103a) CH2(D1-92a)
CH2SCH2(D1-103a) CH2(D1-93a)
CH2SCH2(D1-103a) CH2(D1-95a)
CH2SCH2(D1-103a) CH2(D1-96a)
CH2SCH2(D1-103a) CH2(D1-98a)
CH2SCH2(D1-103a) CH2(D1-108a)
CH2SCH2(D1-103a) CH2(D1-108b,Z=2-Cl)
CH2SCH2(D1-103a) CH2(D1-108b,Z=3-Me)
CH2SCH2(D1-103a) CH2(D1-108b,Z=4-OMe)
CH2SCH2(D1-103a) CH2(D1-108b,Z=2-SMe)
CH2SCH2(D1-103a) CH2(D1-108b,Z=3-CF3)
CH2SCH2(D1-103a) CH2(D1-108b,Z=4-OCF3)
CH2SCH2(D1-103a) CH2(D1-108b,Z=2-SCF3)
CH2SCH2(D1-103a) CH2CH2CN
CH2SCH2(D1-103a) CH2CH2CF3
CH2SCH2(D1-103a) CH2CH2OMe
CH2SCH2(D1-103a) CH2CH2SMe
CH2SCH2(D1-103a) CH2CH2S(O)Me
CH2SCH2(D1-103a) CH2CH2S(O)2Me
CH2SCH2(D1-103a) D1-32a
CH2SCH2(D1-103a) D1-33a
CH2SCH2(D1-103a) D1-34a
CH2SCH2(D1-103a) D1-37a
CH2SCH2(D1-103a) D1-81a
CH2SCH2(D1-103a) D1-82a
CH2SCH2(D1-103a) D1-84a
CH2SCH2(D1-103a) D1-85a
CH2SCH2(D1-103a) D1-87a
CH2SCH2(D1-103a) D1-92a
CH2SCH2(D1-103a) D1-93a
CH2SCH2(D1-103a) D1-95a
CH2SCH2(D1-103a) D1-96a
CH2SCH2(D1-103a) D1-98a
CH2SCH2(D1-103a) D1-108a
CH2SCH2(D1-103a) D1-108b(Z=2-Cl)
CH2SCH2(D1-103a) D1-108b(Z=3-Me)
CH2SCH2(D1-103a) D1-108b(Z=4-OMe)
CH2SCH2(D1-103a) D1-108b(Z=2-SMe)
CH2SCH2(D1-103a) D1-108b(Z=3-CF3)
CH2SCH2(D1-103a) D1-108b(Z=4-OCF3)
CH2SCH2(D1-103a) D1-108b(Z=2-SCF3)
CH2SCH2(D1-103a) C(O)Me
CH2SCH2(D1-103a) C(O)CF3
CH2SCH2(D1-103a) C(O)OMe
CH2S(O)CH2(D1-103a) Me
CH2S(O)CH2(D1-103a) Et
CH2S(O)CH2(D1-103a) Pr-n
CH2S(O)CH2(D1-103a) Pr-i
CH2S(O)CH2(D1-103a) Pr-c
CH2S(O)CH2(D1-103a) Bu-n
CH2S(O)CH2(D1-103a) Bu-i
CH2S(O)CH2(D1-103a) Bu-c
CH2S(O)CH2(D1-103a) Bu-s
CH2S(O)CH2(D1-103a) Bu-t
CH2S(O)CH2(D1-103a) Pen-n
CH2S(O)CH2(D1-103a) Pen-c
CH2S(O)CH2(D1-103a) Hex-n
CH2S(O)CH2(D1-103a) Hex-c
CH2S(O)CH2(D1-103a) CH2Pr-c
CH2S(O)CH2(D1-103a) CH2Bu-c
CH2S(O)CH2(D1-103a) CH2Pen-c
CH2S(O)CH2(D1-103a) CH2Hex-c
CH2S(O)CH2(D1-103a) CH2CH=CH2
CH2S(O)CH2(D1-103a) CH2CH=C(Cl)2
CH2S(O)CH2(D1-103a) CH2C≡CH
CH2S(O)CH2(D1-103a) CH2CN
CH2S(O)CH2(D1-103a) CH2CF3
CH2S(O)CH2(D1-103a) CH2OMe
CH2S(O)CH2(D1-103a) CH2OCF3
CH2S(O)CH2(D1-103a) CH2SMe
CH2S(O)CH2(D1-103a) CH2S(O)Me
CH2S(O)CH2(D1-103a) CH2S(O)2Me
CH2S(O)CH2(D1-103a) CH2SCF3
CH2S(O)CH2(D1-103a) CH2S(O)CF3
CH2S(O)CH2(D1-103a) CH2S(O)2CF3
CH2S(O)CH2(D1-103a) CH2CH(OMe)2
CH2S(O)CH2(D1-103a) CH2CH(SMe)2
CH2S(O)CH2(D1-103a) CH2C(O)Me
CH2S(O)CH2(D1-103a) CH2C(O)CF3
CH2S(O)CH2(D1-103a) CH2C(O)OMe
CH2S(O)CH2(D1-103a) CH2(D1-32a)
CH2S(O)CH2(D1-103a) CH2(D1-33a)
CH2S(O)CH2(D1-103a) CH2(D1-34a)
CH2S(O)CH2(D1-103a) CH2(D1-37a)
CH2S(O)CH2(D1-103a) CH2(D1-81a)
CH2S(O)CH2(D1-103a) CH2(D1-82a)
CH2S(O)CH2(D1-103a) CH2(D1-84a)
CH2S(O)CH2(D1-103a) CH2(D1-85a)
CH2S(O)CH2(D1-103a) CH2(D1-87a)
CH2S(O)CH2(D1-103a) CH2(D1-92a)
CH2S(O)CH2(D1-103a) CH2(D1-93a)
CH2S(O)CH2(D1-103a) CH2(D1-95a)
CH2S(O)CH2(D1-103a) CH2(D1-96a)
CH2S(O)CH2(D1-103a) CH2(D1-98a)
CH2S(O)CH2(D1-103a) CH2(D1-108a)
CH2S(O)CH2(D1-103a) CH2(D1-108b,Z=2-Cl)
CH2S(O)CH2(D1-103a) CH2(D1-108b,Z=3-Me)
CH2S(O)CH2(D1-103a) CH2(D1-108b,Z=4-OMe)
CH2S(O)CH2(D1-103a) CH2(D1-108b,Z=2-SMe)
CH2S(O)CH2(D1-103a) CH2(D1-108b,Z=3-CF3)
CH2S(O)CH2(D1-103a) CH2(D1-108b,Z=4-OCF3)
CH2S(O)CH2(D1-103a) CH2(D1-108b,Z=2-SCF3)
CH2S(O)CH2(D1-103a) CH2CH2CN
CH2S(O)CH2(D1-103a) CH2CH2CF3
CH2S(O)CH2(D1-103a) CH2CH2OMe
CH2S(O)CH2(D1-103a) CH2CH2SMe
CH2S(O)CH2(D1-103a) CH2CH2S(O)Me
CH2S(O)CH2(D1-103a) CH2CH2S(O)2Me
CH2S(O)CH2(D1-103a) D1-32a
CH2S(O)CH2(D1-103a) D1-33a
CH2S(O)CH2(D1-103a) D1-34a
CH2S(O)CH2(D1-103a) D1-37a
CH2S(O)CH2(D1-103a) D1-81a
CH2S(O)CH2(D1-103a) D1-82a
CH2S(O)CH2(D1-103a) D1-84a
CH2S(O)CH2(D1-103a) D1-85a
CH2S(O)CH2(D1-103a) D1-87a
CH2S(O)CH2(D1-103a) D1-92a
CH2S(O)CH2(D1-103a) D1-93a
CH2S(O)CH2(D1-103a) D1-95a
CH2S(O)CH2(D1-103a) D1-96a
CH2S(O)CH2(D1-103a) D1-98a
CH2S(O)CH2(D1-103a) D1-108a
CH2S(O)CH2(D1-103a) D1-108b(Z=2-Cl)
CH2S(O)CH2(D1-103a) D1-108b(Z=3-Me)
CH2S(O)CH2(D1-103a) D1-108b(Z=4-OMe)
CH2S(O)CH2(D1-103a) D1-108b(Z=2-SMe)
CH2S(O)CH2(D1-103a) D1-108b(Z=3-CF3)
CH2S(O)CH2(D1-103a) D1-108b(Z=4-OCF3)
CH2S(O)CH2(D1-103a) D1-108b(Z=2-SCF3)
CH2S(O)CH2(D1-103a) C(O)Me
CH2S(O)CH2(D1-103a) C(O)CF3
CH2S(O)CH2(D1-103a) C(O)OMe
CH2S(O)2CH2(D1-103a) Me
CH2S(O)2CH2(D1-103a) Et
CH2S(O)2CH2(D1-103a) Pr-n
CH2S(O)2CH2(D1-103a) Pr-i
CH2S(O)2CH2(D1-103a) Pr-c
CH2S(O)2CH2(D1-103a) Bu-n
CH2S(O)2CH2(D1-103a) Bu-i
CH2S(O)2CH2(D1-103a) Bu-c
CH2S(O)2CH2(D1-103a) Bu-s
CH2S(O)2CH2(D1-103a) Bu-t
CH2S(O)2CH2(D1-103a) Pen-n
CH2S(O)2CH2(D1-103a) Pen-c
CH2S(O)2CH2(D1-103a) Hex-n
CH2S(O)2CH2(D1-103a) Hex-c
CH2S(O)2CH2(D1-103a) CH2Pr-c
CH2S(O)2CH2(D1-103a) CH2Bu-c
CH2S(O)2CH2(D1-103a) CH2Pen-c
CH2S(O)2CH2(D1-103a) CH2Hex-c
CH2S(O)2CH2(D1-103a) CH2CH=CH2
CH2S(O)2CH2(D1-103a) CH2CH=C(Cl)2
CH2S(O)2CH2(D1-103a) CH2C≡CH
CH2S(O)2CH2(D1-103a) CH2CN
CH2S(O)2CH2(D1-103a) CH2CF3
CH2S(O)2CH2(D1-103a) CH2OMe
CH2S(O)2CH2(D1-103a) CH2OCF3
CH2S(O)2CH2(D1-103a) CH2SMe
CH2S(O)2CH2(D1-103a) CH2S(O)Me
CH2S(O)2CH2(D1-103a) CH2S(O)2Me
CH2S(O)2CH2(D1-103a) CH2SCF3
CH2S(O)2CH2(D1-103a) CH2S(O)CF3
CH2S(O)2CH2(D1-103a) CH2S(O)2CF3
CH2S(O)2CH2(D1-103a) CH2CH(OMe)2
CH2S(O)2CH2(D1-103a) CH2CH(SMe)2
CH2S(O)2CH2(D1-103a) CH2C(O)Me
CH2S(O)2CH2(D1-103a) CH2C(O)CF3
CH2S(O)2CH2(D1-103a) CH2C(O)OMe
CH2S(O)2CH2(D1-103a) CH2(D1-32a)
CH2S(O)2CH2(D1-103a) CH2(D1-33a)
CH2S(O)2CH2(D1-103a) CH2(D1-34a)
CH2S(O)2CH2(D1-103a) CH2(D1-37a)
CH2S(O)2CH2(D1-103a) CH2(D1-81a)
CH2S(O)2CH2(D1-103a) CH2(D1-82a)
CH2S(O)2CH2(D1-103a) CH2(D1-84a)
CH2S(O)2CH2(D1-103a) CH2(D1-85a)
CH2S(O)2CH2(D1-103a) CH2(D1-87a)
CH2S(O)2CH2(D1-103a) CH2(D1-92a)
CH2S(O)2CH2(D1-103a) CH2(D1-93a)
CH2S(O)2CH2(D1-103a) CH2(D1-95a)
CH2S(O)2CH2(D1-103a) CH2(D1-96a)
CH2S(O)2CH2(D1-103a) CH2(D1-98a)
CH2S(O)2CH2(D1-103a) CH2(D1-108a)
CH2S(O)2CH2(D1-103a) CH2(D1-108b,Z=2-Cl)
CH2S(O)2CH2(D1-103a) CH2(D1-108b,Z=3-Me)
CH2S(O)2CH2(D1-103a) CH2(D1-108b,Z=4-OMe)
CH2S(O)2CH2(D1-103a) CH2(D1-108b,Z=2-SMe)
CH2S(O)2CH2(D1-103a) CH2(D1-108b,Z=3-CF3)
CH2S(O)2CH2(D1-103a) CH2(D1-108b,Z=4-OCF3)
CH2S(O)2CH2(D1-103a) CH2(D1-108b,Z=2-SCF3)
CH2S(O)2CH2(D1-103a) CH2CH2CN
CH2S(O)2CH2(D1-103a) CH2CH2CF3
CH2S(O)2CH2(D1-103a) CH2CH2OMe
CH2S(O)2CH2(D1-103a) CH2CH2SMe
CH2S(O)2CH2(D1-103a) CH2CH2S(O)Me
CH2S(O)2CH2(D1-103a) CH2CH2S(O)2Me
CH2S(O)2CH2(D1-103a) D1-32a
CH2S(O)2CH2(D1-103a) D1-33a
CH2S(O)2CH2(D1-103a) D1-34a
CH2S(O)2CH2(D1-103a) D1-37a
CH2S(O)2CH2(D1-103a) D1-81a
CH2S(O)2CH2(D1-103a) D1-82a
CH2S(O)2CH2(D1-103a) D1-84a
CH2S(O)2CH2(D1-103a) D1-85a
CH2S(O)2CH2(D1-103a) D1-87a
CH2S(O)2CH2(D1-103a) D1-92a
CH2S(O)2CH2(D1-103a) D1-93a
CH2S(O)2CH2(D1-103a) D1-95a
CH2S(O)2CH2(D1-103a) D1-96a
CH2S(O)2CH2(D1-103a) D1-98a
CH2S(O)2CH2(D1-103a) D1-108a
CH2S(O)2CH2(D1-103a) D1-108b(Z=2-Cl)
CH2S(O)2CH2(D1-103a) D1-108b(Z=3-Me)
CH2S(O)2CH2(D1-103a) D1-108b(Z=4-OMe)
CH2S(O)2CH2(D1-103a) D1-108b(Z=2-SMe)
CH2S(O)2CH2(D1-103a) D1-108b(Z=3-CF3)
CH2S(O)2CH2(D1-103a) D1-108b(Z=4-OCF3)
CH2S(O)2CH2(D1-103a) D1-108b(Z=2-SCF3)
CH2S(O)2CH2(D1-103a) C(O)Me
CH2S(O)2CH2(D1-103a) C(O)CF3
CH2S(O)2CH2(D1-103a) C(O)OMe
CH(Me)SCH2(D1-103a) Me
CH(Me)SCH2(D1-103a) Et
CH(Me)SCH2(D1-103a) Pr-n
CH(Me)SCH2(D1-103a) Pr-i
CH(Me)SCH2(D1-103a) Pr-c
CH(Me)SCH2(D1-103a) Bu-n
CH(Me)SCH2(D1-103a) Bu-i
CH(Me)SCH2(D1-103a) Bu-c
CH(Me)SCH2(D1-103a) Bu-s
CH(Me)SCH2(D1-103a) Bu-t
CH(Me)SCH2(D1-103a) Pen-n
CH(Me)SCH2(D1-103a) Pen-c
CH(Me)SCH2(D1-103a) Hex-n
CH(Me)SCH2(D1-103a) Hex-c
CH(Me)SCH2(D1-103a) CH2Pr-c
CH(Me)SCH2(D1-103a) CH2Bu-c
CH(Me)SCH2(D1-103a) CH2Pen-c
CH(Me)SCH2(D1-103a) CH2Hex-c
CH(Me)SCH2(D1-103a) CH2CH=CH2
CH(Me)SCH2(D1-103a) CH2CH=C(Cl)2
CH(Me)SCH2(D1-103a) CH2C≡CH
CH(Me)SCH2(D1-103a) CH2CN
CH(Me)SCH2(D1-103a) CH2CF3
CH(Me)SCH2(D1-103a) CH2OMe
CH(Me)SCH2(D1-103a) CH2OCF3
CH(Me)SCH2(D1-103a) CH2SMe
CH(Me)SCH2(D1-103a) CH2S(O)Me
CH(Me)SCH2(D1-103a) CH2S(O)2Me
CH(Me)SCH2(D1-103a) CH2SCF3
CH(Me)SCH2(D1-103a) CH2S(O)CF3
CH(Me)SCH2(D1-103a) CH2S(O)2CF3
CH(Me)SCH2(D1-103a) CH2CH(OMe)2
CH(Me)SCH2(D1-103a) CH2CH(SMe)2
CH(Me)SCH2(D1-103a) CH2C(O)Me
CH(Me)SCH2(D1-103a) CH2C(O)CF3
CH(Me)SCH2(D1-103a) CH2C(O)OMe
CH(Me)SCH2(D1-103a) CH2(D1-32a)
CH(Me)SCH2(D1-103a) CH2(D1-33a)
CH(Me)SCH2(D1-103a) CH2(D1-34a)
CH(Me)SCH2(D1-103a) CH2(D1-37a)
CH(Me)SCH2(D1-103a) CH2(D1-81a)
CH(Me)SCH2(D1-103a) CH2(D1-82a)
CH(Me)SCH2(D1-103a) CH2(D1-84a)
CH(Me)SCH2(D1-103a) CH2(D1-85a)
CH(Me)SCH2(D1-103a) CH2(D1-87a)
CH(Me)SCH2(D1-103a) CH2(D1-92a)
CH(Me)SCH2(D1-103a) CH2(D1-93a)
CH(Me)SCH2(D1-103a) CH2(D1-95a)
CH(Me)SCH2(D1-103a) CH2(D1-96a)
CH(Me)SCH2(D1-103a) CH2(D1-98a)
CH(Me)SCH2(D1-103a) CH2(D1-108a)
CH(Me)SCH2(D1-103a) CH2(D1-108b,Z=2-Cl)
CH(Me)SCH2(D1-103a) CH2(D1-108b,Z=3-Me)
CH(Me)SCH2(D1-103a) CH2(D1-108b,Z=4-OMe)
CH(Me)SCH2(D1-103a) CH2(D1-108b,Z=2-SMe)
CH(Me)SCH2(D1-103a) CH2(D1-108b,Z=3-CF3)
CH(Me)SCH2(D1-103a) CH2(D1-108b,Z=4-OCF3)
CH(Me)SCH2(D1-103a) CH2(D1-108b,Z=2-SCF3)
CH(Me)SCH2(D1-103a) CH2CH2CN
CH(Me)SCH2(D1-103a) CH2CH2CF3
CH(Me)SCH2(D1-103a) CH2CH2OMe
CH(Me)SCH2(D1-103a) CH2CH2SMe
CH(Me)SCH2(D1-103a) CH2CH2S(O)Me
CH(Me)SCH2(D1-103a) CH2CH2S(O)2Me
CH(Me)SCH2(D1-103a) D1-32a
CH(Me)SCH2(D1-103a) D1-33a
CH(Me)SCH2(D1-103a) D1-34a
CH(Me)SCH2(D1-103a) D1-37a
CH(Me)SCH2(D1-103a) D1-81a
CH(Me)SCH2(D1-103a) D1-82a
CH(Me)SCH2(D1-103a) D1-84a
CH(Me)SCH2(D1-103a) D1-85a
CH(Me)SCH2(D1-103a) D1-87a
CH(Me)SCH2(D1-103a) D1-92a
CH(Me)SCH2(D1-103a) D1-93a
CH(Me)SCH2(D1-103a) D1-95a
CH(Me)SCH2(D1-103a) D1-96a
CH(Me)SCH2(D1-103a) D1-98a
CH(Me)SCH2(D1-103a) D1-108a
CH(Me)SCH2(D1-103a) D1-108b(Z=2-Cl)
CH(Me)SCH2(D1-103a) D1-108b(Z=3-Me)
CH(Me)SCH2(D1-103a) D1-108b(Z=4-OMe)
CH(Me)SCH2(D1-103a) D1-108b(Z=2-SMe)
CH(Me)SCH2(D1-103a) D1-108b(Z=3-CF3)
CH(Me)SCH2(D1-103a) D1-108b(Z=4-OCF3)
CH(Me)SCH2(D1-103a) D1-108b(Z=2-SCF3)
CH(Me)SCH2(D1-103a) C(O)Me
CH(Me)SCH2(D1-103a) C(O)CF3
CH(Me)SCH2(D1-103a) C(O)OMe
CH(Me)S(O)CH2(D1-103a) Me
CH(Me)S(O)CH2(D1-103a) Et
CH(Me)S(O)CH2(D1-103a) Pr-n
CH(Me)S(O)CH2(D1-103a) Pr-i
CH(Me)S(O)CH2(D1-103a) Pr-c
CH(Me)S(O)CH2(D1-103a) Bu-n
CH(Me)S(O)CH2(D1-103a) Bu-i
CH(Me)S(O)CH2(D1-103a) Bu-c
CH(Me)S(O)CH2(D1-103a) Bu-s
CH(Me)S(O)CH2(D1-103a) Bu-t
CH(Me)S(O)CH2(D1-103a) Pen-n
CH(Me)S(O)CH2(D1-103a) Pen-c
CH(Me)S(O)CH2(D1-103a) Hex-n
CH(Me)S(O)CH2(D1-103a) Hex-c
CH(Me)S(O)CH2(D1-103a) CH2Pr-c
CH(Me)S(O)CH2(D1-103a) CH2Bu-c
CH(Me)S(O)CH2(D1-103a) CH2Pen-c
CH(Me)S(O)CH2(D1-103a) CH2Hex-c
CH(Me)S(O)CH2(D1-103a) CH2CH=CH2
CH(Me)S(O)CH2(D1-103a) CH2CH=C(Cl)2
CH(Me)S(O)CH2(D1-103a) CH2C≡CH
CH(Me)S(O)CH2(D1-103a) CH2CN
CH(Me)S(O)CH2(D1-103a) CH2CF3
CH(Me)S(O)CH2(D1-103a) CH2OMe
CH(Me)S(O)CH2(D1-103a) CH2OCF3
CH(Me)S(O)CH2(D1-103a) CH2SMe
CH(Me)S(O)CH2(D1-103a) CH2S(O)Me
CH(Me)S(O)CH2(D1-103a) CH2S(O)2Me
CH(Me)S(O)CH2(D1-103a) CH2SCF3
CH(Me)S(O)CH2(D1-103a) CH2S(O)CF3
CH(Me)S(O)CH2(D1-103a) CH2S(O)2CF3
CH(Me)S(O)CH2(D1-103a) CH2CH(OMe)2
CH(Me)S(O)CH2(D1-103a) CH2CH(SMe)2
CH(Me)S(O)CH2(D1-103a) CH2C(O)Me
CH(Me)S(O)CH2(D1-103a) CH2C(O)CF3
CH(Me)S(O)CH2(D1-103a) CH2C(O)OMe
CH(Me)S(O)CH2(D1-103a) CH2(D1-32a)
CH(Me)S(O)CH2(D1-103a) CH2(D1-33a)
CH(Me)S(O)CH2(D1-103a) CH2(D1-34a)
CH(Me)S(O)CH2(D1-103a) CH2(D1-37a)
CH(Me)S(O)CH2(D1-103a) CH2(D1-81a)
CH(Me)S(O)CH2(D1-103a) CH2(D1-82a)
CH(Me)S(O)CH2(D1-103a) CH2(D1-84a)
CH(Me)S(O)CH2(D1-103a) CH2(D1-85a)
CH(Me)S(O)CH2(D1-103a) CH2(D1-87a)
CH(Me)S(O)CH2(D1-103a) CH2(D1-92a)
CH(Me)S(O)CH2(D1-103a) CH2(D1-93a)
CH(Me)S(O)CH2(D1-103a) CH2(D1-95a)
CH(Me)S(O)CH2(D1-103a) CH2(D1-96a)
CH(Me)S(O)CH2(D1-103a) CH2(D1-98a)
CH(Me)S(O)CH2(D1-103a) CH2(D1-108a)
CH(Me)S(O)CH2(D1-103a) CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)CH2(D1-103a) CH2(D1-108b,Z=3-Me)
CH(Me)S(O)CH2(D1-103a) CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)CH2(D1-103a) CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)CH2(D1-103a) CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)CH2(D1-103a) CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)CH2(D1-103a) CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)CH2(D1-103a) CH2CH2CN
CH(Me)S(O)CH2(D1-103a) CH2CH2CF3
CH(Me)S(O)CH2(D1-103a) CH2CH2OMe
CH(Me)S(O)CH2(D1-103a) CH2CH2SMe
CH(Me)S(O)CH2(D1-103a) CH2CH2S(O)Me
CH(Me)S(O)CH2(D1-103a) CH2CH2S(O)2Me
CH(Me)S(O)CH2(D1-103a) D1-32a
CH(Me)S(O)CH2(D1-103a) D1-33a
CH(Me)S(O)CH2(D1-103a) D1-34a
CH(Me)S(O)CH2(D1-103a) D1-37a
CH(Me)S(O)CH2(D1-103a) D1-81a
CH(Me)S(O)CH2(D1-103a) D1-82a
CH(Me)S(O)CH2(D1-103a) D1-84a
CH(Me)S(O)CH2(D1-103a) D1-85a
CH(Me)S(O)CH2(D1-103a) D1-87a
CH(Me)S(O)CH2(D1-103a) D1-92a
CH(Me)S(O)CH2(D1-103a) D1-93a
CH(Me)S(O)CH2(D1-103a) D1-95a
CH(Me)S(O)CH2(D1-103a) D1-96a
CH(Me)S(O)CH2(D1-103a) D1-98a
CH(Me)S(O)CH2(D1-103a) D1-108a
CH(Me)S(O)CH2(D1-103a) D1-108b(Z=2-Cl)
CH(Me)S(O)CH2(D1-103a) D1-108b(Z=3-Me)
CH(Me)S(O)CH2(D1-103a) D1-108b(Z=4-OMe)
CH(Me)S(O)CH2(D1-103a) D1-108b(Z=2-SMe)
CH(Me)S(O)CH2(D1-103a) D1-108b(Z=3-CF3)
CH(Me)S(O)CH2(D1-103a) D1-108b(Z=4-OCF3)
CH(Me)S(O)CH2(D1-103a) D1-108b(Z=2-SCF3)
CH(Me)S(O)CH2(D1-103a) C(O)Me
CH(Me)S(O)CH2(D1-103a) C(O)CF3
CH(Me)S(O)CH2(D1-103a) C(O)OMe
CH(Me)S(O)2CH2(D1-103a) Me
CH(Me)S(O)2CH2(D1-103a) Et
CH(Me)S(O)2CH2(D1-103a) Pr-n
CH(Me)S(O)2CH2(D1-103a) Pr-i
CH(Me)S(O)2CH2(D1-103a) Pr-c
CH(Me)S(O)2CH2(D1-103a) Bu-n
CH(Me)S(O)2CH2(D1-103a) Bu-i
CH(Me)S(O)2CH2(D1-103a) Bu-c
CH(Me)S(O)2CH2(D1-103a) Bu-s
CH(Me)S(O)2CH2(D1-103a) Bu-t
CH(Me)S(O)2CH2(D1-103a) Pen-n
CH(Me)S(O)2CH2(D1-103a) Pen-c
CH(Me)S(O)2CH2(D1-103a) Hex-n
CH(Me)S(O)2CH2(D1-103a) Hex-c
CH(Me)S(O)2CH2(D1-103a) CH2Pr-c
CH(Me)S(O)2CH2(D1-103a) CH2Bu-c
CH(Me)S(O)2CH2(D1-103a) CH2Pen-c
CH(Me)S(O)2CH2(D1-103a) CH2Hex-c
CH(Me)S(O)2CH2(D1-103a) CH2CH=CH2
CH(Me)S(O)2CH2(D1-103a) CH2CH=C(Cl)2
CH(Me)S(O)2CH2(D1-103a) CH2C≡CH
CH(Me)S(O)2CH2(D1-103a) CH2CN
CH(Me)S(O)2CH2(D1-103a) CH2CF3
CH(Me)S(O)2CH2(D1-103a) CH2OMe
CH(Me)S(O)2CH2(D1-103a) CH2OCF3
CH(Me)S(O)2CH2(D1-103a) CH2SMe
CH(Me)S(O)2CH2(D1-103a) CH2S(O)Me
CH(Me)S(O)2CH2(D1-103a) CH2S(O)2Me
CH(Me)S(O)2CH2(D1-103a) CH2SCF3
CH(Me)S(O)2CH2(D1-103a) CH2S(O)CF3
CH(Me)S(O)2CH2(D1-103a) CH2S(O)2CF3
CH(Me)S(O)2CH2(D1-103a) CH2CH(OMe)2
CH(Me)S(O)2CH2(D1-103a) CH2CH(SMe)2
CH(Me)S(O)2CH2(D1-103a) CH2C(O)Me
CH(Me)S(O)2CH2(D1-103a) CH2C(O)CF3
CH(Me)S(O)2CH2(D1-103a) CH2C(O)OMe
CH(Me)S(O)2CH2(D1-103a) CH2(D1-32a)
CH(Me)S(O)2CH2(D1-103a) CH2(D1-33a)
CH(Me)S(O)2CH2(D1-103a) CH2(D1-34a)
CH(Me)S(O)2CH2(D1-103a) CH2(D1-37a)
CH(Me)S(O)2CH2(D1-103a) CH2(D1-81a)
CH(Me)S(O)2CH2(D1-103a) CH2(D1-82a)
CH(Me)S(O)2CH2(D1-103a) CH2(D1-84a)
CH(Me)S(O)2CH2(D1-103a) CH2(D1-85a)
CH(Me)S(O)2CH2(D1-103a) CH2(D1-87a)
CH(Me)S(O)2CH2(D1-103a) CH2(D1-92a)
CH(Me)S(O)2CH2(D1-103a) CH2(D1-93a)
CH(Me)S(O)2CH2(D1-103a) CH2(D1-95a)
CH(Me)S(O)2CH2(D1-103a) CH2(D1-96a)
CH(Me)S(O)2CH2(D1-103a) CH2(D1-98a)
CH(Me)S(O)2CH2(D1-103a) CH2(D1-108a)
CH(Me)S(O)2CH2(D1-103a) CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)2CH2(D1-103a) CH2(D1-108b,Z=3-Me)
CH(Me)S(O)2CH2(D1-103a) CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)2CH2(D1-103a) CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)2CH2(D1-103a) CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)2CH2(D1-103a) CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)2CH2(D1-103a) CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)2CH2(D1-103a) CH2CH2CN
CH(Me)S(O)2CH2(D1-103a) CH2CH2CF3
CH(Me)S(O)2CH2(D1-103a) CH2CH2OMe
CH(Me)S(O)2CH2(D1-103a) CH2CH2SMe
CH(Me)S(O)2CH2(D1-103a) CH2CH2S(O)Me
CH(Me)S(O)2CH2(D1-103a) CH2CH2S(O)2Me
CH(Me)S(O)2CH2(D1-103a) D1-32a
CH(Me)S(O)2CH2(D1-103a) D1-33a
CH(Me)S(O)2CH2(D1-103a) D1-34a
CH(Me)S(O)2CH2(D1-103a) D1-37a
CH(Me)S(O)2CH2(D1-103a) D1-81a
CH(Me)S(O)2CH2(D1-103a) D1-82a
CH(Me)S(O)2CH2(D1-103a) D1-84a
CH(Me)S(O)2CH2(D1-103a) D1-85a
CH(Me)S(O)2CH2(D1-103a) D1-87a
CH(Me)S(O)2CH2(D1-103a) D1-92a
CH(Me)S(O)2CH2(D1-103a) D1-93a
CH(Me)S(O)2CH2(D1-103a) D1-95a
CH(Me)S(O)2CH2(D1-103a) D1-96a
CH(Me)S(O)2CH2(D1-103a) D1-98a
CH(Me)S(O)2CH2(D1-103a) D1-108a
CH(Me)S(O)2CH2(D1-103a) D1-108b(Z=2-Cl)
CH(Me)S(O)2CH2(D1-103a) D1-108b(Z=3-Me)
CH(Me)S(O)2CH2(D1-103a) D1-108b(Z=4-OMe)
CH(Me)S(O)2CH2(D1-103a) D1-108b(Z=2-SMe)
CH(Me)S(O)2CH2(D1-103a) D1-108b(Z=3-CF3)
CH(Me)S(O)2CH2(D1-103a) D1-108b(Z=4-OCF3)
CH(Me)S(O)2CH2(D1-103a) D1-108b(Z=2-SCF3)
CH(Me)S(O)2CH2(D1-103a) C(O)Me
CH(Me)S(O)2CH2(D1-103a) C(O)CF3
CH(Me)S(O)2CH2(D1-103a) C(O)OMe
CH(Et)SCH2(D1-103a) Me
CH(Et)SCH2(D1-103a) Et
CH(Et)SCH2(D1-103a) Pr-n
CH(Et)SCH2(D1-103a) Pr-i
CH(Et)SCH2(D1-103a) Pr-c
CH(Et)SCH2(D1-103a) Bu-n
CH(Et)SCH2(D1-103a) Bu-i
CH(Et)SCH2(D1-103a) Bu-c
CH(Et)SCH2(D1-103a) Bu-s
CH(Et)SCH2(D1-103a) Bu-t
CH(Et)SCH2(D1-103a) Pen-n
CH(Et)SCH2(D1-103a) Pen-c
CH(Et)SCH2(D1-103a) Hex-n
CH(Et)SCH2(D1-103a) Hex-c
CH(Et)SCH2(D1-103a) CH2Pr-c
CH(Et)SCH2(D1-103a) CH2Bu-c
CH(Et)SCH2(D1-103a) CH2Pen-c
CH(Et)SCH2(D1-103a) CH2Hex-c
CH(Et)SCH2(D1-103a) CH2CH=CH2
CH(Et)SCH2(D1-103a) CH2CH=C(Cl)2
CH(Et)SCH2(D1-103a) CH2C≡CH
CH(Et)SCH2(D1-103a) CH2CN
CH(Et)SCH2(D1-103a) CH2CF3
CH(Et)SCH2(D1-103a) CH2OMe
CH(Et)SCH2(D1-103a) CH2OCF3
CH(Et)SCH2(D1-103a) CH2SMe
CH(Et)SCH2(D1-103a) CH2S(O)Me
CH(Et)SCH2(D1-103a) CH2S(O)2Me
CH(Et)SCH2(D1-103a) CH2SCF3
CH(Et)SCH2(D1-103a) CH2S(O)CF3
CH(Et)SCH2(D1-103a) CH2S(O)2CF3
CH(Et)SCH2(D1-103a) CH2CH(OMe)2
CH(Et)SCH2(D1-103a) CH2CH(SMe)2
CH(Et)SCH2(D1-103a) CH2C(O)Me
CH(Et)SCH2(D1-103a) CH2C(O)CF3
CH(Et)SCH2(D1-103a) CH2C(O)OMe
CH(Et)SCH2(D1-103a) CH2(D1-32a)
CH(Et)SCH2(D1-103a) CH2(D1-33a)
CH(Et)SCH2(D1-103a) CH2(D1-34a)
CH(Et)SCH2(D1-103a) CH2(D1-37a)
CH(Et)SCH2(D1-103a) CH2(D1-81a)
CH(Et)SCH2(D1-103a) CH2(D1-82a)
CH(Et)SCH2(D1-103a) CH2(D1-84a)
CH(Et)SCH2(D1-103a) CH2(D1-85a)
CH(Et)SCH2(D1-103a) CH2(D1-87a)
CH(Et)SCH2(D1-103a) CH2(D1-92a)
CH(Et)SCH2(D1-103a) CH2(D1-93a)
CH(Et)SCH2(D1-103a) CH2(D1-95a)
CH(Et)SCH2(D1-103a) CH2(D1-96a)
CH(Et)SCH2(D1-103a) CH2(D1-98a)
CH(Et)SCH2(D1-103a) CH2(D1-108a)
CH(Et)SCH2(D1-103a) CH2(D1-108b,Z=2-Cl)
CH(Et)SCH2(D1-103a) CH2(D1-108b,Z=3-Me)
CH(Et)SCH2(D1-103a) CH2(D1-108b,Z=4-OMe)
CH(Et)SCH2(D1-103a) CH2(D1-108b,Z=2-SMe)
CH(Et)SCH2(D1-103a) CH2(D1-108b,Z=3-CF3)
CH(Et)SCH2(D1-103a) CH2(D1-108b,Z=4-OCF3)
CH(Et)SCH2(D1-103a) CH2(D1-108b,Z=2-SCF3)
CH(Et)SCH2(D1-103a) CH2CH2CN
CH(Et)SCH2(D1-103a) CH2CH2CF3
CH(Et)SCH2(D1-103a) CH2CH2OMe
CH(Et)SCH2(D1-103a) CH2CH2SMe
CH(Et)SCH2(D1-103a) CH2CH2S(O)Me
CH(Et)SCH2(D1-103a) CH2CH2S(O)2Me
CH(Et)SCH2(D1-103a) D1-32a
CH(Et)SCH2(D1-103a) D1-33a
CH(Et)SCH2(D1-103a) D1-34a
CH(Et)SCH2(D1-103a) D1-37a
CH(Et)SCH2(D1-103a) D1-81a
CH(Et)SCH2(D1-103a) D1-82a
CH(Et)SCH2(D1-103a) D1-84a
CH(Et)SCH2(D1-103a) D1-85a
CH(Et)SCH2(D1-103a) D1-87a
CH(Et)SCH2(D1-103a) D1-92a
CH(Et)SCH2(D1-103a) D1-93a
CH(Et)SCH2(D1-103a) D1-95a
CH(Et)SCH2(D1-103a) D1-96a
CH(Et)SCH2(D1-103a) D1-98a
CH(Et)SCH2(D1-103a) D1-108a
CH(Et)SCH2(D1-103a) D1-108b(Z=2-Cl)
CH(Et)SCH2(D1-103a) D1-108b(Z=3-Me)
CH(Et)SCH2(D1-103a) D1-108b(Z=4-OMe)
CH(Et)SCH2(D1-103a) D1-108b(Z=2-SMe)
CH(Et)SCH2(D1-103a) D1-108b(Z=3-CF3)
CH(Et)SCH2(D1-103a) D1-108b(Z=4-OCF3)
CH(Et)SCH2(D1-103a) D1-108b(Z=2-SCF3)
CH(Et)SCH2(D1-103a) C(O)Me
CH(Et)SCH2(D1-103a) C(O)CF3
CH(Et)SCH2(D1-103a) C(O)OMe
CH(Et)S(O)CH2(D1-103a) Me
CH(Et)S(O)CH2(D1-103a) Et
CH(Et)S(O)CH2(D1-103a) Pr-n
CH(Et)S(O)CH2(D1-103a) Pr-i
CH(Et)S(O)CH2(D1-103a) Pr-c
CH(Et)S(O)CH2(D1-103a) Bu-n
CH(Et)S(O)CH2(D1-103a) Bu-i
CH(Et)S(O)CH2(D1-103a) Bu-c
CH(Et)S(O)CH2(D1-103a) Bu-s
CH(Et)S(O)CH2(D1-103a) Bu-t
CH(Et)S(O)CH2(D1-103a) Pen-n
CH(Et)S(O)CH2(D1-103a) Pen-c
CH(Et)S(O)CH2(D1-103a) Hex-n
CH(Et)S(O)CH2(D1-103a) Hex-c
CH(Et)S(O)CH2(D1-103a) CH2Pr-c
CH(Et)S(O)CH2(D1-103a) CH2Bu-c
CH(Et)S(O)CH2(D1-103a) CH2Pen-c
CH(Et)S(O)CH2(D1-103a) CH2Hex-c
CH(Et)S(O)CH2(D1-103a) CH2CH=CH2
CH(Et)S(O)CH2(D1-103a) CH2CH=C(Cl)2
CH(Et)S(O)CH2(D1-103a) CH2C≡CH
CH(Et)S(O)CH2(D1-103a) CH2CN
CH(Et)S(O)CH2(D1-103a) CH2CF3
CH(Et)S(O)CH2(D1-103a) CH2OMe
CH(Et)S(O)CH2(D1-103a) CH2OCF3
CH(Et)S(O)CH2(D1-103a) CH2SMe
CH(Et)S(O)CH2(D1-103a) CH2S(O)Me
CH(Et)S(O)CH2(D1-103a) CH2S(O)2Me
CH(Et)S(O)CH2(D1-103a) CH2SCF3
CH(Et)S(O)CH2(D1-103a) CH2S(O)CF3
CH(Et)S(O)CH2(D1-103a) CH2S(O)2CF3
CH(Et)S(O)CH2(D1-103a) CH2CH(OMe)2
CH(Et)S(O)CH2(D1-103a) CH2CH(SMe)2
CH(Et)S(O)CH2(D1-103a) CH2C(O)Me
CH(Et)S(O)CH2(D1-103a) CH2C(O)CF3
CH(Et)S(O)CH2(D1-103a) CH2C(O)OMe
CH(Et)S(O)CH2(D1-103a) CH2(D1-32a)
CH(Et)S(O)CH2(D1-103a) CH2(D1-33a)
CH(Et)S(O)CH2(D1-103a) CH2(D1-34a)
CH(Et)S(O)CH2(D1-103a) CH2(D1-37a)
CH(Et)S(O)CH2(D1-103a) CH2(D1-81a)
CH(Et)S(O)CH2(D1-103a) CH2(D1-82a)
CH(Et)S(O)CH2(D1-103a) CH2(D1-84a)
CH(Et)S(O)CH2(D1-103a) CH2(D1-85a)
CH(Et)S(O)CH2(D1-103a) CH2(D1-87a)
CH(Et)S(O)CH2(D1-103a) CH2(D1-92a)
CH(Et)S(O)CH2(D1-103a) CH2(D1-93a)
CH(Et)S(O)CH2(D1-103a) CH2(D1-95a)
CH(Et)S(O)CH2(D1-103a) CH2(D1-96a)
CH(Et)S(O)CH2(D1-103a) CH2(D1-98a)
CH(Et)S(O)CH2(D1-103a) CH2(D1-108a)
CH(Et)S(O)CH2(D1-103a) CH2(D1-108b,Z=2-Cl)
CH(Et)S(O)CH2(D1-103a) CH2(D1-108b,Z=3-Me)
CH(Et)S(O)CH2(D1-103a) CH2(D1-108b,Z=4-OMe)
CH(Et)S(O)CH2(D1-103a) CH2(D1-108b,Z=2-SMe)
CH(Et)S(O)CH2(D1-103a) CH2(D1-108b,Z=3-CF3)
CH(Et)S(O)CH2(D1-103a) CH2(D1-108b,Z=4-OCF3)
CH(Et)S(O)CH2(D1-103a) CH2(D1-108b,Z=2-SCF3)
CH(Et)S(O)CH2(D1-103a) CH2CH2CN
CH(Et)S(O)CH2(D1-103a) CH2CH2CF3
CH(Et)S(O)CH2(D1-103a) CH2CH2OMe
CH(Et)S(O)CH2(D1-103a) CH2CH2SMe
CH(Et)S(O)CH2(D1-103a) CH2CH2S(O)Me
CH(Et)S(O)CH2(D1-103a) CH2CH2S(O)2Me
CH(Et)S(O)CH2(D1-103a) D1-32a
CH(Et)S(O)CH2(D1-103a) D1-33a
CH(Et)S(O)CH2(D1-103a) D1-34a
CH(Et)S(O)CH2(D1-103a) D1-37a
CH(Et)S(O)CH2(D1-103a) D1-81a
CH(Et)S(O)CH2(D1-103a) D1-82a
CH(Et)S(O)CH2(D1-103a) D1-84a
CH(Et)S(O)CH2(D1-103a) D1-85a
CH(Et)S(O)CH2(D1-103a) D1-87a
CH(Et)S(O)CH2(D1-103a) D1-92a
CH(Et)S(O)CH2(D1-103a) D1-93a
CH(Et)S(O)CH2(D1-103a) D1-95a
CH(Et)S(O)CH2(D1-103a) D1-96a
CH(Et)S(O)CH2(D1-103a) D1-98a
CH(Et)S(O)CH2(D1-103a) D1-108a
CH(Et)S(O)CH2(D1-103a) D1-108b(Z=2-Cl)
CH(Et)S(O)CH2(D1-103a) D1-108b(Z=3-Me)
CH(Et)S(O)CH2(D1-103a) D1-108b(Z=4-OMe)
CH(Et)S(O)CH2(D1-103a) D1-108b(Z=2-SMe)
CH(Et)S(O)CH2(D1-103a) D1-108b(Z=3-CF3)
CH(Et)S(O)CH2(D1-103a) D1-108b(Z=4-OCF3)
CH(Et)S(O)CH2(D1-103a) D1-108b(Z=2-SCF3)
CH(Et)S(O)CH2(D1-103a) C(O)Me
CH(Et)S(O)CH2(D1-103a) C(O)CF3
CH(Et)S(O)CH2(D1-103a) C(O)OMe
CH(Et)S(O)2CH2(D1-103a) Me
CH(Et)S(O)2CH2(D1-103a) Et
CH(Et)S(O)2CH2(D1-103a) Pr-n
CH(Et)S(O)2CH2(D1-103a) Pr-i
CH(Et)S(O)2CH2(D1-103a) Pr-c
CH(Et)S(O)2CH2(D1-103a) Bu-n
CH(Et)S(O)2CH2(D1-103a) Bu-i
CH(Et)S(O)2CH2(D1-103a) Bu-c
CH(Et)S(O)2CH2(D1-103a) Bu-s
CH(Et)S(O)2CH2(D1-103a) Bu-t
CH(Et)S(O)2CH2(D1-103a) Pen-n
CH(Et)S(O)2CH2(D1-103a) Pen-c
CH(Et)S(O)2CH2(D1-103a) Hex-n
CH(Et)S(O)2CH2(D1-103a) Hex-c
CH(Et)S(O)2CH2(D1-103a) CH2Pr-c
CH(Et)S(O)2CH2(D1-103a) CH2Bu-c
CH(Et)S(O)2CH2(D1-103a) CH2Pen-c
CH(Et)S(O)2CH2(D1-103a) CH2Hex-c
CH(Et)S(O)2CH2(D1-103a) CH2CH=CH2
CH(Et)S(O)2CH2(D1-103a) CH2CH=C(Cl)2
CH(Et)S(O)2CH2(D1-103a) CH2C≡CH
CH(Et)S(O)2CH2(D1-103a) CH2CN
CH(Et)S(O)2CH2(D1-103a) CH2CF3
CH(Et)S(O)2CH2(D1-103a) CH2OMe
CH(Et)S(O)2CH2(D1-103a) CH2OCF3
CH(Et)S(O)2CH2(D1-103a) CH2SMe
CH(Et)S(O)2CH2(D1-103a) CH2S(O)Me
CH(Et)S(O)2CH2(D1-103a) CH2S(O)2Me
CH(Et)S(O)2CH2(D1-103a) CH2SCF3
CH(Et)S(O)2CH2(D1-103a) CH2S(O)CF3
CH(Et)S(O)2CH2(D1-103a) CH2S(O)2CF3
CH(Et)S(O)2CH2(D1-103a) CH2CH(OMe)2
CH(Et)S(O)2CH2(D1-103a) CH2CH(SMe)2
CH(Et)S(O)2CH2(D1-103a) CH2C(O)Me
CH(Et)S(O)2CH2(D1-103a) CH2C(O)CF3
CH(Et)S(O)2CH2(D1-103a) CH2C(O)OMe
CH(Et)S(O)2CH2(D1-103a) CH2(D1-32a)
CH(Et)S(O)2CH2(D1-103a) CH2(D1-33a)
CH(Et)S(O)2CH2(D1-103a) CH2(D1-34a)
CH(Et)S(O)2CH2(D1-103a) CH2(D1-37a)
CH(Et)S(O)2CH2(D1-103a) CH2(D1-81a)
CH(Et)S(O)2CH2(D1-103a) CH2(D1-82a)
CH(Et)S(O)2CH2(D1-103a) CH2(D1-84a)
CH(Et)S(O)2CH2(D1-103a) CH2(D1-85a)
CH(Et)S(O)2CH2(D1-103a) CH2(D1-87a)
CH(Et)S(O)2CH2(D1-103a) CH2(D1-92a)
CH(Et)S(O)2CH2(D1-103a) CH2(D1-93a)
CH(Et)S(O)2CH2(D1-103a) CH2(D1-95a)
CH(Et)S(O)2CH2(D1-103a) CH2(D1-96a)
CH(Et)S(O)2CH2(D1-103a) CH2(D1-98a)
CH(Et)S(O)2CH2(D1-103a) CH2(D1-108a)
CH(Et)S(O)2CH2(D1-103a) CH2(D1-108b,Z=2-Cl)
CH(Et)S(O)2CH2(D1-103a) CH2(D1-108b,Z=3-Me)
CH(Et)S(O)2CH2(D1-103a) CH2(D1-108b,Z=4-OMe)
CH(Et)S(O)2CH2(D1-103a) CH2(D1-108b,Z=2-SMe)
CH(Et)S(O)2CH2(D1-103a) CH2(D1-108b,Z=3-CF3)
CH(Et)S(O)2CH2(D1-103a) CH2(D1-108b,Z=4-OCF3)
CH(Et)S(O)2CH2(D1-103a) CH2(D1-108b,Z=2-SCF3)
CH(Et)S(O)2CH2(D1-103a) CH2CH2CN
CH(Et)S(O)2CH2(D1-103a) CH2CH2CF3
CH(Et)S(O)2CH2(D1-103a) CH2CH2OMe
CH(Et)S(O)2CH2(D1-103a) CH2CH2SMe
CH(Et)S(O)2CH2(D1-103a) CH2CH2S(O)Me
CH(Et)S(O)2CH2(D1-103a) CH2CH2S(O)2Me
CH(Et)S(O)2CH2(D1-103a) D1-32a
CH(Et)S(O)2CH2(D1-103a) D1-33a
CH(Et)S(O)2CH2(D1-103a) D1-34a
CH(Et)S(O)2CH2(D1-103a) D1-37a
CH(Et)S(O)2CH2(D1-103a) D1-81a
CH(Et)S(O)2CH2(D1-103a) D1-82a
CH(Et)S(O)2CH2(D1-103a) D1-84a
CH(Et)S(O)2CH2(D1-103a) D1-85a
CH(Et)S(O)2CH2(D1-103a) D1-87a
CH(Et)S(O)2CH2(D1-103a) D1-92a
CH(Et)S(O)2CH2(D1-103a) D1-93a
CH(Et)S(O)2CH2(D1-103a) D1-95a
CH(Et)S(O)2CH2(D1-103a) D1-96a
CH(Et)S(O)2CH2(D1-103a) D1-98a
CH(Et)S(O)2CH2(D1-103a) D1-108a
CH(Et)S(O)2CH2(D1-103a) D1-108b(Z=2-Cl)
CH(Et)S(O)2CH2(D1-103a) D1-108b(Z=3-Me)
CH(Et)S(O)2CH2(D1-103a) D1-108b(Z=4-OMe)
CH(Et)S(O)2CH2(D1-103a) D1-108b(Z=2-SMe)
CH(Et)S(O)2CH2(D1-103a) D1-108b(Z=3-CF3)
CH(Et)S(O)2CH2(D1-103a) D1-108b(Z=4-OCF3)
CH(Et)S(O)2CH2(D1-103a) D1-108b(Z=2-SCF3)
CH(Et)S(O)2CH2(D1-103a) C(O)Me
CH(Et)S(O)2CH2(D1-103a) C(O)CF3
CH(Et)S(O)2CH2(D1-103a) C(O)OMe
CH2SCH2CH=CH2 Me
CH2SCH2CH=CH2 Et
CH2SCH2CH=CH2 Pr-n
CH2SCH2CH=CH2 Pr-i
CH2SCH2CH=CH2 Pr-c
CH2SCH2CH=CH2 Bu-n
CH2SCH2CH=CH2 Bu-i
CH2SCH2CH=CH2 Bu-c
CH2SCH2CH=CH2 Bu-s
CH2SCH2CH=CH2 Bu-t
CH2SCH2CH=CH2 Pen-n
CH2SCH2CH=CH2 Pen-c
CH2SCH2CH=CH2 Hex-n
CH2SCH2CH=CH2 Hex-c
CH2SCH2CH=CH2 CH2Pr-c
CH2SCH2CH=CH2 CH2Bu-c
CH2SCH2CH=CH2 CH2Pen-c
CH2SCH2CH=CH2 CH2Hex-c
CH2SCH2CH=CH2 CH2CH=CH2
CH2SCH2CH=CH2 CH2CH=C(Cl)2
CH2SCH2CH=CH2 CH2C≡CH
CH2SCH2CH=CH2 CH2CN
CH2SCH2CH=CH2 CH2CF3
CH2SCH2CH=CH2 CH2OMe
CH2SCH2CH=CH2 CH2OCF3
CH2SCH2CH=CH2 CH2SMe
CH2SCH2CH=CH2 CH2S(O)Me
CH2SCH2CH=CH2 CH2S(O)2Me
CH2SCH2CH=CH2 CH2SCF3
CH2SCH2CH=CH2 CH2S(O)CF3
CH2SCH2CH=CH2 CH2S(O)2CF3
CH2SCH2CH=CH2 CH2CH(OMe)2
CH2SCH2CH=CH2 CH2CH(SMe)2
CH2SCH2CH=CH2 CH2C(O)Me
CH2SCH2CH=CH2 CH2C(O)CF3
CH2SCH2CH=CH2 CH2C(O)OMe
CH2SCH2CH=CH2 CH2(D1-32a)
CH2SCH2CH=CH2 CH2(D1-33a)
CH2SCH2CH=CH2 CH2(D1-34a)
CH2SCH2CH=CH2 CH2(D1-37a)
CH2SCH2CH=CH2 CH2(D1-81a)
CH2SCH2CH=CH2 CH2(D1-82a)
CH2SCH2CH=CH2 CH2(D1-84a)
CH2SCH2CH=CH2 CH2(D1-85a)
CH2SCH2CH=CH2 CH2(D1-87a)
CH2SCH2CH=CH2 CH2(D1-92a)
CH2SCH2CH=CH2 CH2(D1-93a)
CH2SCH2CH=CH2 CH2(D1-95a)
CH2SCH2CH=CH2 CH2(D1-96a)
CH2SCH2CH=CH2 CH2(D1-98a)
CH2SCH2CH=CH2 CH2(D1-108a)
CH2SCH2CH=CH2 CH2(D1-108b,Z=2-Cl)
CH2SCH2CH=CH2 CH2(D1-108b,Z=3-Me)
CH2SCH2CH=CH2 CH2(D1-108b,Z=4-OMe)
CH2SCH2CH=CH2 CH2(D1-108b,Z=2-SMe)
CH2SCH2CH=CH2 CH2(D1-108b,Z=3-CF3)
CH2SCH2CH=CH2 CH2(D1-108b,Z=4-OCF3)
CH2SCH2CH=CH2 CH2(D1-108b,Z=2-SCF3)
CH2SCH2CH=CH2 CH2CH2CN
CH2SCH2CH=CH2 CH2CH2CF3
CH2SCH2CH=CH2 CH2CH2OMe
CH2SCH2CH=CH2 CH2CH2SMe
CH2SCH2CH=CH2 CH2CH2S(O)Me
CH2SCH2CH=CH2 CH2CH2S(O)2Me
CH2SCH2CH=CH2 D1-32a
CH2SCH2CH=CH2 D1-33a
CH2SCH2CH=CH2 D1-34a
CH2SCH2CH=CH2 D1-37a
CH2SCH2CH=CH2 D1-81a
CH2SCH2CH=CH2 D1-82a
CH2SCH2CH=CH2 D1-84a
CH2SCH2CH=CH2 D1-85a
CH2SCH2CH=CH2 D1-87a
CH2SCH2CH=CH2 D1-92a
CH2SCH2CH=CH2 D1-93a
CH2SCH2CH=CH2 D1-95a
CH2SCH2CH=CH2 D1-96a
CH2SCH2CH=CH2 D1-98a
CH2SCH2CH=CH2 D1-108a
CH2SCH2CH=CH2 D1-108b(Z=2-Cl)
CH2SCH2CH=CH2 D1-108b(Z=3-Me)
CH2SCH2CH=CH2 D1-108b(Z=4-OMe)
CH2SCH2CH=CH2 D1-108b(Z=2-SMe)
CH2SCH2CH=CH2 D1-108b(Z=3-CF3)
CH2SCH2CH=CH2 D1-108b(Z=4-OCF3)
CH2SCH2CH=CH2 D1-108b(Z=2-SCF3)
CH2SCH2CH=CH2 C(O)Me
CH2SCH2CH=CH2 C(O)CF3
CH2SCH2CH=CH2 C(O)OMe
CH2S(O)CH2CH=CH2 Me
CH2S(O)CH2CH=CH2 Et
CH2S(O)CH2CH=CH2 Pr-n
CH2S(O)CH2CH=CH2 Pr-i
CH2S(O)CH2CH=CH2 Pr-c
CH2S(O)CH2CH=CH2 Bu-n
CH2S(O)CH2CH=CH2 Bu-i
CH2S(O)CH2CH=CH2 Bu-c
CH2S(O)CH2CH=CH2 Bu-s
CH2S(O)CH2CH=CH2 Bu-t
CH2S(O)CH2CH=CH2 Pen-n
CH2S(O)CH2CH=CH2 Pen-c
CH2S(O)CH2CH=CH2 Hex-n
CH2S(O)CH2CH=CH2 Hex-c
CH2S(O)CH2CH=CH2 CH2Pr-c
CH2S(O)CH2CH=CH2 CH2Bu-c
CH2S(O)CH2CH=CH2 CH2Pen-c
CH2S(O)CH2CH=CH2 CH2Hex-c
CH2S(O)CH2CH=CH2 CH2CH=CH2
CH2S(O)CH2CH=CH2 CH2CH=C(Cl)2
CH2S(O)CH2CH=CH2 CH2C≡CH
CH2S(O)CH2CH=CH2 CH2CN
CH2S(O)CH2CH=CH2 CH2CF3
CH2S(O)CH2CH=CH2 CH2OMe
CH2S(O)CH2CH=CH2 CH2OCF3
CH2S(O)CH2CH=CH2 CH2SMe
CH2S(O)CH2CH=CH2 CH2S(O)Me
CH2S(O)CH2CH=CH2 CH2S(O)2Me
CH2S(O)CH2CH=CH2 CH2SCF3
CH2S(O)CH2CH=CH2 CH2S(O)CF3
CH2S(O)CH2CH=CH2 CH2S(O)2CF3
CH2S(O)CH2CH=CH2 CH2CH(OMe)2
CH2S(O)CH2CH=CH2 CH2CH(SMe)2
CH2S(O)CH2CH=CH2 CH2C(O)Me
CH2S(O)CH2CH=CH2 CH2C(O)CF3
CH2S(O)CH2CH=CH2 CH2C(O)OMe
CH2S(O)CH2CH=CH2 CH2(D1-32a)
CH2S(O)CH2CH=CH2 CH2(D1-33a)
CH2S(O)CH2CH=CH2 CH2(D1-34a)
CH2S(O)CH2CH=CH2 CH2(D1-37a)
CH2S(O)CH2CH=CH2 CH2(D1-81a)
CH2S(O)CH2CH=CH2 CH2(D1-82a)
CH2S(O)CH2CH=CH2 CH2(D1-84a)
CH2S(O)CH2CH=CH2 CH2(D1-85a)
CH2S(O)CH2CH=CH2 CH2(D1-87a)
CH2S(O)CH2CH=CH2 CH2(D1-92a)
CH2S(O)CH2CH=CH2 CH2(D1-93a)
CH2S(O)CH2CH=CH2 CH2(D1-95a)
CH2S(O)CH2CH=CH2 CH2(D1-96a)
CH2S(O)CH2CH=CH2 CH2(D1-98a)
CH2S(O)CH2CH=CH2 CH2(D1-108a)
CH2S(O)CH2CH=CH2 CH2(D1-108b,Z=2-Cl)
CH2S(O)CH2CH=CH2 CH2(D1-108b,Z=3-Me)
CH2S(O)CH2CH=CH2 CH2(D1-108b,Z=4-OMe)
CH2S(O)CH2CH=CH2 CH2(D1-108b,Z=2-SMe)
CH2S(O)CH2CH=CH2 CH2(D1-108b,Z=3-CF3)
CH2S(O)CH2CH=CH2 CH2(D1-108b,Z=4-OCF3)
CH2S(O)CH2CH=CH2 CH2(D1-108b,Z=2-SCF3)
CH2S(O)CH2CH=CH2 CH2CH2CN
CH2S(O)CH2CH=CH2 CH2CH2CF3
CH2S(O)CH2CH=CH2 CH2CH2OMe
CH2S(O)CH2CH=CH2 CH2CH2SMe
CH2S(O)CH2CH=CH2 CH2CH2S(O)Me
CH2S(O)CH2CH=CH2 CH2CH2S(O)2Me
CH2S(O)CH2CH=CH2 D1-32a
CH2S(O)CH2CH=CH2 D1-33a
CH2S(O)CH2CH=CH2 D1-34a
CH2S(O)CH2CH=CH2 D1-37a
CH2S(O)CH2CH=CH2 D1-81a
CH2S(O)CH2CH=CH2 D1-82a
CH2S(O)CH2CH=CH2 D1-84a
CH2S(O)CH2CH=CH2 D1-85a
CH2S(O)CH2CH=CH2 D1-87a
CH2S(O)CH2CH=CH2 D1-92a
CH2S(O)CH2CH=CH2 D1-93a
CH2S(O)CH2CH=CH2 D1-95a
CH2S(O)CH2CH=CH2 D1-96a
CH2S(O)CH2CH=CH2 D1-98a
CH2S(O)CH2CH=CH2 D1-108a
CH2S(O)CH2CH=CH2 D1-108b(Z=2-Cl)
CH2S(O)CH2CH=CH2 D1-108b(Z=3-Me)
CH2S(O)CH2CH=CH2 D1-108b(Z=4-OMe)
CH2S(O)CH2CH=CH2 D1-108b(Z=2-SMe)
CH2S(O)CH2CH=CH2 D1-108b(Z=3-CF3)
CH2S(O)CH2CH=CH2 D1-108b(Z=4-OCF3)
CH2S(O)CH2CH=CH2 D1-108b(Z=2-SCF3)
CH2S(O)CH2CH=CH2 C(O)Me
CH2S(O)CH2CH=CH2 C(O)CF3
CH2S(O)CH2CH=CH2 C(O)OMe
CH2S(O)2CH2CH=CH2 Me
CH2S(O)2CH2CH=CH2 Et
CH2S(O)2CH2CH=CH2 Pr-n
CH2S(O)2CH2CH=CH2 Pr-i
CH2S(O)2CH2CH=CH2 Pr-c
CH2S(O)2CH2CH=CH2 Bu-n
CH2S(O)2CH2CH=CH2 Bu-i
CH2S(O)2CH2CH=CH2 Bu-c
CH2S(O)2CH2CH=CH2 Bu-s
CH2S(O)2CH2CH=CH2 Bu-t
CH2S(O)2CH2CH=CH2 Pen-n
CH2S(O)2CH2CH=CH2 Pen-c
CH2S(O)2CH2CH=CH2 Hex-n
CH2S(O)2CH2CH=CH2 Hex-c
CH2S(O)2CH2CH=CH2 CH2Pr-c
CH2S(O)2CH2CH=CH2 CH2Bu-c
CH2S(O)2CH2CH=CH2 CH2Pen-c
CH2S(O)2CH2CH=CH2 CH2Hex-c
CH2S(O)2CH2CH=CH2 CH2CH=CH2
CH2S(O)2CH2CH=CH2 CH2CH=C(Cl)2
CH2S(O)2CH2CH=CH2 CH2C≡CH
CH2S(O)2CH2CH=CH2 CH2CN
CH2S(O)2CH2CH=CH2 CH2CF3
CH2S(O)2CH2CH=CH2 CH2OMe
CH2S(O)2CH2CH=CH2 CH2OCF3
CH2S(O)2CH2CH=CH2 CH2SMe
CH2S(O)2CH2CH=CH2 CH2S(O)Me
CH2S(O)2CH2CH=CH2 CH2S(O)2Me
CH2S(O)2CH2CH=CH2 CH2SCF3
CH2S(O)2CH2CH=CH2 CH2S(O)CF3
CH2S(O)2CH2CH=CH2 CH2S(O)2CF3
CH2S(O)2CH2CH=CH2 CH2CH(OMe)2
CH2S(O)2CH2CH=CH2 CH2CH(SMe)2
CH2S(O)2CH2CH=CH2 CH2C(O)Me
CH2S(O)2CH2CH=CH2 CH2C(O)CF3
CH2S(O)2CH2CH=CH2 CH2C(O)OMe
CH2S(O)2CH2CH=CH2 CH2(D1-32a)
CH2S(O)2CH2CH=CH2 CH2(D1-33a)
CH2S(O)2CH2CH=CH2 CH2(D1-34a)
CH2S(O)2CH2CH=CH2 CH2(D1-37a)
CH2S(O)2CH2CH=CH2 CH2(D1-81a)
CH2S(O)2CH2CH=CH2 CH2(D1-82a)
CH2S(O)2CH2CH=CH2 CH2(D1-84a)
CH2S(O)2CH2CH=CH2 CH2(D1-85a)
CH2S(O)2CH2CH=CH2 CH2(D1-87a)
CH2S(O)2CH2CH=CH2 CH2(D1-92a)
CH2S(O)2CH2CH=CH2 CH2(D1-93a)
CH2S(O)2CH2CH=CH2 CH2(D1-95a)
CH2S(O)2CH2CH=CH2 CH2(D1-96a)
CH2S(O)2CH2CH=CH2 CH2(D1-98a)
CH2S(O)2CH2CH=CH2 CH2(D1-108a)
CH2S(O)2CH2CH=CH2 CH2(D1-108b,Z=2-Cl)
CH2S(O)2CH2CH=CH2 CH2(D1-108b,Z=3-Me)
CH2S(O)2CH2CH=CH2 CH2(D1-108b,Z=4-OMe)
CH2S(O)2CH2CH=CH2 CH2(D1-108b,Z=2-SMe)
CH2S(O)2CH2CH=CH2 CH2(D1-108b,Z=3-CF3)
CH2S(O)2CH2CH=CH2 CH2(D1-108b,Z=4-OCF3)
CH2S(O)2CH2CH=CH2 CH2(D1-108b,Z=2-SCF3)
CH2S(O)2CH2CH=CH2 CH2CH2CN
CH2S(O)2CH2CH=CH2 CH2CH2CF3
CH2S(O)2CH2CH=CH2 CH2CH2OMe
CH2S(O)2CH2CH=CH2 CH2CH2SMe
CH2S(O)2CH2CH=CH2 CH2CH2S(O)Me
CH2S(O)2CH2CH=CH2 CH2CH2S(O)2Me
CH2S(O)2CH2CH=CH2 D1-32a
CH2S(O)2CH2CH=CH2 D1-33a
CH2S(O)2CH2CH=CH2 D1-34a
CH2S(O)2CH2CH=CH2 D1-37a
CH2S(O)2CH2CH=CH2 D1-81a
CH2S(O)2CH2CH=CH2 D1-82a
CH2S(O)2CH2CH=CH2 D1-84a
CH2S(O)2CH2CH=CH2 D1-85a
CH2S(O)2CH2CH=CH2 D1-87a
CH2S(O)2CH2CH=CH2 D1-92a
CH2S(O)2CH2CH=CH2 D1-93a
CH2S(O)2CH2CH=CH2 D1-95a
CH2S(O)2CH2CH=CH2 D1-96a
CH2S(O)2CH2CH=CH2 D1-98a
CH2S(O)2CH2CH=CH2 D1-108a
CH2S(O)2CH2CH=CH2 D1-108b(Z=2-Cl)
CH2S(O)2CH2CH=CH2 D1-108b(Z=3-Me)
CH2S(O)2CH2CH=CH2 D1-108b(Z=4-OMe)
CH2S(O)2CH2CH=CH2 D1-108b(Z=2-SMe)
CH2S(O)2CH2CH=CH2 D1-108b(Z=3-CF3)
CH2S(O)2CH2CH=CH2 D1-108b(Z=4-OCF3)
CH2S(O)2CH2CH=CH2 D1-108b(Z=2-SCF3)
CH2S(O)2CH2CH=CH2 C(O)Me
CH2S(O)2CH2CH=CH2 C(O)CF3
CH2S(O)2CH2CH=CH2 C(O)OMe
CH(Me)SCH2CH=CH2 Me
CH(Me)SCH2CH=CH2 Et
CH(Me)SCH2CH=CH2 Pr-n
CH(Me)SCH2CH=CH2 Pr-i
CH(Me)SCH2CH=CH2 Pr-c
CH(Me)SCH2CH=CH2 Bu-n
CH(Me)SCH2CH=CH2 Bu-i
CH(Me)SCH2CH=CH2 Bu-c
CH(Me)SCH2CH=CH2 Bu-s
CH(Me)SCH2CH=CH2 Bu-t
CH(Me)SCH2CH=CH2 Pen-n
CH(Me)SCH2CH=CH2 Pen-c
CH(Me)SCH2CH=CH2 Hex-n
CH(Me)SCH2CH=CH2 Hex-c
CH(Me)SCH2CH=CH2 CH2Pr-c
CH(Me)SCH2CH=CH2 CH2Bu-c
CH(Me)SCH2CH=CH2 CH2Pen-c
CH(Me)SCH2CH=CH2 CH2Hex-c
CH(Me)SCH2CH=CH2 CH2CH=CH2
CH(Me)SCH2CH=CH2 CH2CH=C(Cl)2
CH(Me)SCH2CH=CH2 CH2C≡CH
CH(Me)SCH2CH=CH2 CH2CN
CH(Me)SCH2CH=CH2 CH2CF3
CH(Me)SCH2CH=CH2 CH2OMe
CH(Me)SCH2CH=CH2 CH2OCF3
CH(Me)SCH2CH=CH2 CH2SMe
CH(Me)SCH2CH=CH2 CH2S(O)Me
CH(Me)SCH2CH=CH2 CH2S(O)2Me
CH(Me)SCH2CH=CH2 CH2SCF3
CH(Me)SCH2CH=CH2 CH2S(O)CF3
CH(Me)SCH2CH=CH2 CH2S(O)2CF3
CH(Me)SCH2CH=CH2 CH2CH(OMe)2
CH(Me)SCH2CH=CH2 CH2CH(SMe)2
CH(Me)SCH2CH=CH2 CH2C(O)Me
CH(Me)SCH2CH=CH2 CH2C(O)CF3
CH(Me)SCH2CH=CH2 CH2C(O)OMe
CH(Me)SCH2CH=CH2 CH2(D1-32a)
CH(Me)SCH2CH=CH2 CH2(D1-33a)
CH(Me)SCH2CH=CH2 CH2(D1-34a)
CH(Me)SCH2CH=CH2 CH2(D1-37a)
CH(Me)SCH2CH=CH2 CH2(D1-81a)
CH(Me)SCH2CH=CH2 CH2(D1-82a)
CH(Me)SCH2CH=CH2 CH2(D1-84a)
CH(Me)SCH2CH=CH2 CH2(D1-85a)
CH(Me)SCH2CH=CH2 CH2(D1-87a)
CH(Me)SCH2CH=CH2 CH2(D1-92a)
CH(Me)SCH2CH=CH2 CH2(D1-93a)
CH(Me)SCH2CH=CH2 CH2(D1-95a)
CH(Me)SCH2CH=CH2 CH2(D1-96a)
CH(Me)SCH2CH=CH2 CH2(D1-98a)
CH(Me)SCH2CH=CH2 CH2(D1-108a)
CH(Me)SCH2CH=CH2 CH2(D1-108b,Z=2-Cl)
CH(Me)SCH2CH=CH2 CH2(D1-108b,Z=3-Me)
CH(Me)SCH2CH=CH2 CH2(D1-108b,Z=4-OMe)
CH(Me)SCH2CH=CH2 CH2(D1-108b,Z=2-SMe)
CH(Me)SCH2CH=CH2 CH2(D1-108b,Z=3-CF3)
CH(Me)SCH2CH=CH2 CH2(D1-108b,Z=4-OCF3)
CH(Me)SCH2CH=CH2 CH2(D1-108b,Z=2-SCF3)
CH(Me)SCH2CH=CH2 CH2CH2CN
CH(Me)SCH2CH=CH2 CH2CH2CF3
CH(Me)SCH2CH=CH2 CH2CH2OMe
CH(Me)SCH2CH=CH2 CH2CH2SMe
CH(Me)SCH2CH=CH2 CH2CH2S(O)Me
CH(Me)SCH2CH=CH2 CH2CH2S(O)2Me
CH(Me)SCH2CH=CH2 D1-32a
CH(Me)SCH2CH=CH2 D1-33a
CH(Me)SCH2CH=CH2 D1-34a
CH(Me)SCH2CH=CH2 D1-37a
CH(Me)SCH2CH=CH2 D1-81a
CH(Me)SCH2CH=CH2 D1-82a
CH(Me)SCH2CH=CH2 D1-84a
CH(Me)SCH2CH=CH2 D1-85a
CH(Me)SCH2CH=CH2 D1-87a
CH(Me)SCH2CH=CH2 D1-92a
CH(Me)SCH2CH=CH2 D1-93a
CH(Me)SCH2CH=CH2 D1-95a
CH(Me)SCH2CH=CH2 D1-96a
CH(Me)SCH2CH=CH2 D1-98a
CH(Me)SCH2CH=CH2 D1-108a
CH(Me)SCH2CH=CH2 D1-108b(Z=2-Cl)
CH(Me)SCH2CH=CH2 D1-108b(Z=3-Me)
CH(Me)SCH2CH=CH2 D1-108b(Z=4-OMe)
CH(Me)SCH2CH=CH2 D1-108b(Z=2-SMe)
CH(Me)SCH2CH=CH2 D1-108b(Z=3-CF3)
CH(Me)SCH2CH=CH2 D1-108b(Z=4-OCF3)
CH(Me)SCH2CH=CH2 D1-108b(Z=2-SCF3)
CH(Me)SCH2CH=CH2 C(O)Me
CH(Me)SCH2CH=CH2 C(O)CF3
CH(Me)SCH2CH=CH2 C(O)OMe
CH(Me)S(O)CH2CH=CH2 Me
CH(Me)S(O)CH2CH=CH2 Et
CH(Me)S(O)CH2CH=CH2 Pr-n
CH(Me)S(O)CH2CH=CH2 Pr-i
CH(Me)S(O)CH2CH=CH2 Pr-c
CH(Me)S(O)CH2CH=CH2 Bu-n
CH(Me)S(O)CH2CH=CH2 Bu-i
CH(Me)S(O)CH2CH=CH2 Bu-c
CH(Me)S(O)CH2CH=CH2 Bu-s
CH(Me)S(O)CH2CH=CH2 Bu-t
CH(Me)S(O)CH2CH=CH2 Pen-n
CH(Me)S(O)CH2CH=CH2 Pen-c
CH(Me)S(O)CH2CH=CH2 Hex-n
CH(Me)S(O)CH2CH=CH2 Hex-c
CH(Me)S(O)CH2CH=CH2 CH2Pr-c
CH(Me)S(O)CH2CH=CH2 CH2Bu-c
CH(Me)S(O)CH2CH=CH2 CH2Pen-c
CH(Me)S(O)CH2CH=CH2 CH2Hex-c
CH(Me)S(O)CH2CH=CH2 CH2CH=CH2
CH(Me)S(O)CH2CH=CH2 CH2CH=C(Cl)2
CH(Me)S(O)CH2CH=CH2 CH2C≡CH
CH(Me)S(O)CH2CH=CH2 CH2CN
CH(Me)S(O)CH2CH=CH2 CH2CF3
CH(Me)S(O)CH2CH=CH2 CH2OMe
CH(Me)S(O)CH2CH=CH2 CH2OCF3
CH(Me)S(O)CH2CH=CH2 CH2SMe
CH(Me)S(O)CH2CH=CH2 CH2S(O)Me
CH(Me)S(O)CH2CH=CH2 CH2S(O)2Me
CH(Me)S(O)CH2CH=CH2 CH2SCF3
CH(Me)S(O)CH2CH=CH2 CH2S(O)CF3
CH(Me)S(O)CH2CH=CH2 CH2S(O)2CF3
CH(Me)S(O)CH2CH=CH2 CH2CH(OMe)2
CH(Me)S(O)CH2CH=CH2 CH2CH(SMe)2
CH(Me)S(O)CH2CH=CH2 CH2C(O)Me
CH(Me)S(O)CH2CH=CH2 CH2C(O)CF3
CH(Me)S(O)CH2CH=CH2 CH2C(O)OMe
CH(Me)S(O)CH2CH=CH2 CH2(D1-32a)
CH(Me)S(O)CH2CH=CH2 CH2(D1-33a)
CH(Me)S(O)CH2CH=CH2 CH2(D1-34a)
CH(Me)S(O)CH2CH=CH2 CH2(D1-37a)
CH(Me)S(O)CH2CH=CH2 CH2(D1-81a)
CH(Me)S(O)CH2CH=CH2 CH2(D1-82a)
CH(Me)S(O)CH2CH=CH2 CH2(D1-84a)
CH(Me)S(O)CH2CH=CH2 CH2(D1-85a)
CH(Me)S(O)CH2CH=CH2 CH2(D1-87a)
CH(Me)S(O)CH2CH=CH2 CH2(D1-92a)
CH(Me)S(O)CH2CH=CH2 CH2(D1-93a)
CH(Me)S(O)CH2CH=CH2 CH2(D1-95a)
CH(Me)S(O)CH2CH=CH2 CH2(D1-96a)
CH(Me)S(O)CH2CH=CH2 CH2(D1-98a)
CH(Me)S(O)CH2CH=CH2 CH2(D1-108a)
CH(Me)S(O)CH2CH=CH2 CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)CH2CH=CH2 CH2(D1-108b,Z=3-Me)
CH(Me)S(O)CH2CH=CH2 CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)CH2CH=CH2 CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)CH2CH=CH2 CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)CH2CH=CH2 CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)CH2CH=CH2 CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)CH2CH=CH2 CH2CH2CN
CH(Me)S(O)CH2CH=CH2 CH2CH2CF3
CH(Me)S(O)CH2CH=CH2 CH2CH2OMe
CH(Me)S(O)CH2CH=CH2 CH2CH2SMe
CH(Me)S(O)CH2CH=CH2 CH2CH2S(O)Me
CH(Me)S(O)CH2CH=CH2 CH2CH2S(O)2Me
CH(Me)S(O)CH2CH=CH2 D1-32a
CH(Me)S(O)CH2CH=CH2 D1-33a
CH(Me)S(O)CH2CH=CH2 D1-34a
CH(Me)S(O)CH2CH=CH2 D1-37a
CH(Me)S(O)CH2CH=CH2 D1-81a
CH(Me)S(O)CH2CH=CH2 D1-82a
CH(Me)S(O)CH2CH=CH2 D1-84a
CH(Me)S(O)CH2CH=CH2 D1-85a
CH(Me)S(O)CH2CH=CH2 D1-87a
CH(Me)S(O)CH2CH=CH2 D1-92a
CH(Me)S(O)CH2CH=CH2 D1-93a
CH(Me)S(O)CH2CH=CH2 D1-95a
CH(Me)S(O)CH2CH=CH2 D1-96a
CH(Me)S(O)CH2CH=CH2 D1-98a
CH(Me)S(O)CH2CH=CH2 D1-108a
CH(Me)S(O)CH2CH=CH2 D1-108b(Z=2-Cl)
CH(Me)S(O)CH2CH=CH2 D1-108b(Z=3-Me)
CH(Me)S(O)CH2CH=CH2 D1-108b(Z=4-OMe)
CH(Me)S(O)CH2CH=CH2 D1-108b(Z=2-SMe)
CH(Me)S(O)CH2CH=CH2 D1-108b(Z=3-CF3)
CH(Me)S(O)CH2CH=CH2 D1-108b(Z=4-OCF3)
CH(Me)S(O)CH2CH=CH2 D1-108b(Z=2-SCF3)
CH(Me)S(O)CH2CH=CH2 C(O)Me
CH(Me)S(O)CH2CH=CH2 C(O)CF3
CH(Me)S(O)CH2CH=CH2 C(O)OMe
CH(Me)S(O)2CH2CH=CH2 Me
CH(Me)S(O)2CH2CH=CH2 Et
CH(Me)S(O)2CH2CH=CH2 Pr-n
CH(Me)S(O)2CH2CH=CH2 Pr-i
CH(Me)S(O)2CH2CH=CH2 Pr-c
CH(Me)S(O)2CH2CH=CH2 Bu-n
CH(Me)S(O)2CH2CH=CH2 Bu-i
CH(Me)S(O)2CH2CH=CH2 Bu-c
CH(Me)S(O)2CH2CH=CH2 Bu-s
CH(Me)S(O)2CH2CH=CH2 Bu-t
CH(Me)S(O)2CH2CH=CH2 Pen-n
CH(Me)S(O)2CH2CH=CH2 Pen-c
CH(Me)S(O)2CH2CH=CH2 Hex-n
CH(Me)S(O)2CH2CH=CH2 Hex-c
CH(Me)S(O)2CH2CH=CH2 CH2Pr-c
CH(Me)S(O)2CH2CH=CH2 CH2Bu-c
CH(Me)S(O)2CH2CH=CH2 CH2Pen-c
CH(Me)S(O)2CH2CH=CH2 CH2Hex-c
CH(Me)S(O)2CH2CH=CH2 CH2CH=CH2
CH(Me)S(O)2CH2CH=CH2 CH2CH=C(Cl)2
CH(Me)S(O)2CH2CH=CH2 CH2C≡CH
CH(Me)S(O)2CH2CH=CH2 CH2CN
CH(Me)S(O)2CH2CH=CH2 CH2CF3
CH(Me)S(O)2CH2CH=CH2 CH2OMe
CH(Me)S(O)2CH2CH=CH2 CH2OCF3
CH(Me)S(O)2CH2CH=CH2 CH2SMe
CH(Me)S(O)2CH2CH=CH2 CH2S(O)Me
CH(Me)S(O)2CH2CH=CH2 CH2S(O)2Me
CH(Me)S(O)2CH2CH=CH2 CH2SCF3
CH(Me)S(O)2CH2CH=CH2 CH2S(O)CF3
CH(Me)S(O)2CH2CH=CH2 CH2S(O)2CF3
CH(Me)S(O)2CH2CH=CH2 CH2CH(OMe)2
CH(Me)S(O)2CH2CH=CH2 CH2CH(SMe)2
CH(Me)S(O)2CH2CH=CH2 CH2C(O)Me
CH(Me)S(O)2CH2CH=CH2 CH2C(O)CF3
CH(Me)S(O)2CH2CH=CH2 CH2C(O)OMe
CH(Me)S(O)2CH2CH=CH2 CH2(D1-32a)
CH(Me)S(O)2CH2CH=CH2 CH2(D1-33a)
CH(Me)S(O)2CH2CH=CH2 CH2(D1-34a)
CH(Me)S(O)2CH2CH=CH2 CH2(D1-37a)
CH(Me)S(O)2CH2CH=CH2 CH2(D1-81a)
CH(Me)S(O)2CH2CH=CH2 CH2(D1-82a)
CH(Me)S(O)2CH2CH=CH2 CH2(D1-84a)
CH(Me)S(O)2CH2CH=CH2 CH2(D1-85a)
CH(Me)S(O)2CH2CH=CH2 CH2(D1-87a)
CH(Me)S(O)2CH2CH=CH2 CH2(D1-92a)
CH(Me)S(O)2CH2CH=CH2 CH2(D1-93a)
CH(Me)S(O)2CH2CH=CH2 CH2(D1-95a)
CH(Me)S(O)2CH2CH=CH2 CH2(D1-96a)
CH(Me)S(O)2CH2CH=CH2 CH2(D1-98a)
CH(Me)S(O)2CH2CH=CH2 CH2(D1-108a)
CH(Me)S(O)2CH2CH=CH2 CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)2CH2CH=CH2 CH2(D1-108b,Z=3-Me)
CH(Me)S(O)2CH2CH=CH2 CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)2CH2CH=CH2 CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)2CH2CH=CH2 CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)2CH2CH=CH2 CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)2CH2CH=CH2 CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)2CH2CH=CH2 CH2CH2CN
CH(Me)S(O)2CH2CH=CH2 CH2CH2CF3
CH(Me)S(O)2CH2CH=CH2 CH2CH2OMe
CH(Me)S(O)2CH2CH=CH2 CH2CH2SMe
CH(Me)S(O)2CH2CH=CH2 CH2CH2S(O)Me
CH(Me)S(O)2CH2CH=CH2 CH2CH2S(O)2Me
CH(Me)S(O)2CH2CH=CH2 D1-32a
CH(Me)S(O)2CH2CH=CH2 D1-33a
CH(Me)S(O)2CH2CH=CH2 D1-34a
CH(Me)S(O)2CH2CH=CH2 D1-37a
CH(Me)S(O)2CH2CH=CH2 D1-81a
CH(Me)S(O)2CH2CH=CH2 D1-82a
CH(Me)S(O)2CH2CH=CH2 D1-84a
CH(Me)S(O)2CH2CH=CH2 D1-85a
CH(Me)S(O)2CH2CH=CH2 D1-87a
CH(Me)S(O)2CH2CH=CH2 D1-92a
CH(Me)S(O)2CH2CH=CH2 D1-93a
CH(Me)S(O)2CH2CH=CH2 D1-95a
CH(Me)S(O)2CH2CH=CH2 D1-96a
CH(Me)S(O)2CH2CH=CH2 D1-98a
CH(Me)S(O)2CH2CH=CH2 D1-108a
CH(Me)S(O)2CH2CH=CH2 D1-108b(Z=2-Cl)
CH(Me)S(O)2CH2CH=CH2 D1-108b(Z=3-Me)
CH(Me)S(O)2CH2CH=CH2 D1-108b(Z=4-OMe)
CH(Me)S(O)2CH2CH=CH2 D1-108b(Z=2-SMe)
CH(Me)S(O)2CH2CH=CH2 D1-108b(Z=3-CF3)
CH(Me)S(O)2CH2CH=CH2 D1-108b(Z=4-OCF3)
CH(Me)S(O)2CH2CH=CH2 D1-108b(Z=2-SCF3)
CH(Me)S(O)2CH2CH=CH2 C(O)Me
CH(Me)S(O)2CH2CH=CH2 C(O)CF3
CH(Me)S(O)2CH2CH=CH2 C(O)OMe
CH(Et)SCH2CH=CH2 Me
CH(Et)SCH2CH=CH2 Et
CH(Et)SCH2CH=CH2 Pr-n
CH(Et)SCH2CH=CH2 Pr-i
CH(Et)SCH2CH=CH2 Pr-c
CH(Et)SCH2CH=CH2 Bu-n
CH(Et)SCH2CH=CH2 Bu-i
CH(Et)SCH2CH=CH2 Bu-c
CH(Et)SCH2CH=CH2 Bu-s
CH(Et)SCH2CH=CH2 Bu-t
CH(Et)SCH2CH=CH2 Pen-n
CH(Et)SCH2CH=CH2 Pen-c
CH(Et)SCH2CH=CH2 Hex-n
CH(Et)SCH2CH=CH2 Hex-c
CH(Et)SCH2CH=CH2 CH2Pr-c
CH(Et)SCH2CH=CH2 CH2Bu-c
CH(Et)SCH2CH=CH2 CH2Pen-c
CH(Et)SCH2CH=CH2 CH2Hex-c
CH(Et)SCH2CH=CH2 CH2CH=CH2
CH(Et)SCH2CH=CH2 CH2CH=C(Cl)2
CH(Et)SCH2CH=CH2 CH2C≡CH
CH(Et)SCH2CH=CH2 CH2CN
CH(Et)SCH2CH=CH2 CH2CF3
CH(Et)SCH2CH=CH2 CH2OMe
CH(Et)SCH2CH=CH2 CH2OCF3
CH(Et)SCH2CH=CH2 CH2SMe
CH(Et)SCH2CH=CH2 CH2S(O)Me
CH(Et)SCH2CH=CH2 CH2S(O)2Me
CH(Et)SCH2CH=CH2 CH2SCF3
CH(Et)SCH2CH=CH2 CH2S(O)CF3
CH(Et)SCH2CH=CH2 CH2S(O)2CF3
CH(Et)SCH2CH=CH2 CH2CH(OMe)2
CH(Et)SCH2CH=CH2 CH2CH(SMe)2
CH(Et)SCH2CH=CH2 CH2C(O)Me
CH(Et)SCH2CH=CH2 CH2C(O)CF3
CH(Et)SCH2CH=CH2 CH2C(O)OMe
CH(Et)SCH2CH=CH2 CH2(D1-32a)
CH(Et)SCH2CH=CH2 CH2(D1-33a)
CH(Et)SCH2CH=CH2 CH2(D1-34a)
CH(Et)SCH2CH=CH2 CH2(D1-37a)
CH(Et)SCH2CH=CH2 CH2(D1-81a)
CH(Et)SCH2CH=CH2 CH2(D1-82a)
CH(Et)SCH2CH=CH2 CH2(D1-84a)
CH(Et)SCH2CH=CH2 CH2(D1-85a)
CH(Et)SCH2CH=CH2 CH2(D1-87a)
CH(Et)SCH2CH=CH2 CH2(D1-92a)
CH(Et)SCH2CH=CH2 CH2(D1-93a)
CH(Et)SCH2CH=CH2 CH2(D1-95a)
CH(Et)SCH2CH=CH2 CH2(D1-96a)
CH(Et)SCH2CH=CH2 CH2(D1-98a)
CH(Et)SCH2CH=CH2 CH2(D1-108a)
CH(Et)SCH2CH=CH2 CH2(D1-108b,Z=2-Cl)
CH(Et)SCH2CH=CH2 CH2(D1-108b,Z=3-Me)
CH(Et)SCH2CH=CH2 CH2(D1-108b,Z=4-OMe)
CH(Et)SCH2CH=CH2 CH2(D1-108b,Z=2-SMe)
CH(Et)SCH2CH=CH2 CH2(D1-108b,Z=3-CF3)
CH(Et)SCH2CH=CH2 CH2(D1-108b,Z=4-OCF3)
CH(Et)SCH2CH=CH2 CH2(D1-108b,Z=2-SCF3)
CH(Et)SCH2CH=CH2 CH2CH2CN
CH(Et)SCH2CH=CH2 CH2CH2CF3
CH(Et)SCH2CH=CH2 CH2CH2OMe
CH(Et)SCH2CH=CH2 CH2CH2SMe
CH(Et)SCH2CH=CH2 CH2CH2S(O)Me
CH(Et)SCH2CH=CH2 CH2CH2S(O)2Me
CH(Et)SCH2CH=CH2 D1-32a
CH(Et)SCH2CH=CH2 D1-33a
CH(Et)SCH2CH=CH2 D1-34a
CH(Et)SCH2CH=CH2 D1-37a
CH(Et)SCH2CH=CH2 D1-81a
CH(Et)SCH2CH=CH2 D1-82a
CH(Et)SCH2CH=CH2 D1-84a
CH(Et)SCH2CH=CH2 D1-85a
CH(Et)SCH2CH=CH2 D1-87a
CH(Et)SCH2CH=CH2 D1-92a
CH(Et)SCH2CH=CH2 D1-93a
CH(Et)SCH2CH=CH2 D1-95a
CH(Et)SCH2CH=CH2 D1-96a
CH(Et)SCH2CH=CH2 D1-98a
CH(Et)SCH2CH=CH2 D1-108a
CH(Et)SCH2CH=CH2 D1-108b(Z=2-Cl)
CH(Et)SCH2CH=CH2 D1-108b(Z=3-Me)
CH(Et)SCH2CH=CH2 D1-108b(Z=4-OMe)
CH(Et)SCH2CH=CH2 D1-108b(Z=2-SMe)
CH(Et)SCH2CH=CH2 D1-108b(Z=3-CF3)
CH(Et)SCH2CH=CH2 D1-108b(Z=4-OCF3)
CH(Et)SCH2CH=CH2 D1-108b(Z=2-SCF3)
CH(Et)SCH2CH=CH2 C(O)Me
CH(Et)SCH2CH=CH2 C(O)CF3
CH(Et)SCH2CH=CH2 C(O)OMe
CH(Et)S(O)CH2CH=CH2 Me
CH(Et)S(O)CH2CH=CH2 Et
CH(Et)S(O)CH2CH=CH2 Pr-n
CH(Et)S(O)CH2CH=CH2 Pr-i
CH(Et)S(O)CH2CH=CH2 Pr-c
CH(Et)S(O)CH2CH=CH2 Bu-n
CH(Et)S(O)CH2CH=CH2 Bu-i
CH(Et)S(O)CH2CH=CH2 Bu-c
CH(Et)S(O)CH2CH=CH2 Bu-s
CH(Et)S(O)CH2CH=CH2 Bu-t
CH(Et)S(O)CH2CH=CH2 Pen-n
CH(Et)S(O)CH2CH=CH2 Pen-c
CH(Et)S(O)CH2CH=CH2 Hex-n
CH(Et)S(O)CH2CH=CH2 Hex-c
CH(Et)S(O)CH2CH=CH2 CH2Pr-c
CH(Et)S(O)CH2CH=CH2 CH2Bu-c
CH(Et)S(O)CH2CH=CH2 CH2Pen-c
CH(Et)S(O)CH2CH=CH2 CH2Hex-c
CH(Et)S(O)CH2CH=CH2 CH2CH=CH2
CH(Et)S(O)CH2CH=CH2 CH2CH=C(Cl)2
CH(Et)S(O)CH2CH=CH2 CH2C≡CH
CH(Et)S(O)CH2CH=CH2 CH2CN
CH(Et)S(O)CH2CH=CH2 CH2CF3
CH(Et)S(O)CH2CH=CH2 CH2OMe
CH(Et)S(O)CH2CH=CH2 CH2OCF3
CH(Et)S(O)CH2CH=CH2 CH2SMe
CH(Et)S(O)CH2CH=CH2 CH2S(O)Me
CH(Et)S(O)CH2CH=CH2 CH2S(O)2Me
CH(Et)S(O)CH2CH=CH2 CH2SCF3
CH(Et)S(O)CH2CH=CH2 CH2S(O)CF3
CH(Et)S(O)CH2CH=CH2 CH2S(O)2CF3
CH(Et)S(O)CH2CH=CH2 CH2CH(OMe)2
CH(Et)S(O)CH2CH=CH2 CH2CH(SMe)2
CH(Et)S(O)CH2CH=CH2 CH2C(O)Me
CH(Et)S(O)CH2CH=CH2 CH2C(O)CF3
CH(Et)S(O)CH2CH=CH2 CH2C(O)OMe
CH(Et)S(O)CH2CH=CH2 CH2(D1-32a)
CH(Et)S(O)CH2CH=CH2 CH2(D1-33a)
CH(Et)S(O)CH2CH=CH2 CH2(D1-34a)
CH(Et)S(O)CH2CH=CH2 CH2(D1-37a)
CH(Et)S(O)CH2CH=CH2 CH2(D1-81a)
CH(Et)S(O)CH2CH=CH2 CH2(D1-82a)
CH(Et)S(O)CH2CH=CH2 CH2(D1-84a)
CH(Et)S(O)CH2CH=CH2 CH2(D1-85a)
CH(Et)S(O)CH2CH=CH2 CH2(D1-87a)
CH(Et)S(O)CH2CH=CH2 CH2(D1-92a)
CH(Et)S(O)CH2CH=CH2 CH2(D1-93a)
CH(Et)S(O)CH2CH=CH2 CH2(D1-95a)
CH(Et)S(O)CH2CH=CH2 CH2(D1-96a)
CH(Et)S(O)CH2CH=CH2 CH2(D1-98a)
CH(Et)S(O)CH2CH=CH2 CH2(D1-108a)
CH(Et)S(O)CH2CH=CH2 CH2(D1-108b,Z=2-Cl)
CH(Et)S(O)CH2CH=CH2 CH2(D1-108b,Z=3-Me)
CH(Et)S(O)CH2CH=CH2 CH2(D1-108b,Z=4-OMe)
CH(Et)S(O)CH2CH=CH2 CH2(D1-108b,Z=2-SMe)
CH(Et)S(O)CH2CH=CH2 CH2(D1-108b,Z=3-CF3)
CH(Et)S(O)CH2CH=CH2 CH2(D1-108b,Z=4-OCF3)
CH(Et)S(O)CH2CH=CH2 CH2(D1-108b,Z=2-SCF3)
CH(Et)S(O)CH2CH=CH2 CH2CH2CN
CH(Et)S(O)CH2CH=CH2 CH2CH2CF3
CH(Et)S(O)CH2CH=CH2 CH2CH2OMe
CH(Et)S(O)CH2CH=CH2 CH2CH2SMe
CH(Et)S(O)CH2CH=CH2 CH2CH2S(O)Me
CH(Et)S(O)CH2CH=CH2 CH2CH2S(O)2Me
CH(Et)S(O)CH2CH=CH2 D1-32a
CH(Et)S(O)CH2CH=CH2 D1-33a
CH(Et)S(O)CH2CH=CH2 D1-34a
CH(Et)S(O)CH2CH=CH2 D1-37a
CH(Et)S(O)CH2CH=CH2 D1-81a
CH(Et)S(O)CH2CH=CH2 D1-82a
CH(Et)S(O)CH2CH=CH2 D1-84a
CH(Et)S(O)CH2CH=CH2 D1-85a
CH(Et)S(O)CH2CH=CH2 D1-87a
CH(Et)S(O)CH2CH=CH2 D1-92a
CH(Et)S(O)CH2CH=CH2 D1-93a
CH(Et)S(O)CH2CH=CH2 D1-95a
CH(Et)S(O)CH2CH=CH2 D1-96a
CH(Et)S(O)CH2CH=CH2 D1-98a
CH(Et)S(O)CH2CH=CH2 D1-108a
CH(Et)S(O)CH2CH=CH2 D1-108b(Z=2-Cl)
CH(Et)S(O)CH2CH=CH2 D1-108b(Z=3-Me)
CH(Et)S(O)CH2CH=CH2 D1-108b(Z=4-OMe)
CH(Et)S(O)CH2CH=CH2 D1-108b(Z=2-SMe)
CH(Et)S(O)CH2CH=CH2 D1-108b(Z=3-CF3)
CH(Et)S(O)CH2CH=CH2 D1-108b(Z=4-OCF3)
CH(Et)S(O)CH2CH=CH2 D1-108b(Z=2-SCF3)
CH(Et)S(O)CH2CH=CH2 C(O)Me
CH(Et)S(O)CH2CH=CH2 C(O)CF3
CH(Et)S(O)CH2CH=CH2 C(O)OMe
CH(Et)S(O)2CH2CH=CH2 Me
CH(Et)S(O)2CH2CH=CH2 Et
CH(Et)S(O)2CH2CH=CH2 Pr-n
CH(Et)S(O)2CH2CH=CH2 Pr-i
CH(Et)S(O)2CH2CH=CH2 Pr-c
CH(Et)S(O)2CH2CH=CH2 Bu-n
CH(Et)S(O)2CH2CH=CH2 Bu-i
CH(Et)S(O)2CH2CH=CH2 Bu-c
CH(Et)S(O)2CH2CH=CH2 Bu-s
CH(Et)S(O)2CH2CH=CH2 Bu-t
CH(Et)S(O)2CH2CH=CH2 Pen-n
CH(Et)S(O)2CH2CH=CH2 Pen-c
CH(Et)S(O)2CH2CH=CH2 Hex-n
CH(Et)S(O)2CH2CH=CH2 Hex-c
CH(Et)S(O)2CH2CH=CH2 CH2Pr-c
CH(Et)S(O)2CH2CH=CH2 CH2Bu-c
CH(Et)S(O)2CH2CH=CH2 CH2Pen-c
CH(Et)S(O)2CH2CH=CH2 CH2Hex-c
CH(Et)S(O)2CH2CH=CH2 CH2CH=CH2
CH(Et)S(O)2CH2CH=CH2 CH2CH=C(Cl)2
CH(Et)S(O)2CH2CH=CH2 CH2C≡CH
CH(Et)S(O)2CH2CH=CH2 CH2CN
CH(Et)S(O)2CH2CH=CH2 CH2CF3
CH(Et)S(O)2CH2CH=CH2 CH2OMe
CH(Et)S(O)2CH2CH=CH2 CH2OCF3
CH(Et)S(O)2CH2CH=CH2 CH2SMe
CH(Et)S(O)2CH2CH=CH2 CH2S(O)Me
CH(Et)S(O)2CH2CH=CH2 CH2S(O)2Me
CH(Et)S(O)2CH2CH=CH2 CH2SCF3
CH(Et)S(O)2CH2CH=CH2 CH2S(O)CF3
CH(Et)S(O)2CH2CH=CH2 CH2S(O)2CF3
CH(Et)S(O)2CH2CH=CH2 CH2CH(OMe)2
CH(Et)S(O)2CH2CH=CH2 CH2CH(SMe)2
CH(Et)S(O)2CH2CH=CH2 CH2C(O)Me
CH(Et)S(O)2CH2CH=CH2 CH2C(O)CF3
CH(Et)S(O)2CH2CH=CH2 CH2C(O)OMe
CH(Et)S(O)2CH2CH=CH2 CH2(D1-32a)
CH(Et)S(O)2CH2CH=CH2 CH2(D1-33a)
CH(Et)S(O)2CH2CH=CH2 CH2(D1-34a)
CH(Et)S(O)2CH2CH=CH2 CH2(D1-37a)
CH(Et)S(O)2CH2CH=CH2 CH2(D1-81a)
CH(Et)S(O)2CH2CH=CH2 CH2(D1-82a)
CH(Et)S(O)2CH2CH=CH2 CH2(D1-84a)
CH(Et)S(O)2CH2CH=CH2 CH2(D1-85a)
CH(Et)S(O)2CH2CH=CH2 CH2(D1-87a)
CH(Et)S(O)2CH2CH=CH2 CH2(D1-92a)
CH(Et)S(O)2CH2CH=CH2 CH2(D1-93a)
CH(Et)S(O)2CH2CH=CH2 CH2(D1-95a)
CH(Et)S(O)2CH2CH=CH2 CH2(D1-96a)
CH(Et)S(O)2CH2CH=CH2 CH2(D1-98a)
CH(Et)S(O)2CH2CH=CH2 CH2(D1-108a)
CH(Et)S(O)2CH2CH=CH2 CH2(D1-108b,Z=2-Cl)
CH(Et)S(O)2CH2CH=CH2 CH2(D1-108b,Z=3-Me)
CH(Et)S(O)2CH2CH=CH2 CH2(D1-108b,Z=4-OMe)
CH(Et)S(O)2CH2CH=CH2 CH2(D1-108b,Z=2-SMe)
CH(Et)S(O)2CH2CH=CH2 CH2(D1-108b,Z=3-CF3)
CH(Et)S(O)2CH2CH=CH2 CH2(D1-108b,Z=4-OCF3)
CH(Et)S(O)2CH2CH=CH2 CH2(D1-108b,Z=2-SCF3)
CH(Et)S(O)2CH2CH=CH2 CH2CH2CN
CH(Et)S(O)2CH2CH=CH2 CH2CH2CF3
CH(Et)S(O)2CH2CH=CH2 CH2CH2OMe
CH(Et)S(O)2CH2CH=CH2 CH2CH2SMe
CH(Et)S(O)2CH2CH=CH2 CH2CH2S(O)Me
CH(Et)S(O)2CH2CH=CH2 CH2CH2S(O)2Me
CH(Et)S(O)2CH2CH=CH2 D1-32a
CH(Et)S(O)2CH2CH=CH2 D1-33a
CH(Et)S(O)2CH2CH=CH2 D1-34a
CH(Et)S(O)2CH2CH=CH2 D1-37a
CH(Et)S(O)2CH2CH=CH2 D1-81a
CH(Et)S(O)2CH2CH=CH2 D1-82a
CH(Et)S(O)2CH2CH=CH2 D1-84a
CH(Et)S(O)2CH2CH=CH2 D1-85a
CH(Et)S(O)2CH2CH=CH2 D1-87a
CH(Et)S(O)2CH2CH=CH2 D1-92a
CH(Et)S(O)2CH2CH=CH2 D1-93a
CH(Et)S(O)2CH2CH=CH2 D1-95a
CH(Et)S(O)2CH2CH=CH2 D1-96a
CH(Et)S(O)2CH2CH=CH2 D1-98a
CH(Et)S(O)2CH2CH=CH2 D1-108a
CH(Et)S(O)2CH2CH=CH2 D1-108b(Z=2-Cl)
CH(Et)S(O)2CH2CH=CH2 D1-108b(Z=3-Me)
CH(Et)S(O)2CH2CH=CH2 D1-108b(Z=4-OMe)
CH(Et)S(O)2CH2CH=CH2 D1-108b(Z=2-SMe)
CH(Et)S(O)2CH2CH=CH2 D1-108b(Z=3-CF3)
CH(Et)S(O)2CH2CH=CH2 D1-108b(Z=4-OCF3)
CH(Et)S(O)2CH2CH=CH2 D1-108b(Z=2-SCF3)
CH(Et)S(O)2CH2CH=CH2 C(O)Me
CH(Et)S(O)2CH2CH=CH2 C(O)CF3
CH(Et)S(O)2CH2CH=CH2 C(O)OMe
CH2SCH2CH2OMe Me
CH2SCH2CH2OMe Et
CH2SCH2CH2OMe Pr-n
CH2SCH2CH2OMe Pr-i
CH2SCH2CH2OMe Pr-c
CH2SCH2CH2OMe Bu-n
CH2SCH2CH2OMe Bu-i
CH2SCH2CH2OMe Bu-c
CH2SCH2CH2OMe Bu-s
CH2SCH2CH2OMe Bu-t
CH2SCH2CH2OMe Pen-n
CH2SCH2CH2OMe Pen-c
CH2SCH2CH2OMe Hex-n
CH2SCH2CH2OMe Hex-c
CH2SCH2CH2OMe CH2Pr-c
CH2SCH2CH2OMe CH2Bu-c
CH2SCH2CH2OMe CH2Pen-c
CH2SCH2CH2OMe CH2Hex-c
CH2SCH2CH2OMe CH2CH=CH2
CH2SCH2CH2OMe CH2CH=C(Cl)2
CH2SCH2CH2OMe CH2C≡CH
CH2SCH2CH2OMe CH2CN
CH2SCH2CH2OMe CH2CF3
CH2SCH2CH2OMe CH2OMe
CH2SCH2CH2OMe CH2OCF3
CH2SCH2CH2OMe CH2SMe
CH2SCH2CH2OMe CH2S(O)Me
CH2SCH2CH2OMe CH2S(O)2Me
CH2SCH2CH2OMe CH2SCF3
CH2SCH2CH2OMe CH2S(O)CF3
CH2SCH2CH2OMe CH2S(O)2CF3
CH2SCH2CH2OMe CH2CH(OMe)2
CH2SCH2CH2OMe CH2CH(SMe)2
CH2SCH2CH2OMe CH2C(O)Me
CH2SCH2CH2OMe CH2C(O)CF3
CH2SCH2CH2OMe CH2C(O)OMe
CH2SCH2CH2OMe CH2(D1-32a)
CH2SCH2CH2OMe CH2(D1-33a)
CH2SCH2CH2OMe CH2(D1-34a)
CH2SCH2CH2OMe CH2(D1-37a)
CH2SCH2CH2OMe CH2(D1-81a)
CH2SCH2CH2OMe CH2(D1-82a)
CH2SCH2CH2OMe CH2(D1-84a)
CH2SCH2CH2OMe CH2(D1-85a)
CH2SCH2CH2OMe CH2(D1-87a)
CH2SCH2CH2OMe CH2(D1-92a)
CH2SCH2CH2OMe CH2(D1-93a)
CH2SCH2CH2OMe CH2(D1-95a)
CH2SCH2CH2OMe CH2(D1-96a)
CH2SCH2CH2OMe CH2(D1-98a)
CH2SCH2CH2OMe CH2(D1-108a)
CH2SCH2CH2OMe CH2(D1-108b,Z=2-Cl)
CH2SCH2CH2OMe CH2(D1-108b,Z=3-Me)
CH2SCH2CH2OMe CH2(D1-108b,Z=4-OMe)
CH2SCH2CH2OMe CH2(D1-108b,Z=2-SMe)
CH2SCH2CH2OMe CH2(D1-108b,Z=3-CF3)
CH2SCH2CH2OMe CH2(D1-108b,Z=4-OCF3)
CH2SCH2CH2OMe CH2(D1-108b,Z=2-SCF3)
CH2SCH2CH2OMe CH2CH2CN
CH2SCH2CH2OMe CH2CH2CF3
CH2SCH2CH2OMe CH2CH2OMe
CH2SCH2CH2OMe CH2CH2SMe
CH2SCH2CH2OMe CH2CH2S(O)Me
CH2SCH2CH2OMe CH2CH2S(O)2Me
CH2SCH2CH2OMe D1-32a
CH2SCH2CH2OMe D1-33a
CH2SCH2CH2OMe D1-34a
CH2SCH2CH2OMe D1-37a
CH2SCH2CH2OMe D1-81a
CH2SCH2CH2OMe D1-82a
CH2SCH2CH2OMe D1-84a
CH2SCH2CH2OMe D1-85a
CH2SCH2CH2OMe D1-87a
CH2SCH2CH2OMe D1-92a
CH2SCH2CH2OMe D1-93a
CH2SCH2CH2OMe D1-95a
CH2SCH2CH2OMe D1-96a
CH2SCH2CH2OMe D1-98a
CH2SCH2CH2OMe D1-108a
CH2SCH2CH2OMe D1-108b(Z=2-Cl)
CH2SCH2CH2OMe D1-108b(Z=3-Me)
CH2SCH2CH2OMe D1-108b(Z=4-OMe)
CH2SCH2CH2OMe D1-108b(Z=2-SMe)
CH2SCH2CH2OMe D1-108b(Z=3-CF3)
CH2SCH2CH2OMe D1-108b(Z=4-OCF3)
CH2SCH2CH2OMe D1-108b(Z=2-SCF3)
CH2SCH2CH2OMe C(O)Me
CH2SCH2CH2OMe C(O)CF3
CH2SCH2CH2OMe C(O)OMe
CH2S(O)CH2CH2OMe Me
CH2S(O)CH2CH2OMe Et
CH2S(O)CH2CH2OMe Pr-n
CH2S(O)CH2CH2OMe Pr-i
CH2S(O)CH2CH2OMe Pr-c
CH2S(O)CH2CH2OMe Bu-n
CH2S(O)CH2CH2OMe Bu-i
CH2S(O)CH2CH2OMe Bu-c
CH2S(O)CH2CH2OMe Bu-s
CH2S(O)CH2CH2OMe Bu-t
CH2S(O)CH2CH2OMe Pen-n
CH2S(O)CH2CH2OMe Pen-c
CH2S(O)CH2CH2OMe Hex-n
CH2S(O)CH2CH2OMe Hex-c
CH2S(O)CH2CH2OMe CH2Pr-c
CH2S(O)CH2CH2OMe CH2Bu-c
CH2S(O)CH2CH2OMe CH2Pen-c
CH2S(O)CH2CH2OMe CH2Hex-c
CH2S(O)CH2CH2OMe CH2CH=CH2
CH2S(O)CH2CH2OMe CH2CH=C(Cl)2
CH2S(O)CH2CH2OMe CH2C≡CH
CH2S(O)CH2CH2OMe CH2CN
CH2S(O)CH2CH2OMe CH2CF3
CH2S(O)CH2CH2OMe CH2OMe
CH2S(O)CH2CH2OMe CH2OCF3
CH2S(O)CH2CH2OMe CH2SMe
CH2S(O)CH2CH2OMe CH2S(O)Me
CH2S(O)CH2CH2OMe CH2S(O)2Me
CH2S(O)CH2CH2OMe CH2SCF3
CH2S(O)CH2CH2OMe CH2S(O)CF3
CH2S(O)CH2CH2OMe CH2S(O)2CF3
CH2S(O)CH2CH2OMe CH2CH(OMe)2
CH2S(O)CH2CH2OMe CH2CH(SMe)2
CH2S(O)CH2CH2OMe CH2C(O)Me
CH2S(O)CH2CH2OMe CH2C(O)CF3
CH2S(O)CH2CH2OMe CH2C(O)OMe
CH2S(O)CH2CH2OMe CH2(D1-32a)
CH2S(O)CH2CH2OMe CH2(D1-33a)
CH2S(O)CH2CH2OMe CH2(D1-34a)
CH2S(O)CH2CH2OMe CH2(D1-37a)
CH2S(O)CH2CH2OMe CH2(D1-81a)
CH2S(O)CH2CH2OMe CH2(D1-82a)
CH2S(O)CH2CH2OMe CH2(D1-84a)
CH2S(O)CH2CH2OMe CH2(D1-85a)
CH2S(O)CH2CH2OMe CH2(D1-87a)
CH2S(O)CH2CH2OMe CH2(D1-92a)
CH2S(O)CH2CH2OMe CH2(D1-93a)
CH2S(O)CH2CH2OMe CH2(D1-95a)
CH2S(O)CH2CH2OMe CH2(D1-96a)
CH2S(O)CH2CH2OMe CH2(D1-98a)
CH2S(O)CH2CH2OMe CH2(D1-108a)
CH2S(O)CH2CH2OMe CH2(D1-108b,Z=2-Cl)
CH2S(O)CH2CH2OMe CH2(D1-108b,Z=3-Me)
CH2S(O)CH2CH2OMe CH2(D1-108b,Z=4-OMe)
CH2S(O)CH2CH2OMe CH2(D1-108b,Z=2-SMe)
CH2S(O)CH2CH2OMe CH2(D1-108b,Z=3-CF3)
CH2S(O)CH2CH2OMe CH2(D1-108b,Z=4-OCF3)
CH2S(O)CH2CH2OMe CH2(D1-108b,Z=2-SCF3)
CH2S(O)CH2CH2OMe CH2CH2CN
CH2S(O)CH2CH2OMe CH2CH2CF3
CH2S(O)CH2CH2OMe CH2CH2OMe
CH2S(O)CH2CH2OMe CH2CH2SMe
CH2S(O)CH2CH2OMe CH2CH2S(O)Me
CH2S(O)CH2CH2OMe CH2CH2S(O)2Me
CH2S(O)CH2CH2OMe D1-32a
CH2S(O)CH2CH2OMe D1-33a
CH2S(O)CH2CH2OMe D1-34a
CH2S(O)CH2CH2OMe D1-37a
CH2S(O)CH2CH2OMe D1-81a
CH2S(O)CH2CH2OMe D1-82a
CH2S(O)CH2CH2OMe D1-84a
CH2S(O)CH2CH2OMe D1-85a
CH2S(O)CH2CH2OMe D1-87a
CH2S(O)CH2CH2OMe D1-92a
CH2S(O)CH2CH2OMe D1-93a
CH2S(O)CH2CH2OMe D1-95a
CH2S(O)CH2CH2OMe D1-96a
CH2S(O)CH2CH2OMe D1-98a
CH2S(O)CH2CH2OMe D1-108a
CH2S(O)CH2CH2OMe D1-108b(Z=2-Cl)
CH2S(O)CH2CH2OMe D1-108b(Z=3-Me)
CH2S(O)CH2CH2OMe D1-108b(Z=4-OMe)
CH2S(O)CH2CH2OMe D1-108b(Z=2-SMe)
CH2S(O)CH2CH2OMe D1-108b(Z=3-CF3)
CH2S(O)CH2CH2OMe D1-108b(Z=4-OCF3)
CH2S(O)CH2CH2OMe D1-108b(Z=2-SCF3)
CH2S(O)CH2CH2OMe C(O)Me
CH2S(O)CH2CH2OMe C(O)CF3
CH2S(O)CH2CH2OMe C(O)OMe
CH2S(O)2CH2CH2OMe Me
CH2S(O)2CH2CH2OMe Et
CH2S(O)2CH2CH2OMe Pr-n
CH2S(O)2CH2CH2OMe Pr-i
CH2S(O)2CH2CH2OMe Pr-c
CH2S(O)2CH2CH2OMe Bu-n
CH2S(O)2CH2CH2OMe Bu-i
CH2S(O)2CH2CH2OMe Bu-c
CH2S(O)2CH2CH2OMe Bu-s
CH2S(O)2CH2CH2OMe Bu-t
CH2S(O)2CH2CH2OMe Pen-n
CH2S(O)2CH2CH2OMe Pen-c
CH2S(O)2CH2CH2OMe Hex-n
CH2S(O)2CH2CH2OMe Hex-c
CH2S(O)2CH2CH2OMe CH2Pr-c
CH2S(O)2CH2CH2OMe CH2Bu-c
CH2S(O)2CH2CH2OMe CH2Pen-c
CH2S(O)2CH2CH2OMe CH2Hex-c
CH2S(O)2CH2CH2OMe CH2CH=CH2
CH2S(O)2CH2CH2OMe CH2CH=C(Cl)2
CH2S(O)2CH2CH2OMe CH2C≡CH
CH2S(O)2CH2CH2OMe CH2CN
CH2S(O)2CH2CH2OMe CH2CF3
CH2S(O)2CH2CH2OMe CH2OMe
CH2S(O)2CH2CH2OMe CH2OCF3
CH2S(O)2CH2CH2OMe CH2SMe
CH2S(O)2CH2CH2OMe CH2S(O)Me
CH2S(O)2CH2CH2OMe CH2S(O)2Me
CH2S(O)2CH2CH2OMe CH2SCF3
CH2S(O)2CH2CH2OMe CH2S(O)CF3
CH2S(O)2CH2CH2OMe CH2S(O)2CF3
CH2S(O)2CH2CH2OMe CH2CH(OMe)2
CH2S(O)2CH2CH2OMe CH2CH(SMe)2
CH2S(O)2CH2CH2OMe CH2C(O)Me
CH2S(O)2CH2CH2OMe CH2C(O)CF3
CH2S(O)2CH2CH2OMe CH2C(O)OMe
CH2S(O)2CH2CH2OMe CH2(D1-32a)
CH2S(O)2CH2CH2OMe CH2(D1-33a)
CH2S(O)2CH2CH2OMe CH2(D1-34a)
CH2S(O)2CH2CH2OMe CH2(D1-37a)
CH2S(O)2CH2CH2OMe CH2(D1-81a)
CH2S(O)2CH2CH2OMe CH2(D1-82a)
CH2S(O)2CH2CH2OMe CH2(D1-84a)
CH2S(O)2CH2CH2OMe CH2(D1-85a)
CH2S(O)2CH2CH2OMe CH2(D1-87a)
CH2S(O)2CH2CH2OMe CH2(D1-92a)
CH2S(O)2CH2CH2OMe CH2(D1-93a)
CH2S(O)2CH2CH2OMe CH2(D1-95a)
CH2S(O)2CH2CH2OMe CH2(D1-96a)
CH2S(O)2CH2CH2OMe CH2(D1-98a)
CH2S(O)2CH2CH2OMe CH2(D1-108a)
CH2S(O)2CH2CH2OMe CH2(D1-108b,Z=2-Cl)
CH2S(O)2CH2CH2OMe CH2(D1-108b,Z=3-Me)
CH2S(O)2CH2CH2OMe CH2(D1-108b,Z=4-OMe)
CH2S(O)2CH2CH2OMe CH2(D1-108b,Z=2-SMe)
CH2S(O)2CH2CH2OMe CH2(D1-108b,Z=3-CF3)
CH2S(O)2CH2CH2OMe CH2(D1-108b,Z=4-OCF3)
CH2S(O)2CH2CH2OMe CH2(D1-108b,Z=2-SCF3)
CH2S(O)2CH2CH2OMe CH2CH2CN
CH2S(O)2CH2CH2OMe CH2CH2CF3
CH2S(O)2CH2CH2OMe CH2CH2OMe
CH2S(O)2CH2CH2OMe CH2CH2SMe
CH2S(O)2CH2CH2OMe CH2CH2S(O)Me
CH2S(O)2CH2CH2OMe CH2CH2S(O)2Me
CH2S(O)2CH2CH2OMe D1-32a
CH2S(O)2CH2CH2OMe D1-33a
CH2S(O)2CH2CH2OMe D1-34a
CH2S(O)2CH2CH2OMe D1-37a
CH2S(O)2CH2CH2OMe D1-81a
CH2S(O)2CH2CH2OMe D1-82a
CH2S(O)2CH2CH2OMe D1-84a
CH2S(O)2CH2CH2OMe D1-85a
CH2S(O)2CH2CH2OMe D1-87a
CH2S(O)2CH2CH2OMe D1-92a
CH2S(O)2CH2CH2OMe D1-93a
CH2S(O)2CH2CH2OMe D1-95a
CH2S(O)2CH2CH2OMe D1-96a
CH2S(O)2CH2CH2OMe D1-98a
CH2S(O)2CH2CH2OMe D1-108a
CH2S(O)2CH2CH2OMe D1-108b(Z=2-Cl)
CH2S(O)2CH2CH2OMe D1-108b(Z=3-Me)
CH2S(O)2CH2CH2OMe D1-108b(Z=4-OMe)
CH2S(O)2CH2CH2OMe D1-108b(Z=2-SMe)
CH2S(O)2CH2CH2OMe D1-108b(Z=3-CF3)
CH2S(O)2CH2CH2OMe D1-108b(Z=4-OCF3)
CH2S(O)2CH2CH2OMe D1-108b(Z=2-SCF3)
CH2S(O)2CH2CH2OMe C(O)Me
CH2S(O)2CH2CH2OMe C(O)CF3
CH2S(O)2CH2CH2OMe C(O)OMe
CH(Me)SCH2CH2OMe Me
CH(Me)SCH2CH2OMe Et
CH(Me)SCH2CH2OMe Pr-n
CH(Me)SCH2CH2OMe Pr-i
CH(Me)SCH2CH2OMe Pr-c
CH(Me)SCH2CH2OMe Bu-n
CH(Me)SCH2CH2OMe Bu-i
CH(Me)SCH2CH2OMe Bu-c
CH(Me)SCH2CH2OMe Bu-s
CH(Me)SCH2CH2OMe Bu-t
CH(Me)SCH2CH2OMe Pen-n
CH(Me)SCH2CH2OMe Pen-c
CH(Me)SCH2CH2OMe Hex-n
CH(Me)SCH2CH2OMe Hex-c
CH(Me)SCH2CH2OMe CH2Pr-c
CH(Me)SCH2CH2OMe CH2Bu-c
CH(Me)SCH2CH2OMe CH2Pen-c
CH(Me)SCH2CH2OMe CH2Hex-c
CH(Me)SCH2CH2OMe CH2CH=CH2
CH(Me)SCH2CH2OMe CH2CH=C(Cl)2
CH(Me)SCH2CH2OMe CH2C≡CH
CH(Me)SCH2CH2OMe CH2CN
CH(Me)SCH2CH2OMe CH2CF3
CH(Me)SCH2CH2OMe CH2OMe
CH(Me)SCH2CH2OMe CH2OCF3
CH(Me)SCH2CH2OMe CH2SMe
CH(Me)SCH2CH2OMe CH2S(O)Me
CH(Me)SCH2CH2OMe CH2S(O)2Me
CH(Me)SCH2CH2OMe CH2SCF3
CH(Me)SCH2CH2OMe CH2S(O)CF3
CH(Me)SCH2CH2OMe CH2S(O)2CF3
CH(Me)SCH2CH2OMe CH2CH(OMe)2
CH(Me)SCH2CH2OMe CH2CH(SMe)2
CH(Me)SCH2CH2OMe CH2C(O)Me
CH(Me)SCH2CH2OMe CH2C(O)CF3
CH(Me)SCH2CH2OMe CH2C(O)OMe
CH(Me)SCH2CH2OMe CH2(D1-32a)
CH(Me)SCH2CH2OMe CH2(D1-33a)
CH(Me)SCH2CH2OMe CH2(D1-34a)
CH(Me)SCH2CH2OMe CH2(D1-37a)
CH(Me)SCH2CH2OMe CH2(D1-81a)
CH(Me)SCH2CH2OMe CH2(D1-82a)
CH(Me)SCH2CH2OMe CH2(D1-84a)
CH(Me)SCH2CH2OMe CH2(D1-85a)
CH(Me)SCH2CH2OMe CH2(D1-87a)
CH(Me)SCH2CH2OMe CH2(D1-92a)
CH(Me)SCH2CH2OMe CH2(D1-93a)
CH(Me)SCH2CH2OMe CH2(D1-95a)
CH(Me)SCH2CH2OMe CH2(D1-96a)
CH(Me)SCH2CH2OMe CH2(D1-98a)
CH(Me)SCH2CH2OMe CH2(D1-108a)
CH(Me)SCH2CH2OMe CH2(D1-108b,Z=2-Cl)
CH(Me)SCH2CH2OMe CH2(D1-108b,Z=3-Me)
CH(Me)SCH2CH2OMe CH2(D1-108b,Z=4-OMe)
CH(Me)SCH2CH2OMe CH2(D1-108b,Z=2-SMe)
CH(Me)SCH2CH2OMe CH2(D1-108b,Z=3-CF3)
CH(Me)SCH2CH2OMe CH2(D1-108b,Z=4-OCF3)
CH(Me)SCH2CH2OMe CH2(D1-108b,Z=2-SCF3)
CH(Me)SCH2CH2OMe CH2CH2CN
CH(Me)SCH2CH2OMe CH2CH2CF3
CH(Me)SCH2CH2OMe CH2CH2OMe
CH(Me)SCH2CH2OMe CH2CH2SMe
CH(Me)SCH2CH2OMe CH2CH2S(O)Me
CH(Me)SCH2CH2OMe CH2CH2S(O)2Me
CH(Me)SCH2CH2OMe D1-32a
CH(Me)SCH2CH2OMe D1-33a
CH(Me)SCH2CH2OMe D1-34a
CH(Me)SCH2CH2OMe D1-37a
CH(Me)SCH2CH2OMe D1-81a
CH(Me)SCH2CH2OMe D1-82a
CH(Me)SCH2CH2OMe D1-84a
CH(Me)SCH2CH2OMe D1-85a
CH(Me)SCH2CH2OMe D1-87a
CH(Me)SCH2CH2OMe D1-92a
CH(Me)SCH2CH2OMe D1-93a
CH(Me)SCH2CH2OMe D1-95a
CH(Me)SCH2CH2OMe D1-96a
CH(Me)SCH2CH2OMe D1-98a
CH(Me)SCH2CH2OMe D1-108a
CH(Me)SCH2CH2OMe D1-108b(Z=2-Cl)
CH(Me)SCH2CH2OMe D1-108b(Z=3-Me)
CH(Me)SCH2CH2OMe D1-108b(Z=4-OMe)
CH(Me)SCH2CH2OMe D1-108b(Z=2-SMe)
CH(Me)SCH2CH2OMe D1-108b(Z=3-CF3)
CH(Me)SCH2CH2OMe D1-108b(Z=4-OCF3)
CH(Me)SCH2CH2OMe D1-108b(Z=2-SCF3)
CH(Me)SCH2CH2OMe C(O)Me
CH(Me)SCH2CH2OMe C(O)CF3
CH(Me)SCH2CH2OMe C(O)OMe
CH(Me)S(O)CH2CH2OMe Me
CH(Me)S(O)CH2CH2OMe Et
CH(Me)S(O)CH2CH2OMe Pr-n
CH(Me)S(O)CH2CH2OMe Pr-i
CH(Me)S(O)CH2CH2OMe Pr-c
CH(Me)S(O)CH2CH2OMe Bu-n
CH(Me)S(O)CH2CH2OMe Bu-i
CH(Me)S(O)CH2CH2OMe Bu-c
CH(Me)S(O)CH2CH2OMe Bu-s
CH(Me)S(O)CH2CH2OMe Bu-t
CH(Me)S(O)CH2CH2OMe Pen-n
CH(Me)S(O)CH2CH2OMe Pen-c
CH(Me)S(O)CH2CH2OMe Hex-n
CH(Me)S(O)CH2CH2OMe Hex-c
CH(Me)S(O)CH2CH2OMe CH2Pr-c
CH(Me)S(O)CH2CH2OMe CH2Bu-c
CH(Me)S(O)CH2CH2OMe CH2Pen-c
CH(Me)S(O)CH2CH2OMe CH2Hex-c
CH(Me)S(O)CH2CH2OMe CH2CH=CH2
CH(Me)S(O)CH2CH2OMe CH2CH=C(Cl)2
CH(Me)S(O)CH2CH2OMe CH2C≡CH
CH(Me)S(O)CH2CH2OMe CH2CN
CH(Me)S(O)CH2CH2OMe CH2CF3
CH(Me)S(O)CH2CH2OMe CH2OMe
CH(Me)S(O)CH2CH2OMe CH2OCF3
CH(Me)S(O)CH2CH2OMe CH2SMe
CH(Me)S(O)CH2CH2OMe CH2S(O)Me
CH(Me)S(O)CH2CH2OMe CH2S(O)2Me
CH(Me)S(O)CH2CH2OMe CH2SCF3
CH(Me)S(O)CH2CH2OMe CH2S(O)CF3
CH(Me)S(O)CH2CH2OMe CH2S(O)2CF3
CH(Me)S(O)CH2CH2OMe CH2CH(OMe)2
CH(Me)S(O)CH2CH2OMe CH2CH(SMe)2
CH(Me)S(O)CH2CH2OMe CH2C(O)Me
CH(Me)S(O)CH2CH2OMe CH2C(O)CF3
CH(Me)S(O)CH2CH2OMe CH2C(O)OMe
CH(Me)S(O)CH2CH2OMe CH2(D1-32a)
CH(Me)S(O)CH2CH2OMe CH2(D1-33a)
CH(Me)S(O)CH2CH2OMe CH2(D1-34a)
CH(Me)S(O)CH2CH2OMe CH2(D1-37a)
CH(Me)S(O)CH2CH2OMe CH2(D1-81a)
CH(Me)S(O)CH2CH2OMe CH2(D1-82a)
CH(Me)S(O)CH2CH2OMe CH2(D1-84a)
CH(Me)S(O)CH2CH2OMe CH2(D1-85a)
CH(Me)S(O)CH2CH2OMe CH2(D1-87a)
CH(Me)S(O)CH2CH2OMe CH2(D1-92a)
CH(Me)S(O)CH2CH2OMe CH2(D1-93a)
CH(Me)S(O)CH2CH2OMe CH2(D1-95a)
CH(Me)S(O)CH2CH2OMe CH2(D1-96a)
CH(Me)S(O)CH2CH2OMe CH2(D1-98a)
CH(Me)S(O)CH2CH2OMe CH2(D1-108a)
CH(Me)S(O)CH2CH2OMe CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)CH2CH2OMe CH2(D1-108b,Z=3-Me)
CH(Me)S(O)CH2CH2OMe CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)CH2CH2OMe CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)CH2CH2OMe CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)CH2CH2OMe CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)CH2CH2OMe CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)CH2CH2OMe CH2CH2CN
CH(Me)S(O)CH2CH2OMe CH2CH2CF3
CH(Me)S(O)CH2CH2OMe CH2CH2OMe
CH(Me)S(O)CH2CH2OMe CH2CH2SMe
CH(Me)S(O)CH2CH2OMe CH2CH2S(O)Me
CH(Me)S(O)CH2CH2OMe CH2CH2S(O)2Me
CH(Me)S(O)CH2CH2OMe D1-32a
CH(Me)S(O)CH2CH2OMe D1-33a
CH(Me)S(O)CH2CH2OMe D1-34a
CH(Me)S(O)CH2CH2OMe D1-37a
CH(Me)S(O)CH2CH2OMe D1-81a
CH(Me)S(O)CH2CH2OMe D1-82a
CH(Me)S(O)CH2CH2OMe D1-84a
CH(Me)S(O)CH2CH2OMe D1-85a
CH(Me)S(O)CH2CH2OMe D1-87a
CH(Me)S(O)CH2CH2OMe D1-92a
CH(Me)S(O)CH2CH2OMe D1-93a
CH(Me)S(O)CH2CH2OMe D1-95a
CH(Me)S(O)CH2CH2OMe D1-96a
CH(Me)S(O)CH2CH2OMe D1-98a
CH(Me)S(O)CH2CH2OMe D1-108a
CH(Me)S(O)CH2CH2OMe D1-108b(Z=2-Cl)
CH(Me)S(O)CH2CH2OMe D1-108b(Z=3-Me)
CH(Me)S(O)CH2CH2OMe D1-108b(Z=4-OMe)
CH(Me)S(O)CH2CH2OMe D1-108b(Z=2-SMe)
CH(Me)S(O)CH2CH2OMe D1-108b(Z=3-CF3)
CH(Me)S(O)CH2CH2OMe D1-108b(Z=4-OCF3)
CH(Me)S(O)CH2CH2OMe D1-108b(Z=2-SCF3)
CH(Me)S(O)CH2CH2OMe C(O)Me
CH(Me)S(O)CH2CH2OMe C(O)CF3
CH(Me)S(O)CH2CH2OMe C(O)OMe
CH(Me)S(O)2CH2CH2OMe Me
CH(Me)S(O)2CH2CH2OMe Et
CH(Me)S(O)2CH2CH2OMe Pr-n
CH(Me)S(O)2CH2CH2OMe Pr-i
CH(Me)S(O)2CH2CH2OMe Pr-c
CH(Me)S(O)2CH2CH2OMe Bu-n
CH(Me)S(O)2CH2CH2OMe Bu-i
CH(Me)S(O)2CH2CH2OMe Bu-c
CH(Me)S(O)2CH2CH2OMe Bu-s
CH(Me)S(O)2CH2CH2OMe Bu-t
CH(Me)S(O)2CH2CH2OMe Pen-n
CH(Me)S(O)2CH2CH2OMe Pen-c
CH(Me)S(O)2CH2CH2OMe Hex-n
CH(Me)S(O)2CH2CH2OMe Hex-c
CH(Me)S(O)2CH2CH2OMe CH2Pr-c
CH(Me)S(O)2CH2CH2OMe CH2Bu-c
CH(Me)S(O)2CH2CH2OMe CH2Pen-c
CH(Me)S(O)2CH2CH2OMe CH2Hex-c
CH(Me)S(O)2CH2CH2OMe CH2CH=CH2
CH(Me)S(O)2CH2CH2OMe CH2CH=C(Cl)2
CH(Me)S(O)2CH2CH2OMe CH2C≡CH
CH(Me)S(O)2CH2CH2OMe CH2CN
CH(Me)S(O)2CH2CH2OMe CH2CF3
CH(Me)S(O)2CH2CH2OMe CH2OMe
CH(Me)S(O)2CH2CH2OMe CH2OCF3
CH(Me)S(O)2CH2CH2OMe CH2SMe
CH(Me)S(O)2CH2CH2OMe CH2S(O)Me
CH(Me)S(O)2CH2CH2OMe CH2S(O)2Me
CH(Me)S(O)2CH2CH2OMe CH2SCF3
CH(Me)S(O)2CH2CH2OMe CH2S(O)CF3
CH(Me)S(O)2CH2CH2OMe CH2S(O)2CF3
CH(Me)S(O)2CH2CH2OMe CH2CH(OMe)2
CH(Me)S(O)2CH2CH2OMe CH2CH(SMe)2
CH(Me)S(O)2CH2CH2OMe CH2C(O)Me
CH(Me)S(O)2CH2CH2OMe CH2C(O)CF3
CH(Me)S(O)2CH2CH2OMe CH2C(O)OMe
CH(Me)S(O)2CH2CH2OMe CH2(D1-32a)
CH(Me)S(O)2CH2CH2OMe CH2(D1-33a)
CH(Me)S(O)2CH2CH2OMe CH2(D1-34a)
CH(Me)S(O)2CH2CH2OMe CH2(D1-37a)
CH(Me)S(O)2CH2CH2OMe CH2(D1-81a)
CH(Me)S(O)2CH2CH2OMe CH2(D1-82a)
CH(Me)S(O)2CH2CH2OMe CH2(D1-84a)
CH(Me)S(O)2CH2CH2OMe CH2(D1-85a)
CH(Me)S(O)2CH2CH2OMe CH2(D1-87a)
CH(Me)S(O)2CH2CH2OMe CH2(D1-92a)
CH(Me)S(O)2CH2CH2OMe CH2(D1-93a)
CH(Me)S(O)2CH2CH2OMe CH2(D1-95a)
CH(Me)S(O)2CH2CH2OMe CH2(D1-96a)
CH(Me)S(O)2CH2CH2OMe CH2(D1-98a)
CH(Me)S(O)2CH2CH2OMe CH2(D1-108a)
CH(Me)S(O)2CH2CH2OMe CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)2CH2CH2OMe CH2(D1-108b,Z=3-Me)
CH(Me)S(O)2CH2CH2OMe CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)2CH2CH2OMe CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)2CH2CH2OMe CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)2CH2CH2OMe CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)2CH2CH2OMe CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)2CH2CH2OMe CH2CH2CN
CH(Me)S(O)2CH2CH2OMe CH2CH2CF3
CH(Me)S(O)2CH2CH2OMe CH2CH2OMe
CH(Me)S(O)2CH2CH2OMe CH2CH2SMe
CH(Me)S(O)2CH2CH2OMe CH2CH2S(O)Me
CH(Me)S(O)2CH2CH2OMe CH2CH2S(O)2Me
CH(Me)S(O)2CH2CH2OMe D1-32a
CH(Me)S(O)2CH2CH2OMe D1-33a
CH(Me)S(O)2CH2CH2OMe D1-34a
CH(Me)S(O)2CH2CH2OMe D1-37a
CH(Me)S(O)2CH2CH2OMe D1-81a
CH(Me)S(O)2CH2CH2OMe D1-82a
CH(Me)S(O)2CH2CH2OMe D1-84a
CH(Me)S(O)2CH2CH2OMe D1-85a
CH(Me)S(O)2CH2CH2OMe D1-87a
CH(Me)S(O)2CH2CH2OMe D1-92a
CH(Me)S(O)2CH2CH2OMe D1-93a
CH(Me)S(O)2CH2CH2OMe D1-95a
CH(Me)S(O)2CH2CH2OMe D1-96a
CH(Me)S(O)2CH2CH2OMe D1-98a
CH(Me)S(O)2CH2CH2OMe D1-108a
CH(Me)S(O)2CH2CH2OMe D1-108b(Z=2-Cl)
CH(Me)S(O)2CH2CH2OMe D1-108b(Z=3-Me)
CH(Me)S(O)2CH2CH2OMe D1-108b(Z=4-OMe)
CH(Me)S(O)2CH2CH2OMe D1-108b(Z=2-SMe)
CH(Me)S(O)2CH2CH2OMe D1-108b(Z=3-CF3)
CH(Me)S(O)2CH2CH2OMe D1-108b(Z=4-OCF3)
CH(Me)S(O)2CH2CH2OMe D1-108b(Z=2-SCF3)
CH(Me)S(O)2CH2CH2OMe C(O)Me
CH(Me)S(O)2CH2CH2OMe C(O)CF3
CH(Me)S(O)2CH2CH2OMe C(O)OMe
CH(Et)SCH2CH2OMe Me
CH(Et)SCH2CH2OMe Et
CH(Et)SCH2CH2OMe Pr-n
CH(Et)SCH2CH2OMe Pr-i
CH(Et)SCH2CH2OMe Pr-c
CH(Et)SCH2CH2OMe Bu-n
CH(Et)SCH2CH2OMe Bu-i
CH(Et)SCH2CH2OMe Bu-c
CH(Et)SCH2CH2OMe Bu-s
CH(Et)SCH2CH2OMe Bu-t
CH(Et)SCH2CH2OMe Pen-n
CH(Et)SCH2CH2OMe Pen-c
CH(Et)SCH2CH2OMe Hex-n
CH(Et)SCH2CH2OMe Hex-c
CH(Et)SCH2CH2OMe CH2Pr-c
CH(Et)SCH2CH2OMe CH2Bu-c
CH(Et)SCH2CH2OMe CH2Pen-c
CH(Et)SCH2CH2OMe CH2Hex-c
CH(Et)SCH2CH2OMe CH2CH=CH2
CH(Et)SCH2CH2OMe CH2CH=C(Cl)2
CH(Et)SCH2CH2OMe CH2C≡CH
CH(Et)SCH2CH2OMe CH2CN
CH(Et)SCH2CH2OMe CH2CF3
CH(Et)SCH2CH2OMe CH2OMe
CH(Et)SCH2CH2OMe CH2OCF3
CH(Et)SCH2CH2OMe CH2SMe
CH(Et)SCH2CH2OMe CH2S(O)Me
CH(Et)SCH2CH2OMe CH2S(O)2Me
CH(Et)SCH2CH2OMe CH2SCF3
CH(Et)SCH2CH2OMe CH2S(O)CF3
CH(Et)SCH2CH2OMe CH2S(O)2CF3
CH(Et)SCH2CH2OMe CH2CH(OMe)2
CH(Et)SCH2CH2OMe CH2CH(SMe)2
CH(Et)SCH2CH2OMe CH2C(O)Me
CH(Et)SCH2CH2OMe CH2C(O)CF3
CH(Et)SCH2CH2OMe CH2C(O)OMe
CH(Et)SCH2CH2OMe CH2(D1-32a)
CH(Et)SCH2CH2OMe CH2(D1-33a)
CH(Et)SCH2CH2OMe CH2(D1-34a)
CH(Et)SCH2CH2OMe CH2(D1-37a)
CH(Et)SCH2CH2OMe CH2(D1-81a)
CH(Et)SCH2CH2OMe CH2(D1-82a)
CH(Et)SCH2CH2OMe CH2(D1-84a)
CH(Et)SCH2CH2OMe CH2(D1-85a)
CH(Et)SCH2CH2OMe CH2(D1-87a)
CH(Et)SCH2CH2OMe CH2(D1-92a)
CH(Et)SCH2CH2OMe CH2(D1-93a)
CH(Et)SCH2CH2OMe CH2(D1-95a)
CH(Et)SCH2CH2OMe CH2(D1-96a)
CH(Et)SCH2CH2OMe CH2(D1-98a)
CH(Et)SCH2CH2OMe CH2(D1-108a)
CH(Et)SCH2CH2OMe CH2(D1-108b,Z=2-Cl)
CH(Et)SCH2CH2OMe CH2(D1-108b,Z=3-Me)
CH(Et)SCH2CH2OMe CH2(D1-108b,Z=4-OMe)
CH(Et)SCH2CH2OMe CH2(D1-108b,Z=2-SMe)
CH(Et)SCH2CH2OMe CH2(D1-108b,Z=3-CF3)
CH(Et)SCH2CH2OMe CH2(D1-108b,Z=4-OCF3)
CH(Et)SCH2CH2OMe CH2(D1-108b,Z=2-SCF3)
CH(Et)SCH2CH2OMe CH2CH2CN
CH(Et)SCH2CH2OMe CH2CH2CF3
CH(Et)SCH2CH2OMe CH2CH2OMe
CH(Et)SCH2CH2OMe CH2CH2SMe
CH(Et)SCH2CH2OMe CH2CH2S(O)Me
CH(Et)SCH2CH2OMe CH2CH2S(O)2Me
CH(Et)SCH2CH2OMe D1-32a
CH(Et)SCH2CH2OMe D1-33a
CH(Et)SCH2CH2OMe D1-34a
CH(Et)SCH2CH2OMe D1-37a
CH(Et)SCH2CH2OMe D1-81a
CH(Et)SCH2CH2OMe D1-82a
CH(Et)SCH2CH2OMe D1-84a
CH(Et)SCH2CH2OMe D1-85a
CH(Et)SCH2CH2OMe D1-87a
CH(Et)SCH2CH2OMe D1-92a
CH(Et)SCH2CH2OMe D1-93a
CH(Et)SCH2CH2OMe D1-95a
CH(Et)SCH2CH2OMe D1-96a
CH(Et)SCH2CH2OMe D1-98a
CH(Et)SCH2CH2OMe D1-108a
CH(Et)SCH2CH2OMe D1-108b(Z=2-Cl)
CH(Et)SCH2CH2OMe D1-108b(Z=3-Me)
CH(Et)SCH2CH2OMe D1-108b(Z=4-OMe)
CH(Et)SCH2CH2OMe D1-108b(Z=2-SMe)
CH(Et)SCH2CH2OMe D1-108b(Z=3-CF3)
CH(Et)SCH2CH2OMe D1-108b(Z=4-OCF3)
CH(Et)SCH2CH2OMe D1-108b(Z=2-SCF3)
CH(Et)SCH2CH2OMe C(O)Me
CH(Et)SCH2CH2OMe C(O)CF3
CH(Et)SCH2CH2OMe C(O)OMe
CH(Et)S(O)CH2CH2OMe Me
CH(Et)S(O)CH2CH2OMe Et
CH(Et)S(O)CH2CH2OMe Pr-n
CH(Et)S(O)CH2CH2OMe Pr-i
CH(Et)S(O)CH2CH2OMe Pr-c
CH(Et)S(O)CH2CH2OMe Bu-n
CH(Et)S(O)CH2CH2OMe Bu-i
CH(Et)S(O)CH2CH2OMe Bu-c
CH(Et)S(O)CH2CH2OMe Bu-s
CH(Et)S(O)CH2CH2OMe Bu-t
CH(Et)S(O)CH2CH2OMe Pen-n
CH(Et)S(O)CH2CH2OMe Pen-c
CH(Et)S(O)CH2CH2OMe Hex-n
CH(Et)S(O)CH2CH2OMe Hex-c
CH(Et)S(O)CH2CH2OMe CH2Pr-c
CH(Et)S(O)CH2CH2OMe CH2Bu-c
CH(Et)S(O)CH2CH2OMe CH2Pen-c
CH(Et)S(O)CH2CH2OMe CH2Hex-c
CH(Et)S(O)CH2CH2OMe CH2CH=CH2
CH(Et)S(O)CH2CH2OMe CH2CH=C(Cl)2
CH(Et)S(O)CH2CH2OMe CH2C≡CH
CH(Et)S(O)CH2CH2OMe CH2CN
CH(Et)S(O)CH2CH2OMe CH2CF3
CH(Et)S(O)CH2CH2OMe CH2OMe
CH(Et)S(O)CH2CH2OMe CH2OCF3
CH(Et)S(O)CH2CH2OMe CH2SMe
CH(Et)S(O)CH2CH2OMe CH2S(O)Me
CH(Et)S(O)CH2CH2OMe CH2S(O)2Me
CH(Et)S(O)CH2CH2OMe CH2SCF3
CH(Et)S(O)CH2CH2OMe CH2S(O)CF3
CH(Et)S(O)CH2CH2OMe CH2S(O)2CF3
CH(Et)S(O)CH2CH2OMe CH2CH(OMe)2
CH(Et)S(O)CH2CH2OMe CH2CH(SMe)2
CH(Et)S(O)CH2CH2OMe CH2C(O)Me
CH(Et)S(O)CH2CH2OMe CH2C(O)CF3
CH(Et)S(O)CH2CH2OMe CH2C(O)OMe
CH(Et)S(O)CH2CH2OMe CH2(D1-32a)
CH(Et)S(O)CH2CH2OMe CH2(D1-33a)
CH(Et)S(O)CH2CH2OMe CH2(D1-34a)
CH(Et)S(O)CH2CH2OMe CH2(D1-37a)
CH(Et)S(O)CH2CH2OMe CH2(D1-81a)
CH(Et)S(O)CH2CH2OMe CH2(D1-82a)
CH(Et)S(O)CH2CH2OMe CH2(D1-84a)
CH(Et)S(O)CH2CH2OMe CH2(D1-85a)
CH(Et)S(O)CH2CH2OMe CH2(D1-87a)
CH(Et)S(O)CH2CH2OMe CH2(D1-92a)
CH(Et)S(O)CH2CH2OMe CH2(D1-93a)
CH(Et)S(O)CH2CH2OMe CH2(D1-95a)
CH(Et)S(O)CH2CH2OMe CH2(D1-96a)
CH(Et)S(O)CH2CH2OMe CH2(D1-98a)
CH(Et)S(O)CH2CH2OMe CH2(D1-108a)
CH(Et)S(O)CH2CH2OMe CH2(D1-108b,Z=2-Cl)
CH(Et)S(O)CH2CH2OMe CH2(D1-108b,Z=3-Me)
CH(Et)S(O)CH2CH2OMe CH2(D1-108b,Z=4-OMe)
CH(Et)S(O)CH2CH2OMe CH2(D1-108b,Z=2-SMe)
CH(Et)S(O)CH2CH2OMe CH2(D1-108b,Z=3-CF3)
CH(Et)S(O)CH2CH2OMe CH2(D1-108b,Z=4-OCF3)
CH(Et)S(O)CH2CH2OMe CH2(D1-108b,Z=2-SCF3)
CH(Et)S(O)CH2CH2OMe CH2CH2CN
CH(Et)S(O)CH2CH2OMe CH2CH2CF3
CH(Et)S(O)CH2CH2OMe CH2CH2OMe
CH(Et)S(O)CH2CH2OMe CH2CH2SMe
CH(Et)S(O)CH2CH2OMe CH2CH2S(O)Me
CH(Et)S(O)CH2CH2OMe CH2CH2S(O)2Me
CH(Et)S(O)CH2CH2OMe D1-32a
CH(Et)S(O)CH2CH2OMe D1-33a
CH(Et)S(O)CH2CH2OMe D1-34a
CH(Et)S(O)CH2CH2OMe D1-37a
CH(Et)S(O)CH2CH2OMe D1-81a
CH(Et)S(O)CH2CH2OMe D1-82a
CH(Et)S(O)CH2CH2OMe D1-84a
CH(Et)S(O)CH2CH2OMe D1-85a
CH(Et)S(O)CH2CH2OMe D1-87a
CH(Et)S(O)CH2CH2OMe D1-92a
CH(Et)S(O)CH2CH2OMe D1-93a
CH(Et)S(O)CH2CH2OMe D1-95a
CH(Et)S(O)CH2CH2OMe D1-96a
CH(Et)S(O)CH2CH2OMe D1-98a
CH(Et)S(O)CH2CH2OMe D1-108a
CH(Et)S(O)CH2CH2OMe D1-108b(Z=2-Cl)
CH(Et)S(O)CH2CH2OMe D1-108b(Z=3-Me)
CH(Et)S(O)CH2CH2OMe D1-108b(Z=4-OMe)
CH(Et)S(O)CH2CH2OMe D1-108b(Z=2-SMe)
CH(Et)S(O)CH2CH2OMe D1-108b(Z=3-CF3)
CH(Et)S(O)CH2CH2OMe D1-108b(Z=4-OCF3)
CH(Et)S(O)CH2CH2OMe D1-108b(Z=2-SCF3)
CH(Et)S(O)CH2CH2OMe C(O)Me
CH(Et)S(O)CH2CH2OMe C(O)CF3
CH(Et)S(O)CH2CH2OMe C(O)OMe
CH(Et)S(O)2CH2CH2OMe Me
CH(Et)S(O)2CH2CH2OMe Et
CH(Et)S(O)2CH2CH2OMe Pr-n
CH(Et)S(O)2CH2CH2OMe Pr-i
CH(Et)S(O)2CH2CH2OMe Pr-c
CH(Et)S(O)2CH2CH2OMe Bu-n
CH(Et)S(O)2CH2CH2OMe Bu-i
CH(Et)S(O)2CH2CH2OMe Bu-c
CH(Et)S(O)2CH2CH2OMe Bu-s
CH(Et)S(O)2CH2CH2OMe Bu-t
CH(Et)S(O)2CH2CH2OMe Pen-n
CH(Et)S(O)2CH2CH2OMe Pen-c
CH(Et)S(O)2CH2CH2OMe Hex-n
CH(Et)S(O)2CH2CH2OMe Hex-c
CH(Et)S(O)2CH2CH2OMe CH2Pr-c
CH(Et)S(O)2CH2CH2OMe CH2Bu-c
CH(Et)S(O)2CH2CH2OMe CH2Pen-c
CH(Et)S(O)2CH2CH2OMe CH2Hex-c
CH(Et)S(O)2CH2CH2OMe CH2CH=CH2
CH(Et)S(O)2CH2CH2OMe CH2CH=C(Cl)2
CH(Et)S(O)2CH2CH2OMe CH2C≡CH
CH(Et)S(O)2CH2CH2OMe CH2CN
CH(Et)S(O)2CH2CH2OMe CH2CF3
CH(Et)S(O)2CH2CH2OMe CH2OMe
CH(Et)S(O)2CH2CH2OMe CH2OCF3
CH(Et)S(O)2CH2CH2OMe CH2SMe
CH(Et)S(O)2CH2CH2OMe CH2S(O)Me
CH(Et)S(O)2CH2CH2OMe CH2S(O)2Me
CH(Et)S(O)2CH2CH2OMe CH2SCF3
CH(Et)S(O)2CH2CH2OMe CH2S(O)CF3
CH(Et)S(O)2CH2CH2OMe CH2S(O)2CF3
CH(Et)S(O)2CH2CH2OMe CH2CH(OMe)2
CH(Et)S(O)2CH2CH2OMe CH2CH(SMe)2
CH(Et)S(O)2CH2CH2OMe CH2C(O)Me
CH(Et)S(O)2CH2CH2OMe CH2C(O)CF3
CH(Et)S(O)2CH2CH2OMe CH2C(O)OMe
CH(Et)S(O)2CH2CH2OMe CH2(D1-32a)
CH(Et)S(O)2CH2CH2OMe CH2(D1-33a)
CH(Et)S(O)2CH2CH2OMe CH2(D1-34a)
CH(Et)S(O)2CH2CH2OMe CH2(D1-37a)
CH(Et)S(O)2CH2CH2OMe CH2(D1-81a)
CH(Et)S(O)2CH2CH2OMe CH2(D1-82a)
CH(Et)S(O)2CH2CH2OMe CH2(D1-84a)
CH(Et)S(O)2CH2CH2OMe CH2(D1-85a)
CH(Et)S(O)2CH2CH2OMe CH2(D1-87a)
CH(Et)S(O)2CH2CH2OMe CH2(D1-92a)
CH(Et)S(O)2CH2CH2OMe CH2(D1-93a)
CH(Et)S(O)2CH2CH2OMe CH2(D1-95a)
CH(Et)S(O)2CH2CH2OMe CH2(D1-96a)
CH(Et)S(O)2CH2CH2OMe CH2(D1-98a)
CH(Et)S(O)2CH2CH2OMe CH2(D1-108a)
CH(Et)S(O)2CH2CH2OMe CH2(D1-108b,Z=2-Cl)
CH(Et)S(O)2CH2CH2OMe CH2(D1-108b,Z=3-Me)
CH(Et)S(O)2CH2CH2OMe CH2(D1-108b,Z=4-OMe)
CH(Et)S(O)2CH2CH2OMe CH2(D1-108b,Z=2-SMe)
CH(Et)S(O)2CH2CH2OMe CH2(D1-108b,Z=3-CF3)
CH(Et)S(O)2CH2CH2OMe CH2(D1-108b,Z=4-OCF3)
CH(Et)S(O)2CH2CH2OMe CH2(D1-108b,Z=2-SCF3)
CH(Et)S(O)2CH2CH2OMe CH2CH2CN
CH(Et)S(O)2CH2CH2OMe CH2CH2CF3
CH(Et)S(O)2CH2CH2OMe CH2CH2OMe
CH(Et)S(O)2CH2CH2OMe CH2CH2SMe
CH(Et)S(O)2CH2CH2OMe CH2CH2S(O)Me
CH(Et)S(O)2CH2CH2OMe CH2CH2S(O)2Me
CH(Et)S(O)2CH2CH2OMe D1-32a
CH(Et)S(O)2CH2CH2OMe D1-33a
CH(Et)S(O)2CH2CH2OMe D1-34a
CH(Et)S(O)2CH2CH2OMe D1-37a
CH(Et)S(O)2CH2CH2OMe D1-81a
CH(Et)S(O)2CH2CH2OMe D1-82a
CH(Et)S(O)2CH2CH2OMe D1-84a
CH(Et)S(O)2CH2CH2OMe D1-85a
CH(Et)S(O)2CH2CH2OMe D1-87a
CH(Et)S(O)2CH2CH2OMe D1-92a
CH(Et)S(O)2CH2CH2OMe D1-93a
CH(Et)S(O)2CH2CH2OMe D1-95a
CH(Et)S(O)2CH2CH2OMe D1-96a
CH(Et)S(O)2CH2CH2OMe D1-98a
CH(Et)S(O)2CH2CH2OMe D1-108a
CH(Et)S(O)2CH2CH2OMe D1-108b(Z=2-Cl)
CH(Et)S(O)2CH2CH2OMe D1-108b(Z=3-Me)
CH(Et)S(O)2CH2CH2OMe D1-108b(Z=4-OMe)
CH(Et)S(O)2CH2CH2OMe D1-108b(Z=2-SMe)
CH(Et)S(O)2CH2CH2OMe D1-108b(Z=3-CF3)
CH(Et)S(O)2CH2CH2OMe D1-108b(Z=4-OCF3)
CH(Et)S(O)2CH2CH2OMe D1-108b(Z=2-SCF3)
CH(Et)S(O)2CH2CH2OMe C(O)Me
CH(Et)S(O)2CH2CH2OMe C(O)CF3
CH(Et)S(O)2CH2CH2OMe C(O)OMe
CH2SCH2CH2OEt Me
CH2SCH2CH2OEt Et
CH2SCH2CH2OEt Pr-n
CH2SCH2CH2OEt Pr-i
CH2SCH2CH2OEt Pr-c
CH2SCH2CH2OEt Bu-n
CH2SCH2CH2OEt Bu-i
CH2SCH2CH2OEt Bu-c
CH2SCH2CH2OEt Bu-s
CH2SCH2CH2OEt Bu-t
CH2SCH2CH2OEt Pen-n
CH2SCH2CH2OEt Pen-c
CH2SCH2CH2OEt Hex-n
CH2SCH2CH2OEt Hex-c
CH2SCH2CH2OEt CH2Pr-c
CH2SCH2CH2OEt CH2Bu-c
CH2SCH2CH2OEt CH2Pen-c
CH2SCH2CH2OEt CH2Hex-c
CH2SCH2CH2OEt CH2CH=CH2
CH2SCH2CH2OEt CH2CH=C(Cl)2
CH2SCH2CH2OEt CH2C≡CH
CH2SCH2CH2OEt CH2CN
CH2SCH2CH2OEt CH2CF3
CH2SCH2CH2OEt CH2OMe
CH2SCH2CH2OEt CH2OCF3
CH2SCH2CH2OEt CH2SMe
CH2SCH2CH2OEt CH2S(O)Me
CH2SCH2CH2OEt CH2S(O)2Me
CH2SCH2CH2OEt CH2SCF3
CH2SCH2CH2OEt CH2S(O)CF3
CH2SCH2CH2OEt CH2S(O)2CF3
CH2SCH2CH2OEt CH2CH(OMe)2
CH2SCH2CH2OEt CH2CH(SMe)2
CH2SCH2CH2OEt CH2C(O)Me
CH2SCH2CH2OEt CH2C(O)CF3
CH2SCH2CH2OEt CH2C(O)OMe
CH2SCH2CH2OEt CH2(D1-32a)
CH2SCH2CH2OEt CH2(D1-33a)
CH2SCH2CH2OEt CH2(D1-34a)
CH2SCH2CH2OEt CH2(D1-37a)
CH2SCH2CH2OEt CH2(D1-81a)
CH2SCH2CH2OEt CH2(D1-82a)
CH2SCH2CH2OEt CH2(D1-84a)
CH2SCH2CH2OEt CH2(D1-85a)
CH2SCH2CH2OEt CH2(D1-87a)
CH2SCH2CH2OEt CH2(D1-92a)
CH2SCH2CH2OEt CH2(D1-93a)
CH2SCH2CH2OEt CH2(D1-95a)
CH2SCH2CH2OEt CH2(D1-96a)
CH2SCH2CH2OEt CH2(D1-98a)
CH2SCH2CH2OEt CH2(D1-108a)
CH2SCH2CH2OEt CH2(D1-108b,Z=2-Cl)
CH2SCH2CH2OEt CH2(D1-108b,Z=3-Me)
CH2SCH2CH2OEt CH2(D1-108b,Z=4-OEt)
CH2SCH2CH2OEt CH2(D1-108b,Z=2-SMe)
CH2SCH2CH2OEt CH2(D1-108b,Z=3-CF3)
CH2SCH2CH2OEt CH2(D1-108b,Z=4-OCF3)
CH2SCH2CH2OEt CH2(D1-108b,Z=2-SCF3)
CH2SCH2CH2OEt CH2CH2CN
CH2SCH2CH2OEt CH2CH2CF3
CH2SCH2CH2OEt CH2CH2OEt
CH2SCH2CH2OEt CH2CH2SMe
CH2SCH2CH2OEt CH2CH2S(O)Me
CH2SCH2CH2OEt CH2CH2S(O)2Me
CH2SCH2CH2OEt D1-32a
CH2SCH2CH2OEt D1-33a
CH2SCH2CH2OEt D1-34a
CH2SCH2CH2OEt D1-37a
CH2SCH2CH2OEt D1-81a
CH2SCH2CH2OEt D1-82a
CH2SCH2CH2OEt D1-84a
CH2SCH2CH2OEt D1-85a
CH2SCH2CH2OEt D1-87a
CH2SCH2CH2OEt D1-92a
CH2SCH2CH2OEt D1-93a
CH2SCH2CH2OEt D1-95a
CH2SCH2CH2OEt D1-96a
CH2SCH2CH2OEt D1-98a
CH2SCH2CH2OEt D1-108a
CH2SCH2CH2OEt D1-108b(Z=2-Cl)
CH2SCH2CH2OEt D1-108b(Z=3-Me)
CH2SCH2CH2OEt D1-108b(Z=4-OEt)
CH2SCH2CH2OEt D1-108b(Z=2-SMe)
CH2SCH2CH2OEt D1-108b(Z=3-CF3)
CH2SCH2CH2OEt D1-108b(Z=4-OCF3)
CH2SCH2CH2OEt D1-108b(Z=2-SCF3)
CH2SCH2CH2OEt C(O)Me
CH2SCH2CH2OEt C(O)CF3
CH2SCH2CH2OEt C(O)OEt
CH2S(O)CH2CH2OEt Me
CH2S(O)CH2CH2OEt Et
CH2S(O)CH2CH2OEt Pr-n
CH2S(O)CH2CH2OEt Pr-i
CH2S(O)CH2CH2OEt Pr-c
CH2S(O)CH2CH2OEt Bu-n
CH2S(O)CH2CH2OEt Bu-i
CH2S(O)CH2CH2OEt Bu-c
CH2S(O)CH2CH2OEt Bu-s
CH2S(O)CH2CH2OEt Bu-t
CH2S(O)CH2CH2OEt Pen-n
CH2S(O)CH2CH2OEt Pen-c
CH2S(O)CH2CH2OEt Hex-n
CH2S(O)CH2CH2OEt Hex-c
CH2S(O)CH2CH2OEt CH2Pr-c
CH2S(O)CH2CH2OEt CH2Bu-c
CH2S(O)CH2CH2OEt CH2Pen-c
CH2S(O)CH2CH2OEt CH2Hex-c
CH2S(O)CH2CH2OEt CH2CH=CH2
CH2S(O)CH2CH2OEt CH2CH=C(Cl)2
CH2S(O)CH2CH2OEt CH2C≡CH
CH2S(O)CH2CH2OEt CH2CN
CH2S(O)CH2CH2OEt CH2CF3
CH2S(O)CH2CH2OEt CH2OEt
CH2S(O)CH2CH2OEt CH2OCF3
CH2S(O)CH2CH2OEt CH2SMe
CH2S(O)CH2CH2OEt CH2S(O)Me
CH2S(O)CH2CH2OEt CH2S(O)2Me
CH2S(O)CH2CH2OEt CH2SCF3
CH2S(O)CH2CH2OEt CH2S(O)CF3
CH2S(O)CH2CH2OEt CH2S(O)2CF3
CH2S(O)CH2CH2OEt CH2CH(OEt)2
CH2S(O)CH2CH2OEt CH2CH(SMe)2
CH2S(O)CH2CH2OEt CH2C(O)Me
CH2S(O)CH2CH2OEt CH2C(O)CF3
CH2S(O)CH2CH2OEt CH2C(O)OEt
CH2S(O)CH2CH2OEt CH2(D1-32a)
CH2S(O)CH2CH2OEt CH2(D1-33a)
CH2S(O)CH2CH2OEt CH2(D1-34a)
CH2S(O)CH2CH2OEt CH2(D1-37a)
CH2S(O)CH2CH2OEt CH2(D1-81a)
CH2S(O)CH2CH2OEt CH2(D1-82a)
CH2S(O)CH2CH2OEt CH2(D1-84a)
CH2S(O)CH2CH2OEt CH2(D1-85a)
CH2S(O)CH2CH2OEt CH2(D1-87a)
CH2S(O)CH2CH2OEt CH2(D1-92a)
CH2S(O)CH2CH2OEt CH2(D1-93a)
CH2S(O)CH2CH2OEt CH2(D1-95a)
CH2S(O)CH2CH2OEt CH2(D1-96a)
CH2S(O)CH2CH2OEt CH2(D1-98a)
CH2S(O)CH2CH2OEt CH2(D1-108a)
CH2S(O)CH2CH2OEt CH2(D1-108b,Z=2-Cl)
CH2S(O)CH2CH2OEt CH2(D1-108b,Z=3-Me)
CH2S(O)CH2CH2OEt CH2(D1-108b,Z=4-OEt)
CH2S(O)CH2CH2OEt CH2(D1-108b,Z=2-SMe)
CH2S(O)CH2CH2OEt CH2(D1-108b,Z=3-CF3)
CH2S(O)CH2CH2OEt CH2(D1-108b,Z=4-OCF3)
CH2S(O)CH2CH2OEt CH2(D1-108b,Z=2-SCF3)
CH2S(O)CH2CH2OEt CH2CH2CN
CH2S(O)CH2CH2OEt CH2CH2CF3
CH2S(O)CH2CH2OEt CH2CH2OEt
CH2S(O)CH2CH2OEt CH2CH2SMe
CH2S(O)CH2CH2OEt CH2CH2S(O)Me
CH2S(O)CH2CH2OEt CH2CH2S(O)2Me
CH2S(O)CH2CH2OEt D1-32a
CH2S(O)CH2CH2OEt D1-33a
CH2S(O)CH2CH2OEt D1-34a
CH2S(O)CH2CH2OEt D1-37a
CH2S(O)CH2CH2OEt D1-81a
CH2S(O)CH2CH2OEt D1-82a
CH2S(O)CH2CH2OEt D1-84a
CH2S(O)CH2CH2OEt D1-85a
CH2S(O)CH2CH2OEt D1-87a
CH2S(O)CH2CH2OEt D1-92a
CH2S(O)CH2CH2OEt D1-93a
CH2S(O)CH2CH2OEt D1-95a
CH2S(O)CH2CH2OEt D1-96a
CH2S(O)CH2CH2OEt D1-98a
CH2S(O)CH2CH2OEt D1-108a
CH2S(O)CH2CH2OEt D1-108b(Z=2-Cl)
CH2S(O)CH2CH2OEt D1-108b(Z=3-Me)
CH2S(O)CH2CH2OEt D1-108b(Z=4-OEt)
CH2S(O)CH2CH2OEt D1-108b(Z=2-SMe)
CH2S(O)CH2CH2OEt D1-108b(Z=3-CF3)
CH2S(O)CH2CH2OEt D1-108b(Z=4-OCF3)
CH2S(O)CH2CH2OEt D1-108b(Z=2-SCF3)
CH2S(O)CH2CH2OEt C(O)Me
CH2S(O)CH2CH2OEt C(O)CF3
CH2S(O)CH2CH2OEt C(O)OEt
CH2S(O)2CH2CH2OEt Me
CH2S(O)2CH2CH2OEt Et
CH2S(O)2CH2CH2OEt Pr-n
CH2S(O)2CH2CH2OEt Pr-i
CH2S(O)2CH2CH2OEt Pr-c
CH2S(O)2CH2CH2OEt Bu-n
CH2S(O)2CH2CH2OEt Bu-i
CH2S(O)2CH2CH2OEt Bu-c
CH2S(O)2CH2CH2OEt Bu-s
CH2S(O)2CH2CH2OEt Bu-t
CH2S(O)2CH2CH2OEt Pen-n
CH2S(O)2CH2CH2OEt Pen-c
CH2S(O)2CH2CH2OEt Hex-n
CH2S(O)2CH2CH2OEt Hex-c
CH2S(O)2CH2CH2OEt CH2Pr-c
CH2S(O)2CH2CH2OEt CH2Bu-c
CH2S(O)2CH2CH2OEt CH2Pen-c
CH2S(O)2CH2CH2OEt CH2Hex-c
CH2S(O)2CH2CH2OEt CH2CH=CH2
CH2S(O)2CH2CH2OEt CH2CH=C(Cl)2
CH2S(O)2CH2CH2OEt CH2C≡CH
CH2S(O)2CH2CH2OEt CH2CN
CH2S(O)2CH2CH2OEt CH2CF3
CH2S(O)2CH2CH2OEt CH2OEt
CH2S(O)2CH2CH2OEt CH2OCF3
CH2S(O)2CH2CH2OEt CH2SMe
CH2S(O)2CH2CH2OEt CH2S(O)Me
CH2S(O)2CH2CH2OEt CH2S(O)2Me
CH2S(O)2CH2CH2OEt CH2SCF3
CH2S(O)2CH2CH2OEt CH2S(O)CF3
CH2S(O)2CH2CH2OEt CH2S(O)2CF3
CH2S(O)2CH2CH2OEt CH2CH(OEt)2
CH2S(O)2CH2CH2OEt CH2CH(SMe)2
CH2S(O)2CH2CH2OEt CH2C(O)Me
CH2S(O)2CH2CH2OEt CH2C(O)CF3
CH2S(O)2CH2CH2OEt CH2C(O)OEt
CH2S(O)2CH2CH2OEt CH2(D1-32a)
CH2S(O)2CH2CH2OEt CH2(D1-33a)
CH2S(O)2CH2CH2OEt CH2(D1-34a)
CH2S(O)2CH2CH2OEt CH2(D1-37a)
CH2S(O)2CH2CH2OEt CH2(D1-81a)
CH2S(O)2CH2CH2OEt CH2(D1-82a)
CH2S(O)2CH2CH2OEt CH2(D1-84a)
CH2S(O)2CH2CH2OEt CH2(D1-85a)
CH2S(O)2CH2CH2OEt CH2(D1-87a)
CH2S(O)2CH2CH2OEt CH2(D1-92a)
CH2S(O)2CH2CH2OEt CH2(D1-93a)
CH2S(O)2CH2CH2OEt CH2(D1-95a)
CH2S(O)2CH2CH2OEt CH2(D1-96a)
CH2S(O)2CH2CH2OEt CH2(D1-98a)
CH2S(O)2CH2CH2OEt CH2(D1-108a)
CH2S(O)2CH2CH2OEt CH2(D1-108b,Z=2-Cl)
CH2S(O)2CH2CH2OEt CH2(D1-108b,Z=3-Me)
CH2S(O)2CH2CH2OEt CH2(D1-108b,Z=4-OEt)
CH2S(O)2CH2CH2OEt CH2(D1-108b,Z=2-SMe)
CH2S(O)2CH2CH2OEt CH2(D1-108b,Z=3-CF3)
CH2S(O)2CH2CH2OEt CH2(D1-108b,Z=4-OCF3)
CH2S(O)2CH2CH2OEt CH2(D1-108b,Z=2-SCF3)
CH2S(O)2CH2CH2OEt CH2CH2CN
CH2S(O)2CH2CH2OEt CH2CH2CF3
CH2S(O)2CH2CH2OEt CH2CH2OEt
CH2S(O)2CH2CH2OEt CH2CH2SMe
CH2S(O)2CH2CH2OEt CH2CH2S(O)Me
CH2S(O)2CH2CH2OEt CH2CH2S(O)2Me
CH2S(O)2CH2CH2OEt D1-32a
CH2S(O)2CH2CH2OEt D1-33a
CH2S(O)2CH2CH2OEt D1-34a
CH2S(O)2CH2CH2OEt D1-37a
CH2S(O)2CH2CH2OEt D1-81a
CH2S(O)2CH2CH2OEt D1-82a
CH2S(O)2CH2CH2OEt D1-84a
CH2S(O)2CH2CH2OEt D1-85a
CH2S(O)2CH2CH2OEt D1-87a
CH2S(O)2CH2CH2OEt D1-92a
CH2S(O)2CH2CH2OEt D1-93a
CH2S(O)2CH2CH2OEt D1-95a
CH2S(O)2CH2CH2OEt D1-96a
CH2S(O)2CH2CH2OEt D1-98a
CH2S(O)2CH2CH2OEt D1-108a
CH2S(O)2CH2CH2OEt D1-108b(Z=2-Cl)
CH2S(O)2CH2CH2OEt D1-108b(Z=3-Me)
CH2S(O)2CH2CH2OEt D1-108b(Z=4-OEt)
CH2S(O)2CH2CH2OEt D1-108b(Z=2-SMe)
CH2S(O)2CH2CH2OEt D1-108b(Z=3-CF3)
CH2S(O)2CH2CH2OEt D1-108b(Z=4-OCF3)
CH2S(O)2CH2CH2OEt D1-108b(Z=2-SCF3)
CH2S(O)2CH2CH2OEt C(O)Me
CH2S(O)2CH2CH2OEt C(O)CF3
CH2S(O)2CH2CH2OEt C(O)OEt
CH(Me)SCH2CH2OEt Me
CH(Me)SCH2CH2OEt Et
CH(Me)SCH2CH2OEt Pr-n
CH(Me)SCH2CH2OEt Pr-i
CH(Me)SCH2CH2OEt Pr-c
CH(Me)SCH2CH2OEt Bu-n
CH(Me)SCH2CH2OEt Bu-i
CH(Me)SCH2CH2OEt Bu-c
CH(Me)SCH2CH2OEt Bu-s
CH(Me)SCH2CH2OEt Bu-t
CH(Me)SCH2CH2OEt Pen-n
CH(Me)SCH2CH2OEt Pen-c
CH(Me)SCH2CH2OEt Hex-n
CH(Me)SCH2CH2OEt Hex-c
CH(Me)SCH2CH2OEt CH2Pr-c
CH(Me)SCH2CH2OEt CH2Bu-c
CH(Me)SCH2CH2OEt CH2Pen-c
CH(Me)SCH2CH2OEt CH2Hex-c
CH(Me)SCH2CH2OEt CH2CH=CH2
CH(Me)SCH2CH2OEt CH2CH=C(Cl)2
CH(Me)SCH2CH2OEt CH2C≡CH
CH(Me)SCH2CH2OEt CH2CN
CH(Me)SCH2CH2OEt CH2CF3
CH(Me)SCH2CH2OEt CH2OEt
CH(Me)SCH2CH2OEt CH2OCF3
CH(Me)SCH2CH2OEt CH2SMe
CH(Me)SCH2CH2OEt CH2S(O)Me
CH(Me)SCH2CH2OEt CH2S(O)2Me
CH(Me)SCH2CH2OEt CH2SCF3
CH(Me)SCH2CH2OEt CH2S(O)CF3
CH(Me)SCH2CH2OEt CH2S(O)2CF3
CH(Me)SCH2CH2OEt CH2CH(OEt)2
CH(Me)SCH2CH2OEt CH2CH(SMe)2
CH(Me)SCH2CH2OEt CH2C(O)Me
CH(Me)SCH2CH2OEt CH2C(O)CF3
CH(Me)SCH2CH2OEt CH2C(O)OEt
CH(Me)SCH2CH2OEt CH2(D1-32a)
CH(Me)SCH2CH2OEt CH2(D1-33a)
CH(Me)SCH2CH2OEt CH2(D1-34a)
CH(Me)SCH2CH2OEt CH2(D1-37a)
CH(Me)SCH2CH2OEt CH2(D1-81a)
CH(Me)SCH2CH2OEt CH2(D1-82a)
CH(Me)SCH2CH2OEt CH2(D1-84a)
CH(Me)SCH2CH2OEt CH2(D1-85a)
CH(Me)SCH2CH2OEt CH2(D1-87a)
CH(Me)SCH2CH2OEt CH2(D1-92a)
CH(Me)SCH2CH2OEt CH2(D1-93a)
CH(Me)SCH2CH2OEt CH2(D1-95a)
CH(Me)SCH2CH2OEt CH2(D1-96a)
CH(Me)SCH2CH2OEt CH2(D1-98a)
CH(Me)SCH2CH2OEt CH2(D1-108a)
CH(Me)SCH2CH2OEt CH2(D1-108b,Z=2-Cl)
CH(Me)SCH2CH2OEt CH2(D1-108b,Z=3-Me)
CH(Me)SCH2CH2OEt CH2(D1-108b,Z=4-OEt)
CH(Me)SCH2CH2OEt CH2(D1-108b,Z=2-SMe)
CH(Me)SCH2CH2OEt CH2(D1-108b,Z=3-CF3)
CH(Me)SCH2CH2OEt CH2(D1-108b,Z=4-OCF3)
CH(Me)SCH2CH2OEt CH2(D1-108b,Z=2-SCF3)
CH(Me)SCH2CH2OEt CH2CH2CN
CH(Me)SCH2CH2OEt CH2CH2CF3
CH(Me)SCH2CH2OEt CH2CH2OEt
CH(Me)SCH2CH2OEt CH2CH2SMe
CH(Me)SCH2CH2OEt CH2CH2S(O)Me
CH(Me)SCH2CH2OEt CH2CH2S(O)2Me
CH(Me)SCH2CH2OEt D1-32a
CH(Me)SCH2CH2OEt D1-33a
CH(Me)SCH2CH2OEt D1-34a
CH(Me)SCH2CH2OEt D1-37a
CH(Me)SCH2CH2OEt D1-81a
CH(Me)SCH2CH2OEt D1-82a
CH(Me)SCH2CH2OEt D1-84a
CH(Me)SCH2CH2OEt D1-85a
CH(Me)SCH2CH2OEt D1-87a
CH(Me)SCH2CH2OEt D1-92a
CH(Me)SCH2CH2OEt D1-93a
CH(Me)SCH2CH2OEt D1-95a
CH(Me)SCH2CH2OEt D1-96a
CH(Me)SCH2CH2OEt D1-98a
CH(Me)SCH2CH2OEt D1-108a
CH(Me)SCH2CH2OEt D1-108b(Z=2-Cl)
CH(Me)SCH2CH2OEt D1-108b(Z=3-Me)
CH(Me)SCH2CH2OEt D1-108b(Z=4-OEt)
CH(Me)SCH2CH2OEt D1-108b(Z=2-SMe)
CH(Me)SCH2CH2OEt D1-108b(Z=3-CF3)
CH(Me)SCH2CH2OEt D1-108b(Z=4-OCF3)
CH(Me)SCH2CH2OEt D1-108b(Z=2-SCF3)
CH(Me)SCH2CH2OEt C(O)Me
CH(Me)SCH2CH2OEt C(O)CF3
CH(Me)SCH2CH2OEt C(O)OEt
CH(Me)S(O)CH2CH2OEt Me
CH(Me)S(O)CH2CH2OEt Et
CH(Me)S(O)CH2CH2OEt Pr-n
CH(Me)S(O)CH2CH2OEt Pr-i
CH(Me)S(O)CH2CH2OEt Pr-c
CH(Me)S(O)CH2CH2OEt Bu-n
CH(Me)S(O)CH2CH2OEt Bu-i
CH(Me)S(O)CH2CH2OEt Bu-c
CH(Me)S(O)CH2CH2OEt Bu-s
CH(Me)S(O)CH2CH2OEt Bu-t
CH(Me)S(O)CH2CH2OEt Pen-n
CH(Me)S(O)CH2CH2OEt Pen-c
CH(Me)S(O)CH2CH2OEt Hex-n
CH(Me)S(O)CH2CH2OEt Hex-c
CH(Me)S(O)CH2CH2OEt CH2Pr-c
CH(Me)S(O)CH2CH2OEt CH2Bu-c
CH(Me)S(O)CH2CH2OEt CH2Pen-c
CH(Me)S(O)CH2CH2OEt CH2Hex-c
CH(Me)S(O)CH2CH2OEt CH2CH=CH2
CH(Me)S(O)CH2CH2OEt CH2CH=C(Cl)2
CH(Me)S(O)CH2CH2OEt CH2C≡CH
CH(Me)S(O)CH2CH2OEt CH2CN
CH(Me)S(O)CH2CH2OEt CH2CF3
CH(Me)S(O)CH2CH2OEt CH2OEt
CH(Me)S(O)CH2CH2OEt CH2OCF3
CH(Me)S(O)CH2CH2OEt CH2SMe
CH(Me)S(O)CH2CH2OEt CH2S(O)Me
CH(Me)S(O)CH2CH2OEt CH2S(O)2Me
CH(Me)S(O)CH2CH2OEt CH2SCF3
CH(Me)S(O)CH2CH2OEt CH2S(O)CF3
CH(Me)S(O)CH2CH2OEt CH2S(O)2CF3
CH(Me)S(O)CH2CH2OEt CH2CH(OEt)2
CH(Me)S(O)CH2CH2OEt CH2CH(SMe)2
CH(Me)S(O)CH2CH2OEt CH2C(O)Me
CH(Me)S(O)CH2CH2OEt CH2C(O)CF3
CH(Me)S(O)CH2CH2OEt CH2C(O)OEt
CH(Me)S(O)CH2CH2OEt CH2(D1-32a)
CH(Me)S(O)CH2CH2OEt CH2(D1-33a)
CH(Me)S(O)CH2CH2OEt CH2(D1-34a)
CH(Me)S(O)CH2CH2OEt CH2(D1-37a)
CH(Me)S(O)CH2CH2OEt CH2(D1-81a)
CH(Me)S(O)CH2CH2OEt CH2(D1-82a)
CH(Me)S(O)CH2CH2OEt CH2(D1-84a)
CH(Me)S(O)CH2CH2OEt CH2(D1-85a)
CH(Me)S(O)CH2CH2OEt CH2(D1-87a)
CH(Me)S(O)CH2CH2OEt CH2(D1-92a)
CH(Me)S(O)CH2CH2OEt CH2(D1-93a)
CH(Me)S(O)CH2CH2OEt CH2(D1-95a)
CH(Me)S(O)CH2CH2OEt CH2(D1-96a)
CH(Me)S(O)CH2CH2OEt CH2(D1-98a)
CH(Me)S(O)CH2CH2OEt CH2(D1-108a)
CH(Me)S(O)CH2CH2OEt CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)CH2CH2OEt CH2(D1-108b,Z=3-Me)
CH(Me)S(O)CH2CH2OEt CH2(D1-108b,Z=4-OEt)
CH(Me)S(O)CH2CH2OEt CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)CH2CH2OEt CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)CH2CH2OEt CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)CH2CH2OEt CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)CH2CH2OEt CH2CH2CN
CH(Me)S(O)CH2CH2OEt CH2CH2CF3
CH(Me)S(O)CH2CH2OEt CH2CH2OEt
CH(Me)S(O)CH2CH2OEt CH2CH2SMe
CH(Me)S(O)CH2CH2OEt CH2CH2S(O)Me
CH(Me)S(O)CH2CH2OEt CH2CH2S(O)2Me
CH(Me)S(O)CH2CH2OEt D1-32a
CH(Me)S(O)CH2CH2OEt D1-33a
CH(Me)S(O)CH2CH2OEt D1-34a
CH(Me)S(O)CH2CH2OEt D1-37a
CH(Me)S(O)CH2CH2OEt D1-81a
CH(Me)S(O)CH2CH2OEt D1-82a
CH(Me)S(O)CH2CH2OEt D1-84a
CH(Me)S(O)CH2CH2OEt D1-85a
CH(Me)S(O)CH2CH2OEt D1-87a
CH(Me)S(O)CH2CH2OEt D1-92a
CH(Me)S(O)CH2CH2OEt D1-93a
CH(Me)S(O)CH2CH2OEt D1-95a
CH(Me)S(O)CH2CH2OEt D1-96a
CH(Me)S(O)CH2CH2OEt D1-98a
CH(Me)S(O)CH2CH2OEt D1-108a
CH(Me)S(O)CH2CH2OEt D1-108b(Z=2-Cl)
CH(Me)S(O)CH2CH2OEt D1-108b(Z=3-Me)
CH(Me)S(O)CH2CH2OEt D1-108b(Z=4-OEt)
CH(Me)S(O)CH2CH2OEt D1-108b(Z=2-SMe)
CH(Me)S(O)CH2CH2OEt D1-108b(Z=3-CF3)
CH(Me)S(O)CH2CH2OEt D1-108b(Z=4-OCF3)
CH(Me)S(O)CH2CH2OEt D1-108b(Z=2-SCF3)
CH(Me)S(O)CH2CH2OEt C(O)Me
CH(Me)S(O)CH2CH2OEt C(O)CF3
CH(Me)S(O)CH2CH2OEt C(O)OEt
CH(Me)S(O)2CH2CH2OEt Me
CH(Me)S(O)2CH2CH2OEt Et
CH(Me)S(O)2CH2CH2OEt Pr-n
CH(Me)S(O)2CH2CH2OEt Pr-i
CH(Me)S(O)2CH2CH2OEt Pr-c
CH(Me)S(O)2CH2CH2OEt Bu-n
CH(Me)S(O)2CH2CH2OEt Bu-i
CH(Me)S(O)2CH2CH2OEt Bu-c
CH(Me)S(O)2CH2CH2OEt Bu-s
CH(Me)S(O)2CH2CH2OEt Bu-t
CH(Me)S(O)2CH2CH2OEt Pen-n
CH(Me)S(O)2CH2CH2OEt Pen-c
CH(Me)S(O)2CH2CH2OEt Hex-n
CH(Me)S(O)2CH2CH2OEt Hex-c
CH(Me)S(O)2CH2CH2OEt CH2Pr-c
CH(Me)S(O)2CH2CH2OEt CH2Bu-c
CH(Me)S(O)2CH2CH2OEt CH2Pen-c
CH(Me)S(O)2CH2CH2OEt CH2Hex-c
CH(Me)S(O)2CH2CH2OEt CH2CH=CH2
CH(Me)S(O)2CH2CH2OEt CH2CH=C(Cl)2
CH(Me)S(O)2CH2CH2OEt CH2C≡CH
CH(Me)S(O)2CH2CH2OEt CH2CN
CH(Me)S(O)2CH2CH2OEt CH2CF3
CH(Me)S(O)2CH2CH2OEt CH2OEt
CH(Me)S(O)2CH2CH2OEt CH2OCF3
CH(Me)S(O)2CH2CH2OEt CH2SMe
CH(Me)S(O)2CH2CH2OEt CH2S(O)Me
CH(Me)S(O)2CH2CH2OEt CH2S(O)2Me
CH(Me)S(O)2CH2CH2OEt CH2SCF3
CH(Me)S(O)2CH2CH2OEt CH2S(O)CF3
CH(Me)S(O)2CH2CH2OEt CH2S(O)2CF3
CH(Me)S(O)2CH2CH2OEt CH2CH(OEt)2
CH(Me)S(O)2CH2CH2OEt CH2CH(SMe)2
CH(Me)S(O)2CH2CH2OEt CH2C(O)Me
CH(Me)S(O)2CH2CH2OEt CH2C(O)CF3
CH(Me)S(O)2CH2CH2OEt CH2C(O)OEt
CH(Me)S(O)2CH2CH2OEt CH2(D1-32a)
CH(Me)S(O)2CH2CH2OEt CH2(D1-33a)
CH(Me)S(O)2CH2CH2OEt CH2(D1-34a)
CH(Me)S(O)2CH2CH2OEt CH2(D1-37a)
CH(Me)S(O)2CH2CH2OEt CH2(D1-81a)
CH(Me)S(O)2CH2CH2OEt CH2(D1-82a)
CH(Me)S(O)2CH2CH2OEt CH2(D1-84a)
CH(Me)S(O)2CH2CH2OEt CH2(D1-85a)
CH(Me)S(O)2CH2CH2OEt CH2(D1-87a)
CH(Me)S(O)2CH2CH2OEt CH2(D1-92a)
CH(Me)S(O)2CH2CH2OEt CH2(D1-93a)
CH(Me)S(O)2CH2CH2OEt CH2(D1-95a)
CH(Me)S(O)2CH2CH2OEt CH2(D1-96a)
CH(Me)S(O)2CH2CH2OEt CH2(D1-98a)
CH(Me)S(O)2CH2CH2OEt CH2(D1-108a)
CH(Me)S(O)2CH2CH2OEt CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)2CH2CH2OEt CH2(D1-108b,Z=3-Me)
CH(Me)S(O)2CH2CH2OEt CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)2CH2CH2OEt CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)2CH2CH2OEt CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)2CH2CH2OEt CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)2CH2CH2OEt CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)2CH2CH2OEt CH2CH2CN
CH(Me)S(O)2CH2CH2OEt CH2CH2CF3
CH(Me)S(O)2CH2CH2OEt CH2CH2OMe
CH(Me)S(O)2CH2CH2OEt CH2CH2SMe
CH(Me)S(O)2CH2CH2OEt CH2CH2S(O)Me
CH(Me)S(O)2CH2CH2OEt CH2CH2S(O)2Me
CH(Me)S(O)2CH2CH2OEt D1-32a
CH(Me)S(O)2CH2CH2OEt D1-33a
CH(Me)S(O)2CH2CH2OEt D1-34a
CH(Me)S(O)2CH2CH2OEt D1-37a
CH(Me)S(O)2CH2CH2OEt D1-81a
CH(Me)S(O)2CH2CH2OEt D1-82a
CH(Me)S(O)2CH2CH2OEt D1-84a
CH(Me)S(O)2CH2CH2OEt D1-85a
CH(Me)S(O)2CH2CH2OEt D1-87a
CH(Me)S(O)2CH2CH2OEt D1-92a
CH(Me)S(O)2CH2CH2OEt D1-93a
CH(Me)S(O)2CH2CH2OEt D1-95a
CH(Me)S(O)2CH2CH2OEt D1-96a
CH(Me)S(O)2CH2CH2OEt D1-98a
CH(Me)S(O)2CH2CH2OEt D1-108a
CH(Me)S(O)2CH2CH2OEt D1-108b(Z=2-Cl)
CH(Me)S(O)2CH2CH2OEt D1-108b(Z=3-Me)
CH(Me)S(O)2CH2CH2OEt D1-108b(Z=4-OMe)
CH(Me)S(O)2CH2CH2OEt D1-108b(Z=2-SMe)
CH(Me)S(O)2CH2CH2OEt D1-108b(Z=3-CF3)
CH(Me)S(O)2CH2CH2OEt D1-108b(Z=4-OCF3)
CH(Me)S(O)2CH2CH2OEt D1-108b(Z=2-SCF3)
CH(Me)S(O)2CH2CH2OEt C(O)Me
CH(Me)S(O)2CH2CH2OEt C(O)CF3
CH(Me)S(O)2CH2CH2OEt C(O)OEt
CH(Et)SCH2CH2OEt Me
CH(Et)SCH2CH2OEt Et
CH(Et)SCH2CH2OEt Pr-n
CH(Et)SCH2CH2OEt Pr-i
CH(Et)SCH2CH2OEt Pr-c
CH(Et)SCH2CH2OEt Bu-n
CH(Et)SCH2CH2OEt Bu-i
CH(Et)SCH2CH2OEt Bu-c
CH(Et)SCH2CH2OEt Bu-s
CH(Et)SCH2CH2OEt Bu-t
CH(Et)SCH2CH2OEt Pen-n
CH(Et)SCH2CH2OEt Pen-c
CH(Et)SCH2CH2OEt Hex-n
CH(Et)SCH2CH2OEt Hex-c
CH(Et)SCH2CH2OEt CH2Pr-c
CH(Et)SCH2CH2OEt CH2Bu-c
CH(Et)SCH2CH2OEt CH2Pen-c
CH(Et)SCH2CH2OEt CH2Hex-c
CH(Et)SCH2CH2OEt CH2CH=CH2
CH(Et)SCH2CH2OEt CH2CH=C(Cl)2
CH(Et)SCH2CH2OEt CH2C≡CH
CH(Et)SCH2CH2OEt CH2CN
CH(Et)SCH2CH2OEt CH2CF3
CH(Et)SCH2CH2OEt CH2OMe
CH(Et)SCH2CH2OEt CH2OCF3
CH(Et)SCH2CH2OEt CH2SMe
CH(Et)SCH2CH2OEt CH2S(O)Me
CH(Et)SCH2CH2OEt CH2S(O)2Me
CH(Et)SCH2CH2OEt CH2SCF3
CH(Et)SCH2CH2OEt CH2S(O)CF3
CH(Et)SCH2CH2OEt CH2S(O)2CF3
CH(Et)SCH2CH2OEt CH2CH(OMe)2
CH(Et)SCH2CH2OEt CH2CH(SMe)2
CH(Et)SCH2CH2OEt CH2C(O)Me
CH(Et)SCH2CH2OEt CH2C(O)CF3
CH(Et)SCH2CH2OEt CH2C(O)OMe
CH(Et)SCH2CH2OEt CH2(D1-32a)
CH(Et)SCH2CH2OEt CH2(D1-33a)
CH(Et)SCH2CH2OEt CH2(D1-34a)
CH(Et)SCH2CH2OEt CH2(D1-37a)
CH(Et)SCH2CH2OEt CH2(D1-81a)
CH(Et)SCH2CH2OEt CH2(D1-82a)
CH(Et)SCH2CH2OEt CH2(D1-84a)
CH(Et)SCH2CH2OEt CH2(D1-85a)
CH(Et)SCH2CH2OEt CH2(D1-87a)
CH(Et)SCH2CH2OEt CH2(D1-92a)
CH(Et)SCH2CH2OEt CH2(D1-93a)
CH(Et)SCH2CH2OEt CH2(D1-95a)
CH(Et)SCH2CH2OEt CH2(D1-96a)
CH(Et)SCH2CH2OEt CH2(D1-98a)
CH(Et)SCH2CH2OEt CH2(D1-108a)
CH(Et)SCH2CH2OEt CH2(D1-108b,Z=2-Cl)
CH(Et)SCH2CH2OEt CH2(D1-108b,Z=3-Me)
CH(Et)SCH2CH2OEt CH2(D1-108b,Z=4-OMe)
CH(Et)SCH2CH2OEt CH2(D1-108b,Z=2-SMe)
CH(Et)SCH2CH2OEt CH2(D1-108b,Z=3-CF3)
CH(Et)SCH2CH2OEt CH2(D1-108b,Z=4-OCF3)
CH(Et)SCH2CH2OEt CH2(D1-108b,Z=2-SCF3)
CH(Et)SCH2CH2OEt CH2CH2CN
CH(Et)SCH2CH2OEt CH2CH2CF3
CH(Et)SCH2CH2OEt CH2CH2OMe
CH(Et)SCH2CH2OEt CH2CH2SMe
CH(Et)SCH2CH2OEt CH2CH2S(O)Me
CH(Et)SCH2CH2OEt CH2CH2S(O)2Me
CH(Et)SCH2CH2OEt D1-32a
CH(Et)SCH2CH2OEt D1-33a
CH(Et)SCH2CH2OEt D1-34a
CH(Et)SCH2CH2OEt D1-37a
CH(Et)SCH2CH2OEt D1-81a
CH(Et)SCH2CH2OEt D1-82a
CH(Et)SCH2CH2OEt D1-84a
CH(Et)SCH2CH2OEt D1-85a
CH(Et)SCH2CH2OEt D1-87a
CH(Et)SCH2CH2OEt D1-92a
CH(Et)SCH2CH2OEt D1-93a
CH(Et)SCH2CH2OEt D1-95a
CH(Et)SCH2CH2OEt D1-96a
CH(Et)SCH2CH2OEt D1-98a
CH(Et)SCH2CH2OEt D1-108a
CH(Et)SCH2CH2OEt D1-108b(Z=2-Cl)
CH(Et)SCH2CH2OEt D1-108b(Z=3-Me)
CH(Et)SCH2CH2OEt D1-108b(Z=4-OMe)
CH(Et)SCH2CH2OEt D1-108b(Z=2-SMe)
CH(Et)SCH2CH2OEt D1-108b(Z=3-CF3)
CH(Et)SCH2CH2OEt D1-108b(Z=4-OCF3)
CH(Et)SCH2CH2OEt D1-108b(Z=2-SCF3)
CH(Et)SCH2CH2OEt C(O)Me
CH(Et)SCH2CH2OEt C(O)CF3
CH(Et)SCH2CH2OEt C(O)OMe
CH(Et)S(O)CH2CH2OEt Me
CH(Et)S(O)CH2CH2OEt Et
CH(Et)S(O)CH2CH2OEt Pr-n
CH(Et)S(O)CH2CH2OEt Pr-i
CH(Et)S(O)CH2CH2OEt Pr-c
CH(Et)S(O)CH2CH2OEt Bu-n
CH(Et)S(O)CH2CH2OEt Bu-i
CH(Et)S(O)CH2CH2OEt Bu-c
CH(Et)S(O)CH2CH2OEt Bu-s
CH(Et)S(O)CH2CH2OEt Bu-t
CH(Et)S(O)CH2CH2OEt Pen-n
CH(Et)S(O)CH2CH2OEt Pen-c
CH(Et)S(O)CH2CH2OEt Hex-n
CH(Et)S(O)CH2CH2OEt Hex-c
CH(Et)S(O)CH2CH2OEt CH2Pr-c
CH(Et)S(O)CH2CH2OEt CH2Bu-c
CH(Et)S(O)CH2CH2OEt CH2Pen-c
CH(Et)S(O)CH2CH2OEt CH2Hex-c
CH(Et)S(O)CH2CH2OEt CH2CH=CH2
CH(Et)S(O)CH2CH2OEt CH2CH=C(Cl)2
CH(Et)S(O)CH2CH2OEt CH2C≡CH
CH(Et)S(O)CH2CH2OEt CH2CN
CH(Et)S(O)CH2CH2OEt CH2CF3
CH(Et)S(O)CH2CH2OEt CH2OMe
CH(Et)S(O)CH2CH2OEt CH2OCF3
CH(Et)S(O)CH2CH2OEt CH2SMe
CH(Et)S(O)CH2CH2OEt CH2S(O)Me
CH(Et)S(O)CH2CH2OEt CH2S(O)2Me
CH(Et)S(O)CH2CH2OEt CH2SCF3
CH(Et)S(O)CH2CH2OEt CH2S(O)CF3
CH(Et)S(O)CH2CH2OEt CH2S(O)2CF3
CH(Et)S(O)CH2CH2OEt CH2CH(OMe)2
CH(Et)S(O)CH2CH2OEt CH2CH(SMe)2
CH(Et)S(O)CH2CH2OEt CH2C(O)Me
CH(Et)S(O)CH2CH2OEt CH2C(O)CF3
CH(Et)S(O)CH2CH2OEt CH2C(O)OMe
CH(Et)S(O)CH2CH2OEt CH2(D1-32a)
CH(Et)S(O)CH2CH2OEt CH2(D1-33a)
CH(Et)S(O)CH2CH2OEt CH2(D1-34a)
CH(Et)S(O)CH2CH2OEt CH2(D1-37a)
CH(Et)S(O)CH2CH2OEt CH2(D1-81a)
CH(Et)S(O)CH2CH2OEt CH2(D1-82a)
CH(Et)S(O)CH2CH2OEt CH2(D1-84a)
CH(Et)S(O)CH2CH2OEt CH2(D1-85a)
CH(Et)S(O)CH2CH2OEt CH2(D1-87a)
CH(Et)S(O)CH2CH2OEt CH2(D1-92a)
CH(Et)S(O)CH2CH2OEt CH2(D1-93a)
CH(Et)S(O)CH2CH2OEt CH2(D1-95a)
CH(Et)S(O)CH2CH2OEt CH2(D1-96a)
CH(Et)S(O)CH2CH2OEt CH2(D1-98a)
CH(Et)S(O)CH2CH2OEt CH2(D1-108a)
CH(Et)S(O)CH2CH2OEt CH2(D1-108b,Z=2-Cl)
CH(Et)S(O)CH2CH2OEt CH2(D1-108b,Z=3-Me)
CH(Et)S(O)CH2CH2OEt CH2(D1-108b,Z=4-OMe)
CH(Et)S(O)CH2CH2OEt CH2(D1-108b,Z=2-SMe)
CH(Et)S(O)CH2CH2OEt CH2(D1-108b,Z=3-CF3)
CH(Et)S(O)CH2CH2OEt CH2(D1-108b,Z=4-OCF3)
CH(Et)S(O)CH2CH2OEt CH2(D1-108b,Z=2-SCF3)
CH(Et)S(O)CH2CH2OEt CH2CH2CN
CH(Et)S(O)CH2CH2OEt CH2CH2CF3
CH(Et)S(O)CH2CH2OEt CH2CH2OMe
CH(Et)S(O)CH2CH2OEt CH2CH2SMe
CH(Et)S(O)CH2CH2OEt CH2CH2S(O)Me
CH(Et)S(O)CH2CH2OEt CH2CH2S(O)2Me
CH(Et)S(O)CH2CH2OEt D1-32a
CH(Et)S(O)CH2CH2OEt D1-33a
CH(Et)S(O)CH2CH2OEt D1-34a
CH(Et)S(O)CH2CH2OEt D1-37a
CH(Et)S(O)CH2CH2OEt D1-81a
CH(Et)S(O)CH2CH2OEt D1-82a
CH(Et)S(O)CH2CH2OEt D1-84a
CH(Et)S(O)CH2CH2OEt D1-85a
CH(Et)S(O)CH2CH2OEt D1-87a
CH(Et)S(O)CH2CH2OEt D1-92a
CH(Et)S(O)CH2CH2OEt D1-93a
CH(Et)S(O)CH2CH2OEt D1-95a
CH(Et)S(O)CH2CH2OEt D1-96a
CH(Et)S(O)CH2CH2OEt D1-98a
CH(Et)S(O)CH2CH2OEt D1-108a
CH(Et)S(O)CH2CH2OEt D1-108b(Z=2-Cl)
CH(Et)S(O)CH2CH2OEt D1-108b(Z=3-Me)
CH(Et)S(O)CH2CH2OEt D1-108b(Z=4-OMe)
CH(Et)S(O)CH2CH2OEt D1-108b(Z=2-SMe)
CH(Et)S(O)CH2CH2OEt D1-108b(Z=3-CF3)
CH(Et)S(O)CH2CH2OEt D1-108b(Z=4-OCF3)
CH(Et)S(O)CH2CH2OEt D1-108b(Z=2-SCF3)
CH(Et)S(O)CH2CH2OEt C(O)Me
CH(Et)S(O)CH2CH2OEt C(O)CF3
CH(Et)S(O)CH2CH2OEt C(O)OMe
CH(Et)S(O)2CH2CH2OEt Me
CH(Et)S(O)2CH2CH2OEt Et
CH(Et)S(O)2CH2CH2OEt Pr-n
CH(Et)S(O)2CH2CH2OEt Pr-i
CH(Et)S(O)2CH2CH2OEt Pr-c
CH(Et)S(O)2CH2CH2OEt Bu-n
CH(Et)S(O)2CH2CH2OEt Bu-i
CH(Et)S(O)2CH2CH2OEt Bu-c
CH(Et)S(O)2CH2CH2OEt Bu-s
CH(Et)S(O)2CH2CH2OEt Bu-t
CH(Et)S(O)2CH2CH2OEt Pen-n
CH(Et)S(O)2CH2CH2OEt Pen-c
CH(Et)S(O)2CH2CH2OEt Hex-n
CH(Et)S(O)2CH2CH2OEt Hex-c
CH(Et)S(O)2CH2CH2OEt CH2Pr-c
CH(Et)S(O)2CH2CH2OEt CH2Bu-c
CH(Et)S(O)2CH2CH2OEt CH2Pen-c
CH(Et)S(O)2CH2CH2OEt CH2Hex-c
CH(Et)S(O)2CH2CH2OEt CH2CH=CH2
CH(Et)S(O)2CH2CH2OEt CH2CH=C(Cl)2
CH(Et)S(O)2CH2CH2OEt CH2C≡CH
CH(Et)S(O)2CH2CH2OEt CH2CN
CH(Et)S(O)2CH2CH2OEt CH2CF3
CH(Et)S(O)2CH2CH2OEt CH2OMe
CH(Et)S(O)2CH2CH2OEt CH2OCF3
CH(Et)S(O)2CH2CH2OEt CH2SMe
CH(Et)S(O)2CH2CH2OEt CH2S(O)Me
CH(Et)S(O)2CH2CH2OEt CH2S(O)2Me
CH(Et)S(O)2CH2CH2OEt CH2SCF3
CH(Et)S(O)2CH2CH2OEt CH2S(O)CF3
CH(Et)S(O)2CH2CH2OEt CH2S(O)2CF3
CH(Et)S(O)2CH2CH2OEt CH2CH(OMe)2
CH(Et)S(O)2CH2CH2OEt CH2CH(SMe)2
CH(Et)S(O)2CH2CH2OEt CH2C(O)Me
CH(Et)S(O)2CH2CH2OEt CH2C(O)CF3
CH(Et)S(O)2CH2CH2OEt CH2C(O)OMe
CH(Et)S(O)2CH2CH2OEt CH2(D1-32a)
CH(Et)S(O)2CH2CH2OEt CH2(D1-33a)
CH(Et)S(O)2CH2CH2OEt CH2(D1-34a)
CH(Et)S(O)2CH2CH2OEt CH2(D1-37a)
CH(Et)S(O)2CH2CH2OEt CH2(D1-81a)
CH(Et)S(O)2CH2CH2OEt CH2(D1-82a)
CH(Et)S(O)2CH2CH2OEt CH2(D1-84a)
CH(Et)S(O)2CH2CH2OEt CH2(D1-85a)
CH(Et)S(O)2CH2CH2OEt CH2(D1-87a)
CH(Et)S(O)2CH2CH2OEt CH2(D1-92a)
CH(Et)S(O)2CH2CH2OEt CH2(D1-93a)
CH(Et)S(O)2CH2CH2OEt CH2(D1-95a)
CH(Et)S(O)2CH2CH2OEt CH2(D1-96a)
CH(Et)S(O)2CH2CH2OEt CH2(D1-98a)
CH(Et)S(O)2CH2CH2OEt CH2(D1-108a)
CH(Et)S(O)2CH2CH2OEt CH2(D1-108b,Z=2-Cl)
CH(Et)S(O)2CH2CH2OEt CH2(D1-108b,Z=3-Me)
CH(Et)S(O)2CH2CH2OEt CH2(D1-108b,Z=4-OEt)
CH(Et)S(O)2CH2CH2OEt CH2(D1-108b,Z=2-SMe)
CH(Et)S(O)2CH2CH2OEt CH2(D1-108b,Z=3-CF3)
CH(Et)S(O)2CH2CH2OEt CH2(D1-108b,Z=4-OCF3)
CH(Et)S(O)2CH2CH2OEt CH2(D1-108b,Z=2-SCF3)
CH(Et)S(O)2CH2CH2OEt CH2CH2CN
CH(Et)S(O)2CH2CH2OEt CH2CH2CF3
CH(Et)S(O)2CH2CH2OEt CH2CH2OMe
CH(Et)S(O)2CH2CH2OEt CH2CH2SMe
CH(Et)S(O)2CH2CH2OEt CH2CH2S(O)Me
CH(Et)S(O)2CH2CH2OEt CH2CH2S(O)2Me
CH(Et)S(O)2CH2CH2OEt D1-32a
CH(Et)S(O)2CH2CH2OEt D1-33a
CH(Et)S(O)2CH2CH2OEt D1-34a
CH(Et)S(O)2CH2CH2OEt D1-37a
CH(Et)S(O)2CH2CH2OEt D1-81a
CH(Et)S(O)2CH2CH2OEt D1-82a
CH(Et)S(O)2CH2CH2OEt D1-84a
CH(Et)S(O)2CH2CH2OEt D1-85a
CH(Et)S(O)2CH2CH2OEt D1-87a
CH(Et)S(O)2CH2CH2OEt D1-92a
CH(Et)S(O)2CH2CH2OEt D1-93a
CH(Et)S(O)2CH2CH2OEt D1-95a
CH(Et)S(O)2CH2CH2OEt D1-96a
CH(Et)S(O)2CH2CH2OEt D1-98a
CH(Et)S(O)2CH2CH2OEt D1-108a
CH(Et)S(O)2CH2CH2OEt D1-108b(Z=2-Cl)
CH(Et)S(O)2CH2CH2OEt D1-108b(Z=3-Me)
CH(Et)S(O)2CH2CH2OEt D1-108b(Z=4-OMe)
CH(Et)S(O)2CH2CH2OEt D1-108b(Z=2-SMe)
CH(Et)S(O)2CH2CH2OEt D1-108b(Z=3-CF3)
CH(Et)S(O)2CH2CH2OEt D1-108b(Z=4-OCF3)
CH(Et)S(O)2CH2CH2OEt D1-108b(Z=2-SCF3)
CH(Et)S(O)2CH2CH2OEt C(O)Me
CH(Et)S(O)2CH2CH2OEt C(O)CF3
CH(Et)S(O)2CH2CH2OEt C(O)OMe
CH2SCH2(D1-32a) Me
CH2SCH2(D1-32a) Et
CH2SCH2(D1-32a) Pr-n
CH2SCH2(D1-32a) Pr-i
CH2SCH2(D1-32a) Pr-c
CH2SCH2(D1-32a) Bu-n
CH2SCH2(D1-32a) Bu-i
CH2SCH2(D1-32a) Bu-c
CH2SCH2(D1-32a) Bu-s
CH2SCH2(D1-32a) Bu-t
CH2SCH2(D1-32a) Pen-n
CH2SCH2(D1-32a) Pen-c
CH2SCH2(D1-32a) Hex-n
CH2SCH2(D1-32a) Hex-c
CH2SCH2(D1-32a) CH2Pr-c
CH2SCH2(D1-32a) CH2Bu-c
CH2SCH2(D1-32a) CH2Pen-c
CH2SCH2(D1-32a) CH2Hex-c
CH2SCH2(D1-32a) CH2CH=CH2
CH2SCH2(D1-32a) CH2CH=C(Cl)2
CH2SCH2(D1-32a) CH2C≡CH
CH2SCH2(D1-32a) CH2CN
CH2SCH2(D1-32a) CH2CF3
CH2SCH2(D1-32a) CH2OMe
CH2SCH2(D1-32a) CH2OCF3
CH2SCH2(D1-32a) CH2SMe
CH2SCH2(D1-32a) CH2S(O)Me
CH2SCH2(D1-32a) CH2S(O)2Me
CH2SCH2(D1-32a) CH2SCF3
CH2SCH2(D1-32a) CH2S(O)CF3
CH2SCH2(D1-32a) CH2S(O)2CF3
CH2SCH2(D1-32a) CH2CH(OMe)2
CH2SCH2(D1-32a) CH2CH(SMe)2
CH2SCH2(D1-32a) CH2C(O)Me
CH2SCH2(D1-32a) CH2C(O)CF3
CH2SCH2(D1-32a) CH2C(O)OMe
CH2SCH2(D1-32a) CH2(D1-32a)
CH2SCH2(D1-32a) CH2(D1-33a)
CH2SCH2(D1-32a) CH2(D1-34a)
CH2SCH2(D1-32a) CH2(D1-37a)
CH2SCH2(D1-32a) CH2(D1-81a)
CH2SCH2(D1-32a) CH2(D1-82a)
CH2SCH2(D1-32a) CH2(D1-84a)
CH2SCH2(D1-32a) CH2(D1-85a)
CH2SCH2(D1-32a) CH2(D1-87a)
CH2SCH2(D1-32a) CH2(D1-92a)
CH2SCH2(D1-32a) CH2(D1-93a)
CH2SCH2(D1-32a) CH2(D1-95a)
CH2SCH2(D1-32a) CH2(D1-96a)
CH2SCH2(D1-32a) CH2(D1-98a)
CH2SCH2(D1-32a) CH2(D1-108a)
CH2SCH2(D1-32a) CH2(D1-108b,Z=2-Cl)
CH2SCH2(D1-32a) CH2(D1-108b,Z=3-Me)
CH2SCH2(D1-32a) CH2(D1-108b,Z=4-OMe)
CH2SCH2(D1-32a) CH2(D1-108b,Z=2-SMe)
CH2SCH2(D1-32a) CH2(D1-108b,Z=3-CF3)
CH2SCH2(D1-32a) CH2(D1-108b,Z=4-OCF3)
CH2SCH2(D1-32a) CH2(D1-108b,Z=2-SCF3)
CH2SCH2(D1-32a) CH2CH2CN
CH2SCH2(D1-32a) CH2CH2CF3
CH2SCH2(D1-32a) CH2CH2OMe
CH2SCH2(D1-32a) CH2CH2SMe
CH2SCH2(D1-32a) CH2CH2S(O)Me
CH2SCH2(D1-32a) CH2CH2S(O)2Me
CH2SCH2(D1-32a) D1-32a
CH2SCH2(D1-32a) D1-33a
CH2SCH2(D1-32a) D1-34a
CH2SCH2(D1-32a) D1-37a
CH2SCH2(D1-32a) D1-81a
CH2SCH2(D1-32a) D1-82a
CH2SCH2(D1-32a) D1-84a
CH2SCH2(D1-32a) D1-85a
CH2SCH2(D1-32a) D1-87a
CH2SCH2(D1-32a) D1-92a
CH2SCH2(D1-32a) D1-93a
CH2SCH2(D1-32a) D1-95a
CH2SCH2(D1-32a) D1-96a
CH2SCH2(D1-32a) D1-98a
CH2SCH2(D1-32a) D1-108a
CH2SCH2(D1-32a) D1-108b(Z=2-Cl)
CH2SCH2(D1-32a) D1-108b(Z=3-Me)
CH2SCH2(D1-32a) D1-108b(Z=4-OMe)
CH2SCH2(D1-32a) D1-108b(Z=2-SMe)
CH2SCH2(D1-32a) D1-108b(Z=3-CF3)
CH2SCH2(D1-32a) D1-108b(Z=4-OCF3)
CH2SCH2(D1-32a) D1-108b(Z=2-SCF3)
CH2SCH2(D1-32a) C(O)Me
CH2SCH2(D1-32a) C(O)CF3
CH2SCH2(D1-32a) C(O)OMe
CH2S(O)CH2(D1-32a) Me
CH2S(O)CH2(D1-32a) Et
CH2S(O)CH2(D1-32a) Pr-n
CH2S(O)CH2(D1-32a) Pr-i
CH2S(O)CH2(D1-32a) Pr-c
CH2S(O)CH2(D1-32a) Bu-n
CH2S(O)CH2(D1-32a) Bu-i
CH2S(O)CH2(D1-32a) Bu-c
CH2S(O)CH2(D1-32a) Bu-s
CH2S(O)CH2(D1-32a) Bu-t
CH2S(O)CH2(D1-32a) Pen-n
CH2S(O)CH2(D1-32a) Pen-c
CH2S(O)CH2(D1-32a) Hex-n
CH2S(O)CH2(D1-32a) Hex-c
CH2S(O)CH2(D1-32a) CH2Pr-c
CH2S(O)CH2(D1-32a) CH2Bu-c
CH2S(O)CH2(D1-32a) CH2Pen-c
CH2S(O)CH2(D1-32a) CH2Hex-c
CH2S(O)CH2(D1-32a) CH2CH=CH2
CH2S(O)CH2(D1-32a) CH2CH=C(Cl)2
CH2S(O)CH2(D1-32a) CH2C≡CH
CH2S(O)CH2(D1-32a) CH2CN
CH2S(O)CH2(D1-32a) CH2CF3
CH2S(O)CH2(D1-32a) CH2OMe
CH2S(O)CH2(D1-32a) CH2OCF3
CH2S(O)CH2(D1-32a) CH2SMe
CH2S(O)CH2(D1-32a) CH2S(O)Me
CH2S(O)CH2(D1-32a) CH2S(O)2Me
CH2S(O)CH2(D1-32a) CH2SCF3
CH2S(O)CH2(D1-32a) CH2S(O)CF3
CH2S(O)CH2(D1-32a) CH2S(O)2CF3
CH2S(O)CH2(D1-32a) CH2CH(OMe)2
CH2S(O)CH2(D1-32a) CH2CH(SMe)2
CH2S(O)CH2(D1-32a) CH2C(O)Me
CH2S(O)CH2(D1-32a) CH2C(O)CF3
CH2S(O)CH2(D1-32a) CH2C(O)OMe
CH2S(O)CH2(D1-32a) CH2(D1-32a)
CH2S(O)CH2(D1-32a) CH2(D1-33a)
CH2S(O)CH2(D1-32a) CH2(D1-34a)
CH2S(O)CH2(D1-32a) CH2(D1-37a)
CH2S(O)CH2(D1-32a) CH2(D1-81a)
CH2S(O)CH2(D1-32a) CH2(D1-82a)
CH2S(O)CH2(D1-32a) CH2(D1-84a)
CH2S(O)CH2(D1-32a) CH2(D1-85a)
CH2S(O)CH2(D1-32a) CH2(D1-87a)
CH2S(O)CH2(D1-32a) CH2(D1-92a)
CH2S(O)CH2(D1-32a) CH2(D1-93a)
CH2S(O)CH2(D1-32a) CH2(D1-95a)
CH2S(O)CH2(D1-32a) CH2(D1-96a)
CH2S(O)CH2(D1-32a) CH2(D1-98a)
CH2S(O)CH2(D1-32a) CH2(D1-108a)
CH2S(O)CH2(D1-32a) CH2(D1-108b,Z=2-Cl)
CH2S(O)CH2(D1-32a) CH2(D1-108b,Z=3-Me)
CH2S(O)CH2(D1-32a) CH2(D1-108b,Z=4-OMe)
CH2S(O)CH2(D1-32a) CH2(D1-108b,Z=2-SMe)
CH2S(O)CH2(D1-32a) CH2(D1-108b,Z=3-CF3)
CH2S(O)CH2(D1-32a) CH2(D1-108b,Z=4-OCF3)
CH2S(O)CH2(D1-32a) CH2(D1-108b,Z=2-SCF3)
CH2S(O)CH2(D1-32a) CH2CH2CN
CH2S(O)CH2(D1-32a) CH2CH2CF3
CH2S(O)CH2(D1-32a) CH2CH2OMe
CH2S(O)CH2(D1-32a) CH2CH2SMe
CH2S(O)CH2(D1-32a) CH2CH2S(O)Me
CH2S(O)CH2(D1-32a) CH2CH2S(O)2Me
CH2S(O)CH2(D1-32a) D1-32a
CH2S(O)CH2(D1-32a) D1-33a
CH2S(O)CH2(D1-32a) D1-34a
CH2S(O)CH2(D1-32a) D1-37a
CH2S(O)CH2(D1-32a) D1-81a
CH2S(O)CH2(D1-32a) D1-82a
CH2S(O)CH2(D1-32a) D1-84a
CH2S(O)CH2(D1-32a) D1-85a
CH2S(O)CH2(D1-32a) D1-87a
CH2S(O)CH2(D1-32a) D1-92a
CH2S(O)CH2(D1-32a) D1-93a
CH2S(O)CH2(D1-32a) D1-95a
CH2S(O)CH2(D1-32a) D1-96a
CH2S(O)CH2(D1-32a) D1-98a
CH2S(O)CH2(D1-32a) D1-108a
CH2S(O)CH2(D1-32a) D1-108b(Z=2-Cl)
CH2S(O)CH2(D1-32a) D1-108b(Z=3-Me)
CH2S(O)CH2(D1-32a) D1-108b(Z=4-OMe)
CH2S(O)CH2(D1-32a) D1-108b(Z=2-SMe)
CH2S(O)CH2(D1-32a) D1-108b(Z=3-CF3)
CH2S(O)CH2(D1-32a) D1-108b(Z=4-OCF3)
CH2S(O)CH2(D1-32a) D1-108b(Z=2-SCF3)
CH2S(O)CH2(D1-32a) C(O)Me
CH2S(O)CH2(D1-32a) C(O)CF3
CH2S(O)CH2(D1-32a) C(O)OMe
CH2S(O)2CH2(D1-32a) Me
CH2S(O)2CH2(D1-32a) Et
CH2S(O)2CH2(D1-32a) Pr-n
CH2S(O)2CH2(D1-32a) Pr-i
CH2S(O)2CH2(D1-32a) Pr-c
CH2S(O)2CH2(D1-32a) Bu-n
CH2S(O)2CH2(D1-32a) Bu-i
CH2S(O)2CH2(D1-32a) Bu-c
CH2S(O)2CH2(D1-32a) Bu-s
CH2S(O)2CH2(D1-32a) Bu-t
CH2S(O)2CH2(D1-32a) Pen-n
CH2S(O)2CH2(D1-32a) Pen-c
CH2S(O)2CH2(D1-32a) Hex-n
CH2S(O)2CH2(D1-32a) Hex-c
CH2S(O)2CH2(D1-32a) CH2Pr-c
CH2S(O)2CH2(D1-32a) CH2Bu-c
CH2S(O)2CH2(D1-32a) CH2Pen-c
CH2S(O)2CH2(D1-32a) CH2Hex-c
CH2S(O)2CH2(D1-32a) CH2CH=CH2
CH2S(O)2CH2(D1-32a) CH2CH=C(Cl)2
CH2S(O)2CH2(D1-32a) CH2C≡CH
CH2S(O)2CH2(D1-32a) CH2CN
CH2S(O)2CH2(D1-32a) CH2CF3
CH2S(O)2CH2(D1-32a) CH2OMe
CH2S(O)2CH2(D1-32a) CH2OCF3
CH2S(O)2CH2(D1-32a) CH2SMe
CH2S(O)2CH2(D1-32a) CH2S(O)Me
CH2S(O)2CH2(D1-32a) CH2S(O)2Me
CH2S(O)2CH2(D1-32a) CH2SCF3
CH2S(O)2CH2(D1-32a) CH2S(O)CF3
CH2S(O)2CH2(D1-32a) CH2S(O)2CF3
CH2S(O)2CH2(D1-32a) CH2CH(OMe)2
CH2S(O)2CH2(D1-32a) CH2CH(SMe)2
CH2S(O)2CH2(D1-32a) CH2C(O)Me
CH2S(O)2CH2(D1-32a) CH2C(O)CF3
CH2S(O)2CH2(D1-32a) CH2C(O)OMe
CH2S(O)2CH2(D1-32a) CH2(D1-32a)
CH2S(O)2CH2(D1-32a) CH2(D1-33a)
CH2S(O)2CH2(D1-32a) CH2(D1-34a)
CH2S(O)2CH2(D1-32a) CH2(D1-37a)
CH2S(O)2CH2(D1-32a) CH2(D1-81a)
CH2S(O)2CH2(D1-32a) CH2(D1-82a)
CH2S(O)2CH2(D1-32a) CH2(D1-84a)
CH2S(O)2CH2(D1-32a) CH2(D1-85a)
CH2S(O)2CH2(D1-32a) CH2(D1-87a)
CH2S(O)2CH2(D1-32a) CH2(D1-92a)
CH2S(O)2CH2(D1-32a) CH2(D1-93a)
CH2S(O)2CH2(D1-32a) CH2(D1-95a)
CH2S(O)2CH2(D1-32a) CH2(D1-96a)
CH2S(O)2CH2(D1-32a) CH2(D1-98a)
CH2S(O)2CH2(D1-32a) CH2(D1-108a)
CH2S(O)2CH2(D1-32a) CH2(D1-108b,Z=2-Cl)
CH2S(O)2CH2(D1-32a) CH2(D1-108b,Z=3-Me)
CH2S(O)2CH2(D1-32a) CH2(D1-108b,Z=4-OMe)
CH2S(O)2CH2(D1-32a) CH2(D1-108b,Z=2-SMe)
CH2S(O)2CH2(D1-32a) CH2(D1-108b,Z=3-CF3)
CH2S(O)2CH2(D1-32a) CH2(D1-108b,Z=4-OCF3)
CH2S(O)2CH2(D1-32a) CH2(D1-108b,Z=2-SCF3)
CH2S(O)2CH2(D1-32a) CH2CH2CN
CH2S(O)2CH2(D1-32a) CH2CH2CF3
CH2S(O)2CH2(D1-32a) CH2CH2OMe
CH2S(O)2CH2(D1-32a) CH2CH2SMe
CH2S(O)2CH2(D1-32a) CH2CH2S(O)Me
CH2S(O)2CH2(D1-32a) CH2CH2S(O)2Me
CH2S(O)2CH2(D1-32a) D1-32a
CH2S(O)2CH2(D1-32a) D1-33a
CH2S(O)2CH2(D1-32a) D1-34a
CH2S(O)2CH2(D1-32a) D1-37a
CH2S(O)2CH2(D1-32a) D1-81a
CH2S(O)2CH2(D1-32a) D1-82a
CH2S(O)2CH2(D1-32a) D1-84a
CH2S(O)2CH2(D1-32a) D1-85a
CH2S(O)2CH2(D1-32a) D1-87a
CH2S(O)2CH2(D1-32a) D1-92a
CH2S(O)2CH2(D1-32a) D1-93a
CH2S(O)2CH2(D1-32a) D1-95a
CH2S(O)2CH2(D1-32a) D1-96a
CH2S(O)2CH2(D1-32a) D1-98a
CH2S(O)2CH2(D1-32a) D1-108a
CH2S(O)2CH2(D1-32a) D1-108b(Z=2-Cl)
CH2S(O)2CH2(D1-32a) D1-108b(Z=3-Me)
CH2S(O)2CH2(D1-32a) D1-108b(Z=4-OMe)
CH2S(O)2CH2(D1-32a) D1-108b(Z=2-SMe)
CH2S(O)2CH2(D1-32a) D1-108b(Z=3-CF3)
CH2S(O)2CH2(D1-32a) D1-108b(Z=4-OCF3)
CH2S(O)2CH2(D1-32a) D1-108b(Z=2-SCF3)
CH2S(O)2CH2(D1-32a) C(O)Me
CH2S(O)2CH2(D1-32a) C(O)CF3
CH2S(O)2CH2(D1-32a) C(O)OMe
CH(Me)SCH2(D1-32a) Me
CH(Me)SCH2(D1-32a) Et
CH(Me)SCH2(D1-32a) Pr-n
CH(Me)SCH2(D1-32a) Pr-i
CH(Me)SCH2(D1-32a) Pr-c
CH(Me)SCH2(D1-32a) Bu-n
CH(Me)SCH2(D1-32a) Bu-i
CH(Me)SCH2(D1-32a) Bu-c
CH(Me)SCH2(D1-32a) Bu-s
CH(Me)SCH2(D1-32a) Bu-t
CH(Me)SCH2(D1-32a) Pen-n
CH(Me)SCH2(D1-32a) Pen-c
CH(Me)SCH2(D1-32a) Hex-n
CH(Me)SCH2(D1-32a) Hex-c
CH(Me)SCH2(D1-32a) CH2Pr-c
CH(Me)SCH2(D1-32a) CH2Bu-c
CH(Me)SCH2(D1-32a) CH2Pen-c
CH(Me)SCH2(D1-32a) CH2Hex-c
CH(Me)SCH2(D1-32a) CH2CH=CH2
CH(Me)SCH2(D1-32a) CH2CH=C(Cl)2
CH(Me)SCH2(D1-32a) CH2C≡CH
CH(Me)SCH2(D1-32a) CH2CN
CH(Me)SCH2(D1-32a) CH2CF3
CH(Me)SCH2(D1-32a) CH2OMe
CH(Me)SCH2(D1-32a) CH2OCF3
CH(Me)SCH2(D1-32a) CH2SMe
CH(Me)SCH2(D1-32a) CH2S(O)Me
CH(Me)SCH2(D1-32a) CH2S(O)2Me
CH(Me)SCH2(D1-32a) CH2SCF3
CH(Me)SCH2(D1-32a) CH2S(O)CF3
CH(Me)SCH2(D1-32a) CH2S(O)2CF3
CH(Me)SCH2(D1-32a) CH2CH(OMe)2
CH(Me)SCH2(D1-32a) CH2CH(SMe)2
CH(Me)SCH2(D1-32a) CH2C(O)Me
CH(Me)SCH2(D1-32a) CH2C(O)CF3
CH(Me)SCH2(D1-32a) CH2C(O)OMe
CH(Me)SCH2(D1-32a) CH2(D1-32a)
CH(Me)SCH2(D1-32a) CH2(D1-33a)
CH(Me)SCH2(D1-32a) CH2(D1-34a)
CH(Me)SCH2(D1-32a) CH2(D1-37a)
CH(Me)SCH2(D1-32a) CH2(D1-81a)
CH(Me)SCH2(D1-32a) CH2(D1-82a)
CH(Me)SCH2(D1-32a) CH2(D1-84a)
CH(Me)SCH2(D1-32a) CH2(D1-85a)
CH(Me)SCH2(D1-32a) CH2(D1-87a)
CH(Me)SCH2(D1-32a) CH2(D1-92a)
CH(Me)SCH2(D1-32a) CH2(D1-93a)
CH(Me)SCH2(D1-32a) CH2(D1-95a)
CH(Me)SCH2(D1-32a) CH2(D1-96a)
CH(Me)SCH2(D1-32a) CH2(D1-98a)
CH(Me)SCH2(D1-32a) CH2(D1-108a)
CH(Me)SCH2(D1-32a) CH2(D1-108b,Z=2-Cl)
CH(Me)SCH2(D1-32a) CH2(D1-108b,Z=3-Me)
CH(Me)SCH2(D1-32a) CH2(D1-108b,Z=4-OMe)
CH(Me)SCH2(D1-32a) CH2(D1-108b,Z=2-SMe)
CH(Me)SCH2(D1-32a) CH2(D1-108b,Z=3-CF3)
CH(Me)SCH2(D1-32a) CH2(D1-108b,Z=4-OCF3)
CH(Me)SCH2(D1-32a) CH2(D1-108b,Z=2-SCF3)
CH(Me)SCH2(D1-32a) CH2CH2CN
CH(Me)SCH2(D1-32a) CH2CH2CF3
CH(Me)SCH2(D1-32a) CH2CH2OMe
CH(Me)SCH2(D1-32a) CH2CH2SMe
CH(Me)SCH2(D1-32a) CH2CH2S(O)Me
CH(Me)SCH2(D1-32a) CH2CH2S(O)2Me
CH(Me)SCH2(D1-32a) D1-32a
CH(Me)SCH2(D1-32a) D1-33a
CH(Me)SCH2(D1-32a) D1-34a
CH(Me)SCH2(D1-32a) D1-37a
CH(Me)SCH2(D1-32a) D1-81a
CH(Me)SCH2(D1-32a) D1-82a
CH(Me)SCH2(D1-32a) D1-84a
CH(Me)SCH2(D1-32a) D1-85a
CH(Me)SCH2(D1-32a) D1-87a
CH(Me)SCH2(D1-32a) D1-92a
CH(Me)SCH2(D1-32a) D1-93a
CH(Me)SCH2(D1-32a) D1-95a
CH(Me)SCH2(D1-32a) D1-96a
CH(Me)SCH2(D1-32a) D1-98a
CH(Me)SCH2(D1-32a) D1-108a
CH(Me)SCH2(D1-32a) D1-108b(Z=2-Cl)
CH(Me)SCH2(D1-32a) D1-108b(Z=3-Me)
CH(Me)SCH2(D1-32a) D1-108b(Z=4-OMe)
CH(Me)SCH2(D1-32a) D1-108b(Z=2-SMe)
CH(Me)SCH2(D1-32a) D1-108b(Z=3-CF3)
CH(Me)SCH2(D1-32a) D1-108b(Z=4-OCF3)
CH(Me)SCH2(D1-32a) D1-108b(Z=2-SCF3)
CH(Me)SCH2(D1-32a) C(O)Me
CH(Me)SCH2(D1-32a) C(O)CF3
CH(Me)SCH2(D1-32a) C(O)OMe
CH(Me)S(O)CH2(D1-32a) Me
CH(Me)S(O)CH2(D1-32a) Et
CH(Me)S(O)CH2(D1-32a) Pr-n
CH(Me)S(O)CH2(D1-32a) Pr-i
CH(Me)S(O)CH2(D1-32a) Pr-c
CH(Me)S(O)CH2(D1-32a) Bu-n
CH(Me)S(O)CH2(D1-32a) Bu-i
CH(Me)S(O)CH2(D1-32a) Bu-c
CH(Me)S(O)CH2(D1-32a) Bu-s
CH(Me)S(O)CH2(D1-32a) Bu-t
CH(Me)S(O)CH2(D1-32a) Pen-n
CH(Me)S(O)CH2(D1-32a) Pen-c
CH(Me)S(O)CH2(D1-32a) Hex-n
CH(Me)S(O)CH2(D1-32a) Hex-c
CH(Me)S(O)CH2(D1-32a) CH2Pr-c
CH(Me)S(O)CH2(D1-32a) CH2Bu-c
CH(Me)S(O)CH2(D1-32a) CH2Pen-c
CH(Me)S(O)CH2(D1-32a) CH2Hex-c
CH(Me)S(O)CH2(D1-32a) CH2CH=CH2
CH(Me)S(O)CH2(D1-32a) CH2CH=C(Cl)2
CH(Me)S(O)CH2(D1-32a) CH2C≡CH
CH(Me)S(O)CH2(D1-32a) CH2CN
CH(Me)S(O)CH2(D1-32a) CH2CF3
CH(Me)S(O)CH2(D1-32a) CH2OMe
CH(Me)S(O)CH2(D1-32a) CH2OCF3
CH(Me)S(O)CH2(D1-32a) CH2SMe
CH(Me)S(O)CH2(D1-32a) CH2S(O)Me
CH(Me)S(O)CH2(D1-32a) CH2S(O)2Me
CH(Me)S(O)CH2(D1-32a) CH2SCF3
CH(Me)S(O)CH2(D1-32a) CH2S(O)CF3
CH(Me)S(O)CH2(D1-32a) CH2S(O)2CF3
CH(Me)S(O)CH2(D1-32a) CH2CH(OMe)2
CH(Me)S(O)CH2(D1-32a) CH2CH(SMe)2
CH(Me)S(O)CH2(D1-32a) CH2C(O)Me
CH(Me)S(O)CH2(D1-32a) CH2C(O)CF3
CH(Me)S(O)CH2(D1-32a) CH2C(O)OMe
CH(Me)S(O)CH2(D1-32a) CH2(D1-32a)
CH(Me)S(O)CH2(D1-32a) CH2(D1-33a)
CH(Me)S(O)CH2(D1-32a) CH2(D1-34a)
CH(Me)S(O)CH2(D1-32a) CH2(D1-37a)
CH(Me)S(O)CH2(D1-32a) CH2(D1-81a)
CH(Me)S(O)CH2(D1-32a) CH2(D1-82a)
CH(Me)S(O)CH2(D1-32a) CH2(D1-84a)
CH(Me)S(O)CH2(D1-32a) CH2(D1-85a)
CH(Me)S(O)CH2(D1-32a) CH2(D1-87a)
CH(Me)S(O)CH2(D1-32a) CH2(D1-92a)
CH(Me)S(O)CH2(D1-32a) CH2(D1-93a)
CH(Me)S(O)CH2(D1-32a) CH2(D1-95a)
CH(Me)S(O)CH2(D1-32a) CH2(D1-96a)
CH(Me)S(O)CH2(D1-32a) CH2(D1-98a)
CH(Me)S(O)CH2(D1-32a) CH2(D1-108a)
CH(Me)S(O)CH2(D1-32a) CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)CH2(D1-32a) CH2(D1-108b,Z=3-Me)
CH(Me)S(O)CH2(D1-32a) CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)CH2(D1-32a) CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)CH2(D1-32a) CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)CH2(D1-32a) CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)CH2(D1-32a) CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)CH2(D1-32a) CH2CH2CN
CH(Me)S(O)CH2(D1-32a) CH2CH2CF3
CH(Me)S(O)CH2(D1-32a) CH2CH2OMe
CH(Me)S(O)CH2(D1-32a) CH2CH2SMe
CH(Me)S(O)CH2(D1-32a) CH2CH2S(O)Me
CH(Me)S(O)CH2(D1-32a) CH2CH2S(O)2Me
CH(Me)S(O)CH2(D1-32a) D1-32a
CH(Me)S(O)CH2(D1-32a) D1-33a
CH(Me)S(O)CH2(D1-32a) D1-34a
CH(Me)S(O)CH2(D1-32a) D1-37a
CH(Me)S(O)CH2(D1-32a) D1-81a
CH(Me)S(O)CH2(D1-32a) D1-82a
CH(Me)S(O)CH2(D1-32a) D1-84a
CH(Me)S(O)CH2(D1-32a) D1-85a
CH(Me)S(O)CH2(D1-32a) D1-87a
CH(Me)S(O)CH2(D1-32a) D1-92a
CH(Me)S(O)CH2(D1-32a) D1-93a
CH(Me)S(O)CH2(D1-32a) D1-95a
CH(Me)S(O)CH2(D1-32a) D1-96a
CH(Me)S(O)CH2(D1-32a) D1-98a
CH(Me)S(O)CH2(D1-32a) D1-108a
CH(Me)S(O)CH2(D1-32a) D1-108b(Z=2-Cl)
CH(Me)S(O)CH2(D1-32a) D1-108b(Z=3-Me)
CH(Me)S(O)CH2(D1-32a) D1-108b(Z=4-OMe)
CH(Me)S(O)CH2(D1-32a) D1-108b(Z=2-SMe)
CH(Me)S(O)CH2(D1-32a) D1-108b(Z=3-CF3)
CH(Me)S(O)CH2(D1-32a) D1-108b(Z=4-OCF3)
CH(Me)S(O)CH2(D1-32a) D1-108b(Z=2-SCF3)
CH(Me)S(O)CH2(D1-32a) C(O)Me
CH(Me)S(O)CH2(D1-32a) C(O)CF3
CH(Me)S(O)CH2(D1-32a) C(O)OMe
CH(Me)S(O)2CH2(D1-32a) Me
CH(Me)S(O)2CH2(D1-32a) Et
CH(Me)S(O)2CH2(D1-32a) Pr-n
CH(Me)S(O)2CH2(D1-32a) Pr-i
CH(Me)S(O)2CH2(D1-32a) Pr-c
CH(Me)S(O)2CH2(D1-32a) Bu-n
CH(Me)S(O)2CH2(D1-32a) Bu-i
CH(Me)S(O)2CH2(D1-32a) Bu-c
CH(Me)S(O)2CH2(D1-32a) Bu-s
CH(Me)S(O)2CH2(D1-32a) Bu-t
CH(Me)S(O)2CH2(D1-32a) Pen-n
CH(Me)S(O)2CH2(D1-32a) Pen-c
CH(Me)S(O)2CH2(D1-32a) Hex-n
CH(Me)S(O)2CH2(D1-32a) Hex-c
CH(Me)S(O)2CH2(D1-32a) CH2Pr-c
CH(Me)S(O)2CH2(D1-32a) CH2Bu-c
CH(Me)S(O)2CH2(D1-32a) CH2Pen-c
CH(Me)S(O)2CH2(D1-32a) CH2Hex-c
CH(Me)S(O)2CH2(D1-32a) CH2CH=CH2
CH(Me)S(O)2CH2(D1-32a) CH2CH=C(Cl)2
CH(Me)S(O)2CH2(D1-32a) CH2C≡CH
CH(Me)S(O)2CH2(D1-32a) CH2CN
CH(Me)S(O)2CH2(D1-32a) CH2CF3
CH(Me)S(O)2CH2(D1-32a) CH2OMe
CH(Me)S(O)2CH2(D1-32a) CH2OCF3
CH(Me)S(O)2CH2(D1-32a) CH2SMe
CH(Me)S(O)2CH2(D1-32a) CH2S(O)Me
CH(Me)S(O)2CH2(D1-32a) CH2S(O)2Me
CH(Me)S(O)2CH2(D1-32a) CH2SCF3
CH(Me)S(O)2CH2(D1-32a) CH2S(O)CF3
CH(Me)S(O)2CH2(D1-32a) CH2S(O)2CF3
CH(Me)S(O)2CH2(D1-32a) CH2CH(OMe)2
CH(Me)S(O)2CH2(D1-32a) CH2CH(SMe)2
CH(Me)S(O)2CH2(D1-32a) CH2C(O)Me
CH(Me)S(O)2CH2(D1-32a) CH2C(O)CF3
CH(Me)S(O)2CH2(D1-32a) CH2C(O)OMe
CH(Me)S(O)2CH2(D1-32a) CH2(D1-32a)
CH(Me)S(O)2CH2(D1-32a) CH2(D1-33a)
CH(Me)S(O)2CH2(D1-32a) CH2(D1-34a)
CH(Me)S(O)2CH2(D1-32a) CH2(D1-37a)
CH(Me)S(O)2CH2(D1-32a) CH2(D1-81a)
CH(Me)S(O)2CH2(D1-32a) CH2(D1-82a)
CH(Me)S(O)2CH2(D1-32a) CH2(D1-84a)
CH(Me)S(O)2CH2(D1-32a) CH2(D1-85a)
CH(Me)S(O)2CH2(D1-32a) CH2(D1-87a)
CH(Me)S(O)2CH2(D1-32a) CH2(D1-92a)
CH(Me)S(O)2CH2(D1-32a) CH2(D1-93a)
CH(Me)S(O)2CH2(D1-32a) CH2(D1-95a)
CH(Me)S(O)2CH2(D1-32a) CH2(D1-96a)
CH(Me)S(O)2CH2(D1-32a) CH2(D1-98a)
CH(Me)S(O)2CH2(D1-32a) CH2(D1-108a)
CH(Me)S(O)2CH2(D1-32a) CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)2CH2(D1-32a) CH2(D1-108b,Z=3-Me)
CH(Me)S(O)2CH2(D1-32a) CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)2CH2(D1-32a) CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)2CH2(D1-32a) CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)2CH2(D1-32a) CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)2CH2(D1-32a) CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)2CH2(D1-32a) CH2CH2CN
CH(Me)S(O)2CH2(D1-32a) CH2CH2CF3
CH(Me)S(O)2CH2(D1-32a) CH2CH2OMe
CH(Me)S(O)2CH2(D1-32a) CH2CH2SMe
CH(Me)S(O)2CH2(D1-32a) CH2CH2S(O)Me
CH(Me)S(O)2CH2(D1-32a) CH2CH2S(O)2Me
CH(Me)S(O)2CH2(D1-32a) D1-32a
CH(Me)S(O)2CH2(D1-32a) D1-33a
CH(Me)S(O)2CH2(D1-32a) D1-34a
CH(Me)S(O)2CH2(D1-32a) D1-37a
CH(Me)S(O)2CH2(D1-32a) D1-81a
CH(Me)S(O)2CH2(D1-32a) D1-82a
CH(Me)S(O)2CH2(D1-32a) D1-84a
CH(Me)S(O)2CH2(D1-32a) D1-85a
CH(Me)S(O)2CH2(D1-32a) D1-87a
CH(Me)S(O)2CH2(D1-32a) D1-92a
CH(Me)S(O)2CH2(D1-32a) D1-93a
CH(Me)S(O)2CH2(D1-32a) D1-95a
CH(Me)S(O)2CH2(D1-32a) D1-96a
CH(Me)S(O)2CH2(D1-32a) D1-98a
CH(Me)S(O)2CH2(D1-32a) D1-108a
CH(Me)S(O)2CH2(D1-32a) D1-108b(Z=2-Cl)
CH(Me)S(O)2CH2(D1-32a) D1-108b(Z=3-Me)
CH(Me)S(O)2CH2(D1-32a) D1-108b(Z=4-OMe)
CH(Me)S(O)2CH2(D1-32a) D1-108b(Z=2-SMe)
CH(Me)S(O)2CH2(D1-32a) D1-108b(Z=3-CF3)
CH(Me)S(O)2CH2(D1-32a) D1-108b(Z=4-OCF3)
CH(Me)S(O)2CH2(D1-32a) D1-108b(Z=2-SCF3)
CH(Me)S(O)2CH2(D1-32a) C(O)Me
CH(Me)S(O)2CH2(D1-32a) C(O)CF3
CH(Me)S(O)2CH2(D1-32a) C(O)OMe
CH(Et)SCH2(D1-32a) Me
CH(Et)SCH2(D1-32a) Et
CH(Et)SCH2(D1-32a) Pr-n
CH(Et)SCH2(D1-32a) Pr-i
CH(Et)SCH2(D1-32a) Pr-c
CH(Et)SCH2(D1-32a) Bu-n
CH(Et)SCH2(D1-32a) Bu-i
CH(Et)SCH2(D1-32a) Bu-c
CH(Et)SCH2(D1-32a) Bu-s
CH(Et)SCH2(D1-32a) Bu-t
CH(Et)SCH2(D1-32a) Pen-n
CH(Et)SCH2(D1-32a) Pen-c
CH(Et)SCH2(D1-32a) Hex-n
CH(Et)SCH2(D1-32a) Hex-c
CH(Et)SCH2(D1-32a) CH2Pr-c
CH(Et)SCH2(D1-32a) CH2Bu-c
CH(Et)SCH2(D1-32a) CH2Pen-c
CH(Et)SCH2(D1-32a) CH2Hex-c
CH(Et)SCH2(D1-32a) CH2CH=CH2
CH(Et)SCH2(D1-32a) CH2CH=C(Cl)2
CH(Et)SCH2(D1-32a) CH2C≡CH
CH(Et)SCH2(D1-32a) CH2CN
CH(Et)SCH2(D1-32a) CH2CF3
CH(Et)SCH2(D1-32a) CH2OMe
CH(Et)SCH2(D1-32a) CH2OCF3
CH(Et)SCH2(D1-32a) CH2SMe
CH(Et)SCH2(D1-32a) CH2S(O)Me
CH(Et)SCH2(D1-32a) CH2S(O)2Me
CH(Et)SCH2(D1-32a) CH2SCF3
CH(Et)SCH2(D1-32a) CH2S(O)CF3
CH(Et)SCH2(D1-32a) CH2S(O)2CF3
CH(Et)SCH2(D1-32a) CH2CH(OMe)2
CH(Et)SCH2(D1-32a) CH2CH(SMe)2
CH(Et)SCH2(D1-32a) CH2C(O)Me
CH(Et)SCH2(D1-32a) CH2C(O)CF3
CH(Et)SCH2(D1-32a) CH2C(O)OMe
CH(Et)SCH2(D1-32a) CH2(D1-32a)
CH(Et)SCH2(D1-32a) CH2(D1-33a)
CH(Et)SCH2(D1-32a) CH2(D1-34a)
CH(Et)SCH2(D1-32a) CH2(D1-37a)
CH(Et)SCH2(D1-32a) CH2(D1-81a)
CH(Et)SCH2(D1-32a) CH2(D1-82a)
CH(Et)SCH2(D1-32a) CH2(D1-84a)
CH(Et)SCH2(D1-32a) CH2(D1-85a)
CH(Et)SCH2(D1-32a) CH2(D1-87a)
CH(Et)SCH2(D1-32a) CH2(D1-92a)
CH(Et)SCH2(D1-32a) CH2(D1-93a)
CH(Et)SCH2(D1-32a) CH2(D1-95a)
CH(Et)SCH2(D1-32a) CH2(D1-96a)
CH(Et)SCH2(D1-32a) CH2(D1-98a)
CH(Et)SCH2(D1-32a) CH2(D1-108a)
CH(Et)SCH2(D1-32a) CH2(D1-108b,Z=2-Cl)
CH(Et)SCH2(D1-32a) CH2(D1-108b,Z=3-Me)
CH(Et)SCH2(D1-32a) CH2(D1-108b,Z=4-OMe)
CH(Et)SCH2(D1-32a) CH2(D1-108b,Z=2-SMe)
CH(Et)SCH2(D1-32a) CH2(D1-108b,Z=3-CF3)
CH(Et)SCH2(D1-32a) CH2(D1-108b,Z=4-OCF3)
CH(Et)SCH2(D1-32a) CH2(D1-108b,Z=2-SCF3)
CH(Et)SCH2(D1-32a) CH2CH2CN
CH(Et)SCH2(D1-32a) CH2CH2CF3
CH(Et)SCH2(D1-32a) CH2CH2OMe
CH(Et)SCH2(D1-32a) CH2CH2SMe
CH(Et)SCH2(D1-32a) CH2CH2S(O)Me
CH(Et)SCH2(D1-32a) CH2CH2S(O)2Me
CH(Et)SCH2(D1-32a) D1-32a
CH(Et)SCH2(D1-32a) D1-33a
CH(Et)SCH2(D1-32a) D1-34a
CH(Et)SCH2(D1-32a) D1-37a
CH(Et)SCH2(D1-32a) D1-81a
CH(Et)SCH2(D1-32a) D1-82a
CH(Et)SCH2(D1-32a) D1-84a
CH(Et)SCH2(D1-32a) D1-85a
CH(Et)SCH2(D1-32a) D1-87a
CH(Et)SCH2(D1-32a) D1-92a
CH(Et)SCH2(D1-32a) D1-93a
CH(Et)SCH2(D1-32a) D1-95a
CH(Et)SCH2(D1-32a) D1-96a
CH(Et)SCH2(D1-32a) D1-98a
CH(Et)SCH2(D1-32a) D1-108a
CH(Et)SCH2(D1-32a) D1-108b(Z=2-Cl)
CH(Et)SCH2(D1-32a) D1-108b(Z=3-Me)
CH(Et)SCH2(D1-32a) D1-108b(Z=4-OMe)
CH(Et)SCH2(D1-32a) D1-108b(Z=2-SMe)
CH(Et)SCH2(D1-32a) D1-108b(Z=3-CF3)
CH(Et)SCH2(D1-32a) D1-108b(Z=4-OCF3)
CH(Et)SCH2(D1-32a) D1-108b(Z=2-SCF3)
CH(Et)SCH2(D1-32a) C(O)Me
CH(Et)SCH2(D1-32a) C(O)CF3
CH(Et)SCH2(D1-32a) C(O)OMe
CH(Et)S(O)CH2(D1-32a) Me
CH(Et)S(O)CH2(D1-32a) Et
CH(Et)S(O)CH2(D1-32a) Pr-n
CH(Et)S(O)CH2(D1-32a) Pr-i
CH(Et)S(O)CH2(D1-32a) Pr-c
CH(Et)S(O)CH2(D1-32a) Bu-n
CH(Et)S(O)CH2(D1-32a) Bu-i
CH(Et)S(O)CH2(D1-32a) Bu-c
CH(Et)S(O)CH2(D1-32a) Bu-s
CH(Et)S(O)CH2(D1-32a) Bu-t
CH(Et)S(O)CH2(D1-32a) Pen-n
CH(Et)S(O)CH2(D1-32a) Pen-c
CH(Et)S(O)CH2(D1-32a) Hex-n
CH(Et)S(O)CH2(D1-32a) Hex-c
CH(Et)S(O)CH2(D1-32a) CH2Pr-c
CH(Et)S(O)CH2(D1-32a) CH2Bu-c
CH(Et)S(O)CH2(D1-32a) CH2Pen-c
CH(Et)S(O)CH2(D1-32a) CH2Hex-c
CH(Et)S(O)CH2(D1-32a) CH2CH=CH2
CH(Et)S(O)CH2(D1-32a) CH2CH=C(Cl)2
CH(Et)S(O)CH2(D1-32a) CH2C≡CH
CH(Et)S(O)CH2(D1-32a) CH2CN
CH(Et)S(O)CH2(D1-32a) CH2CF3
CH(Et)S(O)CH2(D1-32a) CH2OMe
CH(Et)S(O)CH2(D1-32a) CH2OCF3
CH(Et)S(O)CH2(D1-32a) CH2SMe
CH(Et)S(O)CH2(D1-32a) CH2S(O)Me
CH(Et)S(O)CH2(D1-32a) CH2S(O)2Me
CH(Et)S(O)CH2(D1-32a) CH2SCF3
CH(Et)S(O)CH2(D1-32a) CH2S(O)CF3
CH(Et)S(O)CH2(D1-32a) CH2S(O)2CF3
CH(Et)S(O)CH2(D1-32a) CH2CH(OMe)2
CH(Et)S(O)CH2(D1-32a) CH2CH(SMe)2
CH(Et)S(O)CH2(D1-32a) CH2C(O)Me
CH(Et)S(O)CH2(D1-32a) CH2C(O)CF3
CH(Et)S(O)CH2(D1-32a) CH2C(O)OMe
CH(Et)S(O)CH2(D1-32a) CH2(D1-32a)
CH(Et)S(O)CH2(D1-32a) CH2(D1-33a)
CH(Et)S(O)CH2(D1-32a) CH2(D1-34a)
CH(Et)S(O)CH2(D1-32a) CH2(D1-37a)
CH(Et)S(O)CH2(D1-32a) CH2(D1-81a)
CH(Et)S(O)CH2(D1-32a) CH2(D1-82a)
CH(Et)S(O)CH2(D1-32a) CH2(D1-84a)
CH(Et)S(O)CH2(D1-32a) CH2(D1-85a)
CH(Et)S(O)CH2(D1-32a) CH2(D1-87a)
CH(Et)S(O)CH2(D1-32a) CH2(D1-92a)
CH(Et)S(O)CH2(D1-32a) CH2(D1-93a)
CH(Et)S(O)CH2(D1-32a) CH2(D1-95a)
CH(Et)S(O)CH2(D1-32a) CH2(D1-96a)
CH(Et)S(O)CH2(D1-32a) CH2(D1-98a)
CH(Et)S(O)CH2(D1-32a) CH2(D1-108a)
CH(Et)S(O)CH2(D1-32a) CH2(D1-108b,Z=2-Cl)
CH(Et)S(O)CH2(D1-32a) CH2(D1-108b,Z=3-Me)
CH(Et)S(O)CH2(D1-32a) CH2(D1-108b,Z=4-OMe)
CH(Et)S(O)CH2(D1-32a) CH2(D1-108b,Z=2-SMe)
CH(Et)S(O)CH2(D1-32a) CH2(D1-108b,Z=3-CF3)
CH(Et)S(O)CH2(D1-32a) CH2(D1-108b,Z=4-OCF3)
CH(Et)S(O)CH2(D1-32a) CH2(D1-108b,Z=2-SCF3)
CH(Et)S(O)CH2(D1-32a) CH2CH2CN
CH(Et)S(O)CH2(D1-32a) CH2CH2CF3
CH(Et)S(O)CH2(D1-32a) CH2CH2OMe
CH(Et)S(O)CH2(D1-32a) CH2CH2SMe
CH(Et)S(O)CH2(D1-32a) CH2CH2S(O)Me
CH(Et)S(O)CH2(D1-32a) CH2CH2S(O)2Me
CH(Et)S(O)CH2(D1-32a) D1-32a
CH(Et)S(O)CH2(D1-32a) D1-33a
CH(Et)S(O)CH2(D1-32a) D1-34a
CH(Et)S(O)CH2(D1-32a) D1-37a
CH(Et)S(O)CH2(D1-32a) D1-81a
CH(Et)S(O)CH2(D1-32a) D1-82a
CH(Et)S(O)CH2(D1-32a) D1-84a
CH(Et)S(O)CH2(D1-32a) D1-85a
CH(Et)S(O)CH2(D1-32a) D1-87a
CH(Et)S(O)CH2(D1-32a) D1-92a
CH(Et)S(O)CH2(D1-32a) D1-93a
CH(Et)S(O)CH2(D1-32a) D1-95a
CH(Et)S(O)CH2(D1-32a) D1-96a
CH(Et)S(O)CH2(D1-32a) D1-98a
CH(Et)S(O)CH2(D1-32a) D1-108a
CH(Et)S(O)CH2(D1-32a) D1-108b(Z=2-Cl)
CH(Et)S(O)CH2(D1-32a) D1-108b(Z=3-Me)
CH(Et)S(O)CH2(D1-32a) D1-108b(Z=4-OMe)
CH(Et)S(O)CH2(D1-32a) D1-108b(Z=2-SMe)
CH(Et)S(O)CH2(D1-32a) D1-108b(Z=3-CF3)
CH(Et)S(O)CH2(D1-32a) D1-108b(Z=4-OCF3)
CH(Et)S(O)CH2(D1-32a) D1-108b(Z=2-SCF3)
CH(Et)S(O)CH2(D1-32a) C(O)Me
CH(Et)S(O)CH2(D1-32a) C(O)CF3
CH(Et)S(O)CH2(D1-32a) C(O)OMe
CH(Et)S(O)2CH2(D1-32a) Me
CH(Et)S(O)2CH2(D1-32a) Et
CH(Et)S(O)2CH2(D1-32a) Pr-n
CH(Et)S(O)2CH2(D1-32a) Pr-i
CH(Et)S(O)2CH2(D1-32a) Pr-c
CH(Et)S(O)2CH2(D1-32a) Bu-n
CH(Et)S(O)2CH2(D1-32a) Bu-i
CH(Et)S(O)2CH2(D1-32a) Bu-c
CH(Et)S(O)2CH2(D1-32a) Bu-s
CH(Et)S(O)2CH2(D1-32a) Bu-t
CH(Et)S(O)2CH2(D1-32a) Pen-n
CH(Et)S(O)2CH2(D1-32a) Pen-c
CH(Et)S(O)2CH2(D1-32a) Hex-n
CH(Et)S(O)2CH2(D1-32a) Hex-c
CH(Et)S(O)2CH2(D1-32a) CH2Pr-c
CH(Et)S(O)2CH2(D1-32a) CH2Bu-c
CH(Et)S(O)2CH2(D1-32a) CH2Pen-c
CH(Et)S(O)2CH2(D1-32a) CH2Hex-c
CH(Et)S(O)2CH2(D1-32a) CH2CH=CH2
CH(Et)S(O)2CH2(D1-32a) CH2CH=C(Cl)2
CH(Et)S(O)2CH2(D1-32a) CH2C≡CH
CH(Et)S(O)2CH2(D1-32a) CH2CN
CH(Et)S(O)2CH2(D1-32a) CH2CF3
CH(Et)S(O)2CH2(D1-32a) CH2OMe
CH(Et)S(O)2CH2(D1-32a) CH2OCF3
CH(Et)S(O)2CH2(D1-32a) CH2SMe
CH(Et)S(O)2CH2(D1-32a) CH2S(O)Me
CH(Et)S(O)2CH2(D1-32a) CH2S(O)2Me
CH(Et)S(O)2CH2(D1-32a) CH2SCF3
CH(Et)S(O)2CH2(D1-32a) CH2S(O)CF3
CH(Et)S(O)2CH2(D1-32a) CH2S(O)2CF3
CH(Et)S(O)2CH2(D1-32a) CH2CH(OMe)2
CH(Et)S(O)2CH2(D1-32a) CH2CH(SMe)2
CH(Et)S(O)2CH2(D1-32a) CH2C(O)Me
CH(Et)S(O)2CH2(D1-32a) CH2C(O)CF3
CH(Et)S(O)2CH2(D1-32a) CH2C(O)OMe
CH(Et)S(O)2CH2(D1-32a) CH2(D1-32a)
CH(Et)S(O)2CH2(D1-32a) CH2(D1-33a)
CH(Et)S(O)2CH2(D1-32a) CH2(D1-34a)
CH(Et)S(O)2CH2(D1-32a) CH2(D1-37a)
CH(Et)S(O)2CH2(D1-32a) CH2(D1-81a)
CH(Et)S(O)2CH2(D1-32a) CH2(D1-82a)
CH(Et)S(O)2CH2(D1-32a) CH2(D1-84a)
CH(Et)S(O)2CH2(D1-32a) CH2(D1-85a)
CH(Et)S(O)2CH2(D1-32a) CH2(D1-87a)
CH(Et)S(O)2CH2(D1-32a) CH2(D1-92a)
CH(Et)S(O)2CH2(D1-32a) CH2(D1-93a)
CH(Et)S(O)2CH2(D1-32a) CH2(D1-95a)
CH(Et)S(O)2CH2(D1-32a) CH2(D1-96a)
CH(Et)S(O)2CH2(D1-32a) CH2(D1-98a)
CH(Et)S(O)2CH2(D1-32a) CH2(D1-108a)
CH(Et)S(O)2CH2(D1-32a) CH2(D1-108b,Z=2-Cl)
CH(Et)S(O)2CH2(D1-32a) CH2(D1-108b,Z=3-Me)
CH(Et)S(O)2CH2(D1-32a) CH2(D1-108b,Z=4-OMe)
CH(Et)S(O)2CH2(D1-32a) CH2(D1-108b,Z=2-SMe)
CH(Et)S(O)2CH2(D1-32a) CH2(D1-108b,Z=3-CF3)
CH(Et)S(O)2CH2(D1-32a) CH2(D1-108b,Z=4-OCF3)
CH(Et)S(O)2CH2(D1-32a) CH2(D1-108b,Z=2-SCF3)
CH(Et)S(O)2CH2(D1-32a) CH2CH2CN
CH(Et)S(O)2CH2(D1-32a) CH2CH2CF3
CH(Et)S(O)2CH2(D1-32a) CH2CH2OMe
CH(Et)S(O)2CH2(D1-32a) CH2CH2SMe
CH(Et)S(O)2CH2(D1-32a) CH2CH2S(O)Me
CH(Et)S(O)2CH2(D1-32a) CH2CH2S(O)2Me
CH(Et)S(O)2CH2(D1-32a) D1-32a
CH(Et)S(O)2CH2(D1-32a) D1-33a
CH(Et)S(O)2CH2(D1-32a) D1-34a
CH(Et)S(O)2CH2(D1-32a) D1-37a
CH(Et)S(O)2CH2(D1-32a) D1-81a
CH(Et)S(O)2CH2(D1-32a) D1-82a
CH(Et)S(O)2CH2(D1-32a) D1-84a
CH(Et)S(O)2CH2(D1-32a) D1-85a
CH(Et)S(O)2CH2(D1-32a) D1-87a
CH(Et)S(O)2CH2(D1-32a) D1-92a
CH(Et)S(O)2CH2(D1-32a) D1-93a
CH(Et)S(O)2CH2(D1-32a) D1-95a
CH(Et)S(O)2CH2(D1-32a) D1-96a
CH(Et)S(O)2CH2(D1-32a) D1-98a
CH(Et)S(O)2CH2(D1-32a) D1-108a
CH(Et)S(O)2CH2(D1-32a) D1-108b(Z=2-Cl)
CH(Et)S(O)2CH2(D1-32a) D1-108b(Z=3-Me)
CH(Et)S(O)2CH2(D1-32a) D1-108b(Z=4-OMe)
CH(Et)S(O)2CH2(D1-32a) D1-108b(Z=2-SMe)
CH(Et)S(O)2CH2(D1-32a) D1-108b(Z=3-CF3)
CH(Et)S(O)2CH2(D1-32a) D1-108b(Z=4-OCF3)
CH(Et)S(O)2CH2(D1-32a) D1-108b(Z=2-SCF3)
CH(Et)S(O)2CH2(D1-32a) C(O)Me
CH(Et)S(O)2CH2(D1-32a) C(O)CF3
CH2SCH2(D1-33a) Me
CH2SCH2(D1-33a) Et
CH2SCH2(D1-33a) Pr-n
CH2SCH2(D1-33a) Pr-i
CH2SCH2(D1-33a) Pr-c
CH2SCH2(D1-33a) Bu-n
CH2SCH2(D1-33a) Bu-i
CH2SCH2(D1-33a) Bu-c
CH2SCH2(D1-33a) Bu-s
CH2SCH2(D1-33a) Bu-t
CH2SCH2(D1-33a) Pen-n
CH2SCH2(D1-33a) Pen-c
CH2SCH2(D1-33a) Hex-n
CH2SCH2(D1-33a) Hex-c
CH2SCH2(D1-33a) CH2Pr-c
CH2SCH2(D1-33a) CH2Bu-c
CH2SCH2(D1-33a) CH2Pen-c
CH2SCH2(D1-33a) CH2Hex-c
CH2SCH2(D1-33a) CH2CH=CH2
CH2SCH2(D1-33a) CH2CH=C(Cl)2
CH2SCH2(D1-33a) CH2C≡CH
CH2SCH2(D1-33a) CH2CN
CH2SCH2(D1-33a) CH2CF3
CH2SCH2(D1-33a) CH2OMe
CH2SCH2(D1-33a) CH2OCF3
CH2SCH2(D1-33a) CH2SMe
CH2SCH2(D1-33a) CH2S(O)Me
CH2SCH2(D1-33a) CH2S(O)2Me
CH2SCH2(D1-33a) CH2SCF3
CH2SCH2(D1-33a) CH2S(O)CF3
CH2SCH2(D1-33a) CH2S(O)2CF3
CH2SCH2(D1-33a) CH2CH(OMe)2
CH2SCH2(D1-33a) CH2CH(SMe)2
CH2SCH2(D1-33a) CH2C(O)Me
CH2SCH2(D1-33a) CH2C(O)CF3
CH2SCH2(D1-33a) CH2C(O)OMe
CH2SCH2(D1-33a) CH2(D1-32a)
CH2SCH2(D1-33a) CH2(D1-33a)
CH2SCH2(D1-33a) CH2(D1-34a)
CH2SCH2(D1-33a) CH2(D1-37a)
CH2SCH2(D1-33a) CH2(D1-81a)
CH2SCH2(D1-33a) CH2(D1-82a)
CH2SCH2(D1-33a) CH2(D1-84a)
CH2SCH2(D1-33a) CH2(D1-85a)
CH2SCH2(D1-33a) CH2(D1-87a)
CH2SCH2(D1-33a) CH2(D1-92a)
CH2SCH2(D1-33a) CH2(D1-93a)
CH2SCH2(D1-33a) CH2(D1-95a)
CH2SCH2(D1-33a) CH2(D1-96a)
CH2SCH2(D1-33a) CH2(D1-98a)
CH2SCH2(D1-33a) CH2(D1-108a)
CH2SCH2(D1-33a) CH2(D1-108b,Z=2-Cl)
CH2SCH2(D1-33a) CH2(D1-108b,Z=3-Me)
CH2SCH2(D1-33a) CH2(D1-108b,Z=4-OMe)
CH2SCH2(D1-33a) CH2(D1-108b,Z=2-SMe)
CH2SCH2(D1-33a) CH2(D1-108b,Z=3-CF3)
CH2SCH2(D1-33a) CH2(D1-108b,Z=4-OCF3)
CH2SCH2(D1-33a) CH2(D1-108b,Z=2-SCF3)
CH2SCH2(D1-33a) CH2CH2CN
CH2SCH2(D1-33a) CH2CH2CF3
CH2SCH2(D1-33a) CH2CH2OMe
CH2SCH2(D1-33a) CH2CH2SMe
CH2SCH2(D1-33a) CH2CH2S(O)Me
CH2SCH2(D1-33a) CH2CH2S(O)2Me
CH2SCH2(D1-33a) D1-32a
CH2SCH2(D1-33a) D1-33a
CH2SCH2(D1-33a) D1-34a
CH2SCH2(D1-33a) D1-37a
CH2SCH2(D1-33a) D1-81a
CH2SCH2(D1-33a) D1-82a
CH2SCH2(D1-33a) D1-84a
CH2SCH2(D1-33a) D1-85a
CH2SCH2(D1-33a) D1-87a
CH2SCH2(D1-33a) D1-92a
CH2SCH2(D1-33a) D1-93a
CH2SCH2(D1-33a) D1-95a
CH2SCH2(D1-33a) D1-96a
CH2SCH2(D1-33a) D1-98a
CH2SCH2(D1-33a) D1-108a
CH2SCH2(D1-33a) D1-108b(Z=2-Cl)
CH2SCH2(D1-33a) D1-108b(Z=3-Me)
CH2SCH2(D1-33a) D1-108b(Z=4-OMe)
CH2SCH2(D1-33a) D1-108b(Z=2-SMe)
CH2SCH2(D1-33a) D1-108b(Z=3-CF3)
CH2SCH2(D1-33a) D1-108b(Z=4-OCF3)
CH2SCH2(D1-33a) D1-108b(Z=2-SCF3)
CH2SCH2(D1-33a) C(O)Me
CH2SCH2(D1-33a) C(O)CF3
CH2SCH2(D1-33a) C(O)OMe
CH2S(O)CH2(D1-33a) Me
CH2S(O)CH2(D1-33a) Et
CH2S(O)CH2(D1-33a) Pr-n
CH2S(O)CH2(D1-33a) Pr-i
CH2S(O)CH2(D1-33a) Pr-c
CH2S(O)CH2(D1-33a) Bu-n
CH2S(O)CH2(D1-33a) Bu-i
CH2S(O)CH2(D1-33a) Bu-c
CH2S(O)CH2(D1-33a) Bu-s
CH2S(O)CH2(D1-33a) Bu-t
CH2S(O)CH2(D1-33a) Pen-n
CH2S(O)CH2(D1-33a) Pen-c
CH2S(O)CH2(D1-33a) Hex-n
CH2S(O)CH2(D1-33a) Hex-c
CH2S(O)CH2(D1-33a) CH2Pr-c
CH2S(O)CH2(D1-33a) CH2Bu-c
CH2S(O)CH2(D1-33a) CH2Pen-c
CH2S(O)CH2(D1-33a) CH2Hex-c
CH2S(O)CH2(D1-33a) CH2CH=CH2
CH2S(O)CH2(D1-33a) CH2CH=C(Cl)2
CH2S(O)CH2(D1-33a) CH2C≡CH
CH2S(O)CH2(D1-33a) CH2CN
CH2S(O)CH2(D1-33a) CH2CF3
CH2S(O)CH2(D1-33a) CH2OMe
CH2S(O)CH2(D1-33a) CH2OCF3
CH2S(O)CH2(D1-33a) CH2SMe
CH2S(O)CH2(D1-33a) CH2S(O)Me
CH2S(O)CH2(D1-33a) CH2S(O)2Me
CH2S(O)CH2(D1-33a) CH2SCF3
CH2S(O)CH2(D1-33a) CH2S(O)CF3
CH2S(O)CH2(D1-33a) CH2S(O)2CF3
CH2S(O)CH2(D1-33a) CH2CH(OMe)2
CH2S(O)CH2(D1-33a) CH2CH(SMe)2
CH2S(O)CH2(D1-33a) CH2C(O)Me
CH2S(O)CH2(D1-33a) CH2C(O)CF3
CH2S(O)CH2(D1-33a) CH2C(O)OMe
CH2S(O)CH2(D1-33a) CH2(D1-32a)
CH2S(O)CH2(D1-33a) CH2(D1-33a)
CH2S(O)CH2(D1-33a) CH2(D1-34a)
CH2S(O)CH2(D1-33a) CH2(D1-37a)
CH2S(O)CH2(D1-33a) CH2(D1-81a)
CH2S(O)CH2(D1-33a) CH2(D1-82a)
CH2S(O)CH2(D1-33a) CH2(D1-84a)
CH2S(O)CH2(D1-33a) CH2(D1-85a)
CH2S(O)CH2(D1-33a) CH2(D1-87a)
CH2S(O)CH2(D1-33a) CH2(D1-92a)
CH2S(O)CH2(D1-33a) CH2(D1-93a)
CH2S(O)CH2(D1-33a) CH2(D1-95a)
CH2S(O)CH2(D1-33a) CH2(D1-96a)
CH2S(O)CH2(D1-33a) CH2(D1-98a)
CH2S(O)CH2(D1-33a) CH2(D1-108a)
CH2S(O)CH2(D1-33a) CH2(D1-108b,Z=2-Cl)
CH2S(O)CH2(D1-33a) CH2(D1-108b,Z=3-Me)
CH2S(O)CH2(D1-33a) CH2(D1-108b,Z=4-OMe)
CH2S(O)CH2(D1-33a) CH2(D1-108b,Z=2-SMe)
CH2S(O)CH2(D1-33a) CH2(D1-108b,Z=3-CF3)
CH2S(O)CH2(D1-33a) CH2(D1-108b,Z=4-OCF3)
CH2S(O)CH2(D1-33a) CH2(D1-108b,Z=2-SCF3)
CH2S(O)CH2(D1-33a) CH2CH2CN
CH2S(O)CH2(D1-33a) CH2CH2CF3
CH2S(O)CH2(D1-33a) CH2CH2OMe
CH2S(O)CH2(D1-33a) CH2CH2SMe
CH2S(O)CH2(D1-33a) CH2CH2S(O)Me
CH2S(O)CH2(D1-33a) CH2CH2S(O)2Me
CH2S(O)CH2(D1-33a) D1-32a
CH2S(O)CH2(D1-33a) D1-33a
CH2S(O)CH2(D1-33a) D1-34a
CH2S(O)CH2(D1-33a) D1-37a
CH2S(O)CH2(D1-33a) D1-81a
CH2S(O)CH2(D1-33a) D1-82a
CH2S(O)CH2(D1-33a) D1-84a
CH2S(O)CH2(D1-33a) D1-85a
CH2S(O)CH2(D1-33a) D1-87a
CH2S(O)CH2(D1-33a) D1-92a
CH2S(O)CH2(D1-33a) D1-93a
CH2S(O)CH2(D1-33a) D1-95a
CH2S(O)CH2(D1-33a) D1-96a
CH2S(O)CH2(D1-33a) D1-98a
CH2S(O)CH2(D1-33a) D1-108a
CH2S(O)CH2(D1-33a) D1-108b(Z=2-Cl)
CH2S(O)CH2(D1-33a) D1-108b(Z=3-Me)
CH2S(O)CH2(D1-33a) D1-108b(Z=4-OMe)
CH2S(O)CH2(D1-33a) D1-108b(Z=2-SMe)
CH2S(O)CH2(D1-33a) D1-108b(Z=3-CF3)
CH2S(O)CH2(D1-33a) D1-108b(Z=4-OCF3)
CH2S(O)CH2(D1-33a) D1-108b(Z=2-SCF3)
CH2S(O)CH2(D1-33a) C(O)Me
CH2S(O)CH2(D1-33a) C(O)CF3
CH2S(O)CH2(D1-33a) C(O)OMe
CH2S(O)2CH2(D1-33a) Me
CH2S(O)2CH2(D1-33a) Et
CH2S(O)2CH2(D1-33a) Pr-n
CH2S(O)2CH2(D1-33a) Pr-i
CH2S(O)2CH2(D1-33a) Pr-c
CH2S(O)2CH2(D1-33a) Bu-n
CH2S(O)2CH2(D1-33a) Bu-i
CH2S(O)2CH2(D1-33a) Bu-c
CH2S(O)2CH2(D1-33a) Bu-s
CH2S(O)2CH2(D1-33a) Bu-t
CH2S(O)2CH2(D1-33a) Pen-n
CH2S(O)2CH2(D1-33a) Pen-c
CH2S(O)2CH2(D1-33a) Hex-n
CH2S(O)2CH2(D1-33a) Hex-c
CH2S(O)2CH2(D1-33a) CH2Pr-c
CH2S(O)2CH2(D1-33a) CH2Bu-c
CH2S(O)2CH2(D1-33a) CH2Pen-c
CH2S(O)2CH2(D1-33a) CH2Hex-c
CH2S(O)2CH2(D1-33a) CH2CH=CH2
CH2S(O)2CH2(D1-33a) CH2CH=C(Cl)2
CH2S(O)2CH2(D1-33a) CH2C≡CH
CH2S(O)2CH2(D1-33a) CH2CN
CH2S(O)2CH2(D1-33a) CH2CF3
CH2S(O)2CH2(D1-33a) CH2OMe
CH2S(O)2CH2(D1-33a) CH2OCF3
CH2S(O)2CH2(D1-33a) CH2SMe
CH2S(O)2CH2(D1-33a) CH2S(O)Me
CH2S(O)2CH2(D1-33a) CH2S(O)2Me
CH2S(O)2CH2(D1-33a) CH2SCF3
CH2S(O)2CH2(D1-33a) CH2S(O)CF3
CH2S(O)2CH2(D1-33a) CH2S(O)2CF3
CH2S(O)2CH2(D1-33a) CH2CH(OMe)2
CH2S(O)2CH2(D1-33a) CH2CH(SMe)2
CH2S(O)2CH2(D1-33a) CH2C(O)Me
CH2S(O)2CH2(D1-33a) CH2C(O)CF3
CH2S(O)2CH2(D1-33a) CH2C(O)OMe
CH2S(O)2CH2(D1-33a) CH2(D1-32a)
CH2S(O)2CH2(D1-33a) CH2(D1-33a)
CH2S(O)2CH2(D1-33a) CH2(D1-34a)
CH2S(O)2CH2(D1-33a) CH2(D1-37a)
CH2S(O)2CH2(D1-33a) CH2(D1-81a)
CH2S(O)2CH2(D1-33a) CH2(D1-82a)
CH2S(O)2CH2(D1-33a) CH2(D1-84a)
CH2S(O)2CH2(D1-33a) CH2(D1-85a)
CH2S(O)2CH2(D1-33a) CH2(D1-87a)
CH2S(O)2CH2(D1-33a) CH2(D1-92a)
CH2S(O)2CH2(D1-33a) CH2(D1-93a)
CH2S(O)2CH2(D1-33a) CH2(D1-95a)
CH2S(O)2CH2(D1-33a) CH2(D1-96a)
CH2S(O)2CH2(D1-33a) CH2(D1-98a)
CH2S(O)2CH2(D1-33a) CH2(D1-108a)
CH2S(O)2CH2(D1-33a) CH2(D1-108b,Z=2-Cl)
CH2S(O)2CH2(D1-33a) CH2(D1-108b,Z=3-Me)
CH2S(O)2CH2(D1-33a) CH2(D1-108b,Z=4-OMe)
CH2S(O)2CH2(D1-33a) CH2(D1-108b,Z=2-SMe)
CH2S(O)2CH2(D1-33a) CH2(D1-108b,Z=3-CF3)
CH2S(O)2CH2(D1-33a) CH2(D1-108b,Z=4-OCF3)
CH2S(O)2CH2(D1-33a) CH2(D1-108b,Z=2-SCF3)
CH2S(O)2CH2(D1-33a) CH2CH2CN
CH2S(O)2CH2(D1-33a) CH2CH2CF3
CH2S(O)2CH2(D1-33a) CH2CH2OMe
CH2S(O)2CH2(D1-33a) CH2CH2SMe
CH2S(O)2CH2(D1-33a) CH2CH2S(O)Me
CH2S(O)2CH2(D1-33a) CH2CH2S(O)2Me
CH2S(O)2CH2(D1-33a) D1-32a
CH2S(O)2CH2(D1-33a) D1-33a
CH2S(O)2CH2(D1-33a) D1-34a
CH2S(O)2CH2(D1-33a) D1-37a
CH2S(O)2CH2(D1-33a) D1-81a
CH2S(O)2CH2(D1-33a) D1-82a
CH2S(O)2CH2(D1-33a) D1-84a
CH2S(O)2CH2(D1-33a) D1-85a
CH2S(O)2CH2(D1-33a) D1-87a
CH2S(O)2CH2(D1-33a) D1-92a
CH2S(O)2CH2(D1-33a) D1-93a
CH2S(O)2CH2(D1-33a) D1-95a
CH2S(O)2CH2(D1-33a) D1-96a
CH2S(O)2CH2(D1-33a) D1-98a
CH2S(O)2CH2(D1-33a) D1-108a
CH2S(O)2CH2(D1-33a) D1-108b(Z=2-Cl)
CH2S(O)2CH2(D1-33a) D1-108b(Z=3-Me)
CH2S(O)2CH2(D1-33a) D1-108b(Z=4-OMe)
CH2S(O)2CH2(D1-33a) D1-108b(Z=2-SMe)
CH2S(O)2CH2(D1-33a) D1-108b(Z=3-CF3)
CH2S(O)2CH2(D1-33a) D1-108b(Z=4-OCF3)
CH2S(O)2CH2(D1-33a) D1-108b(Z=2-SCF3)
CH2S(O)2CH2(D1-33a) C(O)Me
CH2S(O)2CH2(D1-33a) C(O)CF3
CH2S(O)2CH2(D1-33a) C(O)OMe
CH(Me)SCH2(D1-33a) Me
CH(Me)SCH2(D1-33a) Et
CH(Me)SCH2(D1-33a) Pr-n
CH(Me)SCH2(D1-33a) Pr-i
CH(Me)SCH2(D1-33a) Pr-c
CH(Me)SCH2(D1-33a) Bu-n
CH(Me)SCH2(D1-33a) Bu-i
CH(Me)SCH2(D1-33a) Bu-c
CH(Me)SCH2(D1-33a) Bu-s
CH(Me)SCH2(D1-33a) Bu-t
CH(Me)SCH2(D1-33a) Pen-n
CH(Me)SCH2(D1-33a) Pen-c
CH(Me)SCH2(D1-33a) Hex-n
CH(Me)SCH2(D1-33a) Hex-c
CH(Me)SCH2(D1-33a) CH2Pr-c
CH(Me)SCH2(D1-33a) CH2Bu-c
CH(Me)SCH2(D1-33a) CH2Pen-c
CH(Me)SCH2(D1-33a) CH2Hex-c
CH(Me)SCH2(D1-33a) CH2CH=CH2
CH(Me)SCH2(D1-33a) CH2CH=C(Cl)2
CH(Me)SCH2(D1-33a) CH2C≡CH
CH(Me)SCH2(D1-33a) CH2CN
CH(Me)SCH2(D1-33a) CH2CF3
CH(Me)SCH2(D1-33a) CH2OMe
CH(Me)SCH2(D1-33a) CH2OCF3
CH(Me)SCH2(D1-33a) CH2SMe
CH(Me)SCH2(D1-33a) CH2S(O)Me
CH(Me)SCH2(D1-33a) CH2S(O)2Me
CH(Me)SCH2(D1-33a) CH2SCF3
CH(Me)SCH2(D1-33a) CH2S(O)CF3
CH(Me)SCH2(D1-33a) CH2S(O)2CF3
CH(Me)SCH2(D1-33a) CH2CH(OMe)2
CH(Me)SCH2(D1-33a) CH2CH(SMe)2
CH(Me)SCH2(D1-33a) CH2C(O)Me
CH(Me)SCH2(D1-33a) CH2C(O)CF3
CH(Me)SCH2(D1-33a) CH2C(O)OMe
CH(Me)SCH2(D1-33a) CH2(D1-32a)
CH(Me)SCH2(D1-33a) CH2(D1-33a)
CH(Me)SCH2(D1-33a) CH2(D1-34a)
CH(Me)SCH2(D1-33a) CH2(D1-37a)
CH(Me)SCH2(D1-33a) CH2(D1-81a)
CH(Me)SCH2(D1-33a) CH2(D1-82a)
CH(Me)SCH2(D1-33a) CH2(D1-84a)
CH(Me)SCH2(D1-33a) CH2(D1-85a)
CH(Me)SCH2(D1-33a) CH2(D1-87a)
CH(Me)SCH2(D1-33a) CH2(D1-92a)
CH(Me)SCH2(D1-33a) CH2(D1-93a)
CH(Me)SCH2(D1-33a) CH2(D1-95a)
CH(Me)SCH2(D1-33a) CH2(D1-96a)
CH(Me)SCH2(D1-33a) CH2(D1-98a)
CH(Me)SCH2(D1-33a) CH2(D1-108a)
CH(Me)SCH2(D1-33a) CH2(D1-108b,Z=2-Cl)
CH(Me)SCH2(D1-33a) CH2(D1-108b,Z=3-Me)
CH(Me)SCH2(D1-33a) CH2(D1-108b,Z=4-OMe)
CH(Me)SCH2(D1-33a) CH2(D1-108b,Z=2-SMe)
CH(Me)SCH2(D1-33a) CH2(D1-108b,Z=3-CF3)
CH(Me)SCH2(D1-33a) CH2(D1-108b,Z=4-OCF3)
CH(Me)SCH2(D1-33a) CH2(D1-108b,Z=2-SCF3)
CH(Me)SCH2(D1-33a) CH2CH2CN
CH(Me)SCH2(D1-33a) CH2CH2CF3
CH(Me)SCH2(D1-33a) CH2CH2OMe
CH(Me)SCH2(D1-33a) CH2CH2SMe
CH(Me)SCH2(D1-33a) CH2CH2S(O)Me
CH(Me)SCH2(D1-33a) CH2CH2S(O)2Me
CH(Me)SCH2(D1-33a) D1-32a
CH(Me)SCH2(D1-33a) D1-33a
CH(Me)SCH2(D1-33a) D1-34a
CH(Me)SCH2(D1-33a) D1-37a
CH(Me)SCH2(D1-33a) D1-81a
CH(Me)SCH2(D1-33a) D1-82a
CH(Me)SCH2(D1-33a) D1-84a
CH(Me)SCH2(D1-33a) D1-85a
CH(Me)SCH2(D1-33a) D1-87a
CH(Me)SCH2(D1-33a) D1-92a
CH(Me)SCH2(D1-33a) D1-93a
CH(Me)SCH2(D1-33a) D1-95a
CH(Me)SCH2(D1-33a) D1-96a
CH(Me)SCH2(D1-33a) D1-98a
CH(Me)SCH2(D1-33a) D1-108a
CH(Me)SCH2(D1-33a) D1-108b(Z=2-Cl)
CH(Me)SCH2(D1-33a) D1-108b(Z=3-Me)
CH(Me)SCH2(D1-33a) D1-108b(Z=4-OMe)
CH(Me)SCH2(D1-33a) D1-108b(Z=2-SMe)
CH(Me)SCH2(D1-33a) D1-108b(Z=3-CF3)
CH(Me)SCH2(D1-33a) D1-108b(Z=4-OCF3)
CH(Me)SCH2(D1-33a) D1-108b(Z=2-SCF3)
CH(Me)SCH2(D1-33a) C(O)Me
CH(Me)SCH2(D1-33a) C(O)CF3
CH(Me)SCH2(D1-33a) C(O)OMe
CH(Me)S(O)CH2(D1-33a) Me
CH(Me)S(O)CH2(D1-33a) Et
CH(Me)S(O)CH2(D1-33a) Pr-n
CH(Me)S(O)CH2(D1-33a) Pr-i
CH(Me)S(O)CH2(D1-33a) Pr-c
CH(Me)S(O)CH2(D1-33a) Bu-n
CH(Me)S(O)CH2(D1-33a) Bu-i
CH(Me)S(O)CH2(D1-33a) Bu-c
CH(Me)S(O)CH2(D1-33a) Bu-s
CH(Me)S(O)CH2(D1-33a) Bu-t
CH(Me)S(O)CH2(D1-33a) Pen-n
CH(Me)S(O)CH2(D1-33a) Pen-c
CH(Me)S(O)CH2(D1-33a) Hex-n
CH(Me)S(O)CH2(D1-33a) Hex-c
CH(Me)S(O)CH2(D1-33a) CH2Pr-c
CH(Me)S(O)CH2(D1-33a) CH2Bu-c
CH(Me)S(O)CH2(D1-33a) CH2Pen-c
CH(Me)S(O)CH2(D1-33a) CH2Hex-c
CH(Me)S(O)CH2(D1-33a) CH2CH=CH2
CH(Me)S(O)CH2(D1-33a) CH2CH=C(Cl)2
CH(Me)S(O)CH2(D1-33a) CH2C≡CH
CH(Me)S(O)CH2(D1-33a) CH2CN
CH(Me)S(O)CH2(D1-33a) CH2CF3
CH(Me)S(O)CH2(D1-33a) CH2OMe
CH(Me)S(O)CH2(D1-33a) CH2OCF3
CH(Me)S(O)CH2(D1-33a) CH2SMe
CH(Me)S(O)CH2(D1-33a) CH2S(O)Me
CH(Me)S(O)CH2(D1-33a) CH2S(O)2Me
CH(Me)S(O)CH2(D1-33a) CH2SCF3
CH(Me)S(O)CH2(D1-33a) CH2S(O)CF3
CH(Me)S(O)CH2(D1-33a) CH2S(O)2CF3
CH(Me)S(O)CH2(D1-33a) CH2CH(OMe)2
CH(Me)S(O)CH2(D1-33a) CH2CH(SMe)2
CH(Me)S(O)CH2(D1-33a) CH2C(O)Me
CH(Me)S(O)CH2(D1-33a) CH2C(O)CF3
CH(Me)S(O)CH2(D1-33a) CH2C(O)OMe
CH(Me)S(O)CH2(D1-33a) CH2(D1-32a)
CH(Me)S(O)CH2(D1-33a) CH2(D1-33a)
CH(Me)S(O)CH2(D1-33a) CH2(D1-34a)
CH(Me)S(O)CH2(D1-33a) CH2(D1-37a)
CH(Me)S(O)CH2(D1-33a) CH2(D1-81a)
CH(Me)S(O)CH2(D1-33a) CH2(D1-82a)
CH(Me)S(O)CH2(D1-33a) CH2(D1-84a)
CH(Me)S(O)CH2(D1-33a) CH2(D1-85a)
CH(Me)S(O)CH2(D1-33a) CH2(D1-87a)
CH(Me)S(O)CH2(D1-33a) CH2(D1-92a)
CH(Me)S(O)CH2(D1-33a) CH2(D1-93a)
CH(Me)S(O)CH2(D1-33a) CH2(D1-95a)
CH(Me)S(O)CH2(D1-33a) CH2(D1-96a)
CH(Me)S(O)CH2(D1-33a) CH2(D1-98a)
CH(Me)S(O)CH2(D1-33a) CH2(D1-108a)
CH(Me)S(O)CH2(D1-33a) CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)CH2(D1-33a) CH2(D1-108b,Z=3-Me)
CH(Me)S(O)CH2(D1-33a) CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)CH2(D1-33a) CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)CH2(D1-33a) CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)CH2(D1-33a) CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)CH2(D1-33a) CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)CH2(D1-33a) CH2CH2CN
CH(Me)S(O)CH2(D1-33a) CH2CH2CF3
CH(Me)S(O)CH2(D1-33a) CH2CH2OMe
CH(Me)S(O)CH2(D1-33a) CH2CH2SMe
CH(Me)S(O)CH2(D1-33a) CH2CH2S(O)Me
CH(Me)S(O)CH2(D1-33a) CH2CH2S(O)2Me
CH(Me)S(O)CH2(D1-33a) D1-32a
CH(Me)S(O)CH2(D1-33a) D1-33a
CH(Me)S(O)CH2(D1-33a) D1-34a
CH(Me)S(O)CH2(D1-33a) D1-37a
CH(Me)S(O)CH2(D1-33a) D1-81a
CH(Me)S(O)CH2(D1-33a) D1-82a
CH(Me)S(O)CH2(D1-33a) D1-84a
CH(Me)S(O)CH2(D1-33a) D1-85a
CH(Me)S(O)CH2(D1-33a) D1-87a
CH(Me)S(O)CH2(D1-33a) D1-92a
CH(Me)S(O)CH2(D1-33a) D1-93a
CH(Me)S(O)CH2(D1-33a) D1-95a
CH(Me)S(O)CH2(D1-33a) D1-96a
CH(Me)S(O)CH2(D1-33a) D1-98a
CH(Me)S(O)CH2(D1-33a) D1-108a
CH(Me)S(O)CH2(D1-33a) D1-108b(Z=2-Cl)
CH(Me)S(O)CH2(D1-33a) D1-108b(Z=3-Me)
CH(Me)S(O)CH2(D1-33a) D1-108b(Z=4-OMe)
CH(Me)S(O)CH2(D1-33a) D1-108b(Z=2-SMe)
CH(Me)S(O)CH2(D1-33a) D1-108b(Z=3-CF3)
CH(Me)S(O)CH2(D1-33a) D1-108b(Z=4-OCF3)
CH(Me)S(O)CH2(D1-33a) D1-108b(Z=2-SCF3)
CH(Me)S(O)CH2(D1-33a) C(O)Me
CH(Me)S(O)CH2(D1-33a) C(O)CF3
CH(Me)S(O)CH2(D1-33a) C(O)OMe
CH(Me)S(O)2CH2(D1-33a) Me
CH(Me)S(O)2CH2(D1-33a) Et
CH(Me)S(O)2CH2(D1-33a) Pr-n
CH(Me)S(O)2CH2(D1-33a) Pr-i
CH(Me)S(O)2CH2(D1-33a) Pr-c
CH(Me)S(O)2CH2(D1-33a) Bu-n
CH(Me)S(O)2CH2(D1-33a) Bu-i
CH(Me)S(O)2CH2(D1-33a) Bu-c
CH(Me)S(O)2CH2(D1-33a) Bu-s
CH(Me)S(O)2CH2(D1-33a) Bu-t
CH(Me)S(O)2CH2(D1-33a) Pen-n
CH(Me)S(O)2CH2(D1-33a) Pen-c
CH(Me)S(O)2CH2(D1-33a) Hex-n
CH(Me)S(O)2CH2(D1-33a) Hex-c
CH(Me)S(O)2CH2(D1-33a) CH2Pr-c
CH(Me)S(O)2CH2(D1-33a) CH2Bu-c
CH(Me)S(O)2CH2(D1-33a) CH2Pen-c
CH(Me)S(O)2CH2(D1-33a) CH2Hex-c
CH(Me)S(O)2CH2(D1-33a) CH2CH=CH2
CH(Me)S(O)2CH2(D1-33a) CH2CH=C(Cl)2
CH(Me)S(O)2CH2(D1-33a) CH2C≡CH
CH(Me)S(O)2CH2(D1-33a) CH2CN
CH(Me)S(O)2CH2(D1-33a) CH2CF3
CH(Me)S(O)2CH2(D1-33a) CH2OMe
CH(Me)S(O)2CH2(D1-33a) CH2OCF3
CH(Me)S(O)2CH2(D1-33a) CH2SMe
CH(Me)S(O)2CH2(D1-33a) CH2S(O)Me
CH(Me)S(O)2CH2(D1-33a) CH2S(O)2Me
CH(Me)S(O)2CH2(D1-33a) CH2SCF3
CH(Me)S(O)2CH2(D1-33a) CH2S(O)CF3
CH(Me)S(O)2CH2(D1-33a) CH2S(O)2CF3
CH(Me)S(O)2CH2(D1-33a) CH2CH(OMe)2
CH(Me)S(O)2CH2(D1-33a) CH2CH(SMe)2
CH(Me)S(O)2CH2(D1-33a) CH2C(O)Me
CH(Me)S(O)2CH2(D1-33a) CH2C(O)CF3
CH(Me)S(O)2CH2(D1-33a) CH2C(O)OMe
CH(Me)S(O)2CH2(D1-33a) CH2(D1-32a)
CH(Me)S(O)2CH2(D1-33a) CH2(D1-33a)
CH(Me)S(O)2CH2(D1-33a) CH2(D1-34a)
CH(Me)S(O)2CH2(D1-33a) CH2(D1-37a)
CH(Me)S(O)2CH2(D1-33a) CH2(D1-81a)
CH(Me)S(O)2CH2(D1-33a) CH2(D1-82a)
CH(Me)S(O)2CH2(D1-33a) CH2(D1-84a)
CH(Me)S(O)2CH2(D1-33a) CH2(D1-85a)
CH(Me)S(O)2CH2(D1-33a) CH2(D1-87a)
CH(Me)S(O)2CH2(D1-33a) CH2(D1-92a)
CH(Me)S(O)2CH2(D1-33a) CH2(D1-93a)
CH(Me)S(O)2CH2(D1-33a) CH2(D1-95a)
CH(Me)S(O)2CH2(D1-33a) CH2(D1-96a)
CH(Me)S(O)2CH2(D1-33a) CH2(D1-98a)
CH(Me)S(O)2CH2(D1-33a) CH2(D1-108a)
CH(Me)S(O)2CH2(D1-33a) CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)2CH2(D1-33a) CH2(D1-108b,Z=3-Me)
CH(Me)S(O)2CH2(D1-33a) CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)2CH2(D1-33a) CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)2CH2(D1-33a) CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)2CH2(D1-33a) CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)2CH2(D1-33a) CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)2CH2(D1-33a) CH2CH2CN
CH(Me)S(O)2CH2(D1-33a) CH2CH2CF3
CH(Me)S(O)2CH2(D1-33a) CH2CH2OMe
CH(Me)S(O)2CH2(D1-33a) CH2CH2SMe
CH(Me)S(O)2CH2(D1-33a) CH2CH2S(O)Me
CH(Me)S(O)2CH2(D1-33a) CH2CH2S(O)2Me
CH(Me)S(O)2CH2(D1-33a) D1-32a
CH(Me)S(O)2CH2(D1-33a) D1-33a
CH(Me)S(O)2CH2(D1-33a) D1-34a
CH(Me)S(O)2CH2(D1-33a) D1-37a
CH(Me)S(O)2CH2(D1-33a) D1-81a
CH(Me)S(O)2CH2(D1-33a) D1-82a
CH(Me)S(O)2CH2(D1-33a) D1-84a
CH(Me)S(O)2CH2(D1-33a) D1-85a
CH(Me)S(O)2CH2(D1-33a) D1-87a
CH(Me)S(O)2CH2(D1-33a) D1-92a
CH(Me)S(O)2CH2(D1-33a) D1-93a
CH(Me)S(O)2CH2(D1-33a) D1-95a
CH(Me)S(O)2CH2(D1-33a) D1-96a
CH(Me)S(O)2CH2(D1-33a) D1-98a
CH(Me)S(O)2CH2(D1-33a) D1-108a
CH(Me)S(O)2CH2(D1-33a) D1-108b(Z=2-Cl)
CH(Me)S(O)2CH2(D1-33a) D1-108b(Z=3-Me)
CH(Me)S(O)2CH2(D1-33a) D1-108b(Z=4-OMe)
CH(Me)S(O)2CH2(D1-33a) D1-108b(Z=2-SMe)
CH(Me)S(O)2CH2(D1-33a) D1-108b(Z=3-CF3)
CH(Me)S(O)2CH2(D1-33a) D1-108b(Z=4-OCF3)
CH(Me)S(O)2CH2(D1-33a) D1-108b(Z=2-SCF3)
CH(Me)S(O)2CH2(D1-33a) C(O)Me
CH(Me)S(O)2CH2(D1-33a) C(O)CF3
CH(Me)S(O)2CH2(D1-33a) C(O)OMe
CH(Et)SCH2(D1-33a) Me
CH(Et)SCH2(D1-33a) Et
CH(Et)SCH2(D1-33a) Pr-n
CH(Et)SCH2(D1-33a) Pr-i
CH(Et)SCH2(D1-33a) Pr-c
CH(Et)SCH2(D1-33a) Bu-n
CH(Et)SCH2(D1-33a) Bu-i
CH(Et)SCH2(D1-33a) Bu-c
CH(Et)SCH2(D1-33a) Bu-s
CH(Et)SCH2(D1-33a) Bu-t
CH(Et)SCH2(D1-33a) Pen-n
CH(Et)SCH2(D1-33a) Pen-c
CH(Et)SCH2(D1-33a) Hex-n
CH(Et)SCH2(D1-33a) Hex-c
CH(Et)SCH2(D1-33a) CH2Pr-c
CH(Et)SCH2(D1-33a) CH2Bu-c
CH(Et)SCH2(D1-33a) CH2Pen-c
CH(Et)SCH2(D1-33a) CH2Hex-c
CH(Et)SCH2(D1-33a) CH2CH=CH2
CH(Et)SCH2(D1-33a) CH2CH=C(Cl)2
CH(Et)SCH2(D1-33a) CH2C≡CH
CH(Et)SCH2(D1-33a) CH2CN
CH(Et)SCH2(D1-33a) CH2CF3
CH(Et)SCH2(D1-33a) CH2OMe
CH(Et)SCH2(D1-33a) CH2OCF3
CH(Et)SCH2(D1-33a) CH2SMe
CH(Et)SCH2(D1-33a) CH2S(O)Me
CH(Et)SCH2(D1-33a) CH2S(O)2Me
CH(Et)SCH2(D1-33a) CH2SCF3
CH(Et)SCH2(D1-33a) CH2S(O)CF3
CH(Et)SCH2(D1-33a) CH2S(O)2CF3
CH(Et)SCH2(D1-33a) CH2CH(OMe)2
CH(Et)SCH2(D1-33a) CH2CH(SMe)2
CH(Et)SCH2(D1-33a) CH2C(O)Me
CH(Et)SCH2(D1-33a) CH2C(O)CF3
CH(Et)SCH2(D1-33a) CH2C(O)OMe
CH(Et)SCH2(D1-33a) CH2(D1-32a)
CH(Et)SCH2(D1-33a) CH2(D1-33a)
CH(Et)SCH2(D1-33a) CH2(D1-34a)
CH(Et)SCH2(D1-33a) CH2(D1-37a)
CH(Et)SCH2(D1-33a) CH2(D1-81a)
CH(Et)SCH2(D1-33a) CH2(D1-82a)
CH(Et)SCH2(D1-33a) CH2(D1-84a)
CH(Et)SCH2(D1-33a) CH2(D1-85a)
CH(Et)SCH2(D1-33a) CH2(D1-87a)
CH(Et)SCH2(D1-33a) CH2(D1-92a)
CH(Et)SCH2(D1-33a) CH2(D1-93a)
CH(Et)SCH2(D1-33a) CH2(D1-95a)
CH(Et)SCH2(D1-33a) CH2(D1-96a)
CH(Et)SCH2(D1-33a) CH2(D1-98a)
CH(Et)SCH2(D1-33a) CH2(D1-108a)
CH(Et)SCH2(D1-33a) CH2(D1-108b,Z=2-Cl)
CH(Et)SCH2(D1-33a) CH2(D1-108b,Z=3-Me)
CH(Et)SCH2(D1-33a) CH2(D1-108b,Z=4-OMe)
CH(Et)SCH2(D1-33a) CH2(D1-108b,Z=2-SMe)
CH(Et)SCH2(D1-33a) CH2(D1-108b,Z=3-CF3)
CH(Et)SCH2(D1-33a) CH2(D1-108b,Z=4-OCF3)
CH(Et)SCH2(D1-33a) CH2(D1-108b,Z=2-SCF3)
CH(Et)SCH2(D1-33a) CH2CH2CN
CH(Et)SCH2(D1-33a) CH2CH2CF3
CH(Et)SCH2(D1-33a) CH2CH2OMe
CH(Et)SCH2(D1-33a) CH2CH2SMe
CH(Et)SCH2(D1-33a) CH2CH2S(O)Me
CH(Et)SCH2(D1-33a) CH2CH2S(O)2Me
CH(Et)SCH2(D1-33a) D1-32a
CH(Et)SCH2(D1-33a) D1-33a
CH(Et)SCH2(D1-33a) D1-34a
CH(Et)SCH2(D1-33a) D1-37a
CH(Et)SCH2(D1-33a) D1-81a
CH(Et)SCH2(D1-33a) D1-82a
CH(Et)SCH2(D1-33a) D1-84a
CH(Et)SCH2(D1-33a) D1-85a
CH(Et)SCH2(D1-33a) D1-87a
CH(Et)SCH2(D1-33a) D1-92a
CH(Et)SCH2(D1-33a) D1-93a
CH(Et)SCH2(D1-33a) D1-95a
CH(Et)SCH2(D1-33a) D1-96a
CH(Et)SCH2(D1-33a) D1-98a
CH(Et)SCH2(D1-33a) D1-108a
CH(Et)SCH2(D1-33a) D1-108b(Z=2-Cl)
CH(Et)SCH2(D1-33a) D1-108b(Z=3-Me)
CH(Et)SCH2(D1-33a) D1-108b(Z=4-OMe)
CH(Et)SCH2(D1-33a) D1-108b(Z=2-SMe)
CH(Et)SCH2(D1-33a) D1-108b(Z=3-CF3)
CH(Et)SCH2(D1-33a) D1-108b(Z=4-OCF3)
CH(Et)SCH2(D1-33a) D1-108b(Z=2-SCF3)
CH(Et)SCH2(D1-33a) C(O)Me
CH(Et)SCH2(D1-33a) C(O)CF3
CH(Et)SCH2(D1-33a) C(O)OMe
CH(Et)S(O)CH2(D1-33a) Me
CH(Et)S(O)CH2(D1-33a) Et
CH(Et)S(O)CH2(D1-33a) Pr-n
CH(Et)S(O)CH2(D1-33a) Pr-i
CH(Et)S(O)CH2(D1-33a) Pr-c
CH(Et)S(O)CH2(D1-33a) Bu-n
CH(Et)S(O)CH2(D1-33a) Bu-i
CH(Et)S(O)CH2(D1-33a) Bu-c
CH(Et)S(O)CH2(D1-33a) Bu-s
CH(Et)S(O)CH2(D1-33a) Bu-t
CH(Et)S(O)CH2(D1-33a) Pen-n
CH(Et)S(O)CH2(D1-33a) Pen-c
CH(Et)S(O)CH2(D1-33a) Hex-n
CH(Et)S(O)CH2(D1-33a) Hex-c
CH(Et)S(O)CH2(D1-33a) CH2Pr-c
CH(Et)S(O)CH2(D1-33a) CH2Bu-c
CH(Et)S(O)CH2(D1-33a) CH2Pen-c
CH(Et)S(O)CH2(D1-33a) CH2Hex-c
CH(Et)S(O)CH2(D1-33a) CH2CH=CH2
CH(Et)S(O)CH2(D1-33a) CH2CH=C(Cl)2
CH(Et)S(O)CH2(D1-33a) CH2C≡CH
CH(Et)S(O)CH2(D1-33a) CH2CN
CH(Et)S(O)CH2(D1-33a) CH2CF3
CH(Et)S(O)CH2(D1-33a) CH2OMe
CH(Et)S(O)CH2(D1-33a) CH2OCF3
CH(Et)S(O)CH2(D1-33a) CH2SMe
CH(Et)S(O)CH2(D1-33a) CH2S(O)Me
CH(Et)S(O)CH2(D1-33a) CH2S(O)2Me
CH(Et)S(O)CH2(D1-33a) CH2SCF3
CH(Et)S(O)CH2(D1-33a) CH2S(O)CF3
CH(Et)S(O)CH2(D1-33a) CH2S(O)2CF3
CH(Et)S(O)CH2(D1-33a) CH2CH(OMe)2
CH(Et)S(O)CH2(D1-33a) CH2CH(SMe)2
CH(Et)S(O)CH2(D1-33a) CH2C(O)Me
CH(Et)S(O)CH2(D1-33a) CH2C(O)CF3
CH(Et)S(O)CH2(D1-33a) CH2C(O)OMe
CH(Et)S(O)CH2(D1-33a) CH2(D1-32a)
CH(Et)S(O)CH2(D1-33a) CH2(D1-33a)
CH(Et)S(O)CH2(D1-33a) CH2(D1-34a)
CH(Et)S(O)CH2(D1-33a) CH2(D1-37a)
CH(Et)S(O)CH2(D1-33a) CH2(D1-81a)
CH(Et)S(O)CH2(D1-33a) CH2(D1-82a)
CH(Et)S(O)CH2(D1-33a) CH2(D1-84a)
CH(Et)S(O)CH2(D1-33a) CH2(D1-85a)
CH(Et)S(O)CH2(D1-33a) CH2(D1-87a)
CH(Et)S(O)CH2(D1-33a) CH2(D1-92a)
CH(Et)S(O)CH2(D1-33a) CH2(D1-93a)
CH(Et)S(O)CH2(D1-33a) CH2(D1-95a)
CH(Et)S(O)CH2(D1-33a) CH2(D1-96a)
CH(Et)S(O)CH2(D1-33a) CH2(D1-98a)
CH(Et)S(O)CH2(D1-33a) CH2(D1-108a)
CH(Et)S(O)CH2(D1-33a) CH2(D1-108b,Z=2-Cl)
CH(Et)S(O)CH2(D1-33a) CH2(D1-108b,Z=3-Me)
CH(Et)S(O)CH2(D1-33a) CH2(D1-108b,Z=4-OMe)
CH(Et)S(O)CH2(D1-33a) CH2(D1-108b,Z=2-SMe)
CH(Et)S(O)CH2(D1-33a) CH2(D1-108b,Z=3-CF3)
CH(Et)S(O)CH2(D1-33a) CH2(D1-108b,Z=4-OCF3)
CH(Et)S(O)CH2(D1-33a) CH2(D1-108b,Z=2-SCF3)
CH(Et)S(O)CH2(D1-33a) CH2CH2CN
CH(Et)S(O)CH2(D1-33a) CH2CH2CF3
CH(Et)S(O)CH2(D1-33a) CH2CH2OMe
CH(Et)S(O)CH2(D1-33a) CH2CH2SMe
CH(Et)S(O)CH2(D1-33a) CH2CH2S(O)Me
CH(Et)S(O)CH2(D1-33a) CH2CH2S(O)2Me
CH(Et)S(O)CH2(D1-33a) D1-32a
CH(Et)S(O)CH2(D1-33a) D1-33a
CH(Et)S(O)CH2(D1-33a) D1-34a
CH(Et)S(O)CH2(D1-33a) D1-37a
CH(Et)S(O)CH2(D1-33a) D1-81a
CH(Et)S(O)CH2(D1-33a) D1-82a
CH(Et)S(O)CH2(D1-33a) D1-84a
CH(Et)S(O)CH2(D1-33a) D1-85a
CH(Et)S(O)CH2(D1-33a) D1-87a
CH(Et)S(O)CH2(D1-33a) D1-92a
CH(Et)S(O)CH2(D1-33a) D1-93a
CH(Et)S(O)CH2(D1-33a) D1-95a
CH(Et)S(O)CH2(D1-33a) D1-96a
CH(Et)S(O)CH2(D1-33a) D1-98a
CH(Et)S(O)CH2(D1-33a) D1-108a
CH(Et)S(O)CH2(D1-33a) D1-108b(Z=2-Cl)
CH(Et)S(O)CH2(D1-33a) D1-108b(Z=3-Me)
CH(Et)S(O)CH2(D1-33a) D1-108b(Z=4-OMe)
CH(Et)S(O)CH2(D1-33a) D1-108b(Z=2-SMe)
CH(Et)S(O)CH2(D1-33a) D1-108b(Z=3-CF3)
CH(Et)S(O)CH2(D1-33a) D1-108b(Z=4-OCF3)
CH(Et)S(O)CH2(D1-33a) D1-108b(Z=2-SCF3)
CH(Et)S(O)CH2(D1-33a) C(O)Me
CH(Et)S(O)CH2(D1-33a) C(O)CF3
CH(Et)S(O)CH2(D1-33a) C(O)OMe
CH(Et)S(O)2CH2(D1-33a) Me
CH(Et)S(O)2CH2(D1-33a) Et
CH(Et)S(O)2CH2(D1-33a) Pr-n
CH(Et)S(O)2CH2(D1-33a) Pr-i
CH(Et)S(O)2CH2(D1-33a) Pr-c
CH(Et)S(O)2CH2(D1-33a) Bu-n
CH(Et)S(O)2CH2(D1-33a) Bu-i
CH(Et)S(O)2CH2(D1-33a) Bu-c
CH(Et)S(O)2CH2(D1-33a) Bu-s
CH(Et)S(O)2CH2(D1-33a) Bu-t
CH(Et)S(O)2CH2(D1-33a) Pen-n
CH(Et)S(O)2CH2(D1-33a) Pen-c
CH(Et)S(O)2CH2(D1-33a) Hex-n
CH(Et)S(O)2CH2(D1-33a) Hex-c
CH(Et)S(O)2CH2(D1-33a) CH2Pr-c
CH(Et)S(O)2CH2(D1-33a) CH2Bu-c
CH(Et)S(O)2CH2(D1-33a) CH2Pen-c
CH(Et)S(O)2CH2(D1-33a) CH2Hex-c
CH(Et)S(O)2CH2(D1-33a) CH2CH=CH2
CH(Et)S(O)2CH2(D1-33a) CH2CH=C(Cl)2
CH(Et)S(O)2CH2(D1-33a) CH2C≡CH
CH(Et)S(O)2CH2(D1-33a) CH2CN
CH(Et)S(O)2CH2(D1-33a) CH2CF3
CH(Et)S(O)2CH2(D1-33a) CH2OMe
CH(Et)S(O)2CH2(D1-33a) CH2OCF3
CH(Et)S(O)2CH2(D1-33a) CH2SMe
CH(Et)S(O)2CH2(D1-33a) CH2S(O)Me
CH(Et)S(O)2CH2(D1-33a) CH2S(O)2Me
CH(Et)S(O)2CH2(D1-33a) CH2SCF3
CH(Et)S(O)2CH2(D1-33a) CH2S(O)CF3
CH(Et)S(O)2CH2(D1-33a) CH2S(O)2CF3
CH(Et)S(O)2CH2(D1-33a) CH2CH(OMe)2
CH(Et)S(O)2CH2(D1-33a) CH2CH(SMe)2
CH(Et)S(O)2CH2(D1-33a) CH2C(O)Me
CH(Et)S(O)2CH2(D1-33a) CH2C(O)CF3
CH(Et)S(O)2CH2(D1-33a) CH2C(O)OMe
CH(Et)S(O)2CH2(D1-33a) CH2(D1-32a)
CH(Et)S(O)2CH2(D1-33a) CH2(D1-33a)
CH(Et)S(O)2CH2(D1-33a) CH2(D1-34a)
CH(Et)S(O)2CH2(D1-33a) CH2(D1-37a)
CH(Et)S(O)2CH2(D1-33a) CH2(D1-81a)
CH(Et)S(O)2CH2(D1-33a) CH2(D1-82a)
CH(Et)S(O)2CH2(D1-33a) CH2(D1-84a)
CH(Et)S(O)2CH2(D1-33a) CH2(D1-85a)
CH(Et)S(O)2CH2(D1-33a) CH2(D1-87a)
CH(Et)S(O)2CH2(D1-33a) CH2(D1-92a)
CH(Et)S(O)2CH2(D1-33a) CH2(D1-93a)
CH(Et)S(O)2CH2(D1-33a) CH2(D1-95a)
CH(Et)S(O)2CH2(D1-33a) CH2(D1-96a)
CH(Et)S(O)2CH2(D1-33a) CH2(D1-98a)
CH(Et)S(O)2CH2(D1-33a) CH2(D1-108a)
CH(Et)S(O)2CH2(D1-33a) CH2(D1-108b,Z=2-Cl)
CH(Et)S(O)2CH2(D1-33a) CH2(D1-108b,Z=3-Me)
CH(Et)S(O)2CH2(D1-33a) CH2(D1-108b,Z=4-OMe)
CH(Et)S(O)2CH2(D1-33a) CH2(D1-108b,Z=2-SMe)
CH(Et)S(O)2CH2(D1-33a) CH2(D1-108b,Z=3-CF3)
CH(Et)S(O)2CH2(D1-33a) CH2(D1-108b,Z=4-OCF3)
CH(Et)S(O)2CH2(D1-33a) CH2(D1-108b,Z=2-SCF3)
CH(Et)S(O)2CH2(D1-33a) CH2CH2CN
CH(Et)S(O)2CH2(D1-33a) CH2CH2CF3
CH(Et)S(O)2CH2(D1-33a) CH2CH2OMe
CH(Et)S(O)2CH2(D1-33a) CH2CH2SMe
CH(Et)S(O)2CH2(D1-33a) CH2CH2S(O)Me
CH(Et)S(O)2CH2(D1-33a) CH2CH2S(O)2Me
CH(Et)S(O)2CH2(D1-33a) D1-32a
CH(Et)S(O)2CH2(D1-33a) D1-33a
CH(Et)S(O)2CH2(D1-33a) D1-34a
CH(Et)S(O)2CH2(D1-33a) D1-37a
CH(Et)S(O)2CH2(D1-33a) D1-81a
CH(Et)S(O)2CH2(D1-33a) D1-82a
CH(Et)S(O)2CH2(D1-33a) D1-84a
CH(Et)S(O)2CH2(D1-33a) D1-85a
CH(Et)S(O)2CH2(D1-33a) D1-87a
CH(Et)S(O)2CH2(D1-33a) D1-92a
CH(Et)S(O)2CH2(D1-33a) D1-93a
CH(Et)S(O)2CH2(D1-33a) D1-95a
CH(Et)S(O)2CH2(D1-33a) D1-96a
CH(Et)S(O)2CH2(D1-33a) D1-98a
CH(Et)S(O)2CH2(D1-33a) D1-108a
CH(Et)S(O)2CH2(D1-33a) D1-108b(Z=2-Cl)
CH(Et)S(O)2CH2(D1-33a) D1-108b(Z=3-Me)
CH(Et)S(O)2CH2(D1-33a) D1-108b(Z=4-OMe)
CH(Et)S(O)2CH2(D1-33a) D1-108b(Z=2-SMe)
CH(Et)S(O)2CH2(D1-33a) D1-108b(Z=3-CF3)
CH(Et)S(O)2CH2(D1-33a) D1-108b(Z=4-OCF3)
CH(Et)S(O)2CH2(D1-33a) D1-108b(Z=2-SCF3)
CH(Et)S(O)2CH2(D1-33a) C(O)Me
CH(Et)S(O)2CH2(D1-33a) C(O)CF3
CH(Et)S(O)2CH2(D1-33a) C(O)OMe
CH2SCH2(D1-34a) Me
CH2SCH2(D1-34a) Et
CH2SCH2(D1-34a) Pr-n
CH2SCH2(D1-34a) Pr-i
CH2SCH2(D1-34a) Pr-c
CH2SCH2(D1-34a) Bu-n
CH2SCH2(D1-34a) Bu-i
CH2SCH2(D1-34a) Bu-c
CH2SCH2(D1-34a) Bu-s
CH2SCH2(D1-34a) Bu-t
CH2SCH2(D1-34a) Pen-n
CH2SCH2(D1-34a) Pen-c
CH2SCH2(D1-34a) Hex-n
CH2SCH2(D1-34a) Hex-c
CH2SCH2(D1-34a) CH2Pr-c
CH2SCH2(D1-34a) CH2Bu-c
CH2SCH2(D1-34a) CH2Pen-c
CH2SCH2(D1-34a) CH2Hex-c
CH2SCH2(D1-34a) CH2CH=CH2
CH2SCH2(D1-34a) CH2CH=C(Cl)2
CH2SCH2(D1-34a) CH2C≡CH
CH2SCH2(D1-34a) CH2CN
CH2SCH2(D1-34a) CH2CF3
CH2SCH2(D1-34a) CH2OMe
CH2SCH2(D1-34a) CH2OCF3
CH2SCH2(D1-34a) CH2SMe
CH2SCH2(D1-34a) CH2S(O)Me
CH2SCH2(D1-34a) CH2S(O)2Me
CH2SCH2(D1-34a) CH2SCF3
CH2SCH2(D1-34a) CH2S(O)CF3
CH2SCH2(D1-34a) CH2S(O)2CF3
CH2SCH2(D1-34a) CH2CH(OMe)2
CH2SCH2(D1-34a) CH2CH(SMe)2
CH2SCH2(D1-34a) CH2C(O)Me
CH2SCH2(D1-34a) CH2C(O)CF3
CH2SCH2(D1-34a) CH2C(O)OMe
CH2SCH2(D1-34a) CH2(D1-32a)
CH2SCH2(D1-34a) CH2(D1-33a)
CH2SCH2(D1-34a) CH2(D1-34a)
CH2SCH2(D1-34a) CH2(D1-37a)
CH2SCH2(D1-34a) CH2(D1-81a)
CH2SCH2(D1-34a) CH2(D1-82a)
CH2SCH2(D1-34a) CH2(D1-84a)
CH2SCH2(D1-34a) CH2(D1-85a)
CH2SCH2(D1-34a) CH2(D1-87a)
CH2SCH2(D1-34a) CH2(D1-92a)
CH2SCH2(D1-34a) CH2(D1-93a)
CH2SCH2(D1-34a) CH2(D1-95a)
CH2SCH2(D1-34a) CH2(D1-96a)
CH2SCH2(D1-34a) CH2(D1-98a)
CH2SCH2(D1-34a) CH2(D1-108a)
CH2SCH2(D1-34a) CH2(D1-108b,Z=2-Cl)
CH2SCH2(D1-34a) CH2(D1-108b,Z=3-Me)
CH2SCH2(D1-34a) CH2(D1-108b,Z=4-OMe)
CH2SCH2(D1-34a) CH2(D1-108b,Z=2-SMe)
CH2SCH2(D1-34a) CH2(D1-108b,Z=3-CF3)
CH2SCH2(D1-34a) CH2(D1-108b,Z=4-OCF3)
CH2SCH2(D1-34a) CH2(D1-108b,Z=2-SCF3)
CH2SCH2(D1-34a) CH2CH2CN
CH2SCH2(D1-34a) CH2CH2CF3
CH2SCH2(D1-34a) CH2CH2OMe
CH2SCH2(D1-34a) CH2CH2SMe
CH2SCH2(D1-34a) CH2CH2S(O)Me
CH2SCH2(D1-34a) CH2CH2S(O)2Me
CH2SCH2(D1-34a) D1-32a
CH2SCH2(D1-34a) D1-33a
CH2SCH2(D1-34a) D1-34a
CH2SCH2(D1-34a) D1-37a
CH2SCH2(D1-34a) D1-81a
CH2SCH2(D1-34a) D1-82a
CH2SCH2(D1-34a) D1-84a
CH2SCH2(D1-34a) D1-85a
CH2SCH2(D1-34a) D1-87a
CH2SCH2(D1-34a) D1-92a
CH2SCH2(D1-34a) D1-93a
CH2SCH2(D1-34a) D1-95a
CH2SCH2(D1-34a) D1-96a
CH2SCH2(D1-34a) D1-98a
CH2SCH2(D1-34a) D1-108a
CH2SCH2(D1-34a) D1-108b(Z=2-Cl)
CH2SCH2(D1-34a) D1-108b(Z=3-Me)
CH2SCH2(D1-34a) D1-108b(Z=4-OMe)
CH2SCH2(D1-34a) D1-108b(Z=2-SMe)
CH2SCH2(D1-34a) D1-108b(Z=3-CF3)
CH2SCH2(D1-34a) D1-108b(Z=4-OCF3)
CH2SCH2(D1-34a) D1-108b(Z=2-SCF3)
CH2SCH2(D1-34a) C(O)Me
CH2SCH2(D1-34a) C(O)CF3
CH2SCH2(D1-34a) C(O)OMe
CH2S(O)CH2(D1-34a) Me
CH2S(O)CH2(D1-34a) Et
CH2S(O)CH2(D1-34a) Pr-n
CH2S(O)CH2(D1-34a) Pr-i
CH2S(O)CH2(D1-34a) Pr-c
CH2S(O)CH2(D1-34a) Bu-n
CH2S(O)CH2(D1-34a) Bu-i
CH2S(O)CH2(D1-34a) Bu-c
CH2S(O)CH2(D1-34a) Bu-s
CH2S(O)CH2(D1-34a) Bu-t
CH2S(O)CH2(D1-34a) Pen-n
CH2S(O)CH2(D1-34a) Pen-c
CH2S(O)CH2(D1-34a) Hex-n
CH2S(O)CH2(D1-34a) Hex-c
CH2S(O)CH2(D1-34a) CH2Pr-c
CH2S(O)CH2(D1-34a) CH2Bu-c
CH2S(O)CH2(D1-34a) CH2Pen-c
CH2S(O)CH2(D1-34a) CH2Hex-c
CH2S(O)CH2(D1-34a) CH2CH=CH2
CH2S(O)CH2(D1-34a) CH2CH=C(Cl)2
CH2S(O)CH2(D1-34a) CH2C≡CH
CH2S(O)CH2(D1-34a) CH2CN
CH2S(O)CH2(D1-34a) CH2CF3
CH2S(O)CH2(D1-34a) CH2OMe
CH2S(O)CH2(D1-34a) CH2OCF3
CH2S(O)CH2(D1-34a) CH2SMe
CH2S(O)CH2(D1-34a) CH2S(O)Me
CH2S(O)CH2(D1-34a) CH2S(O)2Me
CH2S(O)CH2(D1-34a) CH2SCF3
CH2S(O)CH2(D1-34a) CH2S(O)CF3
CH2S(O)CH2(D1-34a) CH2S(O)2CF3
CH2S(O)CH2(D1-34a) CH2CH(OMe)2
CH2S(O)CH2(D1-34a) CH2CH(SMe)2
CH2S(O)CH2(D1-34a) CH2C(O)Me
CH2S(O)CH2(D1-34a) CH2C(O)CF3
CH2S(O)CH2(D1-34a) CH2C(O)OMe
CH2S(O)CH2(D1-34a) CH2(D1-32a)
CH2S(O)CH2(D1-34a) CH2(D1-33a)
CH2S(O)CH2(D1-34a) CH2(D1-34a)
CH2S(O)CH2(D1-34a) CH2(D1-37a)
CH2S(O)CH2(D1-34a) CH2(D1-81a)
CH2S(O)CH2(D1-34a) CH2(D1-82a)
CH2S(O)CH2(D1-34a) CH2(D1-84a)
CH2S(O)CH2(D1-34a) CH2(D1-85a)
CH2S(O)CH2(D1-34a) CH2(D1-87a)
CH2S(O)CH2(D1-34a) CH2(D1-92a)
CH2S(O)CH2(D1-34a) CH2(D1-93a)
CH2S(O)CH2(D1-34a) CH2(D1-95a)
CH2S(O)CH2(D1-34a) CH2(D1-96a)
CH2S(O)CH2(D1-34a) CH2(D1-98a)
CH2S(O)CH2(D1-34a) CH2(D1-108a)
CH2S(O)CH2(D1-34a) CH2(D1-108b,Z=2-Cl)
CH2S(O)CH2(D1-34a) CH2(D1-108b,Z=3-Me)
CH2S(O)CH2(D1-34a) CH2(D1-108b,Z=4-OMe)
CH2S(O)CH2(D1-34a) CH2(D1-108b,Z=2-SMe)
CH2S(O)CH2(D1-34a) CH2(D1-108b,Z=3-CF3)
CH2S(O)CH2(D1-34a) CH2(D1-108b,Z=4-OCF3)
CH2S(O)CH2(D1-34a) CH2(D1-108b,Z=2-SCF3)
CH2S(O)CH2(D1-34a) CH2CH2CN
CH2S(O)CH2(D1-34a) CH2CH2CF3
CH2S(O)CH2(D1-34a) CH2CH2OMe
CH2S(O)CH2(D1-34a) CH2CH2SMe
CH2S(O)CH2(D1-34a) CH2CH2S(O)Me
CH2S(O)CH2(D1-34a) CH2CH2S(O)2Me
CH2S(O)CH2(D1-34a) D1-32a
CH2S(O)CH2(D1-34a) D1-33a
CH2S(O)CH2(D1-34a) D1-34a
CH2S(O)CH2(D1-34a) D1-37a
CH2S(O)CH2(D1-34a) D1-81a
CH2S(O)CH2(D1-34a) D1-82a
CH2S(O)CH2(D1-34a) D1-84a
CH2S(O)CH2(D1-34a) D1-85a
CH2S(O)CH2(D1-34a) D1-87a
CH2S(O)CH2(D1-34a) D1-92a
CH2S(O)CH2(D1-34a) D1-93a
CH2S(O)CH2(D1-34a) D1-95a
CH2S(O)CH2(D1-34a) D1-96a
CH2S(O)CH2(D1-34a) D1-98a
CH2S(O)CH2(D1-34a) D1-108a
CH2S(O)CH2(D1-34a) D1-108b(Z=2-Cl)
CH2S(O)CH2(D1-34a) D1-108b(Z=3-Me)
CH2S(O)CH2(D1-34a) D1-108b(Z=4-OMe)
CH2S(O)CH2(D1-34a) D1-108b(Z=2-SMe)
CH2S(O)CH2(D1-34a) D1-108b(Z=3-CF3)
CH2S(O)CH2(D1-34a) D1-108b(Z=4-OCF3)
CH2S(O)CH2(D1-34a) D1-108b(Z=2-SCF3)
CH2S(O)CH2(D1-34a) C(O)Me
CH2S(O)CH2(D1-34a) C(O)CF3
CH2S(O)CH2(D1-34a) C(O)OMe
CH2S(O)2CH2(D1-34a) Me
CH2S(O)2CH2(D1-34a) Et
CH2S(O)2CH2(D1-34a) Pr-n
CH2S(O)2CH2(D1-34a) Pr-i
CH2S(O)2CH2(D1-34a) Pr-c
CH2S(O)2CH2(D1-34a) Bu-n
CH2S(O)2CH2(D1-34a) Bu-i
CH2S(O)2CH2(D1-34a) Bu-c
CH2S(O)2CH2(D1-34a) Bu-s
CH2S(O)2CH2(D1-34a) Bu-t
CH2S(O)2CH2(D1-34a) Pen-n
CH2S(O)2CH2(D1-34a) Pen-c
CH2S(O)2CH2(D1-34a) Hex-n
CH2S(O)2CH2(D1-34a) Hex-c
CH2S(O)2CH2(D1-34a) CH2Pr-c
CH2S(O)2CH2(D1-34a) CH2Bu-c
CH2S(O)2CH2(D1-34a) CH2Pen-c
CH2S(O)2CH2(D1-34a) CH2Hex-c
CH2S(O)2CH2(D1-34a) CH2CH=CH2
CH2S(O)2CH2(D1-34a) CH2CH=C(Cl)2
CH2S(O)2CH2(D1-34a) CH2C≡CH
CH2S(O)2CH2(D1-34a) CH2CN
CH2S(O)2CH2(D1-34a) CH2CF3
CH2S(O)2CH2(D1-34a) CH2OMe
CH2S(O)2CH2(D1-34a) CH2OCF3
CH2S(O)2CH2(D1-34a) CH2SMe
CH2S(O)2CH2(D1-34a) CH2S(O)Me
CH2S(O)2CH2(D1-34a) CH2S(O)2Me
CH2S(O)2CH2(D1-34a) CH2SCF3
CH2S(O)2CH2(D1-34a) CH2S(O)CF3
CH2S(O)2CH2(D1-34a) CH2S(O)2CF3
CH2S(O)2CH2(D1-34a) CH2CH(OMe)2
CH2S(O)2CH2(D1-34a) CH2CH(SMe)2
CH2S(O)2CH2(D1-34a) CH2C(O)Me
CH2S(O)2CH2(D1-34a) CH2C(O)CF3
CH2S(O)2CH2(D1-34a) CH2C(O)OMe
CH2S(O)2CH2(D1-34a) CH2(D1-32a)
CH2S(O)2CH2(D1-34a) CH2(D1-33a)
CH2S(O)2CH2(D1-34a) CH2(D1-34a)
CH2S(O)2CH2(D1-34a) CH2(D1-37a)
CH2S(O)2CH2(D1-34a) CH2(D1-81a)
CH2S(O)2CH2(D1-34a) CH2(D1-82a)
CH2S(O)2CH2(D1-34a) CH2(D1-84a)
CH2S(O)2CH2(D1-34a) CH2(D1-85a)
CH2S(O)2CH2(D1-34a) CH2(D1-87a)
CH2S(O)2CH2(D1-34a) CH2(D1-92a)
CH2S(O)2CH2(D1-34a) CH2(D1-93a)
CH2S(O)2CH2(D1-34a) CH2(D1-95a)
CH2S(O)2CH2(D1-34a) CH2(D1-96a)
CH2S(O)2CH2(D1-34a) CH2(D1-98a)
CH2S(O)2CH2(D1-34a) CH2(D1-108a)
CH2S(O)2CH2(D1-34a) CH2(D1-108b,Z=2-Cl)
CH2S(O)2CH2(D1-34a) CH2(D1-108b,Z=3-Me)
CH2S(O)2CH2(D1-34a) CH2(D1-108b,Z=4-OMe)
CH2S(O)2CH2(D1-34a) CH2(D1-108b,Z=2-SMe)
CH2S(O)2CH2(D1-34a) CH2(D1-108b,Z=3-CF3)
CH2S(O)2CH2(D1-34a) CH2(D1-108b,Z=4-OCF3)
CH2S(O)2CH2(D1-34a) CH2(D1-108b,Z=2-SCF3)
CH2S(O)2CH2(D1-34a) CH2CH2CN
CH2S(O)2CH2(D1-34a) CH2CH2CF3
CH2S(O)2CH2(D1-34a) CH2CH2OMe
CH2S(O)2CH2(D1-34a) CH2CH2SMe
CH2S(O)2CH2(D1-34a) CH2CH2S(O)Me
CH2S(O)2CH2(D1-34a) CH2CH2S(O)2Me
CH2S(O)2CH2(D1-34a) D1-32a
CH2S(O)2CH2(D1-34a) D1-33a
CH2S(O)2CH2(D1-34a) D1-34a
CH2S(O)2CH2(D1-34a) D1-37a
CH2S(O)2CH2(D1-34a) D1-81a
CH2S(O)2CH2(D1-34a) D1-82a
CH2S(O)2CH2(D1-34a) D1-84a
CH2S(O)2CH2(D1-34a) D1-85a
CH2S(O)2CH2(D1-34a) D1-87a
CH2S(O)2CH2(D1-34a) D1-92a
CH2S(O)2CH2(D1-34a) D1-93a
CH2S(O)2CH2(D1-34a) D1-95a
CH2S(O)2CH2(D1-34a) D1-96a
CH2S(O)2CH2(D1-34a) D1-98a
CH2S(O)2CH2(D1-34a) D1-108a
CH2S(O)2CH2(D1-34a) D1-108b(Z=2-Cl)
CH2S(O)2CH2(D1-34a) D1-108b(Z=3-Me)
CH2S(O)2CH2(D1-34a) D1-108b(Z=4-OMe)
CH2S(O)2CH2(D1-34a) D1-108b(Z=2-SMe)
CH2S(O)2CH2(D1-34a) D1-108b(Z=3-CF3)
CH2S(O)2CH2(D1-34a) D1-108b(Z=4-OCF3)
CH2S(O)2CH2(D1-34a) D1-108b(Z=2-SCF3)
CH2S(O)2CH2(D1-34a) C(O)Me
CH2S(O)2CH2(D1-34a) C(O)CF3
CH2S(O)2CH2(D1-34a) C(O)OMe
CH(Me)SCH2(D1-34a) Me
CH(Me)SCH2(D1-34a) Et
CH(Me)SCH2(D1-34a) Pr-n
CH(Me)SCH2(D1-34a) Pr-i
CH(Me)SCH2(D1-34a) Pr-c
CH(Me)SCH2(D1-34a) Bu-n
CH(Me)SCH2(D1-34a) Bu-i
CH(Me)SCH2(D1-34a) Bu-c
CH(Me)SCH2(D1-34a) Bu-s
CH(Me)SCH2(D1-34a) Bu-t
CH(Me)SCH2(D1-34a) Pen-n
CH(Me)SCH2(D1-34a) Pen-c
CH(Me)SCH2(D1-34a) Hex-n
CH(Me)SCH2(D1-34a) Hex-c
CH(Me)SCH2(D1-34a) CH2Pr-c
CH(Me)SCH2(D1-34a) CH2Bu-c
CH(Me)SCH2(D1-34a) CH2Pen-c
CH(Me)SCH2(D1-34a) CH2Hex-c
CH(Me)SCH2(D1-34a) CH2CH=CH2
CH(Me)SCH2(D1-34a) CH2CH=C(Cl)2
CH(Me)SCH2(D1-34a) CH2C≡CH
CH(Me)SCH2(D1-34a) CH2CN
CH(Me)SCH2(D1-34a) CH2CF3
CH(Me)SCH2(D1-34a) CH2OMe
CH(Me)SCH2(D1-34a) CH2OCF3
CH(Me)SCH2(D1-34a) CH2SMe
CH(Me)SCH2(D1-34a) CH2S(O)Me
CH(Me)SCH2(D1-34a) CH2S(O)2Me
CH(Me)SCH2(D1-34a) CH2SCF3
CH(Me)SCH2(D1-34a) CH2S(O)CF3
CH(Me)SCH2(D1-34a) CH2S(O)2CF3
CH(Me)SCH2(D1-34a) CH2CH(OMe)2
CH(Me)SCH2(D1-34a) CH2CH(SMe)2
CH(Me)SCH2(D1-34a) CH2C(O)Me
CH(Me)SCH2(D1-34a) CH2C(O)CF3
CH(Me)SCH2(D1-34a) CH2C(O)OMe
CH(Me)SCH2(D1-34a) CH2(D1-32a)
CH(Me)SCH2(D1-34a) CH2(D1-33a)
CH(Me)SCH2(D1-34a) CH2(D1-34a)
CH(Me)SCH2(D1-34a) CH2(D1-37a)
CH(Me)SCH2(D1-34a) CH2(D1-81a)
CH(Me)SCH2(D1-34a) CH2(D1-82a)
CH(Me)SCH2(D1-34a) CH2(D1-84a)
CH(Me)SCH2(D1-34a) CH2(D1-85a)
CH(Me)SCH2(D1-34a) CH2(D1-87a)
CH(Me)SCH2(D1-34a) CH2(D1-92a)
CH(Me)SCH2(D1-34a) CH2(D1-93a)
CH(Me)SCH2(D1-34a) CH2(D1-95a)
CH(Me)SCH2(D1-34a) CH2(D1-96a)
CH(Me)SCH2(D1-34a) CH2(D1-98a)
CH(Me)SCH2(D1-34a) CH2(D1-108a)
CH(Me)SCH2(D1-34a) CH2(D1-108b,Z=2-Cl)
CH(Me)SCH2(D1-34a) CH2(D1-108b,Z=3-Me)
CH(Me)SCH2(D1-34a) CH2(D1-108b,Z=4-OMe)
CH(Me)SCH2(D1-34a) CH2(D1-108b,Z=2-SMe)
CH(Me)SCH2(D1-34a) CH2(D1-108b,Z=3-CF3)
CH(Me)SCH2(D1-34a) CH2(D1-108b,Z=4-OCF3)
CH(Me)SCH2(D1-34a) CH2(D1-108b,Z=2-SCF3)
CH(Me)SCH2(D1-34a) CH2CH2CN
CH(Me)SCH2(D1-34a) CH2CH2CF3
CH(Me)SCH2(D1-34a) CH2CH2OMe
CH(Me)SCH2(D1-34a) CH2CH2SMe
CH(Me)SCH2(D1-34a) CH2CH2S(O)Me
CH(Me)SCH2(D1-34a) CH2CH2S(O)2Me
CH(Me)SCH2(D1-34a) D1-32a
CH(Me)SCH2(D1-34a) D1-33a
CH(Me)SCH2(D1-34a) D1-34a
CH(Me)SCH2(D1-34a) D1-37a
CH(Me)SCH2(D1-34a) D1-81a
CH(Me)SCH2(D1-34a) D1-82a
CH(Me)SCH2(D1-34a) D1-84a
CH(Me)SCH2(D1-34a) D1-85a
CH(Me)SCH2(D1-34a) D1-87a
CH(Me)SCH2(D1-34a) D1-92a
CH(Me)SCH2(D1-34a) D1-93a
CH(Me)SCH2(D1-34a) D1-95a
CH(Me)SCH2(D1-34a) D1-96a
CH(Me)SCH2(D1-34a) D1-98a
CH(Me)SCH2(D1-34a) D1-108a
CH(Me)SCH2(D1-34a) D1-108b(Z=2-Cl)
CH(Me)SCH2(D1-34a) D1-108b(Z=3-Me)
CH(Me)SCH2(D1-34a) D1-108b(Z=4-OMe)
CH(Me)SCH2(D1-34a) D1-108b(Z=2-SMe)
CH(Me)SCH2(D1-34a) D1-108b(Z=3-CF3)
CH(Me)SCH2(D1-34a) D1-108b(Z=4-OCF3)
CH(Me)SCH2(D1-34a) D1-108b(Z=2-SCF3)
CH(Me)SCH2(D1-34a) C(O)Me
CH(Me)SCH2(D1-34a) C(O)CF3
CH(Me)SCH2(D1-34a) C(O)OMe
CH(Me)S(O)CH2(D1-34a) Me
CH(Me)S(O)CH2(D1-34a) Et
CH(Me)S(O)CH2(D1-34a) Pr-n
CH(Me)S(O)CH2(D1-34a) Pr-i
CH(Me)S(O)CH2(D1-34a) Pr-c
CH(Me)S(O)CH2(D1-34a) Bu-n
CH(Me)S(O)CH2(D1-34a) Bu-i
CH(Me)S(O)CH2(D1-34a) Bu-c
CH(Me)S(O)CH2(D1-34a) Bu-s
CH(Me)S(O)CH2(D1-34a) Bu-t
CH(Me)S(O)CH2(D1-34a) Pen-n
CH(Me)S(O)CH2(D1-34a) Pen-c
CH(Me)S(O)CH2(D1-34a) Hex-n
CH(Me)S(O)CH2(D1-34a) Hex-c
CH(Me)S(O)CH2(D1-34a) CH2Pr-c
CH(Me)S(O)CH2(D1-34a) CH2Bu-c
CH(Me)S(O)CH2(D1-34a) CH2Pen-c
CH(Me)S(O)CH2(D1-34a) CH2Hex-c
CH(Me)S(O)CH2(D1-34a) CH2CH=CH2
CH(Me)S(O)CH2(D1-34a) CH2CH=C(Cl)2
CH(Me)S(O)CH2(D1-34a) CH2C≡CH
CH(Me)S(O)CH2(D1-34a) CH2CN
CH(Me)S(O)CH2(D1-34a) CH2CF3
CH(Me)S(O)CH2(D1-34a) CH2OMe
CH(Me)S(O)CH2(D1-34a) CH2OCF3
CH(Me)S(O)CH2(D1-34a) CH2SMe
CH(Me)S(O)CH2(D1-34a) CH2S(O)Me
CH(Me)S(O)CH2(D1-34a) CH2S(O)2Me
CH(Me)S(O)CH2(D1-34a) CH2SCF3
CH(Me)S(O)CH2(D1-34a) CH2S(O)CF3
CH(Me)S(O)CH2(D1-34a) CH2S(O)2CF3
CH(Me)S(O)CH2(D1-34a) CH2CH(OMe)2
CH(Me)S(O)CH2(D1-34a) CH2CH(SMe)2
CH(Me)S(O)CH2(D1-34a) CH2C(O)Me
CH(Me)S(O)CH2(D1-34a) CH2C(O)CF3
CH(Me)S(O)CH2(D1-34a) CH2C(O)OMe
CH(Me)S(O)CH2(D1-34a) CH2(D1-32a)
CH(Me)S(O)CH2(D1-34a) CH2(D1-33a)
CH(Me)S(O)CH2(D1-34a) CH2(D1-34a)
CH(Me)S(O)CH2(D1-34a) CH2(D1-37a)
CH(Me)S(O)CH2(D1-34a) CH2(D1-81a)
CH(Me)S(O)CH2(D1-34a) CH2(D1-82a)
CH(Me)S(O)CH2(D1-34a) CH2(D1-84a)
CH(Me)S(O)CH2(D1-34a) CH2(D1-85a)
CH(Me)S(O)CH2(D1-34a) CH2(D1-87a)
CH(Me)S(O)CH2(D1-34a) CH2(D1-92a)
CH(Me)S(O)CH2(D1-34a) CH2(D1-93a)
CH(Me)S(O)CH2(D1-34a) CH2(D1-95a)
CH(Me)S(O)CH2(D1-34a) CH2(D1-96a)
CH(Me)S(O)CH2(D1-34a) CH2(D1-98a)
CH(Me)S(O)CH2(D1-34a) CH2(D1-108a)
CH(Me)S(O)CH2(D1-34a) CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)CH2(D1-34a) CH2(D1-108b,Z=3-Me)
CH(Me)S(O)CH2(D1-34a) CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)CH2(D1-34a) CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)CH2(D1-34a) CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)CH2(D1-34a) CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)CH2(D1-34a) CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)CH2(D1-34a) CH2CH2CN
CH(Me)S(O)CH2(D1-34a) CH2CH2CF3
CH(Me)S(O)CH2(D1-34a) CH2CH2OMe
CH(Me)S(O)CH2(D1-34a) CH2CH2SMe
CH(Me)S(O)CH2(D1-34a) CH2CH2S(O)Me
CH(Me)S(O)CH2(D1-34a) CH2CH2S(O)2Me
CH(Me)S(O)CH2(D1-34a) D1-32a
CH(Me)S(O)CH2(D1-34a) D1-33a
CH(Me)S(O)CH2(D1-34a) D1-34a
CH(Me)S(O)CH2(D1-34a) D1-37a
CH(Me)S(O)CH2(D1-34a) D1-81a
CH(Me)S(O)CH2(D1-34a) D1-82a
CH(Me)S(O)CH2(D1-34a) D1-84a
CH(Me)S(O)CH2(D1-34a) D1-85a
CH(Me)S(O)CH2(D1-34a) D1-87a
CH(Me)S(O)CH2(D1-34a) D1-92a
CH(Me)S(O)CH2(D1-34a) D1-93a
CH(Me)S(O)CH2(D1-34a) D1-95a
CH(Me)S(O)CH2(D1-34a) D1-96a
CH(Me)S(O)CH2(D1-34a) D1-98a
CH(Me)S(O)CH2(D1-34a) D1-108a
CH(Me)S(O)CH2(D1-34a) D1-108b(Z=2-Cl)
CH(Me)S(O)CH2(D1-34a) D1-108b(Z=3-Me)
CH(Me)S(O)CH2(D1-34a) D1-108b(Z=4-OMe)
CH(Me)S(O)CH2(D1-34a) D1-108b(Z=2-SMe)
CH(Me)S(O)CH2(D1-34a) D1-108b(Z=3-CF3)
CH(Me)S(O)CH2(D1-34a) D1-108b(Z=4-OCF3)
CH(Me)S(O)CH2(D1-34a) D1-108b(Z=2-SCF3)
CH(Me)S(O)CH2(D1-34a) C(O)Me
CH(Me)S(O)CH2(D1-34a) C(O)CF3
CH(Me)S(O)CH2(D1-34a) C(O)OMe
CH(Me)S(O)2CH2(D1-34a) Me
CH(Me)S(O)2CH2(D1-34a) Et
CH(Me)S(O)2CH2(D1-34a) Pr-n
CH(Me)S(O)2CH2(D1-34a) Pr-i
CH(Me)S(O)2CH2(D1-34a) Pr-c
CH(Me)S(O)2CH2(D1-34a) Bu-n
CH(Me)S(O)2CH2(D1-34a) Bu-i
CH(Me)S(O)2CH2(D1-34a) Bu-c
CH(Me)S(O)2CH2(D1-34a) Bu-s
CH(Me)S(O)2CH2(D1-34a) Bu-t
CH(Me)S(O)2CH2(D1-34a) Pen-n
CH(Me)S(O)2CH2(D1-34a) Pen-c
CH(Me)S(O)2CH2(D1-34a) Hex-n
CH(Me)S(O)2CH2(D1-34a) Hex-c
CH(Me)S(O)2CH2(D1-34a) CH2Pr-c
CH(Me)S(O)2CH2(D1-34a) CH2Bu-c
CH(Me)S(O)2CH2(D1-34a) CH2Pen-c
CH(Me)S(O)2CH2(D1-34a) CH2Hex-c
CH(Me)S(O)2CH2(D1-34a) CH2CH=CH2
CH(Me)S(O)2CH2(D1-34a) CH2CH=C(Cl)2
CH(Me)S(O)2CH2(D1-34a) CH2C≡CH
CH(Me)S(O)2CH2(D1-34a) CH2CN
CH(Me)S(O)2CH2(D1-34a) CH2CF3
CH(Me)S(O)2CH2(D1-34a) CH2OMe
CH(Me)S(O)2CH2(D1-34a) CH2OCF3
CH(Me)S(O)2CH2(D1-34a) CH2SMe
CH(Me)S(O)2CH2(D1-34a) CH2S(O)Me
CH(Me)S(O)2CH2(D1-34a) CH2S(O)2Me
CH(Me)S(O)2CH2(D1-34a) CH2SCF3
CH(Me)S(O)2CH2(D1-34a) CH2S(O)CF3
CH(Me)S(O)2CH2(D1-34a) CH2S(O)2CF3
CH(Me)S(O)2CH2(D1-34a) CH2CH(OMe)2
CH(Me)S(O)2CH2(D1-34a) CH2CH(SMe)2
CH(Me)S(O)2CH2(D1-34a) CH2C(O)Me
CH(Me)S(O)2CH2(D1-34a) CH2C(O)CF3
CH(Me)S(O)2CH2(D1-34a) CH2C(O)OMe
CH(Me)S(O)2CH2(D1-34a) CH2(D1-32a)
CH(Me)S(O)2CH2(D1-34a) CH2(D1-33a)
CH(Me)S(O)2CH2(D1-34a) CH2(D1-34a)
CH(Me)S(O)2CH2(D1-34a) CH2(D1-37a)
CH(Me)S(O)2CH2(D1-34a) CH2(D1-81a)
CH(Me)S(O)2CH2(D1-34a) CH2(D1-82a)
CH(Me)S(O)2CH2(D1-34a) CH2(D1-84a)
CH(Me)S(O)2CH2(D1-34a) CH2(D1-85a)
CH(Me)S(O)2CH2(D1-34a) CH2(D1-87a)
CH(Me)S(O)2CH2(D1-34a) CH2(D1-92a)
CH(Me)S(O)2CH2(D1-34a) CH2(D1-93a)
CH(Me)S(O)2CH2(D1-34a) CH2(D1-95a)
CH(Me)S(O)2CH2(D1-34a) CH2(D1-96a)
CH(Me)S(O)2CH2(D1-34a) CH2(D1-98a)
CH(Me)S(O)2CH2(D1-34a) CH2(D1-108a)
CH(Me)S(O)2CH2(D1-34a) CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)2CH2(D1-34a) CH2(D1-108b,Z=3-Me)
CH(Me)S(O)2CH2(D1-34a) CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)2CH2(D1-34a) CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)2CH2(D1-34a) CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)2CH2(D1-34a) CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)2CH2(D1-34a) CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)2CH2(D1-34a) CH2CH2CN
CH(Me)S(O)2CH2(D1-34a) CH2CH2CF3
CH(Me)S(O)2CH2(D1-34a) CH2CH2OMe
CH(Me)S(O)2CH2(D1-34a) CH2CH2SMe
CH(Me)S(O)2CH2(D1-34a) CH2CH2S(O)Me
CH(Me)S(O)2CH2(D1-34a) CH2CH2S(O)2Me
CH(Me)S(O)2CH2(D1-34a) D1-32a
CH(Me)S(O)2CH2(D1-34a) D1-33a
CH(Me)S(O)2CH2(D1-34a) D1-34a
CH(Me)S(O)2CH2(D1-34a) D1-37a
CH(Me)S(O)2CH2(D1-34a) D1-81a
CH(Me)S(O)2CH2(D1-34a) D1-82a
CH(Me)S(O)2CH2(D1-34a) D1-84a
CH(Me)S(O)2CH2(D1-34a) D1-85a
CH(Me)S(O)2CH2(D1-34a) D1-87a
CH(Me)S(O)2CH2(D1-34a) D1-92a
CH(Me)S(O)2CH2(D1-34a) D1-93a
CH(Me)S(O)2CH2(D1-34a) D1-95a
CH(Me)S(O)2CH2(D1-34a) D1-96a
CH(Me)S(O)2CH2(D1-34a) D1-98a
CH(Me)S(O)2CH2(D1-34a) D1-108a
CH(Me)S(O)2CH2(D1-34a) D1-108b(Z=2-Cl)
CH(Me)S(O)2CH2(D1-34a) D1-108b(Z=3-Me)
CH(Me)S(O)2CH2(D1-34a) D1-108b(Z=4-OMe)
CH(Me)S(O)2CH2(D1-34a) D1-108b(Z=2-SMe)
CH(Me)S(O)2CH2(D1-34a) D1-108b(Z=3-CF3)
CH(Me)S(O)2CH2(D1-34a) D1-108b(Z=4-OCF3)
CH(Me)S(O)2CH2(D1-34a) D1-108b(Z=2-SCF3)
CH(Me)S(O)2CH2(D1-34a) C(O)Me
CH(Me)S(O)2CH2(D1-34a) C(O)CF3
CH(Me)S(O)2CH2(D1-34a) C(O)OMe
CH(Et)SCH2(D1-34a) Me
CH(Et)SCH2(D1-34a) Et
CH(Et)SCH2(D1-34a) Pr-n
CH(Et)SCH2(D1-34a) Pr-i
CH(Et)SCH2(D1-34a) Pr-c
CH(Et)SCH2(D1-34a) Bu-n
CH(Et)SCH2(D1-34a) Bu-i
CH(Et)SCH2(D1-34a) Bu-c
CH(Et)SCH2(D1-34a) Bu-s
CH(Et)SCH2(D1-34a) Bu-t
CH(Et)SCH2(D1-34a) Pen-n
CH(Et)SCH2(D1-34a) Pen-c
CH(Et)SCH2(D1-34a) Hex-n
CH(Et)SCH2(D1-34a) Hex-c
CH(Et)SCH2(D1-34a) CH2Pr-c
CH(Et)SCH2(D1-34a) CH2Bu-c
CH(Et)SCH2(D1-34a) CH2Pen-c
CH(Et)SCH2(D1-34a) CH2Hex-c
CH(Et)SCH2(D1-34a) CH2CH=CH2
CH(Et)SCH2(D1-34a) CH2CH=C(Cl)2
CH(Et)SCH2(D1-34a) CH2C≡CH
CH(Et)SCH2(D1-34a) CH2CN
CH(Et)SCH2(D1-34a) CH2CF3
CH(Et)SCH2(D1-34a) CH2OMe
CH(Et)SCH2(D1-34a) CH2OCF3
CH(Et)SCH2(D1-34a) CH2SMe
CH(Et)SCH2(D1-34a) CH2S(O)Me
CH(Et)SCH2(D1-34a) CH2S(O)2Me
CH(Et)SCH2(D1-34a) CH2SCF3
CH(Et)SCH2(D1-34a) CH2S(O)CF3
CH(Et)SCH2(D1-34a) CH2S(O)2CF3
CH(Et)SCH2(D1-34a) CH2CH(OMe)2
CH(Et)SCH2(D1-34a) CH2CH(SMe)2
CH(Et)SCH2(D1-34a) CH2C(O)Me
CH(Et)SCH2(D1-34a) CH2C(O)CF3
CH(Et)SCH2(D1-34a) CH2C(O)OMe
CH(Et)SCH2(D1-34a) CH2(D1-32a)
CH(Et)SCH2(D1-34a) CH2(D1-33a)
CH(Et)SCH2(D1-34a) CH2(D1-34a)
CH(Et)SCH2(D1-34a) CH2(D1-37a)
CH(Et)SCH2(D1-34a) CH2(D1-81a)
CH(Et)SCH2(D1-34a) CH2(D1-82a)
CH(Et)SCH2(D1-34a) CH2(D1-84a)
CH(Et)SCH2(D1-34a) CH2(D1-85a)
CH(Et)SCH2(D1-34a) CH2(D1-87a)
CH(Et)SCH2(D1-34a) CH2(D1-92a)
CH(Et)SCH2(D1-34a) CH2(D1-93a)
CH(Et)SCH2(D1-34a) CH2(D1-95a)
CH(Et)SCH2(D1-34a) CH2(D1-96a)
CH(Et)SCH2(D1-34a) CH2(D1-98a)
CH(Et)SCH2(D1-34a) CH2(D1-108a)
CH(Et)SCH2(D1-34a) CH2(D1-108b,Z=2-Cl)
CH(Et)SCH2(D1-34a) CH2(D1-108b,Z=3-Me)
CH(Et)SCH2(D1-34a) CH2(D1-108b,Z=4-OMe)
CH(Et)SCH2(D1-34a) CH2(D1-108b,Z=2-SMe)
CH(Et)SCH2(D1-34a) CH2(D1-108b,Z=3-CF3)
CH(Et)SCH2(D1-34a) CH2(D1-108b,Z=4-OCF3)
CH(Et)SCH2(D1-34a) CH2(D1-108b,Z=2-SCF3)
CH(Et)SCH2(D1-34a) CH2CH2CN
CH(Et)SCH2(D1-34a) CH2CH2CF3
CH(Et)SCH2(D1-34a) CH2CH2OMe
CH(Et)SCH2(D1-34a) CH2CH2SMe
CH(Et)SCH2(D1-34a) CH2CH2S(O)Me
CH(Et)SCH2(D1-34a) CH2CH2S(O)2Me
CH(Et)SCH2(D1-34a) D1-32a
CH(Et)SCH2(D1-34a) D1-33a
CH(Et)SCH2(D1-34a) D1-34a
CH(Et)SCH2(D1-34a) D1-37a
CH(Et)SCH2(D1-34a) D1-81a
CH(Et)SCH2(D1-34a) D1-82a
CH(Et)SCH2(D1-34a) D1-84a
CH(Et)SCH2(D1-34a) D1-85a
CH(Et)SCH2(D1-34a) D1-87a
CH(Et)SCH2(D1-34a) D1-92a
CH(Et)SCH2(D1-34a) D1-93a
CH(Et)SCH2(D1-34a) D1-95a
CH(Et)SCH2(D1-34a) D1-96a
CH(Et)SCH2(D1-34a) D1-98a
CH(Et)SCH2(D1-34a) D1-108a
CH(Et)SCH2(D1-34a) D1-108b(Z=2-Cl)
CH(Et)SCH2(D1-34a) D1-108b(Z=3-Me)
CH(Et)SCH2(D1-34a) D1-108b(Z=4-OMe)
CH(Et)SCH2(D1-34a) D1-108b(Z=2-SMe)
CH(Et)SCH2(D1-34a) D1-108b(Z=3-CF3)
CH(Et)SCH2(D1-34a) D1-108b(Z=4-OCF3)
CH(Et)SCH2(D1-34a) D1-108b(Z=2-SCF3)
CH(Et)SCH2(D1-34a) C(O)Me
CH(Et)SCH2(D1-34a) C(O)CF3
CH(Et)SCH2(D1-34a) C(O)OMe
CH(Et)S(O)CH2(D1-34a) Me
CH(Et)S(O)CH2(D1-34a) Et
CH(Et)S(O)CH2(D1-34a) Pr-n
CH(Et)S(O)CH2(D1-34a) Pr-i
CH(Et)S(O)CH2(D1-34a) Pr-c
CH(Et)S(O)CH2(D1-34a) Bu-n
CH(Et)S(O)CH2(D1-34a) Bu-i
CH(Et)S(O)CH2(D1-34a) Bu-c
CH(Et)S(O)CH2(D1-34a) Bu-s
CH(Et)S(O)CH2(D1-34a) Bu-t
CH(Et)S(O)CH2(D1-34a) Pen-n
CH(Et)S(O)CH2(D1-34a) Pen-c
CH(Et)S(O)CH2(D1-34a) Hex-n
CH(Et)S(O)CH2(D1-34a) Hex-c
CH(Et)S(O)CH2(D1-34a) CH2Pr-c
CH(Et)S(O)CH2(D1-34a) CH2Bu-c
CH(Et)S(O)CH2(D1-34a) CH2Pen-c
CH(Et)S(O)CH2(D1-34a) CH2Hex-c
CH(Et)S(O)CH2(D1-34a) CH2CH=CH2
CH(Et)S(O)CH2(D1-34a) CH2CH=C(Cl)2
CH(Et)S(O)CH2(D1-34a) CH2C≡CH
CH(Et)S(O)CH2(D1-34a) CH2CN
CH(Et)S(O)CH2(D1-34a) CH2CF3
CH(Et)S(O)CH2(D1-34a) CH2OMe
CH(Et)S(O)CH2(D1-34a) CH2OCF3
CH(Et)S(O)CH2(D1-34a) CH2SMe
CH(Et)S(O)CH2(D1-34a) CH2S(O)Me
CH(Et)S(O)CH2(D1-34a) CH2S(O)2Me
CH(Et)S(O)CH2(D1-34a) CH2SCF3
CH(Et)S(O)CH2(D1-34a) CH2S(O)CF3
CH(Et)S(O)CH2(D1-34a) CH2S(O)2CF3
CH(Et)S(O)CH2(D1-34a) CH2CH(OMe)2
CH(Et)S(O)CH2(D1-34a) CH2CH(SMe)2
CH(Et)S(O)CH2(D1-34a) CH2C(O)Me
CH(Et)S(O)CH2(D1-34a) CH2C(O)CF3
CH(Et)S(O)CH2(D1-34a) CH2C(O)OMe
CH(Et)S(O)CH2(D1-34a) CH2(D1-32a)
CH(Et)S(O)CH2(D1-34a) CH2(D1-33a)
CH(Et)S(O)CH2(D1-34a) CH2(D1-34a)
CH(Et)S(O)CH2(D1-34a) CH2(D1-37a)
CH(Et)S(O)CH2(D1-34a) CH2(D1-81a)
CH(Et)S(O)CH2(D1-34a) CH2(D1-82a)
CH(Et)S(O)CH2(D1-34a) CH2(D1-84a)
CH(Et)S(O)CH2(D1-34a) CH2(D1-85a)
CH(Et)S(O)CH2(D1-34a) CH2(D1-87a)
CH(Et)S(O)CH2(D1-34a) CH2(D1-92a)
CH(Et)S(O)CH2(D1-34a) CH2(D1-93a)
CH(Et)S(O)CH2(D1-34a) CH2(D1-95a)
CH(Et)S(O)CH2(D1-34a) CH2(D1-96a)
CH(Et)S(O)CH2(D1-34a) CH2(D1-98a)
CH(Et)S(O)CH2(D1-34a) CH2(D1-108a)
CH(Et)S(O)CH2(D1-34a) CH2(D1-108b,Z=2-Cl)
CH(Et)S(O)CH2(D1-34a) CH2(D1-108b,Z=3-Me)
CH(Et)S(O)CH2(D1-34a) CH2(D1-108b,Z=4-OMe)
CH(Et)S(O)CH2(D1-34a) CH2(D1-108b,Z=2-SMe)
CH(Et)S(O)CH2(D1-34a) CH2(D1-108b,Z=3-CF3)
CH(Et)S(O)CH2(D1-34a) CH2(D1-108b,Z=4-OCF3)
CH(Et)S(O)CH2(D1-34a) CH2(D1-108b,Z=2-SCF3)
CH(Et)S(O)CH2(D1-34a) CH2CH2CN
CH(Et)S(O)CH2(D1-34a) CH2CH2CF3
CH(Et)S(O)CH2(D1-34a) CH2CH2OMe
CH(Et)S(O)CH2(D1-34a) CH2CH2SMe
CH(Et)S(O)CH2(D1-34a) CH2CH2S(O)Me
CH(Et)S(O)CH2(D1-34a) CH2CH2S(O)2Me
CH(Et)S(O)CH2(D1-34a) D1-32a
CH(Et)S(O)CH2(D1-34a) D1-33a
CH(Et)S(O)CH2(D1-34a) D1-34a
CH(Et)S(O)CH2(D1-34a) D1-37a
CH(Et)S(O)CH2(D1-34a) D1-81a
CH(Et)S(O)CH2(D1-34a) D1-82a
CH(Et)S(O)CH2(D1-34a) D1-84a
CH(Et)S(O)CH2(D1-34a) D1-85a
CH(Et)S(O)CH2(D1-34a) D1-87a
CH(Et)S(O)CH2(D1-34a) D1-92a
CH(Et)S(O)CH2(D1-34a) D1-93a
CH(Et)S(O)CH2(D1-34a) D1-95a
CH(Et)S(O)CH2(D1-34a) D1-96a
CH(Et)S(O)CH2(D1-34a) D1-98a
CH(Et)S(O)CH2(D1-34a) D1-108a
CH(Et)S(O)CH2(D1-34a) D1-108b(Z=2-Cl)
CH(Et)S(O)CH2(D1-34a) D1-108b(Z=3-Me)
CH(Et)S(O)CH2(D1-34a) D1-108b(Z=4-OMe)
CH(Et)S(O)CH2(D1-34a) D1-108b(Z=2-SMe)
CH(Et)S(O)CH2(D1-34a) D1-108b(Z=3-CF3)
CH(Et)S(O)CH2(D1-34a) D1-108b(Z=4-OCF3)
CH(Et)S(O)CH2(D1-34a) D1-108b(Z=2-SCF3)
CH(Et)S(O)CH2(D1-34a) C(O)Me
CH(Et)S(O)CH2(D1-34a) C(O)CF3
CH(Et)S(O)CH2(D1-34a) C(O)OMe
CH(Et)S(O)2CH2(D1-34a) Me
CH(Et)S(O)2CH2(D1-34a) Et
CH(Et)S(O)2CH2(D1-34a) Pr-n
CH(Et)S(O)2CH2(D1-34a) Pr-i
CH(Et)S(O)2CH2(D1-34a) Pr-c
CH(Et)S(O)2CH2(D1-34a) Bu-n
CH(Et)S(O)2CH2(D1-34a) Bu-i
CH(Et)S(O)2CH2(D1-34a) Bu-c
CH(Et)S(O)2CH2(D1-34a) Bu-s
CH(Et)S(O)2CH2(D1-34a) Bu-t
CH(Et)S(O)2CH2(D1-34a) Pen-n
CH(Et)S(O)2CH2(D1-34a) Pen-c
CH(Et)S(O)2CH2(D1-34a) Hex-n
CH(Et)S(O)2CH2(D1-34a) Hex-c
CH(Et)S(O)2CH2(D1-34a) CH2Pr-c
CH(Et)S(O)2CH2(D1-34a) CH2Bu-c
CH(Et)S(O)2CH2(D1-34a) CH2Pen-c
CH(Et)S(O)2CH2(D1-34a) CH2Hex-c
CH(Et)S(O)2CH2(D1-34a) CH2CH=CH2
CH(Et)S(O)2CH2(D1-34a) CH2CH=C(Cl)2
CH(Et)S(O)2CH2(D1-34a) CH2C≡CH
CH(Et)S(O)2CH2(D1-34a) CH2CN
CH(Et)S(O)2CH2(D1-34a) CH2CF3
CH(Et)S(O)2CH2(D1-34a) CH2OMe
CH(Et)S(O)2CH2(D1-34a) CH2OCF3
CH(Et)S(O)2CH2(D1-34a) CH2SMe
CH(Et)S(O)2CH2(D1-34a) CH2S(O)Me
CH(Et)S(O)2CH2(D1-34a) CH2S(O)2Me
CH(Et)S(O)2CH2(D1-34a) CH2SCF3
CH(Et)S(O)2CH2(D1-34a) CH2S(O)CF3
CH(Et)S(O)2CH2(D1-34a) CH2S(O)2CF3
CH(Et)S(O)2CH2(D1-34a) CH2CH(OMe)2
CH(Et)S(O)2CH2(D1-34a) CH2CH(SMe)2
CH(Et)S(O)2CH2(D1-34a) CH2C(O)Me
CH(Et)S(O)2CH2(D1-34a) CH2C(O)CF3
CH(Et)S(O)2CH2(D1-34a) CH2C(O)OMe
CH(Et)S(O)2CH2(D1-34a) CH2(D1-32a)
CH(Et)S(O)2CH2(D1-34a) CH2(D1-33a)
CH(Et)S(O)2CH2(D1-34a) CH2(D1-34a)
CH(Et)S(O)2CH2(D1-34a) CH2(D1-37a)
CH(Et)S(O)2CH2(D1-34a) CH2(D1-81a)
CH(Et)S(O)2CH2(D1-34a) CH2(D1-82a)
CH(Et)S(O)2CH2(D1-34a) CH2(D1-84a)
CH(Et)S(O)2CH2(D1-34a) CH2(D1-85a)
CH(Et)S(O)2CH2(D1-34a) CH2(D1-87a)
CH(Et)S(O)2CH2(D1-34a) CH2(D1-92a)
CH(Et)S(O)2CH2(D1-34a) CH2(D1-93a)
CH(Et)S(O)2CH2(D1-34a) CH2(D1-95a)
CH(Et)S(O)2CH2(D1-34a) CH2(D1-96a)
CH(Et)S(O)2CH2(D1-34a) CH2(D1-98a)
CH(Et)S(O)2CH2(D1-34a) CH2(D1-108a)
CH(Et)S(O)2CH2(D1-34a) CH2(D1-108b,Z=2-Cl)
CH(Et)S(O)2CH2(D1-34a) CH2(D1-108b,Z=3-Me)
CH(Et)S(O)2CH2(D1-34a) CH2(D1-108b,Z=4-OMe)
CH(Et)S(O)2CH2(D1-34a) CH2(D1-108b,Z=2-SMe)
CH(Et)S(O)2CH2(D1-34a) CH2(D1-108b,Z=3-CF3)
CH(Et)S(O)2CH2(D1-34a) CH2(D1-108b,Z=4-OCF3)
CH(Et)S(O)2CH2(D1-34a) CH2(D1-108b,Z=2-SCF3)
CH(Et)S(O)2CH2(D1-34a) CH2CH2CN
CH(Et)S(O)2CH2(D1-34a) CH2CH2CF3
CH(Et)S(O)2CH2(D1-34a) CH2CH2OMe
CH(Et)S(O)2CH2(D1-34a) CH2CH2SMe
CH(Et)S(O)2CH2(D1-34a) CH2CH2S(O)Me
CH(Et)S(O)2CH2(D1-34a) CH2CH2S(O)2Me
CH(Et)S(O)2CH2(D1-34a) D1-32a
CH(Et)S(O)2CH2(D1-34a) D1-33a
CH(Et)S(O)2CH2(D1-34a) D1-34a
CH(Et)S(O)2CH2(D1-34a) D1-37a
CH(Et)S(O)2CH2(D1-34a) D1-81a
CH(Et)S(O)2CH2(D1-34a) D1-82a
CH(Et)S(O)2CH2(D1-34a) D1-84a
CH(Et)S(O)2CH2(D1-34a) D1-85a
CH(Et)S(O)2CH2(D1-34a) D1-87a
CH(Et)S(O)2CH2(D1-34a) D1-92a
CH(Et)S(O)2CH2(D1-34a) D1-93a
CH(Et)S(O)2CH2(D1-34a) D1-95a
CH(Et)S(O)2CH2(D1-34a) D1-96a
CH(Et)S(O)2CH2(D1-34a) D1-98a
CH(Et)S(O)2CH2(D1-34a) D1-108a
CH(Et)S(O)2CH2(D1-34a) D1-108b(Z=2-Cl)
CH(Et)S(O)2CH2(D1-34a) D1-108b(Z=3-Me)
CH(Et)S(O)2CH2(D1-34a) D1-108b(Z=4-OMe)
CH(Et)S(O)2CH2(D1-34a) D1-108b(Z=2-SMe)
CH(Et)S(O)2CH2(D1-34a) D1-108b(Z=3-CF3)
CH(Et)S(O)2CH2(D1-34a) D1-108b(Z=4-OCF3)
CH(Et)S(O)2CH2(D1-34a) D1-108b(Z=2-SCF3)
CH(Et)S(O)2CH2(D1-34a) C(O)Me
CH(Et)S(O)2CH2(D1-34a) C(O)CF3
CH(Et)S(O)2CH2(D1-34a) C(O)OMe
CH2S{D1-32b(X1=5-CF3)} Me
CH2S{D1-32b(X1=5-CF3)} Et
CH2S{D1-32b(X1=5-CF3)} Pr-n
CH2S{D1-32b(X1=5-CF3)} Pr-i
CH2S{D1-32b(X1=5-CF3)} Pr-c
CH2S{D1-32b(X1=5-CF3)} Bu-n
CH2S{D1-32b(X1=5-CF3)} Bu-i
CH2S{D1-32b(X1=5-CF3)} Bu-c
CH2S{D1-32b(X1=5-CF3)} Bu-s
CH2S{D1-32b(X1=5-CF3)} Bu-t
CH2S{D1-32b(X1=5-CF3)} Pen-n
CH2S{D1-32b(X1=5-CF3)} Pen-c
CH2S{D1-32b(X1=5-CF3)} Hex-n
CH2S{D1-32b(X1=5-CF3)} Hex-c
CH2S{D1-32b(X1=5-CF3)} CH2Pr-c
CH2S{D1-32b(X1=5-CF3)} CH2Bu-c
CH2S{D1-32b(X1=5-CF3)} CH2Pen-c
CH2S{D1-32b(X1=5-CF3)} CH2Hex-c
CH2S{D1-32b(X1=5-CF3)} CH2CH=CH2
CH2S{D1-32b(X1=5-CF3)} CH2CH=C(Cl)2
CH2S{D1-32b(X1=5-CF3)} CH2C≡CH
CH2S{D1-32b(X1=5-CF3)} CH2CN
CH2S{D1-32b(X1=5-CF3)} CH2CF3
CH2S{D1-32b(X1=5-CF3)} CH2OMe
CH2S{D1-32b(X1=5-CF3)} CH2OCF3
CH2S{D1-32b(X1=5-CF3)} CH2SMe
CH2S{D1-32b(X1=5-CF3)} CH2S(O)Me
CH2S{D1-32b(X1=5-CF3)} CH2S(O)2Me
CH2S{D1-32b(X1=5-CF3)} CH2SCF3
CH2S{D1-32b(X1=5-CF3)} CH2S(O)CF3
CH2S{D1-32b(X1=5-CF3)} CH2S(O)2CF3
CH2S{D1-32b(X1=5-CF3)} CH2CH(OMe)2
CH2S{D1-32b(X1=5-CF3)} CH2CH(SMe)2
CH2S{D1-32b(X1=5-CF3)} CH2C(O)Me
CH2S{D1-32b(X1=5-CF3)} CH2C(O)CF3
CH2S{D1-32b(X1=5-CF3)} CH2C(O)OMe
CH2S{D1-32b(X1=5-CF3)} CH2(D1-32a)
CH2S{D1-32b(X1=5-CF3)} CH2(D1-33a)
CH2S{D1-32b(X1=5-CF3)} CH2(D1-34a)
CH2S{D1-32b(X1=5-CF3)} CH2(D1-37a)
CH2S{D1-32b(X1=5-CF3)} CH2(D1-81a)
CH2S{D1-32b(X1=5-CF3)} CH2(D1-82a)
CH2S{D1-32b(X1=5-CF3)} CH2(D1-84a)
CH2S{D1-32b(X1=5-CF3)} CH2(D1-85a)
CH2S{D1-32b(X1=5-CF3)} CH2(D1-87a)
CH2S{D1-32b(X1=5-CF3)} CH2(D1-92a)
CH2S{D1-32b(X1=5-CF3)} CH2(D1-93a)
CH2S{D1-32b(X1=5-CF3)} CH2(D1-95a)
CH2S{D1-32b(X1=5-CF3)} CH2(D1-96a)
CH2S{D1-32b(X1=5-CF3)} CH2(D1-98a)
CH2S{D1-32b(X1=5-CF3)} CH2(D1-108a)
CH2S{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-Cl)
CH2S{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=3-Me)
CH2S{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=4-OMe)
CH2S{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-SMe)
CH2S{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=3-CF3)
CH2S{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=4-OCF3)
CH2S{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-SCF3)
CH2S{D1-32b(X1=5-CF3)} CH2CH2CN
CH2S{D1-32b(X1=5-CF3)} CH2CH2CF3
CH2S{D1-32b(X1=5-CF3)} CH2CH2OMe
CH2S{D1-32b(X1=5-CF3)} CH2CH2SMe
CH2S{D1-32b(X1=5-CF3)} CH2CH2S(O)Me
CH2S{D1-32b(X1=5-CF3)} CH2CH2S(O)2Me
CH2S{D1-32b(X1=5-CF3)} D1-32a
CH2S{D1-32b(X1=5-CF3)} D1-33a
CH2S{D1-32b(X1=5-CF3)} D1-34a
CH2S{D1-32b(X1=5-CF3)} D1-37a
CH2S{D1-32b(X1=5-CF3)} D1-81a
CH2S{D1-32b(X1=5-CF3)} D1-82a
CH2S{D1-32b(X1=5-CF3)} D1-84a
CH2S{D1-32b(X1=5-CF3)} D1-85a
CH2S{D1-32b(X1=5-CF3)} D1-87a
CH2S{D1-32b(X1=5-CF3)} D1-92a
CH2S{D1-32b(X1=5-CF3)} D1-93a
CH2S{D1-32b(X1=5-CF3)} D1-95a
CH2S{D1-32b(X1=5-CF3)} D1-96a
CH2S{D1-32b(X1=5-CF3)} D1-98a
CH2S{D1-32b(X1=5-CF3)} D1-108a
CH2S{D1-32b(X1=5-CF3)} D1-108b(Z=2-Cl)
CH2S{D1-32b(X1=5-CF3)} D1-108b(Z=3-Me)
CH2S{D1-32b(X1=5-CF3)} D1-108b(Z=4-OMe)
CH2S{D1-32b(X1=5-CF3)} D1-108b(Z=2-SMe)
CH2S{D1-32b(X1=5-CF3)} D1-108b(Z=3-CF3)
CH2S{D1-32b(X1=5-CF3)} D1-108b(Z=4-OCF3)
CH2S{D1-32b(X1=5-CF3)} D1-108b(Z=2-SCF3)
CH2S{D1-32b(X1=5-CF3)} C(O)Me
CH2S{D1-32b(X1=5-CF3)} C(O)CF3
CH2S{D1-32b(X1=5-CF3)} C(O)OMe
CH2S(O){D1-32b(X1=5-CF3)} Me
CH2S(O){D1-32b(X1=5-CF3)} Et
CH2S(O){D1-32b(X1=5-CF3)} Pr-n
CH2S(O){D1-32b(X1=5-CF3)} Pr-i
CH2S(O){D1-32b(X1=5-CF3)} Pr-c
CH2S(O){D1-32b(X1=5-CF3)} Bu-n
CH2S(O){D1-32b(X1=5-CF3)} Bu-i
CH2S(O){D1-32b(X1=5-CF3)} Bu-c
CH2S(O){D1-32b(X1=5-CF3)} Bu-s
CH2S(O){D1-32b(X1=5-CF3)} Bu-t
CH2S(O){D1-32b(X1=5-CF3)} Pen-n
CH2S(O){D1-32b(X1=5-CF3)} Pen-c
CH2S(O){D1-32b(X1=5-CF3)} Hex-n
CH2S(O){D1-32b(X1=5-CF3)} Hex-c
CH2S(O){D1-32b(X1=5-CF3)} CH2Pr-c
CH2S(O){D1-32b(X1=5-CF3)} CH2Bu-c
CH2S(O){D1-32b(X1=5-CF3)} CH2Pen-c
CH2S(O){D1-32b(X1=5-CF3)} CH2Hex-c
CH2S(O){D1-32b(X1=5-CF3)} CH2CH=CH2
CH2S(O){D1-32b(X1=5-CF3)} CH2CH=C(Cl)2
CH2S(O){D1-32b(X1=5-CF3)} CH2C≡CH
CH2S(O){D1-32b(X1=5-CF3)} CH2CN
CH2S(O){D1-32b(X1=5-CF3)} CH2CF3
CH2S(O){D1-32b(X1=5-CF3)} CH2OMe
CH2S(O){D1-32b(X1=5-CF3)} CH2OCF3
CH2S(O){D1-32b(X1=5-CF3)} CH2SMe
CH2S(O){D1-32b(X1=5-CF3)} CH2S(O)Me
CH2S(O){D1-32b(X1=5-CF3)} CH2S(O)2Me
CH2S(O){D1-32b(X1=5-CF3)} CH2SCF3
CH2S(O){D1-32b(X1=5-CF3)} CH2S(O)CF3
CH2S(O){D1-32b(X1=5-CF3)} CH2S(O)2CF3
CH2S(O){D1-32b(X1=5-CF3)} CH2CH(OMe)2
CH2S(O){D1-32b(X1=5-CF3)} CH2CH(SMe)2
CH2S(O){D1-32b(X1=5-CF3)} CH2C(O)Me
CH2S(O){D1-32b(X1=5-CF3)} CH2C(O)CF3
CH2S(O){D1-32b(X1=5-CF3)} CH2C(O)OMe
CH2S(O){D1-32b(X1=5-CF3)} CH2(D1-32a)
CH2S(O){D1-32b(X1=5-CF3)} CH2(D1-33a)
CH2S(O){D1-32b(X1=5-CF3)} CH2(D1-34a)
CH2S(O){D1-32b(X1=5-CF3)} CH2(D1-37a)
CH2S(O){D1-32b(X1=5-CF3)} CH2(D1-81a)
CH2S(O){D1-32b(X1=5-CF3)} CH2(D1-82a)
CH2S(O){D1-32b(X1=5-CF3)} CH2(D1-84a)
CH2S(O){D1-32b(X1=5-CF3)} CH2(D1-85a)
CH2S(O){D1-32b(X1=5-CF3)} CH2(D1-87a)
CH2S(O){D1-32b(X1=5-CF3)} CH2(D1-92a)
CH2S(O){D1-32b(X1=5-CF3)} CH2(D1-93a)
CH2S(O){D1-32b(X1=5-CF3)} CH2(D1-95a)
CH2S(O){D1-32b(X1=5-CF3)} CH2(D1-96a)
CH2S(O){D1-32b(X1=5-CF3)} CH2(D1-98a)
CH2S(O){D1-32b(X1=5-CF3)} CH2(D1-108a)
CH2S(O){D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-Cl)
CH2S(O){D1-32b(X1=5-CF3)} CH2(D1-108b,Z=3-Me)
CH2S(O){D1-32b(X1=5-CF3)} CH2(D1-108b,Z=4-OMe)
CH2S(O){D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-SMe)
CH2S(O){D1-32b(X1=5-CF3)} CH2(D1-108b,Z=3-CF3)
CH2S(O){D1-32b(X1=5-CF3)} CH2(D1-108b,Z=4-OCF3)
CH2S(O){D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-SCF3)
CH2S(O){D1-32b(X1=5-CF3)} CH2CH2CN
CH2S(O){D1-32b(X1=5-CF3)} CH2CH2CF3
CH2S(O){D1-32b(X1=5-CF3)} CH2CH2OMe
CH2S(O){D1-32b(X1=5-CF3)} CH2CH2SMe
CH2S(O){D1-32b(X1=5-CF3)} CH2CH2S(O)Me
CH2S(O){D1-32b(X1=5-CF3)} CH2CH2S(O)2Me
CH2S(O){D1-32b(X1=5-CF3)} D1-32a
CH2S(O){D1-32b(X1=5-CF3)} D1-33a
CH2S(O){D1-32b(X1=5-CF3)} D1-34a
CH2S(O){D1-32b(X1=5-CF3)} D1-37a
CH2S(O){D1-32b(X1=5-CF3)} D1-81a
CH2S(O){D1-32b(X1=5-CF3)} D1-82a
CH2S(O){D1-32b(X1=5-CF3)} D1-84a
CH2S(O){D1-32b(X1=5-CF3)} D1-85a
CH2S(O){D1-32b(X1=5-CF3)} D1-87a
CH2S(O){D1-32b(X1=5-CF3)} D1-92a
CH2S(O){D1-32b(X1=5-CF3)} D1-93a
CH2S(O){D1-32b(X1=5-CF3)} D1-95a
CH2S(O){D1-32b(X1=5-CF3)} D1-96a
CH2S(O){D1-32b(X1=5-CF3)} D1-98a
CH2S(O){D1-32b(X1=5-CF3)} D1-108a
CH2S(O){D1-32b(X1=5-CF3)} D1-108b(Z=2-Cl)
CH2S(O){D1-32b(X1=5-CF3)} D1-108b(Z=3-Me)
CH2S(O){D1-32b(X1=5-CF3)} D1-108b(Z=4-OMe)
CH2S(O){D1-32b(X1=5-CF3)} D1-108b(Z=2-SMe)
CH2S(O){D1-32b(X1=5-CF3)} D1-108b(Z=3-CF3)
CH2S(O){D1-32b(X1=5-CF3)} D1-108b(Z=4-OCF3)
CH2S(O){D1-32b(X1=5-CF3)} D1-108b(Z=2-SCF3)
CH2S(O){D1-32b(X1=5-CF3)} C(O)Me
CH2S(O){D1-32b(X1=5-CF3)} C(O)CF3
CH2S(O){D1-32b(X1=5-CF3)} C(O)OMe
CH2S(O)2{D1-32b(X1=5-CF3)} Me
CH2S(O)2{D1-32b(X1=5-CF3)} Et
CH2S(O)2{D1-32b(X1=5-CF3)} Pr-n
CH2S(O)2{D1-32b(X1=5-CF3)} Pr-i
CH2S(O)2{D1-32b(X1=5-CF3)} Pr-c
CH2S(O)2{D1-32b(X1=5-CF3)} Bu-n
CH2S(O)2{D1-32b(X1=5-CF3)} Bu-i
CH2S(O)2{D1-32b(X1=5-CF3)} Bu-c
CH2S(O)2{D1-32b(X1=5-CF3)} Bu-s
CH2S(O)2{D1-32b(X1=5-CF3)} Bu-t
CH2S(O)2{D1-32b(X1=5-CF3)} Pen-n
CH2S(O)2{D1-32b(X1=5-CF3)} Pen-c
CH2S(O)2{D1-32b(X1=5-CF3)} Hex-n
CH2S(O)2{D1-32b(X1=5-CF3)} Hex-c
CH2S(O)2{D1-32b(X1=5-CF3)} CH2Pr-c
CH2S(O)2{D1-32b(X1=5-CF3)} CH2Bu-c
CH2S(O)2{D1-32b(X1=5-CF3)} CH2Pen-c
CH2S(O)2{D1-32b(X1=5-CF3)} CH2Hex-c
CH2S(O)2{D1-32b(X1=5-CF3)} CH2CH=CH2
CH2S(O)2{D1-32b(X1=5-CF3)} CH2CH=C(Cl)2
CH2S(O)2{D1-32b(X1=5-CF3)} CH2C≡CH
CH2S(O)2{D1-32b(X1=5-CF3)} CH2CN
CH2S(O)2{D1-32b(X1=5-CF3)} CH2CF3
CH2S(O)2{D1-32b(X1=5-CF3)} CH2OMe
CH2S(O)2{D1-32b(X1=5-CF3)} CH2OCF3
CH2S(O)2{D1-32b(X1=5-CF3)} CH2SMe
CH2S(O)2{D1-32b(X1=5-CF3)} CH2S(O)Me
CH2S(O)2{D1-32b(X1=5-CF3)} CH2S(O)2Me
CH2S(O)2{D1-32b(X1=5-CF3)} CH2SCF3
CH2S(O)2{D1-32b(X1=5-CF3)} CH2S(O)CF3
CH2S(O)2{D1-32b(X1=5-CF3)} CH2S(O)2CF3
CH2S(O)2{D1-32b(X1=5-CF3)} CH2CH(OMe)2
CH2S(O)2{D1-32b(X1=5-CF3)} CH2CH(SMe)2
CH2S(O)2{D1-32b(X1=5-CF3)} CH2C(O)Me
CH2S(O)2{D1-32b(X1=5-CF3)} CH2C(O)CF3
CH2S(O)2{D1-32b(X1=5-CF3)} CH2C(O)OMe
CH2S(O)2{D1-32b(X1=5-CF3)} CH2(D1-32a)
CH2S(O)2{D1-32b(X1=5-CF3)} CH2(D1-33a)
CH2S(O)2{D1-32b(X1=5-CF3)} CH2(D1-34a)
CH2S(O)2{D1-32b(X1=5-CF3)} CH2(D1-37a)
CH2S(O)2{D1-32b(X1=5-CF3)} CH2(D1-81a)
CH2S(O)2{D1-32b(X1=5-CF3)} CH2(D1-82a)
CH2S(O)2{D1-32b(X1=5-CF3)} CH2(D1-84a)
CH2S(O)2{D1-32b(X1=5-CF3)} CH2(D1-85a)
CH2S(O)2{D1-32b(X1=5-CF3)} CH2(D1-87a)
CH2S(O)2{D1-32b(X1=5-CF3)} CH2(D1-92a)
CH2S(O)2{D1-32b(X1=5-CF3)} CH2(D1-93a)
CH2S(O)2{D1-32b(X1=5-CF3)} CH2(D1-95a)
CH2S(O)2{D1-32b(X1=5-CF3)} CH2(D1-96a)
CH2S(O)2{D1-32b(X1=5-CF3)} CH2(D1-98a)
CH2S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108a)
CH2S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-Cl)
CH2S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=3-Me)
CH2S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=4-OMe)
CH2S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-SMe)
CH2S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=3-CF3)
CH2S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=4-OCF3)
CH2S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-SCF3)
CH2S(O)2{D1-32b(X1=5-CF3)} CH2CH2CN
CH2S(O)2{D1-32b(X1=5-CF3)} CH2CH2CF3
CH2S(O)2{D1-32b(X1=5-CF3)} CH2CH2OMe
CH2S(O)2{D1-32b(X1=5-CF3)} CH2CH2SMe
CH2S(O)2{D1-32b(X1=5-CF3)} CH2CH2S(O)Me
CH2S(O)2{D1-32b(X1=5-CF3)} CH2CH2S(O)2Me
CH2S(O)2{D1-32b(X1=5-CF3)} D1-32a
CH2S(O)2{D1-32b(X1=5-CF3)} D1-33a
CH2S(O)2{D1-32b(X1=5-CF3)} D1-34a
CH2S(O)2{D1-32b(X1=5-CF3)} D1-37a
CH2S(O)2{D1-32b(X1=5-CF3)} D1-81a
CH2S(O)2{D1-32b(X1=5-CF3)} D1-82a
CH2S(O)2{D1-32b(X1=5-CF3)} D1-84a
CH2S(O)2{D1-32b(X1=5-CF3)} D1-85a
CH2S(O)2{D1-32b(X1=5-CF3)} D1-87a
CH2S(O)2{D1-32b(X1=5-CF3)} D1-92a
CH2S(O)2{D1-32b(X1=5-CF3)} D1-93a
CH2S(O)2{D1-32b(X1=5-CF3)} D1-95a
CH2S(O)2{D1-32b(X1=5-CF3)} D1-96a
CH2S(O)2{D1-32b(X1=5-CF3)} D1-98a
CH2S(O)2{D1-32b(X1=5-CF3)} D1-108a
CH2S(O)2{D1-32b(X1=5-CF3)} D1-108b(Z=2-Cl)
CH2S(O)2{D1-32b(X1=5-CF3)} D1-108b(Z=3-Me)
CH2S(O)2{D1-32b(X1=5-CF3)} D1-108b(Z=4-OMe)
CH2S(O)2{D1-32b(X1=5-CF3)} D1-108b(Z=2-SMe)
CH2S(O)2{D1-32b(X1=5-CF3)} D1-108b(Z=3-CF3)
CH2S(O)2{D1-32b(X1=5-CF3)} D1-108b(Z=4-OCF3)
CH2S(O)2{D1-32b(X1=5-CF3)} D1-108b(Z=2-SCF3)
CH2S(O)2{D1-32b(X1=5-CF3)} C(O)Me
CH2S(O)2{D1-32b(X1=5-CF3)} C(O)CF3
CH2S(O)2{D1-32b(X1=5-CF3)} C(O)OMe
CH(Me)S{D1-32b(X1=5-CF3)} Me
CH(Me)S{D1-32b(X1=5-CF3)} Et
CH(Me)S{D1-32b(X1=5-CF3)} Pr-n
CH(Me)S{D1-32b(X1=5-CF3)} Pr-i
CH(Me)S{D1-32b(X1=5-CF3)} Pr-c
CH(Me)S{D1-32b(X1=5-CF3)} Bu-n
CH(Me)S{D1-32b(X1=5-CF3)} Bu-i
CH(Me)S{D1-32b(X1=5-CF3)} Bu-c
CH(Me)S{D1-32b(X1=5-CF3)} Bu-s
CH(Me)S{D1-32b(X1=5-CF3)} Bu-t
CH(Me)S{D1-32b(X1=5-CF3)} Pen-n
CH(Me)S{D1-32b(X1=5-CF3)} Pen-c
CH(Me)S{D1-32b(X1=5-CF3)} Hex-n
CH(Me)S{D1-32b(X1=5-CF3)} Hex-c
CH(Me)S{D1-32b(X1=5-CF3)} CH2Pr-c
CH(Me)S{D1-32b(X1=5-CF3)} CH2Bu-c
CH(Me)S{D1-32b(X1=5-CF3)} CH2Pen-c
CH(Me)S{D1-32b(X1=5-CF3)} CH2Hex-c
CH(Me)S{D1-32b(X1=5-CF3)} CH2CH=CH2
CH(Me)S{D1-32b(X1=5-CF3)} CH2CH=C(Cl)2
CH(Me)S{D1-32b(X1=5-CF3)} CH2C≡CH
CH(Me)S{D1-32b(X1=5-CF3)} CH2CN
CH(Me)S{D1-32b(X1=5-CF3)} CH2CF3
CH(Me)S{D1-32b(X1=5-CF3)} CH2OMe
CH(Me)S{D1-32b(X1=5-CF3)} CH2OCF3
CH(Me)S{D1-32b(X1=5-CF3)} CH2SMe
CH(Me)S{D1-32b(X1=5-CF3)} CH2S(O)Me
CH(Me)S{D1-32b(X1=5-CF3)} CH2S(O)2Me
CH(Me)S{D1-32b(X1=5-CF3)} CH2SCF3
CH(Me)S{D1-32b(X1=5-CF3)} CH2S(O)CF3
CH(Me)S{D1-32b(X1=5-CF3)} CH2S(O)2CF3
CH(Me)S{D1-32b(X1=5-CF3)} CH2CH(OMe)2
CH(Me)S{D1-32b(X1=5-CF3)} CH2CH(SMe)2
CH(Me)S{D1-32b(X1=5-CF3)} CH2C(O)Me
CH(Me)S{D1-32b(X1=5-CF3)} CH2C(O)CF3
CH(Me)S{D1-32b(X1=5-CF3)} CH2C(O)OMe
CH(Me)S{D1-32b(X1=5-CF3)} CH2(D1-32a)
CH(Me)S{D1-32b(X1=5-CF3)} CH2(D1-33a)
CH(Me)S{D1-32b(X1=5-CF3)} CH2(D1-34a)
CH(Me)S{D1-32b(X1=5-CF3)} CH2(D1-37a)
CH(Me)S{D1-32b(X1=5-CF3)} CH2(D1-81a)
CH(Me)S{D1-32b(X1=5-CF3)} CH2(D1-82a)
CH(Me)S{D1-32b(X1=5-CF3)} CH2(D1-84a)
CH(Me)S{D1-32b(X1=5-CF3)} CH2(D1-85a)
CH(Me)S{D1-32b(X1=5-CF3)} CH2(D1-87a)
CH(Me)S{D1-32b(X1=5-CF3)} CH2(D1-92a)
CH(Me)S{D1-32b(X1=5-CF3)} CH2(D1-93a)
CH(Me)S{D1-32b(X1=5-CF3)} CH2(D1-95a)
CH(Me)S{D1-32b(X1=5-CF3)} CH2(D1-96a)
CH(Me)S{D1-32b(X1=5-CF3)} CH2(D1-98a)
CH(Me)S{D1-32b(X1=5-CF3)} CH2(D1-108a)
CH(Me)S{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-Cl)
CH(Me)S{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=3-Me)
CH(Me)S{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=4-OMe)
CH(Me)S{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-SMe)
CH(Me)S{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=3-CF3)
CH(Me)S{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=4-OCF3)
CH(Me)S{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-SCF3)
CH(Me)S{D1-32b(X1=5-CF3)} CH2CH2CN
CH(Me)S{D1-32b(X1=5-CF3)} CH2CH2CF3
CH(Me)S{D1-32b(X1=5-CF3)} CH2CH2OMe
CH(Me)S{D1-32b(X1=5-CF3)} CH2CH2SMe
CH(Me)S{D1-32b(X1=5-CF3)} CH2CH2S(O)Me
CH(Me)S{D1-32b(X1=5-CF3)} CH2CH2S(O)2Me
CH(Me)S{D1-32b(X1=5-CF3)} D1-32a
CH(Me)S{D1-32b(X1=5-CF3)} D1-33a
CH(Me)S{D1-32b(X1=5-CF3)} D1-34a
CH(Me)S{D1-32b(X1=5-CF3)} D1-37a
CH(Me)S{D1-32b(X1=5-CF3)} D1-81a
CH(Me)S{D1-32b(X1=5-CF3)} D1-82a
CH(Me)S{D1-32b(X1=5-CF3)} D1-84a
CH(Me)S{D1-32b(X1=5-CF3)} D1-85a
CH(Me)S{D1-32b(X1=5-CF3)} D1-87a
CH(Me)S{D1-32b(X1=5-CF3)} D1-92a
CH(Me)S{D1-32b(X1=5-CF3)} D1-93a
CH(Me)S{D1-32b(X1=5-CF3)} D1-95a
CH(Me)S{D1-32b(X1=5-CF3)} D1-96a
CH(Me)S{D1-32b(X1=5-CF3)} D1-98a
CH(Me)S{D1-32b(X1=5-CF3)} D1-108a
CH(Me)S{D1-32b(X1=5-CF3)} D1-108b(Z=2-Cl)
CH(Me)S{D1-32b(X1=5-CF3)} D1-108b(Z=3-Me)
CH(Me)S{D1-32b(X1=5-CF3)} D1-108b(Z=4-OMe)
CH(Me)S{D1-32b(X1=5-CF3)} D1-108b(Z=2-SMe)
CH(Me)S{D1-32b(X1=5-CF3)} D1-108b(Z=3-CF3)
CH(Me)S{D1-32b(X1=5-CF3)} D1-108b(Z=4-OCF3)
CH(Me)S{D1-32b(X1=5-CF3)} D1-108b(Z=2-SCF3)
CH(Me)S{D1-32b(X1=5-CF3)} C(O)Me
CH(Me)S{D1-32b(X1=5-CF3)} C(O)CF3
CH(Me)S{D1-32b(X1=5-CF3)} C(O)OMe
CH(Me)S(O){D1-32b(X1=5-CF3)} Me
CH(Me)S(O){D1-32b(X1=5-CF3)} Et
CH(Me)S(O){D1-32b(X1=5-CF3)} Pr-n
CH(Me)S(O){D1-32b(X1=5-CF3)} Pr-i
CH(Me)S(O){D1-32b(X1=5-CF3)} Pr-c
CH(Me)S(O){D1-32b(X1=5-CF3)} Bu-n
CH(Me)S(O){D1-32b(X1=5-CF3)} Bu-i
CH(Me)S(O){D1-32b(X1=5-CF3)} Bu-c
CH(Me)S(O){D1-32b(X1=5-CF3)} Bu-s
CH(Me)S(O){D1-32b(X1=5-CF3)} Bu-t
CH(Me)S(O){D1-32b(X1=5-CF3)} Pen-n
CH(Me)S(O){D1-32b(X1=5-CF3)} Pen-c
CH(Me)S(O){D1-32b(X1=5-CF3)} Hex-n
CH(Me)S(O){D1-32b(X1=5-CF3)} Hex-c
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2Pr-c
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2Bu-c
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2Pen-c
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2Hex-c
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2CH=CH2
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2CH=C(Cl)2
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2C≡CH
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2CN
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2CF3
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2OMe
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2OCF3
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2SMe
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2S(O)Me
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2S(O)2Me
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2SCF3
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2S(O)CF3
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2S(O)2CF3
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2CH(OMe)2
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2CH(SMe)2
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2C(O)Me
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2C(O)CF3
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2C(O)OMe
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2(D1-32a)
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2(D1-33a)
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2(D1-34a)
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2(D1-37a)
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2(D1-81a)
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2(D1-82a)
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2(D1-84a)
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2(D1-85a)
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2(D1-87a)
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2(D1-92a)
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2(D1-93a)
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2(D1-95a)
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2(D1-96a)
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2(D1-98a)
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2(D1-108a)
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-Cl)
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2(D1-108b,Z=3-Me)
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2(D1-108b,Z=4-OMe)
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-SMe)
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2(D1-108b,Z=3-CF3)
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2CH2CN
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2CH2CF3
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2CH2OMe
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2CH2SMe
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2CH2S(O)Me
CH(Me)S(O){D1-32b(X1=5-CF3)} CH2CH2S(O)2Me
CH(Me)S(O){D1-32b(X1=5-CF3)} D1-32a
CH(Me)S(O){D1-32b(X1=5-CF3)} D1-33a
CH(Me)S(O){D1-32b(X1=5-CF3)} D1-34a
CH(Me)S(O){D1-32b(X1=5-CF3)} D1-37a
CH(Me)S(O){D1-32b(X1=5-CF3)} D1-81a
CH(Me)S(O){D1-32b(X1=5-CF3)} D1-82a
CH(Me)S(O){D1-32b(X1=5-CF3)} D1-84a
CH(Me)S(O){D1-32b(X1=5-CF3)} D1-85a
CH(Me)S(O){D1-32b(X1=5-CF3)} D1-87a
CH(Me)S(O){D1-32b(X1=5-CF3)} D1-92a
CH(Me)S(O){D1-32b(X1=5-CF3)} D1-93a
CH(Me)S(O){D1-32b(X1=5-CF3)} D1-95a
CH(Me)S(O){D1-32b(X1=5-CF3)} D1-96a
CH(Me)S(O){D1-32b(X1=5-CF3)} D1-98a
CH(Me)S(O){D1-32b(X1=5-CF3)} D1-108a
CH(Me)S(O){D1-32b(X1=5-CF3)} D1-108b(Z=2-Cl)
CH(Me)S(O){D1-32b(X1=5-CF3)} D1-108b(Z=3-Me)
CH(Me)S(O){D1-32b(X1=5-CF3)} D1-108b(Z=4-OMe)
CH(Me)S(O){D1-32b(X1=5-CF3)} D1-108b(Z=2-SMe)
CH(Me)S(O){D1-32b(X1=5-CF3)} D1-108b(Z=3-CF3)
CH(Me)S(O){D1-32b(X1=5-CF3)} D1-108b(Z=4-OCF3)
CH(Me)S(O){D1-32b(X1=5-CF3)} D1-108b(Z=2-SCF3)
CH(Me)S(O){D1-32b(X1=5-CF3)} C(O)Me
CH(Me)S(O){D1-32b(X1=5-CF3)} C(O)CF3
CH(Me)S(O){D1-32b(X1=5-CF3)} C(O)OMe
CH(Me)S(O)2{D1-32b(X1=5-CF3)} Me
CH(Me)S(O)2{D1-32b(X1=5-CF3)} Et
CH(Me)S(O)2{D1-32b(X1=5-CF3)} Pr-n
CH(Me)S(O)2{D1-32b(X1=5-CF3)} Pr-i
CH(Me)S(O)2{D1-32b(X1=5-CF3)} Pr-c
CH(Me)S(O)2{D1-32b(X1=5-CF3)} Bu-n
CH(Me)S(O)2{D1-32b(X1=5-CF3)} Bu-i
CH(Me)S(O)2{D1-32b(X1=5-CF3)} Bu-c
CH(Me)S(O)2{D1-32b(X1=5-CF3)} Bu-s
CH(Me)S(O)2{D1-32b(X1=5-CF3)} Bu-t
CH(Me)S(O)2{D1-32b(X1=5-CF3)} Pen-n
CH(Me)S(O)2{D1-32b(X1=5-CF3)} Pen-c
CH(Me)S(O)2{D1-32b(X1=5-CF3)} Hex-n
CH(Me)S(O)2{D1-32b(X1=5-CF3)} Hex-c
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2Pr-c
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2Bu-c
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2Pen-c
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2Hex-c
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2CH=CH2
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2CH=C(Cl)2
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2C≡CH
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2CN
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2CF3
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2OMe
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2OCF3
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2SMe
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2S(O)Me
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2S(O)2Me
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2SCF3
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2S(O)CF3
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2S(O)2CF3
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2CH(OMe)2
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2CH(SMe)2
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2C(O)Me
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2C(O)CF3
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2C(O)OMe
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-32a)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-33a)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-34a)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-37a)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-81a)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-82a)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-84a)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-85a)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-87a)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-92a)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-93a)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-95a)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-96a)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-98a)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108a)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=3-Me)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2CH2CN
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2CH2CF3
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2CH2OMe
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2CH2SMe
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2CH2S(O)Me
CH(Me)S(O)2{D1-32b(X1=5-CF3)} CH2CH2S(O)2Me
CH(Me)S(O)2{D1-32b(X1=5-CF3)} D1-32a
CH(Me)S(O)2{D1-32b(X1=5-CF3)} D1-33a
CH(Me)S(O)2{D1-32b(X1=5-CF3)} D1-34a
CH(Me)S(O)2{D1-32b(X1=5-CF3)} D1-37a
CH(Me)S(O)2{D1-32b(X1=5-CF3)} D1-81a
CH(Me)S(O)2{D1-32b(X1=5-CF3)} D1-82a
CH(Me)S(O)2{D1-32b(X1=5-CF3)} D1-84a
CH(Me)S(O)2{D1-32b(X1=5-CF3)} D1-85a
CH(Me)S(O)2{D1-32b(X1=5-CF3)} D1-87a
CH(Me)S(O)2{D1-32b(X1=5-CF3)} D1-92a
CH(Me)S(O)2{D1-32b(X1=5-CF3)} D1-93a
CH(Me)S(O)2{D1-32b(X1=5-CF3)} D1-95a
CH(Me)S(O)2{D1-32b(X1=5-CF3)} D1-96a
CH(Me)S(O)2{D1-32b(X1=5-CF3)} D1-98a
CH(Me)S(O)2{D1-32b(X1=5-CF3)} D1-108a
CH(Me)S(O)2{D1-32b(X1=5-CF3)} D1-108b(Z=2-Cl)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} D1-108b(Z=3-Me)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} D1-108b(Z=4-OMe)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} D1-108b(Z=2-SMe)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} D1-108b(Z=3-CF3)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} D1-108b(Z=4-OCF3)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} D1-108b(Z=2-SCF3)
CH(Me)S(O)2{D1-32b(X1=5-CF3)} C(O)Me
CH(Me)S(O)2{D1-32b(X1=5-CF3)} C(O)CF3
CH(Me)S(O)2{D1-32b(X1=5-CF3)} C(O)OMe
CH(Et)S{D1-32b(X1=5-CF3)} Me
CH(Et)S{D1-32b(X1=5-CF3)} Et
CH(Et)S{D1-32b(X1=5-CF3)} Pr-n
CH(Et)S{D1-32b(X1=5-CF3)} Pr-i
CH(Et)S{D1-32b(X1=5-CF3)} Pr-c
CH(Et)S{D1-32b(X1=5-CF3)} Bu-n
CH(Et)S{D1-32b(X1=5-CF3)} Bu-i
CH(Et)S{D1-32b(X1=5-CF3)} Bu-c
CH(Et)S{D1-32b(X1=5-CF3)} Bu-s
CH(Et)S{D1-32b(X1=5-CF3)} Bu-t
CH(Et)S{D1-32b(X1=5-CF3)} Pen-n
CH(Et)S{D1-32b(X1=5-CF3)} Pen-c
CH(Et)S{D1-32b(X1=5-CF3)} Hex-n
CH(Et)S{D1-32b(X1=5-CF3)} Hex-c
CH(Et)S{D1-32b(X1=5-CF3)} CH2Pr-c
CH(Et)S{D1-32b(X1=5-CF3)} CH2Bu-c
CH(Et)S{D1-32b(X1=5-CF3)} CH2Pen-c
CH(Et)S{D1-32b(X1=5-CF3)} CH2Hex-c
CH(Et)S{D1-32b(X1=5-CF3)} CH2CH=CH2
CH(Et)S{D1-32b(X1=5-CF3)} CH2CH=C(Cl)2
CH(Et)S{D1-32b(X1=5-CF3)} CH2C≡CH
CH(Et)S{D1-32b(X1=5-CF3)} CH2CN
CH(Et)S{D1-32b(X1=5-CF3)} CH2CF3
CH(Et)S{D1-32b(X1=5-CF3)} CH2OMe
CH(Et)S{D1-32b(X1=5-CF3)} CH2OCF3
CH(Et)S{D1-32b(X1=5-CF3)} CH2SMe
CH(Et)S{D1-32b(X1=5-CF3)} CH2S(O)Me
CH(Et)S{D1-32b(X1=5-CF3)} CH2S(O)2Me
CH(Et)S{D1-32b(X1=5-CF3)} CH2SCF3
CH(Et)S{D1-32b(X1=5-CF3)} CH2S(O)CF3
CH(Et)S{D1-32b(X1=5-CF3)} CH2S(O)2CF3
CH(Et)S{D1-32b(X1=5-CF3)} CH2CH(OMe)2
CH(Et)S{D1-32b(X1=5-CF3)} CH2CH(SMe)2
CH(Et)S{D1-32b(X1=5-CF3)} CH2C(O)Me
CH(Et)S{D1-32b(X1=5-CF3)} CH2C(O)CF3
CH(Et)S{D1-32b(X1=5-CF3)} CH2C(O)OMe
CH(Et)S{D1-32b(X1=5-CF3)} CH2(D1-32a)
CH(Et)S{D1-32b(X1=5-CF3)} CH2(D1-33a)
CH(Et)S{D1-32b(X1=5-CF3)} CH2(D1-34a)
CH(Et)S{D1-32b(X1=5-CF3)} CH2(D1-37a)
CH(Et)S{D1-32b(X1=5-CF3)} CH2(D1-81a)
CH(Et)S{D1-32b(X1=5-CF3)} CH2(D1-82a)
CH(Et)S{D1-32b(X1=5-CF3)} CH2(D1-84a)
CH(Et)S{D1-32b(X1=5-CF3)} CH2(D1-85a)
CH(Et)S{D1-32b(X1=5-CF3)} CH2(D1-87a)
CH(Et)S{D1-32b(X1=5-CF3)} CH2(D1-92a)
CH(Et)S{D1-32b(X1=5-CF3)} CH2(D1-93a)
CH(Et)S{D1-32b(X1=5-CF3)} CH2(D1-95a)
CH(Et)S{D1-32b(X1=5-CF3)} CH2(D1-96a)
CH(Et)S{D1-32b(X1=5-CF3)} CH2(D1-98a)
CH(Et)S{D1-32b(X1=5-CF3)} CH2(D1-108a)
CH(Et)S{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-Cl)
CH(Et)S{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=3-Me)
CH(Et)S{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=4-OMe)
CH(Et)S{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-SMe)
CH(Et)S{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=3-CF3)
CH(Et)S{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=4-OCF3)
CH(Et)S{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-SCF3)
CH(Et)S{D1-32b(X1=5-CF3)} CH2CH2CN
CH(Et)S{D1-32b(X1=5-CF3)} CH2CH2CF3
CH(Et)S{D1-32b(X1=5-CF3)} CH2CH2OMe
CH(Et)S{D1-32b(X1=5-CF3)} CH2CH2SMe
CH(Et)S{D1-32b(X1=5-CF3)} CH2CH2S(O)Me
CH(Et)S{D1-32b(X1=5-CF3)} CH2CH2S(O)2Me
CH(Et)S{D1-32b(X1=5-CF3)} D1-32a
CH(Et)S{D1-32b(X1=5-CF3)} D1-33a
CH(Et)S{D1-32b(X1=5-CF3)} D1-34a
CH(Et)S{D1-32b(X1=5-CF3)} D1-37a
CH(Et)S{D1-32b(X1=5-CF3)} D1-81a
CH(Et)S{D1-32b(X1=5-CF3)} D1-82a
CH(Et)S{D1-32b(X1=5-CF3)} D1-84a
CH(Et)S{D1-32b(X1=5-CF3)} D1-85a
CH(Et)S{D1-32b(X1=5-CF3)} D1-87a
CH(Et)S{D1-32b(X1=5-CF3)} D1-92a
CH(Et)S{D1-32b(X1=5-CF3)} D1-93a
CH(Et)S{D1-32b(X1=5-CF3)} D1-95a
CH(Et)S{D1-32b(X1=5-CF3)} D1-96a
CH(Et)S{D1-32b(X1=5-CF3)} D1-98a
CH(Et)S{D1-32b(X1=5-CF3)} D1-108a
CH(Et)S{D1-32b(X1=5-CF3)} D1-108b(Z=2-Cl)
CH(Et)S{D1-32b(X1=5-CF3)} D1-108b(Z=3-Me)
CH(Et)S{D1-32b(X1=5-CF3)} D1-108b(Z=4-OMe)
CH(Et)S{D1-32b(X1=5-CF3)} D1-108b(Z=2-SMe)
CH(Et)S{D1-32b(X1=5-CF3)} D1-108b(Z=3-CF3)
CH(Et)S{D1-32b(X1=5-CF3)} D1-108b(Z=4-OCF3)
CH(Et)S{D1-32b(X1=5-CF3)} D1-108b(Z=2-SCF3)
CH(Et)S{D1-32b(X1=5-CF3)} C(O)Me
CH(Et)S{D1-32b(X1=5-CF3)} C(O)CF3
CH(Et)S{D1-32b(X1=5-CF3)} C(O)OMe
CH(Et)S(O){D1-32b(X1=5-CF3)} Me
CH(Et)S(O){D1-32b(X1=5-CF3)} Et
CH(Et)S(O){D1-32b(X1=5-CF3)} Pr-n
CH(Et)S(O){D1-32b(X1=5-CF3)} Pr-i
CH(Et)S(O){D1-32b(X1=5-CF3)} Pr-c
CH(Et)S(O){D1-32b(X1=5-CF3)} Bu-n
CH(Et)S(O){D1-32b(X1=5-CF3)} Bu-i
CH(Et)S(O){D1-32b(X1=5-CF3)} Bu-c
CH(Et)S(O){D1-32b(X1=5-CF3)} Bu-s
CH(Et)S(O){D1-32b(X1=5-CF3)} Bu-t
CH(Et)S(O){D1-32b(X1=5-CF3)} Pen-n
CH(Et)S(O){D1-32b(X1=5-CF3)} Pen-c
CH(Et)S(O){D1-32b(X1=5-CF3)} Hex-n
CH(Et)S(O){D1-32b(X1=5-CF3)} Hex-c
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2Pr-c
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2Bu-c
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2Pen-c
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2Hex-c
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2CH=CH2
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2CH=C(Cl)2
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2C≡CH
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2CN
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2CF3
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2OMe
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2OCF3
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2SMe
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2S(O)Me
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2S(O)2Me
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2SCF3
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2S(O)CF3
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2S(O)2CF3
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2CH(OMe)2
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2CH(SMe)2
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2C(O)Me
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2C(O)CF3
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2C(O)OMe
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2(D1-32a)
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2(D1-33a)
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2(D1-34a)
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2(D1-37a)
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2(D1-81a)
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2(D1-82a)
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2(D1-84a)
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2(D1-85a)
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2(D1-87a)
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2(D1-92a)
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2(D1-93a)
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2(D1-95a)
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2(D1-96a)
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2(D1-98a)
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2(D1-108a)
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-Cl)
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2(D1-108b,Z=3-Me)
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2(D1-108b,Z=4-OMe)
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-SMe)
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2(D1-108b,Z=3-CF3)
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2(D1-108b,Z=4-OCF3)
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-SCF3)
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2CH2CN
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2CH2CF3
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2CH2OMe
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2CH2SMe
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2CH2S(O)Me
CH(Et)S(O){D1-32b(X1=5-CF3)} CH2CH2S(O)2Me
CH(Et)S(O){D1-32b(X1=5-CF3)} D1-32a
CH(Et)S(O){D1-32b(X1=5-CF3)} D1-33a
CH(Et)S(O){D1-32b(X1=5-CF3)} D1-34a
CH(Et)S(O){D1-32b(X1=5-CF3)} D1-37a
CH(Et)S(O){D1-32b(X1=5-CF3)} D1-81a
CH(Et)S(O){D1-32b(X1=5-CF3)} D1-82a
CH(Et)S(O){D1-32b(X1=5-CF3)} D1-84a
CH(Et)S(O){D1-32b(X1=5-CF3)} D1-85a
CH(Et)S(O){D1-32b(X1=5-CF3)} D1-87a
CH(Et)S(O){D1-32b(X1=5-CF3)} D1-92a
CH(Et)S(O){D1-32b(X1=5-CF3)} D1-93a
CH(Et)S(O){D1-32b(X1=5-CF3)} D1-95a
CH(Et)S(O){D1-32b(X1=5-CF3)} D1-96a
CH(Et)S(O){D1-32b(X1=5-CF3)} D1-98a
CH(Et)S(O){D1-32b(X1=5-CF3)} D1-108a
CH(Et)S(O){D1-32b(X1=5-CF3)} D1-108b(Z=2-Cl)
CH(Et)S(O){D1-32b(X1=5-CF3)} D1-108b(Z=3-Me)
CH(Et)S(O){D1-32b(X1=5-CF3)} D1-108b(Z=4-OMe)
CH(Et)S(O){D1-32b(X1=5-CF3)} D1-108b(Z=2-SMe)
CH(Et)S(O){D1-32b(X1=5-CF3)} D1-108b(Z=3-CF3)
CH(Et)S(O){D1-32b(X1=5-CF3)} D1-108b(Z=4-OCF3)
CH(Et)S(O){D1-32b(X1=5-CF3)} D1-108b(Z=2-SCF3)
CH(Et)S(O){D1-32b(X1=5-CF3)} C(O)Me
CH(Et)S(O){D1-32b(X1=5-CF3)} C(O)CF3
CH(Et)S(O){D1-32b(X1=5-CF3)} C(O)OMe
CH(Et)S(O)2{D1-32b(X1=5-CF3)} Me
CH(Et)S(O)2{D1-32b(X1=5-CF3)} Et
CH(Et)S(O)2{D1-32b(X1=5-CF3)} Pr-n
CH(Et)S(O)2{D1-32b(X1=5-CF3)} Pr-i
CH(Et)S(O)2{D1-32b(X1=5-CF3)} Pr-c
CH(Et)S(O)2{D1-32b(X1=5-CF3)} Bu-n
CH(Et)S(O)2{D1-32b(X1=5-CF3)} Bu-i
CH(Et)S(O)2{D1-32b(X1=5-CF3)} Bu-c
CH(Et)S(O)2{D1-32b(X1=5-CF3)} Bu-s
CH(Et)S(O)2{D1-32b(X1=5-CF3)} Bu-t
CH(Et)S(O)2{D1-32b(X1=5-CF3)} Pen-n
CH(Et)S(O)2{D1-32b(X1=5-CF3)} Pen-c
CH(Et)S(O)2{D1-32b(X1=5-CF3)} Hex-n
CH(Et)S(O)2{D1-32b(X1=5-CF3)} Hex-c
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2Pr-c
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2Bu-c
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2Pen-c
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2Hex-c
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2CH=CH2
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2CH=C(Cl)2
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2C≡CH
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2CN
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2CF3
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2OMe
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2OCF3
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2SMe
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2S(O)Me
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2S(O)2Me
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2SCF3
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2S(O)CF3
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2S(O)2CF3
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2CH(OMe)2
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2CH(SMe)2
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2C(O)Me
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2C(O)CF3
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2C(O)OMe
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-32a)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-33a)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-34a)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-37a)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-81a)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-82a)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-84a)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-85a)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-87a)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-92a)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-93a)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-95a)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-96a)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-98a)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108a)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-Cl)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=3-Me)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=4-OMe)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-SMe)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=3-CF3)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=4-OCF3)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2(D1-108b,Z=2-SCF3)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2CH2CN
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2CH2CF3
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2CH2OMe
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2CH2SMe
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2CH2S(O)Me
CH(Et)S(O)2{D1-32b(X1=5-CF3)} CH2CH2S(O)2Me
CH(Et)S(O)2{D1-32b(X1=5-CF3)} D1-32a
CH(Et)S(O)2{D1-32b(X1=5-CF3)} D1-33a
CH(Et)S(O)2{D1-32b(X1=5-CF3)} D1-34a
CH(Et)S(O)2{D1-32b(X1=5-CF3)} D1-37a
CH(Et)S(O)2{D1-32b(X1=5-CF3)} D1-81a
CH(Et)S(O)2{D1-32b(X1=5-CF3)} D1-82a
CH(Et)S(O)2{D1-32b(X1=5-CF3)} D1-84a
CH(Et)S(O)2{D1-32b(X1=5-CF3)} D1-85a
CH(Et)S(O)2{D1-32b(X1=5-CF3)} D1-87a
CH(Et)S(O)2{D1-32b(X1=5-CF3)} D1-92a
CH(Et)S(O)2{D1-32b(X1=5-CF3)} D1-93a
CH(Et)S(O)2{D1-32b(X1=5-CF3)} D1-95a
CH(Et)S(O)2{D1-32b(X1=5-CF3)} D1-96a
CH(Et)S(O)2{D1-32b(X1=5-CF3)} D1-98a
CH(Et)S(O)2{D1-32b(X1=5-CF3)} D1-108a
CH(Et)S(O)2{D1-32b(X1=5-CF3)} D1-108b(Z=2-Cl)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} D1-108b(Z=3-Me)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} D1-108b(Z=4-OMe)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} D1-108b(Z=2-SMe)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} D1-108b(Z=3-CF3)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} D1-108b(Z=4-OCF3)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} D1-108b(Z=2-SCF3)
CH(Et)S(O)2{D1-32b(X1=5-CF3)} C(O)Me
CH(Et)S(O)2{D1-32b(X1=5-CF3)} C(O)CF3
CH2SCH2C≡CH Me
CH2SCH2C≡CH Et
CH2SCH2C≡CH Pr-n
CH2SCH2C≡CH Pr-i
CH2SCH2C≡CH Pr-c
CH2SCH2C≡CH Bu-n
CH2SCH2C≡CH Bu-i
CH2SCH2C≡CH Bu-c
CH2SCH2C≡CH Bu-s
CH2SCH2C≡CH Bu-t
CH2SCH2C≡CH Pen-n
CH2SCH2C≡CH Pen-c
CH2SCH2C≡CH Hex-n
CH2SCH2C≡CH Hex-c
CH2SCH2C≡CH CH2Pr-c
CH2SCH2C≡CH CH2Bu-c
CH2SCH2C≡CH CH2Pen-c
CH2SCH2C≡CH CH2Hex-c
CH2SCH2C≡CH CH2CH=CH2
CH2SCH2C≡CH CH2CH=C(Cl)2
CH2SCH2C≡CH CH2C≡CH
CH2SCH2C≡CH CH2CN
CH2SCH2C≡CH CH2CF3
CH2SCH2C≡CH CH2OMe
CH2SCH2C≡CH CH2OCF3
CH2SCH2C≡CH CH2SMe
CH2SCH2C≡CH CH2S(O)Me
CH2SCH2C≡CH CH2S(O)2Me
CH2SCH2C≡CH CH2SCF3
CH2SCH2C≡CH CH2S(O)CF3
CH2SCH2C≡CH CH2S(O)2CF3
CH2SCH2C≡CH CH2CH(OMe)2
CH2SCH2C≡CH CH2CH(SMe)2
CH2SCH2C≡CH CH2C(O)Me
CH2SCH2C≡CH CH2C(O)CF3
CH2SCH2C≡CH CH2C(O)OMe
CH2SCH2C≡CH CH2(D1-32a)
CH2SCH2C≡CH CH2(D1-33a)
CH2SCH2C≡CH CH2(D1-34a)
CH2SCH2C≡CH CH2(D1-37a)
CH2SCH2C≡CH CH2(D1-81a)
CH2SCH2C≡CH CH2(D1-82a)
CH2SCH2C≡CH CH2(D1-84a)
CH2SCH2C≡CH CH2(D1-85a)
CH2SCH2C≡CH CH2(D1-87a)
CH2SCH2C≡CH CH2(D1-92a)
CH2SCH2C≡CH CH2(D1-93a)
CH2SCH2C≡CH CH2(D1-95a)
CH2SCH2C≡CH CH2(D1-96a)
CH2SCH2C≡CH CH2(D1-98a)
CH2SCH2C≡CH CH2(D1-108a)
CH2SCH2C≡CH CH2(D1-108b,Z=2-Cl)
CH2SCH2C≡CH CH2(D1-108b,Z=3-Me)
CH2SCH2C≡CH CH2(D1-108b,Z=4-OMe)
CH2SCH2C≡CH CH2(D1-108b,Z=2-SMe)
CH2SCH2C≡CH CH2(D1-108b,Z=3-CF3)
CH2SCH2C≡CH CH2(D1-108b,Z=4-OCF3)
CH2SCH2C≡CH CH2(D1-108b,Z=2-SCF3)
CH2SCH2C≡CH CH2CH2CN
CH2SCH2C≡CH CH2CH2CF3
CH2SCH2C≡CH CH2CH2OMe
CH2SCH2C≡CH CH2CH2SMe
CH2SCH2C≡CH CH2CH2S(O)Me
CH2SCH2C≡CH CH2CH2S(O)2Me
CH2SCH2C≡CH D1-32a
CH2SCH2C≡CH D1-33a
CH2SCH2C≡CH D1-34a
CH2SCH2C≡CH D1-37a
CH2SCH2C≡CH D1-81a
CH2SCH2C≡CH D1-82a
CH2SCH2C≡CH D1-84a
CH2SCH2C≡CH D1-85a
CH2SCH2C≡CH D1-87a
CH2SCH2C≡CH D1-92a
CH2SCH2C≡CH D1-93a
CH2SCH2C≡CH D1-95a
CH2SCH2C≡CH D1-96a
CH2SCH2C≡CH D1-98a
CH2SCH2C≡CH D1-108a
CH2SCH2C≡CH D1-108b(Z=2-Cl)
CH2SCH2C≡CH D1-108b(Z=3-Me)
CH2SCH2C≡CH D1-108b(Z=4-OMe)
CH2SCH2C≡CH D1-108b(Z=2-SMe)
CH2SCH2C≡CH D1-108b(Z=3-CF3)
CH2SCH2C≡CH D1-108b(Z=4-OCF3)
CH2SCH2C≡CH D1-108b(Z=2-SCF3)
CH2SCH2C≡CH C(O)Me
CH2SCH2C≡CH C(O)CF3
CH2SCH2C≡CH C(O)OMe
CH2S(O)CH2C≡CH Me
CH2S(O)CH2C≡CH Et
CH2S(O)CH2C≡CH Pr-n
CH2S(O)CH2C≡CH Pr-i
CH2S(O)CH2C≡CH Pr-c
CH2S(O)CH2C≡CH Bu-n
CH2S(O)CH2C≡CH Bu-i
CH2S(O)CH2C≡CH Bu-c
CH2S(O)CH2C≡CH Bu-s
CH2S(O)CH2C≡CH Bu-t
CH2S(O)CH2C≡CH Pen-n
CH2S(O)CH2C≡CH Pen-c
CH2S(O)CH2C≡CH Hex-n
CH2S(O)CH2C≡CH Hex-c
CH2S(O)CH2C≡CH CH2Pr-c
CH2S(O)CH2C≡CH CH2Bu-c
CH2S(O)CH2C≡CH CH2Pen-c
CH2S(O)CH2C≡CH CH2Hex-c
CH2S(O)CH2C≡CH CH2CH=CH2
CH2S(O)CH2C≡CH CH2CH=C(Cl)2
CH2S(O)CH2C≡CH CH2C≡CH
CH2S(O)CH2C≡CH CH2CN
CH2S(O)CH2C≡CH CH2CF3
CH2S(O)CH2C≡CH CH2OMe
CH2S(O)CH2C≡CH CH2OCF3
CH2S(O)CH2C≡CH CH2SMe
CH2S(O)CH2C≡CH CH2S(O)Me
CH2S(O)CH2C≡CH CH2S(O)2Me
CH2S(O)CH2C≡CH CH2SCF3
CH2S(O)CH2C≡CH CH2S(O)CF3
CH2S(O)CH2C≡CH CH2S(O)2CF3
CH2S(O)CH2C≡CH CH2CH(OMe)2
CH2S(O)CH2C≡CH CH2CH(SMe)2
CH2S(O)CH2C≡CH CH2C(O)Me
CH2S(O)CH2C≡CH CH2C(O)CF3
CH2S(O)CH2C≡CH CH2C(O)OMe
CH2S(O)CH2C≡CH CH2(D1-32a)
CH2S(O)CH2C≡CH CH2(D1-33a)
CH2S(O)CH2C≡CH CH2(D1-34a)
CH2S(O)CH2C≡CH CH2(D1-37a)
CH2S(O)CH2C≡CH CH2(D1-81a)
CH2S(O)CH2C≡CH CH2(D1-82a)
CH2S(O)CH2C≡CH CH2(D1-84a)
CH2S(O)CH2C≡CH CH2(D1-85a)
CH2S(O)CH2C≡CH CH2(D1-87a)
CH2S(O)CH2C≡CH CH2(D1-92a)
CH2S(O)CH2C≡CH CH2(D1-93a)
CH2S(O)CH2C≡CH CH2(D1-95a)
CH2S(O)CH2C≡CH CH2(D1-96a)
CH2S(O)CH2C≡CH CH2(D1-98a)
CH2S(O)CH2C≡CH CH2(D1-108a)
CH2S(O)CH2C≡CH CH2(D1-108b,Z=2-Cl)
CH2S(O)CH2C≡CH CH2(D1-108b,Z=3-Me)
CH2S(O)CH2C≡CH CH2(D1-108b,Z=4-OMe)
CH2S(O)CH2C≡CH CH2(D1-108b,Z=2-SMe)
CH2S(O)CH2C≡CH CH2(D1-108b,Z=3-CF3)
CH2S(O)CH2C≡CH CH2(D1-108b,Z=4-OCF3)
CH2S(O)CH2C≡CH CH2(D1-108b,Z=2-SCF3)
CH2S(O)CH2C≡CH CH2CH2CN
CH2S(O)CH2C≡CH CH2CH2CF3
CH2S(O)CH2C≡CH CH2CH2OMe
CH2S(O)CH2C≡CH CH2CH2SMe
CH2S(O)CH2C≡CH CH2CH2S(O)Me
CH2S(O)CH2C≡CH CH2CH2S(O)2Me
CH2S(O)CH2C≡CH D1-32a
CH2S(O)CH2C≡CH D1-33a
CH2S(O)CH2C≡CH D1-34a
CH2S(O)CH2C≡CH D1-37a
CH2S(O)CH2C≡CH D1-81a
CH2S(O)CH2C≡CH D1-82a
CH2S(O)CH2C≡CH D1-84a
CH2S(O)CH2C≡CH D1-85a
CH2S(O)CH2C≡CH D1-87a
CH2S(O)CH2C≡CH D1-92a
CH2S(O)CH2C≡CH D1-93a
CH2S(O)CH2C≡CH D1-95a
CH2S(O)CH2C≡CH D1-96a
CH2S(O)CH2C≡CH D1-98a
CH2S(O)CH2C≡CH D1-108a
CH2S(O)CH2C≡CH D1-108b(Z=2-Cl)
CH2S(O)CH2C≡CH D1-108b(Z=3-Me)
CH2S(O)CH2C≡CH D1-108b(Z=4-OMe)
CH2S(O)CH2C≡CH D1-108b(Z=2-SMe)
CH2S(O)CH2C≡CH D1-108b(Z=3-CF3)
CH2S(O)CH2C≡CH D1-108b(Z=4-OCF3)
CH2S(O)CH2C≡CH D1-108b(Z=2-SCF3)
CH2S(O)CH2C≡CH C(O)Me
CH2S(O)CH2C≡CH C(O)CF3
CH2S(O)CH2C≡CH C(O)OMe
CH2S(O)2CH2C≡CH Me
CH2S(O)2CH2C≡CH Et
CH2S(O)2CH2C≡CH Pr-n
CH2S(O)2CH2C≡CH Pr-i
CH2S(O)2CH2C≡CH Pr-c
CH2S(O)2CH2C≡CH Bu-n
CH2S(O)2CH2C≡CH Bu-i
CH2S(O)2CH2C≡CH Bu-c
CH2S(O)2CH2C≡CH Bu-s
CH2S(O)2CH2C≡CH Bu-t
CH2S(O)2CH2C≡CH Pen-n
CH2S(O)2CH2C≡CH Pen-c
CH2S(O)2CH2C≡CH Hex-n
CH2S(O)2CH2C≡CH Hex-c
CH2S(O)2CH2C≡CH CH2Pr-c
CH2S(O)2CH2C≡CH CH2Bu-c
CH2S(O)2CH2C≡CH CH2Pen-c
CH2S(O)2CH2C≡CH CH2Hex-c
CH2S(O)2CH2C≡CH CH2CH=CH2
CH2S(O)2CH2C≡CH CH2CH=C(Cl)2
CH2S(O)2CH2C≡CH CH2C≡CH
CH2S(O)2CH2C≡CH CH2CN
CH2S(O)2CH2C≡CH CH2CF3
CH2S(O)2CH2C≡CH CH2OMe
CH2S(O)2CH2C≡CH CH2OCF3
CH2S(O)2CH2C≡CH CH2SMe
CH2S(O)2CH2C≡CH CH2S(O)Me
CH2S(O)2CH2C≡CH CH2S(O)2Me
CH2S(O)2CH2C≡CH CH2SCF3
CH2S(O)2CH2C≡CH CH2S(O)CF3
CH2S(O)2CH2C≡CH CH2S(O)2CF3
CH2S(O)2CH2C≡CH CH2CH(OMe)2
CH2S(O)2CH2C≡CH CH2CH(SMe)2
CH2S(O)2CH2C≡CH CH2C(O)Me
CH2S(O)2CH2C≡CH CH2C(O)CF3
CH2S(O)2CH2C≡CH CH2C(O)OMe
CH2S(O)2CH2C≡CH CH2(D1-32a)
CH2S(O)2CH2C≡CH CH2(D1-33a)
CH2S(O)2CH2C≡CH CH2(D1-34a)
CH2S(O)2CH2C≡CH CH2(D1-37a)
CH2S(O)2CH2C≡CH CH2(D1-81a)
CH2S(O)2CH2C≡CH CH2(D1-82a)
CH2S(O)2CH2C≡CH CH2(D1-84a)
CH2S(O)2CH2C≡CH CH2(D1-85a)
CH2S(O)2CH2C≡CH CH2(D1-87a)
CH2S(O)2CH2C≡CH CH2(D1-92a)
CH2S(O)2CH2C≡CH CH2(D1-93a)
CH2S(O)2CH2C≡CH CH2(D1-95a)
CH2S(O)2CH2C≡CH CH2(D1-96a)
CH2S(O)2CH2C≡CH CH2(D1-98a)
CH2S(O)2CH2C≡CH CH2(D1-108a)
CH2S(O)2CH2C≡CH CH2(D1-108b,Z=2-Cl)
CH2S(O)2CH2C≡CH CH2(D1-108b,Z=3-Me)
CH2S(O)2CH2C≡CH CH2(D1-108b,Z=4-OMe)
CH2S(O)2CH2C≡CH CH2(D1-108b,Z=2-SMe)
CH2S(O)2CH2C≡CH CH2(D1-108b,Z=3-CF3)
CH2S(O)2CH2C≡CH CH2(D1-108b,Z=4-OCF3)
CH2S(O)2CH2C≡CH CH2(D1-108b,Z=2-SCF3)
CH2S(O)2CH2C≡CH CH2CH2CN
CH2S(O)2CH2C≡CH CH2CH2CF3
CH2S(O)2CH2C≡CH CH2CH2OMe
CH2S(O)2CH2C≡CH CH2CH2SMe
CH2S(O)2CH2C≡CH CH2CH2S(O)Me
CH2S(O)2CH2C≡CH CH2CH2S(O)2Me
CH2S(O)2CH2C≡CH D1-32a
CH2S(O)2CH2C≡CH D1-33a
CH2S(O)2CH2C≡CH D1-34a
CH2S(O)2CH2C≡CH D1-37a
CH2S(O)2CH2C≡CH D1-81a
CH2S(O)2CH2C≡CH D1-82a
CH2S(O)2CH2C≡CH D1-84a
CH2S(O)2CH2C≡CH D1-85a
CH2S(O)2CH2C≡CH D1-87a
CH2S(O)2CH2C≡CH D1-92a
CH2S(O)2CH2C≡CH D1-93a
CH2S(O)2CH2C≡CH D1-95a
CH2S(O)2CH2C≡CH D1-96a
CH2S(O)2CH2C≡CH D1-98a
CH2S(O)2CH2C≡CH D1-108a
CH2S(O)2CH2C≡CH D1-108b(Z=2-Cl)
CH2S(O)2CH2C≡CH D1-108b(Z=3-Me)
CH2S(O)2CH2C≡CH D1-108b(Z=4-OMe)
CH2S(O)2CH2C≡CH D1-108b(Z=2-SMe)
CH2S(O)2CH2C≡CH D1-108b(Z=3-CF3)
CH2S(O)2CH2C≡CH D1-108b(Z=4-OCF3)
CH2S(O)2CH2C≡CH D1-108b(Z=2-SCF3)
CH2S(O)2CH2C≡CH C(O)Me
CH2S(O)2CH2C≡CH C(O)CF3
CH2S(O)2CH2C≡CH C(O)OMe
CH(Me)SCH2C≡CH Me
CH(Me)SCH2C≡CH Et
CH(Me)SCH2C≡CH Pr-n
CH(Me)SCH2C≡CH Pr-i
CH(Me)SCH2C≡CH Pr-c
CH(Me)SCH2C≡CH Bu-n
CH(Me)SCH2C≡CH Bu-i
CH(Me)SCH2C≡CH Bu-c
CH(Me)SCH2C≡CH Bu-s
CH(Me)SCH2C≡CH Bu-t
CH(Me)SCH2C≡CH Pen-n
CH(Me)SCH2C≡CH Pen-c
CH(Me)SCH2C≡CH Hex-n
CH(Me)SCH2C≡CH Hex-c
CH(Me)SCH2C≡CH CH2Pr-c
CH(Me)SCH2C≡CH CH2Bu-c
CH(Me)SCH2C≡CH CH2Pen-c
CH(Me)SCH2C≡CH CH2Hex-c
CH(Me)SCH2C≡CH CH2CH=CH2
CH(Me)SCH2C≡CH CH2CH=C(Cl)2
CH(Me)SCH2C≡CH CH2C≡CH
CH(Me)SCH2C≡CH CH2CN
CH(Me)SCH2C≡CH CH2CF3
CH(Me)SCH2C≡CH CH2OMe
CH(Me)SCH2C≡CH CH2OCF3
CH(Me)SCH2C≡CH CH2SMe
CH(Me)SCH2C≡CH CH2S(O)Me
CH(Me)SCH2C≡CH CH2S(O)2Me
CH(Me)SCH2C≡CH CH2SCF3
CH(Me)SCH2C≡CH CH2S(O)CF3
CH(Me)SCH2C≡CH CH2S(O)2CF3
CH(Me)SCH2C≡CH CH2CH(OMe)2
CH(Me)SCH2C≡CH CH2CH(SMe)2
CH(Me)SCH2C≡CH CH2C(O)Me
CH(Me)SCH2C≡CH CH2C(O)CF3
CH(Me)SCH2C≡CH CH2C(O)OMe
CH(Me)SCH2C≡CH CH2(D1-32a)
CH(Me)SCH2C≡CH CH2(D1-33a)
CH(Me)SCH2C≡CH CH2(D1-34a)
CH(Me)SCH2C≡CH CH2(D1-37a)
CH(Me)SCH2C≡CH CH2(D1-81a)
CH(Me)SCH2C≡CH CH2(D1-82a)
CH(Me)SCH2C≡CH CH2(D1-84a)
CH(Me)SCH2C≡CH CH2(D1-85a)
CH(Me)SCH2C≡CH CH2(D1-87a)
CH(Me)SCH2C≡CH CH2(D1-92a)
CH(Me)SCH2C≡CH CH2(D1-93a)
CH(Me)SCH2C≡CH CH2(D1-95a)
CH(Me)SCH2C≡CH CH2(D1-96a)
CH(Me)SCH2C≡CH CH2(D1-98a)
CH(Me)SCH2C≡CH CH2(D1-108a)
CH(Me)SCH2C≡CH CH2(D1-108b,Z=2-Cl)
CH(Me)SCH2C≡CH CH2(D1-108b,Z=3-Me)
CH(Me)SCH2C≡CH CH2(D1-108b,Z=4-OMe)
CH(Me)SCH2C≡CH CH2(D1-108b,Z=2-SMe)
CH(Me)SCH2C≡CH CH2(D1-108b,Z=3-CF3)
CH(Me)SCH2C≡CH CH2(D1-108b,Z=4-OCF3)
CH(Me)SCH2C≡CH CH2(D1-108b,Z=2-SCF3)
CH(Me)SCH2C≡CH CH2CH2CN
CH(Me)SCH2C≡CH CH2CH2CF3
CH(Me)SCH2C≡CH CH2CH2OMe
CH(Me)SCH2C≡CH CH2CH2SMe
CH(Me)SCH2C≡CH CH2CH2S(O)Me
CH(Me)SCH2C≡CH CH2CH2S(O)2Me
CH(Me)SCH2C≡CH D1-32a
CH(Me)SCH2C≡CH D1-33a
CH(Me)SCH2C≡CH D1-34a
CH(Me)SCH2C≡CH D1-37a
CH(Me)SCH2C≡CH D1-81a
CH(Me)SCH2C≡CH D1-82a
CH(Me)SCH2C≡CH D1-84a
CH(Me)SCH2C≡CH D1-85a
CH(Me)SCH2C≡CH D1-87a
CH(Me)SCH2C≡CH D1-92a
CH(Me)SCH2C≡CH D1-93a
CH(Me)SCH2C≡CH D1-95a
CH(Me)SCH2C≡CH D1-96a
CH(Me)SCH2C≡CH D1-98a
CH(Me)SCH2C≡CH D1-108a
CH(Me)SCH2C≡CH D1-108b(Z=2-Cl)
CH(Me)SCH2C≡CH D1-108b(Z=3-Me)
CH(Me)SCH2C≡CH D1-108b(Z=4-OMe)
CH(Me)SCH2C≡CH D1-108b(Z=2-SMe)
CH(Me)SCH2C≡CH D1-108b(Z=3-CF3)
CH(Me)SCH2C≡CH D1-108b(Z=4-OCF3)
CH(Me)SCH2C≡CH D1-108b(Z=2-SCF3)
CH(Me)SCH2C≡CH C(O)Me
CH(Me)SCH2C≡CH C(O)CF3
CH(Me)SCH2C≡CH C(O)OMe
CH(Me)S(O)CH2C≡CH Me
CH(Me)S(O)CH2C≡CH Et
CH(Me)S(O)CH2C≡CH Pr-n
CH(Me)S(O)CH2C≡CH Pr-i
CH(Me)S(O)CH2C≡CH Pr-c
CH(Me)S(O)CH2C≡CH Bu-n
CH(Me)S(O)CH2C≡CH Bu-i
CH(Me)S(O)CH2C≡CH Bu-c
CH(Me)S(O)CH2C≡CH Bu-s
CH(Me)S(O)CH2C≡CH Bu-t
CH(Me)S(O)CH2C≡CH Pen-n
CH(Me)S(O)CH2C≡CH Pen-c
CH(Me)S(O)CH2C≡CH Hex-n
CH(Me)S(O)CH2C≡CH Hex-c
CH(Me)S(O)CH2C≡CH CH2Pr-c
CH(Me)S(O)CH2C≡CH CH2Bu-c
CH(Me)S(O)CH2C≡CH CH2Pen-c
CH(Me)S(O)CH2C≡CH CH2Hex-c
CH(Me)S(O)CH2C≡CH CH2CH=CH2
CH(Me)S(O)CH2C≡CH CH2CH=C(Cl)2
CH(Me)S(O)CH2C≡CH CH2C≡CH
CH(Me)S(O)CH2C≡CH CH2CN
CH(Me)S(O)CH2C≡CH CH2CF3
CH(Me)S(O)CH2C≡CH CH2OMe
CH(Me)S(O)CH2C≡CH CH2OCF3
CH(Me)S(O)CH2C≡CH CH2SMe
CH(Me)S(O)CH2C≡CH CH2S(O)Me
CH(Me)S(O)CH2C≡CH CH2S(O)2Me
CH(Me)S(O)CH2C≡CH CH2SCF3
CH(Me)S(O)CH2C≡CH CH2S(O)CF3
CH(Me)S(O)CH2C≡CH CH2S(O)2CF3
CH(Me)S(O)CH2C≡CH CH2CH(OMe)2
CH(Me)S(O)CH2C≡CH CH2CH(SMe)2
CH(Me)S(O)CH2C≡CH CH2C(O)Me
CH(Me)S(O)CH2C≡CH CH2C(O)CF3
CH(Me)S(O)CH2C≡CH CH2C(O)OMe
CH(Me)S(O)CH2C≡CH CH2(D1-32a)
CH(Me)S(O)CH2C≡CH CH2(D1-33a)
CH(Me)S(O)CH2C≡CH CH2(D1-34a)
CH(Me)S(O)CH2C≡CH CH2(D1-37a)
CH(Me)S(O)CH2C≡CH CH2(D1-81a)
CH(Me)S(O)CH2C≡CH CH2(D1-82a)
CH(Me)S(O)CH2C≡CH CH2(D1-84a)
CH(Me)S(O)CH2C≡CH CH2(D1-85a)
CH(Me)S(O)CH2C≡CH CH2(D1-87a)
CH(Me)S(O)CH2C≡CH CH2(D1-92a)
CH(Me)S(O)CH2C≡CH CH2(D1-93a)
CH(Me)S(O)CH2C≡CH CH2(D1-95a)
CH(Me)S(O)CH2C≡CH CH2(D1-96a)
CH(Me)S(O)CH2C≡CH CH2(D1-98a)
CH(Me)S(O)CH2C≡CH CH2(D1-108a)
CH(Me)S(O)CH2C≡CH CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)CH2C≡CH CH2(D1-108b,Z=3-Me)
CH(Me)S(O)CH2C≡CH CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)CH2C≡CH CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)CH2C≡CH CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)CH2C≡CH CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)CH2C≡CH CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)CH2C≡CH CH2CH2CN
CH(Me)S(O)CH2C≡CH CH2CH2CF3
CH(Me)S(O)CH2C≡CH CH2CH2OMe
CH(Me)S(O)CH2C≡CH CH2CH2SMe
CH(Me)S(O)CH2C≡CH CH2CH2S(O)Me
CH(Me)S(O)CH2C≡CH CH2CH2S(O)2Me
CH(Me)S(O)CH2C≡CH D1-32a
CH(Me)S(O)CH2C≡CH D1-33a
CH(Me)S(O)CH2C≡CH D1-34a
CH(Me)S(O)CH2C≡CH D1-37a
CH(Me)S(O)CH2C≡CH D1-81a
CH(Me)S(O)CH2C≡CH D1-82a
CH(Me)S(O)CH2C≡CH D1-84a
CH(Me)S(O)CH2C≡CH D1-85a
CH(Me)S(O)CH2C≡CH D1-87a
CH(Me)S(O)CH2C≡CH D1-92a
CH(Me)S(O)CH2C≡CH D1-93a
CH(Me)S(O)CH2C≡CH D1-95a
CH(Me)S(O)CH2C≡CH D1-96a
CH(Me)S(O)CH2C≡CH D1-98a
CH(Me)S(O)CH2C≡CH D1-108a
CH(Me)S(O)CH2C≡CH D1-108b(Z=2-Cl)
CH(Me)S(O)CH2C≡CH D1-108b(Z=3-Me)
CH(Me)S(O)CH2C≡CH D1-108b(Z=4-OMe)
CH(Me)S(O)CH2C≡CH D1-108b(Z=2-SMe)
CH(Me)S(O)CH2C≡CH D1-108b(Z=3-CF3)
CH(Me)S(O)CH2C≡CH D1-108b(Z=4-OCF3)
CH(Me)S(O)CH2C≡CH D1-108b(Z=2-SCF3)
CH(Me)S(O)CH2C≡CH C(O)Me
CH(Me)S(O)CH2C≡CH C(O)CF3
CH(Me)S(O)CH2C≡CH C(O)OMe
CH(Me)S(O)2CH2C≡CH Me
CH(Me)S(O)2CH2C≡CH Et
CH(Me)S(O)2CH2C≡CH Pr-n
CH(Me)S(O)2CH2C≡CH Pr-i
CH(Me)S(O)2CH2C≡CH Pr-c
CH(Me)S(O)2CH2C≡CH Bu-n
CH(Me)S(O)2CH2C≡CH Bu-i
CH(Me)S(O)2CH2C≡CH Bu-c
CH(Me)S(O)2CH2C≡CH Bu-s
CH(Me)S(O)2CH2C≡CH Bu-t
CH(Me)S(O)2CH2C≡CH Pen-n
CH(Me)S(O)2CH2C≡CH Pen-c
CH(Me)S(O)2CH2C≡CH Hex-n
CH(Me)S(O)2CH2C≡CH Hex-c
CH(Me)S(O)2CH2C≡CH CH2Pr-c
CH(Me)S(O)2CH2C≡CH CH2Bu-c
CH(Me)S(O)2CH2C≡CH CH2Pen-c
CH(Me)S(O)2CH2C≡CH CH2Hex-c
CH(Me)S(O)2CH2C≡CH CH2CH=CH2
CH(Me)S(O)2CH2C≡CH CH2CH=C(Cl)2
CH(Me)S(O)2CH2C≡CH CH2C≡CH
CH(Me)S(O)2CH2C≡CH CH2CN
CH(Me)S(O)2CH2C≡CH CH2CF3
CH(Me)S(O)2CH2C≡CH CH2OMe
CH(Me)S(O)2CH2C≡CH CH2OCF3
CH(Me)S(O)2CH2C≡CH CH2SMe
CH(Me)S(O)2CH2C≡CH CH2S(O)Me
CH(Me)S(O)2CH2C≡CH CH2S(O)2Me
CH(Me)S(O)2CH2C≡CH CH2SCF3
CH(Me)S(O)2CH2C≡CH CH2S(O)CF3
CH(Me)S(O)2CH2C≡CH CH2S(O)2CF3
CH(Me)S(O)2CH2C≡CH CH2CH(OMe)2
CH(Me)S(O)2CH2C≡CH CH2CH(SMe)2
CH(Me)S(O)2CH2C≡CH CH2C(O)Me
CH(Me)S(O)2CH2C≡CH CH2C(O)CF3
CH(Me)S(O)2CH2C≡CH CH2C(O)OMe
CH(Me)S(O)2CH2C≡CH CH2(D1-32a)
CH(Me)S(O)2CH2C≡CH CH2(D1-33a)
CH(Me)S(O)2CH2C≡CH CH2(D1-34a)
CH(Me)S(O)2CH2C≡CH CH2(D1-37a)
CH(Me)S(O)2CH2C≡CH CH2(D1-81a)
CH(Me)S(O)2CH2C≡CH CH2(D1-82a)
CH(Me)S(O)2CH2C≡CH CH2(D1-84a)
CH(Me)S(O)2CH2C≡CH CH2(D1-85a)
CH(Me)S(O)2CH2C≡CH CH2(D1-87a)
CH(Me)S(O)2CH2C≡CH CH2(D1-92a)
CH(Me)S(O)2CH2C≡CH CH2(D1-93a)
CH(Me)S(O)2CH2C≡CH CH2(D1-95a)
CH(Me)S(O)2CH2C≡CH CH2(D1-96a)
CH(Me)S(O)2CH2C≡CH CH2(D1-98a)
CH(Me)S(O)2CH2C≡CH CH2(D1-108a)
CH(Me)S(O)2CH2C≡CH CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)2CH2C≡CH CH2(D1-108b,Z=3-Me)
CH(Me)S(O)2CH2C≡CH CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)2CH2C≡CH CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)2CH2C≡CH CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)2CH2C≡CH CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)2CH2C≡CH CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)2CH2C≡CH CH2CH2CN
CH(Me)S(O)2CH2C≡CH CH2CH2CF3
CH(Me)S(O)2CH2C≡CH CH2CH2OMe
CH(Me)S(O)2CH2C≡CH CH2CH2SMe
CH(Me)S(O)2CH2C≡CH CH2CH2S(O)Me
CH(Me)S(O)2CH2C≡CH CH2CH2S(O)2Me
CH(Me)S(O)2CH2C≡CH D1-32a
CH(Me)S(O)2CH2C≡CH D1-33a
CH(Me)S(O)2CH2C≡CH D1-34a
CH(Me)S(O)2CH2C≡CH D1-37a
CH(Me)S(O)2CH2C≡CH D1-81a
CH(Me)S(O)2CH2C≡CH D1-82a
CH(Me)S(O)2CH2C≡CH D1-84a
CH(Me)S(O)2CH2C≡CH D1-85a
CH(Me)S(O)2CH2C≡CH D1-87a
CH(Me)S(O)2CH2C≡CH D1-92a
CH(Me)S(O)2CH2C≡CH D1-93a
CH(Me)S(O)2CH2C≡CH D1-95a
CH(Me)S(O)2CH2C≡CH D1-96a
CH(Me)S(O)2CH2C≡CH D1-98a
CH(Me)S(O)2CH2C≡CH D1-108a
CH(Me)S(O)2CH2C≡CH D1-108b(Z=2-Cl)
CH(Me)S(O)2CH2C≡CH D1-108b(Z=3-Me)
CH(Me)S(O)2CH2C≡CH D1-108b(Z=4-OMe)
CH(Me)S(O)2CH2C≡CH D1-108b(Z=2-SMe)
CH(Me)S(O)2CH2C≡CH D1-108b(Z=3-CF3)
CH(Me)S(O)2CH2C≡CH D1-108b(Z=4-OCF3)
CH(Me)S(O)2CH2C≡CH D1-108b(Z=2-SCF3)
CH(Me)S(O)2CH2C≡CH C(O)Me
CH(Me)S(O)2CH2C≡CH C(O)CF3
CH(Me)S(O)2CH2C≡CH C(O)OMe
CH(Et)SCH2C≡CH Me
CH(Et)SCH2C≡CH Et
CH(Et)SCH2C≡CH Pr-n
CH(Et)SCH2C≡CH Pr-i
CH(Et)SCH2C≡CH Pr-c
CH(Et)SCH2C≡CH Bu-n
CH(Et)SCH2C≡CH Bu-i
CH(Et)SCH2C≡CH Bu-c
CH(Et)SCH2C≡CH Bu-s
CH(Et)SCH2C≡CH Bu-t
CH(Et)SCH2C≡CH Pen-n
CH(Et)SCH2C≡CH Pen-c
CH(Et)SCH2C≡CH Hex-n
CH(Et)SCH2C≡CH Hex-c
CH(Et)SCH2C≡CH CH2Pr-c
CH(Et)SCH2C≡CH CH2Bu-c
CH(Et)SCH2C≡CH CH2Pen-c
CH(Et)SCH2C≡CH CH2Hex-c
CH(Et)SCH2C≡CH CH2CH=CH2
CH(Et)SCH2C≡CH CH2CH=C(Cl)2
CH(Et)SCH2C≡CH CH2C≡CH
CH(Et)SCH2C≡CH CH2CN
CH(Et)SCH2C≡CH CH2CF3
CH(Et)SCH2C≡CH CH2OMe
CH(Et)SCH2C≡CH CH2OCF3
CH(Et)SCH2C≡CH CH2SMe
CH(Et)SCH2C≡CH CH2S(O)Me
CH(Et)SCH2C≡CH CH2S(O)2Me
CH(Et)SCH2C≡CH CH2SCF3
CH(Et)SCH2C≡CH CH2S(O)CF3
CH(Et)SCH2C≡CH CH2S(O)2CF3
CH(Et)SCH2C≡CH CH2CH(OMe)2
CH(Et)SCH2C≡CH CH2CH(SMe)2
CH(Et)SCH2C≡CH CH2C(O)Me
CH(Et)SCH2C≡CH CH2C(O)CF3
CH(Et)SCH2C≡CH CH2C(O)OMe
CH(Et)SCH2C≡CH CH2(D1-32a)
CH(Et)SCH2C≡CH CH2(D1-33a)
CH(Et)SCH2C≡CH CH2(D1-34a)
CH(Et)SCH2C≡CH CH2(D1-37a)
CH(Et)SCH2C≡CH CH2(D1-81a)
CH(Et)SCH2C≡CH CH2(D1-82a)
CH(Et)SCH2C≡CH CH2(D1-84a)
CH(Et)SCH2C≡CH CH2(D1-85a)
CH(Et)SCH2C≡CH CH2(D1-87a)
CH(Et)SCH2C≡CH CH2(D1-92a)
CH(Et)SCH2C≡CH CH2(D1-93a)
CH(Et)SCH2C≡CH CH2(D1-95a)
CH(Et)SCH2C≡CH CH2(D1-96a)
CH(Et)SCH2C≡CH CH2(D1-98a)
CH(Et)SCH2C≡CH CH2(D1-108a)
CH(Et)SCH2C≡CH CH2(D1-108b,Z=2-Cl)
CH(Et)SCH2C≡CH CH2(D1-108b,Z=3-Me)
CH(Et)SCH2C≡CH CH2(D1-108b,Z=4-OMe)
CH(Et)SCH2C≡CH CH2(D1-108b,Z=2-SMe)
CH(Et)SCH2C≡CH CH2(D1-108b,Z=3-CF3)
CH(Et)SCH2C≡CH CH2(D1-108b,Z=4-OCF3)
CH(Et)SCH2C≡CH CH2(D1-108b,Z=2-SCF3)
CH(Et)SCH2C≡CH CH2CH2CN
CH(Et)SCH2C≡CH CH2CH2CF3
CH(Et)SCH2C≡CH CH2CH2OMe
CH(Et)SCH2C≡CH CH2CH2SMe
CH(Et)SCH2C≡CH CH2CH2S(O)Me
CH(Et)SCH2C≡CH CH2CH2S(O)2Me
CH(Et)SCH2C≡CH D1-32a
CH(Et)SCH2C≡CH D1-33a
CH(Et)SCH2C≡CH D1-34a
CH(Et)SCH2C≡CH D1-37a
CH(Et)SCH2C≡CH D1-81a
CH(Et)SCH2C≡CH D1-82a
CH(Et)SCH2C≡CH D1-84a
CH(Et)SCH2C≡CH D1-85a
CH(Et)SCH2C≡CH D1-87a
CH(Et)SCH2C≡CH D1-92a
CH(Et)SCH2C≡CH D1-93a
CH(Et)SCH2C≡CH D1-95a
CH(Et)SCH2C≡CH D1-96a
CH(Et)SCH2C≡CH D1-98a
CH(Et)SCH2C≡CH D1-108a
CH(Et)SCH2C≡CH D1-108b(Z=2-Cl)
CH(Et)SCH2C≡CH D1-108b(Z=3-Me)
CH(Et)SCH2C≡CH D1-108b(Z=4-OMe)
CH(Et)SCH2C≡CH D1-108b(Z=2-SMe)
CH(Et)SCH2C≡CH D1-108b(Z=3-CF3)
CH(Et)SCH2C≡CH D1-108b(Z=4-OCF3)
CH(Et)SCH2C≡CH D1-108b(Z=2-SCF3)
CH(Et)SCH2C≡CH C(O)Me
CH(Et)SCH2C≡CH C(O)CF3
CH(Et)SCH2C≡CH C(O)OMe
CH(Et)S(O)CH2C≡CH Me
CH(Et)S(O)CH2C≡CH Et
CH(Et)S(O)CH2C≡CH Pr-n
CH(Et)S(O)CH2C≡CH Pr-i
CH(Et)S(O)CH2C≡CH Pr-c
CH(Et)S(O)CH2C≡CH Bu-n
CH(Et)S(O)CH2C≡CH Bu-i
CH(Et)S(O)CH2C≡CH Bu-c
CH(Et)S(O)CH2C≡CH Bu-s
CH(Et)S(O)CH2C≡CH Bu-t
CH(Et)S(O)CH2C≡CH Pen-n
CH(Et)S(O)CH2C≡CH Pen-c
CH(Et)S(O)CH2C≡CH Hex-n
CH(Et)S(O)CH2C≡CH Hex-c
CH(Et)S(O)CH2C≡CH CH2Pr-c
CH(Et)S(O)CH2C≡CH CH2Bu-c
CH(Et)S(O)CH2C≡CH CH2Pen-c
CH(Et)S(O)CH2C≡CH CH2Hex-c
CH(Et)S(O)CH2C≡CH CH2CH=CH2
CH(Et)S(O)CH2C≡CH CH2CH=C(Cl)2
CH(Et)S(O)CH2C≡CH CH2C≡CH
CH(Et)S(O)CH2C≡CH CH2CN
CH(Et)S(O)CH2C≡CH CH2CF3
CH(Et)S(O)CH2C≡CH CH2OMe
CH(Et)S(O)CH2C≡CH CH2OCF3
CH(Et)S(O)CH2C≡CH CH2SMe
CH(Et)S(O)CH2C≡CH CH2S(O)Me
CH(Et)S(O)CH2C≡CH CH2S(O)2Me
CH(Et)S(O)CH2C≡CH CH2SCF3
CH(Et)S(O)CH2C≡CH CH2S(O)CF3
CH(Et)S(O)CH2C≡CH CH2S(O)2CF3
CH(Et)S(O)CH2C≡CH CH2CH(OMe)2
CH(Et)S(O)CH2C≡CH CH2CH(SMe)2
CH(Et)S(O)CH2C≡CH CH2C(O)Me
CH(Et)S(O)CH2C≡CH CH2C(O)CF3
CH(Et)S(O)CH2C≡CH CH2C(O)OMe
CH(Et)S(O)CH2C≡CH CH2(D1-32a)
CH(Et)S(O)CH2C≡CH CH2(D1-33a)
CH(Et)S(O)CH2C≡CH CH2(D1-34a)
CH(Et)S(O)CH2C≡CH CH2(D1-37a)
CH(Et)S(O)CH2C≡CH CH2(D1-81a)
CH(Et)S(O)CH2C≡CH CH2(D1-82a)
CH(Et)S(O)CH2C≡CH CH2(D1-84a)
CH(Et)S(O)CH2C≡CH CH2(D1-85a)
CH(Et)S(O)CH2C≡CH CH2(D1-87a)
CH(Et)S(O)CH2C≡CH CH2(D1-92a)
CH(Et)S(O)CH2C≡CH CH2(D1-93a)
CH(Et)S(O)CH2C≡CH CH2(D1-95a)
CH(Et)S(O)CH2C≡CH CH2(D1-96a)
CH(Et)S(O)CH2C≡CH CH2(D1-98a)
CH(Et)S(O)CH2C≡CH CH2(D1-108a)
CH(Et)S(O)CH2C≡CH CH2(D1-108b,Z=2-Cl)
CH(Et)S(O)CH2C≡CH CH2(D1-108b,Z=3-Me)
CH(Et)S(O)CH2C≡CH CH2(D1-108b,Z=4-OMe)
CH(Et)S(O)CH2C≡CH CH2(D1-108b,Z=2-SMe)
CH(Et)S(O)CH2C≡CH CH2(D1-108b,Z=3-CF3)
CH(Et)S(O)CH2C≡CH CH2(D1-108b,Z=4-OCF3)
CH(Et)S(O)CH2C≡CH CH2(D1-108b,Z=2-SCF3)
CH(Et)S(O)CH2C≡CH CH2CH2CN
CH(Et)S(O)CH2C≡CH CH2CH2CF3
CH(Et)S(O)CH2C≡CH CH2CH2OMe
CH(Et)S(O)CH2C≡CH CH2CH2SMe
CH(Et)S(O)CH2C≡CH CH2CH2S(O)Me
CH(Et)S(O)CH2C≡CH CH2CH2S(O)2Me
CH(Et)S(O)CH2C≡CH D1-32a
CH(Et)S(O)CH2C≡CH D1-33a
CH(Et)S(O)CH2C≡CH D1-34a
CH(Et)S(O)CH2C≡CH D1-37a
CH(Et)S(O)CH2C≡CH D1-81a
CH(Et)S(O)CH2C≡CH D1-82a
CH(Et)S(O)CH2C≡CH D1-84a
CH(Et)S(O)CH2C≡CH D1-85a
CH(Et)S(O)CH2C≡CH D1-87a
CH(Et)S(O)CH2C≡CH D1-92a
CH(Et)S(O)CH2C≡CH D1-93a
CH(Et)S(O)CH2C≡CH D1-95a
CH(Et)S(O)CH2C≡CH D1-96a
CH(Et)S(O)CH2C≡CH D1-98a
CH(Et)S(O)CH2C≡CH D1-108a
CH(Et)S(O)CH2C≡CH D1-108b(Z=2-Cl)
CH(Et)S(O)CH2C≡CH D1-108b(Z=3-Me)
CH(Et)S(O)CH2C≡CH D1-108b(Z=4-OMe)
CH(Et)S(O)CH2C≡CH D1-108b(Z=2-SMe)
CH(Et)S(O)CH2C≡CH D1-108b(Z=3-CF3)
CH(Et)S(O)CH2C≡CH D1-108b(Z=4-OCF3)
CH(Et)S(O)CH2C≡CH D1-108b(Z=2-SCF3)
CH(Et)S(O)CH2C≡CH C(O)Me
CH(Et)S(O)CH2C≡CH C(O)CF3
CH(Et)S(O)CH2C≡CH C(O)OMe
CH(Et)S(O)2CH2C≡CH Me
CH(Et)S(O)2CH2C≡CH Et
CH(Et)S(O)2CH2C≡CH Pr-n
CH(Et)S(O)2CH2C≡CH Pr-i
CH(Et)S(O)2CH2C≡CH Pr-c
CH(Et)S(O)2CH2C≡CH Bu-n
CH(Et)S(O)2CH2C≡CH Bu-i
CH(Et)S(O)2CH2C≡CH Bu-c
CH(Et)S(O)2CH2C≡CH Bu-s
CH(Et)S(O)2CH2C≡CH Bu-t
CH(Et)S(O)2CH2C≡CH Pen-n
CH(Et)S(O)2CH2C≡CH Pen-c
CH(Et)S(O)2CH2C≡CH Hex-n
CH(Et)S(O)2CH2C≡CH Hex-c
CH(Et)S(O)2CH2C≡CH CH2Pr-c
CH(Et)S(O)2CH2C≡CH CH2Bu-c
CH(Et)S(O)2CH2C≡CH CH2Pen-c
CH(Et)S(O)2CH2C≡CH CH2Hex-c
CH(Et)S(O)2CH2C≡CH CH2CH=CH2
CH(Et)S(O)2CH2C≡CH CH2CH=C(Cl)2
CH(Et)S(O)2CH2C≡CH CH2C≡CH
CH(Et)S(O)2CH2C≡CH CH2CN
CH(Et)S(O)2CH2C≡CH CH2CF3
CH(Et)S(O)2CH2C≡CH CH2OMe
CH(Et)S(O)2CH2C≡CH CH2OCF3
CH(Et)S(O)2CH2C≡CH CH2SMe
CH(Et)S(O)2CH2C≡CH CH2S(O)Me
CH(Et)S(O)2CH2C≡CH CH2S(O)2Me
CH(Et)S(O)2CH2C≡CH CH2SCF3
CH(Et)S(O)2CH2C≡CH CH2S(O)CF3
CH(Et)S(O)2CH2C≡CH CH2S(O)2CF3
CH(Et)S(O)2CH2C≡CH CH2CH(OMe)2
CH(Et)S(O)2CH2C≡CH CH2CH(SMe)2
CH(Et)S(O)2CH2C≡CH CH2C(O)Me
CH(Et)S(O)2CH2C≡CH CH2C(O)CF3
CH(Et)S(O)2CH2C≡CH CH2C(O)OMe
CH(Et)S(O)2CH2C≡CH CH2(D1-32a)
CH(Et)S(O)2CH2C≡CH CH2(D1-33a)
CH(Et)S(O)2CH2C≡CH CH2(D1-34a)
CH(Et)S(O)2CH2C≡CH CH2(D1-37a)
CH(Et)S(O)2CH2C≡CH CH2(D1-81a)
CH(Et)S(O)2CH2C≡CH CH2(D1-82a)
CH(Et)S(O)2CH2C≡CH CH2(D1-84a)
CH(Et)S(O)2CH2C≡CH CH2(D1-85a)
CH(Et)S(O)2CH2C≡CH CH2(D1-87a)
CH(Et)S(O)2CH2C≡CH CH2(D1-92a)
CH(Et)S(O)2CH2C≡CH CH2(D1-93a)
CH(Et)S(O)2CH2C≡CH CH2(D1-95a)
CH(Et)S(O)2CH2C≡CH CH2(D1-96a)
CH(Et)S(O)2CH2C≡CH CH2(D1-98a)
CH(Et)S(O)2CH2C≡CH CH2(D1-108a)
CH(Et)S(O)2CH2C≡CH CH2(D1-108b,Z=2-Cl)
CH(Et)S(O)2CH2C≡CH CH2(D1-108b,Z=3-Me)
CH(Et)S(O)2CH2C≡CH CH2(D1-108b,Z=4-OMe)
CH(Et)S(O)2CH2C≡CH CH2(D1-108b,Z=2-SMe)
CH(Et)S(O)2CH2C≡CH CH2(D1-108b,Z=3-CF3)
CH(Et)S(O)2CH2C≡CH CH2(D1-108b,Z=4-OCF3)
CH(Et)S(O)2CH2C≡CH CH2(D1-108b,Z=2-SCF3)
CH(Et)S(O)2CH2C≡CH CH2CH2CN
CH(Et)S(O)2CH2C≡CH CH2CH2CF3
CH(Et)S(O)2CH2C≡CH CH2CH2OMe
CH(Et)S(O)2CH2C≡CH CH2CH2SMe
CH(Et)S(O)2CH2C≡CH CH2CH2S(O)Me
CH(Et)S(O)2CH2C≡CH CH2CH2S(O)2Me
CH(Et)S(O)2CH2C≡CH D1-32a
CH(Et)S(O)2CH2C≡CH D1-33a
CH(Et)S(O)2CH2C≡CH D1-34a
CH(Et)S(O)2CH2C≡CH D1-37a
CH(Et)S(O)2CH2C≡CH D1-81a
CH(Et)S(O)2CH2C≡CH D1-82a
CH(Et)S(O)2CH2C≡CH D1-84a
CH(Et)S(O)2CH2C≡CH D1-85a
CH(Et)S(O)2CH2C≡CH D1-87a
CH(Et)S(O)2CH2C≡CH D1-92a
CH(Et)S(O)2CH2C≡CH D1-93a
CH(Et)S(O)2CH2C≡CH D1-95a
CH(Et)S(O)2CH2C≡CH D1-96a
CH(Et)S(O)2CH2C≡CH D1-98a
CH(Et)S(O)2CH2C≡CH D1-108a
CH(Et)S(O)2CH2C≡CH D1-108b(Z=2-Cl)
CH(Et)S(O)2CH2C≡CH D1-108b(Z=3-Me)
CH(Et)S(O)2CH2C≡CH D1-108b(Z=4-OMe)
CH(Et)S(O)2CH2C≡CH D1-108b(Z=2-SMe)
CH(Et)S(O)2CH2C≡CH D1-108b(Z=3-CF3)
CH(Et)S(O)2CH2C≡CH D1-108b(Z=4-OCF3)
CH(Et)S(O)2CH2C≡CH D1-108b(Z=2-SCF3)
CH(Et)S(O)2CH2C≡CH C(O)Me
CH(Et)S(O)2CH2C≡CH C(O)CF3
CH(Et)S(O)2CH2C≡CH C(O)OMe
Me Me
Et Me
Pr-n Me
Pr-i Me
Bu-n Me
Bu-i Me
Bu-t Me
Pen-n Me
Hex-n Me
CH(Et)Cl Me
CH2{D1-7b(3-CF3)} Me
CH(CN)Ph Me
SMe Me
SEt Me
SPr-n Me
SPr-i Me
SBu-n Me
SBu-i Me
SBu-t Me
SPen-n Me
SHex-n Me
SPr-c Me
SBu-c Me
SPen-c Me
SHex-c Me
SCH2CH=CH2 Me
SCH2C三CH Me
SCF2H Me
SCF3 Me
SCF2Cl Me
SCH2CF3 Me
S(D1-108c) Me
CH2OH Me
CH2OMe Me
CH2OEt Me
CH2OPr-n Me
CH2OPr-i Me
CH2OBu-n Me
CH2OBu-i Me
CH2OBu-s Me
CH2OBu-t Me
CH2OPen-n Me
CH2OHex-n Me
CH2O(D1-104c) Me
CH(Me)OH Me
CH(Me)OMe Me
CH(Me)OEt Me
CH(Me)OPr-n Me
CH(Me)OPr-i Me
CH(Me)OBu-n Me
CH(Me)OBu-i Me
CH(Me)OBu-s Me
CH(Me)OBu-t Me
CH(Me)OPen-n Me
CH(Me)OHex-n Me
CH(Me)O(D1-104c) Me
CH(Et)OH Me
CH(Et)OMe Me
CH(Et)OEt Me
CH(Et)OPr-n Me
CH(Et)OPr-i Me
CH(Et)OBu-n Me
CH(Et)OBu-i Me
CH(Et)OBu-s Me
CH(Et)OBu-t Me
CH(Et)OPen-n Me
CH(Et)OHex-n Me
CH(Et)O(D1-104c) Me
CH(n-Pr)OH Me
CH(n-Pr)OMe Me
CH(n-Pr)OEt Me
CH(n-Pr)O(D1-104c) Me
CH(i-Pr)OH Me
CH(i-Pr)OMe Me
CH(i-Pr)OEt Me
CH(i-Pr)O(D1-104c) Me
CH(n-Bu)OH Me
CH(n-Bu)OMe Me
CH(n-Bu)OEt Me
CH(n-Bu)O(D1-104c) Me
C(Me)2OH Me
C(Me)2OMe Me
C(Me)2OEt Me
C(Me)2O(D1-104c) Me
CH2CH2OH Me
CH2CH2OMe Me
CH2CH2OEt Me
CH2CH2O(D1-104c) Me
CH(Me)CH2OH Me
CH(Me)CH2OMe Me
CH(Me)CH2OEt Me
CH(Me)CH2O(D1-104c) Me
CH(Et)CH2OH Me
CH(Et)CH2OMe Me
CH(Et)CH2OEt Me
CH(Et)CH2O(D1-104c) Me
CH(n-Pr)CH2OH Me
CH(n-Pr)CH2OMe Me
CH(n-Pr)CH2OEt Me
CH(n-Pr)CH2O(D1-104c) Me
CH(i-Pr)CH2OH Me
CH(i-Pr)CH2OMe Me
CH(i-Pr)CH2OEt Me
CH(i-Pr)CH2O(D1-104c) Me
CH(n-Bu)CH2OH Me
CH(n-Bu)CH2OMe Me
CH(n-Bu)CH2OEt Me
CH(n-Bu)CH2O(D1-104c) Me
C(Me)2CH2OH Me
C(Me)2CH2OMe Me
C(Me)2CH2OEt Me
C(Me)2CH2O(D1-104c) Me
CH2SH Me
CH2SMe Me
CH2SEt Me
CH2SPr-n Me
CH2SPr-i Me
CH2SBu-n Me
CH2SBu-i Me
CH2SBu-t Me
CH2SPen-n Me
CH2SHex-n Me
CH2SPr-c Me
CH2SBu-c Me
CH2SPen-c Me
CH2SHex-c Me
CH2SCH2CH=CH2 Me
CH2SCH2C三CH Me
CH2SCF2H Me
CH2SCF3 Me
CH2SCF2Cl Me
CH2SCH2CF3 Me
CH2S{D1-108c} Me
CH2S(O)Me Me
CH2S(O)Et Me
CH2S(O)Pr-n Me
CH2S(O)Pr-i Me
CH2S(O)Bu-n Me
CH2S(O)Bu-i Me
CH2S(O)Bu-t Me
CH2S(O)Pen-n Me
CH2S(O)Hex-n Me
CH2S(O)Pr-c Me
CH2S(O)Bu-c Me
CH2S(O)Pen-c Me
CH2S(O)Hex-c Me
CH2S(O)CH2CH=CH2 Me
CH2S(O)CH2C三CH Me
CH2S(O)CF2H Me
CH2S(O)CF3 Me
CH2S(O)CF2Cl Me
CH2S(O)CH2CF3 Me
CH2S(O){D1-108c} Me
CH2S(O)2Me Me
CH2S(O)2Et Me
CH2S(O)2Pr-n Me
CH2S(O)2Pr-i Me
CH2S(O)2Bu-n Me
CH2S(O)2Bu-i Me
CH2S(O)2Bu-t Me
CH2S(O)2Pen-n Me
CH2S(O)2Hex-n Me
CH2S(O)2Pr-c Me
CH2S(O)2Bu-c Me
CH2S(O)2Pen-c Me
CH2S(O)2Hex-c Me
CH2S(O)2CH2CH=CH2 Me
CH2S(O)2CH2C三CH Me
CH2S(O)2CF2H Me
CH2S(O)2CF3 Me
CH2S(O)2CF2Cl Me
CH2S(O)2CH2CF3 Me
CH2S(O)2{D1-108c} Me
CH(Me)SH Me
CH(Me)SMe Me
CH(Me)SEt Me
CH(Me)SPr-n Me
CH(Me)SPr-i Me
CH(Me)SBu-n Me
CH(Me)SBu-i Me
CH(Me)SBu-t Me
CH(Me)SPen-n Me
CH(Me)SHex-n Me
CH(Me)SPr-c Me
CH(Me)SBu-c Me
CH(Me)SPen-c Me
CH(Me)SHex-c Me
CH(Me)SCH2CH=CH2 Me
CH(Me)SCH2C三CH Me
CH(Me)SCF2H Me
CH(Me)SCF3 Me
CH(Me)SCF2Cl Me
CH(Me)SCH2CF3 Me
CH(Me)S{D1-108c} Me
CH(Me)S(O)Me Me
CH(Me)S(O)Et Me
CH(Me)S(O)Pr-n Me
CH(Me)S(O)Pr-i Me
CH(Me)S(O)Bu-n Me
CH(Me)S(O)Bu-i Me
CH(Me)S(O)Bu-t Me
CH(Me)S(O)Pen-n Me
CH(Me)S(O)Hex-n Me
CH(Me)S(O)Pr-c Me
CH(Me)S(O)Bu-c Me
CH(Me)S(O)Pen-c Me
CH(Me)S(O)Hex-c Me
CH(Me)S(O)CH2CH=CH2 Me
CH(Me)S(O)CH2C三CH Me
CH(Me)S(O)CF2H Me
CH(Me)S(O)CF3 Me
CH(Me)S(O)CF2Cl Me
CH(Me)S(O)CH2CF3 Me
CH(Me)S(O){D1-108c} Me
CH(Me)S(O)2Me Me
CH(Me)S(O)2Et Me
CH(Me)S(O)2Pr-n Me
CH(Me)S(O)2Pr-i Me
CH(Me)S(O)2Bu-n Me
CH(Me)S(O)2Bu-i Me
CH(Me)S(O)2Bu-t Me
CH(Me)S(O)2Pen-n Me
CH(Me)S(O)2Hex-n Me
CH(Me)S(O)2Pr-c Me
CH(Me)S(O)2Bu-c Me
CH(Me)S(O)2Pen-c Me
CH(Me)S(O)2Hex-c Me
CH(Me)S(O)2CH2CH=CH2 Me
CH(Me)S(O)2CH2C三CH Me
CH(Me)S(O)2CF2H Me
CH(Me)S(O)2CF3 Me
CH(Me)S(O)2CF2Cl Me
CH(Me)S(O)2CH2CF3 Me
CH(Me)S(O)2{D1-108c} Me
CH(Et)SH Me
CH(Et)SMe Me
CH(Et)SEt Me
CH(Et)SPr-n Me
CH(Et)SPr-i Me
CH(Et)SBu-n Me
CH(Et)SBu-i Me
CH(Et)SBu-t Me
CH(Et)SPen-n Me
CH(Et)SHex-n Me
CH(Et)SPr-c Me
CH(Et)SBu-c Me
CH(Et)SPen-c Me
CH(Et)SHex-c Me
CH(Et)SCH2CH=CH2 Me
CH(Et)SCH2C三CH Me
CH(Et)SCF2H Me
CH(Et)SCF3 Me
CH(Et)SCF2Cl Me
CH(Et)SCH2CF3 Me
CH(Et)S{D1-108c} Me
CH(Et)S(O)Me Me
CH(Et)S(O)Et Me
CH(Et)S(O)Pr-n Me
CH(Et)S(O)Pr-i Me
CH(Et)S(O)Bu-n Me
CH(Et)S(O)Bu-i Me
CH(Et)S(O)Bu-t Me
CH(Et)S(O)Pen-n Me
CH(Et)S(O)Hex-n Me
CH(Et)S(O)Pr-c Me
CH(Et)S(O)Bu-c Me
CH(Et)S(O)Pen-c Me
CH(Et)S(O)Hex-c Me
CH(Et)S(O)CH2CH=CH2 Me
CH(Et)S(O)CH2C三CH Me
CH(Et)S(O)CF2H Me
CH(Et)S(O)CF3 Me
CH(Et)S(O)CF2Cl Me
CH(Et)S(O)CH2CF3 Me
CH(Et)S(O){D1-108c} Me
CH(Et)S(O)2Me Me
CH(Et)S(O)2Et Me
CH(Et)S(O)2Pr-n Me
CH(Et)S(O)2Pr-i Me
CH(Et)S(O)2Bu-n Me
CH(Et)S(O)2Bu-i Me
CH(Et)S(O)2Bu-t Me
CH(Et)S(O)2Pen-n Me
CH(Et)S(O)2Hex-n Me
CH(Et)S(O)2Pr-c Me
CH(Et)S(O)2Bu-c Me
CH(Et)S(O)2Pen-c Me
CH(Et)S(O)2Hex-c Me
CH(Et)S(O)2CH2CH=CH2 Me
CH(Et)S(O)2CH2C三CH Me
CH(Et)S(O)2CF2H Me
CH(Et)S(O)2CF3 Me
CH(Et)S(O)2CF2Cl Me
CH(Et)S(O)2CH2CF3 Me
CH(Et)S(O)2{D1-108c} Me
CH(n-Pr)SH Me
CH(n-Pr)SMe Me
CH(n-Pr)SEt Me
CH(n-Pr)SPr-n Me
CH(n-Pr)SPr-i Me
CH(n-Pr)SBu-n Me
CH(n-Pr)SBu-i Me
CH(n-Pr)SBu-t Me
CH(n-Pr)SPen-n Me
CH(n-Pr)SHex-n Me
CH(n-Pr)SPr-c Me
CH(n-Pr)SBu-c Me
CH(n-Pr)SPen-c Me
CH(n-Pr)SHex-c Me
CH(n-Pr)SCH2CH=CH2 Me
CH(n-Pr)SCH2C三CH Me
CH(n-Pr)SCF2H Me
CH(n-Pr)SCF3 Me
CH(n-Pr)SCF2Cl Me
CH(n-Pr)SCH2CF3 Me
CH(n-Pr)S{D1-108c} Me
CH(n-Pr)S(O)Me Me
CH(n-Pr)S(O)Et Me
CH(n-Pr)S(O)Pr-n Me
CH(n-Pr)S(O)Pr-i Me
CH(n-Pr)S(O)Bu-n Me
CH(n-Pr)S(O)Bu-i Me
CH(n-Pr)S(O)Bu-t Me
CH(n-Pr)S(O)Pen-n Me
CH(n-Pr)S(O)Hex-n Me
CH(n-Pr)S(O)Pr-c Me
CH(n-Pr)S(O)Bu-c Me
CH(n-Pr)S(O)Pen-c Me
CH(n-Pr)S(O)Hex-c Me
CH(n-Pr)S(O)CH2CH=CH2 Me
CH(n-Pr)S(O)CH2C三CH Me
CH(n-Pr)S(O)CF2H Me
CH(n-Pr)S(O)CF3 Me
CH(n-Pr)S(O)CF2Cl Me
CH(n-Pr)S(O)CH2CF3 Me
CH(n-Pr)S(O){D1-108c} Me
CH(n-Pr)S(O)2Me Me
CH(n-Pr)S(O)2Et Me
CH(n-Pr)S(O)2Pr-n Me
CH(n-Pr)S(O)2Pr-i Me
CH(n-Pr)S(O)2Bu-n Me
CH(n-Pr)S(O)2Bu-i Me
CH(n-Pr)S(O)2Bu-t Me
CH(n-Pr)S(O)2Pen-n Me
CH(n-Pr)S(O)2Hex-n Me
CH(n-Pr)S(O)2Pr-c Me
CH(n-Pr)S(O)2Bu-c Me
CH(n-Pr)S(O)2Pen-c Me
CH(n-Pr)S(O)2Hex-c Me
CH(n-Pr)S(O)2CH2CH=CH2 Me
CH(n-Pr)S(O)2CH2C三CH Me
CH(n-Pr)S(O)2CF2H Me
CH(n-Pr)S(O)2CF3 Me
CH(n-Pr)S(O)2CF2Cl Me
CH(n-Pr)S(O)2CH2CF3 Me
CH(n-Pr)S(O)2{D1-108c} Me
CH(i-Pr)SH Me
CH(i-Pr)SMe Me
CH(i-Pr)SEt Me
CH(i-Pr)SPr-n Me
CH(i-Pr)SPr-i Me
CH(i-Pr)SBu-n Me
CH(i-Pr)SBu-i Me
CH(i-Pr)SBu-t Me
CH(i-Pr)SPen-n Me
CH(i-Pr)SHex-n Me
CH(i-Pr)SPr-c Me
CH(i-Pr)SBu-c Me
CH(i-Pr)SPen-c Me
CH(i-Pr)SHex-c Me
CH(i-Pr)SCH2CH=CH2 Me
CH(i-Pr)SCH2C三CH Me
CH(i-Pr)SCF2H Me
CH(i-Pr)SCF3 Me
CH(i-Pr)SCF2Cl Me
CH(i-Pr)SCH2CF3 Me
CH(i-Pr)S{D1-108c} Me
CH(i-Pr)S(O)Me Me
CH(i-Pr)S(O)Et Me
CH(i-Pr)S(O)Pr-n Me
CH(i-Pr)S(O)Pr-i Me
CH(i-Pr)S(O)Bu-n Me
CH(i-Pr)S(O)Bu-i Me
CH(i-Pr)S(O)Bu-t Me
CH(i-Pr)S(O)Pen-n Me
CH(i-Pr)S(O)Hex-n Me
CH(i-Pr)S(O)Pr-c Me
CH(i-Pr)S(O)Bu-c Me
CH(i-Pr)S(O)Pen-c Me
CH(i-Pr)S(O)Hex-c Me
CH(i-Pr)S(O)CH2CH=CH2 Me
CH(i-Pr)S(O)CH2C三CH Me
CH(i-Pr)S(O)CF2H Me
CH(i-Pr)S(O)CF3 Me
CH(i-Pr)S(O)CF2Cl Me
CH(i-Pr)S(O)CH2CF3 Me
CH(i-Pr)S(O){D1-108c} Me
CH(i-Pr)S(O)2Me Me
CH(i-Pr)S(O)2Et Me
CH(i-Pr)S(O)2Pr-n Me
CH(i-Pr)S(O)2Pr-i Me
CH(i-Pr)S(O)2Bu-n Me
CH(i-Pr)S(O)2Bu-i Me
CH(i-Pr)S(O)2Bu-t Me
CH(i-Pr)S(O)2Pen-n Me
CH(i-Pr)S(O)2Hex-n Me
CH(i-Pr)S(O)2Pr-c Me
CH(i-Pr)S(O)2Bu-c Me
CH(i-Pr)S(O)2Pen-c Me
CH(i-Pr)S(O)2Hex-c Me
CH(i-Pr)S(O)2CH2CH=CH2 Me
CH(i-Pr)S(O)2CH2C三CH Me
CH(i-Pr)S(O)2CF2H Me
CH(i-Pr)S(O)2CF3 Me
CH(i-Pr)S(O)2CF2Cl Me
CH(i-Pr)S(O)2CH2CF3 Me
CH(i-Pr)S(O)2{D1-108c} Me
CH(n-Bu)SH Me
CH(n-Bu)SMe Me
CH(n-Bu)SEt Me
CH(n-Bu)SPr-n Me
CH(n-Bu)SPr-i Me
CH(n-Bu)SBu-n Me
CH(n-Bu)SBu-i Me
CH(n-Bu)SBu-t Me
CH(n-Bu)SPen-n Me
CH(n-Bu)SHex-n Me
CH(n-Bu)SPr-c Me
CH(n-Bu)SBu-c Me
CH(n-Bu)SPen-c Me
CH(n-Bu)SHex-c Me
CH(n-Bu)SCH2CH=CH2 Me
CH(n-Bu)SCH2C三CH Me
CH(n-Bu)SCF2H Me
CH(n-Bu)SCF3 Me
CH(n-Bu)SCF2Cl Me
CH(n-Bu)SCH2CF3 Me
CH(n-Bu)S{D1-108c} Me
CH(n-Bu)S(O)Me Me
CH(n-Bu)S(O)Et Me
CH(n-Bu)S(O)Pr-n Me
CH(n-Bu)S(O)Pr-i Me
CH(n-Bu)S(O)Bu-n Me
CH(n-Bu)S(O)Bu-i Me
CH(n-Bu)S(O)Bu-t Me
CH(n-Bu)S(O)Pen-n Me
CH(n-Bu)S(O)Hex-n Me
CH(n-Bu)S(O)Pr-c Me
CH(n-Bu)S(O)Bu-c Me
CH(n-Bu)S(O)Pen-c Me
CH(n-Bu)S(O)Hex-c Me
CH(n-Bu)S(O)CH2CH=CH2 Me
CH(n-Bu)S(O)CH2C三CH Me
CH(n-Bu)S(O)CF2H Me
CH(n-Bu)S(O)CF3 Me
CH(n-Bu)S(O)CF2Cl Me
CH(n-Bu)S(O)CH2CF3 Me
CH(n-Bu)S(O){D1-108c} Me
CH(n-Bu)S(O)2Me Me
CH(n-Bu)S(O)2Et Me
CH(n-Bu)S(O)2Pr-n Me
CH(n-Bu)S(O)2Pr-i Me
CH(n-Bu)S(O)2Bu-n Me
CH(n-Bu)S(O)2Bu-i Me
CH(n-Bu)S(O)2Bu-t Me
CH(n-Bu)S(O)2Pen-n Me
CH(n-Bu)S(O)2Hex-n Me
CH(n-Bu)S(O)2Pr-c Me
CH(n-Bu)S(O)2Bu-c Me
CH(n-Bu)S(O)2Pen-c Me
CH(n-Bu)S(O)2Hex-c Me
CH(n-Bu)S(O)2CH2CH=CH2 Me
CH(n-Bu)S(O)2CH2C三CH Me
CH(n-Bu)S(O)2CF2H Me
CH(n-Bu)S(O)2CF3 Me
CH(n-Bu)S(O)2CF2Cl Me
CH(n-Bu)S(O)2CH2CF3 Me
CH(n-Bu)S(O)2{D1-108c} Me
CH(CH2OMe)SH Me
CH(CH2OMe)SMe Me
CH(CH2OMe)SEt Me
CH(CH2OMe)SPr-n Me
CH(CH2OMe)SPr-i Me
CH(CH2OMe)SBu-n Me
CH(CH2OMe)SBu-i Me
CH(CH2OMe)SBu-t Me
CH(CH2OMe)SPen-n Me
CH(CH2OMe)SHex-n Me
CH(CH2OMe)SPr-c Me
CH(CH2OMe)SBu-c Me
CH(CH2OMe)SPen-c Me
CH(CH2OMe)SHex-c Me
CH(CH2OMe)SCH2CH=CH2 Me
CH(CH2OMe)SCH2C三CH Me
CH(CH2OMe)SCF2H Me
CH(CH2OMe)SCF3 Me
CH(CH2OMe)SCF2Cl Me
CH(CH2OMe)SCH2CF3 Me
CH(CH2OMe)S{D1-108c} Me
CH(CH2OMe)SCH2CH2CN Me
CH(CH2OMe)SCH2CH2CF3 Me
CH(CH2OMe)SCH2(D1-103a) Me
CH(CH2OMe)SCH2CH2OMe Me
CH(CH2OMe)SCH2CH2OEt Me
CH(CH2OMe)SCH2(D1-32a) Me
CH(CH2OMe)SCH2(D1-33a) Me
CH(CH2OMe)SCH2(D1-34a) Me
CH(CH2OMe)S{D1-32b(X1=5-CF3)} Me
CH(CH2OMe)SCH2(D1-81a) Me
CH(CH2OMe)SCH2(D1-82a) Me
CH(CH2OMe)SCH2(D1-84a) Me
CH(CH2OMe)SCH2(D1-85a) Me
CH(CH2OMe)SCH2(D1-87a) Me
CH(CH2OMe)SCH2(D1-95a) Me
CH(CH2OMe)SCH2(D1-96a) Me
CH(CH2OMe)SCH2(D1-98a) Me
CH(CH2OMe)SC(O)Me Me
CH(CH2OMe)SC(O)(D1-108a) Me
CH(CH2OMe)S(O)Me Me
CH(CH2OMe)S(O)Et Me
CH(CH2OMe)S(O)Pr-n Me
CH(CH2OMe)S(O)Pr-i Me
CH(CH2OMe)S(O)Bu-n Me
CH(CH2OMe)S(O)Bu-i Me
CH(CH2OMe)S(O)Bu-t Me
CH(CH2OMe)S(O)Pen-n Me
CH(CH2OMe)S(O)Hex-n Me
CH(CH2OMe)S(O)Pr-c Me
CH(CH2OMe)S(O)Bu-c Me
CH(CH2OMe)S(O)Pen-c Me
CH(CH2OMe)S(O)Hex-c Me
CH(CH2OMe)S(O)CH2CH=CH2 Me
CH(CH2OMe)S(O)CH2C三CH Me
CH(CH2OMe)S(O)CF2H Me
CH(CH2OMe)S(O)CF3 Me
CH(CH2OMe)S(O)CF2Cl Me
CH(CH2OMe)S(O)CH2CF3 Me
CH(CH2OMe)S(O){D1-108c} Me
CH(CH2OMe)S(O)CH2CH2CN Me
CH(CH2OMe)S(O)CH2CH2CF3 Me
CH(CH2OMe)S(O)CH2(D1-103a) Me
CH(CH2OMe)S(O)CH2CH2OMe Me
CH(CH2OMe)S(O)CH2CH2OEt Me
CH(CH2OMe)S(O)CH2(D1-32a) Me
CH(CH2OMe)S(O)CH2(D1-33a) Me
CH(CH2OMe)S(O)CH2(D1-34a) Me
CH(CH2OMe)S(O){D1-32b(X1=5-CF3)} Me
CH(CH2OMe)S(O)CH2(D1-81a) Me
CH(CH2OMe)S(O)CH2(D1-82a) Me
CH(CH2OMe)S(O)CH2(D1-84a) Me
CH(CH2OMe)S(O)CH2(D1-85a) Me
CH(CH2OMe)S(O)CH2(D1-87a) Me
CH(CH2OMe)S(O)CH2(D1-95a) Me
CH(CH2OMe)S(O)CH2(D1-96a) Me
CH(CH2OMe)S(O)CH2(D1-98a) Me
CH(CH2OMe)S(O)2Me Me
CH(CH2OMe)S(O)2Et Me
CH(CH2OMe)S(O)2Pr-n Me
CH(CH2OMe)S(O)2Pr-i Me
CH(CH2OMe)S(O)2Bu-n Me
CH(CH2OMe)S(O)2Bu-i Me
CH(CH2OMe)S(O)2Bu-t Me
CH(CH2OMe)S(O)2Pen-n Me
CH(CH2OMe)S(O)2Hex-n Me
CH(CH2OMe)S(O)2Pr-c Me
CH(CH2OMe)S(O)2Bu-c Me
CH(CH2OMe)S(O)2Pen-c Me
CH(CH2OMe)S(O)2Hex-c Me
CH(CH2OMe)S(O)2CH2CH=CH2 Me
CH(CH2OMe)S(O)2CH2C三CH Me
CH(CH2OMe)S(O)2CF2H Me
CH(CH2OMe)S(O)2CF3 Me
CH(CH2OMe)S(O)2CF2Cl Me
CH(CH2OMe)S(O)2CH2CF3 Me
CH(CH2OMe)S(O)2{D1-108c} Me
CH(CH2OMe)S(O)2CH2CH2CN Me
CH(CH2OMe)S(O)2CH2CH2CF3 Me
CH(CH2OMe)S(O)2CH2(D1-103a) Me
CH(CH2OMe)S(O)2CH2CH2OMe Me
CH(CH2OMe)S(O)2CH2CH2OEt Me
CH(CH2OMe)S(O)2CH2(D1-32a) Me
CH(CH2OMe)S(O)2CH2(D1-33a) Me
CH(CH2OMe)S(O)2CH2(D1-34a) Me
CH(CH2OMe)S(O)2{D1-32b(X1=5-CF3)} Me
CH(CH2OMe)S(O)2CH2(D1-81a) Me
CH(CH2OMe)S(O)2CH2(D1-82a) Me
CH(CH2OMe)S(O)2CH2(D1-84a) Me
CH(CH2OMe)S(O)2CH2(D1-85a) Me
CH(CH2OMe)S(O)2CH2(D1-87a) Me
CH(CH2OMe)S(O)2CH2(D1-95a) Me
CH(CH2OMe)S(O)2CH2(D1-96a) Me
CH(CH2OMe)S(O)2CH2(D1-98a) Me
CH(CH2CH=CH2)SH Me
CH(CH2CH=CH2)SMe Me
CH(CH2CH=CH2)SEt Me
CH(CH2CH=CH2)SPr-n Me
CH(CH2CH=CH2)SPr-i Me
CH(CH2CH=CH2)SBu-n Me
CH(CH2CH=CH2)SBu-i Me
CH(CH2CH=CH2)SBu-t Me
CH(CH2CH=CH2)SPen-n Me
CH(CH2CH=CH2)SHex-n Me
CH(CH2CH=CH2)SPr-c Me
CH(CH2CH=CH2)SBu-c Me
CH(CH2CH=CH2)SPen-c Me
CH(CH2CH=CH2)SHex-c Me
CH(CH2CH=CH2)SCH2CH=CH2 Me
CH(CH2CH=CH2)SCH2C三CH Me
CH(CH2CH=CH2)SCF2H Me
CH(CH2CH=CH2)SCF3 Me
CH(CH2CH=CH2)SCF2Cl Me
CH(CH2CH=CH2)SCH2CF3 Me
CH(CH2CH=CH2)S{D1-108c} Me
CH(CH2CH=CH2)SCH2CH2CN Me
CH(CH2CH=CH2)SCH2CH2CF3 Me
CH(CH2CH=CH2)SCH2(D1-103a) Me
CH(CH2CH=CH2)SCH2CH2OMe Me
CH(CH2CH=CH2)SCH2CH2OEt Me
CH(CH2CH=CH2)SCH2(D1-32a) Me
CH(CH2CH=CH2)SCH2(D1-33a) Me
CH(CH2CH=CH2)SCH2(D1-34a) Me
CH(CH2CH=CH2)S{D1-32b(X1=5-CF3)} Me
CH(CH2CH=CH2)SCH2(D1-81a) Me
CH(CH2CH=CH2)SCH2(D1-82a) Me
CH(CH2CH=CH2)SCH2(D1-84a) Me
CH(CH2CH=CH2)SCH2(D1-85a) Me
CH(CH2CH=CH2)SCH2(D1-87a) Me
CH(CH2CH=CH2)SCH2(D1-95a) Me
CH(CH2CH=CH2)SCH2(D1-96a) Me
CH(CH2CH=CH2)SCH2(D1-98a) Me
CH(CH2CH=CH2)SC(O)Me Me
CH(CH2CH=CH2)SC(O)(D1-108a) Me
CH(CH2CH=CH2)S(O)Me Me
CH(CH2CH=CH2)S(O)Et Me
CH(CH2CH=CH2)S(O)Pr-n Me
CH(CH2CH=CH2)S(O)Pr-i Me
CH(CH2CH=CH2)S(O)Bu-n Me
CH(CH2CH=CH2)S(O)Bu-i Me
CH(CH2CH=CH2)S(O)Bu-t Me
CH(CH2CH=CH2)S(O)Pen-n Me
CH(CH2CH=CH2)S(O)Hex-n Me
CH(CH2CH=CH2)S(O)Pr-c Me
CH(CH2CH=CH2)S(O)Bu-c Me
CH(CH2CH=CH2)S(O)Pen-c Me
CH(CH2CH=CH2)S(O)Hex-c Me
CH(CH2CH=CH2)S(O)CH2CH=CH2 Me
CH(CH2CH=CH2)S(O)CH2C三CH Me
CH(CH2CH=CH2)S(O)CF2H Me
CH(CH2CH=CH2)S(O)CF3 Me
CH(CH2CH=CH2)S(O)CF2Cl Me
CH(CH2CH=CH2)S(O)CH2CF3 Me
CH(CH2CH=CH2)S(O){D1-108c} Me
CH(CH2CH=CH2)S(O)CH2CH2CN Me
CH(CH2CH=CH2)S(O)CH2CH2CF3 Me
CH(CH2CH=CH2)S(O)CH2(D1-103a) Me
CH(CH2CH=CH2)S(O)CH2CH2OMe Me
CH(CH2CH=CH2)S(O)CH2CH2OEt Me
CH(CH2CH=CH2)S(O)CH2(D1-32a) Me
CH(CH2CH=CH2)S(O)CH2(D1-33a) Me
CH(CH2CH=CH2)S(O)CH2(D1-34a) Me
CH(CH2CH=CH2)S(O){D1-32b(X1=5-CF3)} Me
CH(CH2CH=CH2)S(O)CH2(D1-81a) Me
CH(CH2CH=CH2)S(O)CH2(D1-82a) Me
CH(CH2CH=CH2)S(O)CH2(D1-84a) Me
CH(CH2CH=CH2)S(O)CH2(D1-85a) Me
CH(CH2CH=CH2)S(O)CH2(D1-87a) Me
CH(CH2CH=CH2)S(O)CH2(D1-95a) Me
CH(CH2CH=CH2)S(O)CH2(D1-96a) Me
CH(CH2CH=CH2)S(O)CH2(D1-98a) Me
CH(CH2CH=CH2)S(O)2Me Me
CH(CH2CH=CH2)S(O)2Et Me
CH(CH2CH=CH2)S(O)2Pr-n Me
CH(CH2CH=CH2)S(O)2Pr-i Me
CH(CH2CH=CH2)S(O)2Bu-n Me
CH(CH2CH=CH2)S(O)2Bu-i Me
CH(CH2CH=CH2)S(O)2Bu-t Me
CH(CH2CH=CH2)S(O)2Pen-n Me
CH(CH2CH=CH2)S(O)2Hex-n Me
CH(CH2CH=CH2)S(O)2Pr-c Me
CH(CH2CH=CH2)S(O)2Bu-c Me
CH(CH2CH=CH2)S(O)2Pen-c Me
CH(CH2CH=CH2)S(O)2Hex-c Me
CH(CH2CH=CH2)S(O)2CH2CH=CH2 Me
CH(CH2CH=CH2)S(O)2CH2C三CH Me
CH(CH2CH=CH2)S(O)2CF2H Me
CH(CH2CH=CH2)S(O)2CF3 Me
CH(CH2CH=CH2)S(O)2CF2Cl Me
CH(CH2CH=CH2)S(O)2CH2CF3 Me
CH(CH2CH=CH2)S(O)2{D1-108c} Me
CH(CH2CH=CH2)S(O)2CH2CH2CN Me
CH(CH2CH=CH2)S(O)2CH2CH2CF3 Me
CH(CH2CH=CH2)S(O)2CH2(D1-103a) Me
CH(CH2CH=CH2)S(O)2CH2CH2OMe Me
CH(CH2CH=CH2)S(O)2CH2CH2OEt Me
CH(CH2CH=CH2)S(O)2CH2(D1-32a) Me
CH(CH2CH=CH2)S(O)2CH2(D1-33a) Me
CH(CH2CH=CH2)S(O)2CH2(D1-34a) Me
CH(CH2CH=CH2)S(O)2{D1-32b(X1=5-CF3)} Me
CH(CH2CH=CH2)S(O)2CH2(D1-81a) Me
CH(CH2CH=CH2)S(O)2CH2(D1-82a) Me
CH(CH2CH=CH2)S(O)2CH2(D1-84a) Me
CH(CH2CH=CH2)S(O)2CH2(D1-85a) Me
CH(CH2CH=CH2)S(O)2CH2(D1-87a) Me
CH(CH2CH=CH2)S(O)2CH2(D1-95a) Me
CH(CH2CH=CH2)S(O)2CH2(D1-96a) Me
CH(CH2CH=CH2)S(O)2CH2(D1-98a) Me
CH(CH2C≡CH)SH Me
CH(CH2C≡CH)SMe Me
CH(CH2C≡CH)SEt Me
CH(CH2C≡CH)SPr-n Me
CH(CH2C≡CH)SPr-i Me
CH(CH2C≡CH)SBu-n Me
CH(CH2C≡CH)SBu-i Me
CH(CH2C≡CH)SBu-t Me
CH(CH2C≡CH)SPen-n Me
CH(CH2C≡CH)SHex-n Me
CH(CH2C≡CH)SPr-c Me
CH(CH2C≡CH)SBu-c Me
CH(CH2C≡CH)SPen-c Me
CH(CH2C≡CH)SHex-c Me
CH(CH2C≡CH)SCH2CH=CH2 Me
CH(CH2C≡CH)SCH2C三CH Me
CH(CH2C≡CH)SCF2H Me
CH(CH2C≡CH)SCF3 Me
CH(CH2C≡CH)SCF2Cl Me
CH(CH2C≡CH)SCH2CF3 Me
CH(CH2C≡CH)S{D1-108c} Me
CH(CH2C≡CH)SCH2CH2CN Me
CH(CH2C≡CH)SCH2CH2CF3 Me
CH(CH2C≡CH)SCH2(D1-103a) Me
CH(CH2C≡CH)SCH2CH2OMe Me
CH(CH2C≡CH)SCH2CH2OEt Me
CH(CH2C≡CH)SCH2(D1-32a) Me
CH(CH2C≡CH)SCH2(D1-33a) Me
CH(CH2C≡CH)SCH2(D1-34a) Me
CH(CH2C≡CH)S{D1-32b(X1=5-CF3)} Me
CH(CH2C≡CH)SCH2(D1-81a) Me
CH(CH2C≡CH)SCH2(D1-82a) Me
CH(CH2C≡CH)SCH2(D1-84a) Me
CH(CH2C≡CH)SCH2(D1-85a) Me
CH(CH2C≡CH)SCH2(D1-87a) Me
CH(CH2C≡CH)SCH2(D1-95a) Me
CH(CH2C≡CH)SCH2(D1-96a) Me
CH(CH2C≡CH)SCH2(D1-98a) Me
CH(CH2C≡CH)SC(O)Me Me
CH(CH2C≡CH)SC(O)(D1-108a) Me
CH(CH2C≡CH)S(O)Me Me
CH(CH2C≡CH)S(O)Et Me
CH(CH2C≡CH)S(O)Pr-n Me
CH(CH2C≡CH)S(O)Pr-i Me
CH(CH2C≡CH)S(O)Bu-n Me
CH(CH2C≡CH)S(O)Bu-i Me
CH(CH2C≡CH)S(O)Bu-t Me
CH(CH2C≡CH)S(O)Pen-n Me
CH(CH2C≡CH)S(O)Hex-n Me
CH(CH2C≡CH)S(O)Pr-c Me
CH(CH2C≡CH)S(O)Bu-c Me
CH(CH2C≡CH)S(O)Pen-c Me
CH(CH2C≡CH)S(O)Hex-c Me
CH(CH2C≡CH)S(O)CH2CH=CH2 Me
CH(CH2C≡CH)S(O)CH2C三CH Me
CH(CH2C≡CH)S(O)CF2H Me
CH(CH2C≡CH)S(O)CF3 Me
CH(CH2C≡CH)S(O)CF2Cl Me
CH(CH2C≡CH)S(O)CH2CF3 Me
CH(CH2C≡CH)S(O){D1-108c} Me
CH(CH2C≡CH)S(O)CH2CH2CN Me
CH(CH2C≡CH)S(O)CH2CH2CF3 Me
CH(CH2C≡CH)S(O)CH2(D1-103a) Me
CH(CH2C≡CH)S(O)CH2CH2OMe Me
CH(CH2C≡CH)S(O)CH2CH2OEt Me
CH(CH2C≡CH)S(O)CH2(D1-32a) Me
CH(CH2C≡CH)S(O)CH2(D1-33a) Me
CH(CH2C≡CH)S(O)CH2(D1-34a) Me
CH(CH2C≡CH)S(O){D1-32b(X1=5-CF3)} Me
CH(CH2C≡CH)S(O)CH2(D1-81a) Me
CH(CH2C≡CH)S(O)CH2(D1-82a) Me
CH(CH2C≡CH)S(O)CH2(D1-84a) Me
CH(CH2C≡CH)S(O)CH2(D1-85a) Me
CH(CH2C≡CH)S(O)CH2(D1-87a) Me
CH(CH2C≡CH)S(O)CH2(D1-95a) Me
CH(CH2C≡CH)S(O)CH2(D1-96a) Me
CH(CH2C≡CH)S(O)CH2(D1-98a) Me
CH(CH2C≡CH)S(O)2Me Me
CH(CH2C≡CH)S(O)2Et Me
CH(CH2C≡CH)S(O)2Pr-n Me
CH(CH2C≡CH)S(O)2Pr-i Me
CH(CH2C≡CH)S(O)2Bu-n Me
CH(CH2C≡CH)S(O)2Bu-i Me
CH(CH2C≡CH)S(O)2Bu-t Me
CH(CH2C≡CH)S(O)2Pen-n Me
CH(CH2C≡CH)S(O)2Hex-n Me
CH(CH2C≡CH)S(O)2Pr-c Me
CH(CH2C≡CH)S(O)2Bu-c Me
CH(CH2C≡CH)S(O)2Pen-c Me
CH(CH2C≡CH)S(O)2Hex-c Me
CH(CH2C≡CH)S(O)2CH2CH=CH2 Me
CH(CH2C≡CH)S(O)2CH2C三CH Me
CH(CH2C≡CH)S(O)2CF2H Me
CH(CH2C≡CH)S(O)2CF3 Me
CH(CH2C≡CH)S(O)2CF2Cl Me
CH(CH2C≡CH)S(O)2CH2CF3 Me
CH(CH2C≡CH)S(O)2{D1-108c} Me
CH(CH2C≡CH)S(O)2CH2CH2CN Me
CH(CH2C≡CH)S(O)2CH2CH2CF3 Me
CH(CH2C≡CH)S(O)2CH2(D1-103a) Me
CH(CH2C≡CH)S(O)2CH2CH2OMe Me
CH(CH2C≡CH)S(O)2CH2CH2OEt Me
CH(CH2C≡CH)S(O)2CH2(D1-32a) Me
CH(CH2C≡CH)S(O)2CH2(D1-33a) Me
CH(CH2C≡CH)S(O)2CH2(D1-34a) Me
CH(CH2C≡CH)S(O)2{D1-32b(X1=5-CF3)} Me
CH(CH2C≡CH)S(O)2CH2(D1-81a) Me
CH(CH2C≡CH)S(O)2CH2(D1-82a) Me
CH(CH2C≡CH)S(O)2CH2(D1-84a) Me
CH(CH2C≡CH)S(O)2CH2(D1-85a) Me
CH(CH2C≡CH)S(O)2CH2(D1-87a) Me
CH(CH2C≡CH)S(O)2CH2(D1-95a) Me
CH(CH2C≡CH)S(O)2CH2(D1-96a) Me
CH(CH2C≡CH)S(O)2CH2(D1-98a) Me
CH(CH2CN)SH Me
CH(CH2CN)SMe Me
CH(CH2CN)SEt Me
CH(CH2CN)SPr-n Me
CH(CH2CN)SPr-i Me
CH(CH2CN)SBu-n Me
CH(CH2CN)SBu-i Me
CH(CH2CN)SBu-t Me
CH(CH2CN)SPen-n Me
CH(CH2CN)SHex-n Me
CH(CH2CN)SPr-c Me
CH(CH2CN)SBu-c Me
CH(CH2CN)SPen-c Me
CH(CH2CN)SHex-c Me
CH(CH2CN)SCH2CH=CH2 Me
CH(CH2CN)SCH2C三CH Me
CH(CH2CN)SCF2H Me
CH(CH2CN)SCF3 Me
CH(CH2CN)SCF2Cl Me
CH(CH2CN)SCH2CF3 Me
CH(CH2CN)S{D1-108c} Me
CH(CH2CN)SCH2CH2CN Me
CH(CH2CN)SCH2CH2CF3 Me
CH(CH2CN)SCH2(D1-103a) Me
CH(CH2CN)SCH2CH2OMe Me
CH(CH2CN)SCH2CH2OEt Me
CH(CH2CN)SCH2(D1-32a) Me
CH(CH2CN)SCH2(D1-33a) Me
CH(CH2CN)SCH2(D1-34a) Me
CH(CH2CN)S{D1-32b(X1=5-CF3)} Me
CH(CH2CN)SCH2(D1-81a) Me
CH(CH2CN)SCH2(D1-82a) Me
CH(CH2CN)SCH2(D1-84a) Me
CH(CH2CN)SCH2(D1-85a) Me
CH(CH2CN)SCH2(D1-87a) Me
CH(CH2CN)SCH2(D1-95a) Me
CH(CH2CN)SCH2(D1-96a) Me
CH(CH2CN)SCH2(D1-98a) Me
CH(CH2CN)SC(O)Me Me
CH(CH2CN)SC(O)(D1-108a) Me
CH(CH2CN)S(O)Me Me
CH(CH2CN)S(O)Et Me
CH(CH2CN)S(O)Pr-n Me
CH(CH2CN)S(O)Pr-i Me
CH(CH2CN)S(O)Bu-n Me
CH(CH2CN)S(O)Bu-i Me
CH(CH2CN)S(O)Bu-t Me
CH(CH2CN)S(O)Pen-n Me
CH(CH2CN)S(O)Hex-n Me
CH(CH2CN)S(O)Pr-c Me
CH(CH2CN)S(O)Bu-c Me
CH(CH2CN)S(O)Pen-c Me
CH(CH2CN)S(O)Hex-c Me
CH(CH2CN)S(O)CH2CH=CH2 Me
CH(CH2CN)S(O)CH2C三CH Me
CH(CH2CN)S(O)CF2H Me
CH(CH2CN)S(O)CF3 Me
CH(CH2CN)S(O)CF2Cl Me
CH(CH2CN)S(O)CH2CF3 Me
CH(CH2CN)S(O){D1-108c} Me
CH(CH2CN)S(O)CH2CH2CN Me
CH(CH2CN)S(O)CH2CH2CF3 Me
CH(CH2CN)S(O)CH2(D1-103a) Me
CH(CH2CN)S(O)CH2CH2OMe Me
CH(CH2CN)S(O)CH2CH2OEt Me
CH(CH2CN)S(O)CH2(D1-32a) Me
CH(CH2CN)S(O)CH2(D1-33a) Me
CH(CH2CN)S(O)CH2(D1-34a) Me
CH(CH2CN)S(O){D1-32b(X1=5-CF3)} Me
CH(CH2CN)S(O)CH2(D1-81a) Me
CH(CH2CN)S(O)CH2(D1-82a) Me
CH(CH2CN)S(O)CH2(D1-84a) Me
CH(CH2CN)S(O)CH2(D1-85a) Me
CH(CH2CN)S(O)CH2(D1-87a) Me
CH(CH2CN)S(O)CH2(D1-95a) Me
CH(CH2CN)S(O)CH2(D1-96a) Me
CH(CH2CN)S(O)CH2(D1-98a) Me
CH(CH2CN)S(O)2Me Me
CH(CH2CN)S(O)2Et Me
CH(CH2CN)S(O)2Pr-n Me
CH(CH2CN)S(O)2Pr-i Me
CH(CH2CN)S(O)2Bu-n Me
CH(CH2CN)S(O)2Bu-i Me
CH(CH2CN)S(O)2Bu-t Me
CH(CH2CN)S(O)2Pen-n Me
CH(CH2CN)S(O)2Hex-n Me
CH(CH2CN)S(O)2Pr-c Me
CH(CH2CN)S(O)2Bu-c Me
CH(CH2CN)S(O)2Pen-c Me
CH(CH2CN)S(O)2Hex-c Me
CH(CH2CN)S(O)2CH2CH=CH2 Me
CH(CH2CN)S(O)2CH2C三CH Me
CH(CH2CN)S(O)2CF2H Me
CH(CH2CN)S(O)2CF3 Me
CH(CH2CN)S(O)2CF2Cl Me
CH(CH2CN)S(O)2CH2CF3 Me
CH(CH2CN)S(O)2{D1-108c} Me
CH(CH2CN)S(O)2CH2CH2CN Me
CH(CH2CN)S(O)2CH2CH2CF3 Me
CH(CH2CN)S(O)2CH2(D1-103a) Me
CH(CH2CN)S(O)2CH2CH2OMe Me
CH(CH2CN)S(O)2CH2CH2OEt Me
CH(CH2CN)S(O)2CH2(D1-32a) Me
CH(CH2CN)S(O)2CH2(D1-33a) Me
CH(CH2CN)S(O)2CH2(D1-34a) Me
CH(CH2CN)S(O)2{D1-32b(X1=5-CF3)} Me
CH(CH2CN)S(O)2CH2(D1-81a) Me
CH(CH2CN)S(O)2CH2(D1-82a) Me
CH(CH2CN)S(O)2CH2(D1-84a) Me
CH(CH2CN)S(O)2CH2(D1-85a) Me
CH(CH2CN)S(O)2CH2(D1-87a) Me
CH(CH2CN)S(O)2CH2(D1-95a) Me
CH(CH2CN)S(O)2CH2(D1-96a) Me
CH(CH2CN)S(O)2CH2(D1-98a) Me
CH(Me)2SH Me
CH(Me)2SMe Me
CH(Me)2SEt Me
CH(Me)2SPr-n Me
CH(Me)2SPr-i Me
CH(Me)2SBu-n Me
CH(Me)2SBu-i Me
CH(Me)2SBu-t Me
CH(Me)2SPen-n Me
CH(Me)2SHex-n Me
CH(Me)2SPr-c Me
CH(Me)2SBu-c Me
CH(Me)2SPen-c Me
CH(Me)2SHex-c Me
CH(Me)2SCH2CH=CH2 Me
CH(Me)2SCH2C三CH Me
CH(Me)2SCF2H Me
CH(Me)2SCF3 Me
CH(Me)2SCF2Cl Me
CH(Me)2SCH2CF3 Me
CH(Me)2S{D1-108c} Me
CH(Me)2SCH2CH2CN Me
CH(Me)2SCH2CH2CF3 Me
CH(Me)2SCH2(D1-103a) Me
CH(Me)2SCH2CH2OMe Me
CH(Me)2SCH2CH2OEt Me
CH(Me)2SCH2(D1-32a) Me
CH(Me)2SCH2(D1-33a) Me
CH(Me)2SCH2(D1-34a) Me
CH(Me)2S{D1-32b(X1=5-CF3)} Me
CH(Me)2SCH2(D1-81a) Me
CH(Me)2SCH2(D1-82a) Me
CH(Me)2SCH2(D1-84a) Me
CH(Me)2SCH2(D1-85a) Me
CH(Me)2SCH2(D1-87a) Me
CH(Me)2SCH2(D1-95a) Me
CH(Me)2SCH2(D1-96a) Me
CH(Me)2SCH2(D1-98a) Me
CH(Me)2SC(O)Me Me
CH(Me)2SC(O)(D1-108a) Me
CH(Me)2S(O)Me Me
CH(Me)2S(O)Et Me
CH(Me)2S(O)Pr-n Me
CH(Me)2S(O)Pr-i Me
CH(Me)2S(O)Bu-n Me
CH(Me)2S(O)Bu-i Me
CH(Me)2S(O)Bu-t Me
CH(Me)2S(O)Pen-n Me
CH(Me)2S(O)Hex-n Me
CH(Me)2S(O)Pr-c Me
CH(Me)2S(O)Bu-c Me
CH(Me)2S(O)Pen-c Me
CH(Me)2S(O)Hex-c Me
CH(Me)2S(O)CH2CH=CH2 Me
CH(Me)2S(O)CH2C三CH Me
CH(Me)2S(O)CF2H Me
CH(Me)2S(O)CF3 Me
CH(Me)2S(O)CF2Cl Me
CH(Me)2S(O)CH2CF3 Me
CH(Me)2S(O){D1-108c} Me
CH(Me)2S(O)CH2CH2CN Me
CH(Me)2S(O)CH2CH2CF3 Me
CH(Me)2S(O)CH2(D1-103a) Me
CH(Me)2S(O)CH2CH2OMe Me
CH(Me)2S(O)CH2CH2OEt Me
CH(Me)2S(O)CH2(D1-32a) Me
CH(Me)2S(O)CH2(D1-33a) Me
CH(Me)2S(O)CH2(D1-34a) Me
CH(Me)2S(O){D1-32b(X1=5-CF3)} Me
CH(Me)2S(O)CH2(D1-81a) Me
CH(Me)2S(O)CH2(D1-82a) Me
CH(Me)2S(O)CH2(D1-84a) Me
CH(Me)2S(O)CH2(D1-85a) Me
CH(Me)2S(O)CH2(D1-87a) Me
CH(Me)2S(O)CH2(D1-95a) Me
CH(Me)2S(O)CH2(D1-96a) Me
CH(Me)2S(O)CH2(D1-98a) Me
CH(Me)2S(O)2Me Me
CH(Me)2S(O)2Et Me
CH(Me)2S(O)2Pr-n Me
CH(Me)2S(O)2Pr-i Me
CH(Me)2S(O)2Bu-n Me
CH(Me)2S(O)2Bu-i Me
CH(Me)2S(O)2Bu-t Me
CH(Me)2S(O)2Pen-n Me
CH(Me)2S(O)2Hex-n Me
CH(Me)2S(O)2Pr-c Me
CH(Me)2S(O)2Bu-c Me
CH(Me)2S(O)2Pen-c Me
CH(Me)2S(O)2Hex-c Me
CH(Me)2S(O)2CH2CH=CH2 Me
CH(Me)2S(O)2CH2C三CH Me
CH(Me)2S(O)2CF2H Me
CH(Me)2S(O)2CF3 Me
CH(Me)2S(O)2CF2Cl Me
CH(Me)2S(O)2CH2CF3 Me
CH(Me)2S(O)2{D1-108c} Me
CH(Me)2S(O)2CH2CH2CN Me
CH(Me)2S(O)2CH2CH2CF3 Me
CH(Me)2S(O)2CH2(D1-103a) Me
CH(Me)2S(O)2CH2CH2OMe Me
CH(Me)2S(O)2CH2CH2OEt Me
CH(Me)2S(O)2CH2(D1-32a) Me
CH(Me)2S(O)2CH2(D1-33a) Me
CH(Me)2S(O)2CH2(D1-34a) Me
CH(Me)2S(O)2{D1-32b(X1=5-CF3)} Me
CH(Me)2S(O)2CH2(D1-81a) Me
CH(Me)2S(O)2CH2(D1-82a) Me
CH(Me)2S(O)2CH2(D1-84a) Me
CH(Me)2S(O)2CH2(D1-85a) Me
CH(Me)2S(O)2CH2(D1-87a) Me
CH(Me)2S(O)2CH2(D1-95a) Me
CH(Me)2S(O)2CH2(D1-96a) Me
CH(Me)2S(O)2CH2(D1-98a) Me
CH2CH2SH Me
CH2CH2SMe Me
CH2CH2SEt Me
CH2CH2SPr-n Me
CH2CH2SPr-i Me
CH2CH2SBu-n Me
CH2CH2SBu-i Me
CH2CH2SBu-t Me
CH2CH2SPen-n Me
CH2CH2SHex-n Me
CH2CH2SPr-c Me
CH2CH2SBu-c Me
CH2CH2SPen-c Me
CH2CH2SHex-c Me
CH2CH2SCH2CH=CH2 Me
CH2CH2SCH2C三CH Me
CH2CH2SCF2H Me
CH2CH2SCF3 Me
CH2CH2SCF2Cl Me
CH2CH2SCH2CF3 Me
CH2CH2S{D1-108c} Me
CH2CH2SCH2CH2CN Me
CH2CH2SCH2CH2CF3 Me
CH2CH2SCH2(D1-103a) Me
CH2CH2SCH2CH2OMe Me
CH2CH2SCH2CH2OEt Me
CH2CH2SCH2(D1-32a) Me
CH2CH2SCH2(D1-33a) Me
CH2CH2SCH2(D1-34a) Me
CH2CH2S{D1-32b(X1=5-CF3)} Me
CH2CH2SCH2(D1-81a) Me
CH2CH2SCH2(D1-82a) Me
CH2CH2SCH2(D1-84a) Me
CH2CH2SCH2(D1-85a) Me
CH2CH2SCH2(D1-87a) Me
CH2CH2SCH2(D1-95a) Me
CH2CH2SCH2(D1-96a) Me
CH2CH2SCH2(D1-98a) Me
CH2CH2SC(O)Me Me
CH2CH2SC(O)(D1-108a) Me
CH2CH2S(O)Me Me
CH2CH2S(O)Et Me
CH2CH2S(O)Pr-n Me
CH2CH2S(O)Pr-i Me
CH2CH2S(O)Bu-n Me
CH2CH2S(O)Bu-i Me
CH2CH2S(O)Bu-t Me
CH2CH2S(O)Pen-n Me
CH2CH2S(O)Hex-n Me
CH2CH2S(O)Pr-c Me
CH2CH2S(O)Bu-c Me
CH2CH2S(O)Pen-c Me
CH2CH2S(O)Hex-c Me
CH2CH2S(O)CH2CH=CH2 Me
CH2CH2S(O)CH2C三CH Me
CH2CH2S(O)CF2H Me
CH2CH2S(O)CF3 Me
CH2CH2S(O)CF2Cl Me
CH2CH2S(O)CH2CF3 Me
CH2CH2S(O){D1-108c} Me
CH2CH2S(O)CH2CH2CN Me
CH2CH2S(O)CH2CH2CF3 Me
CH2CH2S(O)CH2(D1-103a) Me
CH2CH2S(O)CH2CH2OMe Me
CH2CH2S(O)CH2CH2OEt Me
CH2CH2S(O)CH2(D1-32a) Me
CH2CH2S(O)CH2(D1-33a) Me
CH2CH2S(O)CH2(D1-34a) Me
CH2CH2S(O){D1-32b(X1=5-CF3)} Me
CH2CH2S(O)CH2(D1-81a) Me
CH2CH2S(O)CH2(D1-82a) Me
CH2CH2S(O)CH2(D1-84a) Me
CH2CH2S(O)CH2(D1-85a) Me
CH2CH2S(O)CH2(D1-87a) Me
CH2CH2S(O)CH2(D1-95a) Me
CH2CH2S(O)CH2(D1-96a) Me
CH2CH2S(O)CH2(D1-98a) Me
CH2CH2S(O)2Me Me
CH2CH2S(O)2Et Me
CH2CH2S(O)2Pr-n Me
CH2CH2S(O)2Pr-i Me
CH2CH2S(O)2Bu-n Me
CH2CH2S(O)2Bu-i Me
CH2CH2S(O)2Bu-t Me
CH2CH2S(O)2Pen-n Me
CH2CH2S(O)2Hex-n Me
CH2CH2S(O)2Pr-c Me
CH2CH2S(O)2Bu-c Me
CH2CH2S(O)2Pen-c Me
CH2CH2S(O)2Hex-c Me
CH2CH2S(O)2CH2CH=CH2 Me
CH2CH2S(O)2CH2C三CH Me
CH2CH2S(O)2CF2H Me
CH2CH2S(O)2CF3 Me
CH2CH2S(O)2CF2Cl Me
CH2CH2S(O)2CH2CF3 Me
CH2CH2S(O)2{D1-108c} Me
CH2CH2S(O)2CH2CH2CN Me
CH2CH2S(O)2CH2CH2CF3 Me
CH2CH2S(O)2CH2(D1-103a) Me
CH2CH2S(O)2CH2CH2OMe Me
CH2CH2S(O)2CH2CH2OEt Me
CH2CH2S(O)2CH2(D1-32a) Me
CH2CH2S(O)2CH2(D1-33a) Me
CH2CH2S(O)2CH2(D1-34a) Me
CH2CH2S(O)2{D1-32b(X1=5-CF3)} Me
CH2CH2S(O)2CH2(D1-81a) Me
CH2CH2S(O)2CH2(D1-82a) Me
CH2CH2S(O)2CH2(D1-84a) Me
CH2CH2S(O)2CH2(D1-85a) Me
CH2CH2S(O)2CH2(D1-87a) Me
CH2CH2S(O)2CH2(D1-95a) Me
CH2CH2S(O)2CH2(D1-96a) Me
CH2CH2S(O)2CH2(D1-98a) Me
CH(Me)CH2SH Me
CH(Me)CH2SMe Me
CH(Me)CH2SEt Me
CH(Me)CH2SPr-n Me
CH(Me)CH2SPr-i Me
CH(Me)CH2SBu-n Me
CH(Me)CH2SBu-i Me
CH(Me)CH2SBu-t Me
CH(Me)CH2SPen-n Me
CH(Me)CH2SHex-n Me
CH(Me)CH2SPr-c Me
CH(Me)CH2SBu-c Me
CH(Me)CH2SPen-c Me
CH(Me)CH2SHex-c Me
CH(Me)CH2SCH2CH=CH2 Me
CH(Me)CH2SCH2C三CH Me
CH(Me)CH2SCF2H Me
CH(Me)CH2SCF3 Me
CH(Me)CH2SCF2Cl Me
CH(Me)CH2SCH2CF3 Me
CH(Me)CH2S{D1-108c} Me
CH(Me)CH2SCH2CH2CN Me
CH(Me)CH2SCH2CH2CF3 Me
CH(Me)CH2SCH2(D1-103a) Me
CH(Me)CH2SCH2CH2OMe Me
CH(Me)CH2SCH2CH2OEt Me
CH(Me)CH2SCH2(D1-32a) Me
CH(Me)CH2SCH2(D1-33a) Me
CH(Me)CH2SCH2(D1-34a) Me
CH(Me)CH2S{D1-32b(X1=5-CF3)} Me
CH(Me)CH2SCH2(D1-81a) Me
CH(Me)CH2SCH2(D1-82a) Me
CH(Me)CH2SCH2(D1-84a) Me
CH(Me)CH2SCH2(D1-85a) Me
CH(Me)CH2SCH2(D1-87a) Me
CH(Me)CH2SCH2(D1-95a) Me
CH(Me)CH2SCH2(D1-96a) Me
CH(Me)CH2SCH2(D1-98a) Me
CH(Me)CH2SC(O)Me Me
CH(Me)CH2SC(O)(D1-108a) Me
CH(Me)CH2S(O)Me Me
CH(Me)CH2S(O)Et Me
CH(Me)CH2S(O)Pr-n Me
CH(Me)CH2S(O)Pr-i Me
CH(Me)CH2S(O)Bu-n Me
CH(Me)CH2S(O)Bu-i Me
CH(Me)CH2S(O)Bu-t Me
CH(Me)CH2S(O)Pen-n Me
CH(Me)CH2S(O)Hex-n Me
CH(Me)CH2S(O)Pr-c Me
CH(Me)CH2S(O)Bu-c Me
CH(Me)CH2S(O)Pen-c Me
CH(Me)CH2S(O)Hex-c Me
CH(Me)CH2S(O)CH2CH=CH2 Me
CH(Me)CH2S(O)CH2C三CH Me
CH(Me)CH2S(O)CF2H Me
CH(Me)CH2S(O)CF3 Me
CH(Me)CH2S(O)CF2Cl Me
CH(Me)CH2S(O)CH2CF3 Me
CH(Me)CH2S(O){D1-108c} Me
CH(Me)CH2S(O)CH2CH2CN Me
CH(Me)CH2S(O)CH2CH2CF3 Me
CH(Me)CH2S(O)CH2(D1-103a) Me
CH(Me)CH2S(O)CH2CH2OMe Me
CH(Me)CH2S(O)CH2CH2OEt Me
CH(Me)CH2S(O)CH2(D1-32a) Me
CH(Me)CH2S(O)CH2(D1-33a) Me
CH(Me)CH2S(O)CH2(D1-34a) Me
CH(Me)CH2S(O){D1-32b(X1=5-CF3)} Me
CH(Me)CH2S(O)CH2(D1-81a) Me
CH(Me)CH2S(O)CH2(D1-82a) Me
CH(Me)CH2S(O)CH2(D1-84a) Me
CH(Me)CH2S(O)CH2(D1-85a) Me
CH(Me)CH2S(O)CH2(D1-87a) Me
CH(Me)CH2S(O)CH2(D1-95a) Me
CH(Me)CH2S(O)CH2(D1-96a) Me
CH(Me)CH2S(O)CH2(D1-98a) Me
CH(Me)CH2S(O)2Me Me
CH(Me)CH2S(O)2Et Me
CH(Me)CH2S(O)2Pr-n Me
CH(Me)CH2S(O)2Pr-i Me
CH(Me)CH2S(O)2Bu-n Me
CH(Me)CH2S(O)2Bu-i Me
CH(Me)CH2S(O)2Bu-t Me
CH(Me)CH2S(O)2Pen-n Me
CH(Me)CH2S(O)2Hex-n Me
CH(Me)CH2S(O)2Pr-c Me
CH(Me)CH2S(O)2Bu-c Me
CH(Me)CH2S(O)2Pen-c Me
CH(Me)CH2S(O)2Hex-c Me
CH(Me)CH2S(O)2CH2CH=CH2 Me
CH(Me)CH2S(O)2CH2C三CH Me
CH(Me)CH2S(O)2CF2H Me
CH(Me)CH2S(O)2CF3 Me
CH(Me)CH2S(O)2CF2Cl Me
CH(Me)CH2S(O)2CH2CF3 Me
CH(Me)CH2S(O)2{D1-108c} Me
CH(Me)CH2S(O)2CH2CH2CN Me
CH(Me)CH2S(O)2CH2CH2CF3 Me
CH(Me)CH2S(O)2CH2(D1-103a) Me
CH(Me)CH2S(O)2CH2CH2OMe Me
CH(Me)CH2S(O)2CH2CH2OEt Me
CH(Me)CH2S(O)2CH2(D1-32a) Me
CH(Me)CH2S(O)2CH2(D1-33a) Me
CH(Me)CH2S(O)2CH2(D1-34a) Me
CH(Me)CH2S(O)2{D1-32b(X1=5-CF3)} Me
CH(Me)CH2S(O)2CH2(D1-81a) Me
CH(Me)CH2S(O)2CH2(D1-82a) Me
CH(Me)CH2S(O)2CH2(D1-84a) Me
CH(Me)CH2S(O)2CH2(D1-85a) Me
CH(Me)CH2S(O)2CH2(D1-87a) Me
CH(Me)CH2S(O)2CH2(D1-95a) Me
CH(Me)CH2S(O)2CH2(D1-96a) Me
CH(Me)CH2S(O)2CH2(D1-98a) Me
CH(Me)CH(Me)SH Me
CH(Me)CH(Me)SMe Me
CH(Me)CH(Me)SEt Me
CH(Me)CH(Me)SPr-n Me
CH(Me)CH(Me)SPr-i Me
CH(Me)CH(Me)SBu-n Me
CH(Me)CH(Me)SBu-i Me
CH(Me)CH(Me)SBu-t Me
CH(Me)CH(Me)SPen-n Me
CH(Me)CH(Me)SHex-n Me
CH(Me)CH(Me)SPr-c Me
CH(Me)CH(Me)SBu-c Me
CH(Me)CH(Me)SPen-c Me
CH(Me)CH(Me)SHex-c Me
CH(Me)CH(Me)SCH2CH=CH2 Me
CH(Me)CH(Me)SCH2C三CH Me
CH(Me)CH(Me)SCF2H Me
CH(Me)CH(Me)SCF3 Me
CH(Me)CH(Me)SCF2Cl Me
CH(Me)CH(Me)SCH2CF3 Me
CH(Me)CH(Me)S{D1-108c} Me
CH(Me)CH(Me)SCH2CH2CN Me
CH(Me)CH(Me)SCH2CH2CF3 Me
CH(Me)CH(Me)SCH2(D1-103a) Me
CH(Me)CH(Me)SCH2CH2OMe Me
CH(Me)CH(Me)SCH2CH2OEt Me
CH(Me)CH(Me)SCH2(D1-32a) Me
CH(Me)CH(Me)SCH2(D1-33a) Me
CH(Me)CH(Me)SCH2(D1-34a) Me
CH(Me)CH(Me)S{D1-32b(X1=5-CF3)} Me
CH(Me)CH(Me)SCH2(D1-81a) Me
CH(Me)CH(Me)SCH2(D1-82a) Me
CH(Me)CH(Me)SCH2(D1-84a) Me
CH(Me)CH(Me)SCH2(D1-85a) Me
CH(Me)CH(Me)SCH2(D1-87a) Me
CH(Me)CH(Me)SCH2(D1-95a) Me
CH(Me)CH(Me)SCH2(D1-96a) Me
CH(Me)CH(Me)SCH2(D1-98a) Me
CH(Me)CH(Me)SC(O)Me Me
CH(Me)CH(Me)SC(O)(D1-108a) Me
CH(Me)CH(Me)S(O)Me Me
CH(Me)CH(Me)S(O)Et Me
CH(Me)CH(Me)S(O)Pr-n Me
CH(Me)CH(Me)S(O)Pr-i Me
CH(Me)CH(Me)S(O)Bu-n Me
CH(Me)CH(Me)S(O)Bu-i Me
CH(Me)CH(Me)S(O)Bu-t Me
CH(Me)CH(Me)S(O)Pen-n Me
CH(Me)CH(Me)S(O)Hex-n Me
CH(Me)CH(Me)S(O)Pr-c Me
CH(Me)CH(Me)S(O)Bu-c Me
CH(Me)CH(Me)S(O)Pen-c Me
CH(Me)CH(Me)S(O)Hex-c Me
CH(Me)CH(Me)S(O)CH2CH=CH2 Me
CH(Me)CH(Me)S(O)CH2C三CH Me
CH(Me)CH(Me)S(O)CF2H Me
CH(Me)CH(Me)S(O)CF3 Me
CH(Me)CH(Me)S(O)CF2Cl Me
CH(Me)CH(Me)S(O)CH2CF3 Me
CH(Me)CH(Me)S(O){D1-108c} Me
CH(Me)CH(Me)S(O)CH2CH2CN Me
CH(Me)CH(Me)S(O)CH2CH2CF3 Me
CH(Me)CH(Me)S(O)CH2(D1-103a) Me
CH(Me)CH(Me)S(O)CH2CH2OMe Me
CH(Me)CH(Me)S(O)CH2CH2OEt Me
CH(Me)CH(Me)S(O)CH2(D1-32a) Me
CH(Me)CH(Me)S(O)CH2(D1-33a) Me
CH(Me)CH(Me)S(O)CH2(D1-34a) Me
CH(Me)CH(Me)S(O){D1-32b(X1=5-CF3)} Me
CH(Me)CH(Me)S(O)CH2(D1-81a) Me
CH(Me)CH(Me)S(O)CH2(D1-82a) Me
CH(Me)CH(Me)S(O)CH2(D1-84a) Me
CH(Me)CH(Me)S(O)CH2(D1-85a) Me
CH(Me)CH(Me)S(O)CH2(D1-87a) Me
CH(Me)CH(Me)S(O)CH2(D1-95a) Me
CH(Me)CH(Me)S(O)CH2(D1-96a) Me
CH(Me)CH(Me)S(O)CH2(D1-98a) Me
CH(Me)CH(Me)S(O)2Me Me
CH(Me)CH(Me)S(O)2Et Me
CH(Me)CH(Me)S(O)2Pr-n Me
CH(Me)CH(Me)S(O)2Pr-i Me
CH(Me)CH(Me)S(O)2Bu-n Me
CH(Me)CH(Me)S(O)2Bu-i Me
CH(Me)CH(Me)S(O)2Bu-t Me
CH(Me)CH(Me)S(O)2Pen-n Me
CH(Me)CH(Me)S(O)2Hex-n Me
CH(Me)CH(Me)S(O)2Pr-c Me
CH(Me)CH(Me)S(O)2Bu-c Me
CH(Me)CH(Me)S(O)2Pen-c Me
CH(Me)CH(Me)S(O)2Hex-c Me
CH(Me)CH(Me)S(O)2CH2CH=CH2 Me
CH(Me)CH(Me)S(O)2CH2C三CH Me
CH(Me)CH(Me)S(O)2CF2H Me
CH(Me)CH(Me)S(O)2CF3 Me
CH(Me)CH(Me)S(O)2CF2Cl Me
CH(Me)CH(Me)S(O)2CH2CF3 Me
CH(Me)CH(Me)S(O)2{D1-108c} Me
CH(Me)CH(Me)S(O)2CH2CH2CN Me
CH(Me)CH(Me)S(O)2CH2CH2CF3 Me
CH(Me)CH(Me)S(O)2CH2(D1-103a) Me
CH(Me)CH(Me)S(O)2CH2CH2OMe Me
CH(Me)CH(Me)S(O)2CH2CH2OEt Me
CH(Me)CH(Me)S(O)2CH2(D1-32a) Me
CH(Me)CH(Me)S(O)2CH2(D1-33a) Me
CH(Me)CH(Me)S(O)2CH2(D1-34a) Me
CH(Me)CH(Me)S(O)2{D1-32b(X1=5-CF3)} Me
CH(Me)CH(Me)S(O)2CH2(D1-81a) Me
CH(Me)CH(Me)S(O)2CH2(D1-82a) Me
CH(Me)CH(Me)S(O)2CH2(D1-84a) Me
CH(Me)CH(Me)S(O)2CH2(D1-85a) Me
CH(Me)CH(Me)S(O)2CH2(D1-87a) Me
CH(Me)CH(Me)S(O)2CH2(D1-95a) Me
CH(Me)CH(Me)S(O)2CH2(D1-96a) Me
CH(Me)CH(Me)S(O)2CH2(D1-98a) Me
CH2CH(Me)SH Me
CH2CH(Me)SMe Me
CH2CH(Me)SEt Me
CH2CH(Me)SPr-n Me
CH2CH(Me)SPr-i Me
CH2CH(Me)SBu-n Me
CH2CH(Me)SBu-i Me
CH2CH(Me)SBu-t Me
CH2CH(Me)SPen-n Me
CH2CH(Me)SHex-n Me
CH2CH(Me)SPr-c Me
CH2CH(Me)SBu-c Me
CH2CH(Me)SPen-c Me
CH2CH(Me)SHex-c Me
CH2CH(Me)SCH2CH=CH2 Me
CH2CH(Me)SCH2C三CH Me
CH2CH(Me)SCF2H Me
CH2CH(Me)SCF3 Me
CH2CH(Me)SCF2Cl Me
CH2CH(Me)SCH2CF3 Me
CH2CH(Me)S{D1-108c} Me
CH2CH(Me)SCH2CH2CN Me
CH2CH(Me)SCH2CH2CF3 Me
CH2CH(Me)SCH2(D1-103a) Me
CH2CH(Me)SCH2CH2OMe Me
CH2CH(Me)SCH2CH2OEt Me
CH2CH(Me)SCH2(D1-32a) Me
CH2CH(Me)SCH2(D1-33a) Me
CH2CH(Me)SCH2(D1-34a) Me
CH2CH(Me)S{D1-32b(X1=5-CF3)} Me
CH2CH(Me)SCH2(D1-81a) Me
CH2CH(Me)SCH2(D1-82a) Me
CH2CH(Me)SCH2(D1-84a) Me
CH2CH(Me)SCH2(D1-85a) Me
CH2CH(Me)SCH2(D1-87a) Me
CH2CH(Me)SCH2(D1-95a) Me
CH2CH(Me)SCH2(D1-96a) Me
CH2CH(Me)SCH2(D1-98a) Me
CH2CH(Me)SC(O)Me Me
CH2CH(Me)SC(O)(D1-108a) Me
CH2CH(Me)S(O)Me Me
CH2CH(Me)S(O)Et Me
CH2CH(Me)S(O)Pr-n Me
CH2CH(Me)S(O)Pr-i Me
CH2CH(Me)S(O)Bu-n Me
CH2CH(Me)S(O)Bu-i Me
CH2CH(Me)S(O)Bu-t Me
CH2CH(Me)S(O)Pen-n Me
CH2CH(Me)S(O)Hex-n Me
CH2CH(Me)S(O)Pr-c Me
CH2CH(Me)S(O)Bu-c Me
CH2CH(Me)S(O)Pen-c Me
CH2CH(Me)S(O)Hex-c Me
CH2CH(Me)S(O)CH2CH=CH2 Me
CH2CH(Me)S(O)CH2C三CH Me
CH2CH(Me)S(O)CF2H Me
CH2CH(Me)S(O)CF3 Me
CH2CH(Me)S(O)CF2Cl Me
CH2CH(Me)S(O)CH2CF3 Me
CH2CH(Me)S(O){D1-108c} Me
CH2CH(Me)S(O)CH2CH2CN Me
CH2CH(Me)S(O)CH2CH2CF3 Me
CH2CH(Me)S(O)CH2(D1-103a) Me
CH2CH(Me)S(O)CH2CH2OMe Me
CH2CH(Me)S(O)CH2CH2OEt Me
CH2CH(Me)S(O)CH2(D1-32a) Me
CH2CH(Me)S(O)CH2(D1-33a) Me
CH2CH(Me)S(O)CH2(D1-34a) Me
CH2CH(Me)S(O){D1-32b(X1=5-CF3)} Me
CH2CH(Me)S(O)CH2(D1-81a) Me
CH2CH(Me)S(O)CH2(D1-82a) Me
CH2CH(Me)S(O)CH2(D1-84a) Me
CH2CH(Me)S(O)CH2(D1-85a) Me
CH2CH(Me)S(O)CH2(D1-87a) Me
CH2CH(Me)S(O)CH2(D1-95a) Me
CH2CH(Me)S(O)CH2(D1-96a) Me
CH2CH(Me)S(O)CH2(D1-98a) Me
CH2CH(Me)S(O)2Me Me
CH2CH(Me)S(O)2Et Me
CH2CH(Me)S(O)2Pr-n Me
CH2CH(Me)S(O)2Pr-i Me
CH2CH(Me)S(O)2Bu-n Me
CH2CH(Me)S(O)2Bu-i Me
CH2CH(Me)S(O)2Bu-t Me
CH2CH(Me)S(O)2Pen-n Me
CH2CH(Me)S(O)2Hex-n Me
CH2CH(Me)S(O)2Pr-c Me
CH2CH(Me)S(O)2Bu-c Me
CH2CH(Me)S(O)2Pen-c Me
CH2CH(Me)S(O)2Hex-c Me
CH2CH(Me)S(O)2CH2CH=CH2 Me
CH2CH(Me)S(O)2CH2C三CH Me
CH2CH(Me)S(O)2CF2H Me
CH2CH(Me)S(O)2CF3 Me
CH2CH(Me)S(O)2CF2Cl Me
CH2CH(Me)S(O)2CH2CF3 Me
CH2CH(Me)S(O)2{D1-108c} Me
CH2CH(Me)S(O)2CH2CH2CN Me
CH2CH(Me)S(O)2CH2CH2CF3 Me
CH2CH(Me)S(O)2CH2(D1-103a) Me
CH2CH(Me)S(O)2CH2CH2OMe Me
CH2CH(Me)S(O)2CH2CH2OEt Me
CH2CH(Me)S(O)2CH2(D1-32a) Me
CH2CH(Me)S(O)2CH2(D1-33a) Me
CH2CH(Me)S(O)2CH2(D1-34a) Me
CH2CH(Me)S(O)2{D1-32b(X1=5-CF3)} Me
CH2CH(Me)S(O)2CH2(D1-81a) Me
CH2CH(Me)S(O)2CH2(D1-82a) Me
CH2CH(Me)S(O)2CH2(D1-84a) Me
CH2CH(Me)S(O)2CH2(D1-85a) Me
CH2CH(Me)S(O)2CH2(D1-87a) Me
CH2CH(Me)S(O)2CH2(D1-95a) Me
CH2CH(Me)S(O)2CH2(D1-96a) Me
CH2CH(Me)S(O)2CH2(D1-98a) Me
C(O)OH Me
C(O)OMe Me
C(O)OEt Me
C(O)OPr-n Me
C(O)OPr-i Me
C(O)OBu-n Me
C(O)OBu-i Me
C(O)OBu-s Me
C(O)OBu-t Me
C(O)OPen-n Me
C(O)OHex-n Me
CHO Me
C(O)Me Me
C(O)Et Me
C(O)Pr-n Me
C(O)Pr-i Me
C(O)Bu-n Me
C(O)Bu-i Me
C(O)Bu-s Me
C(O)Bu-t Me
C(O)Pen-n Me
C(O)Hex-n Me
C(O)NHC(O)Me Me
C(O)NHMe Me
C(O)NHEt Me
C(O)NHPr-n Me
C(O)NHPr-i Me
C(O)NHBu-n Me
C(O)NHBu-i Me
C(O)NHBu-s Me
C(O)NHBu-t Me
C(O)NHPen-n Me
C(O)NHHex-n Me
CN Me
Ph Me
CH2Cl Me
CH2Br Me
CH2I Me
CH(Me)Cl Me
CH(Me)Br Me
CH(Me)I Me
CH(Et)Cl Me
CH(Et)Br Me
CH(Et)I Me
CH(n-Pr)Cl Me
CH(n-Pr)Br Me
CH(n-Pr)I Me
CH(i-Pr)Cl Me
CH(i-Pr)Br Me
CH(i-Pr)I Me
CH(n-Bu)Cl Me
CH(n-Bu)Br Me
CH(n-Bu)I Me
CH(CH2OMe)Cl Me
CH(CH2OMe)Br Me
CH(CH2OMe)I Me
CH(CH2CH=CH2)Cl Me
CH(CH2CH=CH2)Br Me
CH(CH2CH=CH2)I Me
CH(CH2C三CH)Cl Me
CH(CH2C三CH)Br Me
CH(CH2C三CH)I Me
CH(Me)CH2Cl Me
CH(Me)CH2Br Me
CH(Me)CH2I Me
C(Me)2CH2Cl Me
C(Me)2CH2Br Me
C(Me)2CH2I Me
CH2SCH2(D1-81a) Me
CH2SCH2(D1-81a) Et
CH2SCH2(D1-81a) Pr-n
CH2SCH2(D1-81a) Pr-i
CH2SCH2(D1-81a) Pr-c
CH2SCH2(D1-81a) Bu-n
CH2SCH2(D1-81a) Bu-i
CH2SCH2(D1-81a) Bu-c
CH2SCH2(D1-81a) Bu-s
CH2SCH2(D1-81a) Bu-t
CH2SCH2(D1-81a) Pen-n
CH2SCH2(D1-81a) Pen-c
CH2SCH2(D1-81a) Hex-n
CH2SCH2(D1-81a) Hex-c
CH2SCH2(D1-81a) CH2Pr-c
CH2SCH2(D1-81a) CH2Bu-c
CH2SCH2(D1-81a) CH2Pen-c
CH2SCH2(D1-81a) CH2Hex-c
CH2SCH2(D1-81a) CH2CH=CH2
CH2SCH2(D1-81a) CH2CH=C(Cl)2
CH2SCH2(D1-81a) CH2C≡CH
CH2SCH2(D1-81a) CH2CN
CH2SCH2(D1-81a) CH2CF3
CH2SCH2(D1-81a) CH2OMe
CH2SCH2(D1-81a) CH2OCF3
CH2SCH2(D1-81a) CH2SMe
CH2SCH2(D1-81a) CH2S(O)Me
CH2SCH2(D1-81a) CH2S(O)2Me
CH2SCH2(D1-81a) CH2SCF3
CH2SCH2(D1-81a) CH2S(O)CF3
CH2SCH2(D1-81a) CH2S(O)2CF3
CH2SCH2(D1-81a) CH2CH(OMe)2
CH2SCH2(D1-81a) CH2CH(SMe)2
CH2SCH2(D1-81a) CH2C(O)Me
CH2SCH2(D1-81a) CH2C(O)CF3
CH2SCH2(D1-81a) CH2C(O)OMe
CH2SCH2(D1-81a) CH2(D1-32a)
CH2SCH2(D1-81a) CH2(D1-33a)
CH2SCH2(D1-81a) CH2(D1-34a)
CH2SCH2(D1-81a) CH2(D1-37a)
CH2SCH2(D1-81a) CH2(D1-81a)
CH2SCH2(D1-81a) CH2(D1-82a)
CH2SCH2(D1-81a) CH2(D1-84a)
CH2SCH2(D1-81a) CH2(D1-85a)
CH2SCH2(D1-81a) CH2(D1-87a)
CH2SCH2(D1-81a) CH2(D1-92a)
CH2SCH2(D1-81a) CH2(D1-93a)
CH2SCH2(D1-81a) CH2(D1-95a)
CH2SCH2(D1-81a) CH2(D1-96a)
CH2SCH2(D1-81a) CH2(D1-98a)
CH2SCH2(D1-81a) CH2(D1-108a)
CH2SCH2(D1-81a) CH2(D1-108b,Z=2-Cl)
CH2SCH2(D1-81a) CH2(D1-108b,Z=3-Me)
CH2SCH2(D1-81a) CH2(D1-108b,Z=4-OMe)
CH2SCH2(D1-81a) CH2(D1-108b,Z=2-SMe)
CH2SCH2(D1-81a) CH2(D1-108b,Z=3-CF3)
CH2SCH2(D1-81a) CH2(D1-108b,Z=4-OCF3)
CH2SCH2(D1-81a) CH2(D1-108b,Z=2-SCF3)
CH2SCH2(D1-81a) CH2CH2CN
CH2SCH2(D1-81a) CH2CH2CF3
CH2SCH2(D1-81a) CH2CH2OMe
CH2SCH2(D1-81a) CH2CH2SMe
CH2SCH2(D1-81a) CH2CH2S(O)Me
CH2SCH2(D1-81a) CH2CH2S(O)2Me
CH2SCH2(D1-81a) D1-32a
CH2SCH2(D1-81a) D1-33a
CH2SCH2(D1-81a) D1-34a
CH2SCH2(D1-81a) D1-37a
CH2SCH2(D1-81a) D1-81a
CH2SCH2(D1-81a) D1-82a
CH2SCH2(D1-81a) D1-84a
CH2SCH2(D1-81a) D1-85a
CH2SCH2(D1-81a) D1-87a
CH2SCH2(D1-81a) D1-92a
CH2SCH2(D1-81a) D1-93a
CH2SCH2(D1-81a) D1-95a
CH2SCH2(D1-81a) D1-96a
CH2SCH2(D1-81a) D1-98a
CH2SCH2(D1-81a) D1-108a
CH2SCH2(D1-81a) D1-108b(Z=2-Cl)
CH2SCH2(D1-81a) D1-108b(Z=3-Me)
CH2SCH2(D1-81a) D1-108b(Z=4-OMe)
CH2SCH2(D1-81a) D1-108b(Z=2-SMe)
CH2SCH2(D1-81a) D1-108b(Z=3-CF3)
CH2SCH2(D1-81a) D1-108b(Z=4-OCF3)
CH2SCH2(D1-81a) D1-108b(Z=2-SCF3)
CH2SCH2(D1-81a) C(O)Me
CH2SCH2(D1-81a) C(O)CF3
CH2SCH2(D1-81a) C(O)OMe
CH2S(O)CH2(D1-81a) Me
CH2S(O)CH2(D1-81a) Et
CH2S(O)CH2(D1-81a) Pr-n
CH2S(O)CH2(D1-81a) Pr-i
CH2S(O)CH2(D1-81a) Pr-c
CH2S(O)CH2(D1-81a) Bu-n
CH2S(O)CH2(D1-81a) Bu-i
CH2S(O)CH2(D1-81a) Bu-c
CH2S(O)CH2(D1-81a) Bu-s
CH2S(O)CH2(D1-81a) Bu-t
CH2S(O)CH2(D1-81a) Pen-n
CH2S(O)CH2(D1-81a) Pen-c
CH2S(O)CH2(D1-81a) Hex-n
CH2S(O)CH2(D1-81a) Hex-c
CH2S(O)CH2(D1-81a) CH2Pr-c
CH2S(O)CH2(D1-81a) CH2Bu-c
CH2S(O)CH2(D1-81a) CH2Pen-c
CH2S(O)CH2(D1-81a) CH2Hex-c
CH2S(O)CH2(D1-81a) CH2CH=CH2
CH2S(O)CH2(D1-81a) CH2CH=C(Cl)2
CH2S(O)CH2(D1-81a) CH2C≡CH
CH2S(O)CH2(D1-81a) CH2CN
CH2S(O)CH2(D1-81a) CH2CF3
CH2S(O)CH2(D1-81a) CH2OMe
CH2S(O)CH2(D1-81a) CH2OCF3
CH2S(O)CH2(D1-81a) CH2SMe
CH2S(O)CH2(D1-81a) CH2S(O)Me
CH2S(O)CH2(D1-81a) CH2S(O)2Me
CH2S(O)CH2(D1-81a) CH2SCF3
CH2S(O)CH2(D1-81a) CH2S(O)CF3
CH2S(O)CH2(D1-81a) CH2S(O)2CF3
CH2S(O)CH2(D1-81a) CH2CH(OMe)2
CH2S(O)CH2(D1-81a) CH2CH(SMe)2
CH2S(O)CH2(D1-81a) CH2C(O)Me
CH2S(O)CH2(D1-81a) CH2C(O)CF3
CH2S(O)CH2(D1-81a) CH2C(O)OMe
CH2S(O)CH2(D1-81a) CH2(D1-32a)
CH2S(O)CH2(D1-81a) CH2(D1-33a)
CH2S(O)CH2(D1-81a) CH2(D1-34a)
CH2S(O)CH2(D1-81a) CH2(D1-37a)
CH2S(O)CH2(D1-81a) CH2(D1-81a)
CH2S(O)CH2(D1-81a) CH2(D1-82a)
CH2S(O)CH2(D1-81a) CH2(D1-84a)
CH2S(O)CH2(D1-81a) CH2(D1-85a)
CH2S(O)CH2(D1-81a) CH2(D1-87a)
CH2S(O)CH2(D1-81a) CH2(D1-92a)
CH2S(O)CH2(D1-81a) CH2(D1-93a)
CH2S(O)CH2(D1-81a) CH2(D1-95a)
CH2S(O)CH2(D1-81a) CH2(D1-96a)
CH2S(O)CH2(D1-81a) CH2(D1-98a)
CH2S(O)CH2(D1-81a) CH2(D1-108a)
CH2S(O)CH2(D1-81a) CH2(D1-108b,Z=2-Cl)
CH2S(O)CH2(D1-81a) CH2(D1-108b,Z=3-Me)
CH2S(O)CH2(D1-81a) CH2(D1-108b,Z=4-OMe)
CH2S(O)CH2(D1-81a) CH2(D1-108b,Z=2-SMe)
CH2S(O)CH2(D1-81a) CH2(D1-108b,Z=3-CF3)
CH2S(O)CH2(D1-81a) CH2(D1-108b,Z=4-OCF3)
CH2S(O)CH2(D1-81a) CH2(D1-108b,Z=2-SCF3)
CH2S(O)CH2(D1-81a) CH2CH2CN
CH2S(O)CH2(D1-81a) CH2CH2CF3
CH2S(O)CH2(D1-81a) CH2CH2OMe
CH2S(O)CH2(D1-81a) CH2CH2SMe
CH2S(O)CH2(D1-81a) CH2CH2S(O)Me
CH2S(O)CH2(D1-81a) CH2CH2S(O)2Me
CH2S(O)CH2(D1-81a) D1-32a
CH2S(O)CH2(D1-81a) D1-33a
CH2S(O)CH2(D1-81a) D1-34a
CH2S(O)CH2(D1-81a) D1-37a
CH2S(O)CH2(D1-81a) D1-81a
CH2S(O)CH2(D1-81a) D1-82a
CH2S(O)CH2(D1-81a) D1-84a
CH2S(O)CH2(D1-81a) D1-85a
CH2S(O)CH2(D1-81a) D1-87a
CH2S(O)CH2(D1-81a) D1-92a
CH2S(O)CH2(D1-81a) D1-93a
CH2S(O)CH2(D1-81a) D1-95a
CH2S(O)CH2(D1-81a) D1-96a
CH2S(O)CH2(D1-81a) D1-98a
CH2S(O)CH2(D1-81a) D1-108a
CH2S(O)CH2(D1-81a) D1-108b(Z=2-Cl)
CH2S(O)CH2(D1-81a) D1-108b(Z=3-Me)
CH2S(O)CH2(D1-81a) D1-108b(Z=4-OMe)
CH2S(O)CH2(D1-81a) D1-108b(Z=2-SMe)
CH2S(O)CH2(D1-81a) D1-108b(Z=3-CF3)
CH2S(O)CH2(D1-81a) D1-108b(Z=4-OCF3)
CH2S(O)CH2(D1-81a) D1-108b(Z=2-SCF3)
CH2S(O)CH2(D1-81a) C(O)Me
CH2S(O)CH2(D1-81a) C(O)CF3
CH2S(O)CH2(D1-81a) C(O)OMe
CH2S(O)2CH2(D1-81a) Me
CH2S(O)2CH2(D1-81a) Et
CH2S(O)2CH2(D1-81a) Pr-n
CH2S(O)2CH2(D1-81a) Pr-i
CH2S(O)2CH2(D1-81a) Pr-c
CH2S(O)2CH2(D1-81a) Bu-n
CH2S(O)2CH2(D1-81a) Bu-i
CH2S(O)2CH2(D1-81a) Bu-c
CH2S(O)2CH2(D1-81a) Bu-s
CH2S(O)2CH2(D1-81a) Bu-t
CH2S(O)2CH2(D1-81a) Pen-n
CH2S(O)2CH2(D1-81a) Pen-c
CH2S(O)2CH2(D1-81a) Hex-n
CH2S(O)2CH2(D1-81a) Hex-c
CH2S(O)2CH2(D1-81a) CH2Pr-c
CH2S(O)2CH2(D1-81a) CH2Bu-c
CH2S(O)2CH2(D1-81a) CH2Pen-c
CH2S(O)2CH2(D1-81a) CH2Hex-c
CH2S(O)2CH2(D1-81a) CH2CH=CH2
CH2S(O)2CH2(D1-81a) CH2CH=C(Cl)2
CH2S(O)2CH2(D1-81a) CH2C≡CH
CH2S(O)2CH2(D1-81a) CH2CN
CH2S(O)2CH2(D1-81a) CH2CF3
CH2S(O)2CH2(D1-81a) CH2OMe
CH2S(O)2CH2(D1-81a) CH2OCF3
CH2S(O)2CH2(D1-81a) CH2SMe
CH2S(O)2CH2(D1-81a) CH2S(O)Me
CH2S(O)2CH2(D1-81a) CH2S(O)2Me
CH2S(O)2CH2(D1-81a) CH2SCF3
CH2S(O)2CH2(D1-81a) CH2S(O)CF3
CH2S(O)2CH2(D1-81a) CH2S(O)2CF3
CH2S(O)2CH2(D1-81a) CH2CH(OMe)2
CH2S(O)2CH2(D1-81a) CH2CH(SMe)2
CH2S(O)2CH2(D1-81a) CH2C(O)Me
CH2S(O)2CH2(D1-81a) CH2C(O)CF3
CH2S(O)2CH2(D1-81a) CH2C(O)OMe
CH2S(O)2CH2(D1-81a) CH2(D1-32a)
CH2S(O)2CH2(D1-81a) CH2(D1-33a)
CH2S(O)2CH2(D1-81a) CH2(D1-34a)
CH2S(O)2CH2(D1-81a) CH2(D1-37a)
CH2S(O)2CH2(D1-81a) CH2(D1-81a)
CH2S(O)2CH2(D1-81a) CH2(D1-82a)
CH2S(O)2CH2(D1-81a) CH2(D1-84a)
CH2S(O)2CH2(D1-81a) CH2(D1-85a)
CH2S(O)2CH2(D1-81a) CH2(D1-87a)
CH2S(O)2CH2(D1-81a) CH2(D1-92a)
CH2S(O)2CH2(D1-81a) CH2(D1-93a)
CH2S(O)2CH2(D1-81a) CH2(D1-95a)
CH2S(O)2CH2(D1-81a) CH2(D1-96a)
CH2S(O)2CH2(D1-81a) CH2(D1-98a)
CH2S(O)2CH2(D1-81a) CH2(D1-108a)
CH2S(O)2CH2(D1-81a) CH2(D1-108b,Z=2-Cl)
CH2S(O)2CH2(D1-81a) CH2(D1-108b,Z=3-Me)
CH2S(O)2CH2(D1-81a) CH2(D1-108b,Z=4-OMe)
CH2S(O)2CH2(D1-81a) CH2(D1-108b,Z=2-SMe)
CH2S(O)2CH2(D1-81a) CH2(D1-108b,Z=3-CF3)
CH2S(O)2CH2(D1-81a) CH2(D1-108b,Z=4-OCF3)
CH2S(O)2CH2(D1-81a) CH2(D1-108b,Z=2-SCF3)
CH2S(O)2CH2(D1-81a) CH2CH2CN
CH2S(O)2CH2(D1-81a) CH2CH2CF3
CH2S(O)2CH2(D1-81a) CH2CH2OMe
CH2S(O)2CH2(D1-81a) CH2CH2SMe
CH2S(O)2CH2(D1-81a) CH2CH2S(O)Me
CH2S(O)2CH2(D1-81a) CH2CH2S(O)2Me
CH2S(O)2CH2(D1-81a) D1-32a
CH2S(O)2CH2(D1-81a) D1-33a
CH2S(O)2CH2(D1-81a) D1-34a
CH2S(O)2CH2(D1-81a) D1-37a
CH2S(O)2CH2(D1-81a) D1-81a
CH2S(O)2CH2(D1-81a) D1-82a
CH2S(O)2CH2(D1-81a) D1-84a
CH2S(O)2CH2(D1-81a) D1-85a
CH2S(O)2CH2(D1-81a) D1-87a
CH2S(O)2CH2(D1-81a) D1-92a
CH2S(O)2CH2(D1-81a) D1-93a
CH2S(O)2CH2(D1-81a) D1-95a
CH2S(O)2CH2(D1-81a) D1-96a
CH2S(O)2CH2(D1-81a) D1-98a
CH2S(O)2CH2(D1-81a) D1-108a
CH2S(O)2CH2(D1-81a) D1-108b(Z=2-Cl)
CH2S(O)2CH2(D1-81a) D1-108b(Z=3-Me)
CH2S(O)2CH2(D1-81a) D1-108b(Z=4-OMe)
CH2S(O)2CH2(D1-81a) D1-108b(Z=2-SMe)
CH2S(O)2CH2(D1-81a) D1-108b(Z=3-CF3)
CH2S(O)2CH2(D1-81a) D1-108b(Z=4-OCF3)
CH2S(O)2CH2(D1-81a) D1-108b(Z=2-SCF3)
CH2S(O)2CH2(D1-81a) C(O)Me
CH2S(O)2CH2(D1-81a) C(O)CF3
CH2S(O)2CH2(D1-81a) C(O)OMe
CH(Me)SCH2(D1-81a) Me
CH(Me)SCH2(D1-81a) Et
CH(Me)SCH2(D1-81a) Pr-n
CH(Me)SCH2(D1-81a) Pr-i
CH(Me)SCH2(D1-81a) Pr-c
CH(Me)SCH2(D1-81a) Bu-n
CH(Me)SCH2(D1-81a) Bu-i
CH(Me)SCH2(D1-81a) Bu-c
CH(Me)SCH2(D1-81a) Bu-s
CH(Me)SCH2(D1-81a) Bu-t
CH(Me)SCH2(D1-81a) Pen-n
CH(Me)SCH2(D1-81a) Pen-c
CH(Me)SCH2(D1-81a) Hex-n
CH(Me)SCH2(D1-81a) Hex-c
CH(Me)SCH2(D1-81a) CH2Pr-c
CH(Me)SCH2(D1-81a) CH2Bu-c
CH(Me)SCH2(D1-81a) CH2Pen-c
CH(Me)SCH2(D1-81a) CH2Hex-c
CH(Me)SCH2(D1-81a) CH2CH=CH2
CH(Me)SCH2(D1-81a) CH2CH=C(Cl)2
CH(Me)SCH2(D1-81a) CH2C≡CH
CH(Me)SCH2(D1-81a) CH2CN
CH(Me)SCH2(D1-81a) CH2CF3
CH(Me)SCH2(D1-81a) CH2OMe
CH(Me)SCH2(D1-81a) CH2OCF3
CH(Me)SCH2(D1-81a) CH2SMe
CH(Me)SCH2(D1-81a) CH2S(O)Me
CH(Me)SCH2(D1-81a) CH2S(O)2Me
CH(Me)SCH2(D1-81a) CH2SCF3
CH(Me)SCH2(D1-81a) CH2S(O)CF3
CH(Me)SCH2(D1-81a) CH2S(O)2CF3
CH(Me)SCH2(D1-81a) CH2CH(OMe)2
CH(Me)SCH2(D1-81a) CH2CH(SMe)2
CH(Me)SCH2(D1-81a) CH2C(O)Me
CH(Me)SCH2(D1-81a) CH2C(O)CF3
CH(Me)SCH2(D1-81a) CH2C(O)OMe
CH(Me)SCH2(D1-81a) CH2(D1-32a)
CH(Me)SCH2(D1-81a) CH2(D1-33a)
CH(Me)SCH2(D1-81a) CH2(D1-34a)
CH(Me)SCH2(D1-81a) CH2(D1-37a)
CH(Me)SCH2(D1-81a) CH2(D1-81a)
CH(Me)SCH2(D1-81a) CH2(D1-82a)
CH(Me)SCH2(D1-81a) CH2(D1-84a)
CH(Me)SCH2(D1-81a) CH2(D1-85a)
CH(Me)SCH2(D1-81a) CH2(D1-87a)
CH(Me)SCH2(D1-81a) CH2(D1-92a)
CH(Me)SCH2(D1-81a) CH2(D1-93a)
CH(Me)SCH2(D1-81a) CH2(D1-95a)
CH(Me)SCH2(D1-81a) CH2(D1-96a)
CH(Me)SCH2(D1-81a) CH2(D1-98a)
CH(Me)SCH2(D1-81a) CH2(D1-108a)
CH(Me)SCH2(D1-81a) CH2(D1-108b,Z=2-Cl)
CH(Me)SCH2(D1-81a) CH2(D1-108b,Z=3-Me)
CH(Me)SCH2(D1-81a) CH2(D1-108b,Z=4-OMe)
CH(Me)SCH2(D1-81a) CH2(D1-108b,Z=2-SMe)
CH(Me)SCH2(D1-81a) CH2(D1-108b,Z=3-CF3)
CH(Me)SCH2(D1-81a) CH2(D1-108b,Z=4-OCF3)
CH(Me)SCH2(D1-81a) CH2(D1-108b,Z=2-SCF3)
CH(Me)SCH2(D1-81a) CH2CH2CN
CH(Me)SCH2(D1-81a) CH2CH2CF3
CH(Me)SCH2(D1-81a) CH2CH2OMe
CH(Me)SCH2(D1-81a) CH2CH2SMe
CH(Me)SCH2(D1-81a) CH2CH2S(O)Me
CH(Me)SCH2(D1-81a) CH2CH2S(O)2Me
CH(Me)SCH2(D1-81a) D1-32a
CH(Me)SCH2(D1-81a) D1-33a
CH(Me)SCH2(D1-81a) D1-34a
CH(Me)SCH2(D1-81a) D1-37a
CH(Me)SCH2(D1-81a) D1-81a
CH(Me)SCH2(D1-81a) D1-82a
CH(Me)SCH2(D1-81a) D1-84a
CH(Me)SCH2(D1-81a) D1-85a
CH(Me)SCH2(D1-81a) D1-87a
CH(Me)SCH2(D1-81a) D1-92a
CH(Me)SCH2(D1-81a) D1-93a
CH(Me)SCH2(D1-81a) D1-95a
CH(Me)SCH2(D1-81a) D1-96a
CH(Me)SCH2(D1-81a) D1-98a
CH(Me)SCH2(D1-81a) D1-108a
CH(Me)SCH2(D1-81a) D1-108b(Z=2-Cl)
CH(Me)SCH2(D1-81a) D1-108b(Z=3-Me)
CH(Me)SCH2(D1-81a) D1-108b(Z=4-OMe)
CH(Me)SCH2(D1-81a) D1-108b(Z=2-SMe)
CH(Me)SCH2(D1-81a) D1-108b(Z=3-CF3)
CH(Me)SCH2(D1-81a) D1-108b(Z=4-OCF3)
CH(Me)SCH2(D1-81a) D1-108b(Z=2-SCF3)
CH(Me)SCH2(D1-81a) C(O)Me
CH(Me)SCH2(D1-81a) C(O)CF3
CH(Me)SCH2(D1-81a) C(O)OMe
CH(Me)S(O)CH2(D1-81a) Me
CH(Me)S(O)CH2(D1-81a) Et
CH(Me)S(O)CH2(D1-81a) Pr-n
CH(Me)S(O)CH2(D1-81a) Pr-i
CH(Me)S(O)CH2(D1-81a) Pr-c
CH(Me)S(O)CH2(D1-81a) Bu-n
CH(Me)S(O)CH2(D1-81a) Bu-i
CH(Me)S(O)CH2(D1-81a) Bu-c
CH(Me)S(O)CH2(D1-81a) Bu-s
CH(Me)S(O)CH2(D1-81a) Bu-t
CH(Me)S(O)CH2(D1-81a) Pen-n
CH(Me)S(O)CH2(D1-81a) Pen-c
CH(Me)S(O)CH2(D1-81a) Hex-n
CH(Me)S(O)CH2(D1-81a) Hex-c
CH(Me)S(O)CH2(D1-81a) CH2Pr-c
CH(Me)S(O)CH2(D1-81a) CH2Bu-c
CH(Me)S(O)CH2(D1-81a) CH2Pen-c
CH(Me)S(O)CH2(D1-81a) CH2Hex-c
CH(Me)S(O)CH2(D1-81a) CH2CH=CH2
CH(Me)S(O)CH2(D1-81a) CH2CH=C(Cl)2
CH(Me)S(O)CH2(D1-81a) CH2C≡CH
CH(Me)S(O)CH2(D1-81a) CH2CN
CH(Me)S(O)CH2(D1-81a) CH2CF3
CH(Me)S(O)CH2(D1-81a) CH2OMe
CH(Me)S(O)CH2(D1-81a) CH2OCF3
CH(Me)S(O)CH2(D1-81a) CH2SMe
CH(Me)S(O)CH2(D1-81a) CH2S(O)Me
CH(Me)S(O)CH2(D1-81a) CH2S(O)2Me
CH(Me)S(O)CH2(D1-81a) CH2SCF3
CH(Me)S(O)CH2(D1-81a) CH2S(O)CF3
CH(Me)S(O)CH2(D1-81a) CH2S(O)2CF3
CH(Me)S(O)CH2(D1-81a) CH2CH(OMe)2
CH(Me)S(O)CH2(D1-81a) CH2CH(SMe)2
CH(Me)S(O)CH2(D1-81a) CH2C(O)Me
CH(Me)S(O)CH2(D1-81a) CH2C(O)CF3
CH(Me)S(O)CH2(D1-81a) CH2C(O)OMe
CH(Me)S(O)CH2(D1-81a) CH2(D1-32a)
CH(Me)S(O)CH2(D1-81a) CH2(D1-33a)
CH(Me)S(O)CH2(D1-81a) CH2(D1-34a)
CH(Me)S(O)CH2(D1-81a) CH2(D1-37a)
CH(Me)S(O)CH2(D1-81a) CH2(D1-81a)
CH(Me)S(O)CH2(D1-81a) CH2(D1-82a)
CH(Me)S(O)CH2(D1-81a) CH2(D1-84a)
CH(Me)S(O)CH2(D1-81a) CH2(D1-85a)
CH(Me)S(O)CH2(D1-81a) CH2(D1-87a)
CH(Me)S(O)CH2(D1-81a) CH2(D1-92a)
CH(Me)S(O)CH2(D1-81a) CH2(D1-93a)
CH(Me)S(O)CH2(D1-81a) CH2(D1-95a)
CH(Me)S(O)CH2(D1-81a) CH2(D1-96a)
CH(Me)S(O)CH2(D1-81a) CH2(D1-98a)
CH(Me)S(O)CH2(D1-81a) CH2(D1-108a)
CH(Me)S(O)CH2(D1-81a) CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)CH2(D1-81a) CH2(D1-108b,Z=3-Me)
CH(Me)S(O)CH2(D1-81a) CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)CH2(D1-81a) CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)CH2(D1-81a) CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)CH2(D1-81a) CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)CH2(D1-81a) CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)CH2(D1-81a) CH2CH2CN
CH(Me)S(O)CH2(D1-81a) CH2CH2CF3
CH(Me)S(O)CH2(D1-81a) CH2CH2OMe
CH(Me)S(O)CH2(D1-81a) CH2CH2SMe
CH(Me)S(O)CH2(D1-81a) CH2CH2S(O)Me
CH(Me)S(O)CH2(D1-81a) CH2CH2S(O)2Me
CH(Me)S(O)CH2(D1-81a) D1-32a
CH(Me)S(O)CH2(D1-81a) D1-33a
CH(Me)S(O)CH2(D1-81a) D1-34a
CH(Me)S(O)CH2(D1-81a) D1-37a
CH(Me)S(O)CH2(D1-81a) D1-81a
CH(Me)S(O)CH2(D1-81a) D1-82a
CH(Me)S(O)CH2(D1-81a) D1-84a
CH(Me)S(O)CH2(D1-81a) D1-85a
CH(Me)S(O)CH2(D1-81a) D1-87a
CH(Me)S(O)CH2(D1-81a) D1-92a
CH(Me)S(O)CH2(D1-81a) D1-93a
CH(Me)S(O)CH2(D1-81a) D1-95a
CH(Me)S(O)CH2(D1-81a) D1-96a
CH(Me)S(O)CH2(D1-81a) D1-98a
CH(Me)S(O)CH2(D1-81a) D1-108a
CH(Me)S(O)CH2(D1-81a) D1-108b(Z=2-Cl)
CH(Me)S(O)CH2(D1-81a) D1-108b(Z=3-Me)
CH(Me)S(O)CH2(D1-81a) D1-108b(Z=4-OMe)
CH(Me)S(O)CH2(D1-81a) D1-108b(Z=2-SMe)
CH(Me)S(O)CH2(D1-81a) D1-108b(Z=3-CF3)
CH(Me)S(O)CH2(D1-81a) D1-108b(Z=4-OCF3)
CH(Me)S(O)CH2(D1-81a) D1-108b(Z=2-SCF3)
CH(Me)S(O)CH2(D1-81a) C(O)Me
CH(Me)S(O)CH2(D1-81a) C(O)CF3
CH(Me)S(O)CH2(D1-81a) C(O)OMe
CH(Me)S(O)2CH2(D1-81a) Me
CH(Me)S(O)2CH2(D1-81a) Et
CH(Me)S(O)2CH2(D1-81a) Pr-n
CH(Me)S(O)2CH2(D1-81a) Pr-i
CH(Me)S(O)2CH2(D1-81a) Pr-c
CH(Me)S(O)2CH2(D1-81a) Bu-n
CH(Me)S(O)2CH2(D1-81a) Bu-i
CH(Me)S(O)2CH2(D1-81a) Bu-c
CH(Me)S(O)2CH2(D1-81a) Bu-s
CH(Me)S(O)2CH2(D1-81a) Bu-t
CH(Me)S(O)2CH2(D1-81a) Pen-n
CH(Me)S(O)2CH2(D1-81a) Pen-c
CH(Me)S(O)2CH2(D1-81a) Hex-n
CH(Me)S(O)2CH2(D1-81a) Hex-c
CH(Me)S(O)2CH2(D1-81a) CH2Pr-c
CH(Me)S(O)2CH2(D1-81a) CH2Bu-c
CH(Me)S(O)2CH2(D1-81a) CH2Pen-c
CH(Me)S(O)2CH2(D1-81a) CH2Hex-c
CH(Me)S(O)2CH2(D1-81a) CH2CH=CH2
CH(Me)S(O)2CH2(D1-81a) CH2CH=C(Cl)2
CH(Me)S(O)2CH2(D1-81a) CH2C≡CH
CH(Me)S(O)2CH2(D1-81a) CH2CN
CH(Me)S(O)2CH2(D1-81a) CH2CF3
CH(Me)S(O)2CH2(D1-81a) CH2OMe
CH(Me)S(O)2CH2(D1-81a) CH2OCF3
CH(Me)S(O)2CH2(D1-81a) CH2SMe
CH(Me)S(O)2CH2(D1-81a) CH2S(O)Me
CH(Me)S(O)2CH2(D1-81a) CH2S(O)2Me
CH(Me)S(O)2CH2(D1-81a) CH2SCF3
CH(Me)S(O)2CH2(D1-81a) CH2S(O)CF3
CH(Me)S(O)2CH2(D1-81a) CH2S(O)2CF3
CH(Me)S(O)2CH2(D1-81a) CH2CH(OMe)2
CH(Me)S(O)2CH2(D1-81a) CH2CH(SMe)2
CH(Me)S(O)2CH2(D1-81a) CH2C(O)Me
CH(Me)S(O)2CH2(D1-81a) CH2C(O)CF3
CH(Me)S(O)2CH2(D1-81a) CH2C(O)OMe
CH(Me)S(O)2CH2(D1-81a) CH2(D1-32a)
CH(Me)S(O)2CH2(D1-81a) CH2(D1-33a)
CH(Me)S(O)2CH2(D1-81a) CH2(D1-34a)
CH(Me)S(O)2CH2(D1-81a) CH2(D1-37a)
CH(Me)S(O)2CH2(D1-81a) CH2(D1-81a)
CH(Me)S(O)2CH2(D1-81a) CH2(D1-82a)
CH(Me)S(O)2CH2(D1-81a) CH2(D1-84a)
CH(Me)S(O)2CH2(D1-81a) CH2(D1-85a)
CH(Me)S(O)2CH2(D1-81a) CH2(D1-87a)
CH(Me)S(O)2CH2(D1-81a) CH2(D1-92a)
CH(Me)S(O)2CH2(D1-81a) CH2(D1-93a)
CH(Me)S(O)2CH2(D1-81a) CH2(D1-95a)
CH(Me)S(O)2CH2(D1-81a) CH2(D1-96a)
CH(Me)S(O)2CH2(D1-81a) CH2(D1-98a)
CH(Me)S(O)2CH2(D1-81a) CH2(D1-108a)
CH(Me)S(O)2CH2(D1-81a) CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)2CH2(D1-81a) CH2(D1-108b,Z=3-Me)
CH(Me)S(O)2CH2(D1-81a) CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)2CH2(D1-81a) CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)2CH2(D1-81a) CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)2CH2(D1-81a) CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)2CH2(D1-81a) CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)2CH2(D1-81a) CH2CH2CN
CH(Me)S(O)2CH2(D1-81a) CH2CH2CF3
CH(Me)S(O)2CH2(D1-81a) CH2CH2OMe
CH(Me)S(O)2CH2(D1-81a) CH2CH2SMe
CH(Me)S(O)2CH2(D1-81a) CH2CH2S(O)Me
CH(Me)S(O)2CH2(D1-81a) CH2CH2S(O)2Me
CH(Me)S(O)2CH2(D1-81a) D1-32a
CH(Me)S(O)2CH2(D1-81a) D1-33a
CH(Me)S(O)2CH2(D1-81a) D1-34a
CH(Me)S(O)2CH2(D1-81a) D1-37a
CH(Me)S(O)2CH2(D1-81a) D1-81a
CH(Me)S(O)2CH2(D1-81a) D1-82a
CH(Me)S(O)2CH2(D1-81a) D1-84a
CH(Me)S(O)2CH2(D1-81a) D1-85a
CH(Me)S(O)2CH2(D1-81a) D1-87a
CH(Me)S(O)2CH2(D1-81a) D1-92a
CH(Me)S(O)2CH2(D1-81a) D1-93a
CH(Me)S(O)2CH2(D1-81a) D1-95a
CH(Me)S(O)2CH2(D1-81a) D1-96a
CH(Me)S(O)2CH2(D1-81a) D1-98a
CH(Me)S(O)2CH2(D1-81a) D1-108a
CH(Me)S(O)2CH2(D1-81a) D1-108b(Z=2-Cl)
CH(Me)S(O)2CH2(D1-81a) D1-108b(Z=3-Me)
CH(Me)S(O)2CH2(D1-81a) D1-108b(Z=4-OMe)
CH(Me)S(O)2CH2(D1-81a) D1-108b(Z=2-SMe)
CH(Me)S(O)2CH2(D1-81a) D1-108b(Z=3-CF3)
CH(Me)S(O)2CH2(D1-81a) D1-108b(Z=4-OCF3)
CH(Me)S(O)2CH2(D1-81a) D1-108b(Z=2-SCF3)
CH(Me)S(O)2CH2(D1-81a) C(O)Me
CH(Me)S(O)2CH2(D1-81a) C(O)CF3
CH(Me)S(O)2CH2(D1-81a) C(O)OMe
CH2SCH2(D1-82a) Me
CH2SCH2(D1-82a) Et
CH2SCH2(D1-82a) Pr-n
CH2SCH2(D1-82a) Pr-i
CH2SCH2(D1-82a) Pr-c
CH2SCH2(D1-82a) Bu-n
CH2SCH2(D1-82a) Bu-i
CH2SCH2(D1-82a) Bu-c
CH2SCH2(D1-82a) Bu-s
CH2SCH2(D1-82a) Bu-t
CH2SCH2(D1-82a) Pen-n
CH2SCH2(D1-82a) Pen-c
CH2SCH2(D1-82a) Hex-n
CH2SCH2(D1-82a) Hex-c
CH2SCH2(D1-82a) CH2Pr-c
CH2SCH2(D1-82a) CH2Bu-c
CH2SCH2(D1-82a) CH2Pen-c
CH2SCH2(D1-82a) CH2Hex-c
CH2SCH2(D1-82a) CH2CH=CH2
CH2SCH2(D1-82a) CH2CH=C(Cl)2
CH2SCH2(D1-82a) CH2C≡CH
CH2SCH2(D1-82a) CH2CN
CH2SCH2(D1-82a) CH2CF3
CH2SCH2(D1-82a) CH2OMe
CH2SCH2(D1-82a) CH2OCF3
CH2SCH2(D1-82a) CH2SMe
CH2SCH2(D1-82a) CH2S(O)Me
CH2SCH2(D1-82a) CH2S(O)2Me
CH2SCH2(D1-82a) CH2SCF3
CH2SCH2(D1-82a) CH2S(O)CF3
CH2SCH2(D1-82a) CH2S(O)2CF3
CH2SCH2(D1-82a) CH2CH(OMe)2
CH2SCH2(D1-82a) CH2CH(SMe)2
CH2SCH2(D1-82a) CH2C(O)Me
CH2SCH2(D1-82a) CH2C(O)CF3
CH2SCH2(D1-82a) CH2C(O)OMe
CH2SCH2(D1-82a) CH2(D1-32a)
CH2SCH2(D1-82a) CH2(D1-33a)
CH2SCH2(D1-82a) CH2(D1-34a)
CH2SCH2(D1-82a) CH2(D1-37a)
CH2SCH2(D1-82a) CH2(D1-81a)
CH2SCH2(D1-82a) CH2(D1-82a)
CH2SCH2(D1-82a) CH2(D1-84a)
CH2SCH2(D1-82a) CH2(D1-85a)
CH2SCH2(D1-82a) CH2(D1-87a)
CH2SCH2(D1-82a) CH2(D1-92a)
CH2SCH2(D1-82a) CH2(D1-93a)
CH2SCH2(D1-82a) CH2(D1-95a)
CH2SCH2(D1-82a) CH2(D1-96a)
CH2SCH2(D1-82a) CH2(D1-98a)
CH2SCH2(D1-82a) CH2(D1-108a)
CH2SCH2(D1-82a) CH2(D1-108b,Z=2-Cl)
CH2SCH2(D1-82a) CH2(D1-108b,Z=3-Me)
CH2SCH2(D1-82a) CH2(D1-108b,Z=4-OMe)
CH2SCH2(D1-82a) CH2(D1-108b,Z=2-SMe)
CH2SCH2(D1-82a) CH2(D1-108b,Z=3-CF3)
CH2SCH2(D1-82a) CH2(D1-108b,Z=4-OCF3)
CH2SCH2(D1-82a) CH2(D1-108b,Z=2-SCF3)
CH2SCH2(D1-82a) CH2CH2CN
CH2SCH2(D1-82a) CH2CH2CF3
CH2SCH2(D1-82a) CH2CH2OMe
CH2SCH2(D1-82a) CH2CH2SMe
CH2SCH2(D1-82a) CH2CH2S(O)Me
CH2SCH2(D1-82a) CH2CH2S(O)2Me
CH2SCH2(D1-82a) D1-32a
CH2SCH2(D1-82a) D1-33a
CH2SCH2(D1-82a) D1-34a
CH2SCH2(D1-82a) D1-37a
CH2SCH2(D1-82a) D1-81a
CH2SCH2(D1-82a) D1-82a
CH2SCH2(D1-82a) D1-84a
CH2SCH2(D1-82a) D1-85a
CH2SCH2(D1-82a) D1-87a
CH2SCH2(D1-82a) D1-92a
CH2SCH2(D1-82a) D1-93a
CH2SCH2(D1-82a) D1-95a
CH2SCH2(D1-82a) D1-96a
CH2SCH2(D1-82a) D1-98a
CH2SCH2(D1-82a) D1-108a
CH2SCH2(D1-82a) D1-108b(Z=2-Cl)
CH2SCH2(D1-82a) D1-108b(Z=3-Me)
CH2SCH2(D1-82a) D1-108b(Z=4-OMe)
CH2SCH2(D1-82a) D1-108b(Z=2-SMe)
CH2SCH2(D1-82a) D1-108b(Z=3-CF3)
CH2SCH2(D1-82a) D1-108b(Z=4-OCF3)
CH2SCH2(D1-82a) D1-108b(Z=2-SCF3)
CH2SCH2(D1-82a) C(O)Me
CH2SCH2(D1-82a) C(O)CF3
CH2SCH2(D1-82a) C(O)OMe
CH2S(O)CH2(D1-82a) Me
CH2S(O)CH2(D1-82a) Et
CH2S(O)CH2(D1-82a) Pr-n
CH2S(O)CH2(D1-82a) Pr-i
CH2S(O)CH2(D1-82a) Pr-c
CH2S(O)CH2(D1-82a) Bu-n
CH2S(O)CH2(D1-82a) Bu-i
CH2S(O)CH2(D1-82a) Bu-c
CH2S(O)CH2(D1-82a) Bu-s
CH2S(O)CH2(D1-82a) Bu-t
CH2S(O)CH2(D1-82a) Pen-n
CH2S(O)CH2(D1-82a) Pen-c
CH2S(O)CH2(D1-82a) Hex-n
CH2S(O)CH2(D1-82a) Hex-c
CH2S(O)CH2(D1-82a) CH2Pr-c
CH2S(O)CH2(D1-82a) CH2Bu-c
CH2S(O)CH2(D1-82a) CH2Pen-c
CH2S(O)CH2(D1-82a) CH2Hex-c
CH2S(O)CH2(D1-82a) CH2CH=CH2
CH2S(O)CH2(D1-82a) CH2CH=C(Cl)2
CH2S(O)CH2(D1-82a) CH2C≡CH
CH2S(O)CH2(D1-82a) CH2CN
CH2S(O)CH2(D1-82a) CH2CF3
CH2S(O)CH2(D1-82a) CH2OMe
CH2S(O)CH2(D1-82a) CH2OCF3
CH2S(O)CH2(D1-82a) CH2SMe
CH2S(O)CH2(D1-82a) CH2S(O)Me
CH2S(O)CH2(D1-82a) CH2S(O)2Me
CH2S(O)CH2(D1-82a) CH2SCF3
CH2S(O)CH2(D1-82a) CH2S(O)CF3
CH2S(O)CH2(D1-82a) CH2S(O)2CF3
CH2S(O)CH2(D1-82a) CH2CH(OMe)2
CH2S(O)CH2(D1-82a) CH2CH(SMe)2
CH2S(O)CH2(D1-82a) CH2C(O)Me
CH2S(O)CH2(D1-82a) CH2C(O)CF3
CH2S(O)CH2(D1-82a) CH2C(O)OMe
CH2S(O)CH2(D1-82a) CH2(D1-32a)
CH2S(O)CH2(D1-82a) CH2(D1-33a)
CH2S(O)CH2(D1-82a) CH2(D1-34a)
CH2S(O)CH2(D1-82a) CH2(D1-37a)
CH2S(O)CH2(D1-82a) CH2(D1-81a)
CH2S(O)CH2(D1-82a) CH2(D1-82a)
CH2S(O)CH2(D1-82a) CH2(D1-84a)
CH2S(O)CH2(D1-82a) CH2(D1-85a)
CH2S(O)CH2(D1-82a) CH2(D1-87a)
CH2S(O)CH2(D1-82a) CH2(D1-92a)
CH2S(O)CH2(D1-82a) CH2(D1-93a)
CH2S(O)CH2(D1-82a) CH2(D1-95a)
CH2S(O)CH2(D1-82a) CH2(D1-96a)
CH2S(O)CH2(D1-82a) CH2(D1-98a)
CH2S(O)CH2(D1-82a) CH2(D1-108a)
CH2S(O)CH2(D1-82a) CH2(D1-108b,Z=2-Cl)
CH2S(O)CH2(D1-82a) CH2(D1-108b,Z=3-Me)
CH2S(O)CH2(D1-82a) CH2(D1-108b,Z=4-OMe)
CH2S(O)CH2(D1-82a) CH2(D1-108b,Z=2-SMe)
CH2S(O)CH2(D1-82a) CH2(D1-108b,Z=3-CF3)
CH2S(O)CH2(D1-82a) CH2(D1-108b,Z=4-OCF3)
CH2S(O)CH2(D1-82a) CH2(D1-108b,Z=2-SCF3)
CH2S(O)CH2(D1-82a) CH2CH2CN
CH2S(O)CH2(D1-82a) CH2CH2CF3
CH2S(O)CH2(D1-82a) CH2CH2OMe
CH2S(O)CH2(D1-82a) CH2CH2SMe
CH2S(O)CH2(D1-82a) CH2CH2S(O)Me
CH2S(O)CH2(D1-82a) CH2CH2S(O)2Me
CH2S(O)CH2(D1-82a) D1-32a
CH2S(O)CH2(D1-82a) D1-33a
CH2S(O)CH2(D1-82a) D1-34a
CH2S(O)CH2(D1-82a) D1-37a
CH2S(O)CH2(D1-82a) D1-81a
CH2S(O)CH2(D1-82a) D1-82a
CH2S(O)CH2(D1-82a) D1-84a
CH2S(O)CH2(D1-82a) D1-85a
CH2S(O)CH2(D1-82a) D1-87a
CH2S(O)CH2(D1-82a) D1-92a
CH2S(O)CH2(D1-82a) D1-93a
CH2S(O)CH2(D1-82a) D1-95a
CH2S(O)CH2(D1-82a) D1-96a
CH2S(O)CH2(D1-82a) D1-98a
CH2S(O)CH2(D1-82a) D1-108a
CH2S(O)CH2(D1-82a) D1-108b(Z=2-Cl)
CH2S(O)CH2(D1-82a) D1-108b(Z=3-Me)
CH2S(O)CH2(D1-82a) D1-108b(Z=4-OMe)
CH2S(O)CH2(D1-82a) D1-108b(Z=2-SMe)
CH2S(O)CH2(D1-82a) D1-108b(Z=3-CF3)
CH2S(O)CH2(D1-82a) D1-108b(Z=4-OCF3)
CH2S(O)CH2(D1-82a) D1-108b(Z=2-SCF3)
CH2S(O)CH2(D1-82a) C(O)Me
CH2S(O)CH2(D1-82a) C(O)CF3
CH2S(O)CH2(D1-82a) C(O)OMe
CH2S(O)2CH2(D1-82a) Me
CH2S(O)2CH2(D1-82a) Et
CH2S(O)2CH2(D1-82a) Pr-n
CH2S(O)2CH2(D1-82a) Pr-i
CH2S(O)2CH2(D1-82a) Pr-c
CH2S(O)2CH2(D1-82a) Bu-n
CH2S(O)2CH2(D1-82a) Bu-i
CH2S(O)2CH2(D1-82a) Bu-c
CH2S(O)2CH2(D1-82a) Bu-s
CH2S(O)2CH2(D1-82a) Bu-t
CH2S(O)2CH2(D1-82a) Pen-n
CH2S(O)2CH2(D1-82a) Pen-c
CH2S(O)2CH2(D1-82a) Hex-n
CH2S(O)2CH2(D1-82a) Hex-c
CH2S(O)2CH2(D1-82a) CH2Pr-c
CH2S(O)2CH2(D1-82a) CH2Bu-c
CH2S(O)2CH2(D1-82a) CH2Pen-c
CH2S(O)2CH2(D1-82a) CH2Hex-c
CH2S(O)2CH2(D1-82a) CH2CH=CH2
CH2S(O)2CH2(D1-82a) CH2CH=C(Cl)2
CH2S(O)2CH2(D1-82a) CH2C≡CH
CH2S(O)2CH2(D1-82a) CH2CN
CH2S(O)2CH2(D1-82a) CH2CF3
CH2S(O)2CH2(D1-82a) CH2OMe
CH2S(O)2CH2(D1-82a) CH2OCF3
CH2S(O)2CH2(D1-82a) CH2SMe
CH2S(O)2CH2(D1-82a) CH2S(O)Me
CH2S(O)2CH2(D1-82a) CH2S(O)2Me
CH2S(O)2CH2(D1-82a) CH2SCF3
CH2S(O)2CH2(D1-82a) CH2S(O)CF3
CH2S(O)2CH2(D1-82a) CH2S(O)2CF3
CH2S(O)2CH2(D1-82a) CH2CH(OMe)2
CH2S(O)2CH2(D1-82a) CH2CH(SMe)2
CH2S(O)2CH2(D1-82a) CH2C(O)Me
CH2S(O)2CH2(D1-82a) CH2C(O)CF3
CH2S(O)2CH2(D1-82a) CH2C(O)OMe
CH2S(O)2CH2(D1-82a) CH2(D1-32a)
CH2S(O)2CH2(D1-82a) CH2(D1-33a)
CH2S(O)2CH2(D1-82a) CH2(D1-34a)
CH2S(O)2CH2(D1-82a) CH2(D1-37a)
CH2S(O)2CH2(D1-82a) CH2(D1-81a)
CH2S(O)2CH2(D1-82a) CH2(D1-82a)
CH2S(O)2CH2(D1-82a) CH2(D1-84a)
CH2S(O)2CH2(D1-82a) CH2(D1-85a)
CH2S(O)2CH2(D1-82a) CH2(D1-87a)
CH2S(O)2CH2(D1-82a) CH2(D1-92a)
CH2S(O)2CH2(D1-82a) CH2(D1-93a)
CH2S(O)2CH2(D1-82a) CH2(D1-95a)
CH2S(O)2CH2(D1-82a) CH2(D1-96a)
CH2S(O)2CH2(D1-82a) CH2(D1-98a)
CH2S(O)2CH2(D1-82a) CH2(D1-108a)
CH2S(O)2CH2(D1-82a) CH2(D1-108b,Z=2-Cl)
CH2S(O)2CH2(D1-82a) CH2(D1-108b,Z=3-Me)
CH2S(O)2CH2(D1-82a) CH2(D1-108b,Z=4-OMe)
CH2S(O)2CH2(D1-82a) CH2(D1-108b,Z=2-SMe)
CH2S(O)2CH2(D1-82a) CH2(D1-108b,Z=3-CF3)
CH2S(O)2CH2(D1-82a) CH2(D1-108b,Z=4-OCF3)
CH2S(O)2CH2(D1-82a) CH2(D1-108b,Z=2-SCF3)
CH2S(O)2CH2(D1-82a) CH2CH2CN
CH2S(O)2CH2(D1-82a) CH2CH2CF3
CH2S(O)2CH2(D1-82a) CH2CH2OMe
CH2S(O)2CH2(D1-82a) CH2CH2SMe
CH2S(O)2CH2(D1-82a) CH2CH2S(O)Me
CH2S(O)2CH2(D1-82a) CH2CH2S(O)2Me
CH2S(O)2CH2(D1-82a) D1-32a
CH2S(O)2CH2(D1-82a) D1-33a
CH2S(O)2CH2(D1-82a) D1-34a
CH2S(O)2CH2(D1-82a) D1-37a
CH2S(O)2CH2(D1-82a) D1-81a
CH2S(O)2CH2(D1-82a) D1-82a
CH2S(O)2CH2(D1-82a) D1-84a
CH2S(O)2CH2(D1-82a) D1-85a
CH2S(O)2CH2(D1-82a) D1-87a
CH2S(O)2CH2(D1-82a) D1-92a
CH2S(O)2CH2(D1-82a) D1-93a
CH2S(O)2CH2(D1-82a) D1-95a
CH2S(O)2CH2(D1-82a) D1-96a
CH2S(O)2CH2(D1-82a) D1-98a
CH2S(O)2CH2(D1-82a) D1-108a
CH2S(O)2CH2(D1-82a) D1-108b(Z=2-Cl)
CH2S(O)2CH2(D1-82a) D1-108b(Z=3-Me)
CH2S(O)2CH2(D1-82a) D1-108b(Z=4-OMe)
CH2S(O)2CH2(D1-82a) D1-108b(Z=2-SMe)
CH2S(O)2CH2(D1-82a) D1-108b(Z=3-CF3)
CH2S(O)2CH2(D1-82a) D1-108b(Z=4-OCF3)
CH2S(O)2CH2(D1-82a) D1-108b(Z=2-SCF3)
CH2S(O)2CH2(D1-82a) C(O)Me
CH2S(O)2CH2(D1-82a) C(O)CF3
CH2S(O)2CH2(D1-82a) C(O)OMe
CH(Me)SCH2(D1-84a) Me
CH(Me)SCH2(D1-84a) Et
CH(Me)SCH2(D1-84a) Pr-n
CH(Me)SCH2(D1-84a) Pr-i
CH(Me)SCH2(D1-84a) Pr-c
CH(Me)SCH2(D1-84a) Bu-n
CH(Me)SCH2(D1-84a) Bu-i
CH(Me)SCH2(D1-84a) Bu-c
CH(Me)SCH2(D1-84a) Bu-s
CH(Me)SCH2(D1-84a) Bu-t
CH(Me)SCH2(D1-84a) Pen-n
CH(Me)SCH2(D1-84a) Pen-c
CH(Me)SCH2(D1-84a) Hex-n
CH(Me)SCH2(D1-84a) Hex-c
CH(Me)SCH2(D1-84a) CH2Pr-c
CH(Me)SCH2(D1-84a) CH2Bu-c
CH(Me)SCH2(D1-84a) CH2Pen-c
CH(Me)SCH2(D1-84a) CH2Hex-c
CH(Me)SCH2(D1-84a) CH2CH=CH2
CH(Me)SCH2(D1-84a) CH2CH=C(Cl)2
CH(Me)SCH2(D1-84a) CH2C≡CH
CH(Me)SCH2(D1-84a) CH2CN
CH(Me)SCH2(D1-84a) CH2CF3
CH(Me)SCH2(D1-84a) CH2OMe
CH(Me)SCH2(D1-84a) CH2OCF3
CH(Me)SCH2(D1-84a) CH2SMe
CH(Me)SCH2(D1-84a) CH2S(O)Me
CH(Me)SCH2(D1-84a) CH2S(O)2Me
CH(Me)SCH2(D1-84a) CH2SCF3
CH(Me)SCH2(D1-84a) CH2S(O)CF3
CH(Me)SCH2(D1-84a) CH2S(O)2CF3
CH(Me)SCH2(D1-84a) CH2CH(OMe)2
CH(Me)SCH2(D1-84a) CH2CH(SMe)2
CH(Me)SCH2(D1-84a) CH2C(O)Me
CH(Me)SCH2(D1-84a) CH2C(O)CF3
CH(Me)SCH2(D1-84a) CH2C(O)OMe
CH(Me)SCH2(D1-84a) CH2(D1-32a)
CH(Me)SCH2(D1-84a) CH2(D1-33a)
CH(Me)SCH2(D1-84a) CH2(D1-34a)
CH(Me)SCH2(D1-84a) CH2(D1-37a)
CH(Me)SCH2(D1-84a) CH2(D1-81a)
CH(Me)SCH2(D1-84a) CH2(D1-82a)
CH(Me)SCH2(D1-84a) CH2(D1-84a)
CH(Me)SCH2(D1-84a) CH2(D1-85a)
CH(Me)SCH2(D1-84a) CH2(D1-87a)
CH(Me)SCH2(D1-84a) CH2(D1-92a)
CH(Me)SCH2(D1-84a) CH2(D1-93a)
CH(Me)SCH2(D1-84a) CH2(D1-95a)
CH(Me)SCH2(D1-84a) CH2(D1-96a)
CH(Me)SCH2(D1-84a) CH2(D1-98a)
CH(Me)SCH2(D1-84a) CH2(D1-108a)
CH(Me)SCH2(D1-84a) CH2(D1-108b,Z=2-Cl)
CH(Me)SCH2(D1-84a) CH2(D1-108b,Z=3-Me)
CH(Me)SCH2(D1-84a) CH2(D1-108b,Z=4-OMe)
CH(Me)SCH2(D1-84a) CH2(D1-108b,Z=2-SMe)
CH(Me)SCH2(D1-84a) CH2(D1-108b,Z=3-CF3)
CH(Me)SCH2(D1-84a) CH2(D1-108b,Z=4-OCF3)
CH(Me)SCH2(D1-84a) CH2(D1-108b,Z=2-SCF3)
CH(Me)SCH2(D1-84a) CH2CH2CN
CH(Me)SCH2(D1-84a) CH2CH2CF3
CH(Me)SCH2(D1-84a) CH2CH2OMe
CH(Me)SCH2(D1-84a) CH2CH2SMe
CH(Me)SCH2(D1-84a) CH2CH2S(O)Me
CH(Me)SCH2(D1-84a) CH2CH2S(O)2Me
CH(Me)SCH2(D1-84a) D1-32a
CH(Me)SCH2(D1-84a) D1-33a
CH(Me)SCH2(D1-84a) D1-34a
CH(Me)SCH2(D1-84a) D1-37a
CH(Me)SCH2(D1-84a) D1-81a
CH(Me)SCH2(D1-84a) D1-82a
CH(Me)SCH2(D1-84a) D1-84a
CH(Me)SCH2(D1-84a) D1-85a
CH(Me)SCH2(D1-84a) D1-87a
CH(Me)SCH2(D1-84a) D1-92a
CH(Me)SCH2(D1-84a) D1-93a
CH(Me)SCH2(D1-84a) D1-95a
CH(Me)SCH2(D1-84a) D1-96a
CH(Me)SCH2(D1-84a) D1-98a
CH(Me)SCH2(D1-84a) D1-108a
CH(Me)SCH2(D1-84a) D1-108b(Z=2-Cl)
CH(Me)SCH2(D1-84a) D1-108b(Z=3-Me)
CH(Me)SCH2(D1-84a) D1-108b(Z=4-OMe)
CH(Me)SCH2(D1-84a) D1-108b(Z=2-SMe)
CH(Me)SCH2(D1-84a) D1-108b(Z=3-CF3)
CH(Me)SCH2(D1-84a) D1-108b(Z=4-OCF3)
CH(Me)SCH2(D1-84a) D1-108b(Z=2-SCF3)
CH(Me)SCH2(D1-84a) C(O)Me
CH(Me)SCH2(D1-84a) C(O)CF3
CH(Me)SCH2(D1-84a) C(O)OMe
CH(Me)S(O)CH2(D1-84a) Me
CH(Me)S(O)CH2(D1-84a) Et
CH(Me)S(O)CH2(D1-84a) Pr-n
CH(Me)S(O)CH2(D1-84a) Pr-i
CH(Me)S(O)CH2(D1-84a) Pr-c
CH(Me)S(O)CH2(D1-84a) Bu-n
CH(Me)S(O)CH2(D1-84a) Bu-i
CH(Me)S(O)CH2(D1-84a) Bu-c
CH(Me)S(O)CH2(D1-84a) Bu-s
CH(Me)S(O)CH2(D1-84a) Bu-t
CH(Me)S(O)CH2(D1-84a) Pen-n
CH(Me)S(O)CH2(D1-84a) Pen-c
CH(Me)S(O)CH2(D1-84a) Hex-n
CH(Me)S(O)CH2(D1-84a) Hex-c
CH(Me)S(O)CH2(D1-84a) CH2Pr-c
CH(Me)S(O)CH2(D1-84a) CH2Bu-c
CH(Me)S(O)CH2(D1-84a) CH2Pen-c
CH(Me)S(O)CH2(D1-84a) CH2Hex-c
CH(Me)S(O)CH2(D1-84a) CH2CH=CH2
CH(Me)S(O)CH2(D1-84a) CH2CH=C(Cl)2
CH(Me)S(O)CH2(D1-84a) CH2C≡CH
CH(Me)S(O)CH2(D1-84a) CH2CN
CH(Me)S(O)CH2(D1-84a) CH2CF3
CH(Me)S(O)CH2(D1-84a) CH2OMe
CH(Me)S(O)CH2(D1-84a) CH2OCF3
CH(Me)S(O)CH2(D1-84a) CH2SMe
CH(Me)S(O)CH2(D1-84a) CH2S(O)Me
CH(Me)S(O)CH2(D1-84a) CH2S(O)2Me
CH(Me)S(O)CH2(D1-84a) CH2SCF3
CH(Me)S(O)CH2(D1-84a) CH2S(O)CF3
CH(Me)S(O)CH2(D1-84a) CH2S(O)2CF3
CH(Me)S(O)CH2(D1-84a) CH2CH(OMe)2
CH(Me)S(O)CH2(D1-84a) CH2CH(SMe)2
CH(Me)S(O)CH2(D1-84a) CH2C(O)Me
CH(Me)S(O)CH2(D1-84a) CH2C(O)CF3
CH(Me)S(O)CH2(D1-84a) CH2C(O)OMe
CH(Me)S(O)CH2(D1-84a) CH2(D1-32a)
CH(Me)S(O)CH2(D1-84a) CH2(D1-33a)
CH(Me)S(O)CH2(D1-84a) CH2(D1-34a)
CH(Me)S(O)CH2(D1-84a) CH2(D1-37a)
CH(Me)S(O)CH2(D1-84a) CH2(D1-81a)
CH(Me)S(O)CH2(D1-84a) CH2(D1-82a)
CH(Me)S(O)CH2(D1-84a) CH2(D1-84a)
CH(Me)S(O)CH2(D1-84a) CH2(D1-85a)
CH(Me)S(O)CH2(D1-84a) CH2(D1-87a)
CH(Me)S(O)CH2(D1-84a) CH2(D1-92a)
CH(Me)S(O)CH2(D1-84a) CH2(D1-93a)
CH(Me)S(O)CH2(D1-84a) CH2(D1-95a)
CH(Me)S(O)CH2(D1-84a) CH2(D1-96a)
CH(Me)S(O)CH2(D1-84a) CH2(D1-98a)
CH(Me)S(O)CH2(D1-84a) CH2(D1-108a)
CH(Me)S(O)CH2(D1-84a) CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)CH2(D1-84a) CH2(D1-108b,Z=3-Me)
CH(Me)S(O)CH2(D1-84a) CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)CH2(D1-84a) CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)CH2(D1-84a) CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)CH2(D1-84a) CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)CH2(D1-84a) CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)CH2(D1-84a) CH2CH2CN
CH(Me)S(O)CH2(D1-84a) CH2CH2CF3
CH(Me)S(O)CH2(D1-84a) CH2CH2OMe
CH(Me)S(O)CH2(D1-84a) CH2CH2SMe
CH(Me)S(O)CH2(D1-84a) CH2CH2S(O)Me
CH(Me)S(O)CH2(D1-84a) CH2CH2S(O)2Me
CH(Me)S(O)CH2(D1-84a) D1-32a
CH(Me)S(O)CH2(D1-84a) D1-33a
CH(Me)S(O)CH2(D1-84a) D1-34a
CH(Me)S(O)CH2(D1-84a) D1-37a
CH(Me)S(O)CH2(D1-84a) D1-81a
CH(Me)S(O)CH2(D1-84a) D1-82a
CH(Me)S(O)CH2(D1-84a) D1-84a
CH(Me)S(O)CH2(D1-84a) D1-85a
CH(Me)S(O)CH2(D1-84a) D1-87a
CH(Me)S(O)CH2(D1-84a) D1-92a
CH(Me)S(O)CH2(D1-84a) D1-93a
CH(Me)S(O)CH2(D1-84a) D1-95a
CH(Me)S(O)CH2(D1-84a) D1-96a
CH(Me)S(O)CH2(D1-84a) D1-98a
CH(Me)S(O)CH2(D1-84a) D1-108a
CH(Me)S(O)CH2(D1-84a) D1-108b(Z=2-Cl)
CH(Me)S(O)CH2(D1-84a) D1-108b(Z=3-Me)
CH(Me)S(O)CH2(D1-84a) D1-108b(Z=4-OMe)
CH(Me)S(O)CH2(D1-84a) D1-108b(Z=2-SMe)
CH(Me)S(O)CH2(D1-84a) D1-108b(Z=3-CF3)
CH(Me)S(O)CH2(D1-84a) D1-108b(Z=4-OCF3)
CH(Me)S(O)CH2(D1-84a) D1-108b(Z=2-SCF3)
CH(Me)S(O)CH2(D1-84a) C(O)Me
CH(Me)S(O)CH2(D1-84a) C(O)CF3
CH(Me)S(O)CH2(D1-84a) C(O)OMe
CH(Me)S(O)2CH2(D1-84a) Me
CH(Me)S(O)2CH2(D1-84a) Et
CH(Me)S(O)2CH2(D1-84a) Pr-n
CH(Me)S(O)2CH2(D1-84a) Pr-i
CH(Me)S(O)2CH2(D1-84a) Pr-c
CH(Me)S(O)2CH2(D1-84a) Bu-n
CH(Me)S(O)2CH2(D1-84a) Bu-i
CH(Me)S(O)2CH2(D1-84a) Bu-c
CH(Me)S(O)2CH2(D1-84a) Bu-s
CH(Me)S(O)2CH2(D1-84a) Bu-t
CH(Me)S(O)2CH2(D1-84a) Pen-n
CH(Me)S(O)2CH2(D1-84a) Pen-c
CH(Me)S(O)2CH2(D1-84a) Hex-n
CH(Me)S(O)2CH2(D1-84a) Hex-c
CH(Me)S(O)2CH2(D1-84a) CH2Pr-c
CH(Me)S(O)2CH2(D1-84a) CH2Bu-c
CH(Me)S(O)2CH2(D1-84a) CH2Pen-c
CH(Me)S(O)2CH2(D1-84a) CH2Hex-c
CH(Me)S(O)2CH2(D1-84a) CH2CH=CH2
CH(Me)S(O)2CH2(D1-84a) CH2CH=C(Cl)2
CH(Me)S(O)2CH2(D1-84a) CH2C≡CH
CH(Me)S(O)2CH2(D1-84a) CH2CN
CH(Me)S(O)2CH2(D1-84a) CH2CF3
CH(Me)S(O)2CH2(D1-84a) CH2OMe
CH(Me)S(O)2CH2(D1-84a) CH2OCF3
CH(Me)S(O)2CH2(D1-84a) CH2SMe
CH(Me)S(O)2CH2(D1-84a) CH2S(O)Me
CH(Me)S(O)2CH2(D1-84a) CH2S(O)2Me
CH(Me)S(O)2CH2(D1-84a) CH2SCF3
CH(Me)S(O)2CH2(D1-84a) CH2S(O)CF3
CH(Me)S(O)2CH2(D1-84a) CH2S(O)2CF3
CH(Me)S(O)2CH2(D1-84a) CH2CH(OMe)2
CH(Me)S(O)2CH2(D1-84a) CH2CH(SMe)2
CH(Me)S(O)2CH2(D1-84a) CH2C(O)Me
CH(Me)S(O)2CH2(D1-84a) CH2C(O)CF3
CH(Me)S(O)2CH2(D1-84a) CH2C(O)OMe
CH(Me)S(O)2CH2(D1-84a) CH2(D1-32a)
CH(Me)S(O)2CH2(D1-84a) CH2(D1-33a)
CH(Me)S(O)2CH2(D1-84a) CH2(D1-34a)
CH(Me)S(O)2CH2(D1-84a) CH2(D1-37a)
CH(Me)S(O)2CH2(D1-84a) CH2(D1-81a)
CH(Me)S(O)2CH2(D1-84a) CH2(D1-82a)
CH(Me)S(O)2CH2(D1-84a) CH2(D1-84a)
CH(Me)S(O)2CH2(D1-84a) CH2(D1-85a)
CH(Me)S(O)2CH2(D1-84a) CH2(D1-87a)
CH(Me)S(O)2CH2(D1-84a) CH2(D1-92a)
CH(Me)S(O)2CH2(D1-84a) CH2(D1-93a)
CH(Me)S(O)2CH2(D1-84a) CH2(D1-95a)
CH(Me)S(O)2CH2(D1-84a) CH2(D1-96a)
CH(Me)S(O)2CH2(D1-84a) CH2(D1-98a)
CH(Me)S(O)2CH2(D1-84a) CH2(D1-108a)
CH(Me)S(O)2CH2(D1-84a) CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)2CH2(D1-84a) CH2(D1-108b,Z=3-Me)
CH(Me)S(O)2CH2(D1-84a) CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)2CH2(D1-84a) CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)2CH2(D1-84a) CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)2CH2(D1-84a) CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)2CH2(D1-84a) CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)2CH2(D1-84a) CH2CH2CN
CH(Me)S(O)2CH2(D1-84a) CH2CH2CF3
CH(Me)S(O)2CH2(D1-84a) CH2CH2OMe
CH(Me)S(O)2CH2(D1-84a) CH2CH2SMe
CH(Me)S(O)2CH2(D1-84a) CH2CH2S(O)Me
CH(Me)S(O)2CH2(D1-84a) CH2CH2S(O)2Me
CH(Me)S(O)2CH2(D1-84a) D1-32a
CH(Me)S(O)2CH2(D1-84a) D1-33a
CH(Me)S(O)2CH2(D1-84a) D1-34a
CH(Me)S(O)2CH2(D1-84a) D1-37a
CH(Me)S(O)2CH2(D1-84a) D1-81a
CH(Me)S(O)2CH2(D1-84a) D1-82a
CH(Me)S(O)2CH2(D1-84a) D1-84a
CH(Me)S(O)2CH2(D1-84a) D1-85a
CH(Me)S(O)2CH2(D1-84a) D1-87a
CH(Me)S(O)2CH2(D1-84a) D1-92a
CH(Me)S(O)2CH2(D1-84a) D1-93a
CH(Me)S(O)2CH2(D1-84a) D1-95a
CH(Me)S(O)2CH2(D1-84a) D1-96a
CH(Me)S(O)2CH2(D1-84a) D1-98a
CH(Me)S(O)2CH2(D1-84a) D1-108a
CH(Me)S(O)2CH2(D1-84a) D1-108b(Z=2-Cl)
CH(Me)S(O)2CH2(D1-84a) D1-108b(Z=3-Me)
CH(Me)S(O)2CH2(D1-84a) D1-108b(Z=4-OMe)
CH(Me)S(O)2CH2(D1-84a) D1-108b(Z=2-SMe)
CH(Me)S(O)2CH2(D1-84a) D1-108b(Z=3-CF3)
CH(Me)S(O)2CH2(D1-84a) D1-108b(Z=4-OCF3)
CH(Me)S(O)2CH2(D1-84a) D1-108b(Z=2-SCF3)
CH(Me)S(O)2CH2(D1-84a) C(O)Me
CH(Me)S(O)2CH2(D1-84a) C(O)CF3
CH(Me)S(O)2CH2(D1-84a) C(O)OMe
CH2SCH2(D1-85a) Me
CH2SCH2(D1-85a) Et
CH2SCH2(D1-85a) Pr-n
CH2SCH2(D1-85a) Pr-i
CH2SCH2(D1-85a) Pr-c
CH2SCH2(D1-85a) Bu-n
CH2SCH2(D1-85a) Bu-i
CH2SCH2(D1-85a) Bu-c
CH2SCH2(D1-85a) Bu-s
CH2SCH2(D1-85a) Bu-t
CH2SCH2(D1-85a) Pen-n
CH2SCH2(D1-85a) Pen-c
CH2SCH2(D1-85a) Hex-n
CH2SCH2(D1-85a) Hex-c
CH2SCH2(D1-85a) CH2Pr-c
CH2SCH2(D1-85a) CH2Bu-c
CH2SCH2(D1-85a) CH2Pen-c
CH2SCH2(D1-85a) CH2Hex-c
CH2SCH2(D1-85a) CH2CH=CH2
CH2SCH2(D1-85a) CH2CH=C(Cl)2
CH2SCH2(D1-85a) CH2C≡CH
CH2SCH2(D1-85a) CH2CN
CH2SCH2(D1-85a) CH2CF3
CH2SCH2(D1-85a) CH2OMe
CH2SCH2(D1-85a) CH2OCF3
CH2SCH2(D1-85a) CH2SMe
CH2SCH2(D1-85a) CH2S(O)Me
CH2SCH2(D1-85a) CH2S(O)2Me
CH2SCH2(D1-85a) CH2SCF3
CH2SCH2(D1-85a) CH2S(O)CF3
CH2SCH2(D1-85a) CH2S(O)2CF3
CH2SCH2(D1-85a) CH2CH(OMe)2
CH2SCH2(D1-85a) CH2CH(SMe)2
CH2SCH2(D1-85a) CH2C(O)Me
CH2SCH2(D1-85a) CH2C(O)CF3
CH2SCH2(D1-85a) CH2C(O)OMe
CH2SCH2(D1-85a) CH2(D1-32a)
CH2SCH2(D1-85a) CH2(D1-33a)
CH2SCH2(D1-85a) CH2(D1-34a)
CH2SCH2(D1-85a) CH2(D1-37a)
CH2SCH2(D1-85a) CH2(D1-81a)
CH2SCH2(D1-85a) CH2(D1-82a)
CH2SCH2(D1-85a) CH2(D1-84a)
CH2SCH2(D1-85a) CH2(D1-85a)
CH2SCH2(D1-85a) CH2(D1-87a)
CH2SCH2(D1-85a) CH2(D1-92a)
CH2SCH2(D1-85a) CH2(D1-93a)
CH2SCH2(D1-85a) CH2(D1-95a)
CH2SCH2(D1-85a) CH2(D1-96a)
CH2SCH2(D1-85a) CH2(D1-98a)
CH2SCH2(D1-85a) CH2(D1-108a)
CH2SCH2(D1-85a) CH2(D1-108b,Z=2-Cl)
CH2SCH2(D1-85a) CH2(D1-108b,Z=3-Me)
CH2SCH2(D1-85a) CH2(D1-108b,Z=4-OMe)
CH2SCH2(D1-85a) CH2(D1-108b,Z=2-SMe)
CH2SCH2(D1-85a) CH2(D1-108b,Z=3-CF3)
CH2SCH2(D1-85a) CH2(D1-108b,Z=4-OCF3)
CH2SCH2(D1-85a) CH2(D1-108b,Z=2-SCF3)
CH2SCH2(D1-85a) CH2CH2CN
CH2SCH2(D1-85a) CH2CH2CF3
CH2SCH2(D1-85a) CH2CH2OMe
CH2SCH2(D1-85a) CH2CH2SMe
CH2SCH2(D1-85a) CH2CH2S(O)Me
CH2SCH2(D1-85a) CH2CH2S(O)2Me
CH2SCH2(D1-85a) D1-32a
CH2SCH2(D1-85a) D1-33a
CH2SCH2(D1-85a) D1-34a
CH2SCH2(D1-85a) D1-37a
CH2SCH2(D1-85a) D1-81a
CH2SCH2(D1-85a) D1-82a
CH2SCH2(D1-85a) D1-84a
CH2SCH2(D1-85a) D1-85a
CH2SCH2(D1-85a) D1-87a
CH2SCH2(D1-85a) D1-92a
CH2SCH2(D1-85a) D1-93a
CH2SCH2(D1-85a) D1-95a
CH2SCH2(D1-85a) D1-96a
CH2SCH2(D1-85a) D1-98a
CH2SCH2(D1-85a) D1-108a
CH2SCH2(D1-85a) D1-108b(Z=2-Cl)
CH2SCH2(D1-85a) D1-108b(Z=3-Me)
CH2SCH2(D1-85a) D1-108b(Z=4-OMe)
CH2SCH2(D1-85a) D1-108b(Z=2-SMe)
CH2SCH2(D1-85a) D1-108b(Z=3-CF3)
CH2SCH2(D1-85a) D1-108b(Z=4-OCF3)
CH2SCH2(D1-85a) D1-108b(Z=2-SCF3)
CH2SCH2(D1-85a) C(O)Me
CH2SCH2(D1-85a) C(O)CF3
CH2SCH2(D1-85a) C(O)OMe
CH2S(O)CH2(D1-85a) Me
CH2S(O)CH2(D1-85a) Et
CH2S(O)CH2(D1-85a) Pr-n
CH2S(O)CH2(D1-85a) Pr-i
CH2S(O)CH2(D1-85a) Pr-c
CH2S(O)CH2(D1-85a) Bu-n
CH2S(O)CH2(D1-85a) Bu-i
CH2S(O)CH2(D1-85a) Bu-c
CH2S(O)CH2(D1-85a) Bu-s
CH2S(O)CH2(D1-85a) Bu-t
CH2S(O)CH2(D1-85a) Pen-n
CH2S(O)CH2(D1-85a) Pen-c
CH2S(O)CH2(D1-85a) Hex-n
CH2S(O)CH2(D1-85a) Hex-c
CH2S(O)CH2(D1-85a) CH2Pr-c
CH2S(O)CH2(D1-85a) CH2Bu-c
CH2S(O)CH2(D1-85a) CH2Pen-c
CH2S(O)CH2(D1-85a) CH2Hex-c
CH2S(O)CH2(D1-85a) CH2CH=CH2
CH2S(O)CH2(D1-85a) CH2CH=C(Cl)2
CH2S(O)CH2(D1-85a) CH2C≡CH
CH2S(O)CH2(D1-85a) CH2CN
CH2S(O)CH2(D1-85a) CH2CF3
CH2S(O)CH2(D1-85a) CH2OMe
CH2S(O)CH2(D1-85a) CH2OCF3
CH2S(O)CH2(D1-85a) CH2SMe
CH2S(O)CH2(D1-85a) CH2S(O)Me
CH2S(O)CH2(D1-85a) CH2S(O)2Me
CH2S(O)CH2(D1-85a) CH2SCF3
CH2S(O)CH2(D1-85a) CH2S(O)CF3
CH2S(O)CH2(D1-85a) CH2S(O)2CF3
CH2S(O)CH2(D1-85a) CH2CH(OMe)2
CH2S(O)CH2(D1-85a) CH2CH(SMe)2
CH2S(O)CH2(D1-85a) CH2C(O)Me
CH2S(O)CH2(D1-85a) CH2C(O)CF3
CH2S(O)CH2(D1-85a) CH2C(O)OMe
CH2S(O)CH2(D1-85a) CH2(D1-32a)
CH2S(O)CH2(D1-85a) CH2(D1-33a)
CH2S(O)CH2(D1-85a) CH2(D1-34a)
CH2S(O)CH2(D1-85a) CH2(D1-37a)
CH2S(O)CH2(D1-85a) CH2(D1-81a)
CH2S(O)CH2(D1-85a) CH2(D1-82a)
CH2S(O)CH2(D1-85a) CH2(D1-84a)
CH2S(O)CH2(D1-85a) CH2(D1-85a)
CH2S(O)CH2(D1-85a) CH2(D1-87a)
CH2S(O)CH2(D1-85a) CH2(D1-92a)
CH2S(O)CH2(D1-85a) CH2(D1-93a)
CH2S(O)CH2(D1-85a) CH2(D1-95a)
CH2S(O)CH2(D1-85a) CH2(D1-96a)
CH2S(O)CH2(D1-85a) CH2(D1-98a)
CH2S(O)CH2(D1-85a) CH2(D1-108a)
CH2S(O)CH2(D1-85a) CH2(D1-108b,Z=2-Cl)
CH2S(O)CH2(D1-85a) CH2(D1-108b,Z=3-Me)
CH2S(O)CH2(D1-85a) CH2(D1-108b,Z=4-OMe)
CH2S(O)CH2(D1-85a) CH2(D1-108b,Z=2-SMe)
CH2S(O)CH2(D1-85a) CH2(D1-108b,Z=3-CF3)
CH2S(O)CH2(D1-85a) CH2(D1-108b,Z=4-OCF3)
CH2S(O)CH2(D1-85a) CH2(D1-108b,Z=2-SCF3)
CH2S(O)CH2(D1-85a) CH2CH2CN
CH2S(O)CH2(D1-85a) CH2CH2CF3
CH2S(O)CH2(D1-85a) CH2CH2OMe
CH2S(O)CH2(D1-85a) CH2CH2SMe
CH2S(O)CH2(D1-85a) CH2CH2S(O)Me
CH2S(O)CH2(D1-85a) CH2CH2S(O)2Me
CH2S(O)CH2(D1-85a) D1-32a
CH2S(O)CH2(D1-85a) D1-33a
CH2S(O)CH2(D1-85a) D1-34a
CH2S(O)CH2(D1-85a) D1-37a
CH2S(O)CH2(D1-85a) D1-81a
CH2S(O)CH2(D1-85a) D1-82a
CH2S(O)CH2(D1-85a) D1-84a
CH2S(O)CH2(D1-85a) D1-85a
CH2S(O)CH2(D1-85a) D1-87a
CH2S(O)CH2(D1-85a) D1-92a
CH2S(O)CH2(D1-85a) D1-93a
CH2S(O)CH2(D1-85a) D1-95a
CH2S(O)CH2(D1-85a) D1-96a
CH2S(O)CH2(D1-85a) D1-98a
CH2S(O)CH2(D1-85a) D1-108a
CH2S(O)CH2(D1-85a) D1-108b(Z=2-Cl)
CH2S(O)CH2(D1-85a) D1-108b(Z=3-Me)
CH2S(O)CH2(D1-85a) D1-108b(Z=4-OMe)
CH2S(O)CH2(D1-85a) D1-108b(Z=2-SMe)
CH2S(O)CH2(D1-85a) D1-108b(Z=3-CF3)
CH2S(O)CH2(D1-85a) D1-108b(Z=4-OCF3)
CH2S(O)CH2(D1-85a) D1-108b(Z=2-SCF3)
CH2S(O)CH2(D1-85a) C(O)Me
CH2S(O)CH2(D1-85a) C(O)CF3
CH2S(O)CH2(D1-85a) C(O)OMe
CH2S(O)2CH2(D1-85a) Me
CH2S(O)2CH2(D1-85a) Et
CH2S(O)2CH2(D1-85a) Pr-n
CH2S(O)2CH2(D1-85a) Pr-i
CH2S(O)2CH2(D1-85a) Pr-c
CH2S(O)2CH2(D1-85a) Bu-n
CH2S(O)2CH2(D1-85a) Bu-i
CH2S(O)2CH2(D1-85a) Bu-c
CH2S(O)2CH2(D1-85a) Bu-s
CH2S(O)2CH2(D1-85a) Bu-t
CH2S(O)2CH2(D1-85a) Pen-n
CH2S(O)2CH2(D1-85a) Pen-c
CH2S(O)2CH2(D1-85a) Hex-n
CH2S(O)2CH2(D1-85a) Hex-c
CH2S(O)2CH2(D1-85a) CH2Pr-c
CH2S(O)2CH2(D1-85a) CH2Bu-c
CH2S(O)2CH2(D1-85a) CH2Pen-c
CH2S(O)2CH2(D1-85a) CH2Hex-c
CH2S(O)2CH2(D1-85a) CH2CH=CH2
CH2S(O)2CH2(D1-85a) CH2CH=C(Cl)2
CH2S(O)2CH2(D1-85a) CH2C≡CH
CH2S(O)2CH2(D1-85a) CH2CN
CH2S(O)2CH2(D1-85a) CH2CF3
CH2S(O)2CH2(D1-85a) CH2OMe
CH2S(O)2CH2(D1-85a) CH2OCF3
CH2S(O)2CH2(D1-85a) CH2SMe
CH2S(O)2CH2(D1-85a) CH2S(O)Me
CH2S(O)2CH2(D1-85a) CH2S(O)2Me
CH2S(O)2CH2(D1-85a) CH2SCF3
CH2S(O)2CH2(D1-85a) CH2S(O)CF3
CH2S(O)2CH2(D1-85a) CH2S(O)2CF3
CH2S(O)2CH2(D1-85a) CH2CH(OMe)2
CH2S(O)2CH2(D1-85a) CH2CH(SMe)2
CH2S(O)2CH2(D1-85a) CH2C(O)Me
CH2S(O)2CH2(D1-85a) CH2C(O)CF3
CH2S(O)2CH2(D1-85a) CH2C(O)OMe
CH2S(O)2CH2(D1-85a) CH2(D1-32a)
CH2S(O)2CH2(D1-85a) CH2(D1-33a)
CH2S(O)2CH2(D1-85a) CH2(D1-34a)
CH2S(O)2CH2(D1-85a) CH2(D1-37a)
CH2S(O)2CH2(D1-85a) CH2(D1-81a)
CH2S(O)2CH2(D1-85a) CH2(D1-82a)
CH2S(O)2CH2(D1-85a) CH2(D1-84a)
CH2S(O)2CH2(D1-85a) CH2(D1-85a)
CH2S(O)2CH2(D1-85a) CH2(D1-87a)
CH2S(O)2CH2(D1-85a) CH2(D1-92a)
CH2S(O)2CH2(D1-85a) CH2(D1-93a)
CH2S(O)2CH2(D1-85a) CH2(D1-95a)
CH2S(O)2CH2(D1-85a) CH2(D1-96a)
CH2S(O)2CH2(D1-85a) CH2(D1-98a)
CH2S(O)2CH2(D1-85a) CH2(D1-108a)
CH2S(O)2CH2(D1-85a) CH2(D1-108b,Z=2-Cl)
CH2S(O)2CH2(D1-85a) CH2(D1-108b,Z=3-Me)
CH2S(O)2CH2(D1-85a) CH2(D1-108b,Z=4-OMe)
CH2S(O)2CH2(D1-85a) CH2(D1-108b,Z=2-SMe)
CH2S(O)2CH2(D1-85a) CH2(D1-108b,Z=3-CF3)
CH2S(O)2CH2(D1-85a) CH2(D1-108b,Z=4-OCF3)
CH2S(O)2CH2(D1-85a) CH2(D1-108b,Z=2-SCF3)
CH2S(O)2CH2(D1-85a) CH2CH2CN
CH2S(O)2CH2(D1-85a) CH2CH2CF3
CH2S(O)2CH2(D1-85a) CH2CH2OMe
CH2S(O)2CH2(D1-85a) CH2CH2SMe
CH2S(O)2CH2(D1-85a) CH2CH2S(O)Me
CH2S(O)2CH2(D1-85a) CH2CH2S(O)2Me
CH2S(O)2CH2(D1-85a) D1-32a
CH2S(O)2CH2(D1-85a) D1-33a
CH2S(O)2CH2(D1-85a) D1-34a
CH2S(O)2CH2(D1-85a) D1-37a
CH2S(O)2CH2(D1-85a) D1-81a
CH2S(O)2CH2(D1-85a) D1-82a
CH2S(O)2CH2(D1-85a) D1-84a
CH2S(O)2CH2(D1-85a) D1-85a
CH2S(O)2CH2(D1-85a) D1-87a
CH2S(O)2CH2(D1-85a) D1-92a
CH2S(O)2CH2(D1-85a) D1-93a
CH2S(O)2CH2(D1-85a) D1-95a
CH2S(O)2CH2(D1-85a) D1-96a
CH2S(O)2CH2(D1-85a) D1-98a
CH2S(O)2CH2(D1-85a) D1-108a
CH2S(O)2CH2(D1-85a) D1-108b(Z=2-Cl)
CH2S(O)2CH2(D1-85a) D1-108b(Z=3-Me)
CH2S(O)2CH2(D1-85a) D1-108b(Z=4-OMe)
CH2S(O)2CH2(D1-85a) D1-108b(Z=2-SMe)
CH2S(O)2CH2(D1-85a) D1-108b(Z=3-CF3)
CH2S(O)2CH2(D1-85a) D1-108b(Z=4-OCF3)
CH2S(O)2CH2(D1-85a) D1-108b(Z=2-SCF3)
CH2SCH2(D1-87a) Me
CH2SCH2(D1-87a) Et
CH2SCH2(D1-87a) Pr-n
CH2SCH2(D1-87a) Pr-i
CH2SCH2(D1-87a) Pr-c
CH2SCH2(D1-87a) Bu-n
CH2SCH2(D1-87a) Bu-i
CH2SCH2(D1-87a) Bu-c
CH2SCH2(D1-87a) Bu-s
CH2SCH2(D1-87a) Bu-t
CH2SCH2(D1-87a) Pen-n
CH2SCH2(D1-87a) Pen-c
CH2SCH2(D1-87a) Hex-n
CH2SCH2(D1-87a) Hex-c
CH2SCH2(D1-87a) CH2Pr-c
CH2SCH2(D1-87a) CH2Bu-c
CH2SCH2(D1-87a) CH2Pen-c
CH2SCH2(D1-87a) CH2Hex-c
CH2SCH2(D1-87a) CH2CH=CH2
CH2SCH2(D1-87a) CH2CH=C(Cl)2
CH2SCH2(D1-87a) CH2C≡CH
CH2SCH2(D1-87a) CH2CN
CH2SCH2(D1-87a) CH2CF3
CH2SCH2(D1-87a) CH2OMe
CH2SCH2(D1-87a) CH2OCF3
CH2SCH2(D1-87a) CH2SMe
CH2SCH2(D1-87a) CH2S(O)Me
CH2SCH2(D1-87a) CH2S(O)2Me
CH2SCH2(D1-87a) CH2SCF3
CH2SCH2(D1-87a) CH2S(O)CF3
CH2SCH2(D1-87a) CH2S(O)2CF3
CH2SCH2(D1-87a) CH2CH(OMe)2
CH2SCH2(D1-87a) CH2CH(SMe)2
CH2SCH2(D1-87a) CH2C(O)Me
CH2SCH2(D1-87a) CH2C(O)CF3
CH2SCH2(D1-87a) CH2C(O)OMe
CH2SCH2(D1-87a) CH2(D1-32a)
CH2SCH2(D1-87a) CH2(D1-33a)
CH2SCH2(D1-87a) CH2(D1-34a)
CH2SCH2(D1-87a) CH2(D1-37a)
CH2SCH2(D1-87a) CH2(D1-81a)
CH2SCH2(D1-87a) CH2(D1-82a)
CH2SCH2(D1-87a) CH2(D1-84a)
CH2SCH2(D1-87a) CH2(D1-85a)
CH2SCH2(D1-87a) CH2(D1-87a)
CH2SCH2(D1-87a) CH2(D1-92a)
CH2SCH2(D1-87a) CH2(D1-93a)
CH2SCH2(D1-87a) CH2(D1-95a)
CH2SCH2(D1-87a) CH2(D1-96a)
CH2SCH2(D1-87a) CH2(D1-98a)
CH2SCH2(D1-87a) CH2(D1-108a)
CH2SCH2(D1-87a) CH2(D1-108b,Z=2-Cl)
CH2SCH2(D1-87a) CH2(D1-108b,Z=3-Me)
CH2SCH2(D1-87a) CH2(D1-108b,Z=4-OMe)
CH2SCH2(D1-87a) CH2(D1-108b,Z=2-SMe)
CH2SCH2(D1-87a) CH2(D1-108b,Z=3-CF3)
CH2SCH2(D1-87a) CH2(D1-108b,Z=4-OCF3)
CH2SCH2(D1-87a) CH2(D1-108b,Z=2-SCF3)
CH2SCH2(D1-87a) CH2CH2CN
CH2SCH2(D1-87a) CH2CH2CF3
CH2SCH2(D1-87a) CH2CH2OMe
CH2SCH2(D1-87a) CH2CH2SMe
CH2SCH2(D1-87a) CH2CH2S(O)Me
CH2SCH2(D1-87a) CH2CH2S(O)2Me
CH2SCH2(D1-87a) D1-32a
CH2SCH2(D1-87a) D1-33a
CH2SCH2(D1-87a) D1-34a
CH2SCH2(D1-87a) D1-37a
CH2SCH2(D1-87a) D1-81a
CH2SCH2(D1-87a) D1-82a
CH2SCH2(D1-87a) D1-84a
CH2SCH2(D1-87a) D1-85a
CH2SCH2(D1-87a) D1-87a
CH2SCH2(D1-87a) D1-92a
CH2SCH2(D1-87a) D1-93a
CH2SCH2(D1-87a) D1-95a
CH2SCH2(D1-87a) D1-96a
CH2SCH2(D1-87a) D1-98a
CH2SCH2(D1-87a) D1-108a
CH2SCH2(D1-87a) D1-108b(Z=2-Cl)
CH2SCH2(D1-87a) D1-108b(Z=3-Me)
CH2SCH2(D1-87a) D1-108b(Z=4-OMe)
CH2SCH2(D1-87a) D1-108b(Z=2-SMe)
CH2SCH2(D1-87a) D1-108b(Z=3-CF3)
CH2SCH2(D1-87a) D1-108b(Z=4-OCF3)
CH2SCH2(D1-87a) D1-108b(Z=2-SCF3)
CH2SCH2(D1-87a) C(O)Me
CH2SCH2(D1-87a) C(O)CF3
CH2SCH2(D1-87a) C(O)OMe
CH2S(O)CH2(D1-87a) Me
CH2S(O)CH2(D1-87a) Et
CH2S(O)CH2(D1-87a) Pr-n
CH2S(O)CH2(D1-87a) Pr-i
CH2S(O)CH2(D1-87a) Pr-c
CH2S(O)CH2(D1-87a) Bu-n
CH2S(O)CH2(D1-87a) Bu-i
CH2S(O)CH2(D1-87a) Bu-c
CH2S(O)CH2(D1-87a) Bu-s
CH2S(O)CH2(D1-87a) Bu-t
CH2S(O)CH2(D1-87a) Pen-n
CH2S(O)CH2(D1-87a) Pen-c
CH2S(O)CH2(D1-87a) Hex-n
CH2S(O)CH2(D1-87a) Hex-c
CH2S(O)CH2(D1-87a) CH2Pr-c
CH2S(O)CH2(D1-87a) CH2Bu-c
CH2S(O)CH2(D1-87a) CH2Pen-c
CH2S(O)CH2(D1-87a) CH2Hex-c
CH2S(O)CH2(D1-87a) CH2CH=CH2
CH2S(O)CH2(D1-87a) CH2CH=C(Cl)2
CH2S(O)CH2(D1-87a) CH2C≡CH
CH2S(O)CH2(D1-87a) CH2CN
CH2S(O)CH2(D1-87a) CH2CF3
CH2S(O)CH2(D1-87a) CH2OMe
CH2S(O)CH2(D1-87a) CH2OCF3
CH2S(O)CH2(D1-87a) CH2SMe
CH2S(O)CH2(D1-87a) CH2S(O)Me
CH2S(O)CH2(D1-87a) CH2S(O)2Me
CH2S(O)CH2(D1-87a) CH2SCF3
CH2S(O)CH2(D1-87a) CH2S(O)CF3
CH2S(O)CH2(D1-87a) CH2S(O)2CF3
CH2S(O)CH2(D1-87a) CH2CH(OMe)2
CH2S(O)CH2(D1-87a) CH2CH(SMe)2
CH2S(O)CH2(D1-87a) CH2C(O)Me
CH2S(O)CH2(D1-87a) CH2C(O)CF3
CH2S(O)CH2(D1-87a) CH2C(O)OMe
CH2S(O)CH2(D1-87a) CH2(D1-32a)
CH2S(O)CH2(D1-87a) CH2(D1-33a)
CH2S(O)CH2(D1-87a) CH2(D1-34a)
CH2S(O)CH2(D1-87a) CH2(D1-37a)
CH2S(O)CH2(D1-87a) CH2(D1-81a)
CH2S(O)CH2(D1-87a) CH2(D1-82a)
CH2S(O)CH2(D1-87a) CH2(D1-84a)
CH2S(O)CH2(D1-87a) CH2(D1-85a)
CH2S(O)CH2(D1-87a) CH2(D1-87a)
CH2S(O)CH2(D1-87a) CH2(D1-92a)
CH2S(O)CH2(D1-87a) CH2(D1-93a)
CH2S(O)CH2(D1-87a) CH2(D1-95a)
CH2S(O)CH2(D1-87a) CH2(D1-96a)
CH2S(O)CH2(D1-87a) CH2(D1-98a)
CH2S(O)CH2(D1-87a) CH2(D1-108a)
CH2S(O)CH2(D1-87a) CH2(D1-108b,Z=2-Cl)
CH2S(O)CH2(D1-87a) CH2(D1-108b,Z=3-Me)
CH2S(O)CH2(D1-87a) CH2(D1-108b,Z=4-OMe)
CH2S(O)CH2(D1-87a) CH2(D1-108b,Z=2-SMe)
CH2S(O)CH2(D1-87a) CH2(D1-108b,Z=3-CF3)
CH2S(O)CH2(D1-87a) CH2(D1-108b,Z=4-OCF3)
CH2S(O)CH2(D1-87a) CH2(D1-108b,Z=2-SCF3)
CH2S(O)CH2(D1-87a) CH2CH2CN
CH2S(O)CH2(D1-87a) CH2CH2CF3
CH2S(O)CH2(D1-87a) CH2CH2OMe
CH2S(O)CH2(D1-87a) CH2CH2SMe
CH2S(O)CH2(D1-87a) CH2CH2S(O)Me
CH2S(O)CH2(D1-87a) CH2CH2S(O)2Me
CH2S(O)CH2(D1-87a) D1-32a
CH2S(O)CH2(D1-87a) D1-33a
CH2S(O)CH2(D1-87a) D1-34a
CH2S(O)CH2(D1-87a) D1-37a
CH2S(O)CH2(D1-87a) D1-81a
CH2S(O)CH2(D1-87a) D1-82a
CH2S(O)CH2(D1-87a) D1-84a
CH2S(O)CH2(D1-87a) D1-85a
CH2S(O)CH2(D1-87a) D1-87a
CH2S(O)CH2(D1-87a) D1-92a
CH2S(O)CH2(D1-87a) D1-93a
CH2S(O)CH2(D1-87a) D1-95a
CH2S(O)CH2(D1-87a) D1-96a
CH2S(O)CH2(D1-87a) D1-98a
CH2S(O)CH2(D1-87a) D1-108a
CH2S(O)CH2(D1-87a) D1-108b(Z=2-Cl)
CH2S(O)CH2(D1-87a) D1-108b(Z=3-Me)
CH2S(O)CH2(D1-87a) D1-108b(Z=4-OMe)
CH2S(O)CH2(D1-87a) D1-108b(Z=2-SMe)
CH2S(O)CH2(D1-87a) D1-108b(Z=3-CF3)
CH2S(O)CH2(D1-87a) D1-108b(Z=4-OCF3)
CH2S(O)CH2(D1-87a) D1-108b(Z=2-SCF3)
CH2S(O)CH2(D1-87a) C(O)Me
CH2S(O)CH2(D1-87a) C(O)CF3
CH2S(O)CH2(D1-87a) C(O)OMe
CH2S(O)2CH2(D1-87a) Me
CH2S(O)2CH2(D1-87a) Et
CH2S(O)2CH2(D1-87a) Pr-n
CH2S(O)2CH2(D1-87a) Pr-i
CH2S(O)2CH2(D1-87a) Pr-c
CH2S(O)2CH2(D1-87a) Bu-n
CH2S(O)2CH2(D1-87a) Bu-i
CH2S(O)2CH2(D1-87a) Bu-c
CH2S(O)2CH2(D1-87a) Bu-s
CH2S(O)2CH2(D1-87a) Bu-t
CH2S(O)2CH2(D1-87a) Pen-n
CH2S(O)2CH2(D1-87a) Pen-c
CH2S(O)2CH2(D1-87a) Hex-n
CH2S(O)2CH2(D1-87a) Hex-c
CH2S(O)2CH2(D1-87a) CH2Pr-c
CH2S(O)2CH2(D1-87a) CH2Bu-c
CH2S(O)2CH2(D1-87a) CH2Pen-c
CH2S(O)2CH2(D1-87a) CH2Hex-c
CH2S(O)2CH2(D1-87a) CH2CH=CH2
CH2S(O)2CH2(D1-87a) CH2CH=C(Cl)2
CH2S(O)2CH2(D1-87a) CH2C≡CH
CH2S(O)2CH2(D1-87a) CH2CN
CH2S(O)2CH2(D1-87a) CH2CF3
CH2S(O)2CH2(D1-87a) CH2OMe
CH2S(O)2CH2(D1-87a) CH2OCF3
CH2S(O)2CH2(D1-87a) CH2SMe
CH2S(O)2CH2(D1-87a) CH2S(O)Me
CH2S(O)2CH2(D1-87a) CH2S(O)2Me
CH2S(O)2CH2(D1-87a) CH2SCF3
CH2S(O)2CH2(D1-87a) CH2S(O)CF3
CH2S(O)2CH2(D1-87a) CH2S(O)2CF3
CH2S(O)2CH2(D1-87a) CH2CH(OMe)2
CH2S(O)2CH2(D1-87a) CH2CH(SMe)2
CH2S(O)2CH2(D1-87a) CH2C(O)Me
CH2S(O)2CH2(D1-87a) CH2C(O)CF3
CH2S(O)2CH2(D1-87a) CH2C(O)OMe
CH2S(O)2CH2(D1-87a) CH2(D1-32a)
CH2S(O)2CH2(D1-87a) CH2(D1-33a)
CH2S(O)2CH2(D1-87a) CH2(D1-34a)
CH2S(O)2CH2(D1-87a) CH2(D1-37a)
CH2S(O)2CH2(D1-87a) CH2(D1-81a)
CH2S(O)2CH2(D1-87a) CH2(D1-82a)
CH2S(O)2CH2(D1-87a) CH2(D1-84a)
CH2S(O)2CH2(D1-87a) CH2(D1-85a)
CH2S(O)2CH2(D1-87a) CH2(D1-87a)
CH2S(O)2CH2(D1-87a) CH2(D1-92a)
CH2S(O)2CH2(D1-87a) CH2(D1-93a)
CH2S(O)2CH2(D1-87a) CH2(D1-95a)
CH2S(O)2CH2(D1-87a) CH2(D1-96a)
CH2S(O)2CH2(D1-87a) CH2(D1-98a)
CH2S(O)2CH2(D1-87a) CH2(D1-108a)
CH2S(O)2CH2(D1-87a) CH2(D1-108b,Z=2-Cl)
CH2S(O)2CH2(D1-87a) CH2(D1-108b,Z=3-Me)
CH2S(O)2CH2(D1-87a) CH2(D1-108b,Z=4-OMe)
CH2S(O)2CH2(D1-87a) CH2(D1-108b,Z=2-SMe)
CH2S(O)2CH2(D1-87a) CH2(D1-108b,Z=3-CF3)
CH2S(O)2CH2(D1-87a) CH2(D1-108b,Z=4-OCF3)
CH2S(O)2CH2(D1-87a) CH2(D1-108b,Z=2-SCF3)
CH2S(O)2CH2(D1-87a) CH2CH2CN
CH2S(O)2CH2(D1-87a) CH2CH2CF3
CH2S(O)2CH2(D1-87a) CH2CH2OMe
CH2S(O)2CH2(D1-87a) CH2CH2SMe
CH2S(O)2CH2(D1-87a) CH2CH2S(O)Me
CH2S(O)2CH2(D1-87a) CH2CH2S(O)2Me
CH2S(O)2CH2(D1-87a) D1-32a
CH2S(O)2CH2(D1-87a) D1-33a
CH2S(O)2CH2(D1-87a) D1-34a
CH2S(O)2CH2(D1-87a) D1-37a
CH2S(O)2CH2(D1-87a) D1-81a
CH2S(O)2CH2(D1-87a) D1-82a
CH2S(O)2CH2(D1-87a) D1-84a
CH2S(O)2CH2(D1-87a) D1-85a
CH2S(O)2CH2(D1-87a) D1-87a
CH2S(O)2CH2(D1-87a) D1-92a
CH2S(O)2CH2(D1-87a) D1-93a
CH2S(O)2CH2(D1-87a) D1-95a
CH2S(O)2CH2(D1-87a) D1-96a
CH2S(O)2CH2(D1-87a) D1-98a
CH2S(O)2CH2(D1-87a) D1-108a
CH2S(O)2CH2(D1-87a) D1-108b(Z=2-Cl)
CH2S(O)2CH2(D1-87a) D1-108b(Z=3-Me)
CH2S(O)2CH2(D1-87a) D1-108b(Z=4-OMe)
CH2S(O)2CH2(D1-87a) D1-108b(Z=2-SMe)
CH2S(O)2CH2(D1-87a) D1-108b(Z=3-CF3)
CH2S(O)2CH2(D1-87a) D1-108b(Z=4-OCF3)
CH2S(O)2CH2(D1-87a) D1-108b(Z=2-SCF3)
CH2SCH2(D1-95a) Me
CH2SCH2(D1-95a) Et
CH2SCH2(D1-95a) Pr-n
CH2SCH2(D1-95a) Pr-i
CH2SCH2(D1-95a) Pr-c
CH2SCH2(D1-95a) Bu-n
CH2SCH2(D1-95a) Bu-i
CH2SCH2(D1-95a) Bu-c
CH2SCH2(D1-95a) Bu-s
CH2SCH2(D1-95a) Bu-t
CH2SCH2(D1-95a) Pen-n
CH2SCH2(D1-95a) Pen-c
CH2SCH2(D1-95a) Hex-n
CH2SCH2(D1-95a) Hex-c
CH2SCH2(D1-95a) CH2Pr-c
CH2SCH2(D1-95a) CH2Bu-c
CH2SCH2(D1-95a) CH2Pen-c
CH2SCH2(D1-95a) CH2Hex-c
CH2SCH2(D1-95a) CH2CH=CH2
CH2SCH2(D1-95a) CH2CH=C(Cl)2
CH2SCH2(D1-95a) CH2C≡CH
CH2SCH2(D1-95a) CH2CN
CH2SCH2(D1-95a) CH2CF3
CH2SCH2(D1-95a) CH2OMe
CH2SCH2(D1-95a) CH2OCF3
CH2SCH2(D1-95a) CH2SMe
CH2SCH2(D1-95a) CH2S(O)Me
CH2SCH2(D1-95a) CH2S(O)2Me
CH2SCH2(D1-95a) CH2SCF3
CH2SCH2(D1-95a) CH2S(O)CF3
CH2SCH2(D1-95a) CH2S(O)2CF3
CH2SCH2(D1-95a) CH2CH(OMe)2
CH2SCH2(D1-95a) CH2CH(SMe)2
CH2SCH2(D1-95a) CH2C(O)Me
CH2SCH2(D1-95a) CH2C(O)CF3
CH2SCH2(D1-95a) CH2C(O)OMe
CH2SCH2(D1-95a) CH2(D1-32a)
CH2SCH2(D1-95a) CH2(D1-33a)
CH2SCH2(D1-95a) CH2(D1-34a)
CH2SCH2(D1-95a) CH2(D1-37a)
CH2SCH2(D1-95a) CH2(D1-81a)
CH2SCH2(D1-95a) CH2(D1-82a)
CH2SCH2(D1-95a) CH2(D1-84a)
CH2SCH2(D1-95a) CH2(D1-85a)
CH2SCH2(D1-95a) CH2(D1-87a)
CH2SCH2(D1-95a) CH2(D1-92a)
CH2SCH2(D1-95a) CH2(D1-93a)
CH2SCH2(D1-95a) CH2(D1-95a)
CH2SCH2(D1-95a) CH2(D1-96a)
CH2SCH2(D1-95a) CH2(D1-98a)
CH2SCH2(D1-95a) CH2(D1-108a)
CH2SCH2(D1-95a) CH2(D1-108b,Z=2-Cl)
CH2SCH2(D1-95a) CH2(D1-108b,Z=3-Me)
CH2SCH2(D1-95a) CH2(D1-108b,Z=4-OMe)
CH2SCH2(D1-95a) CH2(D1-108b,Z=2-SMe)
CH2SCH2(D1-95a) CH2(D1-108b,Z=3-CF3)
CH2SCH2(D1-95a) CH2(D1-108b,Z=4-OCF3)
CH2SCH2(D1-95a) CH2(D1-108b,Z=2-SCF3)
CH2SCH2(D1-95a) CH2CH2CN
CH2SCH2(D1-95a) CH2CH2CF3
CH2SCH2(D1-95a) CH2CH2OMe
CH2SCH2(D1-95a) CH2CH2SMe
CH2SCH2(D1-95a) CH2CH2S(O)Me
CH2SCH2(D1-95a) CH2CH2S(O)2Me
CH2SCH2(D1-95a) D1-32a
CH2SCH2(D1-95a) D1-33a
CH2SCH2(D1-95a) D1-34a
CH2SCH2(D1-95a) D1-37a
CH2SCH2(D1-95a) D1-81a
CH2SCH2(D1-95a) D1-82a
CH2SCH2(D1-95a) D1-84a
CH2SCH2(D1-95a) D1-85a
CH2SCH2(D1-95a) D1-87a
CH2SCH2(D1-95a) D1-92a
CH2SCH2(D1-95a) D1-93a
CH2SCH2(D1-95a) D1-95a
CH2SCH2(D1-95a) D1-96a
CH2SCH2(D1-95a) D1-98a
CH2SCH2(D1-95a) D1-108a
CH2SCH2(D1-95a) D1-108b(Z=2-Cl)
CH2SCH2(D1-95a) D1-108b(Z=3-Me)
CH2SCH2(D1-95a) D1-108b(Z=4-OMe)
CH2SCH2(D1-95a) D1-108b(Z=2-SMe)
CH2SCH2(D1-95a) D1-108b(Z=3-CF3)
CH2SCH2(D1-95a) D1-108b(Z=4-OCF3)
CH2SCH2(D1-95a) D1-108b(Z=2-SCF3)
CH2SCH2(D1-95a) C(O)Me
CH2SCH2(D1-95a) C(O)CF3
CH2SCH2(D1-95a) C(O)OMe
CH2S(O)CH2(D1-95a) Me
CH2S(O)CH2(D1-95a) Et
CH2S(O)CH2(D1-95a) Pr-n
CH2S(O)CH2(D1-95a) Pr-i
CH2S(O)CH2(D1-95a) Pr-c
CH2S(O)CH2(D1-95a) Bu-n
CH2S(O)CH2(D1-95a) Bu-i
CH2S(O)CH2(D1-95a) Bu-c
CH2S(O)CH2(D1-95a) Bu-s
CH2S(O)CH2(D1-95a) Bu-t
CH2S(O)CH2(D1-95a) Pen-n
CH2S(O)CH2(D1-95a) Pen-c
CH2S(O)CH2(D1-95a) Hex-n
CH2S(O)CH2(D1-95a) Hex-c
CH2S(O)CH2(D1-95a) CH2Pr-c
CH2S(O)CH2(D1-95a) CH2Bu-c
CH2S(O)CH2(D1-95a) CH2Pen-c
CH2S(O)CH2(D1-95a) CH2Hex-c
CH2S(O)CH2(D1-95a) CH2CH=CH2
CH2S(O)CH2(D1-95a) CH2CH=C(Cl)2
CH2S(O)CH2(D1-95a) CH2C≡CH
CH2S(O)CH2(D1-95a) CH2CN
CH2S(O)CH2(D1-95a) CH2CF3
CH2S(O)CH2(D1-95a) CH2OMe
CH2S(O)CH2(D1-95a) CH2OCF3
CH2S(O)CH2(D1-95a) CH2SMe
CH2S(O)CH2(D1-95a) CH2S(O)Me
CH2S(O)CH2(D1-95a) CH2S(O)2Me
CH2S(O)CH2(D1-95a) CH2SCF3
CH2S(O)CH2(D1-95a) CH2S(O)CF3
CH2S(O)CH2(D1-95a) CH2S(O)2CF3
CH2S(O)CH2(D1-95a) CH2CH(OMe)2
CH2S(O)CH2(D1-95a) CH2CH(SMe)2
CH2S(O)CH2(D1-95a) CH2C(O)Me
CH2S(O)CH2(D1-95a) CH2C(O)CF3
CH2S(O)CH2(D1-95a) CH2C(O)OMe
CH2S(O)CH2(D1-95a) CH2(D1-32a)
CH2S(O)CH2(D1-95a) CH2(D1-33a)
CH2S(O)CH2(D1-95a) CH2(D1-34a)
CH2S(O)CH2(D1-95a) CH2(D1-37a)
CH2S(O)CH2(D1-95a) CH2(D1-81a)
CH2S(O)CH2(D1-95a) CH2(D1-82a)
CH2S(O)CH2(D1-95a) CH2(D1-84a)
CH2S(O)CH2(D1-95a) CH2(D1-85a)
CH2S(O)CH2(D1-95a) CH2(D1-87a)
CH2S(O)CH2(D1-95a) CH2(D1-92a)
CH2S(O)CH2(D1-95a) CH2(D1-93a)
CH2S(O)CH2(D1-95a) CH2(D1-95a)
CH2S(O)CH2(D1-95a) CH2(D1-96a)
CH2S(O)CH2(D1-95a) CH2(D1-98a)
CH2S(O)CH2(D1-95a) CH2(D1-108a)
CH2S(O)CH2(D1-95a) CH2(D1-108b,Z=2-Cl)
CH2S(O)CH2(D1-95a) CH2(D1-108b,Z=3-Me)
CH2S(O)CH2(D1-95a) CH2(D1-108b,Z=4-OMe)
CH2S(O)CH2(D1-95a) CH2(D1-108b,Z=2-SMe)
CH2S(O)CH2(D1-95a) CH2(D1-108b,Z=3-CF3)
CH2S(O)CH2(D1-95a) CH2(D1-108b,Z=4-OCF3)
CH2S(O)CH2(D1-95a) CH2(D1-108b,Z=2-SCF3)
CH2S(O)CH2(D1-95a) CH2CH2CN
CH2S(O)CH2(D1-95a) CH2CH2CF3
CH2S(O)CH2(D1-95a) CH2CH2OMe
CH2S(O)CH2(D1-95a) CH2CH2SMe
CH2S(O)CH2(D1-95a) CH2CH2S(O)Me
CH2S(O)CH2(D1-95a) CH2CH2S(O)2Me
CH2S(O)CH2(D1-95a) D1-32a
CH2S(O)CH2(D1-95a) D1-33a
CH2S(O)CH2(D1-95a) D1-34a
CH2S(O)CH2(D1-95a) D1-37a
CH2S(O)CH2(D1-95a) D1-81a
CH2S(O)CH2(D1-95a) D1-82a
CH2S(O)CH2(D1-95a) D1-84a
CH2S(O)CH2(D1-95a) D1-85a
CH2S(O)CH2(D1-95a) D1-87a
CH2S(O)CH2(D1-95a) D1-92a
CH2S(O)CH2(D1-95a) D1-93a
CH2S(O)CH2(D1-95a) D1-95a
CH2S(O)CH2(D1-95a) D1-96a
CH2S(O)CH2(D1-95a) D1-98a
CH2S(O)CH2(D1-95a) D1-108a
CH2S(O)CH2(D1-95a) D1-108b(Z=2-Cl)
CH2S(O)CH2(D1-95a) D1-108b(Z=3-Me)
CH2S(O)CH2(D1-95a) D1-108b(Z=4-OMe)
CH2S(O)CH2(D1-95a) D1-108b(Z=2-SMe)
CH2S(O)CH2(D1-95a) D1-108b(Z=3-CF3)
CH2S(O)CH2(D1-95a) D1-108b(Z=4-OCF3)
CH2S(O)CH2(D1-95a) D1-108b(Z=2-SCF3)
CH2S(O)CH2(D1-95a) C(O)Me
CH2S(O)CH2(D1-95a) C(O)CF3
CH2S(O)CH2(D1-95a) C(O)OMe
CH2S(O)2CH2(D1-95a) Me
CH2S(O)2CH2(D1-95a) Et
CH2S(O)2CH2(D1-95a) Pr-n
CH2S(O)2CH2(D1-95a) Pr-i
CH2S(O)2CH2(D1-95a) Pr-c
CH2S(O)2CH2(D1-95a) Bu-n
CH2S(O)2CH2(D1-95a) Bu-i
CH2S(O)2CH2(D1-95a) Bu-c
CH2S(O)2CH2(D1-95a) Bu-s
CH2S(O)2CH2(D1-95a) Bu-t
CH2S(O)2CH2(D1-95a) Pen-n
CH2S(O)2CH2(D1-95a) Pen-c
CH2S(O)2CH2(D1-95a) Hex-n
CH2S(O)2CH2(D1-95a) Hex-c
CH2S(O)2CH2(D1-95a) CH2Pr-c
CH2S(O)2CH2(D1-95a) CH2Bu-c
CH2S(O)2CH2(D1-95a) CH2Pen-c
CH2S(O)2CH2(D1-95a) CH2Hex-c
CH2S(O)2CH2(D1-95a) CH2CH=CH2
CH2S(O)2CH2(D1-95a) CH2CH=C(Cl)2
CH2S(O)2CH2(D1-95a) CH2C≡CH
CH2S(O)2CH2(D1-95a) CH2CN
CH2S(O)2CH2(D1-95a) CH2CF3
CH2S(O)2CH2(D1-95a) CH2OMe
CH2S(O)2CH2(D1-95a) CH2OCF3
CH2S(O)2CH2(D1-95a) CH2SMe
CH2S(O)2CH2(D1-95a) CH2S(O)Me
CH2S(O)2CH2(D1-95a) CH2S(O)2Me
CH2S(O)2CH2(D1-95a) CH2SCF3
CH2S(O)2CH2(D1-95a) CH2S(O)CF3
CH2S(O)2CH2(D1-95a) CH2S(O)2CF3
CH2S(O)2CH2(D1-95a) CH2CH(OMe)2
CH2S(O)2CH2(D1-95a) CH2CH(SMe)2
CH2S(O)2CH2(D1-95a) CH2C(O)Me
CH2S(O)2CH2(D1-95a) CH2C(O)CF3
CH2S(O)2CH2(D1-95a) CH2C(O)OMe
CH2S(O)2CH2(D1-95a) CH2(D1-32a)
CH2S(O)2CH2(D1-95a) CH2(D1-33a)
CH2S(O)2CH2(D1-95a) CH2(D1-34a)
CH2S(O)2CH2(D1-95a) CH2(D1-37a)
CH2S(O)2CH2(D1-95a) CH2(D1-81a)
CH2S(O)2CH2(D1-95a) CH2(D1-82a)
CH2S(O)2CH2(D1-95a) CH2(D1-84a)
CH2S(O)2CH2(D1-95a) CH2(D1-85a)
CH2S(O)2CH2(D1-95a) CH2(D1-87a)
CH2S(O)2CH2(D1-95a) CH2(D1-92a)
CH2S(O)2CH2(D1-95a) CH2(D1-93a)
CH2S(O)2CH2(D1-95a) CH2(D1-95a)
CH2S(O)2CH2(D1-95a) CH2(D1-96a)
CH2S(O)2CH2(D1-95a) CH2(D1-98a)
CH2S(O)2CH2(D1-95a) CH2(D1-108a)
CH2S(O)2CH2(D1-95a) CH2(D1-108b,Z=2-Cl)
CH2S(O)2CH2(D1-95a) CH2(D1-108b,Z=3-Me)
CH2S(O)2CH2(D1-95a) CH2(D1-108b,Z=4-OMe)
CH2S(O)2CH2(D1-95a) CH2(D1-108b,Z=2-SMe)
CH2S(O)2CH2(D1-95a) CH2(D1-108b,Z=3-CF3)
CH2S(O)2CH2(D1-95a) CH2(D1-108b,Z=4-OCF3)
CH2S(O)2CH2(D1-95a) CH2(D1-108b,Z=2-SCF3)
CH2S(O)2CH2(D1-95a) CH2CH2CN
CH2S(O)2CH2(D1-95a) CH2CH2CF3
CH2S(O)2CH2(D1-95a) CH2CH2OMe
CH2S(O)2CH2(D1-95a) CH2CH2SMe
CH2S(O)2CH2(D1-95a) CH2CH2S(O)Me
CH2S(O)2CH2(D1-95a) CH2CH2S(O)2Me
CH2S(O)2CH2(D1-95a) D1-32a
CH2S(O)2CH2(D1-95a) D1-33a
CH2S(O)2CH2(D1-95a) D1-34a
CH2S(O)2CH2(D1-95a) D1-37a
CH2S(O)2CH2(D1-95a) D1-81a
CH2S(O)2CH2(D1-95a) D1-82a
CH2S(O)2CH2(D1-95a) D1-84a
CH2S(O)2CH2(D1-95a) D1-85a
CH2S(O)2CH2(D1-95a) D1-87a
CH2S(O)2CH2(D1-95a) D1-92a
CH2S(O)2CH2(D1-95a) D1-93a
CH2S(O)2CH2(D1-95a) D1-95a
CH2S(O)2CH2(D1-95a) D1-96a
CH2S(O)2CH2(D1-95a) D1-98a
CH2S(O)2CH2(D1-95a) D1-108a
CH2S(O)2CH2(D1-95a) D1-108b(Z=2-Cl)
CH2S(O)2CH2(D1-95a) D1-108b(Z=3-Me)
CH2S(O)2CH2(D1-95a) D1-108b(Z=4-OMe)
CH2S(O)2CH2(D1-95a) D1-108b(Z=2-SMe)
CH2S(O)2CH2(D1-95a) D1-108b(Z=3-CF3)
CH2S(O)2CH2(D1-95a) D1-108b(Z=4-OCF3)
CH2S(O)2CH2(D1-95a) D1-108b(Z=2-SCF3)
CH2SCH2(D1-96a) Me
CH2SCH2(D1-96a) Et
CH2SCH2(D1-96a) Pr-n
CH2SCH2(D1-96a) Pr-i
CH2SCH2(D1-96a) Pr-c
CH2SCH2(D1-96a) Bu-n
CH2SCH2(D1-96a) Bu-i
CH2SCH2(D1-96a) Bu-c
CH2SCH2(D1-96a) Bu-s
CH2SCH2(D1-96a) Bu-t
CH2SCH2(D1-96a) Pen-n
CH2SCH2(D1-96a) Pen-c
CH2SCH2(D1-96a) Hex-n
CH2SCH2(D1-96a) Hex-c
CH2SCH2(D1-96a) CH2Pr-c
CH2SCH2(D1-96a) CH2Bu-c
CH2SCH2(D1-96a) CH2Pen-c
CH2SCH2(D1-96a) CH2Hex-c
CH2SCH2(D1-96a) CH2CH=CH2
CH2SCH2(D1-96a) CH2CH=C(Cl)2
CH2SCH2(D1-96a) CH2C≡CH
CH2SCH2(D1-96a) CH2CN
CH2SCH2(D1-96a) CH2CF3
CH2SCH2(D1-96a) CH2OMe
CH2SCH2(D1-96a) CH2OCF3
CH2SCH2(D1-96a) CH2SMe
CH2SCH2(D1-96a) CH2S(O)Me
CH2SCH2(D1-96a) CH2S(O)2Me
CH2SCH2(D1-96a) CH2SCF3
CH2SCH2(D1-96a) CH2S(O)CF3
CH2SCH2(D1-96a) CH2S(O)2CF3
CH2SCH2(D1-96a) CH2CH(OMe)2
CH2SCH2(D1-96a) CH2CH(SMe)2
CH2SCH2(D1-96a) CH2C(O)Me
CH2SCH2(D1-96a) CH2C(O)CF3
CH2SCH2(D1-96a) CH2C(O)OMe
CH2SCH2(D1-96a) CH2(D1-32a)
CH2SCH2(D1-96a) CH2(D1-33a)
CH2SCH2(D1-96a) CH2(D1-34a)
CH2SCH2(D1-96a) CH2(D1-37a)
CH2SCH2(D1-96a) CH2(D1-81a)
CH2SCH2(D1-96a) CH2(D1-82a)
CH2SCH2(D1-96a) CH2(D1-84a)
CH2SCH2(D1-96a) CH2(D1-85a)
CH2SCH2(D1-96a) CH2(D1-87a)
CH2SCH2(D1-96a) CH2(D1-92a)
CH2SCH2(D1-96a) CH2(D1-93a)
CH2SCH2(D1-96a) CH2(D1-95a)
CH2SCH2(D1-96a) CH2(D1-96a)
CH2SCH2(D1-96a) CH2(D1-98a)
CH2SCH2(D1-96a) CH2(D1-108a)
CH2SCH2(D1-96a) CH2(D1-108b,Z=2-Cl)
CH2SCH2(D1-96a) CH2(D1-108b,Z=3-Me)
CH2SCH2(D1-96a) CH2(D1-108b,Z=4-OMe)
CH2SCH2(D1-96a) CH2(D1-108b,Z=2-SMe)
CH2SCH2(D1-96a) CH2(D1-108b,Z=3-CF3)
CH2SCH2(D1-96a) CH2(D1-108b,Z=4-OCF3)
CH2SCH2(D1-96a) CH2(D1-108b,Z=2-SCF3)
CH2SCH2(D1-96a) CH2CH2CN
CH2SCH2(D1-96a) CH2CH2CF3
CH2SCH2(D1-96a) CH2CH2OMe
CH2SCH2(D1-96a) CH2CH2SMe
CH2SCH2(D1-96a) CH2CH2S(O)Me
CH2SCH2(D1-96a) CH2CH2S(O)2Me
CH2SCH2(D1-96a) D1-32a
CH2SCH2(D1-96a) D1-33a
CH2SCH2(D1-96a) D1-34a
CH2SCH2(D1-96a) D1-37a
CH2SCH2(D1-96a) D1-81a
CH2SCH2(D1-96a) D1-82a
CH2SCH2(D1-96a) D1-84a
CH2SCH2(D1-96a) D1-85a
CH2SCH2(D1-96a) D1-87a
CH2SCH2(D1-96a) D1-92a
CH2SCH2(D1-96a) D1-93a
CH2SCH2(D1-96a) D1-95a
CH2SCH2(D1-96a) D1-96a
CH2SCH2(D1-96a) D1-98a
CH2SCH2(D1-96a) D1-108a
CH2SCH2(D1-96a) D1-108b(Z=2-Cl)
CH2SCH2(D1-96a) D1-108b(Z=3-Me)
CH2SCH2(D1-96a) D1-108b(Z=4-OMe)
CH2SCH2(D1-96a) D1-108b(Z=2-SMe)
CH2SCH2(D1-96a) D1-108b(Z=3-CF3)
CH2SCH2(D1-96a) D1-108b(Z=4-OCF3)
CH2SCH2(D1-96a) D1-108b(Z=2-SCF3)
CH2SCH2(D1-96a) C(O)Me
CH2SCH2(D1-96a) C(O)CF3
CH2SCH2(D1-96a) C(O)OMe
CH2S(O)CH2(D1-96a) Me
CH2S(O)CH2(D1-96a) Et
CH2S(O)CH2(D1-96a) Pr-n
CH2S(O)CH2(D1-96a) Pr-i
CH2S(O)CH2(D1-96a) Pr-c
CH2S(O)CH2(D1-96a) Bu-n
CH2S(O)CH2(D1-96a) Bu-i
CH2S(O)CH2(D1-96a) Bu-c
CH2S(O)CH2(D1-96a) Bu-s
CH2S(O)CH2(D1-96a) Bu-t
CH2S(O)CH2(D1-96a) Pen-n
CH2S(O)CH2(D1-96a) Pen-c
CH2S(O)CH2(D1-96a) Hex-n
CH2S(O)CH2(D1-96a) Hex-c
CH2S(O)CH2(D1-96a) CH2Pr-c
CH2S(O)CH2(D1-96a) CH2Bu-c
CH2S(O)CH2(D1-96a) CH2Pen-c
CH2S(O)CH2(D1-96a) CH2Hex-c
CH2S(O)CH2(D1-96a) CH2CH=CH2
CH2S(O)CH2(D1-96a) CH2CH=C(Cl)2
CH2S(O)CH2(D1-96a) CH2C≡CH
CH2S(O)CH2(D1-96a) CH2CN
CH2S(O)CH2(D1-96a) CH2CF3
CH2S(O)CH2(D1-96a) CH2OMe
CH2S(O)CH2(D1-96a) CH2OCF3
CH2S(O)CH2(D1-96a) CH2SMe
CH2S(O)CH2(D1-96a) CH2S(O)Me
CH2S(O)CH2(D1-96a) CH2S(O)2Me
CH2S(O)CH2(D1-96a) CH2SCF3
CH2S(O)CH2(D1-96a) CH2S(O)CF3
CH2S(O)CH2(D1-96a) CH2S(O)2CF3
CH2S(O)CH2(D1-96a) CH2CH(OMe)2
CH2S(O)CH2(D1-96a) CH2CH(SMe)2
CH2S(O)CH2(D1-96a) CH2C(O)Me
CH2S(O)CH2(D1-96a) CH2C(O)CF3
CH2S(O)CH2(D1-96a) CH2C(O)OMe
CH2S(O)CH2(D1-96a) CH2(D1-32a)
CH2S(O)CH2(D1-96a) CH2(D1-33a)
CH2S(O)CH2(D1-96a) CH2(D1-34a)
CH2S(O)CH2(D1-96a) CH2(D1-37a)
CH2S(O)CH2(D1-96a) CH2(D1-81a)
CH2S(O)CH2(D1-96a) CH2(D1-82a)
CH2S(O)CH2(D1-96a) CH2(D1-84a)
CH2S(O)CH2(D1-96a) CH2(D1-85a)
CH2S(O)CH2(D1-96a) CH2(D1-87a)
CH2S(O)CH2(D1-96a) CH2(D1-92a)
CH2S(O)CH2(D1-96a) CH2(D1-93a)
CH2S(O)CH2(D1-96a) CH2(D1-95a)
CH2S(O)CH2(D1-96a) CH2(D1-96a)
CH2S(O)CH2(D1-96a) CH2(D1-98a)
CH2S(O)CH2(D1-96a) CH2(D1-108a)
CH2S(O)CH2(D1-96a) CH2(D1-108b,Z=2-Cl)
CH2S(O)CH2(D1-96a) CH2(D1-108b,Z=3-Me)
CH2S(O)CH2(D1-96a) CH2(D1-108b,Z=4-OMe)
CH2S(O)CH2(D1-96a) CH2(D1-108b,Z=2-SMe)
CH2S(O)CH2(D1-96a) CH2(D1-108b,Z=3-CF3)
CH2S(O)CH2(D1-96a) CH2(D1-108b,Z=4-OCF3)
CH2S(O)CH2(D1-96a) CH2(D1-108b,Z=2-SCF3)
CH2S(O)CH2(D1-96a) CH2CH2CN
CH2S(O)CH2(D1-96a) CH2CH2CF3
CH2S(O)CH2(D1-96a) CH2CH2OMe
CH2S(O)CH2(D1-96a) CH2CH2SMe
CH2S(O)CH2(D1-96a) CH2CH2S(O)Me
CH2S(O)CH2(D1-96a) CH2CH2S(O)2Me
CH2S(O)CH2(D1-96a) D1-32a
CH2S(O)CH2(D1-96a) D1-33a
CH2S(O)CH2(D1-96a) D1-34a
CH2S(O)CH2(D1-96a) D1-37a
CH2S(O)CH2(D1-96a) D1-81a
CH2S(O)CH2(D1-96a) D1-82a
CH2S(O)CH2(D1-96a) D1-84a
CH2S(O)CH2(D1-96a) D1-85a
CH2S(O)CH2(D1-96a) D1-87a
CH2S(O)CH2(D1-96a) D1-92a
CH2S(O)CH2(D1-96a) D1-93a
CH2S(O)CH2(D1-96a) D1-95a
CH2S(O)CH2(D1-96a) D1-96a
CH2S(O)CH2(D1-96a) D1-98a
CH2S(O)CH2(D1-96a) D1-108a
CH2S(O)CH2(D1-96a) D1-108b(Z=2-Cl)
CH2S(O)CH2(D1-96a) D1-108b(Z=3-Me)
CH2S(O)CH2(D1-96a) D1-108b(Z=4-OMe)
CH2S(O)CH2(D1-96a) D1-108b(Z=2-SMe)
CH2S(O)CH2(D1-96a) D1-108b(Z=3-CF3)
CH2S(O)CH2(D1-96a) D1-108b(Z=4-OCF3)
CH2S(O)CH2(D1-96a) D1-108b(Z=2-SCF3)
CH2S(O)CH2(D1-96a) C(O)Me
CH2S(O)CH2(D1-96a) C(O)CF3
CH2S(O)CH2(D1-96a) C(O)OMe
CH2S(O)2CH2(D1-96a) Me
CH2S(O)2CH2(D1-96a) Et
CH2S(O)2CH2(D1-96a) Pr-n
CH2S(O)2CH2(D1-96a) Pr-i
CH2S(O)2CH2(D1-96a) Pr-c
CH2S(O)2CH2(D1-96a) Bu-n
CH2S(O)2CH2(D1-96a) Bu-i
CH2S(O)2CH2(D1-96a) Bu-c
CH2S(O)2CH2(D1-96a) Bu-s
CH2S(O)2CH2(D1-96a) Bu-t
CH2S(O)2CH2(D1-96a) Pen-n
CH2S(O)2CH2(D1-96a) Pen-c
CH2S(O)2CH2(D1-96a) Hex-n
CH2S(O)2CH2(D1-96a) Hex-c
CH2S(O)2CH2(D1-96a) CH2Pr-c
CH2S(O)2CH2(D1-96a) CH2Bu-c
CH2S(O)2CH2(D1-96a) CH2Pen-c
CH2S(O)2CH2(D1-96a) CH2Hex-c
CH2S(O)2CH2(D1-96a) CH2CH=CH2
CH2S(O)2CH2(D1-96a) CH2CH=C(Cl)2
CH2S(O)2CH2(D1-96a) CH2C≡CH
CH2S(O)2CH2(D1-96a) CH2CN
CH2S(O)2CH2(D1-96a) CH2CF3
CH2S(O)2CH2(D1-96a) CH2OMe
CH2S(O)2CH2(D1-96a) CH2OCF3
CH2S(O)2CH2(D1-96a) CH2SMe
CH2S(O)2CH2(D1-96a) CH2S(O)Me
CH2S(O)2CH2(D1-96a) CH2S(O)2Me
CH2S(O)2CH2(D1-96a) CH2SCF3
CH2S(O)2CH2(D1-96a) CH2S(O)CF3
CH2S(O)2CH2(D1-96a) CH2S(O)2CF3
CH2S(O)2CH2(D1-96a) CH2CH(OMe)2
CH2S(O)2CH2(D1-96a) CH2CH(SMe)2
CH2S(O)2CH2(D1-96a) CH2C(O)Me
CH2S(O)2CH2(D1-96a) CH2C(O)CF3
CH2S(O)2CH2(D1-96a) CH2C(O)OMe
CH2S(O)2CH2(D1-96a) CH2(D1-32a)
CH2S(O)2CH2(D1-96a) CH2(D1-33a)
CH2S(O)2CH2(D1-96a) CH2(D1-34a)
CH2S(O)2CH2(D1-96a) CH2(D1-37a)
CH2S(O)2CH2(D1-96a) CH2(D1-81a)
CH2S(O)2CH2(D1-96a) CH2(D1-82a)
CH2S(O)2CH2(D1-96a) CH2(D1-84a)
CH2S(O)2CH2(D1-96a) CH2(D1-85a)
CH2S(O)2CH2(D1-96a) CH2(D1-87a)
CH2S(O)2CH2(D1-96a) CH2(D1-92a)
CH2S(O)2CH2(D1-96a) CH2(D1-93a)
CH2S(O)2CH2(D1-96a) CH2(D1-95a)
CH2S(O)2CH2(D1-96a) CH2(D1-96a)
CH2S(O)2CH2(D1-96a) CH2(D1-98a)
CH2S(O)2CH2(D1-96a) CH2(D1-108a)
CH2S(O)2CH2(D1-96a) CH2(D1-108b,Z=2-Cl)
CH2S(O)2CH2(D1-96a) CH2(D1-108b,Z=3-Me)
CH2S(O)2CH2(D1-96a) CH2(D1-108b,Z=4-OMe)
CH2S(O)2CH2(D1-96a) CH2(D1-108b,Z=2-SMe)
CH2S(O)2CH2(D1-96a) CH2(D1-108b,Z=3-CF3)
CH2S(O)2CH2(D1-96a) CH2(D1-108b,Z=4-OCF3)
CH2S(O)2CH2(D1-96a) CH2(D1-108b,Z=2-SCF3)
CH2S(O)2CH2(D1-96a) CH2CH2CN
CH2S(O)2CH2(D1-96a) CH2CH2CF3
CH2S(O)2CH2(D1-96a) CH2CH2OMe
CH2S(O)2CH2(D1-96a) CH2CH2SMe
CH2S(O)2CH2(D1-96a) CH2CH2S(O)Me
CH2S(O)2CH2(D1-96a) CH2CH2S(O)2Me
CH2S(O)2CH2(D1-96a) D1-32a
CH2S(O)2CH2(D1-96a) D1-33a
CH2S(O)2CH2(D1-96a) D1-34a
CH2S(O)2CH2(D1-96a) D1-37a
CH2S(O)2CH2(D1-96a) D1-81a
CH2S(O)2CH2(D1-96a) D1-82a
CH2S(O)2CH2(D1-96a) D1-84a
CH2S(O)2CH2(D1-96a) D1-85a
CH2S(O)2CH2(D1-96a) D1-87a
CH2S(O)2CH2(D1-96a) D1-92a
CH2S(O)2CH2(D1-96a) D1-93a
CH2S(O)2CH2(D1-96a) D1-95a
CH2S(O)2CH2(D1-96a) D1-96a
CH2S(O)2CH2(D1-96a) D1-98a
CH2S(O)2CH2(D1-96a) D1-108a
CH2S(O)2CH2(D1-96a) D1-108b(Z=2-Cl)
CH2S(O)2CH2(D1-96a) D1-108b(Z=3-Me)
CH2S(O)2CH2(D1-96a) D1-108b(Z=4-OMe)
CH2S(O)2CH2(D1-96a) D1-108b(Z=2-SMe)
CH2S(O)2CH2(D1-96a) D1-108b(Z=3-CF3)
CH2S(O)2CH2(D1-96a) D1-108b(Z=4-OCF3)
CH2S(O)2CH2(D1-96a) D1-108b(Z=2-SCF3)
CH2SCH2(D1-98a) Me
CH2SCH2(D1-98a) Et
CH2SCH2(D1-98a) Pr-n
CH2SCH2(D1-98a) Pr-i
CH2SCH2(D1-98a) Pr-c
CH2SCH2(D1-98a) Bu-n
CH2SCH2(D1-98a) Bu-i
CH2SCH2(D1-98a) Bu-c
CH2SCH2(D1-98a) Bu-s
CH2SCH2(D1-98a) Bu-t
CH2SCH2(D1-98a) Pen-n
CH2SCH2(D1-98a) Pen-c
CH2SCH2(D1-98a) Hex-n
CH2SCH2(D1-98a) Hex-c
CH2SCH2(D1-98a) CH2Pr-c
CH2SCH2(D1-98a) CH2Bu-c
CH2SCH2(D1-98a) CH2Pen-c
CH2SCH2(D1-98a) CH2Hex-c
CH2SCH2(D1-98a) CH2CH=CH2
CH2SCH2(D1-98a) CH2CH=C(Cl)2
CH2SCH2(D1-98a) CH2C≡CH
CH2SCH2(D1-98a) CH2CN
CH2SCH2(D1-98a) CH2CF3
CH2SCH2(D1-98a) CH2OMe
CH2SCH2(D1-98a) CH2OCF3
CH2SCH2(D1-98a) CH2SMe
CH2SCH2(D1-98a) CH2S(O)Me
CH2SCH2(D1-98a) CH2S(O)2Me
CH2SCH2(D1-98a) CH2SCF3
CH2SCH2(D1-98a) CH2S(O)CF3
CH2SCH2(D1-98a) CH2S(O)2CF3
CH2SCH2(D1-98a) CH2CH(OMe)2
CH2SCH2(D1-98a) CH2CH(SMe)2
CH2SCH2(D1-98a) CH2C(O)Me
CH2SCH2(D1-98a) CH2C(O)CF3
CH2SCH2(D1-98a) CH2C(O)OMe
CH2SCH2(D1-98a) CH2(D1-32a)
CH2SCH2(D1-98a) CH2(D1-33a)
CH2SCH2(D1-98a) CH2(D1-34a)
CH2SCH2(D1-98a) CH2(D1-37a)
CH2SCH2(D1-98a) CH2(D1-81a)
CH2SCH2(D1-98a) CH2(D1-82a)
CH2SCH2(D1-98a) CH2(D1-84a)
CH2SCH2(D1-98a) CH2(D1-85a)
CH2SCH2(D1-98a) CH2(D1-87a)
CH2SCH2(D1-98a) CH2(D1-92a)
CH2SCH2(D1-98a) CH2(D1-93a)
CH2SCH2(D1-98a) CH2(D1-95a)
CH2SCH2(D1-98a) CH2(D1-96a)
CH2SCH2(D1-98a) CH2(D1-98a)
CH2SCH2(D1-98a) CH2(D1-108a)
CH2SCH2(D1-98a) CH2(D1-108b,Z=2-Cl)
CH2SCH2(D1-98a) CH2(D1-108b,Z=3-Me)
CH2SCH2(D1-98a) CH2(D1-108b,Z=4-OMe)
CH2SCH2(D1-98a) CH2(D1-108b,Z=2-SMe)
CH2SCH2(D1-98a) CH2(D1-108b,Z=3-CF3)
CH2SCH2(D1-98a) CH2(D1-108b,Z=4-OCF3)
CH2SCH2(D1-98a) CH2(D1-108b,Z=2-SCF3)
CH2SCH2(D1-98a) CH2CH2CN
CH2SCH2(D1-98a) CH2CH2CF3
CH2SCH2(D1-98a) CH2CH2OMe
CH2SCH2(D1-98a) CH2CH2SMe
CH2SCH2(D1-98a) CH2CH2S(O)Me
CH2SCH2(D1-98a) CH2CH2S(O)2Me
CH2SCH2(D1-98a) D1-32a
CH2SCH2(D1-98a) D1-33a
CH2SCH2(D1-98a) D1-34a
CH2SCH2(D1-98a) D1-37a
CH2SCH2(D1-98a) D1-81a
CH2SCH2(D1-98a) D1-82a
CH2SCH2(D1-98a) D1-84a
CH2SCH2(D1-98a) D1-85a
CH2SCH2(D1-98a) D1-87a
CH2SCH2(D1-98a) D1-92a
CH2SCH2(D1-98a) D1-93a
CH2SCH2(D1-98a) D1-95a
CH2SCH2(D1-98a) D1-96a
CH2SCH2(D1-98a) D1-98a
CH2SCH2(D1-98a) D1-108a
CH2SCH2(D1-98a) D1-108b(Z=2-Cl)
CH2SCH2(D1-98a) D1-108b(Z=3-Me)
CH2SCH2(D1-98a) D1-108b(Z=4-OMe)
CH2SCH2(D1-98a) D1-108b(Z=2-SMe)
CH2SCH2(D1-98a) D1-108b(Z=3-CF3)
CH2SCH2(D1-98a) D1-108b(Z=4-OCF3)
CH2SCH2(D1-98a) D1-108b(Z=2-SCF3)
CH2SCH2(D1-98a) C(O)Me
CH2SCH2(D1-98a) C(O)CF3
CH2SCH2(D1-98a) C(O)OMe
CH2S(O)CH2(D1-98a) Me
CH2S(O)CH2(D1-98a) Et
CH2S(O)CH2(D1-98a) Pr-n
CH2S(O)CH2(D1-98a) Pr-i
CH2S(O)CH2(D1-98a) Pr-c
CH2S(O)CH2(D1-98a) Bu-n
CH2S(O)CH2(D1-98a) Bu-i
CH2S(O)CH2(D1-98a) Bu-c
CH2S(O)CH2(D1-98a) Bu-s
CH2S(O)CH2(D1-98a) Bu-t
CH2S(O)CH2(D1-98a) Pen-n
CH2S(O)CH2(D1-98a) Pen-c
CH2S(O)CH2(D1-98a) Hex-n
CH2S(O)CH2(D1-98a) Hex-c
CH2S(O)CH2(D1-98a) CH2Pr-c
CH2S(O)CH2(D1-98a) CH2Bu-c
CH2S(O)CH2(D1-98a) CH2Pen-c
CH2S(O)CH2(D1-98a) CH2Hex-c
CH2S(O)CH2(D1-98a) CH2CH=CH2
CH2S(O)CH2(D1-98a) CH2CH=C(Cl)2
CH2S(O)CH2(D1-98a) CH2C≡CH
CH2S(O)CH2(D1-98a) CH2CN
CH2S(O)CH2(D1-98a) CH2CF3
CH2S(O)CH2(D1-98a) CH2OMe
CH2S(O)CH2(D1-98a) CH2OCF3
CH2S(O)CH2(D1-98a) CH2SMe
CH2S(O)CH2(D1-98a) CH2S(O)Me
CH2S(O)CH2(D1-98a) CH2S(O)2Me
CH2S(O)CH2(D1-98a) CH2SCF3
CH2S(O)CH2(D1-98a) CH2S(O)CF3
CH2S(O)CH2(D1-98a) CH2S(O)2CF3
CH2S(O)CH2(D1-98a) CH2CH(OMe)2
CH2S(O)CH2(D1-98a) CH2CH(SMe)2
CH2S(O)CH2(D1-98a) CH2C(O)Me
CH2S(O)CH2(D1-98a) CH2C(O)CF3
CH2S(O)CH2(D1-98a) CH2C(O)OMe
CH2S(O)CH2(D1-98a) CH2(D1-32a)
CH2S(O)CH2(D1-98a) CH2(D1-33a)
CH2S(O)CH2(D1-98a) CH2(D1-34a)
CH2S(O)CH2(D1-98a) CH2(D1-37a)
CH2S(O)CH2(D1-98a) CH2(D1-81a)
CH2S(O)CH2(D1-98a) CH2(D1-82a)
CH2S(O)CH2(D1-98a) CH2(D1-84a)
CH2S(O)CH2(D1-98a) CH2(D1-85a)
CH2S(O)CH2(D1-98a) CH2(D1-87a)
CH2S(O)CH2(D1-98a) CH2(D1-92a)
CH2S(O)CH2(D1-98a) CH2(D1-93a)
CH2S(O)CH2(D1-98a) CH2(D1-95a)
CH2S(O)CH2(D1-98a) CH2(D1-96a)
CH2S(O)CH2(D1-98a) CH2(D1-98a)
CH2S(O)CH2(D1-98a) CH2(D1-108a)
CH2S(O)CH2(D1-98a) CH2(D1-108b,Z=2-Cl)
CH2S(O)CH2(D1-98a) CH2(D1-108b,Z=3-Me)
CH2S(O)CH2(D1-98a) CH2(D1-108b,Z=4-OMe)
CH2S(O)CH2(D1-98a) CH2(D1-108b,Z=2-SMe)
CH2S(O)CH2(D1-98a) CH2(D1-108b,Z=3-CF3)
CH2S(O)CH2(D1-98a) CH2(D1-108b,Z=4-OCF3)
CH2S(O)CH2(D1-98a) CH2(D1-108b,Z=2-SCF3)
CH2S(O)CH2(D1-98a) CH2CH2CN
CH2S(O)CH2(D1-98a) CH2CH2CF3
CH2S(O)CH2(D1-98a) CH2CH2OMe
CH2S(O)CH2(D1-98a) CH2CH2SMe
CH2S(O)CH2(D1-98a) CH2CH2S(O)Me
CH2S(O)CH2(D1-98a) CH2CH2S(O)2Me
CH2S(O)CH2(D1-98a) D1-32a
CH2S(O)CH2(D1-98a) D1-33a
CH2S(O)CH2(D1-98a) D1-34a
CH2S(O)CH2(D1-98a) D1-37a
CH2S(O)CH2(D1-98a) D1-81a
CH2S(O)CH2(D1-98a) D1-82a
CH2S(O)CH2(D1-98a) D1-84a
CH2S(O)CH2(D1-98a) D1-85a
CH2S(O)CH2(D1-98a) D1-87a
CH2S(O)CH2(D1-98a) D1-92a
CH2S(O)CH2(D1-98a) D1-93a
CH2S(O)CH2(D1-98a) D1-95a
CH2S(O)CH2(D1-98a) D1-96a
CH2S(O)CH2(D1-98a) D1-98a
CH2S(O)CH2(D1-98a) D1-108a
CH2S(O)CH2(D1-98a) D1-108b(Z=2-Cl)
CH2S(O)CH2(D1-98a) D1-108b(Z=3-Me)
CH2S(O)CH2(D1-98a) D1-108b(Z=4-OMe)
CH2S(O)CH2(D1-98a) D1-108b(Z=2-SMe)
CH2S(O)CH2(D1-98a) D1-108b(Z=3-CF3)
CH2S(O)CH2(D1-98a) D1-108b(Z=4-OCF3)
CH2S(O)CH2(D1-98a) D1-108b(Z=2-SCF3)
CH2S(O)CH2(D1-98a) C(O)Me
CH2S(O)CH2(D1-98a) C(O)CF3
CH2S(O)CH2(D1-98a) C(O)OMe
CH2S(O)2CH2(D1-98a) Me
CH2S(O)2CH2(D1-98a) Et
CH2S(O)2CH2(D1-98a) Pr-n
CH2S(O)2CH2(D1-98a) Pr-i
CH2S(O)2CH2(D1-98a) Pr-c
CH2S(O)2CH2(D1-98a) Bu-n
CH2S(O)2CH2(D1-98a) Bu-i
CH2S(O)2CH2(D1-98a) Bu-c
CH2S(O)2CH2(D1-98a) Bu-s
CH2S(O)2CH2(D1-98a) Bu-t
CH2S(O)2CH2(D1-98a) Pen-n
CH2S(O)2CH2(D1-98a) Pen-c
CH2S(O)2CH2(D1-98a) Hex-n
CH2S(O)2CH2(D1-98a) Hex-c
CH2S(O)2CH2(D1-98a) CH2Pr-c
CH2S(O)2CH2(D1-98a) CH2Bu-c
CH2S(O)2CH2(D1-98a) CH2Pen-c
CH2S(O)2CH2(D1-98a) CH2Hex-c
CH2S(O)2CH2(D1-98a) CH2CH=CH2
CH2S(O)2CH2(D1-98a) CH2CH=C(Cl)2
CH2S(O)2CH2(D1-98a) CH2C≡CH
CH2S(O)2CH2(D1-98a) CH2CN
CH2S(O)2CH2(D1-98a) CH2CF3
CH2S(O)2CH2(D1-98a) CH2OMe
CH2S(O)2CH2(D1-98a) CH2OCF3
CH2S(O)2CH2(D1-98a) CH2SMe
CH2S(O)2CH2(D1-98a) CH2S(O)Me
CH2S(O)2CH2(D1-98a) CH2S(O)2Me
CH2S(O)2CH2(D1-98a) CH2SCF3
CH2S(O)2CH2(D1-98a) CH2S(O)CF3
CH2S(O)2CH2(D1-98a) CH2S(O)2CF3
CH2S(O)2CH2(D1-98a) CH2CH(OMe)2
CH2S(O)2CH2(D1-98a) CH2CH(SMe)2
CH2S(O)2CH2(D1-98a) CH2C(O)Me
CH2S(O)2CH2(D1-98a) CH2C(O)CF3
CH2S(O)2CH2(D1-98a) CH2C(O)OMe
CH2S(O)2CH2(D1-98a) CH2(D1-32a)
CH2S(O)2CH2(D1-98a) CH2(D1-33a)
CH2S(O)2CH2(D1-98a) CH2(D1-34a)
CH2S(O)2CH2(D1-98a) CH2(D1-37a)
CH2S(O)2CH2(D1-98a) CH2(D1-81a)
CH2S(O)2CH2(D1-98a) CH2(D1-82a)
CH2S(O)2CH2(D1-98a) CH2(D1-84a)
CH2S(O)2CH2(D1-98a) CH2(D1-85a)
CH2S(O)2CH2(D1-98a) CH2(D1-87a)
CH2S(O)2CH2(D1-98a) CH2(D1-92a)
CH2S(O)2CH2(D1-98a) CH2(D1-93a)
CH2S(O)2CH2(D1-98a) CH2(D1-95a)
CH2S(O)2CH2(D1-98a) CH2(D1-96a)
CH2S(O)2CH2(D1-98a) CH2(D1-98a)
CH2S(O)2CH2(D1-98a) CH2(D1-108a)
CH2S(O)2CH2(D1-98a) CH2(D1-108b,Z=2-Cl)
CH2S(O)2CH2(D1-98a) CH2(D1-108b,Z=3-Me)
CH2S(O)2CH2(D1-98a) CH2(D1-108b,Z=4-OMe)
CH2S(O)2CH2(D1-98a) CH2(D1-108b,Z=2-SMe)
CH2S(O)2CH2(D1-98a) CH2(D1-108b,Z=3-CF3)
CH2S(O)2CH2(D1-98a) CH2(D1-108b,Z=4-OCF3)
CH2S(O)2CH2(D1-98a) CH2(D1-108b,Z=2-SCF3)
CH2S(O)2CH2(D1-98a) CH2CH2CN
CH2S(O)2CH2(D1-98a) CH2CH2CF3
CH2S(O)2CH2(D1-98a) CH2CH2OMe
CH2S(O)2CH2(D1-98a) CH2CH2SMe
CH2S(O)2CH2(D1-98a) CH2CH2S(O)Me
CH2S(O)2CH2(D1-98a) CH2CH2S(O)2Me
CH2S(O)2CH2(D1-98a) D1-32a
CH2S(O)2CH2(D1-98a) D1-33a
CH2S(O)2CH2(D1-98a) D1-34a
CH2S(O)2CH2(D1-98a) D1-37a
CH2S(O)2CH2(D1-98a) D1-81a
CH2S(O)2CH2(D1-98a) D1-82a
CH2S(O)2CH2(D1-98a) D1-84a
CH2S(O)2CH2(D1-98a) D1-85a
CH2S(O)2CH2(D1-98a) D1-87a
CH2S(O)2CH2(D1-98a) D1-92a
CH2S(O)2CH2(D1-98a) D1-93a
CH2S(O)2CH2(D1-98a) D1-95a
CH2S(O)2CH2(D1-98a) D1-96a
CH2S(O)2CH2(D1-98a) D1-98a
CH2S(O)2CH2(D1-98a) D1-108a
CH2S(O)2CH2(D1-98a) D1-108b(Z=2-Cl)
CH2S(O)2CH2(D1-98a) D1-108b(Z=3-Me)
CH2S(O)2CH2(D1-98a) D1-108b(Z=4-OMe)
CH2S(O)2CH2(D1-98a) D1-108b(Z=2-SMe)
CH2S(O)2CH2(D1-98a) D1-108b(Z=3-CF3)
CH2S(O)2CH2(D1-98a) D1-108b(Z=4-OCF3)
CH2S(O)2CH2(D1-98a) D1-108b(Z=2-SCF3)
CH2SH H
CH2SH Me
CH2SH Et
CH2SH Pr-n
CH2SH Pr-i
CH2SH Pr-c
CH2SH Bu-n
CH2SH Bu-i
CH2SH Bu-c
CH2SH Bu-s
CH2SH Bu-t
CH2SH Pen-n
CH2SH Pen-c
CH2SH Hex-n
CH2SH Hex-c
CH2SH CH2Pr-c
CH2SH CH2Bu-c
CH2SH CH2Pen-c
CH2SH CH2Hex-c
CH2SH CH2CH=CH2
CH2SH CH2CH=C(Cl)2
CH2SH CH2C≡CH
CH2SH CH2CN
CH2SH CH2CF3
CH2SH CH2OMe
CH2SH CH2OCF3
CH2SH CH2SMe
CH2SH CH2S(O)Me
CH2SH CH2S(O)2Me
CH2SH CH2SCF3
CH2SH CH2S(O)CF3
CH2SH CH2S(O)2CF3
CH2SH CH2CH(OMe)2
CH2SH CH2CH(SMe)2
CH2SH CH2C(O)Me
CH2SH CH2C(O)CF3
CH2SH CH2C(O)OMe
CH2SH CH2(D1-32a)
CH2SH CH2(D1-33a)
CH2SH CH2(D1-34a)
CH2SH CH2(D1-37a)
CH2SH CH2(D1-81a)
CH2SH CH2(D1-82a)
CH2SH CH2(D1-84a)
CH2SH CH2(D1-85a)
CH2SH CH2(D1-87a)
CH2SH CH2(D1-92a)
CH2SH CH2(D1-93a)
CH2SH CH2(D1-95a)
CH2SH CH2(D1-96a)
CH2SH CH2(D1-98a)
CH2SH CH2(D1-108a)
CH2SH CH2(D1-108b,Z=2-Cl)
CH2SH CH2(D1-108b,Z=3-Me)
CH2SH CH2(D1-108b,Z=4-OMe)
CH2SH CH2(D1-108b,Z=2-SMe)
CH2SH CH2(D1-108b,Z=3-CF3)
CH2SH CH2(D1-108b,Z=4-OCF3)
CH2SH CH2(D1-108b,Z=2-SCF3)
CH2SH CH2CH2CN
CH2SH CH2CH2CF3
CH2SH CH2CH2OMe
CH2SH CH2CH2SMe
CH2SH CH2CH2S(O)Me
CH2SH CH2CH2S(O)2Me
CH2SH D1-32a
CH2SH D1-33a
CH2SH D1-34a
CH2SH D1-37a
CH2SH D1-81a
CH2SH D1-82a
CH2SH D1-84a
CH2SH D1-85a
CH2SH D1-87a
CH2SH D1-92a
CH2SH D1-93a
CH2SH D1-95a
CH2SH D1-96a
CH2SH D1-98a
CH2SH D1-108a
CH2SH D1-108b(Z=2-Cl)
CH2SH D1-108b(Z=3-Me)
CH2SH D1-108b(Z=4-OMe)
CH2SH D1-108b(Z=2-SMe)
CH2SH D1-108b(Z=3-CF3)
CH2SH D1-108b(Z=4-OCF3)
CH2SH D1-108b(Z=2-SCF3)
CH2SH C(O)Me
CH2SH C(O)CF3
CH2SH C(O)OMe
CH(Me)SH H
CH(Me)SH Me
CH(Me)SH Et
CH(Me)SH Pr-n
CH(Me)SH Pr-i
CH(Me)SH Pr-c
CH(Me)SH Bu-n
CH(Me)SH Bu-i
CH(Me)SH Bu-c
CH(Me)SH Bu-s
CH(Me)SH Bu-t
CH(Me)SH Pen-n
CH(Me)SH Pen-c
CH(Me)SH Hex-n
CH(Me)SH Hex-c
CH(Me)SH CH2Pr-c
CH(Me)SH CH2Bu-c
CH(Me)SH CH2Pen-c
CH(Me)SH CH2Hex-c
CH(Me)SH CH2CH=CH2
CH(Me)SH CH2CH=C(Cl)2
CH(Me)SH CH2C≡CH
CH(Me)SH CH2CN
CH(Me)SH CH2CF3
CH(Me)SH CH2OMe
CH(Me)SH CH2OCF3
CH(Me)SH CH2SMe
CH(Me)SH CH2S(O)Me
CH(Me)SH CH2S(O)2Me
CH(Me)SH CH2SCF3
CH(Me)SH CH2S(O)CF3
CH(Me)SH CH2S(O)2CF3
CH(Me)SH CH2CH(OMe)2
CH(Me)SH CH2CH(SMe)2
CH(Me)SH CH2C(O)Me
CH(Me)SH CH2C(O)CF3
CH(Me)SH CH2C(O)OMe
CH(Me)SH CH2(D1-32a)
CH(Me)SH CH2(D1-33a)
CH(Me)SH CH2(D1-34a)
CH(Me)SH CH2(D1-37a)
CH(Me)SH CH2(D1-81a)
CH(Me)SH CH2(D1-82a)
CH(Me)SH CH2(D1-84a)
CH(Me)SH CH2(D1-85a)
CH(Me)SH CH2(D1-87a)
CH(Me)SH CH2(D1-92a)
CH(Me)SH CH2(D1-93a)
CH(Me)SH CH2(D1-95a)
CH(Me)SH CH2(D1-96a)
CH(Me)SH CH2(D1-98a)
CH(Me)SH CH2(D1-108a)
CH(Me)SH CH2(D1-108b,Z=2-Cl)
CH(Me)SH CH2(D1-108b,Z=3-Me)
CH(Me)SH CH2(D1-108b,Z=4-OMe)
CH(Me)SH CH2(D1-108b,Z=2-SMe)
CH(Me)SH CH2(D1-108b,Z=3-CF3)
CH(Me)SH CH2(D1-108b,Z=4-OCF3)
CH(Me)SH CH2(D1-108b,Z=2-SCF3)
CH(Me)SH CH2CH2CN
CH(Me)SH CH2CH2CF3
CH(Me)SH CH2CH2OMe
CH(Me)SH CH2CH2SMe
CH(Me)SH CH2CH2S(O)Me
CH(Me)SH CH2CH2S(O)2Me
CH(Me)SH D1-32a
CH(Me)SH D1-33a
CH(Me)SH D1-34a
CH(Me)SH D1-37a
CH(Me)SH D1-81a
CH(Me)SH D1-82a
CH(Me)SH D1-84a
CH(Me)SH D1-85a
CH(Me)SH D1-87a
CH(Me)SH D1-92a
CH(Me)SH D1-93a
CH(Me)SH D1-95a
CH(Me)SH D1-96a
CH(Me)SH D1-98a
CH(Me)SH D1-108a
CH(Me)SH D1-108b(Z=2-Cl)
CH(Me)SH D1-108b(Z=3-Me)
CH(Me)SH D1-108b(Z=4-OMe)
CH(Me)SH D1-108b(Z=2-SMe)
CH(Me)SH D1-108b(Z=3-CF3)
CH(Me)SH D1-108b(Z=4-OCF3)
CH(Me)SH D1-108b(Z=2-SCF3)
CH(Me)SH C(O)Me
CH(Me)SH C(O)CF3
CH(Me)SH C(O)OMe
CH(Et)SH H
CH(Et)SH Me
CH(Et)SH Et
CH(Et)SH Pr-n
CH(Et)SH Pr-i
CH(Et)SH Pr-c
CH(Et)SH Bu-n
CH(Et)SH Bu-i
CH(Et)SH Bu-c
CH(Et)SH Bu-s
CH(Et)SH Bu-t
CH(Et)SH Pen-n
CH(Et)SH Pen-c
CH(Et)SH Hex-n
CH(Et)SH Hex-c
CH(Et)SH CH2Pr-c
CH(Et)SH CH2Bu-c
CH(Et)SH CH2Pen-c
CH(Et)SH CH2Hex-c
CH(Et)SH CH2CH=CH2
CH(Et)SH CH2CH=C(Cl)2
CH(Et)SH CH2C≡CH
CH(Et)SH CH2CN
CH(Et)SH CH2CF3
CH(Et)SH CH2OMe
CH(Et)SH CH2OCF3
CH(Et)SH CH2SMe
CH(Et)SH CH2S(O)Me
CH(Et)SH CH2S(O)2Me
CH(Et)SH CH2SCF3
CH(Et)SH CH2S(O)CF3
CH(Et)SH CH2S(O)2CF3
CH(Et)SH CH2CH(OMe)2
CH(Et)SH CH2CH(SMe)2
CH(Et)SH CH2C(O)Me
CH(Et)SH CH2C(O)CF3
CH(Et)SH CH2C(O)OMe
CH(Et)SH CH2(D1-32a)
CH(Et)SH CH2(D1-33a)
CH(Et)SH CH2(D1-34a)
CH(Et)SH CH2(D1-37a)
CH(Et)SH CH2(D1-81a)
CH(Et)SH CH2(D1-82a)
CH(Et)SH CH2(D1-84a)
CH(Et)SH CH2(D1-85a)
CH(Et)SH CH2(D1-87a)
CH(Et)SH CH2(D1-92a)
CH(Et)SH CH2(D1-93a)
CH(Et)SH CH2(D1-95a)
CH(Et)SH CH2(D1-96a)
CH(Et)SH CH2(D1-98a)
CH(Et)SH CH2(D1-108a)
CH(Et)SH CH2(D1-108b,Z=2-Cl)
CH(Et)SH CH2(D1-108b,Z=3-Me)
CH(Et)SH CH2(D1-108b,Z=4-OMe)
CH(Et)SH CH2(D1-108b,Z=2-SMe)
CH(Et)SH CH2(D1-108b,Z=3-CF3)
CH(Et)SH CH2(D1-108b,Z=4-OCF3)
CH(Et)SH CH2(D1-108b,Z=2-SCF3)
CH(Et)SH CH2CH2CN
CH(Et)SH CH2CH2CF3
CH(Et)SH CH2CH2OMe
CH(Et)SH CH2CH2SMe
CH(Et)SH CH2CH2S(O)Me
CH(Et)SH CH2CH2S(O)2Me
CH(Et)SH D1-32a
CH(Et)SH D1-33a
CH(Et)SH D1-34a
CH(Et)SH D1-37a
CH(Et)SH D1-81a
CH(Et)SH D1-82a
CH(Et)SH D1-84a
CH(Et)SH D1-85a
CH(Et)SH D1-87a
CH(Et)SH D1-92a
CH(Et)SH D1-93a
CH(Et)SH D1-95a
CH(Et)SH D1-96a
CH(Et)SH D1-98a
CH(Et)SH D1-108a
CH(Et)SH D1-108b(Z=2-Cl)
CH(Et)SH D1-108b(Z=3-Me)
CH(Et)SH D1-108b(Z=4-OMe)
CH(Et)SH D1-108b(Z=2-SMe)
CH(Et)SH D1-108b(Z=3-CF3)
CH(Et)SH D1-108b(Z=4-OCF3)
CH(Et)SH D1-108b(Z=2-SCF3)
CH(Et)SH C(O)Me
CH(Et)SH C(O)CF3
CH(Et)SH C(O)OMe
CH2SC(O)Me H
CH2SC(O)Me Me
CH2SC(O)Me Et
CH2SC(O)Me Pr-n
CH2SC(O)Me Pr-i
CH2SC(O)Me Pr-c
CH2SC(O)Me Bu-n
CH2SC(O)Me Bu-i
CH2SC(O)Me Bu-c
CH2SC(O)Me Bu-s
CH2SC(O)Me Bu-t
CH2SC(O)Me Pen-n
CH2SC(O)Me Pen-c
CH2SC(O)Me Hex-n
CH2SC(O)Me Hex-c
CH2SC(O)Me CH2Pr-c
CH2SC(O)Me CH2Bu-c
CH2SC(O)Me CH2Pen-c
CH2SC(O)Me CH2Hex-c
CH2SC(O)Me CH2CH=CH2
CH2SC(O)Me CH2CH=C(Cl)2
CH2SC(O)Me CH2C≡CH
CH2SC(O)Me CH2CN
CH2SC(O)Me CH2CF3
CH2SC(O)Me CH2OMe
CH2SC(O)Me CH2OCF3
CH2SC(O)Me CH2SMe
CH2SC(O)Me CH2S(O)Me
CH2SC(O)Me CH2S(O)2Me
CH2SC(O)Me CH2SCF3
CH2SC(O)Me CH2S(O)CF3
CH2SC(O)Me CH2S(O)2CF3
CH2SC(O)Me CH2CH(OMe)2
CH2SC(O)Me CH2CH(SMe)2
CH2SC(O)Me CH2C(O)Me
CH2SC(O)Me CH2C(O)CF3
CH2SC(O)Me CH2C(O)OMe
CH2SC(O)Me CH2(D1-32a)
CH2SC(O)Me CH2(D1-33a)
CH2SC(O)Me CH2(D1-34a)
CH2SC(O)Me CH2(D1-37a)
CH2SC(O)Me CH2(D1-81a)
CH2SC(O)Me CH2(D1-82a)
CH2SC(O)Me CH2(D1-84a)
CH2SC(O)Me CH2(D1-85a)
CH2SC(O)Me CH2(D1-87a)
CH2SC(O)Me CH2(D1-92a)
CH2SC(O)Me CH2(D1-93a)
CH2SC(O)Me CH2(D1-95a)
CH2SC(O)Me CH2(D1-96a)
CH2SC(O)Me CH2(D1-98a)
CH2SC(O)Me CH2(D1-108a)
CH2SC(O)Me CH2(D1-108b,Z=2-Cl)
CH2SC(O)Me CH2(D1-108b,Z=3-Me)
CH2SC(O)Me CH2(D1-108b,Z=4-OMe)
CH2SC(O)Me CH2(D1-108b,Z=2-SMe)
CH2SC(O)Me CH2(D1-108b,Z=3-CF3)
CH2SC(O)Me CH2(D1-108b,Z=4-OCF3)
CH2SC(O)Me CH2(D1-108b,Z=2-SCF3)
CH2SC(O)Me CH2CH2CN
CH2SC(O)Me CH2CH2CF3
CH2SC(O)Me CH2CH2OMe
CH2SC(O)Me CH2CH2SMe
CH2SC(O)Me CH2CH2S(O)Me
CH2SC(O)Me CH2CH2S(O)2Me
CH2SC(O)Me D1-32a
CH2SC(O)Me D1-33a
CH2SC(O)Me D1-34a
CH2SC(O)Me D1-37a
CH2SC(O)Me D1-81a
CH2SC(O)Me D1-82a
CH2SC(O)Me D1-84a
CH2SC(O)Me D1-85a
CH2SC(O)Me D1-87a
CH2SC(O)Me D1-92a
CH2SC(O)Me D1-93a
CH2SC(O)Me D1-95a
CH2SC(O)Me D1-96a
CH2SC(O)Me D1-98a
CH2SC(O)Me D1-108a
CH2SC(O)Me D1-108b(Z=2-Cl)
CH2SC(O)Me D1-108b(Z=3-Me)
CH2SC(O)Me D1-108b(Z=4-OMe)
CH2SC(O)Me D1-108b(Z=2-SMe)
CH2SC(O)Me D1-108b(Z=3-CF3)
CH2SC(O)Me D1-108b(Z=4-OCF3)
CH2SC(O)Me D1-108b(Z=2-SCF3)
CH2SC(O)Me C(O)Me
CH2SC(O)Me C(O)CF3
CH2SC(O)Me C(O)OMe
CH(Me)SC(O)Me H
CH(Me)SC(O)Me Me
CH(Me)SC(O)Me Et
CH(Me)SC(O)Me Pr-n
CH(Me)SC(O)Me Pr-i
CH(Me)SC(O)Me Pr-c
CH(Me)SC(O)Me Bu-n
CH(Me)SC(O)Me Bu-i
CH(Me)SC(O)Me Bu-c
CH(Me)SC(O)Me Bu-s
CH(Me)SC(O)Me Bu-t
CH(Me)SC(O)Me Pen-n
CH(Me)SC(O)Me Pen-c
CH(Me)SC(O)Me Hex-n
CH(Me)SC(O)Me Hex-c
CH(Me)SC(O)Me CH2Pr-c
CH(Me)SC(O)Me CH2Bu-c
CH(Me)SC(O)Me CH2Pen-c
CH(Me)SC(O)Me CH2Hex-c
CH(Me)SC(O)Me CH2CH=CH2
CH(Me)SC(O)Me CH2CH=C(Cl)2
CH(Me)SC(O)Me CH2C≡CH
CH(Me)SC(O)Me CH2CN
CH(Me)SC(O)Me CH2CF3
CH(Me)SC(O)Me CH2OMe
CH(Me)SC(O)Me CH2OCF3
CH(Me)SC(O)Me CH2SMe
CH(Me)SC(O)Me CH2S(O)Me
CH(Me)SC(O)Me CH2S(O)2Me
CH(Me)SC(O)Me CH2SCF3
CH(Me)SC(O)Me CH2S(O)CF3
CH(Me)SC(O)Me CH2S(O)2CF3
CH(Me)SC(O)Me CH2CH(OMe)2
CH(Me)SC(O)Me CH2CH(SMe)2
CH(Me)SC(O)Me CH2C(O)Me
CH(Me)SC(O)Me CH2C(O)CF3
CH(Me)SC(O)Me CH2C(O)OMe
CH(Me)SC(O)Me CH2(D1-32a)
CH(Me)SC(O)Me CH2(D1-33a)
CH(Me)SC(O)Me CH2(D1-34a)
CH(Me)SC(O)Me CH2(D1-37a)
CH(Me)SC(O)Me CH2(D1-81a)
CH(Me)SC(O)Me CH2(D1-82a)
CH(Me)SC(O)Me CH2(D1-84a)
CH(Me)SC(O)Me CH2(D1-85a)
CH(Me)SC(O)Me CH2(D1-87a)
CH(Me)SC(O)Me CH2(D1-92a)
CH(Me)SC(O)Me CH2(D1-93a)
CH(Me)SC(O)Me CH2(D1-95a)
CH(Me)SC(O)Me CH2(D1-96a)
CH(Me)SC(O)Me CH2(D1-98a)
CH(Me)SC(O)Me CH2(D1-108a)
CH(Me)SC(O)Me CH2(D1-108b,Z=2-Cl)
CH(Me)SC(O)Me CH2(D1-108b,Z=3-Me)
CH(Me)SC(O)Me CH2(D1-108b,Z=4-OMe)
CH(Me)SC(O)Me CH2(D1-108b,Z=2-SMe)
CH(Me)SC(O)Me CH2(D1-108b,Z=3-CF3)
CH(Me)SC(O)Me CH2(D1-108b,Z=4-OCF3)
CH(Me)SC(O)Me CH2(D1-108b,Z=2-SCF3)
CH(Me)SC(O)Me CH2CH2CN
CH(Me)SC(O)Me CH2CH2CF3
CH(Me)SC(O)Me CH2CH2OMe
CH(Me)SC(O)Me CH2CH2SMe
CH(Me)SC(O)Me CH2CH2S(O)Me
CH(Me)SC(O)Me CH2CH2S(O)2Me
CH(Me)SC(O)Me D1-32a
CH(Me)SC(O)Me D1-33a
CH(Me)SC(O)Me D1-34a
CH(Me)SC(O)Me D1-37a
CH(Me)SC(O)Me D1-81a
CH(Me)SC(O)Me D1-82a
CH(Me)SC(O)Me D1-84a
CH(Me)SC(O)Me D1-85a
CH(Me)SC(O)Me D1-87a
CH(Me)SC(O)Me D1-92a
CH(Me)SC(O)Me D1-93a
CH(Me)SC(O)Me D1-95a
CH(Me)SC(O)Me D1-96a
CH(Me)SC(O)Me D1-98a
CH(Me)SC(O)Me D1-108a
CH(Me)SC(O)Me D1-108b(Z=2-Cl)
CH(Me)SC(O)Me D1-108b(Z=3-Me)
CH(Me)SC(O)Me D1-108b(Z=4-OMe)
CH(Me)SC(O)Me D1-108b(Z=2-SMe)
CH(Me)SC(O)Me D1-108b(Z=3-CF3)
CH(Me)SC(O)Me D1-108b(Z=4-OCF3)
CH(Me)SC(O)Me D1-108b(Z=2-SCF3)
CH(Me)SC(O)Me C(O)Me
CH(Me)SC(O)Me C(O)CF3
CH(Me)SC(O)Me C(O)OMe
CH(Et)SC(O)Me H
CH(Et)SC(O)Me Me
CH(Et)SC(O)Me Et
CH(Et)SC(O)Me Pr-n
CH(Et)SC(O)Me Pr-i
CH(Et)SC(O)Me Pr-c
CH(Et)SC(O)Me Bu-n
CH(Et)SC(O)Me Bu-i
CH(Et)SC(O)Me Bu-c
CH(Et)SC(O)Me Bu-s
CH(Et)SC(O)Me Bu-t
CH(Et)SC(O)Me Pen-n
CH(Et)SC(O)Me Pen-c
CH(Et)SC(O)Me Hex-n
CH(Et)SC(O)Me Hex-c
CH(Et)SC(O)Me CH2Pr-c
CH(Et)SC(O)Me CH2Bu-c
CH(Et)SC(O)Me CH2Pen-c
CH(Et)SC(O)Me CH2Hex-c
CH(Et)SC(O)Me CH2CH=CH2
CH(Et)SC(O)Me CH2CH=C(Cl)2
CH(Et)SC(O)Me CH2C≡CH
CH(Et)SC(O)Me CH2CN
CH(Et)SC(O)Me CH2CF3
CH(Et)SC(O)Me CH2OMe
CH(Et)SC(O)Me CH2OCF3
CH(Et)SC(O)Me CH2SMe
CH(Et)SC(O)Me CH2S(O)Me
CH(Et)SC(O)Me CH2S(O)2Me
CH(Et)SC(O)Me CH2SCF3
CH(Et)SC(O)Me CH2S(O)CF3
CH(Et)SC(O)Me CH2S(O)2CF3
CH(Et)SC(O)Me CH2CH(OMe)2
CH(Et)SC(O)Me CH2CH(SMe)2
CH(Et)SC(O)Me CH2C(O)Me
CH(Et)SC(O)Me CH2C(O)CF3
CH(Et)SC(O)Me CH2C(O)OMe
CH(Et)SC(O)Me CH2(D1-32a)
CH(Et)SC(O)Me CH2(D1-33a)
CH(Et)SC(O)Me CH2(D1-34a)
CH(Et)SC(O)Me CH2(D1-37a)
CH(Et)SC(O)Me CH2(D1-81a)
CH(Et)SC(O)Me CH2(D1-82a)
CH(Et)SC(O)Me CH2(D1-84a)
CH(Et)SC(O)Me CH2(D1-85a)
CH(Et)SC(O)Me CH2(D1-87a)
CH(Et)SC(O)Me CH2(D1-92a)
CH(Et)SC(O)Me CH2(D1-93a)
CH(Et)SC(O)Me CH2(D1-95a)
CH(Et)SC(O)Me CH2(D1-96a)
CH(Et)SC(O)Me CH2(D1-98a)
CH(Et)SC(O)Me CH2(D1-108a)
CH(Et)SC(O)Me CH2(D1-108b,Z=2-Cl)
CH(Et)SC(O)Me CH2(D1-108b,Z=3-Me)
CH(Et)SC(O)Me CH2(D1-108b,Z=4-OMe)
CH(Et)SC(O)Me CH2(D1-108b,Z=2-SMe)
CH(Et)SC(O)Me CH2(D1-108b,Z=3-CF3)
CH(Et)SC(O)Me CH2(D1-108b,Z=4-OCF3)
CH(Et)SC(O)Me CH2(D1-108b,Z=2-SCF3)
CH(Et)SC(O)Me CH2CH2CN
CH(Et)SC(O)Me CH2CH2CF3
CH(Et)SC(O)Me CH2CH2OMe
CH(Et)SC(O)Me CH2CH2SMe
CH(Et)SC(O)Me CH2CH2S(O)Me
CH(Et)SC(O)Me CH2CH2S(O)2Me
CH(Et)SC(O)Me D1-32a
CH(Et)SC(O)Me D1-33a
CH(Et)SC(O)Me D1-34a
CH(Et)SC(O)Me D1-37a
CH(Et)SC(O)Me D1-81a
CH(Et)SC(O)Me D1-82a
CH(Et)SC(O)Me D1-84a
CH(Et)SC(O)Me D1-85a
CH(Et)SC(O)Me D1-87a
CH(Et)SC(O)Me D1-92a
CH(Et)SC(O)Me D1-93a
CH(Et)SC(O)Me D1-95a
CH(Et)SC(O)Me D1-96a
CH(Et)SC(O)Me D1-98a
CH(Et)SC(O)Me D1-108a
CH(Et)SC(O)Me D1-108b(Z=2-Cl)
CH(Et)SC(O)Me D1-108b(Z=3-Me)
CH(Et)SC(O)Me D1-108b(Z=4-OMe)
CH(Et)SC(O)Me D1-108b(Z=2-SMe)
CH(Et)SC(O)Me D1-108b(Z=3-CF3)
CH(Et)SC(O)Me D1-108b(Z=4-OCF3)
CH(Et)SC(O)Me D1-108b(Z=2-SCF3)
CH(Et)SC(O)Me C(O)Me
CH(Et)SC(O)Me C(O)CF3
CH(Et)SC(O)Me C(O)OMe
CH2SC(O)(D1-108a) H
CH2SC(O)(D1-108a) Me
CH2SC(O)(D1-108a) Et
CH2SC(O)(D1-108a) Pr-n
CH2SC(O)(D1-108a) Pr-i
CH2SC(O)(D1-108a) Pr-c
CH2SC(O)(D1-108a) Bu-n
CH2SC(O)(D1-108a) Bu-i
CH2SC(O)(D1-108a) Bu-c
CH2SC(O)(D1-108a) Bu-s
CH2SC(O)(D1-108a) Bu-t
CH2SC(O)(D1-108a) Pen-n
CH2SC(O)(D1-108a) Pen-c
CH2SC(O)(D1-108a) Hex-n
CH2SC(O)(D1-108a) Hex-c
CH2SC(O)(D1-108a) CH2Pr-c
CH2SC(O)(D1-108a) CH2Bu-c
CH2SC(O)(D1-108a) CH2Pen-c
CH2SC(O)(D1-108a) CH2Hex-c
CH2SC(O)(D1-108a) CH2CH=CH2
CH2SC(O)(D1-108a) CH2CH=C(Cl)2
CH2SC(O)(D1-108a) CH2C≡CH
CH2SC(O)(D1-108a) CH2CN
CH2SC(O)(D1-108a) CH2CF3
CH2SC(O)(D1-108a) CH2OMe
CH2SC(O)(D1-108a) CH2OCF3
CH2SC(O)(D1-108a) CH2SMe
CH2SC(O)(D1-108a) CH2S(O)Me
CH2SC(O)(D1-108a) CH2S(O)2Me
CH2SC(O)(D1-108a) CH2SCF3
CH2SC(O)(D1-108a) CH2S(O)CF3
CH2SC(O)(D1-108a) CH2S(O)2CF3
CH2SC(O)(D1-108a) CH2CH(OMe)2
CH2SC(O)(D1-108a) CH2CH(SMe)2
CH2SC(O)(D1-108a) CH2C(O)Me
CH2SC(O)(D1-108a) CH2C(O)CF3
CH2SC(O)(D1-108a) CH2C(O)OMe
CH2SC(O)(D1-108a) CH2(D1-32a)
CH2SC(O)(D1-108a) CH2(D1-33a)
CH2SC(O)(D1-108a) CH2(D1-34a)
CH2SC(O)(D1-108a) CH2(D1-37a)
CH2SC(O)(D1-108a) CH2(D1-81a)
CH2SC(O)(D1-108a) CH2(D1-82a)
CH2SC(O)(D1-108a) CH2(D1-84a)
CH2SC(O)(D1-108a) CH2(D1-85a)
CH2SC(O)(D1-108a) CH2(D1-87a)
CH2SC(O)(D1-108a) CH2(D1-92a)
CH2SC(O)(D1-108a) CH2(D1-93a)
CH2SC(O)(D1-108a) CH2(D1-95a)
CH2SC(O)(D1-108a) CH2(D1-96a)
CH2SC(O)(D1-108a) CH2(D1-98a)
CH2SC(O)(D1-108a) CH2(D1-108a)
CH2SC(O)(D1-108a) CH2(D1-108b,Z=2-Cl)
CH2SC(O)(D1-108a) CH2(D1-108b,Z=3-Me)
CH2SC(O)(D1-108a) CH2(D1-108b,Z=4-OMe)
CH2SC(O)(D1-108a) CH2(D1-108b,Z=2-SMe)
CH2SC(O)(D1-108a) CH2(D1-108b,Z=3-CF3)
CH2SC(O)(D1-108a) CH2(D1-108b,Z=4-OCF3)
CH2SC(O)(D1-108a) CH2(D1-108b,Z=2-SCF3)
CH2SC(O)(D1-108a) CH2CH2CN
CH2SC(O)(D1-108a) CH2CH2CF3
CH2SC(O)(D1-108a) CH2CH2OMe
CH2SC(O)(D1-108a) CH2CH2SMe
CH2SC(O)(D1-108a) CH2CH2S(O)Me
CH2SC(O)(D1-108a) CH2CH2S(O)2Me
CH2SC(O)(D1-108a) D1-32a
CH2SC(O)(D1-108a) D1-33a
CH2SC(O)(D1-108a) D1-34a
CH2SC(O)(D1-108a) D1-37a
CH2SC(O)(D1-108a) D1-81a
CH2SC(O)(D1-108a) D1-82a
CH2SC(O)(D1-108a) D1-84a
CH2SC(O)(D1-108a) D1-85a
CH2SC(O)(D1-108a) D1-87a
CH2SC(O)(D1-108a) D1-92a
CH2SC(O)(D1-108a) D1-93a
CH2SC(O)(D1-108a) D1-95a
CH2SC(O)(D1-108a) D1-96a
CH2SC(O)(D1-108a) D1-98a
CH2SC(O)(D1-108a) D1-108a
CH2SC(O)(D1-108a) D1-108b(Z=2-Cl)
CH2SC(O)(D1-108a) D1-108b(Z=3-Me)
CH2SC(O)(D1-108a) D1-108b(Z=4-OMe)
CH2SC(O)(D1-108a) D1-108b(Z=2-SMe)
CH2SC(O)(D1-108a) D1-108b(Z=3-CF3)
CH2SC(O)(D1-108a) D1-108b(Z=4-OCF3)
CH2SC(O)(D1-108a) D1-108b(Z=2-SCF3)
CH2SC(O)(D1-108a) C(O)Me
CH2SC(O)(D1-108a) C(O)CF3
CH2SC(O)(D1-108a) C(O)OMe
CH(Me)SC(O)(D1-108a) H
CH(Me)SC(O)(D1-108a) Me
CH(Me)SC(O)(D1-108a) Et
CH(Me)SC(O)(D1-108a) Pr-n
CH(Me)SC(O)(D1-108a) Pr-i
CH(Me)SC(O)(D1-108a) Pr-c
CH(Me)SC(O)(D1-108a) Bu-n
CH(Me)SC(O)(D1-108a) Bu-i
CH(Me)SC(O)(D1-108a) Bu-c
CH(Me)SC(O)(D1-108a) Bu-s
CH(Me)SC(O)(D1-108a) Bu-t
CH(Me)SC(O)(D1-108a) Pen-n
CH(Me)SC(O)(D1-108a) Pen-c
CH(Me)SC(O)(D1-108a) Hex-n
CH(Me)SC(O)(D1-108a) Hex-c
CH(Me)SC(O)(D1-108a) CH2Pr-c
CH(Me)SC(O)(D1-108a) CH2Bu-c
CH(Me)SC(O)(D1-108a) CH2Pen-c
CH(Me)SC(O)(D1-108a) CH2Hex-c
CH(Me)SC(O)(D1-108a) CH2CH=CH2
CH(Me)SC(O)(D1-108a) CH2CH=C(Cl)2
CH(Me)SC(O)(D1-108a) CH2C≡CH
CH(Me)SC(O)(D1-108a) CH2CN
CH(Me)SC(O)(D1-108a) CH2CF3
CH(Me)SC(O)(D1-108a) CH2OMe
CH(Me)SC(O)(D1-108a) CH2OCF3
CH(Me)SC(O)(D1-108a) CH2SMe
CH(Me)SC(O)(D1-108a) CH2S(O)Me
CH(Me)SC(O)(D1-108a) CH2S(O)2Me
CH(Me)SC(O)(D1-108a) CH2SCF3
CH(Me)SC(O)(D1-108a) CH2S(O)CF3
CH(Me)SC(O)(D1-108a) CH2S(O)2CF3
CH(Me)SC(O)(D1-108a) CH2CH(OMe)2
CH(Me)SC(O)(D1-108a) CH2CH(SMe)2
CH(Me)SC(O)(D1-108a) CH2C(O)Me
CH(Me)SC(O)(D1-108a) CH2C(O)CF3
CH(Me)SC(O)(D1-108a) CH2C(O)OMe
CH(Me)SC(O)(D1-108a) CH2(D1-32a)
CH(Me)SC(O)(D1-108a) CH2(D1-33a)
CH(Me)SC(O)(D1-108a) CH2(D1-34a)
CH(Me)SC(O)(D1-108a) CH2(D1-37a)
CH(Me)SC(O)(D1-108a) CH2(D1-81a)
CH(Me)SC(O)(D1-108a) CH2(D1-82a)
CH(Me)SC(O)(D1-108a) CH2(D1-84a)
CH(Me)SC(O)(D1-108a) CH2(D1-85a)
CH(Me)SC(O)(D1-108a) CH2(D1-87a)
CH(Me)SC(O)(D1-108a) CH2(D1-92a)
CH(Me)SC(O)(D1-108a) CH2(D1-93a)
CH(Me)SC(O)(D1-108a) CH2(D1-95a)
CH(Me)SC(O)(D1-108a) CH2(D1-96a)
CH(Me)SC(O)(D1-108a) CH2(D1-98a)
CH(Me)SC(O)(D1-108a) CH2(D1-108a)
CH(Me)SC(O)(D1-108a) CH2(D1-108b,Z=2-Cl)
CH(Me)SC(O)(D1-108a) CH2(D1-108b,Z=3-Me)
CH(Me)SC(O)(D1-108a) CH2(D1-108b,Z=4-OMe)
CH(Me)SC(O)(D1-108a) CH2(D1-108b,Z=2-SMe)
CH(Me)SC(O)(D1-108a) CH2(D1-108b,Z=3-CF3)
CH(Me)SC(O)(D1-108a) CH2(D1-108b,Z=4-OCF3)
CH(Me)SC(O)(D1-108a) CH2(D1-108b,Z=2-SCF3)
CH(Me)SC(O)(D1-108a) CH2CH2CN
CH(Me)SC(O)(D1-108a) CH2CH2CF3
CH(Me)SC(O)(D1-108a) CH2CH2OMe
CH(Me)SC(O)(D1-108a) CH2CH2SMe
CH(Me)SC(O)(D1-108a) CH2CH2S(O)Me
CH(Me)SC(O)(D1-108a) CH2CH2S(O)2Me
CH(Me)SC(O)(D1-108a) D1-32a
CH(Me)SC(O)(D1-108a) D1-33a
CH(Me)SC(O)(D1-108a) D1-34a
CH(Me)SC(O)(D1-108a) D1-37a
CH(Me)SC(O)(D1-108a) D1-81a
CH(Me)SC(O)(D1-108a) D1-82a
CH(Me)SC(O)(D1-108a) D1-84a
CH(Me)SC(O)(D1-108a) D1-85a
CH(Me)SC(O)(D1-108a) D1-87a
CH(Me)SC(O)(D1-108a) D1-92a
CH(Me)SC(O)(D1-108a) D1-93a
CH(Me)SC(O)(D1-108a) D1-95a
CH(Me)SC(O)(D1-108a) D1-96a
CH(Me)SC(O)(D1-108a) D1-98a
CH(Me)SC(O)(D1-108a) D1-108a
CH(Me)SC(O)(D1-108a) D1-108b(Z=2-Cl)
CH(Me)SC(O)(D1-108a) D1-108b(Z=3-Me)
CH(Me)SC(O)(D1-108a) D1-108b(Z=4-OMe)
CH(Me)SC(O)(D1-108a) D1-108b(Z=2-SMe)
CH(Me)SC(O)(D1-108a) D1-108b(Z=3-CF3)
CH(Me)SC(O)(D1-108a) D1-108b(Z=4-OCF3)
CH(Me)SC(O)(D1-108a) D1-108b(Z=2-SCF3)
CH(Me)SC(O)(D1-108a) C(O)Me
CH(Me)SC(O)(D1-108a) C(O)CF3
CH(Me)SC(O)(D1-108a) C(O)OMe
CH(Et)SC(O)(D1-108a) H
CH(Et)SC(O)(D1-108a) Me
CH(Et)SC(O)(D1-108a) Et
CH(Et)SC(O)(D1-108a) Pr-n
CH(Et)SC(O)(D1-108a) Pr-i
CH(Et)SC(O)(D1-108a) Pr-c
CH(Et)SC(O)(D1-108a) Bu-n
CH(Et)SC(O)(D1-108a) Bu-i
CH(Et)SC(O)(D1-108a) Bu-c
CH(Et)SC(O)(D1-108a) Bu-s
CH(Et)SC(O)(D1-108a) Bu-t
CH(Et)SC(O)(D1-108a) Pen-n
CH(Et)SC(O)(D1-108a) Pen-c
CH(Et)SC(O)(D1-108a) Hex-n
CH(Et)SC(O)(D1-108a) Hex-c
CH(Et)SC(O)(D1-108a) CH2Pr-c
CH(Et)SC(O)(D1-108a) CH2Bu-c
CH(Et)SC(O)(D1-108a) CH2Pen-c
CH(Et)SC(O)(D1-108a) CH2Hex-c
CH(Et)SC(O)(D1-108a) CH2CH=CH2
CH(Et)SC(O)(D1-108a) CH2CH=C(Cl)2
CH(Et)SC(O)(D1-108a) CH2C≡CH
CH(Et)SC(O)(D1-108a) CH2CN
CH(Et)SC(O)(D1-108a) CH2CF3
CH(Et)SC(O)(D1-108a) CH2OMe
CH(Et)SC(O)(D1-108a) CH2OCF3
CH(Et)SC(O)(D1-108a) CH2SMe
CH(Et)SC(O)(D1-108a) CH2S(O)Me
CH(Et)SC(O)(D1-108a) CH2S(O)2Me
CH(Et)SC(O)(D1-108a) CH2SCF3
CH(Et)SC(O)(D1-108a) CH2S(O)CF3
CH(Et)SC(O)(D1-108a) CH2S(O)2CF3
CH(Et)SC(O)(D1-108a) CH2CH(OMe)2
CH(Et)SC(O)(D1-108a) CH2CH(SMe)2
CH(Et)SC(O)(D1-108a) CH2C(O)Me
CH(Et)SC(O)(D1-108a) CH2C(O)CF3
CH(Et)SC(O)(D1-108a) CH2C(O)OMe
CH(Et)SC(O)(D1-108a) CH2(D1-32a)
CH(Et)SC(O)(D1-108a) CH2(D1-33a)
CH(Et)SC(O)(D1-108a) CH2(D1-34a)
CH(Et)SC(O)(D1-108a) CH2(D1-37a)
CH(Et)SC(O)(D1-108a) CH2(D1-81a)
CH(Et)SC(O)(D1-108a) CH2(D1-82a)
CH(Et)SC(O)(D1-108a) CH2(D1-84a)
CH(Et)SC(O)(D1-108a) CH2(D1-85a)
CH(Et)SC(O)(D1-108a) CH2(D1-87a)
CH(Et)SC(O)(D1-108a) CH2(D1-92a)
CH(Et)SC(O)(D1-108a) CH2(D1-93a)
CH(Et)SC(O)(D1-108a) CH2(D1-95a)
CH(Et)SC(O)(D1-108a) CH2(D1-96a)
CH(Et)SC(O)(D1-108a) CH2(D1-98a)
CH(Et)SC(O)(D1-108a) CH2(D1-108a)
CH(Et)SC(O)(D1-108a) CH2(D1-108b,Z=2-Cl)
CH(Et)SC(O)(D1-108a) CH2(D1-108b,Z=3-Me)
CH(Et)SC(O)(D1-108a) CH2(D1-108b,Z=4-OMe)
CH(Et)SC(O)(D1-108a) CH2(D1-108b,Z=2-SMe)
CH(Et)SC(O)(D1-108a) CH2(D1-108b,Z=3-CF3)
CH(Et)SC(O)(D1-108a) CH2(D1-108b,Z=4-OCF3)
CH(Et)SC(O)(D1-108a) CH2(D1-108b,Z=2-SCF3)
CH(Et)SC(O)(D1-108a) CH2CH2CN
CH(Et)SC(O)(D1-108a) CH2CH2CF3
CH(Et)SC(O)(D1-108a) CH2CH2OMe
CH(Et)SC(O)(D1-108a) CH2CH2SMe
CH(Et)SC(O)(D1-108a) CH2CH2S(O)Me
CH(Et)SC(O)(D1-108a) CH2CH2S(O)2Me
CH(Et)SC(O)(D1-108a) D1-32a
CH(Et)SC(O)(D1-108a) D1-33a
CH(Et)SC(O)(D1-108a) D1-34a
CH(Et)SC(O)(D1-108a) D1-37a
CH(Et)SC(O)(D1-108a) D1-81a
CH(Et)SC(O)(D1-108a) D1-82a
CH(Et)SC(O)(D1-108a) D1-84a
CH(Et)SC(O)(D1-108a) D1-85a
CH(Et)SC(O)(D1-108a) D1-87a
CH(Et)SC(O)(D1-108a) D1-92a
CH(Et)SC(O)(D1-108a) D1-93a
CH(Et)SC(O)(D1-108a) D1-95a
CH(Et)SC(O)(D1-108a) D1-96a
CH(Et)SC(O)(D1-108a) D1-98a
CH(Et)SC(O)(D1-108a) D1-108a
CH(Et)SC(O)(D1-108a) D1-108b(Z=2-Cl)
CH(Et)SC(O)(D1-108a) D1-108b(Z=3-Me)
CH(Et)SC(O)(D1-108a) D1-108b(Z=4-OMe)
CH(Et)SC(O)(D1-108a) D1-108b(Z=2-SMe)
CH(Et)SC(O)(D1-108a) D1-108b(Z=3-CF3)
CH(Et)SC(O)(D1-108a) D1-108b(Z=4-OCF3)
CH(Et)SC(O)(D1-108a) D1-108b(Z=2-SCF3)
CH(Et)SC(O)(D1-108a) C(O)Me
CH(Et)SC(O)(D1-108a) C(O)CF3
CH(Et)SC(O)(D1-108a) C(O)OMe
Me H
Et H
Pr-n H
Pr-i H
Bu-n H
Bu-i H
Bu-t H
Pen-n H
Hex-n H
CH(Et)Cl H
CH2{D1-7b(3-CF3)} H
CH(CN)Ph H
SMe H
SEt H
SPr-n H
SPr-i H
SBu-n H
SBu-i H
SBu-t H
SPen-n H
SHex-n H
SPr-c H
SBu-c H
SPen-c H
SHex-c H
SCH2CH=CH2 H
SCH2C三CH H
SCF2H H
SCF3 H
SCF2Cl H
SCH2CF3 H
S(D1-108c) H
CH2OH H
CH2OMe H
CH2OEt H
CH2OPr-n H
CH2OPr-i H
CH2OBu-n H
CH2OBu-i H
CH2OBu-s H
CH2OBu-t H
CH2OPen-n H
CH2OHex-n H
CH2O(D1-104c) H
CH(Me)OH H
CH(Me)OMe H
CH(Me)OEt H
CH(Me)OPr-n H
CH(Me)OPr-i H
CH(Me)OBu-n H
CH(Me)OBu-i H
CH(Me)OBu-s H
CH(Me)OBu-t H
CH(Me)OPen-n H
CH(Me)OHex-n H
CH(Me)O(D1-104c) H
CH(Et)OH H
CH(Et)OMe H
CH(Et)OEt H
CH(Et)OPr-n H
CH(Et)OPr-i H
CH(Et)OBu-n H
CH(Et)OBu-i H
CH(Et)OBu-s H
CH(Et)OBu-t H
CH(Et)OPen-n H
CH(Et)OHex-n H
CH(Et)O(D1-104c) H
CH(n-Pr)OH H
CH(n-Pr)OMe H
CH(n-Pr)OEt H
CH(n-Pr)O(D1-104c) H
CH(i-Pr)OH H
CH(i-Pr)OMe H
CH(i-Pr)OEt H
CH(i-Pr)O(D1-104c) H
CH(n-Bu)OH H
CH(n-Bu)OMe H
CH(n-Bu)OEt H
CH(n-Bu)O(D1-104c) H
C(Me)2OH H
C(Me)2OMe H
C(Me)2OEt H
C(Me)2O(D1-104c) H
CH2CH2OH H
CH2CH2OMe H
CH2CH2OEt H
CH2CH2O(D1-104c) H
CH(Me)CH2OH H
CH(Me)CH2OMe H
CH(Me)CH2OEt H
CH(Me)CH2O(D1-104c) H
CH(Et)CH2OH H
CH(Et)CH2OMe H
CH(Et)CH2OEt H
CH(Et)CH2O(D1-104c) H
CH(n-Pr)CH2OH H
CH(n-Pr)CH2OMe H
CH(n-Pr)CH2OEt H
CH(n-Pr)CH2O(D1-104c) H
CH(i-Pr)CH2OH H
CH(i-Pr)CH2OMe H
CH(i-Pr)CH2OEt H
CH(i-Pr)CH2O(D1-104c) H
CH(n-Bu)CH2OH H
CH(n-Bu)CH2OMe H
CH(n-Bu)CH2OEt H
CH(n-Bu)CH2O(D1-104c) H
C(Me)2CH2OH H
C(Me)2CH2OMe H
C(Me)2CH2OEt H
C(Me)2CH2O(D1-104c) H
CH2SH H
CH2SMe H
CH2SEt H
CH2SPr-n H
CH2SPr-i H
CH2SBu-n H
CH2SBu-i H
CH2SBu-t H
CH2SPen-n H
CH2SHex-n H
CH2SPr-c H
CH2SBu-c H
CH2SPen-c H
CH2SHex-c H
CH2SCH2CH=CH2 H
CH2SCH2C三CH H
CH2SCF2H H
CH2SCF3 H
CH2SCF2Cl H
CH2SCH2CF3 H
CH2S{D1-108c} H
CH2S(O)Me H
CH2S(O)Et H
CH2S(O)Pr-n H
CH2S(O)Pr-i H
CH2S(O)Bu-n H
CH2S(O)Bu-i H
CH2S(O)Bu-t H
CH2S(O)Pen-n H
CH2S(O)Hex-n H
CH2S(O)Pr-c H
CH2S(O)Bu-c H
CH2S(O)Pen-c H
CH2S(O)Hex-c H
CH2S(O)CH2CH=CH2 H
CH2S(O)CH2C三CH H
CH2S(O)CF2H H
CH2S(O)CF3 H
CH2S(O)CF2Cl H
CH2S(O)CH2CF3 H
CH2S(O){D1-108c} H
CH2S(O)2Me H
CH2S(O)2Et H
CH2S(O)2Pr-n H
CH2S(O)2Pr-i H
CH2S(O)2Bu-n H
CH2S(O)2Bu-i H
CH2S(O)2Bu-t H
CH2S(O)2Pen-n H
CH2S(O)2Hex-n H
CH2S(O)2Pr-c H
CH2S(O)2Bu-c H
CH2S(O)2Pen-c H
CH2S(O)2Hex-c H
CH2S(O)2CH2CH=CH2 H
CH2S(O)2CH2C三CH H
CH2S(O)2CF2H H
CH2S(O)2CF3 H
CH2S(O)2CF2Cl H
CH2S(O)2CH2CF3 H
CH2S(O)2{D1-108c} H
CH(Me)SH H
CH(Me)SMe H
CH(Me)SEt H
CH(Me)SPr-n H
CH(Me)SPr-i H
CH(Me)SBu-n H
CH(Me)SBu-i H
CH(Me)SBu-t H
CH(Me)SPen-n H
CH(Me)SHex-n H
CH(Me)SPr-c H
CH(Me)SBu-c H
CH(Me)SPen-c H
CH(Me)SHex-c H
CH(Me)SCH2CH=CH2 H
CH(Me)SCH2C三CH H
CH(Me)SCF2H H
CH(Me)SCF3 H
CH(Me)SCF2Cl H
CH(Me)SCH2CF3 H
CH(Me)S{D1-108c} H
CH(Me)S(O)Me H
CH(Me)S(O)Et H
CH(Me)S(O)Pr-n H
CH(Me)S(O)Pr-i H
CH(Me)S(O)Bu-n H
CH(Me)S(O)Bu-i H
CH(Me)S(O)Bu-t H
CH(Me)S(O)Pen-n H
CH(Me)S(O)Hex-n H
CH(Me)S(O)Pr-c H
CH(Me)S(O)Bu-c H
CH(Me)S(O)Pen-c H
CH(Me)S(O)Hex-c H
CH(Me)S(O)CH2CH=CH2 H
CH(Me)S(O)CH2C三CH H
CH(Me)S(O)CF2H H
CH(Me)S(O)CF3 H
CH(Me)S(O)CF2Cl H
CH(Me)S(O)CH2CF3 H
CH(Me)S(O){D1-108c} H
CH(Me)S(O)2Me H
CH(Me)S(O)2Et H
CH(Me)S(O)2Pr-n H
CH(Me)S(O)2Pr-i H
CH(Me)S(O)2Bu-n H
CH(Me)S(O)2Bu-i H
CH(Me)S(O)2Bu-t H
CH(Me)S(O)2Pen-n H
CH(Me)S(O)2Hex-n H
CH(Me)S(O)2Pr-c H
CH(Me)S(O)2Bu-c H
CH(Me)S(O)2Pen-c H
CH(Me)S(O)2Hex-c H
CH(Me)S(O)2CH2CH=CH2 H
CH(Me)S(O)2CH2C三CH H
CH(Me)S(O)2CF2H H
CH(Me)S(O)2CF3 H
CH(Me)S(O)2CF2Cl H
CH(Me)S(O)2CH2CF3 H
CH(Me)S(O)2{D1-108c} H
CH(Et)SH H
CH(Et)SMe H
CH(Et)SEt H
CH(Et)SPr-n H
CH(Et)SPr-i H
CH(Et)SBu-n H
CH(Et)SBu-i H
CH(Et)SBu-t H
CH(Et)SPen-n H
CH(Et)SHex-n H
CH(Et)SPr-c H
CH(Et)SBu-c H
CH(Et)SPen-c H
CH(Et)SHex-c H
CH(Et)SCH2CH=CH2 H
CH(Et)SCH2C三CH H
CH(Et)SCF2H H
CH(Et)SCF3 H
CH(Et)SCF2Cl H
CH(Et)SCH2CF3 H
CH(Et)S{D1-108c} H
CH(Et)S(O)Me H
CH(Et)S(O)Et H
CH(Et)S(O)Pr-n H
CH(Et)S(O)Pr-i H
CH(Et)S(O)Bu-n H
CH(Et)S(O)Bu-i H
CH(Et)S(O)Bu-t H
CH(Et)S(O)Pen-n H
CH(Et)S(O)Hex-n H
CH(Et)S(O)Pr-c H
CH(Et)S(O)Bu-c H
CH(Et)S(O)Pen-c H
CH(Et)S(O)Hex-c H
CH(Et)S(O)CH2CH=CH2 H
CH(Et)S(O)CH2C三CH H
CH(Et)S(O)CF2H H
CH(Et)S(O)CF3 H
CH(Et)S(O)CF2Cl H
CH(Et)S(O)CH2CF3 H
CH(Et)S(O){D1-108c} H
CH(Et)S(O)2Me H
CH(Et)S(O)2Et H
CH(Et)S(O)2Pr-n H
CH(Et)S(O)2Pr-i H
CH(Et)S(O)2Bu-n H
CH(Et)S(O)2Bu-i H
CH(Et)S(O)2Bu-t H
CH(Et)S(O)2Pen-n H
CH(Et)S(O)2Hex-n H
CH(Et)S(O)2Pr-c H
CH(Et)S(O)2Bu-c H
CH(Et)S(O)2Pen-c H
CH(Et)S(O)2Hex-c H
CH(Et)S(O)2CH2CH=CH2 H
CH(Et)S(O)2CH2C三CH H
CH(Et)S(O)2CF2H H
CH(Et)S(O)2CF3 H
CH(Et)S(O)2CF2Cl H
CH(Et)S(O)2CH2CF3 H
CH(Et)S(O)2{D1-108c} H
CH(n-Pr)SH H
CH(n-Pr)SMe H
CH(n-Pr)SEt H
CH(n-Pr)SPr-n H
CH(n-Pr)SPr-i H
CH(n-Pr)SBu-n H
CH(n-Pr)SBu-i H
CH(n-Pr)SBu-t H
CH(n-Pr)SPen-n H
CH(n-Pr)SHex-n H
CH(n-Pr)SPr-c H
CH(n-Pr)SBu-c H
CH(n-Pr)SPen-c H
CH(n-Pr)SHex-c H
CH(n-Pr)SCH2CH=CH2 H
CH(n-Pr)SCH2C三CH H
CH(n-Pr)SCF2H H
CH(n-Pr)SCF3 H
CH(n-Pr)SCF2Cl H
CH(n-Pr)SCH2CF3 H
CH(n-Pr)S{D1-108c} H
CH(n-Pr)S(O)Me H
CH(n-Pr)S(O)Et H
CH(n-Pr)S(O)Pr-n H
CH(n-Pr)S(O)Pr-i H
CH(n-Pr)S(O)Bu-n H
CH(n-Pr)S(O)Bu-i H
CH(n-Pr)S(O)Bu-t H
CH(n-Pr)S(O)Pen-n H
CH(n-Pr)S(O)Hex-n H
CH(n-Pr)S(O)Pr-c H
CH(n-Pr)S(O)Bu-c H
CH(n-Pr)S(O)Pen-c H
CH(n-Pr)S(O)Hex-c H
CH(n-Pr)S(O)CH2CH=CH2 H
CH(n-Pr)S(O)CH2C三CH H
CH(n-Pr)S(O)CF2H H
CH(n-Pr)S(O)CF3 H
CH(n-Pr)S(O)CF2Cl H
CH(n-Pr)S(O)CH2CF3 H
CH(n-Pr)S(O){D1-108c} H
CH(n-Pr)S(O)2Me H
CH(n-Pr)S(O)2Et H
CH(n-Pr)S(O)2Pr-n H
CH(n-Pr)S(O)2Pr-i H
CH(n-Pr)S(O)2Bu-n H
CH(n-Pr)S(O)2Bu-i H
CH(n-Pr)S(O)2Bu-t H
CH(n-Pr)S(O)2Pen-n H
CH(n-Pr)S(O)2Hex-n H
CH(n-Pr)S(O)2Pr-c H
CH(n-Pr)S(O)2Bu-c H
CH(n-Pr)S(O)2Pen-c H
CH(n-Pr)S(O)2Hex-c H
CH(n-Pr)S(O)2CH2CH=CH2 H
CH(n-Pr)S(O)2CH2C三CH H
CH(n-Pr)S(O)2CF2H H
CH(n-Pr)S(O)2CF3 H
CH(n-Pr)S(O)2CF2Cl H
CH(n-Pr)S(O)2CH2CF3 H
CH(n-Pr)S(O)2{D1-108c} H
CH(i-Pr)SH H
CH(i-Pr)SMe H
CH(i-Pr)SEt H
CH(i-Pr)SPr-n H
CH(i-Pr)SPr-i H
CH(i-Pr)SBu-n H
CH(i-Pr)SBu-i H
CH(i-Pr)SBu-t H
CH(i-Pr)SPen-n H
CH(i-Pr)SHex-n H
CH(i-Pr)SPr-c H
CH(i-Pr)SBu-c H
CH(i-Pr)SPen-c H
CH(i-Pr)SHex-c H
CH(i-Pr)SCH2CH=CH2 H
CH(i-Pr)SCH2C三CH H
CH(i-Pr)SCF2H H
CH(i-Pr)SCF3 H
CH(i-Pr)SCF2Cl H
CH(i-Pr)SCH2CF3 H
CH(i-Pr)S{D1-108c} H
CH(i-Pr)S(O)Me H
CH(i-Pr)S(O)Et H
CH(i-Pr)S(O)Pr-n H
CH(i-Pr)S(O)Pr-i H
CH(i-Pr)S(O)Bu-n H
CH(i-Pr)S(O)Bu-i H
CH(i-Pr)S(O)Bu-t H
CH(i-Pr)S(O)Pen-n H
CH(i-Pr)S(O)Hex-n H
CH(i-Pr)S(O)Pr-c H
CH(i-Pr)S(O)Bu-c H
CH(i-Pr)S(O)Pen-c H
CH(i-Pr)S(O)Hex-c H
CH(i-Pr)S(O)CH2CH=CH2 H
CH(i-Pr)S(O)CH2C三CH H
CH(i-Pr)S(O)CF2H H
CH(i-Pr)S(O)CF3 H
CH(i-Pr)S(O)CF2Cl H
CH(i-Pr)S(O)CH2CF3 H
CH(i-Pr)S(O){D1-108c} H
CH(i-Pr)S(O)2Me H
CH(i-Pr)S(O)2Et H
CH(i-Pr)S(O)2Pr-n H
CH(i-Pr)S(O)2Pr-i H
CH(i-Pr)S(O)2Bu-n H
CH(i-Pr)S(O)2Bu-i H
CH(i-Pr)S(O)2Bu-t H
CH(i-Pr)S(O)2Pen-n H
CH(i-Pr)S(O)2Hex-n H
CH(i-Pr)S(O)2Pr-c H
CH(i-Pr)S(O)2Bu-c H
CH(i-Pr)S(O)2Pen-c H
CH(i-Pr)S(O)2Hex-c H
CH(i-Pr)S(O)2CH2CH=CH2 H
CH(i-Pr)S(O)2CH2C三CH H
CH(i-Pr)S(O)2CF2H H
CH(i-Pr)S(O)2CF3 H
CH(i-Pr)S(O)2CF2Cl H
CH(i-Pr)S(O)2CH2CF3 H
CH(i-Pr)S(O)2{D1-108c} H
CH(n-Bu)SH H
CH(n-Bu)SMe H
CH(n-Bu)SEt H
CH(n-Bu)SPr-n H
CH(n-Bu)SPr-i H
CH(n-Bu)SBu-n H
CH(n-Bu)SBu-i H
CH(n-Bu)SBu-t H
CH(n-Bu)SPen-n H
CH(n-Bu)SHex-n H
CH(n-Bu)SPr-c H
CH(n-Bu)SBu-c H
CH(n-Bu)SPen-c H
CH(n-Bu)SHex-c H
CH(n-Bu)SCH2CH=CH2 H
CH(n-Bu)SCH2C三CH H
CH(n-Bu)SCF2H H
CH(n-Bu)SCF3 H
CH(n-Bu)SCF2Cl H
CH(n-Bu)SCH2CF3 H
CH(n-Bu)S{D1-108c} H
CH(n-Bu)S(O)Me H
CH(n-Bu)S(O)Et H
CH(n-Bu)S(O)Pr-n H
CH(n-Bu)S(O)Pr-i H
CH(n-Bu)S(O)Bu-n H
CH(n-Bu)S(O)Bu-i H
CH(n-Bu)S(O)Bu-t H
CH(n-Bu)S(O)Pen-n H
CH(n-Bu)S(O)Hex-n H
CH(n-Bu)S(O)Pr-c H
CH(n-Bu)S(O)Bu-c H
CH(n-Bu)S(O)Pen-c H
CH(n-Bu)S(O)Hex-c H
CH(n-Bu)S(O)CH2CH=CH2 H
CH(n-Bu)S(O)CH2C三CH H
CH(n-Bu)S(O)CF2H H
CH(n-Bu)S(O)CF3 H
CH(n-Bu)S(O)CF2Cl H
CH(n-Bu)S(O)CH2CF3 H
CH(n-Bu)S(O){D1-108c} H
CH(n-Bu)S(O)2Me H
CH(n-Bu)S(O)2Et H
CH(n-Bu)S(O)2Pr-n H
CH(n-Bu)S(O)2Pr-i H
CH(n-Bu)S(O)2Bu-n H
CH(n-Bu)S(O)2Bu-i H
CH(n-Bu)S(O)2Bu-t H
CH(n-Bu)S(O)2Pen-n H
CH(n-Bu)S(O)2Hex-n H
CH(n-Bu)S(O)2Pr-c H
CH(n-Bu)S(O)2Bu-c H
CH(n-Bu)S(O)2Pen-c H
CH(n-Bu)S(O)2Hex-c H
CH(n-Bu)S(O)2CH2CH=CH2 H
CH(n-Bu)S(O)2CH2C三CH H
CH(n-Bu)S(O)2CF2H H
CH(n-Bu)S(O)2CF3 H
CH(n-Bu)S(O)2CF2Cl H
CH(n-Bu)S(O)2CH2CF3 H
CH(n-Bu)S(O)2{D1-108c} H
CH(CH2OMe)SH H
CH(CH2OMe)SMe H
CH(CH2OMe)SEt H
CH(CH2OMe)SPr-n H
CH(CH2OMe)SPr-i H
CH(CH2OMe)SBu-n H
CH(CH2OMe)SBu-i H
CH(CH2OMe)SBu-t H
CH(CH2OMe)SPen-n H
CH(CH2OMe)SHex-n H
CH(CH2OMe)SPr-c H
CH(CH2OMe)SBu-c H
CH(CH2OMe)SPen-c H
CH(CH2OMe)SHex-c H
CH(CH2OMe)SCH2CH=CH2 H
CH(CH2OMe)SCH2C三CH H
CH(CH2OMe)SCF2H H
CH(CH2OMe)SCF3 H
CH(CH2OMe)SCF2Cl H
CH(CH2OMe)SCH2CF3 H
CH(CH2OMe)S{D1-108c} H
CH(CH2OMe)S(O)Me H
CH(CH2OMe)S(O)Et H
CH(CH2OMe)S(O)Pr-n H
CH(CH2OMe)S(O)Pr-i H
CH(CH2OMe)S(O)Bu-n H
CH(CH2OMe)S(O)Bu-i H
CH(CH2OMe)S(O)Bu-t H
CH(CH2OMe)S(O)Pen-n H
CH(CH2OMe)S(O)Hex-n H
CH(CH2OMe)S(O)Pr-c H
CH(CH2OMe)S(O)Bu-c H
CH(CH2OMe)S(O)Pen-c H
CH(CH2OMe)S(O)Hex-c H
CH(CH2OMe)S(O)CH2CH=CH2 H
CH(CH2OMe)S(O)CH2C三CH H
CH(CH2OMe)S(O)CF2H H
CH(CH2OMe)S(O)CF3 H
CH(CH2OMe)S(O)CF2Cl H
CH(CH2OMe)S(O)CH2CF3 H
CH(CH2OMe)S(O){D1-108c} H
CH(CH2OMe)S(O)2Me H
CH(CH2OMe)S(O)2Et H
CH(CH2OMe)S(O)2Pr-n H
CH(CH2OMe)S(O)2Pr-i H
CH(CH2OMe)S(O)2Bu-n H
CH(CH2OMe)S(O)2Bu-i H
CH(CH2OMe)S(O)2Bu-t H
CH(CH2OMe)S(O)2Pen-n H
CH(CH2OMe)S(O)2Hex-n H
CH(CH2OMe)S(O)2Pr-c H
CH(CH2OMe)S(O)2Bu-c H
CH(CH2OMe)S(O)2Pen-c H
CH(CH2OMe)S(O)2Hex-c H
CH(CH2OMe)S(O)2CH2CH=CH2 H
CH(CH2OMe)S(O)2CH2C三CH H
CH(CH2OMe)S(O)2CF2H H
CH(CH2OMe)S(O)2CF3 H
CH(CH2OMe)S(O)2CF2Cl H
CH(CH2OMe)S(O)2CH2CF3 H
CH(CH2OMe)S(O)2{D1-108c} H
CH(CH2CH=CH2)SH H
CH(CH2CH=CH2)SMe H
CH(CH2CH=CH2)SEt H
CH(CH2CH=CH2)SPr-n H
CH(CH2CH=CH2)SPr-i H
CH(CH2CH=CH2)SBu-n H
CH(CH2CH=CH2)SBu-i H
CH(CH2CH=CH2)SBu-t H
CH(CH2CH=CH2)SPen-n H
CH(CH2CH=CH2)SHex-n H
CH(CH2CH=CH2)SPr-c H
CH(CH2CH=CH2)SBu-c H
CH(CH2CH=CH2)SPen-c H
CH(CH2CH=CH2)SHex-c H
CH(CH2CH=CH2)SCH2CH=CH2 H
CH(CH2CH=CH2)SCH2C三CH H
CH(CH2CH=CH2)SCF2H H
CH(CH2CH=CH2)SCF3 H
CH(CH2CH=CH2)SCF2Cl H
CH(CH2CH=CH2)SCH2CF3 H
CH(CH2CH=CH2)S{D1-108c} H
CH(CH2CH=CH2)S(O)Me H
CH(CH2CH=CH2)S(O)Et H
CH(CH2CH=CH2)S(O)Pr-n H
CH(CH2CH=CH2)S(O)Pr-i H
CH(CH2CH=CH2)S(O)Bu-n H
CH(CH2CH=CH2)S(O)Bu-i H
CH(CH2CH=CH2)S(O)Bu-t H
CH(CH2CH=CH2)S(O)Pen-n H
CH(CH2CH=CH2)S(O)Hex-n H
CH(CH2CH=CH2)S(O)Pr-c H
CH(CH2CH=CH2)S(O)Bu-c H
CH(CH2CH=CH2)S(O)Pen-c H
CH(CH2CH=CH2)S(O)Hex-c H
CH(CH2CH=CH2)S(O)CH2CH=CH2 H
CH(CH2CH=CH2)S(O)CH2C三CH H
CH(CH2CH=CH2)S(O)CF2H H
CH(CH2CH=CH2)S(O)CF3 H
CH(CH2CH=CH2)S(O)CF2Cl H
CH(CH2CH=CH2)S(O)CH2CF3 H
CH(CH2CH=CH2)S(O){D1-108c} H
CH(CH2CH=CH2)S(O)2Me H
CH(CH2CH=CH2)S(O)2Et H
CH(CH2CH=CH2)S(O)2Pr-n H
CH(CH2CH=CH2)S(O)2Pr-i H
CH(CH2CH=CH2)S(O)2Bu-n H
CH(CH2CH=CH2)S(O)2Bu-i H
CH(CH2CH=CH2)S(O)2Bu-t H
CH(CH2CH=CH2)S(O)2Pen-n H
CH(CH2CH=CH2)S(O)2Hex-n H
CH(CH2CH=CH2)S(O)2Pr-c H
CH(CH2CH=CH2)S(O)2Bu-c H
CH(CH2CH=CH2)S(O)2Pen-c H
CH(CH2CH=CH2)S(O)2Hex-c H
CH(CH2CH=CH2)S(O)2CH2CH=CH2 H
CH(CH2CH=CH2)S(O)2CH2C三CH H
CH(CH2CH=CH2)S(O)2CF2H H
CH(CH2CH=CH2)S(O)2CF3 H
CH(CH2CH=CH2)S(O)2CF2Cl H
CH(CH2CH=CH2)S(O)2CH2CF3 H
CH(CH2CH=CH2)S(O)2{D1-108c} H
CH(CH2C≡CH)SH H
CH(CH2C≡CH)SMe H
CH(CH2C≡CH)SEt H
CH(CH2C≡CH)SPr-n H
CH(CH2C≡CH)SPr-i H
CH(CH2C≡CH)SBu-n H
CH(CH2C≡CH)SBu-i H
CH(CH2C≡CH)SBu-t H
CH(CH2C≡CH)SPen-n H
CH(CH2C≡CH)SHex-n H
CH(CH2C≡CH)SPr-c H
CH(CH2C≡CH)SBu-c H
CH(CH2C≡CH)SPen-c H
CH(CH2C≡CH)SHex-c H
CH(CH2C≡CH)SCH2CH=CH2 H
CH(CH2C≡CH)SCH2C三CH H
CH(CH2C≡CH)SCF2H H
CH(CH2C≡CH)SCF3 H
CH(CH2C≡CH)SCF2Cl H
CH(CH2C≡CH)SCH2CF3 H
CH(CH2C≡CH)S{D1-108c} H
CH(CH2C≡CH)S(O)Me H
CH(CH2C≡CH)S(O)Et H
CH(CH2C≡CH)S(O)Pr-n H
CH(CH2C≡CH)S(O)Pr-i H
CH(CH2C≡CH)S(O)Bu-n H
CH(CH2C≡CH)S(O)Bu-i H
CH(CH2C≡CH)S(O)Bu-t H
CH(CH2C≡CH)S(O)Pen-n H
CH(CH2C≡CH)S(O)Hex-n H
CH(CH2C≡CH)S(O)Pr-c H
CH(CH2C≡CH)S(O)Bu-c H
CH(CH2C≡CH)S(O)Pen-c H
CH(CH2C≡CH)S(O)Hex-c H
CH(CH2C≡CH)S(O)CH2CH=CH2 H
CH(CH2C≡CH)S(O)CH2C三CH H
CH(CH2C≡CH)S(O)CF2H H
CH(CH2C≡CH)S(O)CF3 H
CH(CH2C≡CH)S(O)CF2Cl H
CH(CH2C≡CH)S(O)CH2CF3 H
CH(CH2C≡CH)S(O){D1-108c} H
CH(CH2C≡CH)S(O)2Me H
CH(CH2C≡CH)S(O)2Et H
CH(CH2C≡CH)S(O)2Pr-n H
CH(CH2C≡CH)S(O)2Pr-i H
CH(CH2C≡CH)S(O)2Bu-n H
CH(CH2C≡CH)S(O)2Bu-i H
CH(CH2C≡CH)S(O)2Bu-t H
CH(CH2C≡CH)S(O)2Pen-n H
CH(CH2C≡CH)S(O)2Hex-n H
CH(CH2C≡CH)S(O)2Pr-c H
CH(CH2C≡CH)S(O)2Bu-c H
CH(CH2C≡CH)S(O)2Pen-c H
CH(CH2C≡CH)S(O)2Hex-c H
CH(CH2C≡CH)S(O)2CH2CH=CH2 H
CH(CH2C≡CH)S(O)2CH2C三CH H
CH(CH2C≡CH)S(O)2CF2H H
CH(CH2C≡CH)S(O)2CF3 H
CH(CH2C≡CH)S(O)2CF2Cl H
CH(CH2C≡CH)S(O)2CH2CF3 H
CH(CH2C≡CH)S(O)2{D1-108c} H
CH(CH2CN)SH H
CH(CH2CN)SMe H
CH(CH2CN)SEt H
CH(CH2CN)SPr-n H
CH(CH2CN)SPr-i H
CH(CH2CN)SBu-n H
CH(CH2CN)SBu-i H
CH(CH2CN)SBu-t H
CH(CH2CN)SPen-n H
CH(CH2CN)SHex-n H
CH(CH2CN)SPr-c H
CH(CH2CN)SBu-c H
CH(CH2CN)SPen-c H
CH(CH2CN)SHex-c H
CH(CH2CN)SCH2CH=CH2 H
CH(CH2CN)SCH2C三CH H
CH(CH2CN)SCF2H H
CH(CH2CN)SCF3 H
CH(CH2CN)SCF2Cl H
CH(CH2CN)SCH2CF3 H
CH(CH2CN)S{D1-108c} H
CH(CH2CN)S(O)Me H
CH(CH2CN)S(O)Et H
CH(CH2CN)S(O)Pr-n H
CH(CH2CN)S(O)Pr-i H
CH(CH2CN)S(O)Bu-n H
CH(CH2CN)S(O)Bu-i H
CH(CH2CN)S(O)Bu-t H
CH(CH2CN)S(O)Pen-n H
CH(CH2CN)S(O)Hex-n H
CH(CH2CN)S(O)Pr-c H
CH(CH2CN)S(O)Bu-c H
CH(CH2CN)S(O)Pen-c H
CH(CH2CN)S(O)Hex-c H
CH(CH2CN)S(O)CH2CH=CH2 H
CH(CH2CN)S(O)CH2C三CH H
CH(CH2CN)S(O)CF2H H
CH(CH2CN)S(O)CF3 H
CH(CH2CN)S(O)CF2Cl H
CH(CH2CN)S(O)CH2CF3 H
CH(CH2CN)S(O){D1-108c} H
CH(CH2CN)S(O)2Me H
CH(CH2CN)S(O)2Et H
CH(CH2CN)S(O)2Pr-n H
CH(CH2CN)S(O)2Pr-i H
CH(CH2CN)S(O)2Bu-n H
CH(CH2CN)S(O)2Bu-i H
CH(CH2CN)S(O)2Bu-t H
CH(CH2CN)S(O)2Pen-n H
CH(CH2CN)S(O)2Hex-n H
CH(CH2CN)S(O)2Pr-c H
CH(CH2CN)S(O)2Bu-c H
CH(CH2CN)S(O)2Pen-c H
CH(CH2CN)S(O)2Hex-c H
CH(CH2CN)S(O)2CH2CH=CH2 H
CH(CH2CN)S(O)2CH2C三CH H
CH(CH2CN)S(O)2CF2H H
CH(CH2CN)S(O)2CF3 H
CH(CH2CN)S(O)2CF2Cl H
CH(CH2CN)S(O)2CH2CF3 H
CH(CH2CN)S(O)2{D1-108c} H
CH(Me)2SH H
CH(Me)2SMe H
CH(Me)2SEt H
CH(Me)2SPr-n H
CH(Me)2SPr-i H
CH(Me)2SBu-n H
CH(Me)2SBu-i H
CH(Me)2SBu-t H
CH(Me)2SPen-n H
CH(Me)2SHex-n H
CH(Me)2SPr-c H
CH(Me)2SBu-c H
CH(Me)2SPen-c H
CH(Me)2SHex-c H
CH(Me)2SCH2CH=CH2 H
CH(Me)2SCH2C三CH H
CH(Me)2SCF2H H
CH(Me)2SCF3 H
CH(Me)2SCF2Cl H
CH(Me)2SCH2CF3 H
CH(Me)2S{D1-108c} H
CH(Me)2S(O)Me H
CH(Me)2S(O)Et H
CH(Me)2S(O)Pr-n H
CH(Me)2S(O)Pr-i H
CH(Me)2S(O)Bu-n H
CH(Me)2S(O)Bu-i H
CH(Me)2S(O)Bu-t H
CH(Me)2S(O)Pen-n H
CH(Me)2S(O)Hex-n H
CH(Me)2S(O)Pr-c H
CH(Me)2S(O)Bu-c H
CH(Me)2S(O)Pen-c H
CH(Me)2S(O)Hex-c H
CH(Me)2S(O)CH2CH=CH2 H
CH(Me)2S(O)CH2C三CH H
CH(Me)2S(O)CF2H H
CH(Me)2S(O)CF3 H
CH(Me)2S(O)CF2Cl H
CH(Me)2S(O)CH2CF3 H
CH(Me)2S(O){D1-108c} H
CH(Me)2S(O)2Me H
CH(Me)2S(O)2Et H
CH(Me)2S(O)2Pr-n H
CH(Me)2S(O)2Pr-i H
CH(Me)2S(O)2Bu-n H
CH(Me)2S(O)2Bu-i H
CH(Me)2S(O)2Bu-t H
CH(Me)2S(O)2Pen-n H
CH(Me)2S(O)2Hex-n H
CH(Me)2S(O)2Pr-c H
CH(Me)2S(O)2Bu-c H
CH(Me)2S(O)2Pen-c H
CH(Me)2S(O)2Hex-c H
CH(Me)2S(O)2CH2CH=CH2 H
CH(Me)2S(O)2CH2C三CH H
CH(Me)2S(O)2CF2H H
CH(Me)2S(O)2CF3 H
CH(Me)2S(O)2CF2Cl H
CH(Me)2S(O)2CH2CF3 H
CH(Me)2S(O)2{D1-108c} H
CH2CH2SH H
CH2CH2SMe H
CH2CH2SEt H
CH2CH2SPr-n H
CH2CH2SPr-i H
CH2CH2SBu-n H
CH2CH2SBu-i H
CH2CH2SBu-t H
CH2CH2SPen-n H
CH2CH2SHex-n H
CH2CH2SPr-c H
CH2CH2SBu-c H
CH2CH2SPen-c H
CH2CH2SHex-c H
CH2CH2SCH2CH=CH2 H
CH2CH2SCH2C三CH H
CH2CH2SCF2H H
CH2CH2SCF3 H
CH2CH2SCF2Cl H
CH2CH2SCH2CF3 H
CH2CH2S{D1-108c} H
CH2CH2S(O)Me H
CH2CH2S(O)Et H
CH2CH2S(O)Pr-n H
CH2CH2S(O)Pr-i H
CH2CH2S(O)Bu-n H
CH2CH2S(O)Bu-i H
CH2CH2S(O)Bu-t H
CH2CH2S(O)Pen-n H
CH2CH2S(O)Hex-n H
CH2CH2S(O)Pr-c H
CH2CH2S(O)Bu-c H
CH2CH2S(O)Pen-c H
CH2CH2S(O)Hex-c H
CH2CH2S(O)CH2CH=CH2 H
CH2CH2S(O)CH2C三CH H
CH2CH2S(O)CF2H H
CH2CH2S(O)CF3 H
CH2CH2S(O)CF2Cl H
CH2CH2S(O)CH2CF3 H
CH2CH2S(O){D1-108c} H
CH2CH2S(O)2Me H
CH2CH2S(O)2Et H
CH2CH2S(O)2Pr-n H
CH2CH2S(O)2Pr-i H
CH2CH2S(O)2Bu-n H
CH2CH2S(O)2Bu-i H
CH2CH2S(O)2Bu-t H
CH2CH2S(O)2Pen-n H
CH2CH2S(O)2Hex-n H
CH2CH2S(O)2Pr-c H
CH2CH2S(O)2Bu-c H
CH2CH2S(O)2Pen-c H
CH2CH2S(O)2Hex-c H
CH2CH2S(O)2CH2CH=CH2 H
CH2CH2S(O)2CH2C三CH H
CH2CH2S(O)2CF2H H
CH2CH2S(O)2CF3 H
CH2CH2S(O)2CF2Cl H
CH2CH2S(O)2CH2CF3 H
CH2CH2S(O)2{D1-108c} H
CH(Me)CH2SH H
CH(Me)CH2SMe H
CH(Me)CH2SEt H
CH(Me)CH2SPr-n H
CH(Me)CH2SPr-i H
CH(Me)CH2SBu-n H
CH(Me)CH2SBu-i H
CH(Me)CH2SBu-t H
CH(Me)CH2SPen-n H
CH(Me)CH2SHex-n H
CH(Me)CH2SPr-c H
CH(Me)CH2SBu-c H
CH(Me)CH2SPen-c H
CH(Me)CH2SHex-c H
CH(Me)CH2SCH2CH=CH2 H
CH(Me)CH2SCH2C三CH H
CH(Me)CH2SCF2H H
CH(Me)CH2SCF3 H
CH(Me)CH2SCF2Cl H
CH(Me)CH2SCH2CF3 H
CH(Me)CH2S{D1-108c} H
CH(Me)CH2S(O)Me H
CH(Me)CH2S(O)Et H
CH(Me)CH2S(O)Pr-n H
CH(Me)CH2S(O)Pr-i H
CH(Me)CH2S(O)Bu-n H
CH(Me)CH2S(O)Bu-i H
CH(Me)CH2S(O)Bu-t H
CH(Me)CH2S(O)Pen-n H
CH(Me)CH2S(O)Hex-n H
CH(Me)CH2S(O)Pr-c H
CH(Me)CH2S(O)Bu-c H
CH(Me)CH2S(O)Pen-c H
CH(Me)CH2S(O)Hex-c H
CH(Me)CH2S(O)CH2CH=CH2 H
CH(Me)CH2S(O)CH2C三CH H
CH(Me)CH2S(O)CF2H H
CH(Me)CH2S(O)CF3 H
CH(Me)CH2S(O)CF2Cl H
CH(Me)CH2S(O)CH2CF3 H
CH(Me)CH2S(O){D1-108c} H
CH(Me)CH2S(O)2Me H
CH(Me)CH2S(O)2Et H
CH(Me)CH2S(O)2Pr-n H
CH(Me)CH2S(O)2Pr-i H
CH(Me)CH2S(O)2Bu-n H
CH(Me)CH2S(O)2Bu-i H
CH(Me)CH2S(O)2Bu-t H
CH(Me)CH2S(O)2Pen-n H
CH(Me)CH2S(O)2Hex-n H
CH(Me)CH2S(O)2Pr-c H
CH(Me)CH2S(O)2Bu-c H
CH(Me)CH2S(O)2Pen-c H
CH(Me)CH2S(O)2Hex-c H
CH(Me)CH2S(O)2CH2CH=CH2 H
CH(Me)CH2S(O)2CH2C三CH H
CH(Me)CH2S(O)2CF2H H
CH(Me)CH2S(O)2CF3 H
CH(Me)CH2S(O)2CF2Cl H
CH(Me)CH2S(O)2CH2CF3 H
CH(Me)CH2S(O)2{D1-108c} H
CH(Me)CH(Me)SH H
CH(Me)CH(Me)SMe H
CH(Me)CH(Me)SEt H
CH(Me)CH(Me)SPr-n H
CH(Me)CH(Me)SPr-i H
CH(Me)CH(Me)SBu-n H
CH(Me)CH(Me)SBu-i H
CH(Me)CH(Me)SBu-t H
CH(Me)CH(Me)SPen-n H
CH(Me)CH(Me)SHex-n H
CH(Me)CH(Me)SPr-c H
CH(Me)CH(Me)SBu-c H
CH(Me)CH(Me)SPen-c H
CH(Me)CH(Me)SHex-c H
CH(Me)CH(Me)SCH2CH=CH2 H
CH(Me)CH(Me)SCH2C三CH H
CH(Me)CH(Me)SCF2H H
CH(Me)CH(Me)SCF3 H
CH(Me)CH(Me)SCF2Cl H
CH(Me)CH(Me)SCH2CF3 H
CH(Me)CH(Me)S{D1-108c} H
CH(Me)CH(Me)S(O)Me H
CH(Me)CH(Me)S(O)Et H
CH(Me)CH(Me)S(O)Pr-n H
CH(Me)CH(Me)S(O)Pr-i H
CH(Me)CH(Me)S(O)Bu-n H
CH(Me)CH(Me)S(O)Bu-i H
CH(Me)CH(Me)S(O)Bu-t H
CH(Me)CH(Me)S(O)Pen-n H
CH(Me)CH(Me)S(O)Hex-n H
CH(Me)CH(Me)S(O)Pr-c H
CH(Me)CH(Me)S(O)Bu-c H
CH(Me)CH(Me)S(O)Pen-c H
CH(Me)CH(Me)S(O)Hex-c H
CH(Me)CH(Me)S(O)CH2CH=CH2 H
CH(Me)CH(Me)S(O)CH2C三CH H
CH(Me)CH(Me)S(O)CF2H H
CH(Me)CH(Me)S(O)CF3 H
CH(Me)CH(Me)S(O)CF2Cl H
CH(Me)CH(Me)S(O)CH2CF3 H
CH(Me)CH(Me)S(O){D1-108c} H
CH(Me)CH(Me)S(O)2Me H
CH(Me)CH(Me)S(O)2Et H
CH(Me)CH(Me)S(O)2Pr-n H
CH(Me)CH(Me)S(O)2Pr-i H
CH(Me)CH(Me)S(O)2Bu-n H
CH(Me)CH(Me)S(O)2Bu-i H
CH(Me)CH(Me)S(O)2Bu-t H
CH(Me)CH(Me)S(O)2Pen-n H
CH(Me)CH(Me)S(O)2Hex-n H
CH(Me)CH(Me)S(O)2Pr-c H
CH(Me)CH(Me)S(O)2Bu-c H
CH(Me)CH(Me)S(O)2Pen-c H
CH(Me)CH(Me)S(O)2Hex-c H
CH(Me)CH(Me)S(O)2CH2CH=CH2 H
CH(Me)CH(Me)S(O)2CH2C三CH H
CH(Me)CH(Me)S(O)2CF2H H
CH(Me)CH(Me)S(O)2CF3 H
CH(Me)CH(Me)S(O)2CF2Cl H
CH(Me)CH(Me)S(O)2CH2CF3 H
CH(Me)CH(Me)S(O)2{D1-108c} H
CH2CH(Me)SH H
CH2CH(Me)SMe H
CH2CH(Me)SEt H
CH2CH(Me)SPr-n H
CH2CH(Me)SPr-i H
CH2CH(Me)SBu-n H
CH2CH(Me)SBu-i H
CH2CH(Me)SBu-t H
CH2CH(Me)SPen-n H
CH2CH(Me)SHex-n H
CH2CH(Me)SPr-c H
CH2CH(Me)SBu-c H
CH2CH(Me)SPen-c H
CH2CH(Me)SHex-c H
CH2CH(Me)SCH2CH=CH2 H
CH2CH(Me)SCH2C三CH H
CH2CH(Me)SCF2H H
CH2CH(Me)SCF3 H
CH2CH(Me)SCF2Cl H
CH2CH(Me)SCH2CF3 H
CH2CH(Me)S{D1-108c} H
CH2CH(Me)S(O)Me H
CH2CH(Me)S(O)Et H
CH2CH(Me)S(O)Pr-n H
CH2CH(Me)S(O)Pr-i H
CH2CH(Me)S(O)Bu-n H
CH2CH(Me)S(O)Bu-i H
CH2CH(Me)S(O)Bu-t H
CH2CH(Me)S(O)Pen-n H
CH2CH(Me)S(O)Hex-n H
CH2CH(Me)S(O)Pr-c H
CH2CH(Me)S(O)Bu-c H
CH2CH(Me)S(O)Pen-c H
CH2CH(Me)S(O)Hex-c H
CH2CH(Me)S(O)CH2CH=CH2 H
CH2CH(Me)S(O)CH2C三CH H
CH2CH(Me)S(O)CF2H H
CH2CH(Me)S(O)CF3 H
CH2CH(Me)S(O)CF2Cl H
CH2CH(Me)S(O)CH2CF3 H
CH2CH(Me)S(O){D1-108c} H
CH2CH(Me)S(O)2Me H
CH2CH(Me)S(O)2Et H
CH2CH(Me)S(O)2Pr-n H
CH2CH(Me)S(O)2Pr-i H
CH2CH(Me)S(O)2Bu-n H
CH2CH(Me)S(O)2Bu-i H
CH2CH(Me)S(O)2Bu-t H
CH2CH(Me)S(O)2Pen-n H
CH2CH(Me)S(O)2Hex-n H
CH2CH(Me)S(O)2Pr-c H
CH2CH(Me)S(O)2Bu-c H
CH2CH(Me)S(O)2Pen-c H
CH2CH(Me)S(O)2Hex-c H
CH2CH(Me)S(O)2CH2CH=CH2 H
CH2CH(Me)S(O)2CH2C三CH H
CH2CH(Me)S(O)2CF2H H
CH2CH(Me)S(O)2CF3 H
CH2CH(Me)S(O)2CF2Cl H
CH2CH(Me)S(O)2CH2CF3 H
CH2CH(Me)S(O)2{D1-108c} H
C(O)OH H
C(O)OMe H
C(O)OEt H
C(O)OPr-n H
C(O)OPr-i H
C(O)OBu-n H
C(O)OBu-i H
C(O)OBu-s H
C(O)OBu-t H
C(O)OPen-n H
C(O)OHex-n H
CHO H
C(O)Me H
C(O)Et H
C(O)Pr-n H
C(O)Pr-i H
C(O)Bu-n H
C(O)Bu-i H
C(O)Bu-s H
C(O)Bu-t H
C(O)Pen-n H
C(O)Hex-n H
C(O)NHC(O)Me H
C(O)NHMe H
C(O)NHEt H
C(O)NHPr-n H
C(O)NHPr-i H
C(O)NHBu-n H
C(O)NHBu-i H
C(O)NHBu-s H
C(O)NHBu-t H
C(O)NHPen-n H
C(O)NHHex-n H
CN H
Ph H
CH2Cl H
CH2Br H
CH2I H
CH(Me)Cl H
CH(Me)Br H
CH(Me)I H
CH(Et)Cl H
CH(Et)Br H
CH(Et)I H
CH(n-Pr)Cl H
CH(n-Pr)Br H
CH(n-Pr)I H
CH(i-Pr)Cl H
CH(i-Pr)Br H
CH(i-Pr)I H
CH(n-Bu)Cl H
CH(n-Bu)Br H
CH(n-Bu)I H
CH(CH2OMe)Cl H
CH(CH2OMe)Br H
CH(CH2OMe)I H
CH(CH2CH=CH2)Cl H
CH(CH2CH=CH2)Br H
CH(CH2CH=CH2)I H
CH(CH2C三CH)Cl H
CH(CH2C三CH)Br H
CH(CH2C三CH)I H
CH(Me)CH2Cl H
CH(Me)CH2Br H
CH(Me)CH2I H
C(Me)2CH2Cl H
C(Me)2CH2Br H
C(Me)2CH2I H
CH2SCH2Pr-c Me
CH2SCH2Pr-c Et
CH2SCH2Pr-c Pr-n
CH2SCH2Pr-c Pr-i
CH2SCH2Pr-c Pr-c
CH2SCH2Pr-c Bu-n
CH2SCH2Pr-c Bu-i
CH2SCH2Pr-c Bu-c
CH2SCH2Pr-c Bu-s
CH2SCH2Pr-c Bu-t
CH2SCH2Pr-c Pen-n
CH2SCH2Pr-c Pen-c
CH2SCH2Pr-c Hex-n
CH2SCH2Pr-c Hex-c
CH2SCH2Pr-c CH2Pr-c
CH2SCH2Pr-c CH2Bu-c
CH2SCH2Pr-c CH2Pen-c
CH2SCH2Pr-c CH2Hex-c
CH2SCH2Pr-c CH2CH=CH2
CH2SCH2Pr-c CH2CH=C(Cl)2
CH2SCH2Pr-c CH2Pr-c
CH2SCH2Pr-c CH2CN
CH2SCH2Pr-c CH2CF3
CH2SCH2Pr-c CH2OMe
CH2SCH2Pr-c CH2OCF3
CH2SCH2Pr-c CH2SMe
CH2SCH2Pr-c CH2S(O)Me
CH2SCH2Pr-c CH2S(O)2Me
CH2SCH2Pr-c CH2SCF3
CH2SCH2Pr-c CH2S(O)CF3
CH2SCH2Pr-c CH2S(O)2CF3
CH2SCH2Pr-c CH2CH(OMe)2
CH2SCH2Pr-c CH2CH(SMe)2
CH2SCH2Pr-c CH2C(O)Me
CH2SCH2Pr-c CH2C(O)CF3
CH2SCH2Pr-c CH2C(O)OMe
CH2SCH2Pr-c CH2(D1-32a)
CH2SCH2Pr-c CH2(D1-33a)
CH2SCH2Pr-c CH2(D1-34a)
CH2SCH2Pr-c CH2(D1-37a)
CH2SCH2Pr-c CH2(D1-81a)
CH2SCH2Pr-c CH2(D1-82a)
CH2SCH2Pr-c CH2(D1-84a)
CH2SCH2Pr-c CH2(D1-85a)
CH2SCH2Pr-c CH2(D1-87a)
CH2SCH2Pr-c CH2(D1-92a)
CH2SCH2Pr-c CH2(D1-93a)
CH2SCH2Pr-c CH2(D1-95a)
CH2SCH2Pr-c CH2(D1-96a)
CH2SCH2Pr-c CH2(D1-98a)
CH2SCH2Pr-c CH2(D1-108a)
CH2SCH2Pr-c CH2(D1-108b,Z=2-Cl)
CH2SCH2Pr-c CH2(D1-108b,Z=3-Me)
CH2SCH2Pr-c CH2(D1-108b,Z=4-OMe)
CH2SCH2Pr-c CH2(D1-108b,Z=2-SMe)
CH2SCH2Pr-c CH2(D1-108b,Z=3-CF3)
CH2SCH2Pr-c CH2(D1-108b,Z=4-OCF3)
CH2SCH2Pr-c CH2(D1-108b,Z=2-SCF3)
CH2SCH2Pr-c CH2CH2CN
CH2SCH2Pr-c CH2CH2CF3
CH2SCH2Pr-c CH2CH2OMe
CH2SCH2Pr-c CH2CH2SMe
CH2SCH2Pr-c CH2CH2S(O)Me
CH2SCH2Pr-c CH2CH2S(O)2Me
CH2SCH2Pr-c D1-32a
CH2SCH2Pr-c D1-33a
CH2SCH2Pr-c D1-34a
CH2SCH2Pr-c D1-37a
CH2SCH2Pr-c D1-81a
CH2SCH2Pr-c D1-82a
CH2SCH2Pr-c D1-84a
CH2SCH2Pr-c D1-85a
CH2SCH2Pr-c D1-87a
CH2SCH2Pr-c D1-92a
CH2SCH2Pr-c D1-93a
CH2SCH2Pr-c D1-95a
CH2SCH2Pr-c D1-96a
CH2SCH2Pr-c D1-98a
CH2SCH2Pr-c D1-108a
CH2SCH2Pr-c D1-108b(Z=2-Cl)
CH2SCH2Pr-c D1-108b(Z=3-Me)
CH2SCH2Pr-c D1-108b(Z=4-OMe)
CH2SCH2Pr-c D1-108b(Z=2-SMe)
CH2SCH2Pr-c D1-108b(Z=3-CF3)
CH2SCH2Pr-c D1-108b(Z=4-OCF3)
CH2SCH2Pr-c D1-108b(Z=2-SCF3)
CH2SCH2Pr-c C(O)Me
CH2SCH2Pr-c C(O)CF3
CH2SCH2Pr-c C(O)OMe
CH2S(O)CH2Pr-c Me
CH2S(O)CH2Pr-c Et
CH2S(O)CH2Pr-c Pr-n
CH2S(O)CH2Pr-c Pr-i
CH2S(O)CH2Pr-c Pr-c
CH2S(O)CH2Pr-c Bu-n
CH2S(O)CH2Pr-c Bu-i
CH2S(O)CH2Pr-c Bu-c
CH2S(O)CH2Pr-c Bu-s
CH2S(O)CH2Pr-c Bu-t
CH2S(O)CH2Pr-c Pen-n
CH2S(O)CH2Pr-c Pen-c
CH2S(O)CH2Pr-c Hex-n
CH2S(O)CH2Pr-c Hex-c
CH2S(O)CH2Pr-c CH2Pr-c
CH2S(O)CH2Pr-c CH2Bu-c
CH2S(O)CH2Pr-c CH2Pen-c
CH2S(O)CH2Pr-c CH2Hex-c
CH2S(O)CH2Pr-c CH2CH=CH2
CH2S(O)CH2Pr-c CH2CH=C(Cl)2
CH2S(O)CH2Pr-c CH2C≡CH
CH2S(O)CH2Pr-c CH2CN
CH2S(O)CH2Pr-c CH2CF3
CH2S(O)CH2Pr-c CH2OMe
CH2S(O)CH2Pr-c CH2OCF3
CH2S(O)CH2Pr-c CH2SMe
CH2S(O)CH2Pr-c CH2S(O)Me
CH2S(O)CH2Pr-c CH2S(O)2Me
CH2S(O)CH2Pr-c CH2SCF3
CH2S(O)CH2Pr-c CH2S(O)CF3
CH2S(O)CH2Pr-c CH2S(O)2CF3
CH2S(O)CH2Pr-c CH2CH(OMe)2
CH2S(O)CH2Pr-c CH2CH(SMe)2
CH2S(O)CH2Pr-c CH2C(O)Me
CH2S(O)CH2Pr-c CH2C(O)CF3
CH2S(O)CH2Pr-c CH2C(O)OMe
CH2S(O)CH2Pr-c CH2(D1-32a)
CH2S(O)CH2Pr-c CH2(D1-33a)
CH2S(O)CH2Pr-c CH2(D1-34a)
CH2S(O)CH2Pr-c CH2(D1-37a)
CH2S(O)CH2Pr-c CH2(D1-81a)
CH2S(O)CH2Pr-c CH2(D1-82a)
CH2S(O)CH2Pr-c CH2(D1-84a)
CH2S(O)CH2Pr-c CH2(D1-85a)
CH2S(O)CH2Pr-c CH2(D1-87a)
CH2S(O)CH2Pr-c CH2(D1-92a)
CH2S(O)CH2Pr-c CH2(D1-93a)
CH2S(O)CH2Pr-c CH2(D1-95a)
CH2S(O)CH2Pr-c CH2(D1-96a)
CH2S(O)CH2Pr-c CH2(D1-98a)
CH2S(O)CH2Pr-c CH2(D1-108a)
CH2S(O)CH2Pr-c CH2(D1-108b,Z=2-Cl)
CH2S(O)CH2Pr-c CH2(D1-108b,Z=3-Me)
CH2S(O)CH2Pr-c CH2(D1-108b,Z=4-OMe)
CH2S(O)CH2Pr-c CH2(D1-108b,Z=2-SMe)
CH2S(O)CH2Pr-c CH2(D1-108b,Z=3-CF3)
CH2S(O)CH2Pr-c CH2(D1-108b,Z=4-OCF3)
CH2S(O)CH2Pr-c CH2(D1-108b,Z=2-SCF3)
CH2S(O)CH2Pr-c CH2CH2CN
CH2S(O)CH2Pr-c CH2CH2CF3
CH2S(O)CH2Pr-c CH2CH2OMe
CH2S(O)CH2Pr-c CH2CH2SMe
CH2S(O)CH2Pr-c CH2CH2S(O)Me
CH2S(O)CH2Pr-c CH2CH2S(O)2Me
CH2S(O)CH2Pr-c D1-32a
CH2S(O)CH2Pr-c D1-33a
CH2S(O)CH2Pr-c D1-34a
CH2S(O)CH2Pr-c D1-37a
CH2S(O)CH2Pr-c D1-81a
CH2S(O)CH2Pr-c D1-82a
CH2S(O)CH2Pr-c D1-84a
CH2S(O)CH2Pr-c D1-85a
CH2S(O)CH2Pr-c D1-87a
CH2S(O)CH2Pr-c D1-92a
CH2S(O)CH2Pr-c D1-93a
CH2S(O)CH2Pr-c D1-95a
CH2S(O)CH2Pr-c D1-96a
CH2S(O)CH2Pr-c D1-98a
CH2S(O)CH2Pr-c D1-108a
CH2S(O)CH2Pr-c D1-108b(Z=2-Cl)
CH2S(O)CH2Pr-c D1-108b(Z=3-Me)
CH2S(O)CH2Pr-c D1-108b(Z=4-OMe)
CH2S(O)CH2Pr-c D1-108b(Z=2-SMe)
CH2S(O)CH2Pr-c D1-108b(Z=3-CF3)
CH2S(O)CH2Pr-c D1-108b(Z=4-OCF3)
CH2S(O)CH2Pr-c D1-108b(Z=2-SCF3)
CH2S(O)CH2Pr-c C(O)Me
CH2S(O)CH2Pr-c C(O)CF3
CH2S(O)CH2Pr-c C(O)OMe
CH2S(O)2CH2Pr-c Me
CH2S(O)2CH2Pr-c Et
CH2S(O)2CH2Pr-c Pr-n
CH2S(O)2CH2Pr-c Pr-i
CH2S(O)2CH2Pr-c Pr-c
CH2S(O)2CH2Pr-c Bu-n
CH2S(O)2CH2Pr-c Bu-i
CH2S(O)2CH2Pr-c Bu-c
CH2S(O)2CH2Pr-c Bu-s
CH2S(O)2CH2Pr-c Bu-t
CH2S(O)2CH2Pr-c Pen-n
CH2S(O)2CH2Pr-c Pen-c
CH2S(O)2CH2Pr-c Hex-n
CH2S(O)2CH2Pr-c Hex-c
CH2S(O)2CH2Pr-c CH2Pr-c
CH2S(O)2CH2Pr-c CH2Bu-c
CH2S(O)2CH2Pr-c CH2Pen-c
CH2S(O)2CH2Pr-c CH2Hex-c
CH2S(O)2CH2Pr-c CH2CH=CH2
CH2S(O)2CH2Pr-c CH2CH=C(Cl)2
CH2S(O)2CH2Pr-c CH2C≡CH
CH2S(O)2CH2Pr-c CH2CN
CH2S(O)2CH2Pr-c CH2CF3
CH2S(O)2CH2Pr-c CH2OMe
CH2S(O)2CH2Pr-c CH2OCF3
CH2S(O)2CH2Pr-c CH2SMe
CH2S(O)2CH2Pr-c CH2S(O)Me
CH2S(O)2CH2Pr-c CH2S(O)2Me
CH2S(O)2CH2Pr-c CH2SCF3
CH2S(O)2CH2Pr-c CH2S(O)CF3
CH2S(O)2CH2Pr-c CH2S(O)2CF3
CH2S(O)2CH2Pr-c CH2CH(OMe)2
CH2S(O)2CH2Pr-c CH2CH(SMe)2
CH2S(O)2CH2Pr-c CH2C(O)Me
CH2S(O)2CH2Pr-c CH2C(O)CF3
CH2S(O)2CH2Pr-c CH2C(O)OMe
CH2S(O)2CH2Pr-c CH2(D1-32a)
CH2S(O)2CH2Pr-c CH2(D1-33a)
CH2S(O)2CH2Pr-c CH2(D1-34a)
CH2S(O)2CH2Pr-c CH2(D1-37a)
CH2S(O)2CH2Pr-c CH2(D1-81a)
CH2S(O)2CH2Pr-c CH2(D1-82a)
CH2S(O)2CH2Pr-c CH2(D1-84a)
CH2S(O)2CH2Pr-c CH2(D1-85a)
CH2S(O)2CH2Pr-c CH2(D1-87a)
CH2S(O)2CH2Pr-c CH2(D1-92a)
CH2S(O)2CH2Pr-c CH2(D1-93a)
CH2S(O)2CH2Pr-c CH2(D1-95a)
CH2S(O)2CH2Pr-c CH2(D1-96a)
CH2S(O)2CH2Pr-c CH2(D1-98a)
CH2S(O)2CH2Pr-c CH2(D1-108a)
CH2S(O)2CH2Pr-c CH2(D1-108b,Z=2-Cl)
CH2S(O)2CH2Pr-c CH2(D1-108b,Z=3-Me)
CH2S(O)2CH2Pr-c CH2(D1-108b,Z=4-OMe)
CH2S(O)2CH2Pr-c CH2(D1-108b,Z=2-SMe)
CH2S(O)2CH2Pr-c CH2(D1-108b,Z=3-CF3)
CH2S(O)2CH2Pr-c CH2(D1-108b,Z=4-OCF3)
CH2S(O)2CH2Pr-c CH2(D1-108b,Z=2-SCF3)
CH2S(O)2CH2Pr-c CH2CH2CN
CH2S(O)2CH2Pr-c CH2CH2CF3
CH2S(O)2CH2Pr-c CH2CH2OMe
CH2S(O)2CH2Pr-c CH2CH2SMe
CH2S(O)2CH2Pr-c CH2CH2S(O)Me
CH2S(O)2CH2Pr-c CH2CH2S(O)2Me
CH2S(O)2CH2Pr-c D1-32a
CH2S(O)2CH2Pr-c D1-33a
CH2S(O)2CH2Pr-c D1-34a
CH2S(O)2CH2Pr-c D1-37a
CH2S(O)2CH2Pr-c D1-81a
CH2S(O)2CH2Pr-c D1-82a
CH2S(O)2CH2Pr-c D1-84a
CH2S(O)2CH2Pr-c D1-85a
CH2S(O)2CH2Pr-c D1-87a
CH2S(O)2CH2Pr-c D1-92a
CH2S(O)2CH2Pr-c D1-93a
CH2S(O)2CH2Pr-c D1-95a
CH2S(O)2CH2Pr-c D1-96a
CH2S(O)2CH2Pr-c D1-98a
CH2S(O)2CH2Pr-c D1-108a
CH2S(O)2CH2Pr-c D1-108b(Z=2-Cl)
CH2S(O)2CH2Pr-c D1-108b(Z=3-Me)
CH2S(O)2CH2Pr-c D1-108b(Z=4-OMe)
CH2S(O)2CH2Pr-c D1-108b(Z=2-SMe)
CH2S(O)2CH2Pr-c D1-108b(Z=3-CF3)
CH2S(O)2CH2Pr-c D1-108b(Z=4-OCF3)
CH2S(O)2CH2Pr-c D1-108b(Z=2-SCF3)
CH2S(O)2CH2Pr-c C(O)Me
CH2S(O)2CH2Pr-c C(O)CF3
CH2S(O)2CH2Pr-c C(O)OMe
CH(Me)SCH2Pr-c Me
CH(Me)SCH2Pr-c Et
CH(Me)SCH2Pr-c Pr-n
CH(Me)SCH2Pr-c Pr-i
CH(Me)SCH2Pr-c Pr-c
CH(Me)SCH2Pr-c Bu-n
CH(Me)SCH2Pr-c Bu-i
CH(Me)SCH2Pr-c Bu-c
CH(Me)SCH2Pr-c Bu-s
CH(Me)SCH2Pr-c Bu-t
CH(Me)SCH2Pr-c Pen-n
CH(Me)SCH2Pr-c Pen-c
CH(Me)SCH2Pr-c Hex-n
CH(Me)SCH2Pr-c Hex-c
CH(Me)SCH2Pr-c CH2Pr-c
CH(Me)SCH2Pr-c CH2Bu-c
CH(Me)SCH2Pr-c CH2Pen-c
CH(Me)SCH2Pr-c CH2Hex-c
CH(Me)SCH2Pr-c CH2CH=CH2
CH(Me)SCH2Pr-c CH2CH=C(Cl)2
CH(Me)SCH2Pr-c CH2C≡CH
CH(Me)SCH2Pr-c CH2CN
CH(Me)SCH2Pr-c CH2CF3
CH(Me)SCH2Pr-c CH2OMe
CH(Me)SCH2Pr-c CH2OCF3
CH(Me)SCH2Pr-c CH2SMe
CH(Me)SCH2Pr-c CH2S(O)Me
CH(Me)SCH2Pr-c CH2S(O)2Me
CH(Me)SCH2Pr-c CH2SCF3
CH(Me)SCH2Pr-c CH2S(O)CF3
CH(Me)SCH2Pr-c CH2S(O)2CF3
CH(Me)SCH2Pr-c CH2CH(OMe)2
CH(Me)SCH2Pr-c CH2CH(SMe)2
CH(Me)SCH2Pr-c CH2C(O)Me
CH(Me)SCH2Pr-c CH2C(O)CF3
CH(Me)SCH2Pr-c CH2C(O)OMe
CH(Me)SCH2Pr-c CH2(D1-32a)
CH(Me)SCH2Pr-c CH2(D1-33a)
CH(Me)SCH2Pr-c CH2(D1-34a)
CH(Me)SCH2Pr-c CH2(D1-37a)
CH(Me)SCH2Pr-c CH2(D1-81a)
CH(Me)SCH2Pr-c CH2(D1-82a)
CH(Me)SCH2Pr-c CH2(D1-84a)
CH(Me)SCH2Pr-c CH2(D1-85a)
CH(Me)SCH2Pr-c CH2(D1-87a)
CH(Me)SCH2Pr-c CH2(D1-92a)
CH(Me)SCH2Pr-c CH2(D1-93a)
CH(Me)SCH2Pr-c CH2(D1-95a)
CH(Me)SCH2Pr-c CH2(D1-96a)
CH(Me)SCH2Pr-c CH2(D1-98a)
CH(Me)SCH2Pr-c CH2(D1-108a)
CH(Me)SCH2Pr-c CH2(D1-108b,Z=2-Cl)
CH(Me)SCH2Pr-c CH2(D1-108b,Z=3-Me)
CH(Me)SCH2Pr-c CH2(D1-108b,Z=4-OMe)
CH(Me)SCH2Pr-c CH2(D1-108b,Z=2-SMe)
CH(Me)SCH2Pr-c CH2(D1-108b,Z=3-CF3)
CH(Me)SCH2Pr-c CH2(D1-108b,Z=4-OCF3)
CH(Me)SCH2Pr-c CH2(D1-108b,Z=2-SCF3)
CH(Me)SCH2Pr-c CH2CH2CN
CH(Me)SCH2Pr-c CH2CH2CF3
CH(Me)SCH2Pr-c CH2CH2OMe
CH(Me)SCH2Pr-c CH2CH2SMe
CH(Me)SCH2Pr-c CH2CH2S(O)Me
CH(Me)SCH2Pr-c CH2CH2S(O)2Me
CH(Me)SCH2Pr-c D1-32a
CH(Me)SCH2Pr-c D1-33a
CH(Me)SCH2Pr-c D1-34a
CH(Me)SCH2Pr-c D1-37a
CH(Me)SCH2Pr-c D1-81a
CH(Me)SCH2Pr-c D1-82a
CH(Me)SCH2Pr-c D1-84a
CH(Me)SCH2Pr-c D1-85a
CH(Me)SCH2Pr-c D1-87a
CH(Me)SCH2Pr-c D1-92a
CH(Me)SCH2Pr-c D1-93a
CH(Me)SCH2Pr-c D1-95a
CH(Me)SCH2Pr-c D1-96a
CH(Me)SCH2Pr-c D1-98a
CH(Me)SCH2Pr-c D1-108a
CH(Me)SCH2Pr-c D1-108b(Z=2-Cl)
CH(Me)SCH2Pr-c D1-108b(Z=3-Me)
CH(Me)SCH2Pr-c D1-108b(Z=4-OMe)
CH(Me)SCH2Pr-c D1-108b(Z=2-SMe)
CH(Me)SCH2Pr-c D1-108b(Z=3-CF3)
CH(Me)SCH2Pr-c D1-108b(Z=4-OCF3)
CH(Me)SCH2Pr-c D1-108b(Z=2-SCF3)
CH(Me)SCH2Pr-c C(O)Me
CH(Me)SCH2Pr-c C(O)CF3
CH(Me)SCH2Pr-c C(O)OMe
CH(Me)S(O)CH2Pr-c Me
CH(Me)S(O)CH2Pr-c Et
CH(Me)S(O)CH2Pr-c Pr-n
CH(Me)S(O)CH2Pr-c Pr-i
CH(Me)S(O)CH2Pr-c Pr-c
CH(Me)S(O)CH2Pr-c Bu-n
CH(Me)S(O)CH2Pr-c Bu-i
CH(Me)S(O)CH2Pr-c Bu-c
CH(Me)S(O)CH2Pr-c Bu-s
CH(Me)S(O)CH2Pr-c Bu-t
CH(Me)S(O)CH2Pr-c Pen-n
CH(Me)S(O)CH2Pr-c Pen-c
CH(Me)S(O)CH2Pr-c Hex-n
CH(Me)S(O)CH2Pr-c Hex-c
CH(Me)S(O)CH2Pr-c CH2Pr-c
CH(Me)S(O)CH2Pr-c CH2Bu-c
CH(Me)S(O)CH2Pr-c CH2Pen-c
CH(Me)S(O)CH2Pr-c CH2Hex-c
CH(Me)S(O)CH2Pr-c CH2CH=CH2
CH(Me)S(O)CH2Pr-c CH2CH=C(Cl)2
CH(Me)S(O)CH2Pr-c CH2C≡CH
CH(Me)S(O)CH2Pr-c CH2CN
CH(Me)S(O)CH2Pr-c CH2CF3
CH(Me)S(O)CH2Pr-c CH2OMe
CH(Me)S(O)CH2Pr-c CH2OCF3
CH(Me)S(O)CH2Pr-c CH2SMe
CH(Me)S(O)CH2Pr-c CH2S(O)Me
CH(Me)S(O)CH2Pr-c CH2S(O)2Me
CH(Me)S(O)CH2Pr-c CH2SCF3
CH(Me)S(O)CH2Pr-c CH2S(O)CF3
CH(Me)S(O)CH2Pr-c CH2S(O)2CF3
CH(Me)S(O)CH2Pr-c CH2CH(OMe)2
CH(Me)S(O)CH2Pr-c CH2CH(SMe)2
CH(Me)S(O)CH2Pr-c CH2C(O)Me
CH(Me)S(O)CH2Pr-c CH2C(O)CF3
CH(Me)S(O)CH2Pr-c CH2C(O)OMe
CH(Me)S(O)CH2Pr-c CH2(D1-32a)
CH(Me)S(O)CH2Pr-c CH2(D1-33a)
CH(Me)S(O)CH2Pr-c CH2(D1-34a)
CH(Me)S(O)CH2Pr-c CH2(D1-37a)
CH(Me)S(O)CH2Pr-c CH2(D1-81a)
CH(Me)S(O)CH2Pr-c CH2(D1-82a)
CH(Me)S(O)CH2Pr-c CH2(D1-84a)
CH(Me)S(O)CH2Pr-c CH2(D1-85a)
CH(Me)S(O)CH2Pr-c CH2(D1-87a)
CH(Me)S(O)CH2Pr-c CH2(D1-92a)
CH(Me)S(O)CH2Pr-c CH2(D1-93a)
CH(Me)S(O)CH2Pr-c CH2(D1-95a)
CH(Me)S(O)CH2Pr-c CH2(D1-96a)
CH(Me)S(O)CH2Pr-c CH2(D1-98a)
CH(Me)S(O)CH2Pr-c CH2(D1-108a)
CH(Me)S(O)CH2Pr-c CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)CH2Pr-c CH2(D1-108b,Z=3-Me)
CH(Me)S(O)CH2Pr-c CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)CH2Pr-c CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)CH2Pr-c CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)CH2Pr-c CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)CH2Pr-c CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)CH2Pr-c CH2CH2CN
CH(Me)S(O)CH2Pr-c CH2CH2CF3
CH(Me)S(O)CH2Pr-c CH2CH2OMe
CH(Me)S(O)CH2Pr-c CH2CH2SMe
CH(Me)S(O)CH2Pr-c CH2CH2S(O)Me
CH(Me)S(O)CH2Pr-c CH2CH2S(O)2Me
CH(Me)S(O)CH2Pr-c D1-32a
CH(Me)S(O)CH2Pr-c D1-33a
CH(Me)S(O)CH2Pr-c D1-34a
CH(Me)S(O)CH2Pr-c D1-37a
CH(Me)S(O)CH2Pr-c D1-81a
CH(Me)S(O)CH2Pr-c D1-82a
CH(Me)S(O)CH2Pr-c D1-84a
CH(Me)S(O)CH2Pr-c D1-85a
CH(Me)S(O)CH2Pr-c D1-87a
CH(Me)S(O)CH2Pr-c D1-92a
CH(Me)S(O)CH2Pr-c D1-93a
CH(Me)S(O)CH2Pr-c D1-95a
CH(Me)S(O)CH2Pr-c D1-96a
CH(Me)S(O)CH2Pr-c D1-98a
CH(Me)S(O)CH2Pr-c D1-108a
CH(Me)S(O)CH2Pr-c D1-108b(Z=2-Cl)
CH(Me)S(O)CH2Pr-c D1-108b(Z=3-Me)
CH(Me)S(O)CH2Pr-c D1-108b(Z=4-OMe)
CH(Me)S(O)CH2Pr-c D1-108b(Z=2-SMe)
CH(Me)S(O)CH2Pr-c D1-108b(Z=3-CF3)
CH(Me)S(O)CH2Pr-c D1-108b(Z=4-OCF3)
CH(Me)S(O)CH2Pr-c D1-108b(Z=2-SCF3)
CH(Me)S(O)CH2Pr-c C(O)Me
CH(Me)S(O)CH2Pr-c C(O)CF3
CH(Me)S(O)CH2Pr-c C(O)OMe
CH(Me)S(O)2CH2Pr-c Me
CH(Me)S(O)2CH2Pr-c Et
CH(Me)S(O)2CH2Pr-c Pr-n
CH(Me)S(O)2CH2Pr-c Pr-i
CH(Me)S(O)2CH2Pr-c Pr-c
CH(Me)S(O)2CH2Pr-c Bu-n
CH(Me)S(O)2CH2Pr-c Bu-i
CH(Me)S(O)2CH2Pr-c Bu-c
CH(Me)S(O)2CH2Pr-c Bu-s
CH(Me)S(O)2CH2Pr-c Bu-t
CH(Me)S(O)2CH2Pr-c Pen-n
CH(Me)S(O)2CH2Pr-c Pen-c
CH(Me)S(O)2CH2Pr-c Hex-n
CH(Me)S(O)2CH2Pr-c Hex-c
CH(Me)S(O)2CH2Pr-c CH2Pr-c
CH(Me)S(O)2CH2Pr-c CH2Bu-c
CH(Me)S(O)2CH2Pr-c CH2Pen-c
CH(Me)S(O)2CH2Pr-c CH2Hex-c
CH(Me)S(O)2CH2Pr-c CH2CH=CH2
CH(Me)S(O)2CH2Pr-c CH2CH=C(Cl)2
CH(Me)S(O)2CH2Pr-c CH2C≡CH
CH(Me)S(O)2CH2Pr-c CH2CN
CH(Me)S(O)2CH2Pr-c CH2CF3
CH(Me)S(O)2CH2Pr-c CH2OMe
CH(Me)S(O)2CH2Pr-c CH2OCF3
CH(Me)S(O)2CH2Pr-c CH2SMe
CH(Me)S(O)2CH2Pr-c CH2S(O)Me
CH(Me)S(O)2CH2Pr-c CH2S(O)2Me
CH(Me)S(O)2CH2Pr-c CH2SCF3
CH(Me)S(O)2CH2Pr-c CH2S(O)CF3
CH(Me)S(O)2CH2Pr-c CH2S(O)2CF3
CH(Me)S(O)2CH2Pr-c CH2CH(OMe)2
CH(Me)S(O)2CH2Pr-c CH2CH(SMe)2
CH(Me)S(O)2CH2Pr-c CH2C(O)Me
CH(Me)S(O)2CH2Pr-c CH2C(O)CF3
CH(Me)S(O)2CH2Pr-c CH2C(O)OMe
CH(Me)S(O)2CH2Pr-c CH2(D1-32a)
CH(Me)S(O)2CH2Pr-c CH2(D1-33a)
CH(Me)S(O)2CH2Pr-c CH2(D1-34a)
CH(Me)S(O)2CH2Pr-c CH2(D1-37a)
CH(Me)S(O)2CH2Pr-c CH2(D1-81a)
CH(Me)S(O)2CH2Pr-c CH2(D1-82a)
CH(Me)S(O)2CH2Pr-c CH2(D1-84a)
CH(Me)S(O)2CH2Pr-c CH2(D1-85a)
CH(Me)S(O)2CH2Pr-c CH2(D1-87a)
CH(Me)S(O)2CH2Pr-c CH2(D1-92a)
CH(Me)S(O)2CH2Pr-c CH2(D1-93a)
CH(Me)S(O)2CH2Pr-c CH2(D1-95a)
CH(Me)S(O)2CH2Pr-c CH2(D1-96a)
CH(Me)S(O)2CH2Pr-c CH2(D1-98a)
CH(Me)S(O)2CH2Pr-c CH2(D1-108a)
CH(Me)S(O)2CH2Pr-c CH2(D1-108b,Z=2-Cl)
CH(Me)S(O)2CH2Pr-c CH2(D1-108b,Z=3-Me)
CH(Me)S(O)2CH2Pr-c CH2(D1-108b,Z=4-OMe)
CH(Me)S(O)2CH2Pr-c CH2(D1-108b,Z=2-SMe)
CH(Me)S(O)2CH2Pr-c CH2(D1-108b,Z=3-CF3)
CH(Me)S(O)2CH2Pr-c CH2(D1-108b,Z=4-OCF3)
CH(Me)S(O)2CH2Pr-c CH2(D1-108b,Z=2-SCF3)
CH(Me)S(O)2CH2Pr-c CH2CH2CN
CH(Me)S(O)2CH2Pr-c CH2CH2CF3
CH(Me)S(O)2CH2Pr-c CH2CH2OMe
CH(Me)S(O)2CH2Pr-c CH2CH2SMe
CH(Me)S(O)2CH2Pr-c CH2CH2S(O)Me
CH(Me)S(O)2CH2Pr-c CH2CH2S(O)2Me
CH(Me)S(O)2CH2Pr-c D1-32a
CH(Me)S(O)2CH2Pr-c D1-33a
CH(Me)S(O)2CH2Pr-c D1-34a
CH(Me)S(O)2CH2Pr-c D1-37a
CH(Me)S(O)2CH2Pr-c D1-81a
CH(Me)S(O)2CH2Pr-c D1-82a
CH(Me)S(O)2CH2Pr-c D1-84a
CH(Me)S(O)2CH2Pr-c D1-85a
CH(Me)S(O)2CH2Pr-c D1-87a
CH(Me)S(O)2CH2Pr-c D1-92a
CH(Me)S(O)2CH2Pr-c D1-93a
CH(Me)S(O)2CH2Pr-c D1-95a
CH(Me)S(O)2CH2Pr-c D1-96a
CH(Me)S(O)2CH2Pr-c D1-98a
CH(Me)S(O)2CH2Pr-c D1-108a
CH(Me)S(O)2CH2Pr-c D1-108b(Z=2-Cl)
CH(Me)S(O)2CH2Pr-c D1-108b(Z=3-Me)
CH(Me)S(O)2CH2Pr-c D1-108b(Z=4-OMe)
CH(Me)S(O)2CH2Pr-c D1-108b(Z=2-SMe)
CH(Me)S(O)2CH2Pr-c D1-108b(Z=3-CF3)
CH(Me)S(O)2CH2Pr-c D1-108b(Z=4-OCF3)
CH(Me)S(O)2CH2Pr-c D1-108b(Z=2-SCF3)
CH(Me)S(O)2CH2Pr-c C(O)Me
CH(Me)S(O)2CH2Pr-c C(O)CF3
CH(Me)S(O)2CH2Pr-c C(O)OMe
CH(Et)SCH2Pr-c Me
CH(Et)SCH2Pr-c Et
CH(Et)SCH2Pr-c Pr-n
CH(Et)SCH2Pr-c Pr-i
CH(Et)SCH2Pr-c Pr-c
CH(Et)SCH2Pr-c Bu-n
CH(Et)SCH2Pr-c Bu-i
CH(Et)SCH2Pr-c Bu-c
CH(Et)SCH2Pr-c Bu-s
CH(Et)SCH2Pr-c Bu-t
CH(Et)SCH2Pr-c Pen-n
CH(Et)SCH2Pr-c Pen-c
CH(Et)SCH2Pr-c Hex-n
CH(Et)SCH2Pr-c Hex-c
CH(Et)SCH2Pr-c CH2Pr-c
CH(Et)SCH2Pr-c CH2Bu-c
CH(Et)SCH2Pr-c CH2Pen-c
CH(Et)SCH2Pr-c CH2Hex-c
CH(Et)SCH2Pr-c CH2CH=CH2
CH(Et)SCH2Pr-c CH2CH=C(Cl)2
CH(Et)SCH2Pr-c CH2C≡CH
CH(Et)SCH2Pr-c CH2CN
CH(Et)SCH2Pr-c CH2CF3
CH(Et)SCH2Pr-c CH2OMe
CH(Et)SCH2Pr-c CH2OCF3
CH(Et)SCH2Pr-c CH2SMe
CH(Et)SCH2Pr-c CH2S(O)Me
CH(Et)SCH2Pr-c CH2S(O)2Me
CH(Et)SCH2Pr-c CH2SCF3
CH(Et)SCH2Pr-c CH2S(O)CF3
CH(Et)SCH2Pr-c CH2S(O)2CF3
CH(Et)SCH2Pr-c CH2CH(OMe)2
CH(Et)SCH2Pr-c CH2CH(SMe)2
CH(Et)SCH2Pr-c CH2C(O)Me
CH(Et)SCH2Pr-c CH2C(O)CF3
CH(Et)SCH2Pr-c CH2C(O)OMe
CH(Et)SCH2Pr-c CH2(D1-32a)
CH(Et)SCH2Pr-c CH2(D1-33a)
CH(Et)SCH2Pr-c CH2(D1-34a)
CH(Et)SCH2Pr-c CH2(D1-37a)
CH(Et)SCH2Pr-c CH2(D1-81a)
CH(Et)SCH2Pr-c CH2(D1-82a)
CH(Et)SCH2Pr-c CH2(D1-84a)
CH(Et)SCH2Pr-c CH2(D1-85a)
CH(Et)SCH2Pr-c CH2(D1-87a)
CH(Et)SCH2Pr-c CH2(D1-92a)
CH(Et)SCH2Pr-c CH2(D1-93a)
CH(Et)SCH2Pr-c CH2(D1-95a)
CH(Et)SCH2Pr-c CH2(D1-96a)
CH(Et)SCH2Pr-c CH2(D1-98a)
CH(Et)SCH2Pr-c CH2(D1-108a)
CH(Et)SCH2Pr-c CH2(D1-108b,Z=2-Cl)
CH(Et)SCH2Pr-c CH2(D1-108b,Z=3-Me)
CH(Et)SCH2Pr-c CH2(D1-108b,Z=4-OMe)
CH(Et)SCH2Pr-c CH2(D1-108b,Z=2-SMe)
CH(Et)SCH2Pr-c CH2(D1-108b,Z=3-CF3)
CH(Et)SCH2Pr-c CH2(D1-108b,Z=4-OCF3)
CH(Et)SCH2Pr-c CH2(D1-108b,Z=2-SCF3)
CH(Et)SCH2Pr-c CH2CH2CN
CH(Et)SCH2Pr-c CH2CH2CF3
CH(Et)SCH2Pr-c CH2CH2OMe
CH(Et)SCH2Pr-c CH2CH2SMe
CH(Et)SCH2Pr-c CH2CH2S(O)Me
CH(Et)SCH2Pr-c CH2CH2S(O)2Me
CH(Et)SCH2Pr-c D1-32a
CH(Et)SCH2Pr-c D1-33a
CH(Et)SCH2Pr-c D1-34a
CH(Et)SCH2Pr-c D1-37a
CH(Et)SCH2Pr-c D1-81a
CH(Et)SCH2Pr-c D1-82a
CH(Et)SCH2Pr-c D1-84a
CH(Et)SCH2Pr-c D1-85a
CH(Et)SCH2Pr-c D1-87a
CH(Et)SCH2Pr-c D1-92a
CH(Et)SCH2Pr-c D1-93a
CH(Et)SCH2Pr-c D1-95a
CH(Et)SCH2Pr-c D1-96a
CH(Et)SCH2Pr-c D1-98a
CH(Et)SCH2Pr-c D1-108a
CH(Et)SCH2Pr-c D1-108b(Z=2-Cl)
CH(Et)SCH2Pr-c D1-108b(Z=3-Me)
CH(Et)SCH2Pr-c D1-108b(Z=4-OMe)
CH(Et)SCH2Pr-c D1-108b(Z=2-SMe)
CH(Et)SCH2Pr-c D1-108b(Z=3-CF3)
CH(Et)SCH2Pr-c D1-108b(Z=4-OCF3)
CH(Et)SCH2Pr-c D1-108b(Z=2-SCF3)
CH(Et)SCH2Pr-c C(O)Me
CH(Et)SCH2Pr-c C(O)CF3
CH(Et)SCH2Pr-c C(O)OMe
CH(Et)S(O)CH2Pr-c Me
CH(Et)S(O)CH2Pr-c Et
CH(Et)S(O)CH2Pr-c Pr-n
CH(Et)S(O)CH2Pr-c Pr-i
CH(Et)S(O)CH2Pr-c Pr-c
CH(Et)S(O)CH2Pr-c Bu-n
CH(Et)S(O)CH2Pr-c Bu-i
CH(Et)S(O)CH2Pr-c Bu-c
CH(Et)S(O)CH2Pr-c Bu-s
CH(Et)S(O)CH2Pr-c Bu-t
CH(Et)S(O)CH2Pr-c Pen-n
CH(Et)S(O)CH2Pr-c Pen-c
CH(Et)S(O)CH2Pr-c Hex-n
CH(Et)S(O)CH2Pr-c Hex-c
CH(Et)S(O)CH2Pr-c CH2Pr-c
CH(Et)S(O)CH2Pr-c CH2Bu-c
CH(Et)S(O)CH2Pr-c CH2Pen-c
CH(Et)S(O)CH2Pr-c CH2Hex-c
CH(Et)S(O)CH2Pr-c CH2CH=CH2
CH(Et)S(O)CH2Pr-c CH2CH=C(Cl)2
CH(Et)S(O)CH2Pr-c CH2C≡CH
CH(Et)S(O)CH2Pr-c CH2CN
CH(Et)S(O)CH2Pr-c CH2CF3
CH(Et)S(O)CH2Pr-c CH2OMe
CH(Et)S(O)CH2Pr-c CH2OCF3
CH(Et)S(O)CH2Pr-c CH2SMe
CH(Et)S(O)CH2Pr-c CH2S(O)Me
CH(Et)S(O)CH2Pr-c CH2S(O)2Me
CH(Et)S(O)CH2Pr-c CH2SCF3
CH(Et)S(O)CH2Pr-c CH2S(O)CF3
CH(Et)S(O)CH2Pr-c CH2S(O)2CF3
CH(Et)S(O)CH2Pr-c CH2CH(OMe)2
CH(Et)S(O)CH2Pr-c CH2CH(SMe)2
CH(Et)S(O)CH2Pr-c CH2C(O)Me
CH(Et)S(O)CH2Pr-c CH2C(O)CF3
CH(Et)S(O)CH2Pr-c CH2C(O)OMe
CH(Et)S(O)CH2Pr-c CH2(D1-32a)
CH(Et)S(O)CH2Pr-c CH2(D1-33a)
CH(Et)S(O)CH2Pr-c CH2(D1-34a)
CH(Et)S(O)CH2Pr-c CH2(D1-37a)
CH(Et)S(O)CH2Pr-c CH2(D1-81a)
CH(Et)S(O)CH2Pr-c CH2(D1-82a)
CH(Et)S(O)CH2Pr-c CH2(D1-84a)
CH(Et)S(O)CH2Pr-c CH2(D1-85a)
CH(Et)S(O)CH2Pr-c CH2(D1-87a)
CH(Et)S(O)CH2Pr-c CH2(D1-92a)
CH(Et)S(O)CH2Pr-c CH2(D1-93a)
CH(Et)S(O)CH2Pr-c CH2(D1-95a)
CH(Et)S(O)CH2Pr-c CH2(D1-96a)
CH(Et)S(O)CH2Pr-c CH2(D1-98a)
CH(Et)S(O)CH2Pr-c CH2(D1-108a)
CH(Et)S(O)CH2Pr-c CH2(D1-108b,Z=2-Cl)
CH(Et)S(O)CH2Pr-c CH2(D1-108b,Z=3-Me)
CH(Et)S(O)CH2Pr-c CH2(D1-108b,Z=4-OMe)
CH(Et)S(O)CH2Pr-c CH2(D1-108b,Z=2-SMe)
CH(Et)S(O)CH2Pr-c CH2(D1-108b,Z=3-CF3)
CH(Et)S(O)CH2Pr-c CH2(D1-108b,Z=4-OCF3)
CH(Et)S(O)CH2Pr-c CH2(D1-108b,Z=2-SCF3)
CH(Et)S(O)CH2Pr-c CH2CH2CN
CH(Et)S(O)CH2Pr-c CH2CH2CF3
CH(Et)S(O)CH2Pr-c CH2CH2OMe
CH(Et)S(O)CH2Pr-c CH2CH2SMe
CH(Et)S(O)CH2Pr-c CH2CH2S(O)Me
CH(Et)S(O)CH2Pr-c CH2CH2S(O)2Me
CH(Et)S(O)CH2Pr-c D1-32a
CH(Et)S(O)CH2Pr-c D1-33a
CH(Et)S(O)CH2Pr-c D1-34a
CH(Et)S(O)CH2Pr-c D1-37a
CH(Et)S(O)CH2Pr-c D1-81a
CH(Et)S(O)CH2Pr-c D1-82a
CH(Et)S(O)CH2Pr-c D1-84a
CH(Et)S(O)CH2Pr-c D1-85a
CH(Et)S(O)CH2Pr-c D1-87a
CH(Et)S(O)CH2Pr-c D1-92a
CH(Et)S(O)CH2Pr-c D1-93a
CH(Et)S(O)CH2Pr-c D1-95a
CH(Et)S(O)CH2Pr-c D1-96a
CH(Et)S(O)CH2Pr-c D1-98a
CH(Et)S(O)CH2Pr-c D1-108a
CH(Et)S(O)CH2Pr-c D1-108b(Z=2-Cl)
CH(Et)S(O)CH2Pr-c D1-108b(Z=3-Me)
CH(Et)S(O)CH2Pr-c D1-108b(Z=4-OMe)
CH(Et)S(O)CH2Pr-c D1-108b(Z=2-SMe)
CH(Et)S(O)CH2Pr-c D1-108b(Z=3-CF3)
CH(Et)S(O)CH2Pr-c D1-108b(Z=4-OCF3)
CH(Et)S(O)CH2Pr-c D1-108b(Z=2-SCF3)
CH(Et)S(O)CH2Pr-c C(O)Me
CH(Et)S(O)CH2Pr-c C(O)CF3
CH(Et)S(O)CH2Pr-c C(O)OMe
CH(Et)S(O)2CH2Pr-c Me
CH(Et)S(O)2CH2Pr-c Et
CH(Et)S(O)2CH2Pr-c Pr-n
CH(Et)S(O)2CH2Pr-c Pr-i
CH(Et)S(O)2CH2Pr-c Pr-c
CH(Et)S(O)2CH2Pr-c Bu-n
CH(Et)S(O)2CH2Pr-c Bu-i
CH(Et)S(O)2CH2Pr-c Bu-c
CH(Et)S(O)2CH2Pr-c Bu-s
CH(Et)S(O)2CH2Pr-c Bu-t
CH(Et)S(O)2CH2Pr-c Pen-n
CH(Et)S(O)2CH2Pr-c Pen-c
CH(Et)S(O)2CH2Pr-c Hex-n
CH(Et)S(O)2CH2Pr-c Hex-c
CH(Et)S(O)2CH2Pr-c CH2Pr-c
CH(Et)S(O)2CH2Pr-c CH2Bu-c
CH(Et)S(O)2CH2Pr-c CH2Pen-c
CH(Et)S(O)2CH2Pr-c CH2Hex-c
CH(Et)S(O)2CH2Pr-c CH2CH=CH2
CH(Et)S(O)2CH2Pr-c CH2CH=C(Cl)2
CH(Et)S(O)2CH2Pr-c CH2C≡CH
CH(Et)S(O)2CH2Pr-c CH2CN
CH(Et)S(O)2CH2Pr-c CH2CF3
CH(Et)S(O)2CH2Pr-c CH2OMe
CH(Et)S(O)2CH2Pr-c CH2OCF3
CH(Et)S(O)2CH2Pr-c CH2SMe
CH(Et)S(O)2CH2Pr-c CH2S(O)Me
CH(Et)S(O)2CH2Pr-c CH2S(O)2Me
CH(Et)S(O)2CH2Pr-c CH2SCF3
CH(Et)S(O)2CH2Pr-c CH2S(O)CF3
CH(Et)S(O)2CH2Pr-c CH2S(O)2CF3
CH(Et)S(O)2CH2Pr-c CH2CH(OMe)2
CH(Et)S(O)2CH2Pr-c CH2CH(SMe)2
CH(Et)S(O)2CH2Pr-c CH2C(O)Me
CH(Et)S(O)2CH2Pr-c CH2C(O)CF3
CH(Et)S(O)2CH2Pr-c CH2C(O)OMe
CH(Et)S(O)2CH2Pr-c CH2(D1-32a)
CH(Et)S(O)2CH2Pr-c CH2(D1-33a)
CH(Et)S(O)2CH2Pr-c CH2(D1-34a)
CH(Et)S(O)2CH2Pr-c CH2(D1-37a)
CH(Et)S(O)2CH2Pr-c CH2(D1-81a)
CH(Et)S(O)2CH2Pr-c CH2(D1-82a)
CH(Et)S(O)2CH2Pr-c CH2(D1-84a)
CH(Et)S(O)2CH2Pr-c CH2(D1-85a)
CH(Et)S(O)2CH2Pr-c CH2(D1-87a)
CH(Et)S(O)2CH2Pr-c CH2(D1-92a)
CH(Et)S(O)2CH2Pr-c CH2(D1-93a)
CH(Et)S(O)2CH2Pr-c CH2(D1-95a)
CH(Et)S(O)2CH2Pr-c CH2(D1-96a)
CH(Et)S(O)2CH2Pr-c CH2(D1-98a)
CH(Et)S(O)2CH2Pr-c CH2(D1-108a)
CH(Et)S(O)2CH2Pr-c CH2(D1-108b,Z=2-Cl)
CH(Et)S(O)2CH2Pr-c CH2(D1-108b,Z=3-Me)
CH(Et)S(O)2CH2Pr-c CH2(D1-108b,Z=4-OMe)
CH(Et)S(O)2CH2Pr-c CH2(D1-108b,Z=2-SMe)
CH(Et)S(O)2CH2Pr-c CH2(D1-108b,Z=3-CF3)
CH(Et)S(O)2CH2Pr-c CH2(D1-108b,Z=4-OCF3)
CH(Et)S(O)2CH2Pr-c CH2(D1-108b,Z=2-SCF3)
CH(Et)S(O)2CH2Pr-c CH2CH2CN
CH(Et)S(O)2CH2Pr-c CH2CH2CF3
CH(Et)S(O)2CH2Pr-c CH2CH2OMe
CH(Et)S(O)2CH2Pr-c CH2CH2SMe
CH(Et)S(O)2CH2Pr-c CH2CH2S(O)Me
CH(Et)S(O)2CH2Pr-c CH2CH2S(O)2Me
CH(Et)S(O)2CH2Pr-c D1-32a
CH(Et)S(O)2CH2Pr-c D1-33a
CH(Et)S(O)2CH2Pr-c D1-34a
CH(Et)S(O)2CH2Pr-c D1-37a
CH(Et)S(O)2CH2Pr-c D1-81a
CH(Et)S(O)2CH2Pr-c D1-82a
CH(Et)S(O)2CH2Pr-c D1-84a
CH(Et)S(O)2CH2Pr-c D1-85a
CH(Et)S(O)2CH2Pr-c D1-87a
CH(Et)S(O)2CH2Pr-c D1-92a
CH(Et)S(O)2CH2Pr-c D1-93a
CH(Et)S(O)2CH2Pr-c D1-95a
CH(Et)S(O)2CH2Pr-c D1-96a
CH(Et)S(O)2CH2Pr-c D1-98a
CH(Et)S(O)2CH2Pr-c D1-108a
CH(Et)S(O)2CH2Pr-c D1-108b(Z=2-Cl)
CH(Et)S(O)2CH2Pr-c D1-108b(Z=3-Me)
CH(Et)S(O)2CH2Pr-c D1-108b(Z=4-OMe)
CH(Et)S(O)2CH2Pr-c D1-108b(Z=2-SMe)
CH(Et)S(O)2CH2Pr-c D1-108b(Z=3-CF3)
CH(Et)S(O)2CH2Pr-c D1-108b(Z=4-OCF3)
CH(Et)S(O)2CH2Pr-c D1-108b(Z=2-SCF3)
CH(Et)S(O)2CH2Pr-c C(O)Me
CH(Et)S(O)2CH2Pr-c C(O)CF3
CH(Et)S(O)2CH2Pr-c C(O)OMe
CH2SCH2C(O)OMe Me
CH2SCH2C(O)OEt Me
CH2SCH2C(O)OPr-n Me
CH2SCH2C(O)OPr-i Me
CH2SCH2C(O)OBu-n Me
CH2SCH2C(O)OBu-i Me
CH2SCH2C(O)OBu-t Me
CH2SCH2C(O)OPen-n Me
CH2SCH2C(O)OHex-n Me
CH2SCH2C(O)OMe Et
CH2SCH2C(O)OMe Pr-n
CH2SCH2C(O)OMe Pr-i
CH2SCH2C(O)OMe Pr-c
CH2SCH2C(O)OMe Bu-n
CH2SCH2C(O)OMe Bu-i
CH2SCH2C(O)OMe Bu-c
CH2SCH2C(O)OMe Bu-s
CH2SCH2C(O)OMe Bu-t
CH2SCH2C(O)OMe Pen-n
CH2SCH2C(O)OMe Pen-c
CH2SCH2C(O)OMe Hex-n
CH2SCH2C(O)OMe Hex-c
CH2SCH2C(O)OMe CH2Pr-c
CH2SCH2C(O)OMe CH2Bu-c
CH2SCH2C(O)OMe CH2Pen-c
CH2SCH2C(O)OMe CH2Hex-c
CH2SCH2C(O)OMe CH2CH=CH2
CH2SCH2C(O)OMe CH2CH=C(Cl)2
CH2SCH2C(O)OMe CH2C≡CH
CH2SCH2C(O)OMe CH2CN
CH2SCH2C(O)OMe CH2CF3
CH2SCH2C(O)OMe CH2OMe
CH2SCH2C(O)OMe CH2OCF3
CH2SCH2C(O)OMe CH2SMe
CH2SCH2C(O)OMe CH2S(O)Me
CH2SCH2C(O)OMe CH2S(O)2Me
CH2SCH2C(O)OMe CH2SCF3
CH2SCH2C(O)OMe CH2S(O)CF3
CH2SCH2C(O)OMe CH2S(O)2CF3
CH2SCH2C(O)OMe CH2CH(OMe)2
CH2SCH2C(O)OMe CH2CH(SMe)2
CH2SCH2C(O)OMe CH2C(O)Me
CH2SCH2C(O)OMe CH2C(O)CF3
CH2SCH2C(O)OMe CH2C(O)OMe
CH2S(O)CH2C(O)OMe Me
CH2S(O)CH2C(O)OEt Me
CH2S(O)CH2C(O)OPr-n Me
CH2S(O)CH2C(O)OPr-i Me
CH2S(O)CH2C(O)OBu-n Me
CH2S(O)CH2C(O)OBu-i Me
CH2S(O)CH2C(O)OBu-t Me
CH2S(O)CH2C(O)OPen-n Me
CH2S(O)CH2C(O)OHex-n Me
CH2S(O)CH2C(O)OMe Et
CH2S(O)CH2C(O)OMe Pr-n
CH2S(O)CH2C(O)OMe Pr-i
CH2S(O)CH2C(O)OMe Pr-c
CH2S(O)CH2C(O)OMe Bu-n
CH2S(O)CH2C(O)OMe Bu-i
CH2S(O)CH2C(O)OMe Bu-c
CH2S(O)CH2C(O)OMe Bu-s
CH2S(O)CH2C(O)OMe Bu-t
CH2S(O)CH2C(O)OMe Pen-n
CH2S(O)CH2C(O)OMe Pen-c
CH2S(O)CH2C(O)OMe Hex-n
CH2S(O)CH2C(O)OMe Hex-c
CH2S(O)CH2C(O)OMe CH2Pr-c
CH2S(O)CH2C(O)OMe CH2Bu-c
CH2S(O)CH2C(O)OMe CH2Pen-c
CH2S(O)CH2C(O)OMe CH2Hex-c
CH2S(O)CH2C(O)OMe CH2CH=CH2
CH2S(O)CH2C(O)OMe CH2CH=C(Cl)2
CH2S(O)CH2C(O)OMe CH2C≡CH
CH2S(O)CH2C(O)OMe CH2CN
CH2S(O)CH2C(O)OMe CH2CF3
CH2S(O)CH2C(O)OMe CH2OMe
CH2S(O)CH2C(O)OMe CH2OCF3
CH2S(O)CH2C(O)OMe CH2SMe
CH2S(O)CH2C(O)OMe CH2S(O)Me
CH2S(O)CH2C(O)OMe CH2S(O)2Me
CH2S(O)CH2C(O)OMe CH2SCF3
CH2S(O)CH2C(O)OMe CH2S(O)CF3
CH2S(O)CH2C(O)OMe CH2S(O)2CF3
CH2S(O)CH2C(O)OMe CH2CH(OMe)2
CH2S(O)CH2C(O)OMe CH2CH(SMe)2
CH2S(O)CH2C(O)OMe CH2C(O)Me
CH2S(O)CH2C(O)OMe CH2C(O)CF3
CH2S(O)CH2C(O)OMe CH2C(O)OMe
CH2S(O)2CH2C(O)OMe Me
CH2S(O)2CH2C(O)OEt Me
CH2S(O)2CH2C(O)OPr-n Me
CH2S(O)2CH2C(O)OPr-i Me
CH2S(O)2CH2C(O)OBu-n Me
CH2S(O)2CH2C(O)OBu-i Me
CH2S(O)2CH2C(O)OBu-t Me
CH2S(O)2CH2C(O)OPen-n Me
CH2S(O)2CH2C(O)OHex-n Me
CH2S(O)2CH2C(O)OMe Et
CH2S(O)2CH2C(O)OMe Pr-n
CH2S(O)2CH2C(O)OMe Pr-i
CH2S(O)2CH2C(O)OMe Pr-c
CH2S(O)2CH2C(O)OMe Bu-n
CH2S(O)2CH2C(O)OMe Bu-i
CH2S(O)2CH2C(O)OMe Bu-c
CH2S(O)2CH2C(O)OMe Bu-s
CH2S(O)2CH2C(O)OMe Bu-t
CH2S(O)2CH2C(O)OMe Pen-n
CH2S(O)2CH2C(O)OMe Pen-c
CH2S(O)2CH2C(O)OMe Hex-n
CH2S(O)2CH2C(O)OMe Hex-c
CH2S(O)2CH2C(O)OMe CH2Pr-c
CH2S(O)2CH2C(O)OMe CH2Bu-c
CH2S(O)2CH2C(O)OMe CH2Pen-c
CH2S(O)2CH2C(O)OMe CH2Hex-c
CH2S(O)2CH2C(O)OMe CH2CH=CH2
CH2S(O)2CH2C(O)OMe CH2CH=C(Cl)2
CH2S(O)2CH2C(O)OMe CH2C≡CH
CH2S(O)2CH2C(O)OMe CH2CN
CH2S(O)2CH2C(O)OMe CH2CF3
CH2S(O)2CH2C(O)OMe CH2OMe
CH2S(O)2CH2C(O)OMe CH2OCF3
CH2S(O)2CH2C(O)OMe CH2SMe
CH2S(O)2CH2C(O)OMe CH2S(O)Me
CH2S(O)2CH2C(O)OMe CH2S(O)2Me
CH2S(O)2CH2C(O)OMe CH2SCF3
CH2S(O)2CH2C(O)OMe CH2S(O)CF3
CH2S(O)2CH2C(O)OMe CH2S(O)2CF3
CH2S(O)2CH2C(O)OMe CH2CH(OMe)2
CH2S(O)2CH2C(O)OMe CH2CH(SMe)2
CH2S(O)2CH2C(O)OMe CH2C(O)Me
CH2S(O)2CH2C(O)OMe CH2C(O)CF3
CH2S(O)2CH2C(O)OMe CH2C(O)OMe
CH(Me)SCH2C(O)OMe Me
CH(Me)SCH2C(O)OEt Me
CH(Me)SCH2C(O)OPr-n Me
CH(Me)SCH2C(O)OPr-i Me
CH(Me)SCH2C(O)OBu-n Me
CH(Me)SCH2C(O)OBu-i Me
CH(Me)SCH2C(O)OBu-t Me
CH(Me)SCH2C(O)OPen-n Me
CH(Me)SCH2C(O)OHex-n Me
CH(Me)SCH2C(O)OMe Et
CH(Me)SCH2C(O)OMe Pr-n
CH(Me)SCH2C(O)OMe Pr-i
CH(Me)SCH2C(O)OMe Pr-c
CH(Me)SCH2C(O)OMe Bu-n
CH(Me)SCH2C(O)OMe Bu-i
CH(Me)SCH2C(O)OMe Bu-c
CH(Me)SCH2C(O)OMe Bu-s
CH(Me)SCH2C(O)OMe Bu-t
CH(Me)SCH2C(O)OMe Pen-n
CH(Me)SCH2C(O)OMe Pen-c
CH(Me)SCH2C(O)OMe Hex-n
CH(Me)SCH2C(O)OMe Hex-c
CH(Me)SCH2C(O)OMe CH2Pr-c
CH(Me)SCH2C(O)OMe CH2Bu-c
CH(Me)SCH2C(O)OMe CH2Pen-c
CH(Me)SCH2C(O)OMe CH2Hex-c
CH(Me)SCH2C(O)OMe CH2CH=CH2
CH(Me)SCH2C(O)OMe CH2CH=C(Cl)2
CH(Me)SCH2C(O)OMe CH2C≡CH
CH(Me)SCH2C(O)OMe CH2CN
CH(Me)SCH2C(O)OMe CH2CF3
CH(Me)SCH2C(O)OMe CH2OMe
CH(Me)SCH2C(O)OMe CH2OCF3
CH(Me)SCH2C(O)OMe CH2SMe
CH(Me)SCH2C(O)OMe CH2S(O)Me
CH(Me)SCH2C(O)OMe CH2S(O)2Me
CH(Me)SCH2C(O)OMe CH2SCF3
CH(Me)SCH2C(O)OMe CH2S(O)CF3
CH(Me)SCH2C(O)OMe CH2S(O)2CF3
CH(Me)SCH2C(O)OMe CH2CH(OMe)2
CH(Me)SCH2C(O)OMe CH2CH(SMe)2
CH(Me)SCH2C(O)OMe CH2C(O)Me
CH(Me)SCH2C(O)OMe CH2C(O)CF3
CH(Me)SCH2C(O)OMe CH2C(O)OMe
CH(Me)S(O)CH2C(O)OMe Me
CH(Me)S(O)CH2C(O)OEt Me
CH(Me)S(O)CH2C(O)OPr-n Me
CH(Me)S(O)CH2C(O)OPr-i Me
CH(Me)S(O)CH2C(O)OBu-n Me
CH(Me)S(O)CH2C(O)OBu-i Me
CH(Me)S(O)CH2C(O)OBu-t Me
CH(Me)S(O)CH2C(O)OPen-n Me
CH(Me)S(O)CH2C(O)OHex-n Me
CH(Me)S(O)CH2C(O)OMe Et
CH(Me)S(O)CH2C(O)OMe Pr-n
CH(Me)S(O)CH2C(O)OMe Pr-i
CH(Me)S(O)CH2C(O)OMe Pr-c
CH(Me)S(O)CH2C(O)OMe Bu-n
CH(Me)S(O)CH2C(O)OMe Bu-i
CH(Me)S(O)CH2C(O)OMe Bu-c
CH(Me)S(O)CH2C(O)OMe Bu-s
CH(Me)S(O)CH2C(O)OMe Bu-t
CH(Me)S(O)CH2C(O)OMe Pen-n
CH(Me)S(O)CH2C(O)OMe Pen-c
CH(Me)S(O)CH2C(O)OMe Hex-n
CH(Me)S(O)CH2C(O)OMe Hex-c
CH(Me)S(O)CH2C(O)OMe CH2Pr-c
CH(Me)S(O)CH2C(O)OMe CH2Bu-c
CH(Me)S(O)CH2C(O)OMe CH2Pen-c
CH(Me)S(O)CH2C(O)OMe CH2Hex-c
CH(Me)S(O)CH2C(O)OMe CH2CH=CH2
CH(Me)S(O)CH2C(O)OMe CH2CH=C(Cl)2
CH(Me)S(O)CH2C(O)OMe CH2C≡CH
CH(Me)S(O)CH2C(O)OMe CH2CN
CH(Me)S(O)CH2C(O)OMe CH2CF3
CH(Me)S(O)CH2C(O)OMe CH2OMe
CH(Me)S(O)CH2C(O)OMe CH2OCF3
CH(Me)S(O)CH2C(O)OMe CH2SMe
CH(Me)S(O)CH2C(O)OMe CH2S(O)Me
CH(Me)S(O)CH2C(O)OMe CH2S(O)2Me
CH(Me)S(O)CH2C(O)OMe CH2SCF3
CH(Me)S(O)CH2C(O)OMe CH2S(O)CF3
CH(Me)S(O)CH2C(O)OMe CH2S(O)2CF3
CH(Me)S(O)CH2C(O)OMe CH2CH(OMe)2
CH(Me)S(O)CH2C(O)OMe CH2CH(SMe)2
CH(Me)S(O)CH2C(O)OMe CH2C(O)Me
CH(Me)S(O)CH2C(O)OMe CH2C(O)CF3
CH(Me)S(O)CH2C(O)OMe CH2C(O)OMe
CH(Me)S(O)2CH2C(O)OMe Me
CH(Me)S(O)2CH2C(O)OEt Me
CH(Me)S(O)2CH2C(O)OPr-n Me
CH(Me)S(O)2CH2C(O)OPr-i Me
CH(Me)S(O)2CH2C(O)OBu-n Me
CH(Me)S(O)2CH2C(O)OBu-i Me
CH(Me)S(O)2CH2C(O)OBu-t Me
CH(Me)S(O)2CH2C(O)OPen-n Me
CH(Me)S(O)2CH2C(O)OHex-n Me
CH(Me)S(O)2CH2C(O)OMe Et
CH(Me)S(O)2CH2C(O)OMe Pr-n
CH(Me)S(O)2CH2C(O)OMe Pr-i
CH(Me)S(O)2CH2C(O)OMe Pr-c
CH(Me)S(O)2CH2C(O)OMe Bu-n
CH(Me)S(O)2CH2C(O)OMe Bu-i
CH(Me)S(O)2CH2C(O)OMe Bu-c
CH(Me)S(O)2CH2C(O)OMe Bu-s
CH(Me)S(O)2CH2C(O)OMe Bu-t
CH(Me)S(O)2CH2C(O)OMe Pen-n
CH(Me)S(O)2CH2C(O)OMe Pen-c
CH(Me)S(O)2CH2C(O)OMe Hex-n
CH(Me)S(O)2CH2C(O)OMe Hex-c
CH(Me)S(O)2CH2C(O)OMe CH2Pr-c
CH(Me)S(O)2CH2C(O)OMe CH2Bu-c
CH(Me)S(O)2CH2C(O)OMe CH2Pen-c
CH(Me)S(O)2CH2C(O)OMe CH2Hex-c
CH(Me)S(O)2CH2C(O)OMe CH2CH=CH2
CH(Me)S(O)2CH2C(O)OMe CH2CH=C(Cl)2
CH(Me)S(O)2CH2C(O)OMe CH2C≡CH
CH(Me)S(O)2CH2C(O)OMe CH2CN
CH(Me)S(O)2CH2C(O)OMe CH2CF3
CH(Me)S(O)2CH2C(O)OMe CH2OMe
CH(Me)S(O)2CH2C(O)OMe CH2OCF3
CH(Me)S(O)2CH2C(O)OMe CH2SMe
CH(Me)S(O)2CH2C(O)OMe CH2S(O)Me
CH(Me)S(O)2CH2C(O)OMe CH2S(O)2Me
CH(Me)S(O)2CH2C(O)OMe CH2SCF3
CH(Me)S(O)2CH2C(O)OMe CH2S(O)CF3
CH(Me)S(O)2CH2C(O)OMe CH2S(O)2CF3
CH(Me)S(O)2CH2C(O)OMe CH2CH(OMe)2
CH(Me)S(O)2CH2C(O)OMe CH2CH(SMe)2
CH(Me)S(O)2CH2C(O)OMe CH2C(O)Me
CH(Me)S(O)2CH2C(O)OMe CH2C(O)CF3
CH(Me)S(O)2CH2C(O)OMe CH2C(O)OMe
CH(Et)SCH2C(O)OMe Me
CH(Et)SCH2C(O)OEt Me
CH(Et)SCH2C(O)OPr-n Me
CH(Et)SCH2C(O)OPr-i Me
CH(Et)SCH2C(O)OBu-n Me
CH(Et)SCH2C(O)OBu-i Me
CH(Et)SCH2C(O)OBu-t Me
CH(Et)SCH2C(O)OPen-n Me
CH(Et)SCH2C(O)OHex-n Me
CH(Et)SCH2C(O)OMe Et
CH(Et)SCH2C(O)OMe Pr-n
CH(Et)SCH2C(O)OMe Pr-i
CH(Et)SCH2C(O)OMe Pr-c
CH(Et)SCH2C(O)OMe Bu-n
CH(Et)SCH2C(O)OMe Bu-i
CH(Et)SCH2C(O)OMe Bu-c
CH(Et)SCH2C(O)OMe Bu-s
CH(Et)SCH2C(O)OMe Bu-t
CH(Et)SCH2C(O)OMe Pen-n
CH(Et)SCH2C(O)OMe Pen-c
CH(Et)SCH2C(O)OMe Hex-n
CH(Et)SCH2C(O)OMe Hex-c
CH(Et)SCH2C(O)OMe CH2Pr-c
CH(Et)SCH2C(O)OMe CH2Bu-c
CH(Et)SCH2C(O)OMe CH2Pen-c
CH(Et)SCH2C(O)OMe CH2Hex-c
CH(Et)SCH2C(O)OMe CH2CH=CH2
CH(Et)SCH2C(O)OMe CH2CH=C(Cl)2
CH(Et)SCH2C(O)OMe CH2C≡CH
CH(Et)SCH2C(O)OMe CH2CN
CH(Et)SCH2C(O)OMe CH2CF3
CH(Et)SCH2C(O)OMe CH2OMe
CH(Et)SCH2C(O)OMe CH2OCF3
CH(Et)SCH2C(O)OMe CH2SMe
CH(Et)SCH2C(O)OMe CH2S(O)Me
CH(Et)SCH2C(O)OMe CH2S(O)2Me
CH(Et)SCH2C(O)OMe CH2SCF3
CH(Et)SCH2C(O)OMe CH2S(O)CF3
CH(Et)SCH2C(O)OMe CH2S(O)2CF3
CH(Et)SCH2C(O)OMe CH2CH(OMe)2
CH(Et)SCH2C(O)OMe CH2CH(SMe)2
CH(Et)SCH2C(O)OMe CH2C(O)Me
CH(Et)SCH2C(O)OMe CH2C(O)CF3
CH(Et)SCH2C(O)OMe CH2C(O)OMe
CH(Et)S(O)CH2C(O)OMe Me
CH(Et)S(O)CH2C(O)OEt Me
CH(Et)S(O)CH2C(O)OPr-n Me
CH(Et)S(O)CH2C(O)OPr-i Me
CH(Et)S(O)CH2C(O)OBu-n Me
CH(Et)S(O)CH2C(O)OBu-i Me
CH(Et)S(O)CH2C(O)OBu-t Me
CH(Et)S(O)CH2C(O)OPen-n Me
CH(Et)S(O)CH2C(O)OHex-n Me
CH(Et)S(O)CH2C(O)OMe Et
CH(Et)S(O)CH2C(O)OMe Pr-n
CH(Et)S(O)CH2C(O)OMe Pr-i
CH(Et)S(O)CH2C(O)OMe Pr-c
CH(Et)S(O)CH2C(O)OMe Bu-n
CH(Et)S(O)CH2C(O)OMe Bu-i
CH(Et)S(O)CH2C(O)OMe Bu-c
CH(Et)S(O)CH2C(O)OMe Bu-s
CH(Et)S(O)CH2C(O)OMe Bu-t
CH(Et)S(O)CH2C(O)OMe Pen-n
CH(Et)S(O)CH2C(O)OMe Pen-c
CH(Et)S(O)CH2C(O)OMe Hex-n
CH(Et)S(O)CH2C(O)OMe Hex-c
CH(Et)S(O)CH2C(O)OMe CH2Pr-c
CH(Et)S(O)CH2C(O)OMe CH2Bu-c
CH(Et)S(O)CH2C(O)OMe CH2Pen-c
CH(Et)S(O)CH2C(O)OMe CH2Hex-c
CH(Et)S(O)CH2C(O)OMe CH2CH=CH2
CH(Et)S(O)CH2C(O)OMe CH2CH=C(Cl)2
CH(Et)S(O)CH2C(O)OMe CH2C≡CH
CH(Et)S(O)CH2C(O)OMe CH2CN
CH(Et)S(O)CH2C(O)OMe CH2CF3
CH(Et)S(O)CH2C(O)OMe CH2OMe
CH(Et)S(O)CH2C(O)OMe CH2OCF3
CH(Et)S(O)CH2C(O)OMe CH2SMe
CH(Et)S(O)CH2C(O)OMe CH2S(O)Me
CH(Et)S(O)CH2C(O)OMe CH2S(O)2Me
CH(Et)S(O)CH2C(O)OMe CH2SCF3
CH(Et)S(O)CH2C(O)OMe CH2S(O)CF3
CH(Et)S(O)CH2C(O)OMe CH2S(O)2CF3
CH(Et)S(O)CH2C(O)OMe CH2CH(OMe)2
CH(Et)S(O)CH2C(O)OMe CH2CH(SMe)2
CH(Et)S(O)CH2C(O)OMe CH2C(O)Me
CH(Et)S(O)CH2C(O)OMe CH2C(O)CF3
CH(Et)S(O)CH2C(O)OMe CH2C(O)OMe
CH(Et)S(O)2CH2C(O)OMe Me
CH(Et)S(O)2CH2C(O)OEt Me
CH(Et)S(O)2CH2C(O)OPr-n Me
CH(Et)S(O)2CH2C(O)OPr-i Me
CH(Et)S(O)2CH2C(O)OBu-n Me
CH(Et)S(O)2CH2C(O)OBu-i Me
CH(Et)S(O)2CH2C(O)OBu-t Me
CH(Et)S(O)2CH2C(O)OPen-n Me
CH(Et)S(O)2CH2C(O)OHex-n Me
CH(Et)S(O)2CH2C(O)OMe Et
CH(Et)S(O)2CH2C(O)OMe Pr-n
CH(Et)S(O)2CH2C(O)OMe Pr-i
CH(Et)S(O)2CH2C(O)OMe Pr-c
CH(Et)S(O)2CH2C(O)OMe Bu-n
CH(Et)S(O)2CH2C(O)OMe Bu-i
CH(Et)S(O)2CH2C(O)OMe Bu-c
CH(Et)S(O)2CH2C(O)OMe Bu-s
CH(Et)S(O)2CH2C(O)OMe Bu-t
CH(Et)S(O)2CH2C(O)OMe Pen-n
CH(Et)S(O)2CH2C(O)OMe Pen-c
CH(Et)S(O)2CH2C(O)OMe Hex-n
CH(Et)S(O)2CH2C(O)OMe Hex-c
CH(Et)S(O)2CH2C(O)OMe CH2Pr-c
CH(Et)S(O)2CH2C(O)OMe CH2Bu-c
CH(Et)S(O)2CH2C(O)OMe CH2Pen-c
CH(Et)S(O)2CH2C(O)OMe CH2Hex-c
CH(Et)S(O)2CH2C(O)OMe CH2CH=CH2
CH(Et)S(O)2CH2C(O)OMe CH2CH=C(Cl)2
CH(Et)S(O)2CH2C(O)OMe CH2C≡CH
CH(Et)S(O)2CH2C(O)OMe CH2CN
CH(Et)S(O)2CH2C(O)OMe CH2CF3
CH(Et)S(O)2CH2C(O)OMe CH2OMe
CH(Et)S(O)2CH2C(O)OMe CH2OCF3
CH(Et)S(O)2CH2C(O)OMe CH2SMe
CH(Et)S(O)2CH2C(O)OMe CH2S(O)Me
CH(Et)S(O)2CH2C(O)OMe CH2S(O)2Me
CH(Et)S(O)2CH2C(O)OMe CH2SCF3
CH(Et)S(O)2CH2C(O)OMe CH2S(O)CF3
CH(Et)S(O)2CH2C(O)OMe CH2S(O)2CF3
CH(Et)S(O)2CH2C(O)OMe CH2CH(OMe)2
CH(Et)S(O)2CH2C(O)OMe CH2CH(SMe)2
CH(Et)S(O)2CH2C(O)OMe CH2C(O)Me
CH(Et)S(O)2CH2C(O)OMe CH2C(O)CF3
CH(Et)S(O)2CH2C(O)OMe CH2C(O)OMe
CH2SCH2C(O)Me Me
CH2SCH2C(O)Et Me
CH2SCH2C(O)Pr-n Me
CH2SCH2C(O)Pr-i Me
CH2SCH2C(O)Pr-c Me
CH2SCH2C(O)Bu-n Me
CH2SCH2C(O)Bu-i Me
CH2SCH2C(O)Bu-c Me
CH2SCH2C(O)Bu-t Me
CH2SCH2C(O)Pen-n Me
CH2SCH2C(O)Pen-c Me
CH2SCH2C(O)Hex-n Me
CH2SCH2C(O)Hex-c Me
CH2SCH2C(O)Me Et
CH2SCH2C(O)Me Pr-n
CH2SCH2C(O)Me Pr-i
CH2SCH2C(O)Me Pr-c
CH2SCH2C(O)Me Bu-n
CH2SCH2C(O)Me Bu-i
CH2SCH2C(O)Me Bu-c
CH2SCH2C(O)Me Bu-s
CH2SCH2C(O)Me Bu-t
CH2SCH2C(O)Me Pen-n
CH2SCH2C(O)Me Pen-c
CH2SCH2C(O)Me Hex-n
CH2SCH2C(O)Me Hex-c
CH2SCH2C(O)Me CH2Pr-c
CH2SCH2C(O)Me CH2Bu-c
CH2SCH2C(O)Me CH2Pen-c
CH2SCH2C(O)Me CH2Hex-c
CH2SCH2C(O)Me CH2CH=CH2
CH2SCH2C(O)Me CH2CH=C(Cl)2
CH2SCH2C(O)Me CH2C≡CH
CH2SCH2C(O)Me CH2CN
CH2SCH2C(O)Me CH2CF3
CH2SCH2C(O)Me CH2OMe
CH2SCH2C(O)Me CH2OCF3
CH2SCH2C(O)Me CH2SMe
CH2SCH2C(O)Me CH2S(O)Me
CH2SCH2C(O)Me CH2S(O)2Me
CH2SCH2C(O)Me CH2SCF3
CH2SCH2C(O)Me CH2S(O)CF3
CH2SCH2C(O)Me CH2S(O)2CF3
CH2SCH2C(O)Me CH2CH(OMe)2
CH2SCH2C(O)Me CH2CH(SMe)2
CH2SCH2C(O)Me CH2C(O)Me
CH2SCH2C(O)Me CH2C(O)CF3
CH2SCH2C(O)Me CH2C(O)OMe
CH2S(O)CH2C(O)Me Me
CH2S(O)CH2C(O)Et Me
CH2S(O)CH2C(O)Pr-n Me
CH2S(O)CH2C(O)Pr-i Me
CH2S(O)CH2C(O)Pr-c Me
CH2S(O)CH2C(O)Bu-n Me
CH2S(O)CH2C(O)Bu-i Me
CH2S(O)CH2C(O)Bu-c Me
CH2S(O)CH2C(O)Bu-t Me
CH2S(O)CH2C(O)Pen-n Me
CH2S(O)CH2C(O)Pen-c Me
CH2S(O)CH2C(O)Hex-n Me
CH2S(O)CH2C(O)Hex-c Me
CH2S(O)CH2C(O)Me Et
CH2S(O)CH2C(O)Me Pr-n
CH2S(O)CH2C(O)Me Pr-i
CH2S(O)CH2C(O)Me Pr-c
CH2S(O)CH2C(O)Me Bu-n
CH2S(O)CH2C(O)Me Bu-i
CH2S(O)CH2C(O)Me Bu-c
CH2S(O)CH2C(O)Me Bu-s
CH2S(O)CH2C(O)Me Bu-t
CH2S(O)CH2C(O)Me Pen-n
CH2S(O)CH2C(O)Me Pen-c
CH2S(O)CH2C(O)Me Hex-n
CH2S(O)CH2C(O)Me Hex-c
CH2S(O)CH2C(O)Me CH2Pr-c
CH2S(O)CH2C(O)Me CH2Bu-c
CH2S(O)CH2C(O)Me CH2Pen-c
CH2S(O)CH2C(O)Me CH2Hex-c
CH2S(O)CH2C(O)Me CH2CH=CH2
CH2S(O)CH2C(O)Me CH2CH=C(Cl)2
CH2S(O)CH2C(O)Me CH2C≡CH
CH2S(O)CH2C(O)Me CH2CN
CH2S(O)CH2C(O)Me CH2CF3
CH2S(O)CH2C(O)Me CH2OMe
CH2S(O)CH2C(O)Me CH2OCF3
CH2S(O)CH2C(O)Me CH2SMe
CH2S(O)CH2C(O)Me CH2S(O)Me
CH2S(O)CH2C(O)Me CH2S(O)2Me
CH2S(O)CH2C(O)Me CH2SCF3
CH2S(O)CH2C(O)Me CH2S(O)CF3
CH2S(O)CH2C(O)Me CH2S(O)2CF3
CH2S(O)CH2C(O)Me CH2CH(OMe)2
CH2S(O)CH2C(O)Me CH2CH(SMe)2
CH2S(O)CH2C(O)Me CH2C(O)Me
CH2S(O)CH2C(O)Me CH2C(O)CF3
CH2S(O)CH2C(O)Me CH2C(O)OMe
CH2S(O)2CH2C(O)Me Me
CH2S(O)2CH2C(O)Et Me
CH2S(O)2CH2C(O)Pr-n Me
CH2S(O)2CH2C(O)Pr-i Me
CH2S(O)2CH2C(O)Pr-c Me
CH2S(O)2CH2C(O)Bu-n Me
CH2S(O)2CH2C(O)Bu-i Me
CH2S(O)2CH2C(O)Bu-c Me
CH2S(O)2CH2C(O)Bu-t Me
CH2S(O)2CH2C(O)Pen-n Me
CH2S(O)2CH2C(O)Pen-c Me
CH2S(O)2CH2C(O)Hex-n Me
CH2S(O)2CH2C(O)Hex-c Me
CH2S(O)2CH2C(O)Me Et
CH2S(O)2CH2C(O)Me Pr-n
CH2S(O)2CH2C(O)Me Pr-i
CH2S(O)2CH2C(O)Me Pr-c
CH2S(O)2CH2C(O)Me Bu-n
CH2S(O)2CH2C(O)Me Bu-i
CH2S(O)2CH2C(O)Me Bu-c
CH2S(O)2CH2C(O)Me Bu-s
CH2S(O)2CH2C(O)Me Bu-t
CH2S(O)2CH2C(O)Me Pen-n
CH2S(O)2CH2C(O)Me Pen-c
CH2S(O)2CH2C(O)Me Hex-n
CH2S(O)2CH2C(O)Me Hex-c
CH2S(O)2CH2C(O)Me CH2Pr-c
CH2S(O)2CH2C(O)Me CH2Bu-c
CH2S(O)2CH2C(O)Me CH2Pen-c
CH2S(O)2CH2C(O)Me CH2Hex-c
CH2S(O)2CH2C(O)Me CH2CH=CH2
CH2S(O)2CH2C(O)Me CH2CH=C(Cl)2
CH2S(O)2CH2C(O)Me CH2C≡CH
CH2S(O)2CH2C(O)Me CH2CN
CH2S(O)2CH2C(O)Me CH2CF3
CH2S(O)2CH2C(O)Me CH2OMe
CH2S(O)2CH2C(O)Me CH2OCF3
CH2S(O)2CH2C(O)Me CH2SMe
CH2S(O)2CH2C(O)Me CH2S(O)Me
CH2S(O)2CH2C(O)Me CH2S(O)2Me
CH2S(O)2CH2C(O)Me CH2SCF3
CH2S(O)2CH2C(O)Me CH2S(O)CF3
CH2S(O)2CH2C(O)Me CH2S(O)2CF3
CH2S(O)2CH2C(O)Me CH2CH(OMe)2
CH2S(O)2CH2C(O)Me CH2CH(SMe)2
CH2S(O)2CH2C(O)Me CH2C(O)Me
CH2S(O)2CH2C(O)Me CH2C(O)CF3
CH2S(O)2CH2C(O)Me CH2C(O)OMe
CH(Me)SCH2C(O)Me Me
CH(Me)SCH2C(O)Et Me
CH(Me)SCH2C(O)Pr-n Me
CH(Me)SCH2C(O)Pr-i Me
CH(Me)SCH2C(O)Pr-c Me
CH(Me)SCH2C(O)Bu-n Me
CH(Me)SCH2C(O)Bu-i Me
CH(Me)SCH2C(O)Bu-c Me
CH(Me)SCH2C(O)Bu-t Me
CH(Me)SCH2C(O)Pen-n Me
CH(Me)SCH2C(O)Pen-c Me
CH(Me)SCH2C(O)Hex-n Me
CH(Me)SCH2C(O)Hex-c Me
CH(Me)SCH2C(O)Me Et
CH(Me)SCH2C(O)Me Pr-n
CH(Me)SCH2C(O)Me Pr-i
CH(Me)SCH2C(O)Me Pr-c
CH(Me)SCH2C(O)Me Bu-n
CH(Me)SCH2C(O)Me Bu-i
CH(Me)SCH2C(O)Me Bu-c
CH(Me)SCH2C(O)Me Bu-s
CH(Me)SCH2C(O)Me Bu-t
CH(Me)SCH2C(O)Me Pen-n
CH(Me)SCH2C(O)Me Pen-c
CH(Me)SCH2C(O)Me Hex-n
CH(Me)SCH2C(O)Me Hex-c
CH(Me)SCH2C(O)Me CH2Pr-c
CH(Me)SCH2C(O)Me CH2Bu-c
CH(Me)SCH2C(O)Me CH2Pen-c
CH(Me)SCH2C(O)Me CH2Hex-c
CH(Me)SCH2C(O)Me CH2CH=CH2
CH(Me)SCH2C(O)Me CH2CH=C(Cl)2
CH(Me)SCH2C(O)Me CH2C≡CH
CH(Me)SCH2C(O)Me CH2CN
CH(Me)SCH2C(O)Me CH2CF3
CH(Me)SCH2C(O)Me CH2OMe
CH(Me)SCH2C(O)Me CH2OCF3
CH(Me)SCH2C(O)Me CH2SMe
CH(Me)SCH2C(O)Me CH2S(O)Me
CH(Me)SCH2C(O)Me CH2S(O)2Me
CH(Me)SCH2C(O)Me CH2SCF3
CH(Me)SCH2C(O)Me CH2S(O)CF3
CH(Me)SCH2C(O)Me CH2S(O)2CF3
CH(Me)SCH2C(O)Me CH2CH(OMe)2
CH(Me)SCH2C(O)Me CH2CH(SMe)2
CH(Me)SCH2C(O)Me CH2C(O)Me
CH(Me)SCH2C(O)Me CH2C(O)CF3
CH(Me)SCH2C(O)Me CH2C(O)OMe
CH(Me)S(O)CH2C(O)Me Me
CH(Me)S(O)CH2C(O)Et Me
CH(Me)S(O)CH2C(O)Pr-n Me
CH(Me)S(O)CH2C(O)Pr-i Me
CH(Me)S(O)CH2C(O)Pr-c Me
CH(Me)S(O)CH2C(O)Bu-n Me
CH(Me)S(O)CH2C(O)Bu-i Me
CH(Me)S(O)CH2C(O)Bu-t Me
CH(Me)S(O)CH2C(O)Pen-n Me
CH(Me)S(O)CH2C(O)Pen-c Me
CH(Me)S(O)CH2C(O)Hex-n Me
CH(Me)S(O)CH2C(O)Hex-c Me
CH(Me)S(O)CH2C(O)Me Et
CH(Me)S(O)CH2C(O)Me Pr-n
CH(Me)S(O)CH2C(O)Me Pr-i
CH(Me)S(O)CH2C(O)Me Pr-c
CH(Me)S(O)CH2C(O)Me Bu-n
CH(Me)S(O)CH2C(O)Me Bu-i
CH(Me)S(O)CH2C(O)Me Bu-c
CH(Me)S(O)CH2C(O)Me Bu-s
CH(Me)S(O)CH2C(O)Me Bu-t
CH(Me)S(O)CH2C(O)Me Pen-n
CH(Me)S(O)CH2C(O)Me Pen-c
CH(Me)S(O)CH2C(O)Me Hex-n
CH(Me)S(O)CH2C(O)Me Hex-c
CH(Me)S(O)CH2C(O)Me CH2Pr-c
CH(Me)S(O)CH2C(O)Me CH2Bu-c
CH(Me)S(O)CH2C(O)Me CH2Pen-c
CH(Me)S(O)CH2C(O)Me CH2Hex-c
CH(Me)S(O)CH2C(O)Me CH2CH=CH2
CH(Me)S(O)CH2C(O)Me CH2CH=C(Cl)2
CH(Me)S(O)CH2C(O)Me CH2C≡CH
CH(Me)S(O)CH2C(O)Me CH2CN
CH(Me)S(O)CH2C(O)Me CH2CF3
CH(Me)S(O)CH2C(O)Me CH2OMe
CH(Me)S(O)CH2C(O)Me CH2OCF3
CH(Me)S(O)CH2C(O)Me CH2SMe
CH(Me)S(O)CH2C(O)Me CH2S(O)Me
CH(Me)S(O)CH2C(O)Me CH2S(O)2Me
CH(Me)S(O)CH2C(O)Me CH2SCF3
CH(Me)S(O)CH2C(O)Me CH2S(O)CF3
CH(Me)S(O)CH2C(O)Me CH2S(O)2CF3
CH(Me)S(O)CH2C(O)Me CH2CH(OMe)2
CH(Me)S(O)CH2C(O)Me CH2CH(SMe)2
CH(Me)S(O)CH2C(O)Me CH2C(O)Me
CH(Me)S(O)CH2C(O)Me CH2C(O)CF3
CH(Me)S(O)CH2C(O)Me CH2C(O)OMe
CH(Me)S(O)2CH2C(O)Me Me
CH(Me)S(O)2CH2C(O)Et Me
CH(Me)S(O)2CH2C(O)Pr-n Me
CH(Me)S(O)2CH2C(O)Pr-i Me
CH(Me)S(O)2CH2C(O)Pr-c Me
CH(Me)S(O)2CH2C(O)Bu-n Me
CH(Me)S(O)2CH2C(O)Bu-i Me
CH(Me)S(O)2CH2C(O)Bu-t Me
CH(Me)S(O)2CH2C(O)Pen-n Me
CH(Me)S(O)2CH2C(O)Pen-c Me
CH(Me)S(O)2CH2C(O)Hex-n Me
CH(Me)S(O)2CH2C(O)Hex-c Me
CH(Me)S(O)2CH2C(O)Me Et
CH(Me)S(O)2CH2C(O)Me Pr-n
CH(Me)S(O)2CH2C(O)Me Pr-i
CH(Me)S(O)2CH2C(O)Me Pr-c
CH(Me)S(O)2CH2C(O)Me Bu-n
CH(Me)S(O)2CH2C(O)Me Bu-i
CH(Me)S(O)2CH2C(O)Me Bu-c
CH(Me)S(O)2CH2C(O)Me Bu-s
CH(Me)S(O)2CH2C(O)Me Bu-t
CH(Me)S(O)2CH2C(O)Me Pen-n
CH(Me)S(O)2CH2C(O)Me Pen-c
CH(Me)S(O)2CH2C(O)Me Hex-n
CH(Me)S(O)2CH2C(O)Me Hex-c
CH(Me)S(O)2CH2C(O)Me CH2Pr-c
CH(Me)S(O)2CH2C(O)Me CH2Bu-c
CH(Me)S(O)2CH2C(O)Me CH2Pen-c
CH(Me)S(O)2CH2C(O)Me CH2Hex-c
CH(Me)S(O)2CH2C(O)Me CH2CH=CH2
CH(Me)S(O)2CH2C(O)Me CH2CH=C(Cl)2
CH(Me)S(O)2CH2C(O)Me CH2C≡CH
CH(Me)S(O)2CH2C(O)Me CH2CN
CH(Me)S(O)2CH2C(O)Me CH2CF3
CH(Me)S(O)2CH2C(O)Me CH2OMe
CH(Me)S(O)2CH2C(O)Me CH2OCF3
CH(Me)S(O)2CH2C(O)Me CH2SMe
CH(Me)S(O)2CH2C(O)Me CH2S(O)Me
CH(Me)S(O)2CH2C(O)Me CH2S(O)2Me
CH(Me)S(O)2CH2C(O)Me CH2SCF3
CH(Me)S(O)2CH2C(O)Me CH2S(O)CF3
CH(Me)S(O)2CH2C(O)Me CH2S(O)2CF3
CH(Me)S(O)2CH2C(O)Me CH2CH(OMe)2
CH(Me)S(O)2CH2C(O)Me CH2CH(SMe)2
CH(Me)S(O)2CH2C(O)Me CH2C(O)Me
CH(Me)S(O)2CH2C(O)Me CH2C(O)CF3
CH(Me)S(O)2CH2C(O)Me CH2C(O)OMe
CH(Et)SCH2C(O)Me Me
CH(Et)SCH2C(O)Et Me
CH(Et)SCH2C(O)Pr-n Me
CH(Et)SCH2C(O)Pr-i Me
CH(Et)SCH2C(O)Pr-c Me
CH(Et)SCH2C(O)Bu-n Me
CH(Et)SCH2C(O)Bu-i Me
CH(Et)SCH2C(O)Bu-c Me
CH(Et)SCH2C(O)Bu-t Me
CH(Et)SCH2C(O)Pen-n Me
CH(Et)SCH2C(O)Pen-c Me
CH(Et)SCH2C(O)Hex-n Me
CH(Et)SCH2C(O)Hex-c Me
CH(Et)SCH2C(O)Me Et
CH(Et)SCH2C(O)Me Pr-n
CH(Et)SCH2C(O)Me Pr-i
CH(Et)SCH2C(O)Me Pr-c
CH(Et)SCH2C(O)Me Bu-n
CH(Et)SCH2C(O)Me Bu-i
CH(Et)SCH2C(O)Me Bu-c
CH(Et)SCH2C(O)Me Bu-s
CH(Et)SCH2C(O)Me Bu-t
CH(Et)SCH2C(O)Me Pen-n
CH(Et)SCH2C(O)Me Pen-c
CH(Et)SCH2C(O)Me Hex-n
CH(Et)SCH2C(O)Me Hex-c
CH(Et)SCH2C(O)Me CH2Pr-c
CH(Et)SCH2C(O)Me CH2Bu-c
CH(Et)SCH2C(O)Me CH2Pen-c
CH(Et)SCH2C(O)Me CH2Hex-c
CH(Et)SCH2C(O)Me CH2CH=CH2
CH(Et)SCH2C(O)Me CH2CH=C(Cl)2
CH(Et)SCH2C(O)Me CH2C≡CH
CH(Et)SCH2C(O)Me CH2CN
CH(Et)SCH2C(O)Me CH2CF3
CH(Et)SCH2C(O)Me CH2OMe
CH(Et)SCH2C(O)Me CH2OCF3
CH(Et)SCH2C(O)Me CH2SMe
CH(Et)SCH2C(O)Me CH2S(O)Me
CH(Et)SCH2C(O)Me CH2S(O)2Me
CH(Et)SCH2C(O)Me CH2SCF3
CH(Et)SCH2C(O)Me CH2S(O)CF3
CH(Et)SCH2C(O)Me CH2S(O)2CF3
CH(Et)SCH2C(O)Me CH2CH(OMe)2
CH(Et)SCH2C(O)Me CH2CH(SMe)2
CH(Et)SCH2C(O)Me CH2C(O)Me
CH(Et)SCH2C(O)Me CH2C(O)CF3
CH(Et)SCH2C(O)Me CH2C(O)OMe
CH(Et)S(O)CH2C(O)Me Me
CH(Et)S(O)CH2C(O)Et Me
CH(Et)S(O)CH2C(O)Pr-n Me
CH(Et)S(O)CH2C(O)Pr-i Me
CH(Et)S(O)CH2C(O)Pr-c Me
CH(Et)S(O)CH2C(O)Bu-n Me
CH(Et)S(O)CH2C(O)Bu-i Me
CH(Et)S(O)CH2C(O)Bu-t Me
CH(Et)S(O)CH2C(O)Pen-n Me
CH(Et)S(O)CH2C(O)Pen-c Me
CH(Et)S(O)CH2C(O)Hex-n Me
CH(Et)S(O)CH2C(O)Hex-c Me
CH(Et)S(O)CH2C(O)Me Et
CH(Et)S(O)CH2C(O)Me Pr-n
CH(Et)S(O)CH2C(O)Me Pr-i
CH(Et)S(O)CH2C(O)Me Pr-c
CH(Et)S(O)CH2C(O)Me Bu-n
CH(Et)S(O)CH2C(O)Me Bu-i
CH(Et)S(O)CH2C(O)Me Bu-c
CH(Et)S(O)CH2C(O)Me Bu-s
CH(Et)S(O)CH2C(O)Me Bu-t
CH(Et)S(O)CH2C(O)Me Pen-n
CH(Et)S(O)CH2C(O)Me Pen-c
CH(Et)S(O)CH2C(O)Me Hex-n
CH(Et)S(O)CH2C(O)Me Hex-c
CH(Et)S(O)CH2C(O)Me CH2Pr-c
CH(Et)S(O)CH2C(O)Me CH2Bu-c
CH(Et)S(O)CH2C(O)Me CH2Pen-c
CH(Et)S(O)CH2C(O)Me CH2Hex-c
CH(Et)S(O)CH2C(O)Me CH2CH=CH2
CH(Et)S(O)CH2C(O)Me CH2CH=C(Cl)2
CH(Et)S(O)CH2C(O)Me CH2C≡CH
CH(Et)S(O)CH2C(O)Me CH2CN
CH(Et)S(O)CH2C(O)Me CH2CF3
CH(Et)S(O)CH2C(O)Me CH2OMe
CH(Et)S(O)CH2C(O)Me CH2OCF3
CH(Et)S(O)CH2C(O)Me CH2SMe
CH(Et)S(O)CH2C(O)Me CH2S(O)Me
CH(Et)S(O)CH2C(O)Me CH2S(O)2Me
CH(Et)S(O)CH2C(O)Me CH2SCF3
CH(Et)S(O)CH2C(O)Me CH2S(O)CF3
CH(Et)S(O)CH2C(O)Me CH2S(O)2CF3
CH(Et)S(O)CH2C(O)Me CH2CH(OMe)2
CH(Et)S(O)CH2C(O)Me CH2CH(SMe)2
CH(Et)S(O)CH2C(O)Me CH2C(O)Me
CH(Et)S(O)CH2C(O)Me CH2C(O)CF3
CH(Et)S(O)CH2C(O)Me CH2C(O)OMe
CH(Et)S(O)2CH2C(O)Me Me
CH(Et)S(O)2CH2C(O)Et Me
CH(Et)S(O)2CH2C(O)Pr-n Me
CH(Et)S(O)2CH2C(O)Pr-i Me
CH(Et)S(O)2CH2C(O)Pr-c Me
CH(Et)S(O)2CH2C(O)Bu-n Me
CH(Et)S(O)2CH2C(O)Bu-i Me
CH(Et)S(O)2CH2C(O)Bu-t Me
CH(Et)S(O)2CH2C(O)Pen-n Me
CH(Et)S(O)2CH2C(O)Pen-c Me
CH(Et)S(O)2CH2C(O)Hex-n Me
CH(Et)S(O)2CH2C(O)Hex-c Me
CH(Et)S(O)2CH2C(O)Me Et
CH(Et)S(O)2CH2C(O)Me Pr-n
CH(Et)S(O)2CH2C(O)Me Pr-i
CH(Et)S(O)2CH2C(O)Me Pr-c
CH(Et)S(O)2CH2C(O)Me Bu-n
CH(Et)S(O)2CH2C(O)Me Bu-i
CH(Et)S(O)2CH2C(O)Me Bu-c
CH(Et)S(O)2CH2C(O)Me Bu-s
CH(Et)S(O)2CH2C(O)Me Bu-t
CH(Et)S(O)2CH2C(O)Me Pen-n
CH(Et)S(O)2CH2C(O)Me Pen-c
CH(Et)S(O)2CH2C(O)Me Hex-n
CH(Et)S(O)2CH2C(O)Me Hex-c
CH(Et)S(O)2CH2C(O)Me CH2Pr-c
CH(Et)S(O)2CH2C(O)Me CH2Bu-c
CH(Et)S(O)2CH2C(O)Me CH2Pen-c
CH(Et)S(O)2CH2C(O)Me CH2Hex-c
CH(Et)S(O)2CH2C(O)Me CH2CH=CH2
CH(Et)S(O)2CH2C(O)Me CH2CH=C(Cl)2
CH(Et)S(O)2CH2C(O)Me CH2C≡CH
CH(Et)S(O)2CH2C(O)Me CH2CN
CH(Et)S(O)2CH2C(O)Me CH2CF3
CH(Et)S(O)2CH2C(O)Me CH2OMe
CH(Et)S(O)2CH2C(O)Me CH2OCF3
CH(Et)S(O)2CH2C(O)Me CH2SMe
CH(Et)S(O)2CH2C(O)Me CH2S(O)Me
CH(Et)S(O)2CH2C(O)Me CH2S(O)2Me
CH(Et)S(O)2CH2C(O)Me CH2SCF3
CH(Et)S(O)2CH2C(O)Me CH2S(O)CF3
CH(Et)S(O)2CH2C(O)Me CH2S(O)2CF3
CH(Et)S(O)2CH2C(O)Me CH2CH(OMe)2
CH(Et)S(O)2CH2C(O)Me CH2CH(SMe)2
CH(Et)S(O)2CH2C(O)Me CH2C(O)Me
CH(Et)S(O)2CH2C(O)Me CH2C(O)CF3
CH(Et)S(O)2CH2C(O)Me CH2C(O)OMe
CH2SCH2C(O)NHMe Me
CH2SCH2C(O)NHEt Me
CH2SCH2C(O)NHPr-n Me
CH2SCH2C(O)NHPr-i Me
CH2SCH2C(O)NHPr-c Me
CH2SCH2C(O)NHBu-n Me
CH2SCH2C(O)NHBu-i Me
CH2SCH2C(O)NHBu-c Me
CH2SCH2C(O)NHBu-t Me
CH2SCH2C(O)NHPen-n Me
CH2SCH2C(O)NHPen-c Me
CH2SCH2C(O)NHHex-n Me
CH2SCH2C(O)NHHex-c Me
CH2SCH2C(O)N(Me)2 Me
CH2SCH2C(O)N(Et)2 Me
CH2SCH2C(O)NHMe Et
CH2SCH2C(O)NHMe Pr-n
CH2SCH2C(O)NHMe Pr-i
CH2SCH2C(O)NHMe Pr-c
CH2SCH2C(O)NHMe Bu-n
CH2SCH2C(O)NHMe Bu-i
CH2SCH2C(O)NHMe Bu-c
CH2SCH2C(O)NHMe Bu-s
CH2SCH2C(O)NHMe Bu-t
CH2SCH2C(O)NHMe Pen-n
CH2SCH2C(O)NHMe Pen-c
CH2SCH2C(O)NHMe Hex-n
CH2SCH2C(O)NHMe Hex-c
CH2SCH2C(O)NHMe CH2Pr-c
CH2SCH2C(O)NHMe CH2Bu-c
CH2SCH2C(O)NHMe CH2Pen-c
CH2SCH2C(O)NHMe CH2Hex-c
CH2SCH2C(O)NHMe CH2CH=CH2
CH2SCH2C(O)NHMe CH2CH=C(Cl)2
CH2SCH2C(O)NHMe CH2C≡CH
CH2SCH2C(O)NHMe CH2CN
CH2SCH2C(O)NHMe CH2CF3
CH2SCH2C(O)NHMe CH2OMe
CH2SCH2C(O)NHMe CH2OCF3
CH2SCH2C(O)NHMe CH2SMe
CH2SCH2C(O)NHMe CH2S(O)Me
CH2SCH2C(O)NHMe CH2S(O)2Me
CH2SCH2C(O)NHMe CH2SCF3
CH2SCH2C(O)NHMe CH2S(O)CF3
CH2SCH2C(O)NHMe CH2S(O)2CF3
CH2SCH2C(O)NHMe CH2CH(OMe)2
CH2SCH2C(O)NHMe CH2CH(SMe)2
CH2SCH2C(O)NHMe CH2C(O)Me
CH2SCH2C(O)NHMe CH2C(O)CF3
CH2SCH2C(O)NHMe CH2C(O)OMe
CH2S(O)CH2C(O)NHMe Me
CH2S(O)CH2C(O)NHEt Me
CH2S(O)CH2C(O)NHPr-n Me
CH2S(O)CH2C(O)NHPr-i Me
CH2S(O)CH2C(O)NHPr-c Me
CH2S(O)CH2C(O)NHBu-n Me
CH2S(O)CH2C(O)NHBu-i Me
CH2S(O)CH2C(O)NHBu-c Me
CH2S(O)CH2C(O)NHBu-t Me
CH2S(O)CH2C(O)NHPen-n Me
CH2S(O)CH2C(O)NHPen-c Me
CH2S(O)CH2C(O)NHHex-n Me
CH2S(O)CH2C(O)NHHex-c Me
CH2S(O)CH2C(O)N(Me)2 Me
CH2S(O)CH2C(O)N(Et)2 Me
CH2S(O)CH2C(O)NHMe Et
CH2S(O)CH2C(O)NHMe Pr-n
CH2S(O)CH2C(O)NHMe Pr-i
CH2S(O)CH2C(O)NHMe Pr-c
CH2S(O)CH2C(O)NHMe Bu-n
CH2S(O)CH2C(O)NHMe Bu-i
CH2S(O)CH2C(O)NHMe Bu-c
CH2S(O)CH2C(O)NHMe Bu-s
CH2S(O)CH2C(O)NHMe Bu-t
CH2S(O)CH2C(O)NHMe Pen-n
CH2S(O)CH2C(O)NHMe Pen-c
CH2S(O)CH2C(O)NHMe Hex-n
CH2S(O)CH2C(O)NHMe Hex-c
CH2S(O)CH2C(O)NHMe CH2Pr-c
CH2S(O)CH2C(O)NHMe CH2Bu-c
CH2S(O)CH2C(O)NHMe CH2Pen-c
CH2S(O)CH2C(O)NHMe CH2Hex-c
CH2S(O)CH2C(O)NHMe CH2CH=CH2
CH2S(O)CH2C(O)NHMe CH2CH=C(Cl)2
CH2S(O)CH2C(O)NHMe CH2C≡CH
CH2S(O)CH2C(O)NHMe CH2CN
CH2S(O)CH2C(O)NHMe CH2CF3
CH2S(O)CH2C(O)NHMe CH2OMe
CH2S(O)CH2C(O)NHMe CH2OCF3
CH2S(O)CH2C(O)NHMe CH2SMe
CH2S(O)CH2C(O)NHMe CH2S(O)Me
CH2S(O)CH2C(O)NHMe CH2S(O)2Me
CH2S(O)CH2C(O)NHMe CH2SCF3
CH2S(O)CH2C(O)NHMe CH2S(O)CF3
CH2S(O)CH2C(O)NHMe CH2S(O)2CF3
CH2S(O)CH2C(O)NHMe CH2CH(OMe)2
CH2S(O)CH2C(O)NHMe CH2CH(SMe)2
CH2S(O)CH2C(O)NHMe CH2C(O)Me
CH2S(O)CH2C(O)NHMe CH2C(O)CF3
CH2S(O)CH2C(O)NHMe CH2C(O)OMe
CH2S(O)2CH2C(O)NHMe Me
CH2S(O)2CH2C(O)NHMe Me
CH2S(O)2CH2C(O)NHEt Me
CH2S(O)2CH2C(O)NHPr-n Me
CH2S(O)2CH2C(O)NHPr-i Me
CH2S(O)2CH2C(O)NHPr-c Me
CH2S(O)2CH2C(O)NHBu-n Me
CH2S(O)2CH2C(O)NHBu-i Me
CH2S(O)2CH2C(O)NHBu-c Me
CH2S(O)2CH2C(O)NHBu-t Me
CH2S(O)2CH2C(O)NHPen-n Me
CH2S(O)2CH2C(O)NHPen-c Me
CH2S(O)2CH2C(O)NHHex-n Me
CH2S(O)2CH2C(O)NHHex-c Me
CH2S(O)2CH2C(O)N(Me)2 Me
CH2S(O)2CH2C(O)N(Et)2 Me
CH2S(O)2CH2C(O)NHMe Et
CH2S(O)2CH2C(O)NHMe Pr-n
CH2S(O)2CH2C(O)NHMe Pr-i
CH2S(O)2CH2C(O)NHMe Pr-c
CH2S(O)2CH2C(O)NHMe Bu-n
CH2S(O)2CH2C(O)NHMe Bu-i
CH2S(O)2CH2C(O)NHMe Bu-c
CH2S(O)2CH2C(O)NHMe Bu-s
CH2S(O)2CH2C(O)NHMe Bu-t
CH2S(O)2CH2C(O)NHMe Pen-n
CH2S(O)2CH2C(O)NHMe Pen-c
CH2S(O)2CH2C(O)NHMe Hex-n
CH2S(O)2CH2C(O)NHMe Hex-c
CH2S(O)2CH2C(O)NHMe CH2Pr-c
CH2S(O)2CH2C(O)NHMe CH2Bu-c
CH2S(O)2CH2C(O)NHMe CH2Pen-c
CH2S(O)2CH2C(O)NHMe CH2Hex-c
CH2S(O)2CH2C(O)NHMe CH2CH=CH2
CH2S(O)2CH2C(O)NHMe CH2CH=C(Cl)2
CH2S(O)2CH2C(O)NHMe CH2C≡CH
CH2S(O)2CH2C(O)NHMe CH2CN
CH2S(O)2CH2C(O)NHMe CH2CF3
CH2S(O)2CH2C(O)NHMe CH2OMe
CH2S(O)2CH2C(O)NHMe CH2OCF3
CH2S(O)2CH2C(O)NHMe CH2SMe
CH2S(O)2CH2C(O)NHMe CH2S(O)Me
CH2S(O)2CH2C(O)NHMe CH2S(O)2Me
CH2S(O)2CH2C(O)NHMe CH2SCF3
CH2S(O)2CH2C(O)NHMe CH2S(O)CF3
CH2S(O)2CH2C(O)NHMe CH2S(O)2CF3
CH2S(O)2CH2C(O)NHMe CH2CH(OMe)2
CH2S(O)2CH2C(O)NHMe CH2CH(SMe)2
CH2S(O)2CH2C(O)NHMe CH2C(O)Me
CH2S(O)2CH2C(O)NHMe CH2C(O)CF3
CH2S(O)2CH2C(O)NHMe CH2C(O)OMe
CH(Me)SCH2C(O)NHMe Me
CH(Me)SCH2C(O)NHEt Me
CH(Me)SCH2C(O)NHPr-n Me
CH(Me)SCH2C(O)NHPr-i Me
CH(Me)SCH2C(O)NHPr-c Me
CH(Me)SCH2C(O)NHBu-n Me
CH(Me)SCH2C(O)NHBu-i Me
CH(Me)SCH2C(O)NHBu-c Me
CH(Me)SCH2C(O)NHBu-t Me
CH(Me)SCH2C(O)NHPen-n Me
CH(Me)SCH2C(O)NHPen-c Me
CH(Me)SCH2C(O)NHHex-n Me
CH(Me)SCH2C(O)NHHex-c Me
CH(Me)SCH2C(O)N(Me)2 Me
CH(Me)SCH2C(O)N(Et)2 Me
CH(Me)SCH2C(O)NHMe Et
CH(Me)SCH2C(O)NHMe Pr-n
CH(Me)SCH2C(O)NHMe Pr-i
CH(Me)SCH2C(O)NHMe Pr-c
CH(Me)SCH2C(O)NHMe Bu-n
CH(Me)SCH2C(O)NHMe Bu-i
CH(Me)SCH2C(O)NHMe Bu-c
CH(Me)SCH2C(O)NHMe Bu-s
CH(Me)SCH2C(O)NHMe Bu-t
CH(Me)SCH2C(O)NHMe Pen-n
CH(Me)SCH2C(O)NHMe Pen-c
CH(Me)SCH2C(O)NHMe Hex-n
CH(Me)SCH2C(O)NHMe Hex-c
CH(Me)SCH2C(O)NHMe CH2Pr-c
CH(Me)SCH2C(O)NHMe CH2Bu-c
CH(Me)SCH2C(O)NHMe CH2Pen-c
CH(Me)SCH2C(O)NHMe CH2Hex-c
CH(Me)SCH2C(O)NHMe CH2CH=CH2
CH(Me)SCH2C(O)NHMe CH2CH=C(Cl)2
CH(Me)SCH2C(O)NHMe CH2C≡CH
CH(Me)SCH2C(O)NHMe CH2CN
CH(Me)SCH2C(O)NHMe CH2CF3
CH(Me)SCH2C(O)NHMe CH2OMe
CH(Me)SCH2C(O)NHMe CH2OCF3
CH(Me)SCH2C(O)NHMe CH2SMe
CH(Me)SCH2C(O)NHMe CH2S(O)Me
CH(Me)SCH2C(O)NHMe CH2S(O)2Me
CH(Me)SCH2C(O)NHMe CH2SCF3
CH(Me)SCH2C(O)NHMe CH2S(O)CF3
CH(Me)SCH2C(O)NHMe CH2S(O)2CF3
CH(Me)SCH2C(O)NHMe CH2CH(OMe)2
CH(Me)SCH2C(O)NHMe CH2CH(SMe)2
CH(Me)SCH2C(O)NHMe CH2C(O)Me
CH(Me)SCH2C(O)NHMe CH2C(O)CF3
CH(Me)SCH2C(O)NHMe CH2C(O)OMe
CH(Me)S(O)CH2C(O)NHMe Me
CH(Me)S(O)CH2C(O)NHEt Me
CH(Me)S(O)CH2C(O)NHPr-n Me
CH(Me)S(O)CH2C(O)NHPr-i Me
CH(Me)S(O)CH2C(O)NHPr-c Me
CH(Me)S(O)CH2C(O)NHBu-n Me
CH(Me)S(O)CH2C(O)NHBu-i Me
CH(Me)S(O)CH2C(O)NHBu-c Me
CH(Me)S(O)CH2C(O)NHBu-t Me
CH(Me)S(O)CH2C(O)NHPen-n Me
CH(Me)S(O)CH2C(O)NHPen-c Me
CH(Me)S(O)CH2C(O)NHHex-n Me
CH(Me)S(O)CH2C(O)NHHex-c Me
CH(Et)S(O)CH2C(O)N(Me)2 Me
CH(Et)S(O)CH2C(O)N(Et)2 Me
CH(Me)S(O)CH2C(O)NHMe Et
CH(Me)S(O)CH2C(O)NHMe Pr-n
CH(Me)S(O)CH2C(O)NHMe Pr-i
CH(Me)S(O)CH2C(O)NHMe Pr-c
CH(Me)S(O)CH2C(O)NHMe Bu-n
CH(Me)S(O)CH2C(O)NHMe Bu-i
CH(Me)S(O)CH2C(O)NHMe Bu-c
CH(Me)S(O)CH2C(O)NHMe Bu-s
CH(Me)S(O)CH2C(O)NHMe Bu-t
CH(Me)S(O)CH2C(O)NHMe Pen-n
CH(Me)S(O)CH2C(O)NHMe Pen-c
CH(Me)S(O)CH2C(O)NHMe Hex-n
CH(Me)S(O)CH2C(O)NHMe Hex-c
CH(Me)S(O)CH2C(O)NHMe CH2Pr-c
CH(Me)S(O)CH2C(O)NHMe CH2Bu-c
CH(Me)S(O)CH2C(O)NHMe CH2Pen-c
CH(Me)S(O)CH2C(O)NHMe CH2Hex-c
CH(Me)S(O)CH2C(O)NHMe CH2CH=CH2
CH(Me)S(O)CH2C(O)NHMe CH2CH=C(Cl)2
CH(Me)S(O)CH2C(O)NHMe CH2C≡CH
CH(Me)S(O)CH2C(O)NHMe CH2CN
CH(Me)S(O)CH2C(O)NHMe CH2CF3
CH(Me)S(O)CH2C(O)NHMe CH2OMe
CH(Me)S(O)CH2C(O)NHMe CH2OCF3
CH(Me)S(O)CH2C(O)NHMe CH2SMe
CH(Me)S(O)CH2C(O)NHMe CH2S(O)Me
CH(Me)S(O)CH2C(O)NHMe CH2S(O)2Me
CH(Me)S(O)CH2C(O)NHMe CH2SCF3
CH(Me)S(O)CH2C(O)NHMe CH2S(O)CF3
CH(Me)S(O)CH2C(O)NHMe CH2S(O)2CF3
CH(Me)S(O)CH2C(O)NHMe CH2CH(OMe)2
CH(Me)S(O)CH2C(O)NHMe CH2CH(SMe)2
CH(Me)S(O)CH2C(O)NHMe CH2C(O)Me
CH(Me)S(O)CH2C(O)NHMe CH2C(O)CF3
CH(Me)S(O)CH2C(O)NHMe CH2C(O)OMe
CH(Me)S(O)2CH2C(O)NHMe Me
CH(Me)S(O)2CH2C(O)NHEt Me
CH(Me)S(O)2CH2C(O)NHPr-n Me
CH(Me)S(O)2CH2C(O)NHPr-i Me
CH(Me)S(O)2CH2C(O)NHPr-c Me
CH(Me)S(O)2CH2C(O)NHBu-n Me
CH(Me)S(O)2CH2C(O)NHBu-i Me
CH(Me)S(O)2CH2C(O)NHBu-c Me
CH(Me)S(O)2CH2C(O)NHBu-t Me
CH(Me)S(O)2CH2C(O)NHPen-n Me
CH(Me)S(O)2CH2C(O)NHPen-c Me
CH(Me)S(O)2CH2C(O)NHHex-n Me
CH(Me)S(O)2CH2C(O)NHHex-c Me
CH(Me)S(O)2CH2C(O)N(Me)2 Me
CH(Me)S(O)2CH2C(O)N(Et)2 Me
CH(Me)S(O)2CH2C(O)NHMe Et
CH(Me)S(O)2CH2C(O)NHMe Pr-n
CH(Me)S(O)2CH2C(O)NHMe Pr-i
CH(Me)S(O)2CH2C(O)NHMe Pr-c
CH(Me)S(O)2CH2C(O)NHMe Bu-n
CH(Me)S(O)2CH2C(O)NHMe Bu-i
CH(Me)S(O)2CH2C(O)NHMe Bu-c
CH(Me)S(O)2CH2C(O)NHMe Bu-s
CH(Me)S(O)2CH2C(O)NHMe Bu-t
CH(Me)S(O)2CH2C(O)NHMe Pen-n
CH(Me)S(O)2CH2C(O)NHMe Pen-c
CH(Me)S(O)2CH2C(O)NHMe Hex-n
CH(Me)S(O)2CH2C(O)NHMe Hex-c
CH(Me)S(O)2CH2C(O)NHMe CH2Pr-c
CH(Me)S(O)2CH2C(O)NHMe CH2Bu-c
CH(Me)S(O)2CH2C(O)NHMe CH2Pen-c
CH(Me)S(O)2CH2C(O)NHMe CH2Hex-c
CH(Me)S(O)2CH2C(O)NHMe CH2CH=CH2
CH(Me)S(O)2CH2C(O)NHMe CH2CH=C(Cl)2
CH(Me)S(O)2CH2C(O)NHMe CH2C≡CH
CH(Me)S(O)2CH2C(O)NHMe CH2CN
CH(Me)S(O)2CH2C(O)NHMe CH2CF3
CH(Me)S(O)2CH2C(O)NHMe CH2OMe
CH(Me)S(O)2CH2C(O)NHMe CH2OCF3
CH(Me)S(O)2CH2C(O)NHMe CH2SMe
CH(Me)S(O)2CH2C(O)NHMe CH2S(O)Me
CH(Me)S(O)2CH2C(O)NHMe CH2S(O)2Me
CH(Me)S(O)2CH2C(O)NHMe CH2SCF3
CH(Me)S(O)2CH2C(O)NHMe CH2S(O)CF3
CH(Me)S(O)2CH2C(O)NHMe CH2S(O)2CF3
CH(Me)S(O)2CH2C(O)NHMe CH2CH(OMe)2
CH(Me)S(O)2CH2C(O)NHMe CH2CH(SMe)2
CH(Me)S(O)2CH2C(O)NHMe CH2C(O)Me
CH(Me)S(O)2CH2C(O)NHMe CH2C(O)CF3
CH(Me)S(O)2CH2C(O)NHMe CH2C(O)OMe
CH(Et)SCH2C(O)NHMe Me
CH(Et)SCH2C(O)NHEt Me
CH(Et)SCH2C(O)NHPr-n Me
CH(Et)SCH2C(O)NHPr-i Me
CH(Et)SCH2C(O)NHPr-c Me
CH(Et)SCH2C(O)NHBu-n Me
CH(Et)SCH2C(O)NHBu-i Me
CH(Et)SCH2C(O)NHBu-c Me
CH(Et)SCH2C(O)NHBu-t Me
CH(Et)SCH2C(O)NHPen-n Me
CH(Et)SCH2C(O)NHPen-c Me
CH(Et)SCH2C(O)NHHex-n Me
CH(Et)SCH2C(O)NHHex-c Me
CH(Et)SCH2C(O)N(Me)2 Me
CH(Et)SCH2C(O)N(Et)2 Me
CH(Et)SCH2C(O)NHMe Et
CH(Et)SCH2C(O)NHMe Pr-n
CH(Et)SCH2C(O)NHMe Pr-i
CH(Et)SCH2C(O)NHMe Pr-c
CH(Et)SCH2C(O)NHMe Bu-n
CH(Et)SCH2C(O)NHMe Bu-i
CH(Et)SCH2C(O)NHMe Bu-c
CH(Et)SCH2C(O)NHMe Bu-s
CH(Et)SCH2C(O)NHMe Bu-t
CH(Et)SCH2C(O)NHMe Pen-n
CH(Et)SCH2C(O)NHMe Pen-c
CH(Et)SCH2C(O)NHMe Hex-n
CH(Et)SCH2C(O)NHMe Hex-c
CH(Et)SCH2C(O)NHMe CH2Pr-c
CH(Et)SCH2C(O)NHMe CH2Bu-c
CH(Et)SCH2C(O)NHMe CH2Pen-c
CH(Et)SCH2C(O)NHMe CH2Hex-c
CH(Et)SCH2C(O)NHMe CH2CH=CH2
CH(Et)SCH2C(O)NHMe CH2CH=C(Cl)2
CH(Et)SCH2C(O)NHMe CH2C≡CH
CH(Et)SCH2C(O)NHMe CH2CN
CH(Et)SCH2C(O)NHMe CH2CF3
CH(Et)SCH2C(O)NHMe CH2OMe
CH(Et)SCH2C(O)NHMe CH2OCF3
CH(Et)SCH2C(O)NHMe CH2SMe
CH(Et)SCH2C(O)NHMe CH2S(O)Me
CH(Et)SCH2C(O)NHMe CH2S(O)2Me
CH(Et)SCH2C(O)NHMe CH2SCF3
CH(Et)SCH2C(O)NHMe CH2S(O)CF3
CH(Et)SCH2C(O)NHMe CH2S(O)2CF3
CH(Et)SCH2C(O)NHMe CH2CH(OMe)2
CH(Et)SCH2C(O)NHMe CH2CH(SMe)2
CH(Et)SCH2C(O)NHMe CH2C(O)Me
CH(Et)SCH2C(O)NHMe CH2C(O)CF3
CH(Et)SCH2C(O)NHMe CH2C(O)OMe
CH(Et)S(O)CH2C(O)NHMe Me
CH(Et)S(O)CH2C(O)NHEt Me
CH(Et)S(O)CH2C(O)NHPr-n Me
CH(Et)S(O)CH2C(O)NHPr-i Me
CH(Et)S(O)CH2C(O)NHPr-c Me
CH(Et)S(O)CH2C(O)NHBu-n Me
CH(Et)S(O)CH2C(O)NHBu-i Me
CH(Et)S(O)CH2C(O)NHBu-c Me
CH(Et)S(O)CH2C(O)NHBu-t Me
CH(Et)S(O)CH2C(O)NHPen-n Me
CH(Et)S(O)CH2C(O)NHPen-c Me
CH(Et)S(O)CH2C(O)NHHex-n Me
CH(Et)S(O)CH2C(O)NHHex-c Me
CH(Et)S(O)CH2C(O)N(Me)2 Me
CH(Et)S(O)CH2C(O)N(Et)2 Me
CH(Et)S(O)CH2C(O)NHMe Et
CH(Et)S(O)CH2C(O)NHMe Pr-n
CH(Et)S(O)CH2C(O)NHMe Pr-i
CH(Et)S(O)CH2C(O)NHMe Pr-c
CH(Et)S(O)CH2C(O)NHMe Bu-n
CH(Et)S(O)CH2C(O)NHMe Bu-i
CH(Et)S(O)CH2C(O)NHMe Bu-c
CH(Et)S(O)CH2C(O)NHMe Bu-s
CH(Et)S(O)CH2C(O)NHMe Bu-t
CH(Et)S(O)CH2C(O)NHMe Pen-n
CH(Et)S(O)CH2C(O)NHMe Pen-c
CH(Et)S(O)CH2C(O)NHMe Hex-n
CH(Et)S(O)CH2C(O)NHMe Hex-c
CH(Et)S(O)CH2C(O)NHMe CH2Pr-c
CH(Et)S(O)CH2C(O)NHMe CH2Bu-c
CH(Et)S(O)CH2C(O)NHMe CH2Pen-c
CH(Et)S(O)CH2C(O)NHMe CH2Hex-c
CH(Et)S(O)CH2C(O)NHMe CH2CH=CH2
CH(Et)S(O)CH2C(O)NHMe CH2CH=C(Cl)2
CH(Et)S(O)CH2C(O)NHMe CH2C≡CH
CH(Et)S(O)CH2C(O)NHMe CH2CN
CH(Et)S(O)CH2C(O)NHMe CH2CF3
CH(Et)S(O)CH2C(O)NHMe CH2OMe
CH(Et)S(O)CH2C(O)NHMe CH2OCF3
CH(Et)S(O)CH2C(O)NHMe CH2SMe
CH(Et)S(O)CH2C(O)NHMe CH2S(O)Me
CH(Et)S(O)CH2C(O)NHMe CH2S(O)2Me
CH(Et)S(O)CH2C(O)NHMe CH2SCF3
CH(Et)S(O)CH2C(O)NHMe CH2S(O)CF3
CH(Et)S(O)CH2C(O)NHMe CH2S(O)2CF3
CH(Et)S(O)CH2C(O)NHMe CH2CH(OMe)2
CH(Et)S(O)CH2C(O)NHMe CH2CH(SMe)2
CH(Et)S(O)CH2C(O)NHMe CH2C(O)Me
CH(Et)S(O)CH2C(O)NHMe CH2C(O)CF3
CH(Et)S(O)CH2C(O)NHMe CH2C(O)OMe
CH(Et)S(O)2CH2C(O)NHMe Me
CH(Et)S(O)2CH2C(O)NHEt Me
CH(Et)S(O)2CH2C(O)NHPr-n Me
CH(Et)S(O)2CH2C(O)NHPr-i Me
CH(Et)S(O)2CH2C(O)NHPr-c Me
CH(Et)S(O)2CH2C(O)NHBu-n Me
CH(Et)S(O)2CH2C(O)NHBu-i Me
CH(Et)S(O)2CH2C(O)NHBu-c Me
CH(Et)S(O)2CH2C(O)NHBu-t Me
CH(Et)S(O)2CH2C(O)NHPen-n Me
CH(Et)S(O)2CH2C(O)NHPen-c Me
CH(Et)S(O)2CH2C(O)NHHex-n Me
CH(Et)S(O)2CH2C(O)NHHex-c Me
CH(Et)S(O)2CH2C(O)N(Me)2 Me
CH(Et)S(O)2CH2C(O)N(Et)2 Me
CH(Et)S(O)2CH2C(O)NHMe Et
CH(Et)S(O)2CH2C(O)NHMe Pr-n
CH(Et)S(O)2CH2C(O)NHMe Pr-i
CH(Et)S(O)2CH2C(O)NHMe Pr-c
CH(Et)S(O)2CH2C(O)NHMe Bu-n
CH(Et)S(O)2CH2C(O)NHMe Bu-i
CH(Et)S(O)2CH2C(O)NHMe Bu-c
CH(Et)S(O)2CH2C(O)NHMe Bu-s
CH(Et)S(O)2CH2C(O)NHMe Bu-t
CH(Et)S(O)2CH2C(O)NHMe Pen-n
CH(Et)S(O)2CH2C(O)NHMe Pen-c
CH(Et)S(O)2CH2C(O)NHMe Hex-n
CH(Et)S(O)2CH2C(O)NHMe Hex-c
CH(Et)S(O)2CH2C(O)NHMe CH2Pr-c
CH(Et)S(O)2CH2C(O)NHMe CH2Bu-c
CH(Et)S(O)2CH2C(O)NHMe CH2Pen-c
CH(Et)S(O)2CH2C(O)NHMe CH2Hex-c
CH(Et)S(O)2CH2C(O)NHMe CH2CH=CH2
CH(Et)S(O)2CH2C(O)NHMe CH2CH=C(Cl)2
CH(Et)S(O)2CH2C(O)NHMe CH2C≡CH
CH(Et)S(O)2CH2C(O)NHMe CH2CN
CH(Et)S(O)2CH2C(O)NHMe CH2CF3
CH(Et)S(O)2CH2C(O)NHMe CH2OMe
CH(Et)S(O)2CH2C(O)NHMe CH2OCF3
CH(Et)S(O)2CH2C(O)NHMe CH2SMe
CH(Et)S(O)2CH2C(O)NHMe CH2S(O)Me
CH(Et)S(O)2CH2C(O)NHMe CH2S(O)2Me
CH(Et)S(O)2CH2C(O)NHMe CH2SCF3
CH(Et)S(O)2CH2C(O)NHMe CH2S(O)CF3
CH(Et)S(O)2CH2C(O)NHMe CH2S(O)2CF3
CH(Et)S(O)2CH2C(O)NHMe CH2CH(OMe)2
CH(Et)S(O)2CH2C(O)NHMe CH2CH(SMe)2
CH(Et)S(O)2CH2C(O)NHMe CH2C(O)Me
CH(Et)S(O)2CH2C(O)NHMe CH2C(O)CF3
CH(Et)S(O)2CH2C(O)NHMe CH2C(O)OMe
CH2SCH(Me)C(O)OMe Me
CH2SCH(Me)C(O)OEt Me
CH2SCH(Me)C(O)OPr-n Me
CH2SCH(Me)C(O)OPr-i Me
CH2SCH(Me)C(O)OBu-n Me
CH2SCH(Me)C(O)OBu-i Me
CH2SCH(Me)C(O)OBu-t Me
CH2SCH(Me)C(O)OPen-n Me
CH2SCH(Me)C(O)OHex-n Me
CH2SCH(Me)C(O)OMe Et
CH2SCH(Me)C(O)OMe Pr-n
CH2SCH(Me)C(O)OMe Pr-i
CH2SCH(Me)C(O)OMe Pr-c
CH2SCH(Me)C(O)OMe Bu-n
CH2SCH(Me)C(O)OMe Bu-i
CH2SCH(Me)C(O)OMe Bu-c
CH2SCH(Me)C(O)OMe Bu-s
CH2SCH(Me)C(O)OMe Bu-t
CH2SCH(Me)C(O)OMe Pen-n
CH2SCH(Me)C(O)OMe Pen-c
CH2SCH(Me)C(O)OMe Hex-n
CH2SCH(Me)C(O)OMe Hex-c
CH2SCH(Me)C(O)OMe CH2Pr-c
CH2SCH(Me)C(O)OMe CH2Bu-c
CH2SCH(Me)C(O)OMe CH2Pen-c
CH2SCH(Me)C(O)OMe CH2Hex-c
CH2SCH(Me)C(O)OMe CH2CH=CH2
CH2SCH(Me)C(O)OMe CH2CH=C(Cl)2
CH2SCH(Me)C(O)OMe CH2C≡CH
CH2SCH(Me)C(O)OMe CH2CN
CH2SCH(Me)C(O)OMe CH2CF3
CH2SCH(Me)C(O)OMe CH2OMe
CH2SCH(Me)C(O)OMe CH2OCF3
CH2SCH(Me)C(O)OMe CH2SMe
CH2SCH(Me)C(O)OMe CH2S(O)Me
CH2SCH(Me)C(O)OMe CH2S(O)2Me
CH2SCH(Me)C(O)OMe CH2SCF3
CH2SCH(Me)C(O)OMe CH2S(O)CF3
CH2SCH(Me)C(O)OMe CH2S(O)2CF3
CH2SCH(Me)C(O)OMe CH2CH(OMe)2
CH2SCH(Me)C(O)OMe CH2CH(SMe)2
CH2SCH(Me)C(O)OMe CH2C(O)Me
CH2SCH(Me)C(O)OMe CH2C(O)CF3
CH2SCH(Me)C(O)OMe CH2C(O)OMe
CH2S(O)CH(Me)C(O)OMe Me
CH2S(O)CH(Me)C(O)OEt Me
CH2S(O)CH(Me)C(O)OPr-n Me
CH2S(O)CH(Me)C(O)OPr-i Me
CH2S(O)CH(Me)C(O)OBu-n Me
CH2S(O)CH(Me)C(O)OBu-i Me
CH2S(O)CH(Me)C(O)OBu-t Me
CH2S(O)CH(Me)C(O)OPen-n Me
CH2S(O)CH(Me)C(O)OHex-n Me
CH2S(O)CH(Me)C(O)OMe Et
CH2S(O)CH(Me)C(O)OMe Pr-n
CH2S(O)CH(Me)C(O)OMe Pr-i
CH2S(O)CH(Me)C(O)OMe Pr-c
CH2S(O)CH(Me)C(O)OMe Bu-n
CH2S(O)CH(Me)C(O)OMe Bu-i
CH2S(O)CH(Me)C(O)OMe Bu-c
CH2S(O)CH(Me)C(O)OMe Bu-s
CH2S(O)CH(Me)C(O)OMe Bu-t
CH2S(O)CH(Me)C(O)OMe Pen-n
CH2S(O)CH(Me)C(O)OMe Pen-c
CH2S(O)CH(Me)C(O)OMe Hex-n
CH2S(O)CH(Me)C(O)OMe Hex-c
CH2S(O)CH(Me)C(O)OMe CH2Pr-c
CH2S(O)CH(Me)C(O)OMe CH2Bu-c
CH2S(O)CH(Me)C(O)OMe CH2Pen-c
CH2S(O)CH(Me)C(O)OMe CH2Hex-c
CH2S(O)CH(Me)C(O)OMe CH2CH=CH2
CH2S(O)CH(Me)C(O)OMe CH2CH=C(Cl)2
CH2S(O)CH(Me)C(O)OMe CH2C≡CH
CH2S(O)CH(Me)C(O)OMe CH2CN
CH2S(O)CH(Me)C(O)OMe CH2CF3
CH2S(O)CH(Me)C(O)OMe CH2OMe
CH2S(O)CH(Me)C(O)OMe CH2OCF3
CH2S(O)CH(Me)C(O)OMe CH2SMe
CH2S(O)CH(Me)C(O)OMe CH2S(O)Me
CH2S(O)CH(Me)C(O)OMe CH2S(O)2Me
CH2S(O)CH(Me)C(O)OMe CH2SCF3
CH2S(O)CH(Me)C(O)OMe CH2S(O)CF3
CH2S(O)CH(Me)C(O)OMe CH2S(O)2CF3
CH2S(O)CH(Me)C(O)OMe CH2CH(OMe)2
CH2S(O)CH(Me)C(O)OMe CH2CH(SMe)2
CH2S(O)CH(Me)C(O)OMe CH2C(O)Me
CH2S(O)CH(Me)C(O)OMe CH2C(O)CF3
CH2S(O)CH(Me)C(O)OMe CH2C(O)OMe
CH2S(O)2CH(Me)C(O)OMe Me
CH2S(O)2CH(Me)C(O)OEt Me
CH2S(O)2CH(Me)C(O)OPr-n Me
CH2S(O)2CH(Me)C(O)OPr-i Me
CH2S(O)2CH(Me)C(O)OBu-n Me
CH2S(O)2CH(Me)C(O)OBu-i Me
CH2S(O)2CH(Me)C(O)OBu-t Me
CH2S(O)2CH(Me)C(O)OPen-n Me
CH2S(O)2CH(Me)C(O)OHex-n Me
CH2S(O)2CH(Me)C(O)OMe Et
CH2S(O)2CH(Me)C(O)OMe Pr-n
CH2S(O)2CH(Me)C(O)OMe Pr-i
CH2S(O)2CH(Me)C(O)OMe Pr-c
CH2S(O)2CH(Me)C(O)OMe Bu-n
CH2S(O)2CH(Me)C(O)OMe Bu-i
CH2S(O)2CH(Me)C(O)OMe Bu-c
CH2S(O)2CH(Me)C(O)OMe Bu-s
CH2S(O)2CH(Me)C(O)OMe Bu-t
CH2S(O)2CH(Me)C(O)OMe Pen-n
CH2S(O)2CH(Me)C(O)OMe Pen-c
CH2S(O)2CH(Me)C(O)OMe Hex-n
CH2S(O)2CH(Me)C(O)OMe Hex-c
CH2S(O)2CH(Me)C(O)OMe CH2Pr-c
CH2S(O)2CH(Me)C(O)OMe CH2Bu-c
CH2S(O)2CH(Me)C(O)OMe CH2Pen-c
CH2S(O)2CH(Me)C(O)OMe CH2Hex-c
CH2S(O)2CH(Me)C(O)OMe CH2CH=CH2
CH2S(O)2CH(Me)C(O)OMe CH2CH=C(Cl)2
CH2S(O)2CH(Me)C(O)OMe CH2C≡CH
CH2S(O)2CH(Me)C(O)OMe CH2CN
CH2S(O)2CH(Me)C(O)OMe CH2CF3
CH2S(O)2CH(Me)C(O)OMe CH2OMe
CH2S(O)2CH(Me)C(O)OMe CH2OCF3
CH2S(O)2CH(Me)C(O)OMe CH2SMe
CH2S(O)2CH(Me)C(O)OMe CH2S(O)Me
CH2S(O)2CH(Me)C(O)OMe CH2S(O)2Me
CH2S(O)2CH(Me)C(O)OMe CH2SCF3
CH2S(O)2CH(Me)C(O)OMe CH2S(O)CF3
CH2S(O)2CH(Me)C(O)OMe CH2S(O)2CF3
CH2S(O)2CH(Me)C(O)OMe CH2CH(OMe)2
CH2S(O)2CH(Me)C(O)OMe CH2CH(SMe)2
CH2S(O)2CH(Me)C(O)OMe CH2C(O)Me
CH2S(O)2CH(Me)C(O)OMe CH2C(O)CF3
CH2S(O)2CH(Me)C(O)OMe CH2C(O)OMe
CH(Me)SCH(Me)C(O)OMe Me
CH(Me)SCH(Me)C(O)OEt Me
CH(Me)SCH(Me)C(O)OPr-n Me
CH(Me)SCH(Me)C(O)OPr-i Me
CH(Me)SCH(Me)C(O)OBu-n Me
CH(Me)SCH(Me)C(O)OBu-i Me
CH(Me)SCH(Me)C(O)OBu-t Me
CH(Me)SCH(Me)C(O)OPen-n Me
CH(Me)SCH(Me)C(O)OHex-n Me
CH(Me)SCH(Me)C(O)OMe Et
CH(Me)SCH(Me)C(O)OMe Pr-n
CH(Me)SCH(Me)C(O)OMe Pr-i
CH(Me)SCH(Me)C(O)OMe Pr-c
CH(Me)SCH(Me)C(O)OMe Bu-n
CH(Me)SCH(Me)C(O)OMe Bu-i
CH(Me)SCH(Me)C(O)OMe Bu-c
CH(Me)SCH(Me)C(O)OMe Bu-s
CH(Me)SCH(Me)C(O)OMe Bu-t
CH(Me)SCH(Me)C(O)OMe Pen-n
CH(Me)SCH(Me)C(O)OMe Pen-c
CH(Me)SCH(Me)C(O)OMe Hex-n
CH(Me)SCH(Me)C(O)OMe Hex-c
CH(Me)SCH(Me)C(O)OMe CH2Pr-c
CH(Me)SCH(Me)C(O)OMe CH2Bu-c
CH(Me)SCH(Me)C(O)OMe CH2Pen-c
CH(Me)SCH(Me)C(O)OMe CH2Hex-c
CH(Me)SCH(Me)C(O)OMe CH2CH=CH2
CH(Me)SCH(Me)C(O)OMe CH2CH=C(Cl)2
CH(Me)SCH(Me)C(O)OMe CH2C≡CH
CH(Me)SCH(Me)C(O)OMe CH2CN
CH(Me)SCH(Me)C(O)OMe CH2CF3
CH(Me)SCH(Me)C(O)OMe CH2OMe
CH(Me)SCH(Me)C(O)OMe CH2OCF3
CH(Me)SCH(Me)C(O)OMe CH2SMe
CH(Me)SCH(Me)C(O)OMe CH2S(O)Me
CH(Me)SCH(Me)C(O)OMe CH2S(O)2Me
CH(Me)SCH(Me)C(O)OMe CH2SCF3
CH(Me)SCH(Me)C(O)OMe CH2S(O)CF3
CH(Me)SCH(Me)C(O)OMe CH2S(O)2CF3
CH(Me)SCH(Me)C(O)OMe CH2CH(OMe)2
CH(Me)SCH(Me)C(O)OMe CH2CH(SMe)2
CH(Me)SCH(Me)C(O)OMe CH2C(O)Me
CH(Me)SCH(Me)C(O)OMe CH2C(O)CF3
CH(Me)SCH(Me)C(O)OMe CH2C(O)OMe
CH(Me)S(O)CH(Me)C(O)OMe Me
CH(Me)S(O)CH(Me)C(O)OEt Me
CH(Me)S(O)CH(Me)C(O)OPr-n Me
CH(Me)S(O)CH(Me)C(O)OPr-i Me
CH(Me)S(O)CH(Me)C(O)OBu-n Me
CH(Me)S(O)CH(Me)C(O)OBu-i Me
CH(Me)S(O)CH(Me)C(O)OBu-t Me
CH(Me)S(O)CH(Me)C(O)OPen-n Me
CH(Me)S(O)CH(Me)C(O)OHex-n Me
CH(Me)S(O)CH(Me)C(O)OMe Et
CH(Me)S(O)CH(Me)C(O)OMe Pr-n
CH(Me)S(O)CH(Me)C(O)OMe Pr-i
CH(Me)S(O)CH(Me)C(O)OMe Pr-c
CH(Me)S(O)CH(Me)C(O)OMe Bu-n
CH(Me)S(O)CH(Me)C(O)OMe Bu-i
CH(Me)S(O)CH(Me)C(O)OMe Bu-c
CH(Me)S(O)CH(Me)C(O)OMe Bu-s
CH(Me)S(O)CH(Me)C(O)OMe Bu-t
CH(Me)S(O)CH(Me)C(O)OMe Pen-n
CH(Me)S(O)CH(Me)C(O)OMe Pen-c
CH(Me)S(O)CH(Me)C(O)OMe Hex-n
CH(Me)S(O)CH(Me)C(O)OMe Hex-c
CH(Me)S(O)CH(Me)C(O)OMe CH2Pr-c
CH(Me)S(O)CH(Me)C(O)OMe CH2Bu-c
CH(Me)S(O)CH(Me)C(O)OMe CH2Pen-c
CH(Me)S(O)CH(Me)C(O)OMe CH2Hex-c
CH(Me)S(O)CH(Me)C(O)OMe CH2CH=CH2
CH(Me)S(O)CH(Me)C(O)OMe CH2CH=C(Cl)2
CH(Me)S(O)CH(Me)C(O)OMe CH2C≡CH
CH(Me)S(O)CH(Me)C(O)OMe CH2CN
CH(Me)S(O)CH(Me)C(O)OMe CH2CF3
CH(Me)S(O)CH(Me)C(O)OMe CH2OMe
CH(Me)S(O)CH(Me)C(O)OMe CH2OCF3
CH(Me)S(O)CH(Me)C(O)OMe CH2SMe
CH(Me)S(O)CH(Me)C(O)OMe CH2S(O)Me
CH(Me)S(O)CH(Me)C(O)OMe CH2S(O)2Me
CH(Me)S(O)CH(Me)C(O)OMe CH2SCF3
CH(Me)S(O)CH(Me)C(O)OMe CH2S(O)CF3
CH(Me)S(O)CH(Me)C(O)OMe CH2S(O)2CF3
CH(Me)S(O)CH(Me)C(O)OMe CH2CH(OMe)2
CH(Me)S(O)CH(Me)C(O)OMe CH2CH(SMe)2
CH(Me)S(O)CH(Me)C(O)OMe CH2C(O)Me
CH(Me)S(O)CH(Me)C(O)OMe CH2C(O)CF3
CH(Me)S(O)CH(Me)C(O)OMe CH2C(O)OMe
CH(Me)S(O)2CH(Me)C(O)OMe Me
CH(Me)S(O)2CH(Me)C(O)OEt Me
CH(Me)S(O)2CH(Me)C(O)OPr-n Me
CH(Me)S(O)2CH(Me)C(O)OPr-i Me
CH(Me)S(O)2CH(Me)C(O)OBu-n Me
CH(Me)S(O)2CH(Me)C(O)OBu-i Me
CH(Me)S(O)2CH(Me)C(O)OBu-t Me
CH(Me)S(O)2CH(Me)C(O)OPen-n Me
CH(Me)S(O)2CH(Me)C(O)OMe Et
CH(Me)S(O)2CH(Me)C(O)OMe Pr-n
CH(Me)S(O)2CH(Me)C(O)OMe Pr-i
CH(Me)S(O)2CH(Me)C(O)OMe Pr-c
CH(Me)S(O)2CH(Me)C(O)OMe Bu-n
CH(Me)S(O)2CH(Me)C(O)OMe Bu-i
CH(Me)S(O)2CH(Me)C(O)OMe Bu-c
CH(Me)S(O)2CH(Me)C(O)OMe Bu-s
CH(Me)S(O)2CH(Me)C(O)OMe Bu-t
CH(Me)S(O)2CH(Me)C(O)OMe Pen-n
CH(Me)S(O)2CH(Me)C(O)OMe Pen-c
CH(Me)S(O)2CH(Me)C(O)OMe Hex-n
CH(Me)S(O)2CH(Me)C(O)OMe Hex-c
CH(Me)S(O)2CH(Me)C(O)OMe CH2Pr-c
CH(Me)S(O)2CH(Me)C(O)OMe CH2Bu-c
CH(Me)S(O)2CH(Me)C(O)OMe CH2Pen-c
CH(Me)S(O)2CH(Me)C(O)OMe CH2Hex-c
CH(Me)S(O)2CH(Me)C(O)OMe CH2CH=CH2
CH(Me)S(O)2CH(Me)C(O)OMe CH2CH=C(Cl)2
CH(Me)S(O)2CH(Me)C(O)OMe CH2C≡CH
CH(Me)S(O)2CH(Me)C(O)OMe CH2CN
CH(Me)S(O)2CH(Me)C(O)OMe CH2CF3
CH(Me)S(O)2CH(Me)C(O)OMe CH2OMe
CH(Me)S(O)2CH(Me)C(O)OMe CH2OCF3
CH(Me)S(O)2CH(Me)C(O)OMe CH2SMe
CH(Me)S(O)2CH(Me)C(O)OMe CH2S(O)Me
CH(Me)S(O)2CH(Me)C(O)OMe CH2S(O)2Me
CH(Me)S(O)2CH(Me)C(O)OMe CH2SCF3
CH(Me)S(O)2CH(Me)C(O)OMe CH2S(O)CF3
CH(Me)S(O)2CH(Me)C(O)OMe CH2S(O)2CF3
CH(Me)S(O)2CH(Me)C(O)OMe CH2CH(OMe)2
CH(Me)S(O)2CH(Me)C(O)OMe CH2CH(SMe)2
CH(Me)S(O)2CH(Me)C(O)OMe CH2C(O)Me
CH(Me)S(O)2CH(Me)C(O)OMe CH2C(O)CF3
CH(Me)S(O)2CH(Me)C(O)OMe CH2C(O)OMe
CH(Et)SCH(Me)C(O)OMe Me
CH(Et)SCH(Me)C(O)OEt Me
CH(Et)SCH(Me)C(O)OPr-n Me
CH(Et)SCH(Me)C(O)OPr-i Me
CH(Et)SCH(Me)C(O)OBu-n Me
CH(Et)SCH(Me)C(O)OBu-i Me
CH(Et)SCH(Me)C(O)OBu-t Me
CH(Et)SCH(Me)C(O)OPen-n Me
CH(Et)SCH(Me)C(O)OHex-n Me
CH(Et)SCH(Me)C(O)OMe Et
CH(Et)SCH(Me)C(O)OMe Pr-n
CH(Et)SCH(Me)C(O)OMe Pr-i
CH(Et)SCH(Me)C(O)OMe Pr-c
CH(Et)SCH(Me)C(O)OMe Bu-n
CH(Et)SCH(Me)C(O)OMe Bu-i
CH(Et)SCH(Me)C(O)OMe Bu-c
CH(Et)SCH(Me)C(O)OMe Bu-s
CH(Et)SCH(Me)C(O)OMe Bu-t
CH(Et)SCH(Me)C(O)OMe Pen-n
CH(Et)SCH(Me)C(O)OMe Pen-c
CH(Et)SCH(Me)C(O)OMe Hex-n
CH(Et)SCH(Me)C(O)OMe Hex-c
CH(Et)SCH(Me)C(O)OMe CH2Pr-c
CH(Et)SCH(Me)C(O)OMe CH2Bu-c
CH(Et)SCH(Me)C(O)OMe CH2Pen-c
CH(Et)SCH(Me)C(O)OMe CH2Hex-c
CH(Et)SCH(Me)C(O)OMe CH2CH=CH2
CH(Et)SCH(Me)C(O)OMe CH2CH=C(Cl)2
CH(Et)SCH(Me)C(O)OMe CH2C≡CH
CH(Et)SCH(Me)C(O)OMe CH2CN
CH(Et)SCH(Me)C(O)OMe CH2CF3
CH(Et)SCH(Me)C(O)OMe CH2OMe
CH(Et)SCH(Me)C(O)OMe CH2OCF3
CH(Et)SCH(Me)C(O)OMe CH2SMe
CH(Et)SCH(Me)C(O)OMe CH2S(O)Me
CH(Et)SCH(Me)C(O)OMe CH2S(O)2Me
CH(Et)SCH(Me)C(O)OMe CH2SCF3
CH(Et)SCH(Me)C(O)OMe CH2S(O)CF3
CH(Et)SCH(Me)C(O)OMe CH2S(O)2CF3
CH(Et)SCH(Me)C(O)OMe CH2CH(OMe)2
CH(Et)SCH(Me)C(O)OMe CH2CH(SMe)2
CH(Et)SCH(Me)C(O)OMe CH2C(O)Me
CH(Et)SCH(Me)C(O)OMe CH2C(O)CF3
CH(Et)SCH(Me)C(O)OMe CH2C(O)OMe
CH(Et)S(O)CH(Me)C(O)OMe Me
CH(Et)S(O)CH(Me)C(O)OEt Me
CH(Et)S(O)CH(Me)C(O)OPr-n Me
CH(Et)S(O)CH(Me)C(O)OPr-i Me
CH(Et)S(O)CH(Me)C(O)OBu-n Me
CH(Et)S(O)CH(Me)C(O)OBu-i Me
CH(Et)S(O)CH(Me)C(O)OBu-t Me
CH(Et)S(O)CH(Me)C(O)OPen-n Me
CH(Et)S(O)CH(Me)C(O)OHex-n Me
CH(Et)S(O)CH(Me)C(O)OMe Et
CH(Et)S(O)CH(Me)C(O)OMe Pr-n
CH(Et)S(O)CH(Me)C(O)OMe Pr-i
CH(Et)S(O)CH(Me)C(O)OMe Pr-c
CH(Et)S(O)CH(Me)C(O)OMe Bu-n
CH(Et)S(O)CH(Me)C(O)OMe Bu-i
CH(Et)S(O)CH(Me)C(O)OMe Bu-c
CH(Et)S(O)CH(Me)C(O)OMe Bu-s
CH(Et)S(O)CH(Me)C(O)OMe Bu-t
CH(Et)S(O)CH(Me)C(O)OMe Pen-n
CH(Et)S(O)CH(Me)C(O)OMe Pen-c
CH(Et)S(O)CH(Me)C(O)OMe Hex-n
CH(Et)S(O)CH(Me)C(O)OMe Hex-c
CH(Et)S(O)CH(Me)C(O)OMe CH2Pr-c
CH(Et)S(O)CH(Me)C(O)OMe CH2Bu-c
CH(Et)S(O)CH(Me)C(O)OMe CH2Pen-c
CH(Et)S(O)CH(Me)C(O)OMe CH2Hex-c
CH(Et)S(O)CH(Me)C(O)OMe CH2CH=CH2
CH(Et)S(O)CH(Me)C(O)OMe CH2CH=C(Cl)2
CH(Et)S(O)CH(Me)C(O)OMe CH2C≡CH
CH(Et)S(O)CH(Me)C(O)OMe CH2CN
CH(Et)S(O)CH(Me)C(O)OMe CH2CF3
CH(Et)S(O)CH(Me)C(O)OMe CH2OMe
CH(Et)S(O)CH(Me)C(O)OMe CH2OCF3
CH(Et)S(O)CH(Me)C(O)OMe CH2SMe
CH(Et)S(O)CH(Me)C(O)OMe CH2S(O)Me
CH(Et)S(O)CH(Me)C(O)OMe CH2S(O)2Me
CH(Et)S(O)CH(Me)C(O)OMe CH2SCF3
CH(Et)S(O)CH(Me)C(O)OMe CH2S(O)CF3
CH(Et)S(O)CH(Me)C(O)OMe CH2S(O)2CF3
CH(Et)S(O)CH(Me)C(O)OMe CH2CH(OMe)2
CH(Et)S(O)CH(Me)C(O)OMe CH2CH(SMe)2
CH(Et)S(O)CH(Me)C(O)OMe CH2C(O)Me
CH(Et)S(O)CH(Me)C(O)OMe CH2C(O)CF3
CH(Et)S(O)CH(Me)C(O)OMe CH2C(O)OMe
CH(Et)S(O)2CH(Me)C(O)OMe Me
CH(Et)S(O)2CH(Me)C(O)OEt Me
CH(Et)S(O)2CH(Me)C(O)OPr-n Me
CH(Et)S(O)2CH(Me)C(O)OPr-i Me
CH(Et)S(O)2CH(Me)C(O)OBu-n Me
CH(Et)S(O)2CH(Me)C(O)OBu-i Me
CH(Et)S(O)2CH(Me)C(O)OBu-t Me
CH(Et)S(O)2CH(Me)C(O)OPen-n Me
CH(Et)S(O)2CH(Me)C(O)OHex-n Me
CH(Et)S(O)2CH(Me)C(O)OMe Et
CH(Et)S(O)2CH(Me)C(O)OMe Pr-n
CH(Et)S(O)2CH(Me)C(O)OMe Pr-i
CH(Et)S(O)2CH(Me)C(O)OMe Pr-c
CH(Et)S(O)2CH(Me)C(O)OMe Bu-n
CH(Et)S(O)2CH(Me)C(O)OMe Bu-i
CH(Et)S(O)2CH(Me)C(O)OMe Bu-c
CH(Et)S(O)2CH(Me)C(O)OMe Bu-s
CH(Et)S(O)2CH(Me)C(O)OMe Bu-t
CH(Et)S(O)2CH(Me)C(O)OMe Pen-n
CH(Et)S(O)2CH(Me)C(O)OMe Pen-c
CH(Et)S(O)2CH(Me)C(O)OMe Hex-n
CH(Et)S(O)2CH(Me)C(O)OMe Hex-c
CH(Et)S(O)2CH(Me)C(O)OMe CH2Pr-c
CH(Et)S(O)2CH(Me)C(O)OMe CH2Bu-c
CH(Et)S(O)2CH(Me)C(O)OMe CH2Pen-c
CH(Et)S(O)2CH(Me)C(O)OMe CH2Hex-c
CH(Et)S(O)2CH(Me)C(O)OMe CH2CH=CH2
CH(Et)S(O)2CH(Me)C(O)OMe CH2CH=C(Cl)2
CH(Et)S(O)2CH(Me)C(O)OMe CH2C≡CH
CH(Et)S(O)2CH(Me)C(O)OMe CH2CN
CH(Et)S(O)2CH(Me)C(O)OMe CH2CF3
CH(Et)S(O)2CH(Me)C(O)OMe CH2OMe
CH(Et)S(O)2CH(Me)C(O)OMe CH2OCF3
CH(Et)S(O)2CH(Me)C(O)OMe CH2SMe
CH(Et)S(O)2CH(Me)C(O)OMe CH2S(O)Me
CH(Et)S(O)2CH(Me)C(O)OMe CH2S(O)2Me
CH(Et)S(O)2CH(Me)C(O)OMe CH2SCF3
CH(Et)S(O)2CH(Me)C(O)OMe CH2S(O)CF3
CH(Et)S(O)2CH(Me)C(O)OMe CH2S(O)2CF3
CH(Et)S(O)2CH(Me)C(O)OMe CH2CH(OMe)2
CH(Et)S(O)2CH(Me)C(O)OMe CH2CH(SMe)2
CH(Et)S(O)2CH(Me)C(O)OMe CH2C(O)Me
CH(Et)S(O)2CH(Me)C(O)OMe CH2C(O)CF3
CH(Et)S(O)2CH(Me)C(O)OMe CH2C(O)OMe
----------------------------------------------------
本発明化合物は、農園芸作物及び樹木などを加害する所謂農業害虫、家畜・家禽類に寄生する所謂家畜害虫、家屋等の人間の生活環境で様々な悪影響を与える所謂衛生害虫、倉庫に貯蔵された穀物等を加害する所謂貯穀害虫等としての昆虫類、及び同様の場面で発生、加害するダニ類、甲殻類、軟体動物、線虫類の何れの有害生物も低濃度で有効に防除できる。
-------------------------------------------------- ---
R12b                                R11b
-------------------------------------------------- ---
H Me
H Et
H Pr-n
H Pr-i
H Pr-c
H Bu-n
H Bu-i
H Bu-c
H Bu-s
H Bu-t
H Pen-n
H Pen-c
H Hex-n
H Hex-c
H CH2Pr-c
H CH2Bu-c
H CH2Pen-c
H CH2Hex-c
H CH2CH = CH2
H CH2CH = C (Cl)2
H CH2C≡CH
H CH2CN
H CH2CFThree
H CH2OMe
H CH2OCFThree
H CH2SMe
H CH2S (O) Me
H CH2S (O)2Me
H CH2SCFThree
H CH2S (O) CFThree
H CH2S (O)2CFThree
H CH2CH (OMe)2
H CH2CH (SMe)2
H CH2C (O) Me
H CH2C (O) CFThree
H CH2C (O) OMe
H CH2(D1-32a)
H CH2(D1-33a)
H CH2(D1-34a)
H CH2(D1-37a)
H CH2(D1-81a)
H CH2(D1-82a)
H CH2(D1-84a)
H CH2(D1-85a)
H CH2(D1-87a)
H CH2(D1-92a)
H CH2(D1-93a)
H CH2(D1-95a)
H CH2(D1-96a)
H CH2(D1-98a)
H CH2(D1-108a)
H CH2(D1-108b, Z = 2-Cl)
H CH2(D1-108b, Z = 3-Me)
H CH2(D1-108b, Z = 4-OMe)
H CH2(D1-108b, Z = 2-SMe)
H CH2(D1-108b, Z = 3-CFThree)
H CH2(D1-108b, Z = 4-OCFThree)
H CH2(D1-108b, Z = 2-SCFThree)
H CH2CH2CN
H CH2CH2CFThree
H CH2CH2OMe
H CH2CH2SMe
H CH2CH2S (O) Me
H CH2CH2S (O)2Me
H D1-32a
H D1-33a
H D1-34a
H D1-37a
H D1-81a
H D1-82a
H D1-84a
H D1-85a
H D1-87a
H D1-92a
H D1-93a
H D1-95a
H D1-96a
H D1-98a
H D1-108a
H D1-108b (Z = 2-Cl)
H D1-108b (Z = 3-Me)
H D1-108b (Z = 4-OMe)
H D1-108b (Z = 2-SMe)
H D1-108b (Z = 3-CFThree)
H D1-108b (Z = 4-OCFThree)
H D1-108b (Z = 2-SCFThree)
H C (O) Me
H C (O) CFThree
H C (O) OMe
CFThree                                Me
CFThree                                Et
CFThree                                Pr-n
CFThree                                Pr-i
CFThree                                Pr-c
CFThree                                Bu-n
CFThree                                Bu-i
CFThree                                Bu-c
CFThree                                Bu-s
CFThree                                Bu-t
CFThree                                Pen-n
CFThree                                Pen-c
CFThree                                Hex-n
CFThree                                Hex-c
CFThree                                CH2Pr-c
CFThree                                CH2Bu-c
CFThree                                CH2Pen-c
CFThree                                CH2Hex-c
CFThree                               CH2CH = CH2
CFThree                                CH2CH = C (Cl)2
CFThree                                CH2C≡CH
CFThree                                CH2CN
CFThree                                CH2CFThree
CFThree                                CH2OMe
CFThree                                CH2OCFThree
CFThree                                CH2SMe
CFThree                                CH2S (O) Me
CFThree                                CH2S (O)2Me
CFThree                                CH2SCFThree
CFThree                                CH2S (O) CFThree
CFThree                                CH2S (O)2CFThree
CFThree                                CH2CH (OMe)2
CFThree                                CH2CH (SMe)2
CFThree                                CH2C (O) Me
CFThree                                CH2C (O) CFThree
CFThree                                CH2C (O) OMe
CFThree                                CH2(D1-32a)
CFThree                                CH2(D1-33a)
CFThree                                CH2(D1-34a)
CFThree                                CH2(D1-37a)
CFThree                                CH2(D1-81a)
CFThree                                CH2(D1-82a)
CFThree                                CH2(D1-84a)
CFThree                                CH2(D1-85a)
CFThree                                CH2(D1-87a)
CFThree                                CH2(D1-92a)
CFThree                                CH2(D1-93a)
CFThree                                CH2(D1-95a)
CFThree                                CH2(D1-96a)
CFThree                                CH2(D1-98a)
CFThree                                CH2(D1-108a)
CFThree                                CH2(D1-108b, Z = 2-Cl)
CFThree                                CH2(D1-108b, Z = 3-Me)
CFThree                                CH2(D1-108b, Z = 4-OMe)
CFThree                                CH2(D1-108b, Z = 2-SMe)
CFThree                                CH2(D1-108b, Z = 3-CFThree)
CFThree                                CH2(D1-108b, Z = 4-OCFThree)
CFThree                                CH2(D1-108b, Z = 2-SCFThree)
CFThree                                CH2CH2CN
CFThree                                CH2CH2CFThree
CFThree                                CH2CH2OMe
CFThree                                CH2CH2SMe
CFThree                                CH2CH2S (O) Me
CFThree                                CH2CH2S (O)2Me
CFThree                                D1-32a
CFThree                                D1-33a
CFThree                                D1-34a
CFThree                               D1-37a
CFThree                                D1-81a
CFThree                                D1-82a
CFThree                                D1-84a
CFThree                                D1-85a
CFThree                                D1-87a
CFThree                                D1-92a
CFThree                                D1-93a
CFThree                                D1-95a
CFThree                               D1-96a
CFThree                                D1-98a
CFThree                                D1-108a
CFThree                                D1-108b (Z = 2-Cl)
CFThree                                D1-108b (Z = 3-Me)
CFThree                                D1-108b (Z = 4-OMe)
CFThree                                D1-108b (Z = 2-SMe)
CFThree                                D1-108b (Z = 3-CFThree)
CFThree                                D1-108b (Z = 4-OCFThree)
CFThree                                D1-108b (Z = 2-SCFThree)
CFThree                                C (O) Me
CFThree                                C (O) CFThree
CFThree                                C (O) OMe
Me Me
Me Et
Me Pr-n
Me Pr-i
Me Pr-c
Me Bu-n
Me Bu-i
Me Bu-c
Me Bu-s
Me Bu-t
Me Pen-n
Me Pen-c
Me Hex-n
Me Hex-c
Me CH2Pr-c
Me CH2Bu-c
Me CH2Pen-c
Me CH2Hex-c
Me CH2CH = CH2
Me CH2CH = C (Cl)2
Me CH2C≡CH
Me CH2CN
Me CH2CFThree
Me CH2OMe
Me CH2OCFThree
Me CH2SMe
Me CH2S (O) Me
Me CH2S (O)2Me
Me CH2SCFThree
Me CH2S (O) CFThree
Me CH2S (O)2CFThree
Me CH2CH (OMe)2
Me CH2CH (SMe)2
Me CH2C (O) Me
Me CH2C (O) CFThree
Me CH2C (O) OMe
Me CH2(D1-32a)
Me CH2(D1-33a)
Me CH2(D1-34a)
Me CH2(D1-37a)
Me CH2(D1-81a)
Me CH2(D1-82a)
Me CH2(D1-84a)
Me CH2(D1-85a)
Me CH2(D1-87a)
Me CH2(D1-92a)
Me CH2(D1-93a)
Me CH2(D1-95a)
Me CH2(D1-96a)
Me CH2(D1-98a)
Me CH2(D1-108a)
Me CH2(D1-108b, Z = 2-Cl)
Me CH2(D1-108b, Z = 3-Me)
Me CH2(D1-108b, Z = 4-OMe)
Me CH2(D1-108b, Z = 2-SMe)
Me CH2(D1-108b, Z = 3-CFThree)
Me CH2(D1-108b, Z = 4-OCFThree)
Me CH2(D1-108b, Z = 2-SCFThree)
Me CH2CH2CN
Me CH2CH2CFThree
Me CH2CH2OMe
Me CH2CH2SMe
Me CH2CH2S (O) Me
Me CH2CH2S (O)2Me
Me D1-32a
Me D1-33a
Me D1-34a
Me D1-37a
Me D1-81a
Me D1-82a
Me D1-84a
Me D1-85a
Me D1-87a
Me D1-92a
Me D1-93a
Me D1-95a
Me D1-96a
Me D1-98a
Me D1-108a
Me D1-108b (Z = 2-Cl)
Me D1-108b (Z = 3-Me)
Me D1-108b (Z = 4-OMe)
Me D1-108b (Z = 2-SMe)
Me D1-108b (Z = 3-CFThree)
Me D1-108b (Z = 4-OCFThree)
Me D1-108b (Z = 2-SCFThree)
Me C (O) Me
Me C (O) CFThree
Me C (O) OMe
OMe Me
OMe Et
OMe Pr-n
OMe Pr-i
OMe Pr-c
OMe Bu-n
OMe Bu-i
OMe Bu-c
OMe Bu-s
OMe Bu-t
OMe Pen-n
OMe Pen-c
OMe Hex-n
OMe Hex-c
OMe CH2Pr-c
OMe CH2Bu-c
OMe CH2Pen-c
OMe CH2Hex-c
OMe CH2CH = CH2
OMe CH2CH = C (Cl)2
OMe CH2C≡CH
OMe CH2CN
OMe CH2CFThree
OMe CH2OMe
OMe CH2OCFThree
OMe CH2SMe
OMe CH2S (O) Me
OMe CH2S (O)2Me
OMe CH2SCFThree
OMe CH2S (O) CFThree
OMe CH2S (O)2CFThree
OMe CH2CH (OMe)2
OMe CH2CH (SMe)2
OMe CH2C (O) Me
OMe CH2C (O) CFThree
OMe CH2C (O) OMe
OMe CH2(D1-32a)
OMe CH2(D1-33a)
OMe CH2(D1-34a)
OMe CH2(D1-37a)
OMe CH2(D1-81a)
OMe CH2(D1-82a)
OMe CH2(D1-84a)
OMe CH2(D1-85a)
OMe CH2(D1-87a)
OMe CH2(D1-92a)
OMe CH2(D1-93a)
OMe CH2(D1-95a)
OMe CH2(D1-96a)
OMe CH2(D1-98a)
OMe CH2(D1-108a)
OMe CH2(D1-108b, Z = 2-Cl)
OMe CH2(D1-108b, Z = 3-Me)
OMe CH2(D1-108b, Z = 4-OMe)
OMe CH2(D1-108b, Z = 2-SMe)
OMe CH2(D1-108b, Z = 3-CFThree)
OMe CH2(D1-108b, Z = 4-OCFThree)
OMe CH2(D1-108b, Z = 2-SCFThree)
OMe CH2CH2CN
OMe CH2CH2CFThree
OMe CH2CH2OMe
OMe CH2CH2SMe
OMe CH2CH2S (O) Me
OMe CH2CH2S (O)2Me
OMe D1-32a
OMe D1-33a
OMe D1-34a
OMe D1-37a
OMe D1-81a
OMe D1-82a
OMe D1-84a
OMe D1-85a
OMe D1-87a
OMe D1-92a
OMe D1-93a
OMe D1-95a
OMe D1-96a
OMe D1-98a
OMe D1-108a
OMe D1-108b (Z = 2-Cl)
OMe D1-108b (Z = 3-Me)
OMe D1-108b (Z = 4-OMe)
OMe D1-108b (Z = 2-SMe)
OMe D1-108b (Z = 3-CFThree)
OMe D1-108b (Z = 4-OCFThree)
OMe D1-108b (Z = 2-SCFThree)
OMe C (O) Me
OMe C (O) CFThree
OMe C (O) OMe
SMe Me
SMe Et
SMe Pr-n
SMe Pr-i
SMe Pr-c
SMe Bu-n
SMe Bu-i
SMe Bu-c
SMe Bu-s
SMe Bu-t
SMe Pen-n
SMe Pen-c
SMe Hex-n
SMe Hex-c
SMe CH2Pr-c
SMe CH2Bu-c
SMe CH2Pen-c
SMe CH2Hex-c
SMe CH2CH = CH2
SMe CH2CH = C (Cl)2
SMe CH2C≡CH
SMe CH2CN
SMe CH2CFThree
SMe CH2OMe
SMe CH2OCFThree
SMe CH2SMe
SMe CH2S (O) Me
SMe CH2S (O)2Me
SMe CH2SCFThree
SMe CH2S (O) CFThree
SMe CH2S (O)2CFThree
SMe CH2CH (OMe)2
SMe CH2CH (SMe)2
SMe CH2C (O) Me
SMe CH2C (O) CFThree
SMe CH2C (O) OMe
SMe CH2(D1-32a)
SMe CH2(D1-33a)
SMe CH2(D1-34a)
SMe CH2(D1-37a)
SMe CH2(D1-81a)
SMe CH2(D1-82a)
SMe CH2(D1-84a)
SMe CH2(D1-85a)
SMe CH2(D1-87a)
SMe CH2(D1-92a)
SMe CH2(D1-93a)
SMe CH2(D1-95a)
SMe CH2(D1-96a)
SMe CH2(D1-98a)
SMe CH2(D1-108a)
SMe CH2(D1-108b, Z = 2-Cl)
SMe CH2(D1-108b, Z = 3-Me)
SMe CH2(D1-108b, Z = 4-OMe)
SMe CH2(D1-108b, Z = 2-SMe)
SMe CH2(D1-108b, Z = 3-CFThree)
SMe CH2(D1-108b, Z = 4-OCFThree)
SMe CH2(D1-108b, Z = 2-SCFThree)
SMe CH2CH2CN
SMe CH2CH2CFThree
SMe CH2CH2OMe
SMe CH2CH2SMe
SMe CH2CH2S (O) Me
SMe CH2CH2S (O)2Me
SMe D1-32a
SMe D1-33a
SMe D1-34a
SMe D1-37a
SMe D1-81a
SMe D1-82a
SMe D1-84a
SMe D1-85a
SMe D1-87a
SMe D1-92a
SMe D1-93a
SMe D1-95a
SMe D1-96a
SMe D1-98a
SMe D1-108a
SMe D1-108b (Z = 2-Cl)
SMe D1-108b (Z = 3-Me)
SMe D1-108b (Z = 4-OMe)
SMe D1-108b (Z = 2-SMe)
SMe D1-108b (Z = 3-CFThree)
SMe D1-108b (Z = 4-OCFThree)
SMe D1-108b (Z = 2-SCFThree)
SMe C (O) Me
SMe C (O) CFThree
SMe C (O) OMe
CH2OMe Me
CH2OMe Et
CH2OMe Pr-n
CH2OMe Pr-i
CH2OMe Pr-c
CH2OMe Bu-n
CH2OMe Bu-i
CH2OMe Bu-c
CH2OMe Bu-s
CH2OMe Bu-t
CH2OMe Pen-n
CH2OMe Pen-c
CH2OMe Hex-n
CH2OMe Hex-c
CH2OMe CH2Pr-c
CH2OMe CH2Bu-c
CH2OMe CH2Pen-c
CH2OMe CH2Hex-c
CH2OMe CH2CH = CH2
CH2OMe CH2CH = C (Cl)2
CH2OMe CH2C≡CH
CH2OMe CH2CN
CH2OMe CH2CFThree
CH2OMe CH2OMe
CH2OMe CH2OCFThree
CH2OMe CH2SMe
CH2OMe CH2S (O) Me
CH2OMe CH2S (O)2Me
CH2OMe CH2SCFThree
CH2OMe CH2S (O) CFThree
CH2OMe CH2S (O)2CFThree
CH2OMe CH2CH (OMe)2
CH2OMe CH2CH (SMe)2
CH2OMe CH2C (O) Me
CH2OMe CH2C (O) CFThree
CH2OMe CH2C (O) OMe
CH2OMe CH2(D1-32a)
CH2OMe CH2(D1-33a)
CH2OMe CH2(D1-34a)
CH2OMe CH2(D1-37a)
CH2OMe CH2(D1-81a)
CH2OMe CH2(D1-82a)
CH2OMe CH2(D1-84a)
CH2OMe CH2(D1-85a)
CH2OMe CH2(D1-87a)
CH2OMe CH2(D1-92a)
CH2OMe CH2(D1-93a)
CH2OMe CH2(D1-95a)
CH2OMe CH2(D1-96a)
CH2OMe CH2(D1-98a)
CH2OMe CH2(D1-108a)
CH2OMe CH2(D1-108b, Z = 2-Cl)
CH2OMe CH2(D1-108b, Z = 3-Me)
CH2OMe CH2(D1-108b, Z = 4-OMe)
CH2OMe CH2(D1-108b, Z = 2-SMe)
CH2OMe CH2(D1-108b, Z = 3-CFThree)
CH2OMe CH2(D1-108b, Z = 4-OCFThree)
CH2OMe CH2(D1-108b, Z = 2-SCFThree)
CH2OMe CH2CH2CN
CH2OMe CH2CH2CFThree
CH2OMe CH2CH2OMe
CH2OMe CH2CH2SMe
CH2OMe CH2CH2S (O) Me
CH2OMe CH2CH2S (O)2Me
CH2OMe D1-32a
CH2OMe D1-33a
CH2OMe D1-34a
CH2OMe D1-37a
CH2OMe D1-81a
CH2OMe D1-82a
CH2OMe D1-84a
CH2OMe D1-85a
CH2OMe D1-87a
CH2OMe D1-92a
CH2OMe D1-93a
CH2OMe D1-95a
CH2OMe D1-96a
CH2OMe D1-98a
CH2OMe D1-108a
CH2OMe D1-108b (Z = 2-Cl)
CH2OMe D1-108b (Z = 3-Me)
CH2OMe D1-108b (Z = 4-OMe)
CH2OMe D1-108b (Z = 2-SMe)
CH2OMe D1-108b (Z = 3-CFThree)
CH2OMe D1-108b (Z = 4-OCFThree)
CH2OMe D1-108b (Z = 2-SCFThree)
CH2OMe C (O) Me
CH2OMe C (O) CFThree
CH2OMe C (O) OMe
CH2SMe Me
CH2SMe Et
CH2SMe Pr-n
CH2SMe Pr-i
CH2SMe Pr-c
CH2SMe Bu-n
CH2SMe Bu-i
CH2SMe Bu-c
CH2SMe Bu-s
CH2SMe Bu-t
CH2SMe Pen-n
CH2SMe Pen-c
CH2SMe Hex-n
CH2SMe Hex-c
CH2SMe CH2Pr-c
CH2SMe CH2Bu-c
CH2SMe CH2Pen-c
CH2SMe CH2Hex-c
CH2SMe CH2CH = CH2
CH2SMe CH2CH = C (Cl)2
CH2SMe CH2C≡CH
CH2SMe CH2CN
CH2SMe CH2CFThree
CH2SMe CH2OMe
CH2SMe CH2OCFThree
CH2SMe CH2SMe
CH2SMe CH2S (O) Me
CH2SMe CH2S (O)2Me
CH2SMe CH2SCFThree
CH2SMe CH2S (O) CFThree
CH2SMe CH2S (O)2CFThree
CH2SMe CH2CH (OMe)2
CH2SMe CH2CH (SMe)2
CH2SMe CH2C (O) Me
CH2SMe CH2C (O) CFThree
CH2SMe CH2C (O) OMe
CH2SMe CH2(D1-32a)
CH2SMe CH2(D1-33a)
CH2SMe CH2(D1-34a)
CH2SMe CH2(D1-37a)
CH2SMe CH2(D1-81a)
CH2SMe CH2(D1-82a)
CH2SMe CH2(D1-84a)
CH2SMe CH2(D1-85a)
CH2SMe CH2(D1-87a)
CH2SMe CH2(D1-92a)
CH2SMe CH2(D1-93a)
CH2SMe CH2(D1-95a)
CH2SMe CH2(D1-96a)
CH2SMe CH2(D1-98a)
CH2SMe CH2(D1-108a)
CH2SMe CH2(D1-108b, Z = 2-Cl)
CH2SMe CH2(D1-108b, Z = 3-Me)
CH2SMe CH2(D1-108b, Z = 4-OMe)
CH2SMe CH2(D1-108b, Z = 2-SMe)
CH2SMe CH2(D1-108b, Z = 3-CFThree)
CH2SMe CH2(D1-108b, Z = 4-OCFThree)
CH2SMe CH2(D1-108b, Z = 2-SCFThree)
CH2SMe CH2CH2CN
CH2SMe CH2CH2CFThree
CH2SMe CH2CH2OMe
CH2SMe CH2CH2SMe
CH2SMe CH2CH2S (O) Me
CH2SMe CH2CH2S (O)2Me
CH2SMe D1-32a
CH2SMe D1-33a
CH2SMe D1-34a
CH2SMe D1-37a
CH2SMe D1-81a
CH2SMe D1-82a
CH2SMe D1-84a
CH2SMe D1-85a
CH2SMe D1-87a
CH2SMe D1-92a
CH2SMe D1-93a
CH2SMe D1-95a
CH2SMe D1-96a
CH2SMe D1-98a
CH2SMe D1-108a
CH2SMe D1-108b (Z = 2-Cl)
CH2SMe D1-108b (Z = 3-Me)
CH2SMe D1-108b (Z = 4-OMe)
CH2SMe D1-108b (Z = 2-SMe)
CH2SMe D1-108b (Z = 3-CFThree)
CH2SMe D1-108b (Z = 4-OCFThree)
CH2SMe D1-108b (Z = 2-SCFThree)
CH2SMe C (O) Me
CH2SMe C (O) CFThree
CH2SMe C (O) OMe
CH2S (O) Me Me
CH2S (O) Me Et
CH2S (O) Me Pr-n
CH2S (O) Me Pr-i
CH2S (O) Me Pr-c
CH2S (O) Me Bu-n
CH2S (O) Me Bu-i
CH2S (O) Me Bu-c
CH2S (O) Me Bu-s
CH2S (O) Me Bu-t
CH2S (O) Me Pen-n
CH2S (O) Me Pen-c
CH2S (O) Me Hex-n
CH2S (O) Me Hex-c
CH2S (O) Me CH2Pr-c
CH2S (O) Me CH2Bu-c
CH2S (O) Me CH2Pen-c
CH2S (O) Me CH2Hex-c
CH2S (O) Me CH2CH = CH2
CH2S (O) Me CH2CH = C (Cl)2
CH2S (O) Me CH2C≡CH
CH2S (O) Me CH2CN
CH2S (O) Me CH2CFThree
CH2S (O) Me CH2OMe
CH2S (O) Me CH2OCFThree
CH2S (O) Me CH2SMe
CH2S (O) Me CH2S (O) Me
CH2S (O) Me CH2S (O)2Me
CH2S (O) Me CH2SCFThree
CH2S (O) Me CH2S (O) CFThree
CH2S (O) Me CH2S (O)2CFThree
CH2S (O) Me CH2CH (OMe)2
CH2S (O) Me CH2CH (SMe)2
CH2S (O) Me CH2C (O) Me
CH2S (O) Me CH2C (O) CFThree
CH2S (O) Me CH2C (O) OMe
CH2S (O) Me CH2(D1-32a)
CH2S (O) Me CH2(D1-33a)
CH2S (O) Me CH2(D1-34a)
CH2S (O) Me CH2(D1-37a)
CH2S (O) Me CH2(D1-81a)
CH2S (O) Me CH2(D1-82a)
CH2S (O) Me CH2(D1-84a)
CH2S (O) Me CH2(D1-85a)
CH2S (O) Me CH2(D1-87a)
CH2S (O) Me CH2(D1-92a)
CH2S (O) Me CH2(D1-93a)
CH2S (O) Me CH2(D1-95a)
CH2S (O) Me CH2(D1-96a)
CH2S (O) Me CH2(D1-98a)
CH2S (O) Me CH2(D1-108a)
CH2S (O) Me CH2(D1-108b, Z = 2-Cl)
CH2S (O) Me CH2(D1-108b, Z = 3-Me)
CH2S (O) Me CH2(D1-108b, Z = 4-OMe)
CH2S (O) Me CH2(D1-108b, Z = 2-SMe)
CH2S (O) Me CH2(D1-108b, Z = 3-CFThree)
CH2S (O) Me CH2(D1-108b, Z = 4-OCFThree)
CH2S (O) Me CH2(D1-108b, Z = 2-SCFThree)
CH2S (O) Me CH2CH2CN
CH2S (O) Me CH2CH2CFThree
CH2S (O) Me CH2CH2OMe
CH2S (O) Me CH2CH2SMe
CH2S (O) Me CH2CH2S (O) Me
CH2S (O) Me CH2CH2S (O)2Me
CH2S (O) Me D1-32a
CH2S (O) Me D1-33a
CH2S (O) Me D1-34a
CH2S (O) Me D1-37a
CH2S (O) Me D1-81a
CH2S (O) Me D1-82a
CH2S (O) Me D1-84a
CH2S (O) Me D1-85a
CH2S (O) Me D1-87a
CH2S (O) Me D1-92a
CH2S (O) Me D1-93a
CH2S (O) Me D1-95a
CH2S (O) Me D1-96a
CH2S (O) Me D1-98a
CH2S (O) Me D1-108a
CH2S (O) Me D1-108b (Z = 2-Cl)
CH2S (O) Me D1-108b (Z = 3-Me)
CH2S (O) Me D1-108b (Z = 4-OMe)
CH2S (O) Me D1-108b (Z = 2-SMe)
CH2S (O) Me D1-108b (Z = 3-CFThree)
CH2S (O) Me D1-108b (Z = 4-OCFThree)
CH2S (O) Me D1-108b (Z = 2-SCFThree)
CH2S (O) Me C (O) Me
CH2S (O) Me C (O) CFThree
CH2S (O) Me C (O) OMe
CH2S (O)2Me Me
CH2S (O)2Me Et
CH2S (O)2Me Pr-n
CH2S (O)2Me Pr-i
CH2S (O)2Me Pr-c
CH2S (O)2Me Bu-n
CH2S (O)2Me Bu-i
CH2S (O)2Me Bu-c
CH2S (O)2Me Bu-s
CH2S (O)2Me Bu-t
CH2S (O)2Me Pen-n
CH2S (O)2Me Pen-c
CH2S (O)2Me Hex-n
CH2S (O)2Me Hex-c
CH2S (O)2Me CH2Pr-c
CH2S (O)2Me CH2Bu-c
CH2S (O)2Me CH2Pen-c
CH2S (O)2Me CH2Hex-c
CH2S (O)2Me CH2CH = CH2
CH2S (O)2Me CH2CH = C (Cl)2
CH2S (O)2Me CH2C≡CH
CH2S (O)2Me CH2CN
CH2S (O)2Me CH2CFThree
CH2S (O)2Me CH2OMe
CH2S (O)2Me CH2OCFThree
CH2S (O)2Me CH2SMe
CH2S (O)2Me CH2S (O) Me
CH2S (O)2Me CH2S (O)2Me
CH2S (O)2Me CH2SCFThree
CH2S (O)2Me CH2S (O) CFThree
CH2S (O)2Me CH2S (O)2CFThree
CH2S (O)2Me CH2CH (OMe)2
CH2S (O)2Me CH2CH (SMe)2
CH2S (O)2Me CH2C (O) Me
CH2S (O)2Me CH2C (O) CFThree
CH2S (O)2Me CH2C (O) OMe
CH2S (O)2Me CH2(D1-32a)
CH2S (O)2Me CH2(D1-33a)
CH2S (O)2Me CH2(D1-34a)
CH2S (O)2Me CH2(D1-37a)
CH2S (O)2Me CH2(D1-81a)
CH2S (O)2Me CH2(D1-82a)
CH2S (O)2Me CH2(D1-84a)
CH2S (O)2Me CH2(D1-85a)
CH2S (O)2Me CH2(D1-87a)
CH2S (O)2Me CH2(D1-92a)
CH2S (O)2Me CH2(D1-93a)
CH2S (O)2Me CH2(D1-95a)
CH2S (O)2Me CH2(D1-96a)
CH2S (O)2Me CH2(D1-98a)
CH2S (O)2Me CH2(D1-108a)
CH2S (O)2Me CH2(D1-108b, Z = 2-Cl)
CH2S (O)2Me CH2(D1-108b, Z = 3-Me)
CH2S (O)2Me CH2(D1-108b, Z = 4-OMe)
CH2S (O)2Me CH2(D1-108b, Z = 2-SMe)
CH2S (O)2Me CH2(D1-108b, Z = 3-CFThree)
CH2S (O)2Me CH2(D1-108b, Z = 4-OCFThree)
CH2S (O)2Me CH2(D1-108b, Z = 2-SCFThree)
CH2S (O)2Me CH2CH2CN
CH2S (O)2Me CH2CH2CFThree
CH2S (O)2Me CH2CH2OMe
CH2S (O)2Me CH2CH2SMe
CH2S (O)2Me CH2CH2S (O) Me
CH2S (O)2Me CH2CH2S (O)2Me
CH2S (O)2Me D1-32a
CH2S (O)2Me D1-33a
CH2S (O)2Me D1-34a
CH2S (O)2Me D1-37a
CH2S (O)2Me D1-81a
CH2S (O)2Me D1-82a
CH2S (O)2Me D1-84a
CH2S (O)2Me D1-85a
CH2S (O)2Me D1-87a
CH2S (O)2Me D1-92a
CH2S (O)2Me D1-93a
CH2S (O)2Me D1-95a
CH2S (O)2Me D1-96a
CH2S (O)2Me D1-98a
CH2S (O)2Me D1-108a
CH2S (O)2Me D1-108b (Z = 2-Cl)
CH2S (O)2Me D1-108b (Z = 3-Me)
CH2S (O)2Me D1-108b (Z = 4-OMe)
CH2S (O)2Me D1-108b (Z = 2-SMe)
CH2S (O)2Me D1-108b (Z = 3-CFThree)
CH2S (O)2Me D1-108b (Z = 4-OCFThree)
CH2S (O)2Me D1-108b (Z = 2-SCFThree)
CH2S (O)2Me C (O) Me
CH2S (O)2Me C (O) CFThree
CH2S (O)2Me C (O) OMe
CH (Me) SMe Me
CH (Me) SMe Et
CH (Me) SMe Pr-n
CH (Me) SMe Pr-i
CH (Me) SMe Pr-c
CH (Me) SMe Bu-n
CH (Me) SMe Bu-i
CH (Me) SMe Bu-c
CH (Me) SMe Bu-s
CH (Me) SMe Bu-t
CH (Me) SMe Pen-n
CH (Me) SMe Pen-c
CH (Me) SMe Hex-n
CH (Me) S (O) Me Me
CH (Me) S (O) Me Et
CH (Me) S (O) Me Pr-n
CH (Me) S (O) Me Pr-i
CH (Me) S (O) Me Pr-c
CH (Me) S (O) Me Bu-n
CH (Me) S (O) Me Bu-i
CH (Me) S (O) Me Bu-c
CH (Me) S (O) Me Bu-s
CH (Me) S (O) Me Bu-t
CH (Me) S (O) Me Pen-n
CH (Me) S (O) Me Pen-c
CH (Me) S (O) Me Hex-n
CH (Me) S (O)2Me Me
CH (Me) S (O)2Me Et
CH (Me) S (O)2Me Pr-n
CH (Me) S (O)2Me Pr-i
CH (Me) S (O)2Me Pr-c
CH (Me) S (O)2Me Bu-n
CH (Me) S (O)2Me Bu-i
CH (Me) S (O)2Me Bu-c
CH (Me) S (O)2Me Bu-s
CH (Me) S (O)2Me Bu-t
CH (Me) S (O)2Me Pen-n
CH (Me) S (O)2Me Pen-c
CH (Me) S (O)2Me Hex-n
CH (Et) SMe Me
CH (Et) SMe Et
CH (Et) SMe Pr-n
CH (Et) SMe Pr-i
CH (Et) SMe Pr-c
CH (Et) SMe Bu-n
CH (Et) SMe Bu-i
CH (Et) SMe Bu-c
CH (Et) SMe Bu-s
CH (Et) SMe Bu-t
CH (Et) SMe Pen-n
CH (Et) SMe Pen-c
CH (Et) SMe Hex-n
CH (Et) S (O) Me Me
CH (Et) S (O) Me Et
CH (Et) S (O) Me Pr-n
CH (Et) S (O) Me Pr-i
CH (Et) S (O) Me Pr-c
CH (Et) S (O) Me Bu-n
CH (Et) S (O) Me Bu-i
CH (Et) S (O) Me Bu-c
CH (Et) S (O) Me Bu-s
CH (Et) S (O) Me Bu-t
CH (Et) S (O) Me Pen-n
CH (Et) S (O) Me Pen-c
CH (Et) S (O) Me Hex-n
CH (Et) S (O)2Me Me
CH (Et) S (O)2Me Et
CH (Et) S (O)2Me Pr-n
CH (Et) S (O)2Me Pr-i
CH (Et) S (O)2Me Pr-c
CH (Et) S (O)2Me Bu-n
CH (Et) S (O)2Me Bu-i
CH (Et) S (O)2Me Bu-c
CH (Et) S (O)2Me Bu-s
CH (Et) S (O)2Me Bu-t
CH (Et) S (O)2Me Pen-n
CH (Et) S (O)2Me Pen-c
CH (Et) S (O)2Me Hex-n
CH (Me) SEt Me
CH (Me) SEt Et
CH (Me) SEt Pr-n
CH (Me) SEt Pr-i
CH (Me) SEt Pr-c
CH (Me) SEt Bu-n
CH (Me) SEt Bu-i
CH (Me) SEt Bu-c
CH (Me) SEt Bu-s
CH (Me) SEt Bu-t
CH (Me) SEt Pen-n
CH (Me) SEt Pen-c
CH (Me) SEt Hex-n
CH (Me) S (O) Et Me
CH (Me) S (O) Et Et
CH (Me) S (O) Et Pr-n
CH (Me) S (O) Et Pr-i
CH (Me) S (O) Et Pr-c
CH (Me) S (O) Et Bu-n
CH (Me) S (O) Et Bu-i
CH (Me) S (O) Et Bu-c
CH (Me) S (O) Et Bu-s
CH (Me) S (O) Et Bu-t
CH (Me) S (O) Et Pen-n
CH (Me) S (O) Et Pen-c
CH (Me) S (O) Et Hex-n
CH (Me) S (O)2Et Me
CH (Me) S (O)2Et Et
CH (Me) S (O)2Et Pr-n
CH (Me) S (O)2Et Pr-i
CH (Me) S (O)2Et Pr-c
CH (Me) S (O)2Et Bu-n
CH (Me) S (O)2Et Bu-i
CH (Me) S (O)2Et Bu-c
CH (Me) S (O)2Et Bu-s
CH (Me) S (O)2Et Bu-t
CH (Me) S (O)2Et Pen-n
CH (Me) S (O)2Et Pen-c
CH (Me) S (O)2Et Hex-n
CH (Et) SEt Me
CH (Et) SEt Et
CH (Et) SEt Pr-n
CH (Et) SEt Pr-i
CH (Et) SEt Pr-c
CH (Et) SEt Bu-n
CH (Et) SEt Bu-i
CH (Et) SEt Bu-c
CH (Et) SEt Bu-s
CH (Et) SEt Bu-t
CH (Et) SEt Pen-n
CH (Et) SEt Pen-c
CH (Et) SEt Hex-n
CH (Et) S (O) Et Me
CH (Et) S (O) Et Et
CH (Et) S (O) Et Pr-n
CH (Et) S (O) Et Pr-i
CH (Et) S (O) Et Pr-c
CH (Et) S (O) Et Bu-n
CH (Et) S (O) Et Bu-i
CH (Et) S (O) Et Bu-c
CH (Et) S (O) Et Bu-s
CH (Et) S (O) Et Bu-t
CH (Et) S (O) Et Pen-n
CH (Et) S (O) Et Pen-c
CH (Et) S (O) Et Hex-n
CH (Et) S (O)2Et Me
CH (Et) S (O)2Et Et
CH (Et) S (O)2Et Pr-n
CH (Et) S (O)2Et Pr-i
CH (Et) S (O)2Et Pr-c
CH (Et) S (O)2Et Bu-n
CH (Et) S (O)2Et Bu-i
CH (Et) S (O)2Et Bu-c
CH (Et) S (O)2Et Bu-s
CH (Et) S (O)2Et Bu-t
CH (Et) S (O)2Et Pen-n
CH (Et) S (O)2Et Pen-c
CH (Et) S (O)2Et Hex-n
CH2SCH2CH2CN Me
CH2SCH2CH2CN Et
CH2SCH2CH2CN Pr-n
CH2SCH2CH2CN Pr-i
CH2SCH2CH2CN Pr-c
CH2SCH2CH2CN Bu-n
CH2SCH2CH2CN Bu-i
CH2SCH2CH2CN Bu-c
CH2SCH2CH2CN Bu-s
CH2SCH2CH2CN Bu-t
CH2SCH2CH2CN Pen-n
CH2SCH2CH2CN Pen-c
CH2SCH2CH2CN Hex-n
CH2S (O) CH2CH2CN Me
CH2S (O) CH2CH2CN Et
CH2S (O) CH2CH2CN Pr-n
CH2S (O) CH2CH2CN Pr-i
CH2S (O) CH2CH2CN Pr-c
CH2S (O) CH2CH2CN Bu-n
CH2S (O) CH2CH2CN Bu-i
CH2S (O) CH2CH2CN Bu-c
CH2S (O) CH2CH2CN Bu-s
CH2S (O) CH2CH2CN Bu-t
CH2S (O) CH2CH2CN Pen-n
CH2S (O) CH2CH2CN Pen-c
CH2S (O) CH2CH2CN Hex-n
CH2S (O)2CH2CH2CN Me
CH2S (O)2CH2CH2CN Et
CH2S (O)2CH2CH2CN Pr-n
CH2S (O)2CH2CH2CN Pr-i
CH2S (O)2CH2CH2CN Pr-c
CH2S (O)2CH2CH2CN Bu-n
CH2S (O)2CH2CH2CN Bu-i
CH2S (O)2CH2CH2CN Bu-c
CH2S (O)2CH2CH2CN Bu-s
CH2S (O)2CH2CH2CN Bu-t
CH2S (O)2CH2CH2CN Pen-n
CH2S (O)2CH2CH2CN Pen-c
CH2S (O)2CH2CH2CN Hex-n
CH (Me) SCH2CH2CN Me
CH (Me) SCH2CH2CN Et
CH (Me) SCH2CH2CN Pr-n
CH (Me) SCH2CH2CN Pr-i
CH (Me) SCH2CH2CN Pr-c
CH (Me) SCH2CH2CN Bu-n
CH (Me) SCH2CH2CN Bu-i
CH (Me) SCH2CH2CN Bu-c
CH (Me) SCH2CH2CN Bu-s
CH (Me) SCH2CH2CN Bu-t
CH (Me) SCH2CH2CN Pen-n
CH (Me) SCH2CH2CN Pen-c
CH (Me) SCH2CH2CN Hex-n
CH (Me) S (O) CH2CH2CN Me
CH (Me) S (O) CH2CH2CN Et
CH (Me) S (O) CH2CH2CN Pr-n
CH (Me) S (O) CH2CH2CN Pr-i
CH (Me) S (O) CH2CH2CN Pr-c
CH (Me) S (O) CH2CH2CN Bu-n
CH (Me) S (O) CH2CH2CN Bu-i
CH (Me) S (O) CH2CH2CN Bu-c
CH (Me) S (O) CH2CH2CN Bu-s
CH (Me) S (O) CH2CH2CN Bu-t
CH (Me) S (O) CH2CH2CN Pen-n
CH (Me) S (O) CH2CH2CN Pen-c
CH (Me) S (O) CH2CH2CN Hex-n
CH (Me) S (O)2CH2CH2CN Me
CH (Me) S (O)2CH2CH2CN Et
CH (Me) S (O)2CH2CH2CN Pr-n
CH (Me) S (O)2CH2CH2CN Pr-i
CH (Me) S (O)2CH2CH2CN Pr-c
CH (Me) S (O)2CH2CH2CN Bu-n
CH (Me) S (O)2CH2CH2CN Bu-i
CH (Me) S (O)2CH2CH2CN Bu-c
CH (Me) S (O)2CH2CH2CN Bu-s
CH (Me) S (O)2CH2CH2CN Bu-t
CH (Me) S (O)2CH2CH2CN Pen-n
CH (Me) S (O)2CH2CH2CN Pen-c
CH (Me) S (O)2CH2CH2CN Hex-n
CH (Et) SCH2CH2CN Me
CH (Et) SCH2CH2CN Et
CH (Et) SCH2CH2CN Pr-n
CH (Et) SCH2CH2CN Pr-i
CH (Et) SCH2CH2CN Pr-c
CH (Et) SCH2CH2CN Bu-n
CH (Et) SCH2CH2CN Bu-i
CH (Et) SCH2CH2CN Bu-c
CH (Et) SCH2CH2CN Bu-s
CH (Et) SCH2CH2CN Bu-t
CH (Et) SCH2CH2CN Pen-n
CH (Et) SCH2CH2CN Pen-c
CH (Et) SCH2CH2CN Hex-n
CH (Et) S (O) CH2CH2CN Me
CH (Et) S (O) CH2CH2CN Et
CH (Et) S (O) CH2CH2CN Pr-n
CH (Et) S (O) CH2CH2CN Pr-i
CH (Et) S (O) CH2CH2CN Pr-c
CH (Et) S (O) CH2CH2CN Bu-n
CH (Et) S (O) CH2CH2CN Bu-i
CH (Et) S (O) CH2CH2CN Bu-c
CH (Et) S (O) CH2CH2CN Bu-s
CH (Et) S (O) CH2CH2CN Bu-t
CH (Et) S (O) CH2CH2CN Pen-n
CH (Et) S (O) CH2CH2CN Pen-c
CH (Et) S (O) CH2CH2CN Hex-n
CH (Et) S (O)2CH2CH2CN Me
CH (Et) S (O)2CH2CH2CN Et
CH (Et) S (O)2CH2CH2CN Pr-n
CH (Et) S (O)2CH2CH2CN Pr-i
CH (Et) S (O)2CH2CH2CN Pr-c
CH (Et) S (O)2CH2CH2CN Bu-n
CH (Et) S (O)2CH2CH2CN Bu-i
CH (Et) S (O)2CH2CH2CN Bu-c
CH (Et) S (O)2CH2CH2CN Bu-s
CH (Et) S (O)2CH2CH2CN Bu-t
CH (Et) S (O)2CH2CH2CN Pen-n
CH (Et) S (O)2CH2CH2CN Pen-c
CH (Et) S (O)2CH2CH2CN Hex-n
CH2SC (O) Me Me
CH2CH2SC (O) Me Me
CH (Me) SC (O) Me Me
CH (Me) CH2SC (O) Me Me
CH (Et) SC (O) Me Me
CH (Et) CH2SC (O) Me Me
CH2SCFThree                             Me
CH2SCFThree                             Et
CH2SCFThree                             Pr-n
CH2SCFThree                             Pr-i
CH2SCFThree                             Pr-c
CH2SCFThree                             Bu-n
CH2SCFThree                             Bu-i
CH2SCFThree                             Bu-c
CH2SCFThree                             Bu-s
CH2SCFThree                             Bu-t
CH2SCFThree                             Pen-n
CH2SCFThree                             Pen-c
CH2SCFThree                             Hex-n
CH2SCFThree                             Hex-c
CH2SCFThree                             CH2Pr-c
CH2SCFThree                             CH2Bu-c
CH2SCFThree                             CH2Pen-c
CH2SCFThree                             CH2Hex-c
CH2SCFThree                             CH2CH = CH2
CH2SCFThree                             CH2CH = C (Cl)2
CH2SCFThree                             CH2C≡CH
CH2SCFThree                             CH2CN
CH2SCFThree                             CH2CFThree
CH2SCFThree                             CH2OMe
CH2SCFThree                             CH2OCFThree
CH2SCFThree                             CH2SMe
CH2SCFThree                             CH2S (O) Me
CH2SCFThree                             CH2S (O)2Me
CH2SCFThree                             CH2SCFThree
CH2SCFThree                             CH2S (O) CFThree
CH2SCFThree                             CH2S (O)2CFThree
CH2SCFThree                             CH2CH (OMe)2
CH2SCFThree                             CH2CH (SMe)2
CH2SCFThree                             CH2C (O) Me
CH2SCFThree                             CH2C (O) CFThree
CH2SCFThree                             CH2C (O) OMe
CH2SCFThree                             CH2(D1-32a)
CH2SCFThree                             CH2(D1-33a)
CH2SCFThree                             CH2(D1-34a)
CH2SCFThree                             CH2(D1-37a)
CH2SCFThree                             CH2(D1-81a)
CH2SCFThree                             CH2(D1-82a)
CH2SCFThree                             CH2(D1-84a)
CH2SCFThree                             CH2(D1-85a)
CH2SCFThree                             CH2(D1-87a)
CH2SCFThree                             CH2(D1-92a)
CH2SCFThree                             CH2(D1-93a)
CH2SCFThree                             CH2(D1-95a)
CH2SCFThree                             CH2(D1-96a)
CH2SCFThree                             CH2(D1-98a)
CH2SCFThree                             CH2(D1-108a)
CH2SCFThree                             CH2(D1-108b, Z = 2-Cl)
CH2SCFThree                             CH2(D1-108b, Z = 3-Me)
CH2SCFThree                             CH2(D1-108b, Z = 4-OMe)
CH2SCFThree                             CH2(D1-108b, Z = 2-SMe)
CH2SCFThree                             CH2(D1-108b, Z = 3-CFThree)
CH2SCFThree                             CH2(D1-108b, Z = 4-OCFThree)
CH2SCFThree                             CH2(D1-108b, Z = 2-SCFThree)
CH2SCFThree                             CH2CH2CN
CH2SCFThree                             CH2CH2CFThree
CH2SCFThree                             CH2CH2OMe
CH2SCFThree                             CH2CH2SMe
CH2SCFThree                             CH2CH2S (O) Me
CH2SCFThree                             CH2CH2S (O)2Me
CH2SCFThree                             D1-32a
CH2SCFThree                             D1-33a
CH2SCFThree                             D1-34a
CH2SCFThree                             D1-37a
CH2SCFThree                             D1-81a
CH2SCFThree                             D1-82a
CH2SCFThree                             D1-84a
CH2SCFThree                             D1-85a
CH2SCFThree                             D1-87a
CH2SCFThree                             D1-92a
CH2SCFThree                             D1-93a
CH2SCFThree                             D1-95a
CH2SCFThree                             D1-96a
CH2SCFThree                             D1-98a
CH2SCFThree                             D1-108a
CH2SCFThree                             D1-108b (Z = 2-Cl)
CH2SCFThree                             D1-108b (Z = 3-Me)
CH2SCFThree                             D1-108b (Z = 4-OMe)
CH2SCFThree                             D1-108b (Z = 2-SMe)
CH2SCFThree                             D1-108b (Z = 3-CFThree)
CH2SCFThree                             D1-108b (Z = 4-OCFThree)
CH2SCFThree                             D1-108b (Z = 2-SCFThree)
CH2SCFThree                             C (O) Me
CH2SCFThree                             C (O) CFThree
CH2SCFThree                             C (O) OMe
CH2S (O) CFThree                          Me
CH2S (O) CFThree                          Et
CH2S (O) CFThree                          Pr-n
CH2S (O) CFThree                          Pr-i
CH2S (O) CFThree                          Pr-c
CH2S (O) CFThree                          Bu-n
CH2S (O) CFThree                          Bu-i
CH2S (O) CFThree                          Bu-c
CH2S (O) CFThree                          Bu-s
CH2S (O) CFThree                          Bu-t
CH2S (O) CFThree                          Pen-n
CH2S (O) CFThree                          Pen-c
CH2S (O) CFThree                          Hex-n
CH2S (O) CFThree                          Hex-c
CH2S (O) CFThree                          CH2Pr-c
CH2S (O) CFThree                          CH2Bu-c
CH2S (O) CFThree                          CH2Pen-c
CH2S (O) CFThree                          CH2Hex-c
CH2S (O) CFThree                          CH2CH = CH2
CH2S (O) CFThree                          CH2CH = C (Cl)2
CH2S (O) CFThree                          CH2C≡CH
CH2S (O) CFThree                          CH2CN
CH2S (O) CFThree                          CH2CFThree
CH2S (O) CFThree                          CH2OMe
CH2S (O) CFThree                          CH2OCFThree
CH2S (O) CFThree                          CH2SMe
CH2S (O) CFThree                          CH2S (O) Me
CH2S (O) CFThree                          CH2S (O)2Me
CH2S (O) CFThree                          CH2SCFThree
CH2S (O) CFThree                          CH2S (O) CFThree
CH2S (O) CFThree                          CH2S (O)2CFThree
CH2S (O) CFThree                          CH2CH (OMe)2
CH2S (O) CFThree                          CH2CH (SMe)2
CH2S (O) CFThree                          CH2C (O) Me
CH2S (O) CFThree                          CH2C (O) CFThree
CH2S (O) CFThree                          CH2C (O) OMe
CH2S (O) CFThree                          CH2(D1-32a)
CH2S (O) CFThree                          CH2(D1-33a)
CH2S (O) CFThree                          CH2(D1-34a)
CH2S (O) CFThree                          CH2(D1-37a)
CH2S (O) CFThree                          CH2(D1-81a)
CH2S (O) CFThree                          CH2(D1-82a)
CH2S (O) CFThree                          CH2(D1-84a)
CH2S (O) CFThree                          CH2(D1-85a)
CH2S (O) CFThree                          CH2(D1-87a)
CH2S (O) CFThree                          CH2(D1-92a)
CH2S (O) CFThree                          CH2(D1-93a)
CH2S (O) CFThree                          CH2(D1-95a)
CH2S (O) CFThree                          CH2(D1-96a)
CH2S (O) CFThree                          CH2(D1-98a)
CH2S (O) CFThree                          CH2(D1-108a)
CH2S (O) CFThree                          CH2(D1-108b, Z = 2-Cl)
CH2S (O) CFThree                          CH2(D1-108b, Z = 3-Me)
CH2S (O) CFThree                          CH2(D1-108b, Z = 4-OMe)
CH2S (O) CFThree                          CH2(D1-108b, Z = 2-SMe)
CH2S (O) CFThree                          CH2(D1-108b, Z = 3-CFThree)
CH2S (O) CFThree                          CH2(D1-108b, Z = 4-OCFThree)
CH2S (O) CFThree                          CH2(D1-108b, Z = 2-SCFThree)
CH2S (O) CFThree                          CH2CH2CN
CH2S (O) CFThree                          CH2CH2CFThree
CH2S (O) CFThree                          CH2CH2OMe
CH2S (O) CFThree                          CH2CH2SMe
CH2S (O) CFThree                          CH2CH2S (O) Me
CH2S (O) CFThree                          CH2CH2S (O)2Me
CH2S (O) CFThree                          D1-32a
CH2S (O) CFThree                          D1-33a
CH2S (O) CFThree                          D1-34a
CH2S (O) CFThree                          D1-37a
CH2S (O) CFThree                          D1-81a
CH2S (O) CFThree                          D1-82a
CH2S (O) CFThree                          D1-84a
CH2S (O) CFThree                          D1-85a
CH2S (O) CFThree                          D1-87a
CH2S (O) CFThree                          D1-92a
CH2S (O) CFThree                          D1-93a
CH2S (O) CFThree                          D1-95a
CH2S (O) CFThree                          D1-96a
CH2S (O) CFThree                          D1-98a
CH2S (O) CFThree                          D1-108a
CH2S (O) CFThree                          D1-108b (Z = 2-Cl)
CH2S (O) CFThree                          D1-108b (Z = 3-Me)
CH2S (O) CFThree                          D1-108b (Z = 4-OMe)
CH2S (O) CFThree                          D1-108b (Z = 2-SMe)
CH2S (O) CFThree                          D1-108b (Z = 3-CFThree)
CH2S (O) CFThree                          D1-108b (Z = 4-OCFThree)
CH2S (O) CFThree                          D1-108b (Z = 2-SCFThree)
CH2S (O) CFThree                          C (O) Me
CH2S (O) CFThree                          C (O) CFThree
CH2S (O) CFThree                          C (O) OMe
CH2S (O)2CFThree                          Me
CH2S (O)2CFThree                          Et
CH2S (O)2CFThree                          Pr-n
CH2S (O)2CFThree                          Pr-i
CH2S (O)2CFThree                          Pr-c
CH2S (O)2CFThree                          Bu-n
CH2S (O)2CFThree                          Bu-i
CH2S (O)2CFThree                          Bu-c
CH2S (O)2CFThree                          Bu-s
CH2S (O)2CFThree                          Bu-t
CH2S (O)2CFThree                          Pen-n
CH2S (O)2CFThree                          Pen-c
CH2S (O)2CFThree                          Hex-n
CH2S (O)2CFThree                          Hex-c
CH2S (O)2CFThree                          CH2Pr-c
CH2S (O)2CFThree                          CH2Bu-c
CH2S (O)2CFThree                          CH2Pen-c
CH2S (O)2CFThree                          CH2Hex-c
CH2S (O)2CFThree                          CH2CH = CH2
CH2S (O)2CFThree                          CH2CH = C (Cl)2
CH2S (O)2CFThree                          CH2C≡CH
CH2S (O)2CFThree                          CH2CN
CH2S (O)2CFThree                          CH2CFThree
CH2S (O)2CFThree                          CH2OMe
CH2S (O)2CFThree                          CH2OCFThree
CH2S (O)2CFThree                          CH2SMe
CH2S (O)2CFThree                          CH2S (O) Me
CH2S (O)2CFThree                          CH2S (O)2Me
CH2S (O)2CFThree                          CH2SCFThree
CH2S (O)2CFThree                          CH2S (O) CFThree
CH2S (O)2CFThree                          CH2S (O)2CFThree
CH2S (O)2CFThree                          CH2CH (OMe)2
CH2S (O)2CFThree                          CH2CH (SMe)2
CH2S (O)2CFThree                          CH2C (O) Me
CH2S (O)2CFThree                          CH2C (O) CFThree
CH2S (O)2CFThree                          CH2C (O) OMe
CH2S (O)2CFThree                          CH2(D1-32a)
CH2S (O)2CFThree                          CH2(D1-33a)
CH2S (O)2CFThree                          CH2(D1-34a)
CH2S (O)2CFThree                          CH2(D1-37a)
CH2S (O)2CFThree                          CH2(D1-81a)
CH2S (O)2CFThree                          CH2(D1-82a)
CH2S (O)2CFThree                          CH2(D1-84a)
CH2S (O)2CFThree                          CH2(D1-85a)
CH2S (O)2CFThree                          CH2(D1-87a)
CH2S (O)2CFThree                          CH2(D1-92a)
CH2S (O)2CFThree                          CH2(D1-93a)
CH2S (O)2CFThree                          CH2(D1-95a)
CH2S (O)2CFThree                          CH2(D1-96a)
CH2S (O)2CFThree                          CH2(D1-98a)
CH2S (O)2CFThree                          CH2(D1-108a)
CH2S (O)2CFThree                          CH2(D1-108b, Z = 2-Cl)
CH2S (O)2CFThree                          CH2(D1-108b, Z = 3-Me)
CH2S (O)2CFThree                          CH2(D1-108b, Z = 4-OMe)
CH2S (O)2CFThree                          CH2(D1-108b, Z = 2-SMe)
CH2S (O)2CFThree                          CH2(D1-108b, Z = 3-CFThree)
CH2S (O)2CFThree                          CH2(D1-108b, Z = 4-OCFThree)
CH2S (O)2CFThree                          CH2(D1-108b, Z = 2-SCFThree)
CH2S (O)2CFThree                          CH2CH2CN
CH2S (O)2CFThree                          CH2CH2CFThree
CH2S (O)2CFThree                          CH2CH2OMe
CH2S (O)2CFThree                          CH2CH2SMe
CH2S (O)2CFThree                          CH2CH2S (O) Me
CH2S (O)2CFThree                          CH2CH2S (O)2Me
CH2S (O)2CFThree                          D1-32a
CH2S (O)2CFThree                          D1-33a
CH2S (O)2CFThree                          D1-34a
CH2S (O)2CFThree                          D1-37a
CH2S (O)2CFThree                          D1-81a
CH2S (O)2CFThree                          D1-82a
CH2S (O)2CFThree                          D1-84a
CH2S (O)2CFThree                          D1-85a
CH2S (O)2CFThree                          D1-87a
CH2S (O)2CFThree                          D1-92a
CH2S (O)2CFThree                          D1-93a
CH2S (O)2CFThree                          D1-95a
CH2S (O)2CFThree                          D1-96a
CH2S (O)2CFThree                          D1-98a
CH2S (O)2CFThree                          D1-108a
CH2S (O)2CFThree                          D1-108b (Z = 2-Cl)
CH2S (O)2CFThree                          D1-108b (Z = 3-Me)
CH2S (O)2CFThree                          D1-108b (Z = 4-OMe)
CH2S (O)2CFThree                          D1-108b (Z = 2-SMe)
CH2S (O)2CFThree                          D1-108b (Z = 3-CFThree)
CH2S (O)2CFThree                          D1-108b (Z = 4-OCFThree)
CH2S (O)2CFThree                          D1-108b (Z = 2-SCFThree)
CH2S (O)2CFThree                          C (O) Me
CH2S (O)2CFThree                          C (O) CFThree
CH2S (O)2CFThree                          C (O) OMe
CH2CH2SCFThree                           Me
CH2CH2SCFThree                           Et
CH2CH2SCFThree                           Pr-n
CH2CH2SCFThree                           Pr-i
CH2CH2SCFThree                           Pr-c
CH2CH2SCFThree                           Bu-n
CH2CH2SCFThree                           Bu-i
CH2CH2SCFThree                           Bu-c
CH2CH2SCFThree                           Bu-s
CH2CH2SCFThree                           Bu-t
CH2CH2SCFThree                           Pen-n
CH2CH2SCFThree                           Pen-c
CH2CH2SCFThree                           Hex-n
CH2CH2SCFThree                           Hex-c
CH2CH2SCFThree                           CH2Pr-c
CH2CH2SCFThree                           CH2Bu-c
CH2CH2SCFThree                           CH2Pen-c
CH2CH2SCFThree                           CH2Hex-c
CH2CH2SCFThree                           CH2CH = CH2
CH2CH2SCFThree                           CH2CH = C (Cl)2
CH2CH2SCFThree                           CH2C≡CH
CH2CH2SCFThree                           CH2CN
CH2CH2SCFThree                           CH2CFThree
CH2CH2SCFThree                           CH2OMe
CH2CH2SCFThree                           CH2OCFThree
CH2CH2SCFThree                           CH2SMe
CH2CH2SCFThree                           CH2S (O) Me
CH2CH2SCFThree                           CH2S (O)2Me
CH2CH2SCFThree                           CH2SCFThree
CH2CH2SCFThree                           CH2S (O) CFThree
CH2CH2SCFThree                           CH2S (O)2CFThree
CH2CH2SCFThree                           CH2CH (OMe)2
CH2CH2SCFThree                           CH2CH (SMe)2
CH2CH2SCFThree                           CH2C (O) Me
CH2CH2SCFThree                           CH2C (O) CFThree
CH2CH2SCFThree                           CH2C (O) OMe
CH2CH2SCFThree                           CH2(D1-32a)
CH2CH2SCFThree                           CH2(D1-33a)
CH2CH2SCFThree                           CH2(D1-34a)
CH2CH2SCFThree                           CH2(D1-37a)
CH2CH2SCFThree                           CH2(D1-81a)
CH2CH2SCFThree                           CH2(D1-82a)
CH2CH2SCFThree                           CH2(D1-84a)
CH2CH2SCFThree                           CH2(D1-85a)
CH2CH2SCFThree                           CH2(D1-87a)
CH2CH2SCFThree                           CH2(D1-92a)
CH2CH2SCFThree                           CH2(D1-93a)
CH2CH2SCFThree                           CH2(D1-95a)
CH2CH2SCFThree                           CH2(D1-96a)
CH2CH2SCFThree                           CH2(D1-98a)
CH2CH2SCFThree                           CH2(D1-108a)
CH2CH2SCFThree                           CH2(D1-108b, Z = 2-Cl)
CH2CH2SCFThree                           CH2(D1-108b, Z = 3-Me)
CH2CH2SCFThree                           CH2(D1-108b, Z = 4-OMe)
CH2CH2SCFThree                           CH2(D1-108b, Z = 2-SMe)
CH2CH2SCFThree                           CH2(D1-108b, Z = 3-CFThree)
CH2CH2SCFThree                           CH2(D1-108b, Z = 4-OCFThree)
CH2CH2SCFThree                           CH2(D1-108b, Z = 2-SCFThree)
CH2CH2SCFThree                           CH2CH2CN
CH2CH2SCFThree                           CH2CH2CFThree
CH2CH2SCFThree                           CH2CH2OMe
CH2CH2SCFThree                           CH2CH2SMe
CH2CH2SCFThree                           CH2CH2S (O) Me
CH2CH2SCFThree                           CH2CH2S (O)2Me
CH2CH2SCFThree                           D1-32a
CH2CH2SCFThree                           D1-33a
CH2CH2SCFThree                           D1-34a
CH2CH2SCFThree                           D1-37a
CH2CH2H2SCFThree                          D1-81a
CH2CH2SCFThree                           D1-82a
CH2CH2SCFThree                           D1-84a
CH2CH2SCFThree                           D1-85a
CH2CH2SCFThree                           D1-87a
CH2CH2SCFThree                           D1-92a
CH2CH2SCFThree                           D1-93a
CH2CH2SCFThree                           D1-95a
CH2CH2SCFThree                           D1-96a
CH2CH2SCFThree                           D1-98a
CH2CH2SCFThree                           D1-108a
CH2CH2SCFThree                           D1-108b (Z = 2-Cl)
CH2CH2SCFThree                           D1-108b (Z = 3-Me)
CH2CH2SCFThree                           D1-108b (Z = 4-OMe)
CH2CH2SCFThree                           D1-108b (Z = 2-SMe)
CH2CH2SCFThree                           D1-108b (Z = 3-CFThree)
CH2CH2SCFThree                           D1-108b (Z = 4-OCFThree)
CH2CH2SCFThree                           D1-108b (Z = 2-SCFThree)
CH2CH2SCFThree                           C (O) Me
CH2CH2SCFThree                           C (O) CFThree
CH2CH2SCFThree                           C (O) OMe
CH2CH2S (O) CFThree                        Me
CH2CH2S (O) CFThree                        Et
CH2CH2S (O) CFThree                        Pr-n
CH2CH2S (O) CFThree                        Pr-i
CH2CH2S (O) CFThree                        Pr-c
CH2CH2S (O) CFThree                        Bu-n
CH2CH2S (O) CFThree                        Bu-i
CH2CH2S (O) CFThree                        Bu-c
CH2CH2S (O) CFThree                        Bu-s
CH2CH2S (O) CFThree                        Bu-t
CH2CH2S (O) CFThree                        Pen-n
CH2CH2S (O) CFThree                        Pen-c
CH2CH2S (O) CFThree                        Hex-n
CH2CH2S (O) CFThree                        Hex-c
CH2CH2S (O) CFThree                        CH2Pr-c
CH2CH2S (O) CFThree                        CH2Bu-c
CH2CH2S (O) CFThree                        CH2Pen-c
CH2CH2S (O) CFThree                        CH2Hex-c
CH2CH2S (O) CFThree                        CH2CH = CH2
CH2CH2S (O) CFThree                        CH2CH = C (Cl)2
CH2CH2S (O) CFThree                        CH2C≡CH
CH2CH2S (O) CFThree                        CH2CN
CH2CH2S (O) CFThree                        CH2CFThree
CH2CH2S (O) CFThree                        CH2OMe
CH2CH2S (O) CFThree                        CH2OCFThree
CH2CH2S (O) CFThree                        CH2SMe
CH2CH2S (O) CFThree                        CH2S (O) Me
CH2CH2S (O) CFThree                        CH2S (O)2Me
CH2CH2S (O) CFThree                        CH2SCFThree
CH2CH2S (O) CFThree                        CH2S (O) CFThree
CH2CH2S (O) CFThree                        CH2S (O)2CFThree
CH2CH2S (O) CFThree                        CH2CH (OMe)2
CH2CH2S (O) CFThree                        CH2CH (SMe)2
CH2CH2S (O) CFThree                        CH2C (O) Me
CH2CH2S (O) CFThree                        CH2C (O) CFThree
CH2CH2S (O) CFThree                        CH2C (O) OMe
CH2CH2S (O) CFThree                        CH2(D1-32a)
CH2CH2S (O) CFThree                        CH2(D1-33a)
CH2CH2S (O) CFThree                        CH2(D1-34a)
CH2CH2S (O) CFThree                        CH2(D1-37a)
CH2CH2S (O) CFThree                        CH2(D1-81a)
CH2CH2S (O) CFThree                        CH2(D1-82a)
CH2CH2S (O) CFThree                        CH2(D1-84a)
CH2CH2S (O) CFThree                        CH2(D1-85a)
CH2CH2S (O) CFThree                        CH2(D1-87a)
CH2CH2S (O) CFThree                        CH2(D1-92a)
CH2CH2S (O) CFThree                        CH2(D1-93a)
CH2CH2S (O) CFThree                        CH2(D1-95a)
CH2CH2S (O) CFThree                        CH2(D1-96a)
CH2CH2S (O) CFThree                        CH2(D1-98a)
CH2CH2S (O) CFThree                        CH2(D1-108a)
CH2CH2S (O) CFThree                        CH2(D1-108b, Z = 2-Cl)
CH2CH2S (O) CFThree                        CH2(D1-108b, Z = 3-Me)
CH2CH2S (O) CFThree                        CH2(D1-108b, Z = 4-OMe)
CH2CH2S (O) CFThree                        CH2(D1-108b, Z = 2-SMe)
CH2CH2S (O) CFThree                        CH2(D1-108b, Z = 3-CFThree)
CH2CH2S (O) CFThree                        CH2(D1-108b, Z = 4-OCFThree)
CH2CH2S (O) CFThree                        CH2(D1-108b, Z = 2-SCFThree)
CH2CH2S (O) CFThree                        CH2CH2CN
CH2CH2S (O) CFThree                        CH2CH2CFThree
CH2CH2S (O) CFThree                        CH2CH2OMe
CH2CH2S (O) CFThree                        CH2CH2SMe
CH2CH2S (O) CFThree                        CH2CH2S (O) Me
CH2CH2S (O) CFThree                        CH2CH2S (O)2Me
CH2CH2S (O) CFThree                        D1-32a
CH2CH2S (O) CFThree                        D1-33a
CH2CH2S (O) CFThree                        D1-34a
CH2CH2S (O) CFThree                        D1-37a
CH2CH2S (O) CFThree                        D1-81a
CH2CH2S (O) CFThree                        D1-82a
CH2CH2S (O) CFThree                        D1-84a
CH2CH2S (O) CFThree                        D1-85a
CH2CH2S (O) CFThree                        D1-87a
CH2CH2S (O) CFThree                        D1-92a
CH2CH2S (O) CFThree                        D1-93a
CH2CH2S (O) CFThree                        D1-95a
CH2CH2S (O) CFThree                        D1-96a
CH2CH2S (O) CFThree                        D1-98a
CH2CH2S (O) CFThree                        D1-108a
CH2CH2S (O) CFThree                        D1-108b (Z = 2-Cl)
CH2CH2S (O) CFThree                        D1-108b (Z = 3-Me)
CH2CH2S (O) CFThree                        D1-108b (Z = 4-OMe)
CH2CH2S (O) CFThree                        D1-108b (Z = 2-SMe)
CH2CH2S (O) CFThree                        D1-108b (Z = 3-CFThree)
CH2CH2S (O) CFThree                        D1-108b (Z = 4-OCFThree)
CH2CH2S (O) CFThree                        D1-108b (Z = 2-SCFThree)
CH2CH2S (O) CFThree                        C (O) Me
CH2CH2S (O) CFThree                        C (O) CFThree
CH2CH2S (O) CFThree                        C (O) OMe
CH2CH2S (O)2CFThree                       Me
CH2CH2S (O)2CFThree                       Et
CH2CH2S (O)2CFThree                       Pr-n
CH2CH2S (O)2CFThree                       Pr-i
CH2CH2S (O)2CFThree                       Pr-c
CH2CH2S (O)2CFThree                       Bu-n
CH2CH2S (O)2CFThree                       Bu-i
CH2CH2S (O)2CFThree                       Bu-c
CH2CH2S (O)2CFThree                       Bu-s
CH2CH2S (O)2CFThree                       Bu-t
CH2CH2S (O)2CFThree                       Pen-n
CH2CH2S (O)2CFThree                       Pen-c
CH2CH2S (O)2CFThree                       Hex-n
CH2CH2S (O)2CFThree                       Hex-c
CH2CH2S (O)2CFThree                       CH2Pr-c
CH2CH2S (O)2CFThree                       CH2Bu-c
CH2CH2S (O)2CFThree                       CH2Pen-c
CH2CH2S (O)2CFThree                       CH2Hex-c
CH2CH2S (O)2CFThree                       CH2CH = CH2
CH2CH2S (O)2CFThree                       CH2CH = C (Cl)2
CH2CH2S (O)2CFThree                       CH2C≡CH
CH2CH2S (O)2CFThree                       CH2CN
CH2CH2S (O)2CFThree                       CH2CFThree
CH2CH2S (O)2CFThree                       CH2OMe
CH2CH2S (O)2CFThree                       CH2OCFThree
CH2CH2S (O)2CFThree                       CH2SMe
CH2CH2S (O)2CFThree                       CH2S (O) Me
CH2CH2S (O)2CFThree                       CH2S (O)2Me
CH2CH2S (O)2CFThree                       CH2SCFThree
CH2CH2S (O)2CFThree                       CH2S (O) CFThree
CH2CH2S (O)2CFThree                       CH2S (O)2CFThree
CH2CH2S (O)2CFThree                       CH2CH (OMe)2
CH2CH2S (O)2CFThree                       CH2CH (SMe)2
CH2CH2S (O)2CFThree                       CH2C (O) Me
CH2CH2S (O)2CFThree                       CH2C (O) CFThree
CH2CH2S (O)2CFThree                       CH2C (O) OMe
CH2CH2S (O)2CFThree                       CH2(D1-32a)
CH2CH2S (O)2CFThree                       CH2(D1-33a)
CH2CH2S (O)2CFThree                       CH2(D1-34a)
CH2CH2S (O)2CFThree                       CH2(D1-37a)
CH2CH2S (O)2CFThree                       CH2(D1-81a)
CH2CH2S (O)2CFThree                       CH2(D1-82a)
CH2CH2S (O)2CFThree                       CH2(D1-84a)
CH2CH2S (O)2CFThree                       CH2(D1-85a)
CH2CH2S (O)2CFThree                       CH2(D1-87a)
CH2CH2S (O)2CFThree                       CH2(D1-92a)
CH2CH2S (O)2CFThree                       CH2(D1-93a)
CH2CH2S (O)2CFThree                       CH2(D1-95a)
CH2CH2S (O)2CFThree                       CH2(D1-96a)
CH2CH2S (O)2CFThree                       CH2(D1-98a)
CH2CH2S (O)2CFThree                       CH2(D1-108a)
CH2CH2S (O)2CFThree                       CH2(D1-108b, Z = 2-Cl)
CH2CH2S (O)2CFThree                       CH2(D1-108b, Z = 3-Me)
CH2CH2S (O)2CFThree                       CH2(D1-108b, Z = 4-OMe)
CH2CH2S (O)2CFThree                       CH2(D1-108b, Z = 2-SMe)
CH2CH2S (O)2CFThree                       CH2(D1-108b, Z = 3-CFThree)
CH2CH2S (O)2CFThree                       CH2(D1-108b, Z = 4-OCFThree)
CH2CH2S (O)2CFThree                       CH2(D1-108b, Z = 2-SCFThree)
CH2CH2S (O)2CFThree                       CH2CH2CN
CH2CH2S (O)2CFThree                       CH2CH2CFThree
CH2CH2S (O)2CFThree                       CH2CH2OMe
CH2CH2S (O)2CFThree                       CH2CH2SMe
CH2CH2S (O)2CFThree                       CH2CH2S (O) Me
CH2CH2S (O)2CFThree                       CH2CH2S (O)2Me
CH2CH2S (O)2CFThree                       D1-32a
CH2CH2S (O)2CFThree                       D1-33a
CH2CH2S (O)2CFThree                       D1-34a
CH2CH2S (O)2CFThree                       D1-37a
CH2CH2S (O)2CFThree                       D1-81a
CH2CH2S (O)2CFThree                       D1-82a
CH2CH2S (O)2CFThree                       D1-84a
CH2CH2S (O)2CFThree                       D1-85a
CH2CH2S (O)2CFThree                       D1-87a
CH2CH2S (O)2CFThree                       D1-92a
CH2CH2S (O)2CFThree                       D1-93a
CH2CH2S (O)2CFThree                       D1-95a
CH2CH2S (O)2CFThree                       D1-96a
CH2CH2S (O)2CFThree                       D1-98a
CH2CH2S (O)2CFThree                       D1-108a
CH2CH2S (O)2CFThree                       D1-108b (Z = 2-Cl)
CH2CH2S (O)2CFThree                       D1-108b (Z = 3-Me)
CH2CH2S (O)2CFThree                       D1-108b (Z = 4-OMe)
CH2CH2S (O)2CFThree                       D1-108b (Z = 2-SMe)
CH2CH2S (O)2CFThree                       D1-108b (Z = 3-CFThree)
CH2CH2S (O)2CFThree                       D1-108b (Z = 4-OCFThree)
CH2CH2S (O)2CFThree                       D1-108b (Z = 2-SCFThree)
CH2CH2S (O)2CFThree                       C (O) Me
CH2CH2S (O)2CFThree                       C (O) CFThree
CH2CH2S (O)2CFThree                       C (O) OMe
D1-32a Me
D1-32a Et
D1-32a Pr-n
D1-32a Pr-i
D1-32a Pr-c
D1-32a Bu-n
D1-32a Bu-i
D1-32a Bu-c
D1-32a Bu-s
D1-32a Bu-t
D1-32a Pen-n
D1-32a Pen-c
D1-32a Hex-n
D1-32a Hex-c
D1-32a CH2Pr-c
D1-32a CH2Bu-c
D1-32a CH2Pen-c
D1-32a CH2Hex-c
D1-32a CH2CH = CH2
D1-32a CH2CH = C (Cl)2
D1-32a CH2C≡CH
D1-32a CH2CN
D1-32a CH2CFThree
D1-32a CH2OMe
D1-32a CH2OCFThree
D1-32a CH2SMe
D1-32a CH2S (O) Me
D1-32a CH2S (O)2Me
D1-32a CH2SCFThree
D1-32a CH2S (O) CFThree
D1-32a CH2S (O)2CFThree
D1-32a CH2CH (OMe)2
D1-32a CH2CH (SMe)2
D1-32a CH2C (O) Me
D1-32a CH2C (O) CFThree
D1-32a CH2C (O) OMe
D1-32a CH2(D1-32a)
D1-32a CH2(D1-33a)
D1-32a CH2(D1-34a)
D1-32a CH2(D1-37a)
D1-32a CH2(D1-81a)
D1-32a CH2(D1-82a)
D1-32a CH2(D1-84a)
D1-32a CH2(D1-85a)
D1-32a CH2(D1-87a)
D1-32a CH2(D1-92a)
D1-32a CH2(D1-93a)
D1-32a CH2(D1-95a)
D1-32a CH2(D1-96a)
D1-32a CH2(D1-98a)
D1-32a CH2(D1-108a)
D1-32a CH2(D1-108b, Z = 2-Cl)
D1-32a CH2(D1-108b, Z = 3-Me)
D1-32a CH2(D1-108b, Z = 4-OMe)
D1-32a CH2(D1-108b, Z = 2-SMe)
D1-32a CH2(D1-108b, Z = 3-CFThree)
D1-32a CH2(D1-108b, Z = 4-OCFThree)
D1-32a CH2(D1-108b, Z = 2-SCFThree)
D1-32a CH2CH2CN
D1-32a CH2CH2CFThree
D1-32a CH2CH2OMe
D1-32a CH2CH2SMe
D1-32a CH2CH2S (O) Me
D1-32a CH2CH2S (O)2Me
D1-32a D1-32a
D1-32a D1-33a
D1-32a D1-34a
D1-32a D1-37a
D1-32a D1-81a
D1-32a D1-82a
D1-32a D1-84a
D1-32a D1-85a
D1-32a D1-87a
D1-32a D1-92a
D1-32a D1-93a
D1-32a D1-95a
D1-32a D1-96a
D1-32a D1-98a
D1-32a D1-108a
D1-32a D1-108b (Z = 2-Cl)
D1-32a D1-108b (Z = 3-Me)
D1-32a D1-108b (Z = 4-OMe)
D1-32a D1-108b (Z = 2-SMe)
D1-32a D1-108b (Z = 3-CFThree)
D1-32a D1-108b (Z = 4-OCFThree)
D1-32a D1-108b (Z = 2-SCFThree)
D1-32a C (O) Me
D1-32a C (O) CFThree
D1-32a C (O) OMe
D1-33a Me
D1-33a Et
D1-33a Pr-n
D1-33a Pr-i
D1-33a Pr-c
D1-33a Bu-n
D1-33a Bu-i
D1-33a Bu-c
D1-33a Bu-s
D1-33a Bu-t
D1-33a Pen-n
D1-33a Pen-c
D1-33a Hex-n
D1-33a Hex-c
D1-33a CH2Pr-c
D1-33a CH2Bu-c
D1-33a CH2Pen-c
D1-33a CH2Hex-c
D1-33a CH2CH = CH2
D1-33a CH2CH = C (Cl)2
D1-33a CH2C≡CH
D1-33a CH2CN
D1-33a CH2CFThree
D1-33a CH2OMe
D1-33a CH2OCFThree
D1-33a CH2SMe
D1-33a CH2S (O) Me
D1-33a CH2S (O)2Me
D1-33a CH2SCFThree
D1-33a CH2S (O) CFThree
D1-33a CH2S (O)2CFThree
D1-33a CH2CH (OMe)2
D1-33a CH2CH (SMe)2
D1-33a CH2C (O) Me
D1-33a CH2C (O) CFThree
D1-33a CH2C (O) OMe
D1-33a CH2(D1-32a)
D1-33a CH2(D1-33a)
D1-33a CH2(D1-34a)
D1-33a CH2(D1-37a)
D1-33a CH2(D1-81a)
D1-33a CH2(D1-82a)
D1-33a CH2(D1-84a)
D1-33a CH2(D1-85a)
D1-33a CH2(D1-87a)
D1-33a CH2(D1-92a)
D1-33a CH2(D1-93a)
D1-33a CH2(D1-95a)
D1-33a CH2(D1-96a)
D1-33a CH2(D1-98a)
D1-33a CH2(D1-108a)
D1-33a CH2(D1-108b, Z = 2-Cl)
D1-33a CH2(D1-108b, Z = 3-Me)
D1-33a CH2(D1-108b, Z = 4-OMe)
D1-33a CH2(D1-108b, Z = 2-SMe)
D1-33a CH2(D1-108b, Z = 3-CFThree)
D1-33a CH2(D1-108b, Z = 4-OCFThree)
D1-33a CH2(D1-108b, Z = 2-SCFThree)
D1-33a CH2CH2CN
D1-33a CH2CH2CFThree
D1-33a CH2CH2OMe
D1-33a CH2CH2SMe
D1-33a CH2CH2S (O) Me
D1-33a CH2CH2S (O)2Me
D1-33a D1-32a
D1-33a D1-33a
D1-33a D1-34a
D1-33a D1-37a
D1-33a D1-81a
D1-33a D1-82a
D1-33a D1-84a
D1-33a D1-85a
D1-33a D1-87a
D1-33a D1-92a
D1-33a D1-93a
D1-33a D1-95a
D1-33a D1-96a
D1-33a D1-98a
D1-33a D1-108a
D1-33a D1-108b (Z = 2-Cl)
D1-33a D1-108b (Z = 3-Me)
D1-33a D1-108b (Z = 4-OMe)
D1-33a D1-108b (Z = 2-SMe)
D1-33a D1-108b (Z = 3-CFThree)
D1-33a D1-108b (Z = 4-OCFThree)
D1-33a D1-108b (Z = 2-SCFThree)
D1-33a C (O) Me
D1-33a C (O) CFThree
D1-33a C (O) OMe
D1-34a Me
D1-34a Et
D1-34a Pr-n
D1-34a Pr-i
D1-34a Pr-c
D1-34a Bu-n
D1-34a Bu-i
D1-34a Bu-c
D1-34a Bu-s
D1-34a Bu-t
D1-34a Pen-n
D1-34a Pen-c
D1-34a Hex-n
D1-34a Hex-c
D1-34a CH2Pr-c
D1-34a CH2Bu-c
D1-34a CH2Pen-c
D1-34a CH2Hex-c
D1-34a CH2CH = CH2
D1-34a CH2CH = C (Cl)2
D1-34a CH2C≡CH
D1-34a CH2CN
D1-34a CH2CFThree
D1-34a CH2OMe
D1-34a CH2OCFThree
D1-34a CH2SMe
D1-34a CH2S (O) Me
D1-34a CH2S (O)2Me
D1-34a CH2SCFThree
D1-34a CH2S (O) CFThree
D1-34a CH2S (O)2CFThree
D1-34a CH2CH (OMe)2
D1-34a CH2CH (SMe)2
D1-34a CH2C (O) Me
D1-34a CH2C (O) CFThree
D1-34a CH2C (O) OMe
D1-34a CH2(D1-32a)
D1-34a CH2(D1-33a)
D1-34a CH2(D1-34a)
D1-34a CH2(D1-37a)
D1-34a CH2(D1-81a)
D1-34a CH2(D1-82a)
D1-34a CH2(D1-84a)
D1-34a CH2(D1-85a)
D1-34a CH2(D1-87a)
D1-34a CH2(D1-92a)
D1-34a CH2(D1-93a)
D1-34a CH2(D1-95a)
D1-34a CH2(D1-96a)
D1-34a CH2(D1-98a)
D1-34a CH2(D1-108a)
D1-34a CH2(D1-108b, Z = 2-Cl)
D1-34a CH2(D1-108b, Z = 3-Me)
D1-34a CH2(D1-108b, Z = 4-OMe)
D1-34a CH2(D1-108b, Z = 2-SMe)
D1-34a CH2(D1-108b, Z = 3-CFThree)
D1-34a CH2(D1-108b, Z = 4-OCFThree)
D1-34a CH2(D1-108b, Z = 2-SCFThree)
D1-34a CH2CH2CN
D1-34a CH2CH2CFThree
D1-34a CH2CH2OMe
D1-34a CH2CH2SMe
D1-34a CH2CH2S (O) Me
D1-34a CH2CH2S (O)2Me
D1-34a D1-32a
D1-34a D1-33a
D1-34a D1-34a
D1-34a D1-37a
D1-34a D1-81a
D1-34a D1-82a
D1-34a D1-84a
D1-34a D1-85a
D1-34a D1-87a
D1-34a D1-92a
D1-34a D1-93a
D1-34a D1-95a
D1-34a D1-96a
D1-34a D1-98a
D1-34a D1-108a
D1-34a D1-108b (Z = 2-Cl)
D1-34a D1-108b (Z = 3-Me)
D1-34a D1-108b (Z = 4-OMe)
D1-34a D1-108b (Z = 2-SMe)
D1-34a D1-108b (Z = 3-CFThree)
D1-34a D1-108b (Z = 4-OCFThree)
D1-34a D1-108b (Z = 2-SCFThree)
D1-34a C (O) Me
D1-34a C (O) CFThree
D1-34a C (O) OMe
D1-37a Me
D1-37a Et
D1-37a Pr-n
D1-37a Pr-i
D1-37a Pr-c
D1-37a Bu-n
D1-37a Bu-i
D1-37a Bu-c
D1-37a Bu-s
D1-37a Bu-t
D1-37a Pen-n
D1-37a Pen-c
D1-37a Hex-n
D1-37a Hex-c
D1-37a CH2Pr-c
D1-37a CH2Bu-c
D1-37a CH2Pen-c
D1-37a CH2Hex-c
D1-37a CH2CH = CH2
D1-37a CH2CH = C (Cl)2
D1-37a CH2C≡CH
D1-37a CH2CN
D1-37a CH2CFThree
D1-37a CH2OMe
D1-37a CH2OCFThree
D1-37a CH2SMe
D1-37a CH2S (O) Me
D1-37a CH2S (O)2Me
D1-37a CH2SCFThree
D1-37a CH2S (O) CFThree
D1-37a CH2S (O)2CFThree
D1-37a CH2CH (OMe)2
D1-37a CH2CH (SMe)2
D1-37a CH2C (O) Me
D1-37a CH2C (O) CFThree
D1-37a CH2C (O) OMe
D1-37a CH2(D1-32a)
D1-37a CH2(D1-33a)
D1-37a CH2(D1-34a)
D1-37a CH2(D1-37a)
D1-37a CH2(D1-81a)
D1-37a CH2(D1-82a)
D1-37a CH2(D1-84a)
D1-37a CH2(D1-85a)
D1-37a CH2(D1-87a)
D1-37a CH2(D1-92a)
D1-37a CH2(D1-93a)
D1-37a CH2(D1-95a)
D1-37a CH2(D1-96a)
D1-37a CH2(D1-98a)
D1-37a CH2(D1-108a)
D1-37a CH2(D1-108b, Z = 2-Cl)
D1-37a CH2(D1-108b, Z = 3-Me)
D1-37a CH2(D1-108b, Z = 4-OMe)
D1-37a CH2(D1-108b, Z = 2-SMe)
D1-37a CH2(D1-108b, Z = 3-CFThree)
D1-37a CH2(D1-108b, Z = 4-OCFThree)
D1-37a CH2(D1-108b, Z = 2-SCFThree)
D1-37a CH2CH2CN
D1-37a CH2CH2CFThree
D1-37a CH2CH2OMe
D1-37a CH2CH2SMe
D1-37a CH2CH2S (O) Me
D1-37a CH2CH2S (O)2Me
D1-37a D1-32a
D1-37a D1-33a
D1-37a D1-34a
D1-37a D1-37a
D1-37a D1-81a
D1-37a D1-82a
D1-37a D1-84a
D1-37a D1-85a
D1-37a D1-87a
D1-37a D1-92a
D1-37a D1-93a
D1-37a D1-95a
D1-37a D1-96a
D1-37a D1-98a
D1-37a D1-108a
D1-37a D1-108b (Z = 2-Cl)
D1-37a D1-108b (Z = 3-Me)
D1-37a D1-108b (Z = 4-OMe)
D1-37a D1-108b (Z = 2-SMe)
D1-37a D1-108b (Z = 3-CFThree)
D1-37a D1-108b (Z = 4-OCFThree)
D1-37a D1-108b (Z = 2-SCFThree)
D1-37a C (O) Me
D1-37a C (O) CFThree
D1-37a C (O) OMe
D1-81a Me
D1-81a Et
D1-81a Pr-n
D1-81a Pr-i
D1-81a Pr-c
D1-81a Bu-n
D1-81a Bu-i
D1-81a Bu-c
D1-81a Bu-s
D1-81a Bu-t
D1-81a Pen-n
D1-81a Pen-c
D1-81a Hex-n
D1-81a Hex-c
D1-81a CH2Pr-c
D1-81a CH2Bu-c
D1-81a CH2Pen-c
D1-81a CH2Hex-c
D1-81a CH2CH = CH2
D1-81a CH2CH = C (Cl)2
D1-81a CH2C≡CH
D1-81a CH2CN
D1-81a CH2CFThree
D1-81a CH2OMe
D1-81a CH2OCFThree
D1-81a CH2SMe
D1-81a CH2S (O) Me
D1-81a CH2S (O)2Me
D1-81a CH2SCFThree
D1-81a CH2S (O) CFThree
D1-81a CH2S (O)2CFThree
D1-81a CH2CH (OMe)2
D1-81a CH2CH (SMe)2
D1-81a CH2C (O) Me
D1-81a CH2C (O) CFThree
D1-81a CH2C (O) OMe
D1-81a CH2(D1-32a)
D1-81a CH2(D1-33a)
D1-81a CH2(D1-34a)
D1-81a CH2(D1-37a)
D1-81a CH2(D1-81a)
D1-81a CH2(D1-82a)
D1-81a CH2(D1-84a)
D1-81a CH2(D1-85a)
D1-81a CH2(D1-87a)
D1-81a CH2(D1-92a)
D1-81a CH2(D1-93a)
D1-81a CH2(D1-95a)
D1-81a CH2(D1-96a)
D1-81a CH2(D1-98a)
D1-81a CH2(D1-108a)
D1-81a CH2(D1-108b, Z = 2-Cl)
D1-81a CH2(D1-108b, Z = 3-Me)
D1-81a CH2(D1-108b, Z = 4-OMe)
D1-81a CH2(D1-108b, Z = 2-SMe)
D1-81a CH2(D1-108b, Z = 3-CFThree)
D1-81a CH2(D1-108b, Z = 4-OCFThree)
D1-81a CH2(D1-108b, Z = 2-SCFThree)
D1-81a CH2CH2CN
D1-81a CH2CH2CFThree
D1-81a CH2CH2OMe
D1-81a CH2CH2SMe
D1-81a CH2CH2S (O) Me
D1-81a CH2CH2S (O)2Me
D1-81a D1-32a
D1-81a D1-33a
D1-81a D1-34a
D1-81a D1-37a
D1-81a D1-81a
D1-81a D1-82a
D1-81a D1-84a
D1-81a D1-85a
D1-81a D1-87a
D1-81a D1-92a
D1-81a D1-93a
D1-81a D1-95a
D1-81a D1-96a
D1-81a D1-98a
D1-81a D1-108a
D1-81a D1-108b (Z = 2-Cl)
D1-81a D1-108b (Z = 3-Me)
D1-81a D1-108b (Z = 4-OMe)
D1-81a D1-108b (Z = 2-SMe)
D1-81a D1-108b (Z = 3-CFThree)
D1-81a D1-108b (Z = 4-OCFThree)
D1-81a D1-108b (Z = 2-SCFThree)
D1-81a C (O) Me
D1-81a C (O) CFThree
D1-81a C (O) OMe
D1-82a Me
D1-82a Et
D1-82a Pr-n
D1-82a Pr-i
D1-82a Pr-c
D1-82a Bu-n
D1-82a Bu-i
D1-82a Bu-c
D1-82a Bu-s
D1-82a Bu-t
D1-82a Pen-n
D1-82a Pen-c
D1-82a Hex-n
D1-82a Hex-c
D1-82a CH2Pr-c
D1-82a CH2Bu-c
D1-82a CH2Pen-c
D1-82a CH2Hex-c
D1-82a CH2CH = CH2
D1-82a CH2CH = C (Cl)2
D1-82a CH2C≡CH
D1-82a CH2CN
D1-82a CH2CFThree
D1-82a CH2OMe
D1-82a CH2OCFThree
D1-82a CH2SMe
D1-82a CH2S (O) Me
D1-82a CH2S (O)2Me
D1-82a CH2SCFThree
D1-82a CH2S (O) CFThree
D1-82a CH2S (O)2CFThree
D1-82a CH2CH (OMe)2
D1-82a CH2CH (SMe)2
D1-82a CH2C (O) Me
D1-82a CH2C (O) CFThree
D1-82a CH2C (O) OMe
D1-82a CH2(D1-32a)
D1-82a CH2(D1-33a)
D1-82a CH2(D1-34a)
D1-82a CH2(D1-37a)
D1-82a CH2(D1-81a)
D1-82a CH2(D1-82a)
D1-82a CH2(D1-84a)
D1-82a CH2(D1-85a)
D1-82a CH2(D1-87a)
D1-82a CH2(D1-92a)
D1-82a CH2(D1-93a)
D1-82a CH2(D1-95a)
D1-82a CH2(D1-96a)
D1-82a CH2(D1-98a)
D1-82a CH2(D1-108a)
D1-82a CH2(D1-108b, Z = 2-Cl)
D1-82a CH2(D1-108b, Z = 3-Me)
D1-82a CH2(D1-108b, Z = 4-OMe)
D1-82a CH2(D1-108b, Z = 2-SMe)
D1-82a CH2(D1-108b, Z = 3-CFThree)
D1-82a CH2(D1-108b, Z = 4-OCFThree)
D1-82a CH2(D1-108b, Z = 2-SCFThree)
D1-82a CH2CH2CN
D1-82a CH2CH2CFThree
D1-82a CH2CH2OMe
D1-82a CH2CH2SMe
D1-82a CH2CH2S (O) Me
D1-82a CH2CH2S (O)2Me
D1-82a D1-32a
D1-82a D1-33a
D1-82a D1-34a
D1-82a D1-37a
D1-82a D1-81a
D1-82a D1-82a
D1-82a D1-84a
D1-82a D1-85a
D1-82a D1-87a
D1-82a D1-92a
D1-82a D1-93a
D1-82a D1-95a
D1-82a D1-96a
D1-82a D1-98a
D1-82a D1-108a
D1-82a D1-108b (Z = 2-Cl)
D1-82a D1-108b (Z = 3-Me)
D1-82a D1-108b (Z = 4-OMe)
D1-82a D1-108b (Z = 2-SMe)
D1-82a D1-108b (Z = 3-CFThree)
D1-82a D1-108b (Z = 4-OCFThree)
D1-82a D1-108b (Z = 2-SCFThree)
D1-82a C (O) Me
D1-82a C (O) CFThree
D1-82a C (O) OMe
D1-84a Me
D1-84a Et
D1-84a Pr-n
D1-84a Pr-i
D1-84a Pr-c
D1-84a Bu-n
D1-84a Bu-i
D1-84a Bu-c
D1-84a Bu-s
D1-84a Bu-t
D1-84a Pen-n
D1-84a Pen-c
D1-84a Hex-n
D1-84a Hex-c
D1-84a CH2Pr-c
D1-84a CH2Bu-c
D1-84a CH2Pen-c
D1-84a CH2Hex-c
D1-84a CH2CH = CH2
D1-84a CH2CH = C (Cl)2
D1-84a CH2C≡CH
D1-84a CH2CN
D1-84a CH2CFThree
D1-84a CH2OMe
D1-84a CH2OCFThree
D1-84a CH2SMe
D1-84a CH2S (O) Me
D1-84a CH2S (O)2Me
D1-84a CH2SCFThree
D1-84a CH2S (O) CFThree
D1-84a CH2S (O)2CFThree
D1-84a CH2CH (OMe)2
D1-84a CH2CH (SMe)2
D1-84a CH2C (O) Me
D1-84a CH2C (O) CFThree
D1-84a CH2C (O) OMe
D1-84a CH2(D1-32a)
D1-84a CH2(D1-33a)
D1-84a CH2(D1-34a)
D1-84a CH2(D1-37a)
D1-84a CH2(D1-81a)
D1-84a CH2(D1-82a)
D1-84a CH2(D1-84a)
D1-84a CH2(D1-85a)
D1-84a CH2(D1-87a)
D1-84a CH2(D1-92a)
D1-84a CH2(D1-93a)
D1-84a CH2(D1-95a)
D1-84a CH2(D1-96a)
D1-84a CH2(D1-98a)
D1-84a CH2(D1-108a)
D1-84a CH2(D1-108b, Z = 2-Cl)
D1-84a CH2(D1-108b, Z = 3-Me)
D1-84a CH2(D1-108b, Z = 4-OMe)
D1-84a CH2(D1-108b, Z = 2-SMe)
D1-84a CH2(D1-108b, Z = 3-CFThree)
D1-84a CH2(D1-108b, Z = 4-OCFThree)
D1-84a CH2(D1-108b, Z = 2-SCFThree)
D1-84a CH2CH2CN
D1-84a CH2CH2CFThree
D1-84a CH2CH2OMe
D1-84a CH2CH2SMe
D1-84a CH2CH2S (O) Me
D1-84a CH2CH2S (O)2Me
D1-84a D1-32a
D1-84a D1-33a
D1-84a D1-34a
D1-84a D1-37a
D1-84a D1-81a
D1-84a D1-82a
D1-84a D1-84a
D1-84a D1-85a
D1-84a D1-87a
D1-84a D1-92a
D1-84a D1-93a
D1-84a D1-95a
D1-84a D1-96a
D1-84a D1-98a
D1-84a D1-108a
D1-84a D1-108b (Z = 2-Cl)
D1-84a D1-108b (Z = 3-Me)
D1-84a D1-108b (Z = 4-OMe)
D1-84a D1-108b (Z = 2-SMe)
D1-84a D1-108b (Z = 3-CFThree)
D1-84a D1-108b (Z = 4-OCFThree)
D1-84a D1-108b (Z = 2-SCFThree)
D1-84a C (O) Me
D1-84a C (O) CFThree
D1-84a C (O) OMe
D1-85a Me
D1-85a Et
D1-85a Pr-n
D1-85a Pr-i
D1-85a Pr-c
D1-85a Bu-n
D1-85a Bu-i
D1-85a Bu-c
D1-85a Bu-s
D1-85a Bu-t
D1-85a Pen-n
D1-85a Pen-c
D1-85a Hex-n
D1-85a Hex-c
D1-85a CH2Pr-c
D1-85a CH2Bu-c
D1-85a CH2Pen-c
D1-85a CH2Hex-c
D1-85a CH2CH = CH2
D1-85a CH2CH = C (Cl)2
D1-85a CH2C≡CH
D1-85a CH2CN
D1-85a CH2CFThree
D1-85a CH2OMe
D1-85a CH2OCFThree
D1-85a CH2SMe
D1-85a CH2S (O) Me
D1-85a CH2S (O)2Me
D1-85a CH2SCFThree
D1-85a CH2S (O) CFThree
D1-85a CH2S (O)2CFThree
D1-85a CH2CH (OMe)2
D1-85a CH2CH (SMe)2
D1-85a CH2C (O) Me
D1-85a CH2C (O) CFThree
D1-85a CH2C (O) OMe
D1-85a CH2(D1-32a)
D1-85a CH2(D1-33a)
D1-85a CH2(D1-34a)
D1-85a CH2(D1-37a)
D1-85a CH2(D1-81a)
D1-85a CH2(D1-82a)
D1-85a CH2(D1-84a)
D1-85a CH2(D1-85a)
D1-85a CH2(D1-87a)
D1-85a CH2(D1-92a)
D1-85a CH2(D1-93a)
D1-85a CH2(D1-95a)
D1-85a CH2(D1-96a)
D1-85a CH2(D1-98a)
D1-85a CH2(D1-108a)
D1-85a CH2(D1-108b, Z = 2-Cl)
D1-85a CH2(D1-108b, Z = 3-Me)
D1-85a CH2(D1-108b, Z = 4-OMe)
D1-85a CH2(D1-108b, Z = 2-SMe)
D1-85a CH2(D1-108b, Z = 3-CFThree)
D1-85a CH2(D1-108b, Z = 4-OCFThree)
D1-85a CH2(D1-108b, Z = 2-SCFThree)
D1-85a CH2CH2CN
D1-85a CH2CH2CFThree
D1-85a CH2CH2OMe
D1-85a CH2CH2SMe
D1-85a CH2CH2S (O) Me
D1-85a CH2CH2S (O)2Me
D1-85a D1-32a
D1-85a D1-33a
D1-85a D1-34a
D1-85a D1-37a
D1-85a D1-81a
D1-85a D1-82a
D1-85a D1-84a
D1-85a D1-85a
D1-85a D1-87a
D1-85a D1-92a
D1-85a D1-93a
D1-85a D1-95a
D1-85a D1-96a
D1-85a D1-98a
D1-85a D1-108a
D1-85a D1-108b (Z = 2-Cl)
D1-85a D1-108b (Z = 3-Me)
D1-85a D1-108b (Z = 4-OMe)
D1-85a D1-108b (Z = 2-SMe)
D1-85a D1-108b (Z = 3-CFThree)
D1-85a D1-108b (Z = 4-OCFThree)
D1-85a D1-108b (Z = 2-SCFThree)
D1-85a C (O) Me
D1-85a C (O) CFThree
D1-85a C (O) OMe
D1-87a Me
D1-87a Et
D1-87a Pr-n
D1-87a Pr-i
D1-87a Pr-c
D1-87a Bu-n
D1-87a Bu-i
D1-87a Bu-c
D1-87a Bu-s
D1-87a Bu-t
D1-87a Pen-n
D1-87a Pen-c
D1-87a Hex-n
D1-87a Hex-c
D1-87a CH2Pr-c
D1-87a CH2Bu-c
D1-87a CH2Pen-c
D1-87a CH2Hex-c
D1-87a CH2CH = CH2
D1-87a CH2CH = C (Cl)2
D1-87a CH2C≡CH
D1-87a CH2CN
D1-87a CH2CFThree
D1-87a CH2OMe
D1-87a CH2OCFThree
D1-87a CH2SMe
D1-87a CH2S (O) Me
D1-87a CH2S (O)2Me
D1-87a CH2SCFThree
D1-87a CH2S (O) CFThree
D1-87a CH2S (O)2CFThree
D1-87a CH2CH (OMe)2
D1-87a CH2CH (SMe)2
D1-87a CH2C (O) Me
D1-87a CH2C (O) CFThree
D1-87a CH2C (O) OMe
D1-87a CH2(D1-32a)
D1-87a CH2(D1-33a)
D1-87a CH2(D1-34a)
D1-87a CH2(D1-37a)
D1-87a CH2(D1-81a)
D1-87a CH2(D1-82a)
D1-87a CH2(D1-84a)
D1-87a CH2(D1-85a)
D1-87a CH2(D1-87a)
D1-87a CH2(D1-92a)
D1-87a CH2(D1-93a)
D1-87a CH2(D1-95a)
D1-87a CH2(D1-96a)
D1-87a CH2(D1-98a)
D1-87a CH2(D1-108a)
D1-87a CH2(D1-108b, Z = 2-Cl)
D1-87a CH2(D1-108b, Z = 3-Me)
D1-87a CH2(D1-108b, Z = 4-OMe)
D1-87a CH2(D1-108b, Z = 2-SMe)
D1-87a CH2(D1-108b, Z = 3-CFThree)
D1-87a CH2(D1-108b, Z = 4-OCFThree)
D1-87a CH2(D1-108b, Z = 2-SCFThree)
D1-87a CH2CH2CN
D1-87a CH2CH2CFThree
D1-87a CH2CH2OMe
D1-87a CH2CH2SMe
D1-87a CH2CH2S (O) Me
D1-87a CH2CH2S (O)2Me
D1-87a D1-32a
D1-87a D1-33a
D1-87a D1-34a
D1-87a D1-37a
D1-87a D1-81a
D1-87a D1-82a
D1-87a D1-84a
D1-87a D1-85a
D1-87a D1-87a
D1-87a D1-92a
D1-87a D1-93a
D1-87a D1-95a
D1-87a D1-96a
D1-87a D1-98a
D1-87a D1-108a
D1-87a D1-108b (Z = 2-Cl)
D1-87a D1-108b (Z = 3-Me)
D1-87a D1-108b (Z = 4-OMe)
D1-87a D1-108b (Z = 2-SMe)
D1-87a D1-108b (Z = 3-CFThree)
D1-87a D1-108b (Z = 4-OCFThree)
D1-87a D1-108b (Z = 2-SCFThree)
D1-87a C (O) Me
D1-87a C (O) CFThree
D1-87a C (O) OMe
D1-92a Me
D1-92a Et
D1-92a Pr-n
D1-92a Pr-i
D1-92a Pr-c
D1-92a Bu-n
D1-92a Bu-i
D1-92a Bu-c
D1-92a Bu-s
D1-92a Bu-t
D1-92a Pen-n
D1-92a Pen-c
D1-92a Hex-n
D1-92a Hex-c
D1-92a CH2Pr-c
D1-92a CH2Bu-c
D1-92a CH2Pen-c
D1-92a CH2Hex-c
D1-92a CH2CH = CH2
D1-92a CH2CH = C (Cl)2
D1-92a CH2C≡CH
D1-92a CH2CN
D1-92a CH2CFThree
D1-92a CH2OMe
D1-92a CH2OCFThree
D1-92a CH2SMe
D1-92a CH2S (O) Me
D1-92a CH2S (O)2Me
D1-92a CH2SCFThree
D1-92a CH2S (O) CFThree
D1-92a CH2S (O)2CFThree
D1-92a CH2CH (OMe)2
D1-92a CH2CH (SMe)2
D1-92a CH2C (O) Me
D1-92a CH2C (O) CFThree
D1-92a CH2C (O) OMe
D1-92a CH2(D1-32a)
D1-92a CH2(D1-33a)
D1-92a CH2(D1-34a)
D1-92a CH2(D1-37a)
D1-92a CH2(D1-81a)
D1-92a CH2(D1-82a)
D1-92a CH2(D1-84a)
D1-92a CH2(D1-85a)
D1-92a CH2(D1-87a)
D1-92a CH2(D1-92a)
D1-92a CH2(D1-93a)
D1-92a CH2(D1-95a)
D1-92a CH2(D1-96a)
D1-92a CH2(D1-98a)
D1-92a CH2(D1-108a)
D1-92a CH2(D1-108b, Z = 2-Cl)
D1-92a CH2(D1-108b, Z = 3-Me)
D1-92a CH2(D1-108b, Z = 4-OMe)
D1-92a CH2(D1-108b, Z = 2-SMe)
D1-92a CH2(D1-108b, Z = 3-CFThree)
D1-92a CH2(D1-108b, Z = 4-OCFThree)
D1-92a CH2(D1-108b, Z = 2-SCFThree)
D1-92a CH2CH2CN
D1-92a CH2CH2CFThree
D1-92a CH2CH2OMe
D1-92a CH2CH2SMe
D1-92a CH2CH2S (O) Me
D1-92a CH2CH2S (O)2Me
D1-92a D1-32a
D1-92a D1-33a
D1-92a D1-34a
D1-92a D1-37a
D1-92a D1-81a
D1-92a D1-82a
D1-92a D1-84a
D1-92a D1-85a
D1-92a D1-87a
D1-92a D1-92a
D1-92a D1-93a
D1-92a D1-95a
D1-92a D1-96a
D1-92a D1-98a
D1-92a D1-108a
D1-92a D1-108b (Z = 2-Cl)
D1-92a D1-108b (Z = 3-Me)
D1-92a D1-108b (Z = 4-OMe)
D1-92a D1-108b (Z = 2-SMe)
D1-92a D1-108b (Z = 3-CFThree)
D1-92a D1-108b (Z = 4-OCFThree)
D1-92a D1-108b (Z = 2-SCFThree)
D1-92a C (O) Me
D1-92a C (O) CFThree
D1-92a C (O) OMe
D1-93a Me
D1-93a Et
D1-93a Pr-n
D1-93a Pr-i
D1-93a Pr-c
D1-93a Bu-n
D1-93a Bu-i
D1-93a Bu-c
D1-93a Bu-s
D1-93a Bu-t
D1-93a Pen-n
D1-93a Pen-c
D1-93a Hex-n
D1-93a Hex-c
D1-93a CH2Pr-c
D1-93a CH2Bu-c
D1-93a CH2Pen-c
D1-93a CH2Hex-c
D1-93a CH2CH = CH2
D1-93a CH2CH = C (Cl)2
D1-93a CH2C≡CH
D1-93a CH2CN
D1-93a CH2CFThree
D1-93a CH2OMe
D1-93a CH2OCFThree
D1-93a CH2SMe
D1-93a CH2S (O) Me
D1-93a CH2S (O)2Me
D1-93a CH2SCFThree
D1-93a CH2S (O) CFThree
D1-93a CH2S (O)2CFThree
D1-93a CH2CH (OMe)2
D1-93a CH2CH (SMe)2
D1-93a CH2C (O) Me
D1-93a CH2C (O) CFThree
D1-93a CH2C (O) OMe
D1-93a CH2(D1-32a)
D1-93a CH2(D1-33a)
D1-93a CH2(D1-34a)
D1-93a CH2(D1-37a)
D1-93a CH2(D1-81a)
D1-93a CH2(D1-82a)
D1-93a CH2(D1-84a)
D1-93a CH2(D1-85a)
D1-93a CH2(D1-87a)
D1-93a CH2(D1-92a)
D1-93a CH2(D1-93a)
D1-93a CH2(D1-95a)
D1-93a CH2(D1-96a)
D1-93a CH2(D1-98a)
D1-93a CH2(D1-108a)
D1-93a CH2(D1-108b, Z = 2-Cl)
D1-93a CH2(D1-108b, Z = 3-Me)
D1-93a CH2(D1-108b, Z = 4-OMe)
D1-93a CH2(D1-108b, Z = 2-SMe)
D1-93a CH2(D1-108b, Z = 3-CFThree)
D1-93a CH2(D1-108b, Z = 4-OCFThree)
D1-93a CH2(D1-108b, Z = 2-SCFThree)
D1-93a CH2CH2CN
D1-93a CH2CH2CFThree
D1-93a CH2CH2OMe
D1-93a CH2CH2SMe
D1-93a CH2CH2S (O) Me
D1-93a CH2CH2S (O)2Me
D1-93a D1-32a
D1-93a D1-33a
D1-93a D1-34a
D1-93a D1-37a
D1-93a D1-81a
D1-93a D1-82a
D1-93a D1-84a
D1-93a D1-85a
D1-93a D1-87a
D1-93a D1-92a
D1-93a D1-93a
D1-93a D1-95a
D1-93a D1-96a
D1-93a D1-98a
D1-93a D1-108a
D1-93a D1-108b (Z = 2-Cl)
D1-93a D1-108b (Z = 3-Me)
D1-93a D1-108b (Z = 4-OMe)
D1-93a D1-108b (Z = 2-SMe)
D1-93a D1-108b (Z = 3-CFThree)
D1-93a D1-108b (Z = 4-OCFThree)
D1-93a D1-108b (Z = 2-SCFThree)
D1-93a C (O) Me
D1-93a C (O) CFThree
D1-93a C (O) OMe
D1-95a Me
D1-95a Et
D1-95a Pr-n
D1-95a Pr-i
D1-95a Pr-c
D1-95a Bu-n
D1-95a Bu-i
D1-95a Bu-c
D1-95a Bu-s
D1-95a Bu-t
D1-95a Pen-n
D1-95a Pen-c
D1-95a Hex-n
D1-95a Hex-c
D1-95a CH2Pr-c
D1-95a CH2Bu-c
D1-95a CH2Pen-c
D1-95a CH2Hex-c
D1-95a CH2CH = CH2
D1-95a CH2CH = C (Cl)2
D1-95a CH2C≡CH
D1-95a CH2CN
D1-95a CH2CFThree
D1-95a CH2OMe
D1-95a CH2OCFThree
D1-95a CH2SMe
D1-95a CH2S (O) Me
D1-95a CH2S (O)2Me
D1-95a CH2SCFThree
D1-95a CH2S (O) CFThree
D1-95a CH2S (O)2CFThree
D1-95a CH2CH (OMe)2
D1-95a CH2CH (SMe)2
D1-95a CH2C (O) Me
D1-95a CH2C (O) CFThree
D1-95a CH2C (O) OMe
D1-95a CH2(D1-32a)
D1-95a CH2(D1-33a)
D1-95a CH2(D1-34a)
D1-95a CH2(D1-37a)
D1-95a CH2(D1-81a)
D1-95a CH2(D1-82a)
D1-95a CH2(D1-84a)
D1-95a CH2(D1-85a)
D1-95a CH2(D1-87a)
D1-95a CH2(D1-92a)
D1-95a CH2(D1-93a)
D1-95a CH2(D1-95a)
D1-95a CH2(D1-96a)
D1-95a CH2(D1-98a)
D1-95a CH2(D1-108a)
D1-95a CH2(D1-108b, Z = 2-Cl)
D1-95a CH2(D1-108b, Z = 3-Me)
D1-95a CH2(D1-108b, Z = 4-OMe)
D1-95a CH2(D1-108b, Z = 2-SMe)
D1-95a CH2(D1-108b, Z = 3-CFThree)
D1-95a CH2(D1-108b, Z = 4-OCFThree)
D1-95a CH2(D1-108b, Z = 2-SCFThree)
D1-95a CH2CH2CN
D1-95a CH2CH2CFThree
D1-95a CH2CH2OMe
D1-95a CH2CH2SMe
D1-95a CH2CH2S (O) Me
D1-95a CH2CH2S (O)2Me
D1-95a D1-32a
D1-95a D1-33a
D1-95a D1-34a
D1-95a D1-37a
D1-95a D1-81a
D1-95a D1-82a
D1-95a D1-84a
D1-95a D1-85a
D1-95a D1-87a
D1-95a D1-92a
D1-95a D1-93a
D1-95a D1-95a
D1-95a D1-96a
D1-95a D1-98a
D1-95a D1-108a
D1-95a D1-108b (Z = 2-Cl)
D1-95a D1-108b (Z = 3-Me)
D1-95a D1-108b (Z = 4-OMe)
D1-95a D1-108b (Z = 2-SMe)
D1-95a D1-108b (Z = 3-CFThree)
D1-95a D1-108b (Z = 4-OCFThree)
D1-95a D1-108b (Z = 2-SCFThree)
D1-95a C (O) Me
D1-95a C (O) CFThree
D1-95a C (O) OMe
D1-96a Me
D1-96a Et
D1-96a Pr-n
D1-96a Pr-i
D1-96a Pr-c
D1-96a Bu-n
D1-96a Bu-i
D1-96a Bu-c
D1-96a Bu-s
D1-96a Bu-t
D1-96a Pen-n
D1-96a Pen-c
D1-96a Hex-n
D1-96a Hex-c
D1-96a CH2Pr-c
D1-96a CH2Bu-c
D1-96a CH2Pen-c
D1-96a CH2Hex-c
D1-96a CH2CH = CH2
D1-96a CH2CH = C (Cl)2
D1-96a CH2C≡CH
D1-96a CH2CN
D1-96a CH2CFThree
D1-96a CH2OMe
D1-96a CH2OCFThree
D1-96a CH2SMe
D1-96a CH2S (O) Me
D1-96a CH2S (O)2Me
D1-96a CH2SCFThree
D1-96a CH2S (O) CFThree
D1-96a CH2S (O)2CFThree
D1-96a CH2CH (OMe)2
D1-96a CH2CH (SMe)2
D1-96a CH2C (O) Me
D1-96a CH2C (O) CFThree
D1-96a CH2C (O) OMe
D1-96a CH2(D1-32a)
D1-96a CH2(D1-33a)
D1-96a CH2(D1-34a)
D1-96a CH2(D1-37a)
D1-96a CH2(D1-81a)
D1-96a CH2(D1-82a)
D1-96a CH2(D1-84a)
D1-96a CH2(D1-85a)
D1-96a CH2(D1-87a)
D1-96a CH2(D1-92a)
D1-96a CH2(D1-93a)
D1-96a CH2(D1-95a)
D1-96a CH2(D1-96a)
D1-96a CH2(D1-98a)
D1-96a CH2(D1-108a)
D1-96a CH2(D1-108b, Z = 2-Cl)
D1-96a CH2(D1-108b, Z = 3-Me)
D1-96a CH2(D1-108b, Z = 4-OMe)
D1-96a CH2(D1-108b, Z = 2-SMe)
D1-96a CH2(D1-108b, Z = 3-CFThree)
D1-96a CH2(D1-108b, Z = 4-OCFThree)
D1-96a CH2(D1-108b, Z = 2-SCFThree)
D1-96a CH2CH2CN
D1-96a CH2CH2CFThree
D1-96a CH2CH2OMe
D1-96a CH2CH2SMe
D1-96a CH2CH2S (O) Me
D1-96a CH2CH2S (O)2Me
D1-96a D1-32a
D1-96a D1-33a
D1-96a D1-34a
D1-96a D1-37a
D1-96a D1-81a
D1-96a D1-82a
D1-96a D1-84a
D1-96a D1-85a
D1-96a D1-87a
D1-96a D1-92a
D1-96a D1-93a
D1-96a D1-95a
D1-96a D1-96a
D1-96a D1-98a
D1-96a D1-108a
D1-96a D1-108b (Z = 2-Cl)
D1-96a D1-108b (Z = 3-Me)
D1-96a D1-108b (Z = 4-OMe)
D1-96a D1-108b (Z = 2-SMe)
D1-96a D1-108b (Z = 3-CFThree)
D1-96a D1-108b (Z = 4-OCFThree)
D1-96a D1-108b (Z = 2-SCFThree)
D1-96a C (O) Me
D1-96a C (O) CFThree
D1-96a C (O) OMe
D1-98a Me
D1-98a Et
D1-98a Pr-n
D1-98a Pr-i
D1-98a Pr-c
D1-98a Bu-n
D1-98a Bu-i
D1-98a Bu-c
D1-98a Bu-s
D1-98a Bu-t
D1-98a Pen-n
D1-98a Pen-c
D1-98a Hex-n
D1-98a Hex-c
D1-98a CH2Pr-c
D1-98a CH2Bu-c
D1-98a CH2Pen-c
D1-98a CH2Hex-c
D1-98a CH2CH = CH2
D1-98a CH2CH = C (Cl)2
D1-98a CH2C≡CH
D1-98a CH2CN
D1-98a CH2CFThree
D1-98a CH2OMe
D1-98a CH2OCFThree
D1-98a CH2SMe
D1-98a CH2S (O) Me
D1-98a CH2S (O)2Me
D1-98a CH2SCFThree
D1-98a CH2S (O) CFThree
D1-98a CH2S (O)2CFThree
D1-98a CH2CH (OMe)2
D1-98a CH2CH (SMe)2
D1-98a CH2C (O) Me
D1-98a CH2C (O) CFThree
D1-98a CH2C (O) OMe
D1-98a CH2(D1-32a)
D1-98a CH2(D1-33a)
D1-98a CH2(D1-34a)
D1-98a CH2(D1-37a)
D1-98a CH2(D1-81a)
D1-98a CH2(D1-82a)
D1-98a CH2(D1-84a)
D1-98a CH2(D1-85a)
D1-98a CH2(D1-87a)
D1-98a CH2(D1-92a)
D1-98a CH2(D1-93a)
D1-98a CH2(D1-95a)
D1-98a CH2(D1-96a)
D1-98a CH2(D1-98a)
D1-98a CH2(D1-108a)
D1-98a CH2(D1-108b, Z = 2-Cl)
D1-98a CH2(D1-108b, Z = 3-Me)
D1-98a CH2(D1-108b, Z = 4-OMe)
D1-98a CH2(D1-108b, Z = 2-SMe)
D1-98a CH2(D1-108b, Z = 3-CFThree)
D1-98a CH2(D1-108b, Z = 4-OCFThree)
D1-98a CH2(D1-108b, Z = 2-SCFThree)
D1-98a CH2CH2CN
D1-98a CH2CH2CFThree
D1-98a CH2CH2OMe
D1-98a CH2CH2SMe
D1-98a CH2CH2S (O) Me
D1-98a CH2CH2S (O)2Me
D1-98a D1-32a
D1-98a D1-33a
D1-98a D1-34a
D1-98a D1-37a
D1-98a D1-81a
D1-98a D1-82a
D1-98a D1-84a
D1-98a D1-85a
D1-98a D1-87a
D1-98a D1-92a
D1-98a D1-93a
D1-98a D1-95a
D1-98a D1-96a
D1-98a D1-98a
D1-98a D1-108a
D1-98a D1-108b (Z = 2-Cl)
D1-98a D1-108b (Z = 3-Me)
D1-98a D1-108b (Z = 4-OMe)
D1-98a D1-108b (Z = 2-SMe)
D1-98a D1-108b (Z = 3-CFThree)
D1-98a D1-108b (Z = 4-OCFThree)
D1-98a D1-108b (Z = 2-SCFThree)
D1-98a C (O) Me
D1-98a C (O) CFThree
D1-98a C (O) OMe
D1-108a Me
D1-108a Et
D1-108a Pr-n
D1-108a Pr-i
D1-108a Pr-c
D1-108a Bu-n
D1-108a Bu-i
D1-108a Bu-c
D1-108a Bu-s
D1-108a Bu-t
D1-108a Pen-n
D1-108a Pen-c
D1-108a Hex-n
D1-108a Hex-c
D1-108a CH2Pr-c
D1-108a CH2Bu-c
D1-108a CH2Pen-c
D1-108a CH2Hex-c
D1-108a CH2CH = CH2
D1-108a CH2CH = C (Cl)2
D1-108a CH2C≡CH
D1-108a CH2CN
D1-108a CH2CFThree
D1-108a CH2OMe
D1-108a CH2OCFThree
D1-108a CH2SMe
D1-108a CH2S (O) Me
D1-108a CH2S (O)2Me
D1-108a CH2SCFThree
D1-108a CH2S (O) CFThree
D1-108a CH2S (O)2CFThree
D1-108a CH2CH (OMe)2
D1-108a CH2CH (SMe)2
D1-108a CH2C (O) Me
D1-108a CH2C (O) CFThree
D1-108a CH2C (O) OMe
D1-108a CH2(D1-32a)
D1-108a CH2(D1-33a)
D1-108a CH2(D1-34a)
D1-108a CH2(D1-37a)
D1-108a CH2(D1-81a)
D1-108a CH2(D1-82a)
D1-108a CH2(D1-84a)
D1-108a CH2(D1-85a)
D1-108a CH2(D1-87a)
D1-108a CH2(D1-92a)
D1-108a CH2(D1-93a)
D1-108a CH2(D1-95a)
D1-108a CH2(D1-96a)
D1-108a CH2(D1-98a)
D1-108a CH2(D1-108a)
D1-108a CH2(D1-108b, Z = 2-Cl)
D1-108a CH2(D1-108b, Z = 3-Me)
D1-108a CH2(D1-108b, Z = 4-OMe)
D1-108a CH2(D1-108b, Z = 2-SMe)
D1-108a CH2(D1-108b, Z = 3-CFThree)
D1-108a CH2(D1-108b, Z = 4-OCFThree)
D1-108a CH2(D1-108b, Z = 2-SCFThree)
D1-108a CH2CH2CN
D1-108a CH2CH2CFThree
D1-108a CH2CH2OMe
D1-108a CH2CH2SMe
D1-108a CH2CH2S (O) Me
D1-108a CH2CH2S (O)2Me
D1-108a D1-32a
D1-108a D1-33a
D1-108a D1-34a
D1-108a D1-37a
D1-108a D1-81a
D1-108a D1-82a
D1-108a D1-84a
D1-108a D1-85a
D1-108a D1-87a
D1-108a D1-92a
D1-108a D1-93a
D1-108a D1-95a
D1-108a D1-96a
D1-108a D1-98a
D1-108a D1-108a
D1-108a D1-108b (Z = 2-Cl)
D1-108a D1-108b (Z = 3-Me)
D1-108a D1-108b (Z = 4-OMe)
D1-108a D1-108b (Z = 2-SMe)
D1-108a D1-108b (Z = 3-CFThree)
D1-108a D1-108b (Z = 4-OCFThree)
D1-108a D1-108b (Z = 2-SCFThree)
D1-108a C (O) Me
D1-108a C (O) CFThree
D1-108a C (O) OMe
CH2SCH2CH2CFThree                         Me
CH2SCH2CH2CFThree                         Et
CH2SCH2CH2CFThree                         Pr-n
CH2SCH2CH2CFThree                         Pr-i
CH2SCH2CH2CFThree                         Pr-c
CH2SCH2CH2CFThree                         Bu-n
CH2SCH2CH2CFThree                         Bu-i
CH2SCH2CH2CFThree                         Bu-c
CH2SCH2CH2CFThree                         Bu-s
CH2SCH2CH2CFThree                         Bu-t
CH2SCH2CH2CFThree                         Pen-n
CH2SCH2CH2CFThree                         Pen-c
CH2SCH2CH2CFThree                         Hex-n
CH2SCH2CH2CFThree                         Hex-c
CH2SCH2CH2CFThree                         CH2Pr-c
CH2SCH2CH2CFThree                         CH2Bu-c
CH2SCH2CH2CFThree                         CH2Pen-c
CH2SCH2CH2CFThree                         CH2Hex-c
CH2SCH2CH2CFThree                         CH2CH = CH2
CH2SCH2CH2CFThree                         CH2CH = C (Cl)2
CH2SCH2CH2CFThree                         CH2C≡CH
CH2SCH2CH2CFThree                         CH2CN
CH2SCH2CH2CFThree                         CH2CFThree
CH2SCH2CH2CFThree                         CH2OMe
CH2SCH2CH2CFThree                         CH2OCFThree
CH2SCH2CH2CFThree                         CH2SMe
CH2SCH2CH2CFThree                         CH2S (O) Me
CH2SCH2CH2CFThree                         CH2S (O)2Me
CH2SCH2CH2CFThree                         CH2SCFThree
CH2SCH2CH2CFThree                         CH2S (O) CFThree
CH2SCH2CH2CFThree                         CH2S (O)2CFThree
CH2SCH2CH2CFThree                         CH2CH (OMe)2
CH2SCH2CH2CFThree                         CH2CH (SMe)2
CH2SCH2CH2CFThree                         CH2C (O) Me
CH2SCH2CH2CFThree                         CH2C (O) CFThree
CH2SCH2CH2CFThree                         CH2C (O) OMe
CH2SCH2CH2CFThree                         CH2(D1-32a)
CH2SCH2CH2CFThree                         CH2(D1-33a)
CH2SCH2CH2CFThree                         CH2(D1-34a)
CH2SCH2CH2CFThree                         CH2(D1-37a)
CH2SCH2CH2CFThree                         CH2(D1-81a)
CH2SCH2CH2CFThree                         CH2(D1-82a)
CH2SCH2CH2CFThree                         CH2(D1-84a)
CH2SCH2CH2CFThree                         CH2(D1-85a)
CH2SCH2CH2CFThree                         CH2(D1-87a)
CH2SCH2CH2CFThree                         CH2(D1-92a)
CH2SCH2CH2CFThree                         CH2(D1-93a)
CH2SCH2CH2CFThree                         CH2(D1-95a)
CH2SCH2CH2CFThree                         CH2(D1-96a)
CH2SCH2CH2CFThree                         CH2(D1-98a)
CH2SCH2CH2CFThree                         CH2(D1-108a)
CH2SCH2CH2CFThree                         CH2(D1-108b, Z = 2-Cl)
CH2SCH2CH2CFThree                         CH2(D1-108b, Z = 3-Me)
CH2SCH2CH2CFThree                         CH2(D1-108b, Z = 4-OMe)
CH2SCH2CH2CFThree                         CH2(D1-108b, Z = 2-SMe)
CH2SCH2CH2CFThree                         CH2(D1-108b, Z = 3-CFThree)
CH2SCH2CH2CFThree                         CH2(D1-108b, Z = 4-OCFThree)
CH2SCH2CH2CFThree                         CH2(D1-108b, Z = 2-SCFThree)
CH2SCH2CH2CFThree                         CH2CH2CN
CH2SCH2CH2CFThree                         CH2CH2CFThree
CH2SCH2CH2CFThree                         CH2CH2OMe
CH2SCH2CH2CFThree                         CH2CH2SMe
CH2SCH2CH2CFThree                         CH2CH2S (O) Me
CH2SCH2CH2CFThree                         CH2CH2S (O)2Me
CH2SCH2CH2CFThree                         D1-32a
CH2SCH2CH2CFThree                         D1-33a
CH2SCH2CH2CFThree                         D1-34a
CH2SCH2CH2CFThree                         D1-37a
CH2SCH2CH2CFThree                         D1-81a
CH2SCH2CH2CFThree                         D1-82a
CH2SCH2CH2CFThree                         D1-84a
CH2SCH2CH2CFThree                         D1-85a
CH2SCH2CH2CFThree                         D1-87a
CH2SCH2CH2CFThree                         D1-92a
CH2SCH2CH2CFThree                         D1-93a
CH2SCH2CH2CFThree                         D1-95a
CH2SCH2CH2CFThree                         D1-96a
CH2SCH2CH2CFThree                         D1-98a
CH2SCH2CH2CFThree                         D1-108a
CH2SCH2CH2CFThree                         D1-108b (Z = 2-Cl)
CH2SCH2CH2CFThree                         D1-108b (Z = 3-Me)
CH2SCH2CH2CFThree                         D1-108b (Z = 4-OMe)
CH2SCH2CH2CFThree                         D1-108b (Z = 2-SMe)
CH2SCH2CH2CFThree                         D1-108b (Z = 3-CFThree)
CH2SCH2CH2CFThree                         D1-108b (Z = 4-OCFThree)
CH2SCH2CH2CFThree                         D1-108b (Z = 2-SCFThree)
CH2SCH2CH2CFThree                         C (O) Me
CH2SCH2CH2CFThree                         C (O) CFThree
CH2SCH2CH2CFThree                         C (O) OMe
CH2S (O) CH2CH2CFThree                      Me
CH2S (O) CH2CH2CFThree                      Et
CH2S (O) CH2CH2CFThree                      Pr-n
CH2S (O) CH2CH2CFThree                      Pr-i
CH2S (O) CH2CH2CFThree                      Pr-c
CH2S (O) CH2CH2CFThree                      Bu-n
CH2S (O) CH2CH2CFThree                      Bu-i
CH2S (O) CH2CH2CFThree                      Bu-c
CH2S (O) CH2CH2CFThree                      Bu-s
CH2S (O) CH2CH2CFThree                      Bu-t
CH2S (O) CH2CH2CFThree                      Pen-n
CH2S (O) CH2CH2CFThree                      Pen-c
CH2S (O) CH2CH2CFThree                      Hex-n
CH2S (O) CH2CH2CFThree                      Hex-c
CH2S (O) CH2CH2CFThree                      CH2Pr-c
CH2S (O) CH2CH2CFThree                      CH2Bu-c
CH2S (O) CH2CH2CFThree                      CH2Pen-c
CH2S (O) CH2CH2CFThree                      CH2Hex-c
CH2S (O) CH2CH2CFThree                      CH2CH = CH2
CH2S (O) CH2CH2CFThree                      CH2CH = C (Cl)2
CH2S (O) CH2CH2CFThree                      CH2C≡CH
CH2S (O) CH2CH2CFThree                      CH2CN
CH2S (O) CH2CH2CFThree                      CH2CFThree
CH2S (O) CH2CH2CFThree                      CH2OMe
CH2S (O) CH2CH2CFThree                      CH2OCFThree
CH2S (O) CH2CH2CFThree                      CH2SMe
CH2S (O) CH2CH2CFThree                      CH2S (O) Me
CH2S (O) CH2CH2CFThree                      CH2S (O)2Me
CH2S (O) CH2CH2CFThree                      CH2SCFThree
CH2S (O) CH2CH2CFThree                      CH2S (O) CFThree
CH2S (O) CH2CH2CFThree                      CH2S (O)2CFThree
CH2S (O) CH2CH2CFThree                      CH2CH (OMe)2
CH2S (O) CH2CH2CFThree                      CH2CH (SMe)2
CH2S (O) CH2CH2CFThree                      CH2C (O) Me
CH2S (O) CH2CH2CFThree                      CH2C (O) CFThree
CH2S (O) CH2CH2CFThree                      CH2C (O) OMe
CH2S (O) CH2CH2CFThree                      CH2(D1-32a)
CH2S (O) CH2CH2CFThree                      CH2(D1-33a)
CH2S (O) CH2CH2CFThree                      CH2(D1-34a)
CH2S (O) CH2CH2CFThree                      CH2(D1-37a)
CH2S (O) CH2CH2CFThree                      CH2(D1-81a)
CH2S (O) CH2CH2CFThree                      CH2(D1-82a)
CH2S (O) CH2CH2CFThree                      CH2(D1-84a)
CH2S (O) CH2CH2CFThree                      CH2(D1-85a)
CH2S (O) CH2CH2CFThree                      CH2(D1-87a)
CH2S (O) CH2CH2CFThree                      CH2(D1-92a)
CH2S (O) CH2CH2CFThree                      CH2(D1-93a)
CH2S (O) CH2CH2CFThree                      CH2(D1-95a)
CH2S (O) CH2CH2CFThree                      CH2(D1-96a)
CH2S (O) CH2CH2CFThree                      CH2(D1-98a)
CH2S (O) CH2CH2CFThree                      CH2(D1-108a)
CH2S (O) CH2CH2CFThree                      CH2(D1-108b, Z = 2-Cl)
CH2S (O) CH2CH2CFThree                      CH2(D1-108b, Z = 3-Me)
CH2S (O) CH2CH2CFThree                      CH2(D1-108b, Z = 4-OMe)
CH2S (O) CH2CH2CFThree                      CH2(D1-108b, Z = 2-SMe)
CH2S (O) CH2CH2CFThree                      CH2(D1-108b, Z = 3-CFThree)
CH2S (O) CH2CH2CFThree                      CH2(D1-108b, Z = 4-OCFThree)
CH2S (O) CH2CH2CFThree                      CH2(D1-108b, Z = 2-SCFThree)
CH2S (O) CH2CH2CFThree                      CH2CH2CN
CH2S (O) CH2CH2CFThree                      CH2CH2CFThree
CH2S (O) CH2CH2CFThree                      CH2CH2OMe
CH2S (O) CH2CH2CFThree                      CH2CH2SMe
CH2S (O) CH2CH2CFThree                      CH2CH2S (O) Me
CH2S (O) CH2CH2CFThree                      CH2CH2S (O)2Me
CH2S (O) CH2CH2CFThree                      D1-32a
CH2S (O) CH2CH2CFThree                      D1-33a
CH2S (O) CH2CH2CFThree                      D1-34a
CH2S (O) CH2CH2CFThree                      D1-37a
CH2S (O) CH2CH2CFThree                      D1-81a
CH2S (O) CH2CH2CFThree                      D1-82a
CH2S (O) CH2CH2CFThree                      D1-84a
CH2S (O) CH2CH2CFThree                      D1-85a
CH2S (O) CH2CH2CFThree                      D1-87a
CH2S (O) CH2CH2CFThree                      D1-92a
CH2S (O) CH2CH2CFThree                      D1-93a
CH2S (O) CH2CH2CFThree                      D1-95a
CH2S (O) CH2CH2CFThree                      D1-96a
CH2S (O) CH2CH2CFThree                      D1-98a
CH2S (O) CH2CH2CFThree                      D1-108a
CH2S (O) CH2CH2CFThree                      D1-108b (Z = 2-Cl)
CH2S (O) CH2CH2CFThree                      D1-108b (Z = 3-Me)
CH2S (O) CH2CH2CFThree                      D1-108b (Z = 4-OMe)
CH2S (O) CH2CH2CFThree                      D1-108b (Z = 2-SMe)
CH2S (O) CH2CH2CFThree                      D1-108b (Z = 3-CFThree)
CH2S (O) CH2CH2CFThree                      D1-108b (Z = 4-OCFThree)
CH2S (O) CH2CH2CFThree                      D1-108b (Z = 2-SCFThree)
CH2S (O) CH2CH2CFThree                      C (O) Me
CH2S (O) CH2CH2CFThree                      C (O) CFThree
CH2S (O) CH2CH2CFThree                      C (O) OMe
CH2S (O)2CH2CH2CFThree                      Me
CH2S (O)2CH2CH2CFThree                      Et
CH2S (O)2CH2CH2CFThree                      Pr-n
CH2S (O)2CH2CH2CFThree                      Pr-i
CH2S (O)2CH2CH2CFThree                      Pr-c
CH2S (O)2CH2CH2CFThree                      Bu-n
CH2S (O)2CH2CH2CFThree                      Bu-i
CH2S (O)2CH2CH2CFThree                      Bu-c
CH2S (O)2CH2CH2CFThree                      Bu-s
CH2S (O)2CH2CH2CFThree                      Bu-t
CH2S (O)2CH2CH2CFThree                      Pen-n
CH2S (O)2CH2CH2CFThree                      Pen-c
CH2S (O)2CH2CH2CFThree                      Hex-n
CH2S (O)2CH2CH2CFThree                      Hex-c
CH2S (O)2CH2CH2CFThree                      CH2Pr-c
CH2S (O)2CH2CH2CFThree                      CH2Bu-c
CH2S (O)2CH2CH2CFThree                      CH2Pen-c
CH2S (O)2CH2CH2CFThree                      CH2Hex-c
CH2S (O)2CH2CH2CFThree                      CH2CH = CH2
CH2S (O)2CH2CH2CFThree                      CH2CH = C (Cl)2
CH2S (O)2CH2CH2CFThree                      CH2C≡CH
CH2S (O)2CH2CH2CFThree                      CH2CN
CH2S (O)2CH2CH2CFThree                      CH2CFThree
CH2S (O)2CH2CH2CFThree                      CH2OMe
CH2S (O)2CH2CH2CFThree                      CH2OCFThree
CH2S (O)2CH2CH2CFThree                      CH2SMe
CH2S (O)2CH2CH2CFThree                      CH2S (O) Me
CH2S (O)2CH2CH2CFThree                      CH2S (O)2Me
CH2S (O)2CH2CH2CFThree                      CH2SCFThree
CH2S (O)2CH2CH2CFThree                      CH2S (O) CFThree
CH2S (O)2CH2CH2CFThree                      CH2S (O)2CFThree
CH2S (O)2CH2CH2CFThree                      CH2CH (OMe)2
CH2S (O)2CH2CH2CFThree                      CH2CH (SMe)2
CH2S (O)2CH2CH2CFThree                      CH2C (O) Me
CH2S (O)2CH2CH2CFThree                      CH2C (O) CFThree
CH2S (O)2CH2CH2CFThree                      CH2C (O) OMe
CH2S (O)2CH2CH2CFThree                      CH2(D1-32a)
CH2S (O)2CH2CH2CFThree                      CH2(D1-33a)
CH2S (O)2CH2CH2CFThree                      CH2(D1-34a)
CH2S (O)2CH2CH2CFThree                      CH2(D1-37a)
CH2S (O)2CH2CH2CFThree                      CH2(D1-81a)
CH2S (O)2CH2CH2CFThree                      CH2(D1-82a)
CH2S (O)2CH2CH2CFThree                      CH2(D1-84a)
CH2S (O)2CH2CH2CFThree                      CH2(D1-85a)
CH2S (O)2CH2CH2CFThree                      CH2(D1-87a)
CH2S (O)2CH2CH2CFThree                      CH2(D1-92a)
CH2S (O)2CH2CH2CFThree                      CH2(D1-93a)
CH2S (O)2CH2CH2CFThree                      CH2(D1-95a)
CH2S (O)2CH2CH2CFThree                      CH2(D1-96a)
CH2S (O)2CH2CH2CFThree                      CH2(D1-98a)
CH2S (O)2CH2CH2CFThree                      CH2(D1-108a)
CH2S (O)2CH2CH2CFThree                      CH2(D1-108b, Z = 2-Cl)
CH2S (O)2CH2CH2CFThree                      CH2(D1-108b, Z = 3-Me)
CH2S (O)2CH2CH2CFThree                      CH2(D1-108b, Z = 4-OMe)
CH2S (O)2CH2CH2CFThree                      CH2(D1-108b, Z = 2-SMe)
CH2S (O)2CH2CH2CFThree                      CH2(D1-108b, Z = 3-CFThree)
CH2S (O)2CH2CH2CFThree                      CH2(D1-108b, Z = 4-OCFThree)
CH2S (O)2CH2CH2CFThree                      CH2(D1-108b, Z = 2-SCFThree)
CH2S (O)2CH2CH2CFThree                      CH2CH2CN
CH2S (O)2CH2CH2CFThree                      CH2CH2CFThree
CH2S (O)2CH2CH2CFThree                      CH2CH2OMe
CH2S (O)2CH2CH2CFThree                      CH2CH2SMe
CH2S (O)2CH2CH2CFThree                      CH2CH2S (O) Me
CH2S (O)2CH2CH2CFThree                      CH2CH2S (O)2Me
CH2S (O)2CH2CH2CFThree                      D1-32a
CH2S (O)2CH2CH2CFThree                      D1-33a
CH2S (O)2CH2CH2CFThree                      D1-34a
CH2S (O)2CH2CH2CFThree                      D1-37a
CH2S (O)2CH2CH2CFThree                      D1-81a
CH2S (O)2CH2CH2CFThree                      D1-82a
CH2S (O)2CH2CH2CFThree                      D1-84a
CH2S (O)2CH2CH2CFThree                      D1-85a
CH2S (O)2CH2CH2CFThree                      D1-87a
CH2S (O)2CH2CH2CFThree                      D1-92a
CH2S (O)2CH2CH2CFThree                      D1-93a
CH2S (O)2CH2CH2CFThree                      D1-95a
CH2S (O)2CH2CH2CFThree                      D1-96a
CH2S (O)2CH2CH2CFThree                      D1-98a
CH2S (O)2CH2CH2CFThree                      D1-108a
CH2S (O)2CH2CH2CFThree                      D1-108b (Z = 2-Cl)
CH2S (O)2CH2CH2CFThree                      D1-108b (Z = 3-Me)
CH2S (O)2CH2CH2CFThree                      D1-108b (Z = 4-OMe)
CH2S (O)2CH2CH2CFThree                      D1-108b (Z = 2-SMe)
CH2S (O)2CH2CH2CFThree                      D1-108b (Z = 3-CFThree)
CH2S (O)2CH2CH2CFThree                      D1-108b (Z = 4-OCFThree)
CH2S (O)2CH2CH2CFThree                      D1-108b (Z = 2-SCFThree)
CH2S (O)2CH2CH2CFThree                      C (O) Me
CH2S (O)2CH2CH2CFThree                      C (O) CFThree
CH2S (O)2CH2CH2CFThree                      C (O) OMe
CH (Me) SCH2CH2CFThree                      Me
CH (Me) SCH2CH2CFThree                      Et
CH (Me) SCH2CH2CFThree                      Pr-n
CH (Me) SCH2CH2CFThree                      Pr-i
CH (Me) SCH2CH2CFThree                      Pr-c
CH (Me) SCH2CH2CFThree                      Bu-n
CH (Me) SCH2CH2CFThree                      Bu-i
CH (Me) SCH2CH2CFThree                      Bu-c
CH (Me) SCH2CH2CFThree                      Bu-s
CH (Me) SCH2CH2CFThree                      Bu-t
CH (Me) SCH2CH2CFThree                      Pen-n
CH (Me) SCH2CH2CFThree                      Pen-c
CH (Me) SCH2CH2CFThree                      Hex-n
CH (Me) SCH2CH2CFThree                      Hex-c
CH (Me) SCH2CH2CFThree                      CH2Pr-c
CH (Me) SCH2CH2CFThree                      CH2Bu-c
CH (Me) SCH2CH2CFThree                      CH2Pen-c
CH (Me) SCH2CH2CFThree                      CH2Hex-c
CH (Me) SCH2CH2CFThree                      CH2CH = CH2
CH (Me) SCH2CH2CFThree                      CH2CH = C (Cl)2
CH (Me) SCH2CH2CFThree                      CH2C≡CH
CH (Me) SCH2CH2CFThree                      CH2CN
CH (Me) SCH2CH2CFThree                      CH2CFThree
CH (Me) SCH2CH2CFThree                      CH2OMe
CH (Me) SCH2CH2CFThree                      CH2OCFThree
CH (Me) SCH2CH2CFThree                      CH2SMe
CH (Me) SCH2CH2CFThree                      CH2S (O) Me
CH (Me) SCH2CH2CFThree                      CH2S (O)2Me
CH (Me) SCH2CH2CFThree                      CH2SCFThree
CH (Me) SCH2CH2CFThree                      CH2S (O) CFThree
CH (Me) SCH2CH2CFThree                      CH2S (O)2CFThree
CH (Me) SCH2CH2CFThree                      CH2CH (OMe)2
CH (Me) SCH2CH2CFThree                      CH2CH (SMe)2
CH (Me) SCH2CH2CFThree                      CH2C (O) Me
CH (Me) SCH2CH2CFThree                      CH2C (O) CFThree
CH (Me) SCH2CH2CFThree                      CH2C (O) OMe
CH (Me) SCH2CH2CFThree                      CH2(D1-32a)
CH (Me) SCH2CH2CFThree                      CH2(D1-33a)
CH (Me) SCH2CH2CFThree                      CH2(D1-34a)
CH (Me) SCH2CH2CFThree                      CH2(D1-37a)
CH (Me) SCH2CH2CFThree                      CH2(D1-81a)
CH (Me) SCH2CH2CFThree                      CH2(D1-82a)
CH (Me) SCH2CH2CFThree                      CH2(D1-84a)
CH (Me) SCH2CH2CFThree                      CH2(D1-85a)
CH (Me) SCH2CH2CFThree                      CH2(D1-87a)
CH (Me) SCH2CH2CFThree                      CH2(D1-92a)
CH (Me) SCH2CH2CFThree                      CH2(D1-93a)
CH (Me) SCH2CH2CFThree                      CH2(D1-95a)
CH (Me) SCH2CH2CFThree                      CH2(D1-96a)
CH (Me) SCH2CH2CFThree                      CH2(D1-98a)
CH (Me) SCH2CH2CFThree                      CH2(D1-108a)
CH (Me) SCH2CH2CFThree                      CH2(D1-108b, Z = 2-Cl)
CH (Me) SCH2CH2CFThree                      CH2(D1-108b, Z = 3-Me)
CH (Me) SCH2CH2CFThree                      CH2(D1-108b, Z = 4-OMe)
CH (Me) SCH2CH2CFThree                      CH2(D1-108b, Z = 2-SMe)
CH (Me) SCH2CH2CFThree                      CH2(D1-108b, Z = 3-CFThree)
CH (Me) SCH2CH2CFThree                      CH2(D1-108b, Z = 4-OCFThree)
CH (Me) SCH2CH2CFThree                      CH2(D1-108b, Z = 2-SCFThree)
CH (Me) SCH2CH2CFThree                      CH2CH2CN
CH (Me) SCH2CH2CFThree                      CH2CH2CFThree
CH (Me) SCH2CH2CFThree                      CH2CH2OMe
CH (Me) SCH2CH2CFThree                      CH2CH2SMe
CH (Me) SCH2CH2CFThree                      CH2CH2S (O) Me
CH (Me) SCH2CH2CFThree                      CH2CH2S (O)2Me
CH (Me) SCH2CH2CFThree                      D1-32a
CH (Me) SCH2CH2CFThree                      D1-33a
CH (Me) SCH2CH2CFThree                      D1-34a
CH (Me) SCH2CH2CFThree                      D1-37a
CH (Me) SCH2CH2CFThree                      D1-81a
CH (Me) SCH2CH2CFThree                      D1-82a
CH (Me) SCH2CH2CFThree                      D1-84a
CH (Me) SCH2CH2CFThree                      D1-85a
CH (Me) SCH2CH2CFThree                      D1-87a
CH (Me) SCH2CH2CFThree                      D1-92a
CH (Me) SCH2CH2CFThree                      D1-93a
CH (Me) SCH2CH2CFThree                      D1-95a
CH (Me) SCH2CH2CFThree                      D1-96a
CH (Me) SCH2CH2CFThree                      D1-98a
CH (Me) SCH2CH2CFThree                      D1-108a
CH (Me) SCH2CH2CFThree                      D1-108b (Z = 2-Cl)
CH (Me) SCH2CH2CFThree                      D1-108b (Z = 3-Me)
CH (Me) SCH2CH2CFThree                      D1-108b (Z = 4-OMe)
CH (Me) SCH2CH2CFThree                      D1-108b (Z = 2-SMe)
CH (Me) SCH2CH2CFThree                      D1-108b (Z = 3-CFThree)
CH (Me) SCH2CH2CFThree                      D1-108b (Z = 4-OCFThree)
CH (Me) SCH2CH2CFThree                      D1-108b (Z = 2-SCFThree)
CH (Me) SCH2CH2CFThree                      C (O) Me
CH (Me) SCH2CH2CFThree                      C (O) CFThree
CH (Me) SCH2CH2CFThree                      C (O) OMe
CH (Me) S (O) CH2CH2CFThree                   Me
CH (Me) S (O) CH2CH2CFThree                   Et
CH (Me) S (O) CH2CH2CFThree                   Pr-n
CH (Me) S (O) CH2CH2CFThree                   Pr-i
CH (Me) S (O) CH2CH2CFThree                   Pr-c
CH (Me) S (O) CH2CH2CFThree                   Bu-n
CH (Me) S (O) CH2CH2CFThree                   Bu-i
CH (Me) S (O) CH2CH2CFThree                   Bu-c
CH (Me) S (O) CH2CH2CFThree                   Bu-s
CH (Me) S (O) CH2CH2CFThree                   Bu-t
CH (Me) S (O) CH2CH2CFThree                   Pen-n
CH (Me) S (O) CH2CH2CFThree                   Pen-c
CH (Me) S (O) CH2CH2CFThree                   Hex-n
CH (Me) S (O) CH2CH2CFThree                   Hex-c
CH (Me) S (O) CH2CH2CFThree                   CH2Pr-c
CH (Me) S (O) CH2CH2CFThree                   CH2Bu-c
CH (Me) S (O) CH2CH2CFThree                   CH2Pen-c
CH (Me) S (O) CH2CH2CFThree                   CH2Hex-c
CH (Me) S (O) CH2CH2CFThree                   CH2CH = CH2
CH (Me) S (O) CH2CH2CFThree                   CH2CH = C (Cl)2
CH (Me) S (O) CH2CH2CFThree                   CH2C≡CH
CH (Me) S (O) CH2CH2CFThree                   CH2CN
CH (Me) S (O) CH2CH2CFThree                   CH2CFThree
CH (Me) S (O) CH2CH2CFThree                   CH2OMe
CH (Me) S (O) CH2CH2CFThree                   CH2OCFThree
CH (Me) S (O) CH2CH2CFThree                   CH2SMe
CH (Me) S (O) CH2CH2CFThree                   CH2S (O) Me
CH (Me) S (O) CH2CH2CFThree                   CH2S (O)2Me
CH (Me) S (O) CH2CH2CFThree                   CH2SCFThree
CH (Me) S (O) CH2CH2CFThree                   CH2S (O) CFThree
CH (Me) S (O) CH2CH2CFThree                   CH2S (O)2CFThree
CH (Me) S (O) CH2CH2CFThree                   CH2CH (OMe)2
CH (Me) S (O) CH2CH2CFThree                   CH2CH (SMe)2
CH (Me) S (O) CH2CH2CFThree                   CH2C (O) Me
CH (Me) S (O) CH2CH2CFThree                   CH2C (O) CFThree
CH (Me) S (O) CH2CH2CFThree                   CH2C (O) OMe
CH (Me) S (O) CH2CH2CFThree                   CH2(D1-32a)
CH (Me) S (O) CH2CH2CFThree                   CH2(D1-33a)
CH (Me) S (O) CH2CH2CFThree                   CH2(D1-34a)
CH (Me) S (O) CH2CH2CFThree                   CH2(D1-37a)
CH (Me) S (O) CH2CH2CFThree                   CH2(D1-81a)
CH (Me) S (O) CH2CH2CFThree                   CH2(D1-82a)
CH (Me) S (O) CH2CH2CFThree                   CH2(D1-84a)
CH (Me) S (O) CH2CH2CFThree                   CH2(D1-85a)
CH (Me) S (O) CH2CH2CFThree                   CH2(D1-87a)
CH (Me) S (O) CH2CH2CFThree                   CH2(D1-92a)
CH (Me) S (O) CH2CH2CFThree                   CH2(D1-93a)
CH (Me) S (O) CH2CH2CFThree                   CH2(D1-95a)
CH (Me) S (O) CH2CH2CFThree                   CH2(D1-96a)
CH (Me) S (O) CH2CH2CFThree                   CH2(D1-98a)
CH (Me) S (O) CH2CH2CFThree                   CH2(D1-108a)
CH (Me) S (O) CH2CH2CFThree                   CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O) CH2CH2CFThree                   CH2(D1-108b, Z = 3-Me)
CH (Me) S (O) CH2CH2CFThree                   CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O) CH2CH2CFThree                   CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O) CH2CH2CFThree                   CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O) CH2CH2CFThree                   CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O) CH2CH2CFThree                   CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O) CH2CH2CFThree                   CH2CH2CN
CH (Me) S (O) CH2CH2CFThree                   CH2CH2CFThree
CH (Me) S (O) CH2CH2CFThree                   CH2CH2OMe
CH (Me) S (O) CH2CH2CFThree                   CH2CH2SMe
CH (Me) S (O) CH2CH2CFThree                   CH2CH2S (O) Me
CH (Me) S (O) CH2CH2CFThree                   CH2CH2S (O)2Me
CH (Me) S (O) CH2CH2CFThree                   D1-32a
CH (Me) S (O) CH2CH2CFThree                   D1-33a
CH (Me) S (O) CH2CH2CFThree                   D1-34a
CH (Me) S (O) CH2CH2CFThree                   D1-37a
CH (Me) S (O) CH2CH2CFThree                   D1-81a
CH (Me) S (O) CH2CH2CFThree                   D1-82a
CH (Me) S (O) CH2CH2CFThree                   D1-84a
CH (Me) S (O) CH2CH2CFThree                   D1-85a
CH (Me) S (O) CH2CH2CFThree                   D1-87a
CH (Me) S (O) CH2CH2CFThree                   D1-92a
CH (Me) S (O) CH2CH2CFThree                   D1-93a
CH (Me) S (O) CH2CH2CFThree                   D1-95a
CH (Me) S (O) CH2CH2CFThree                   D1-96a
CH (Me) S (O) CH2CH2CFThree                   D1-98a
CH (Me) S (O) CH2CH2CFThree                   D1-108a
CH (Me) S (O) CH2CH2CFThree                   D1-108b (Z = 2-Cl)
CH (Me) S (O) CH2CH2CFThree                   D1-108b (Z = 3-Me)
CH (Me) S (O) CH2CH2CFThree                   D1-108b (Z = 4-OMe)
CH (Me) S (O) CH2CH2CFThree                   D1-108b (Z = 2-SMe)
CH (Me) S (O) CH2CH2CFThree                   D1-108b (Z = 3-CFThree)
CH (Me) S (O) CH2CH2CFThree                   D1-108b (Z = 4-OCFThree)
CH (Me) S (O) CH2CH2CFThree                   D1-108b (Z = 2-SCFThree)
CH (Me) S (O) CH2CH2CFThree                   C (O) Me
CH (Me) S (O) CH2CH2CFThree                   C (O) CFThree
CH (Me) S (O) CH2CH2CFThree                   C (O) OMe
CH (Me) S (O)2CH2CH2CFThree                   Me
CH (Me) S (O)2CH2CH2CFThree                   Et
CH (Me) S (O)2CH2CH2CFThree                   Pr-n
CH (Me) S (O)2CH2CH2CFThree                   Pr-i
CH (Me) S (O)2CH2CH2CFThree                   Pr-c
CH (Me) S (O)2CH2CH2CFThree                   Bu-n
CH (Me) S (O)2CH2CH2CFThree                   Bu-i
CH (Me) S (O)2CH2CH2CFThree                   Bu-c
CH (Me) S (O)2CH2CH2CFThree                   Bu-s
CH (Me) S (O)2CH2CH2CFThree                   Bu-t
CH (Me) S (O)2CH2CH2CFThree                   Pen-n
CH (Me) S (O)2CH2CH2CFThree                   Pen-c
CH (Me) S (O)2CH2CH2CFThree                   Hex-n
CH (Me) S (O)2CH2CH2CFThree                   Hex-c
CH (Me) S (O)2CH2CH2CFThree                   CH2Pr-c
CH (Me) S (O)2CH2CH2CFThree                   CH2Bu-c
CH (Me) S (O)2CH2CH2CFThree                   CH2Pen-c
CH (Me) S (O)2CH2CH2CFThree                   CH2Hex-c
CH (Me) S (O)2CH2CH2CFThree                   CH2CH = CH2
CH (Me) S (O)2CH2CH2CFThree                   CH2CH = C (Cl)2
CH (Me) S (O)2CH2CH2CFThree                   CH2C≡CH
CH (Me) S (O)2CH2CH2CFThree                   CH2CN
CH (Me) S (O)2CH2CH2CFThree                   CH2CFThree
CH (Me) S (O)2CH2CH2CFThree                   CH2OMe
CH (Me) S (O)2CH2CH2CFThree                   CH2OCFThree
CH (Me) S (O)2CH2CH2CFThree                   CH2SMe
CH (Me) S (O)2CH2CH2CFThree                  CH2S (O) Me
CH (Me) S (O)2CH2CH2CFThree                   CH2S (O)2Me
CH (Me) S (O)2CH2CH2CFThree                   CH2SCFThree
CH (Me) S (O)2CH2CH2CFThree                   CH2S (O) CFThree
CH (Me) S (O)2CH2CH2CFThree                   CH2S (O)2CFThree
CH (Me) S (O)2CH2CH2CFThree                   CH2CH (OMe)2
CH (Me) S (O)2CH2CH2CFThree                   CH2CH (SMe)2
CH (Me) S (O)2CH2CH2CFThree                   CH2C (O) Me
CH (Me) S (O)2CH2CH2CFThree                   CH2C (O) CFThree
CH (Me) S (O)2CH2CH2CFThree                   CH2C (O) OMe
CH (Me) S (O)2CH2CH2CFThree                   CH2(D1-32a)
CH (Me) S (O)2CH2CH2CFThree                   CH2(D1-33a)
CH (Me) S (O)2CH2CH2CFThree                   CH2(D1-34a)
CH (Me) S (O)2CH2CH2CFThree                   CH2(D1-37a)
CH (Me) S (O)2CH2CH2CFThree                   CH2(D1-81a)
CH (Me) S (O)2CH2CH2CFThree                   CH2(D1-82a)
CH (Me) S (O)2CH2CH2CFThree                   CH2(D1-84a)
CH (Me) S (O)2CH2CH2CFThree                   CH2(D1-85a)
CH (Me) S (O)2CH2CH2CFThree                   CH2(D1-87a)
CH (Me) S (O)2CH2CH2CFThree                   CH2(D1-92a)
CH (Me) S (O)2CH2CH2CFThree                   CH2(D1-93a)
CH (Me) S (O)2CH2CH2CFThree                   CH2(D1-95a)
CH (Me) S (O)2CH2CH2CFThree                   CH2(D1-96a)
CH (Me) S (O)2CH2CH2CFThree                   CH2(D1-98a)
CH (Me) S (O)2CH2CH2CFThree                   CH2(D1-108a)
CH (Me) S (O)2CH2CH2CFThree                   CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O)2CH2CH2CFThree                   CH2(D1-108b, Z = 3-Me)
CH (Me) S (O)2CH2CH2CFThree                   CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O)2CH2CH2CFThree                   CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O)2CH2CH2CFThree                   CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O)2CH2CH2CFThree                   CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O)2CH2CH2CFThree                   CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O)2CH2CH2CFThree                   CH2CH2CN
CH (Me) S (O)2CH2CH2CFThree                   CH2CH2CFThree
CH (Me) S (O)2CH2CH2CFThree                   CH2CH2OMe
CH (Me) S (O)2CH2CH2CFThree                   CH2CH2SMe
CH (Me) S (O)2CH2CH2CFThree                   CH2CH2S (O) Me
CH (Me) S (O)2CH2CH2CFThree                   CH2CH2S (O)2Me
CH (Me) S (O)2CH2CH2CFThree                   D1-32a
CH (Me) S (O)2CH2CH2CFThree                   D1-33a
CH (Me) S (O)2CH2CH2CFThree                   D1-34a
CH (Me) S (O)2CH2CH2CFThree                   D1-37a
CH (Me) S (O)2CH2CH2CFThree                   D1-81a
CH (Me) S (O)2CH2CH2CFThree                   D1-82a
CH (Me) S (O)2CH2CH2CFThree                   D1-84a
CH (Me) S (O)2CH2CH2CFThree                   D1-85a
CH (Me) S (O)2CH2CH2CFThree                   D1-87a
CH (Me) S (O)2CH2CH2CFThree                   D1-92a
CH (Me) S (O)2CH2CH2CFThree                   D1-93a
CH (Me) S (O)2CH2CH2CFThree                   D1-95a
CH (Me) S (O)2CH2CH2CFThree                   D1-96a
CH (Me) S (O)2CH2CH2CFThree                   D1-98a
CH (Me) S (O)2CH2CH2CFThree                   D1-108a
CH (Me) S (O)2CH2CH2CFThree                   D1-108b (Z = 2-Cl)
CH (Me) S (O)2CH2CH2CFThree                   D1-108b (Z = 3-Me)
CH (Me) S (O)2CH2CH2CFThree                   D1-108b (Z = 4-OMe)
CH (Me) S (O)2CH2CH2CFThree                   D1-108b (Z = 2-SMe)
CH (Me) S (O)2CH2CH2CFThree                   D1-108b (Z = 3-CFThree)
CH (Me) S (O)2CH2CH2CFThree                   D1-108b (Z = 4-OCFThree)
CH (Me) S (O)2CH2CH2CFThree                   D1-108b (Z = 2-SCFThree)
CH (Me) S (O)2CH2CH2CFThree                   C (O) Me
CH (Me) S (O)2CH2CH2CFThree                   C (O) CFThree
CH (Me) S (O)2CH2CH2CFThree                   C (O) OMe
CH (Et) SCH2CH2CFThree                      Me
CH (Et) SCH2CH2CFThree                      Et
CH (Et) SCH2CH2CFThree                      Pr-n
CH (Et) SCH2CH2CFThree                     Pr-i
CH (Et) SCH2CH2CFThree                      Pr-c
CH (Et) SCH2CH2CFThree                      Bu-n
CH (Et) SCH2CH2CFThree                      Bu-i
CH (Et) SCH2CH2CFThree                      Bu-c
CH (Et) SCH2CH2CFThree                      Bu-s
CH (Et) SCH2CH2CFThree                      Bu-t
CH (Et) SCH2CH2CFThree                      Pen-n
CH (Et) SCH2CH2CFThree                      Pen-c
CH (Et) SCH2CH2CFThree                      Hex-n
CH (Et) SCH2CH2CFThree                      Hex-c
CH (Et) SCH2CH2CFThree                      CH2Pr-c
CH (Et) SCH2CH2CFThree                      CH2Bu-c
CH (Et) SCH2CH2CFThree                      CH2Pen-c
CH (Et) SCH2CH2CFThree                      CH2Hex-c
CH (Et) SCH2CH2CFThree                      CH2CH = CH2
CH (Et) SCH2CH2CFThree                      CH2CH = C (Cl)2
CH (Et) SCH2CH2CFThree                      CH2C≡CH
CH (Et) SCH2CH2CFThree                      CH2CN
CH (Et) SCH2CH2CFThree                      CH2CFThree
CH (Et) SCH2CH2CFThree                      CH2OMe
CH (Et) SCH2CH2CFThree                      CH2OCFThree
CH (Et) SCH2CH2CFThree                      CH2SMe
CH (Et) SCH2CH2CFThree                      CH2S (O) Me
CH (Et) SCH2CH2CFThree                      CH2S (O)2Me
CH (Et) SCH2CH2CFThree                      CH2SCFThree
CH (Et) SCH2CH2CFThree                      CH2S (O) CFThree
CH (Et) SCH2CH2CFThree                      CH2S (O)2CFThree
CH (Et) SCH2CH2CFThree                      CH2CH (OMe)2
CH (Et) SCH2CH2CFThree                      CH2CH (SMe)2
CH (Et) SCH2CH2CFThree                      CH2C (O) Me
CH (Et) SCH2CH2CFThree                      CH2C (O) CFThree
CH (Et) SCH2CH2CFThree                      CH2C (O) OMe
CH (Et) SCH2CH2CFThree                      CH2(D1-32a)
CH (Et) SCH2CH2CFThree                      CH2(D1-33a)
CH (Et) SCH2CH2CFThree                      CH2(D1-34a)
CH (Et) SCH2CH2CFThree                      CH2(D1-37a)
CH (Et) SCH2CH2CFThree                      CH2(D1-81a)
CH (Et) SCH2CH2CFThree                      CH2(D1-82a)
CH (Et) SCH2CH2CFThree                      CH2(D1-84a)
CH (Et) SCH2CH2CFThree                      CH2(D1-85a)
CH (Et) SCH2CH2CFThree                      CH2(D1-87a)
CH (Et) SCH2CH2CFThree                      CH2(D1-92a)
CH (Et) SCH2CH2CFThree                      CH2(D1-93a)
CH (Et) SCH2CH2CFThree                      CH2(D1-95a)
CH (Et) SCH2CH2CFThree                      CH2(D1-96a)
CH (Et) SCH2CH2CFThree                      CH2(D1-98a)
CH (Et) SCH2CH2CFThree                      CH2(D1-108a)
CH (Et) SCH2CH2CFThree                      CH2(D1-108b, Z = 2-Cl)
CH (Et) SCH2CH2CFThree                      CH2(D1-108b, Z = 3-Me)
CH (Et) SCH2CH2CFThree                      CH2(D1-108b, Z = 4-OMe)
CH (Et) SCH2CH2CFThree                      CH2(D1-108b, Z = 2-SMe)
CH (Et) SCH2CH2CFThree                      CH2(D1-108b, Z = 3-CFThree)
CH (Et) SCH2CH2CFThree                      CH2(D1-108b, Z = 4-OCFThree)
CH (Et) SCH2CH2CFThree                      CH2(D1-108b, Z = 2-SCFThree)
CH (Et) SCH2CH2CFThree                      CH2CH2CN
CH (Et) SCH2CH2CFThree                      CH2CH2CFThree
CH (Et) SCH2CH2CFThree                      CH2CH2OMe
CH (Et) SCH2CH2CFThree                      CH2CH2SMe
CH (Et) SCH2CH2CFThree                      CH2CH2S (O) Me
CH (Et) SCH2CH2CFThree                      CH2CH2S (O)2Me
CH (Et) SCH2CH2CFThree                      D1-32a
CH (Et) SCH2CH2CFThree                      D1-33a
CH (Et) SCH2CH2CFThree                      D1-34a
CH (Et) SCH2CH2CFThree                      D1-37a
CH (Et) SCH2CH2CFThree                      D1-81a
CH (Et) SCH2CH2CFThree                      D1-82a
CH (Et) SCH2CH2CFThree                      D1-84a
CH (Et) SCH2CH2CFThree                      D1-85a
CH (Et) SCH2CH2CFThree                      D1-87a
CH (Et) SCH2CH2CFThree                      D1-92a
CH (Et) SCH2CH2CFThree                      D1-93a
CH (Et) SCH2CH2CFThree                      D1-95a
CH (Et) SCH2CH2CFThree                      D1-96a
CH (Et) SCH2CH2CFThree                      D1-98a
CH (Et) SCH2CH2CFThree                      D1-108a
CH (Et) SCH2CH2CFThree                      D1-108b (Z = 2-Cl)
CH (Et) SCH2CH2CFThree                      D1-108b (Z = 3-Me)
CH (Et) SCH2CH2CFThree                      D1-108b (Z = 4-OMe)
CH (Et) SCH2CH2CFThree                      D1-108b (Z = 2-SMe)
CH (Et) SCH2CH2CFThree                      D1-108b (Z = 3-CFThree)
CH (Et) SCH2CH2CFThree                      D1-108b (Z = 4-OCFThree)
CH (Et) SCH2CH2CFThree                      D1-108b (Z = 2-SCFThree)
CH (Et) SCH2CH2CFThree                      C (O) Me
CH (Et) SCH2CH2CFThree                      C (O) CFThree
CH (Et) SCH2CH2CFThree                      C (O) OMe
CH (Et) S (O) CH2CH2CFThree                   Me
CH (Et) S (O) CH2CH2CFThree                   Et
CH (Et) S (O) CH2CH2CFThree                   Pr-n
CH (Et) S (O) CH2CH2CFThree                   Pr-i
CH (Et) S (O) CH2CH2CFThree                   Pr-c
CH (Et) S (O) CH2CH2CFThree                   Bu-n
CH (Et) S (O) CH2CH2CFThree                   Bu-i
CH (Et) S (O) CH2CH2CFThree                   Bu-c
CH (Et) S (O) CH2CH2CFThree                   Bu-s
CH (Et) S (O) CH2CH2CFThree                   Bu-t
CH (Et) S (O) CH2CH2CFThree                   Pen-n
CH (Et) S (O) CH2CH2CFThree                   Pen-c
CH (Et) S (O) CH2CH2CFThree                   Hex-n
CH (Et) S (O) CH2CH2CFThree                   Hex-c
CH (Et) S (O) CH2CH2CFThree                   CH2Pr-c
CH (Et) S (O) CH2CH2CFThree                   CH2Bu-c
CH (Et) S (O) CH2CH2CFThree                   CH2Pen-c
CH (Et) S (O) CH2CH2CFThree                   CH2Hex-c
CH (Et) S (O) CH2CH2CFThree                   CH2CH = CH2
CH (Et) S (O) CH2CH2CFThree                   CH2CH = C (Cl)2
CH (Et) S (O) CH2CH2CFThree                   CH2C≡CH
CH (Et) S (O) CH2CH2CFThree                   CH2CN
CH (Et) S (O) CH2CH2CFThree                   CH2CFThree
CH (Et) S (O) CH2CH2CFThree                   CH2OMe
CH (Et) S (O) CH2CH2CFThree                   CH2OCFThree
CH (Et) S (O) CH2CH2CFThree                   CH2SMe
CH (Et) S (O) CH2CH2CFThree                   CH2S (O) Me
CH (Et) S (O) CH2CH2CFThree                   CH2S (O)2Me
CH (Et) S (O) CH2CH2CFThree                   CH2SCFThree
CH (Et) S (O) CH2CH2CFThree                   CH2S (O) CFThree
CH (Et) S (O) CH2CH2CFThree                   CH2S (O)2CFThree
CH (Et) S (O) CH2CH2CFThree                   CH2CH (OMe)2
CH (Et) S (O) CH2CH2CFThree                   CH2CH (SMe)2
CH (Et) S (O) CH2CH2CFThree                   CH2C (O) Me
CH (Et) S (O) CH2CH2CFThree                   CH2C (O) CFThree
CH (Et) S (O) CH2CH2CFThree                   CH2C (O) OMe
CH (Et) S (O) CH2CH2CFThree                   CH2(D1-32a)
CH (Et) S (O) CH2CH2CFThree                   CH2(D1-33a)
CH (Et) S (O) CH2CH2CFThree                   CH2(D1-34a)
CH (Et) S (O) CH2CH2CFThree                   CH2(D1-37a)
CH (Et) S (O) CH2CH2CFThree                   CH2(D1-81a)
CH (Et) S (O) CH2CH2CFThree                   CH2(D1-82a)
CH (Et) S (O) CH2CH2CFThree                   CH2(D1-84a)
CH (Et) S (O) CH2CH2CFThree                   CH2(D1-85a)
CH (Et) S (O) CH2CH2CFThree                   CH2(D1-87a)
CH (Et) S (O) CH2CH2CFThree                   CH2(D1-92a)
CH (Et) S (O) CH2CH2CFThree                   CH2(D1-93a)
CH (Et) S (O) CH2CH2CFThree                   CH2(D1-95a)
CH (Et) S (O) CH2CH2CFThree                   CH2(D1-96a)
CH (Et) S (O) CH2CH2CFThree                   CH2(D1-98a)
CH (Et) S (O) CH2CH2CFThree                   CH2(D1-108a)
CH (Et) S (O) CH2CH2CFThree                   CH2(D1-108b, Z = 2-Cl)
CH (Et) S (O) CH2CH2CFThree                   CH2(D1-108b, Z = 3-Me)
CH (Et) S (O) CH2CH2CFThree                   CH2(D1-108b, Z = 4-OMe)
CH (Et) S (O) CH2CH2CFThree                   CH2(D1-108b, Z = 2-SMe)
CH (Et) S (O) CH2CH2CFThree                   CH2(D1-108b, Z = 3-CFThree)
CH (Et) S (O) CH2CH2CFThree                   CH2(D1-108b, Z = 4-OCFThree)
CH (Et) S (O) CH2CH2CFThree                   CH2(D1-108b, Z = 2-SCFThree)
CH (Et) S (O) CH2CH2CFThree                   CH2CH2CN
CH (Et) S (O) CH2CH2CFThree                   CH2CH2CFThree
CH (Et) S (O) CH2CH2CFThree                   CH2CH2OMe
CH (Et) S (O) CH2CH2CFThree                   CH2CH2SMe
CH (Et) S (O) CH2CH2CFThree                   CH2CH2S (O) Me
CH (Et) S (O) CH2CH2CFThree                   CH2CH2S (O)2Me
CH (Et) S (O) CH2CH2CFThree                   D1-32a
CH (Et) S (O) CH2CH2CFThree                   D1-33a
CH (Et) S (O) CH2CH2CFThree                   D1-34a
CH (Et) S (O) CH2CH2CFThree                   D1-37a
CH (Et) S (O) CH2CH2CFThree                   D1-81a
CH (Et) S (O) CH2CH2CFThree                   D1-82a
CH (Et) S (O) CH2CH2CFThree                   D1-84a
CH (Et) S (O) CH2CH2CFThree                   D1-85a
CH (Et) S (O) CH2CH2CFThree                   D1-87a
CH (Et) S (O) CH2CH2CFThree                   D1-92a
CH (Et) S (O) CH2CH2CFThree                   D1-93a
CH (Et) S (O) CH2CH2CFThree                   D1-95a
CH (Et) S (O) CH2CH2CFThree                   D1-96a
CH (Et) S (O) CH2CH2CFThree                   D1-98a
CH (Et) S (O) CH2CH2CFThree                   D1-108a
CH (Et) S (O) CH2CH2CFThree                   D1-108b (Z = 2-Cl)
CH (Et) S (O) CH2CH2CFThree                   D1-108b (Z = 3-Me)
CH (Et) S (O) CH2CH2CFThree                   D1-108b (Z = 4-OMe)
CH (Et) S (O) CH2CH2CFThree                   D1-108b (Z = 2-SMe)
CH (Et) S (O) CH2CH2CFThree                   D1-108b (Z = 3-CFThree)
CH (Et) S (O) CH2CH2CFThree                   D1-108b (Z = 4-OCFThree)
CH (Et) S (O) CH2CH2CFThree                   D1-108b (Z = 2-SCFThree)
CH (Et) S (O) CH2CH2CFThree                   C (O) Me
CH (Et) S (O) CH2CH2CFThree                   C (O) CFThree
CH (Et) S (O) CH2CH2CFThree                   C (O) OMe
CH (Et) S (O)2CH2CH2CFThree                   Me
CH (Et) S (O)2CH2CH2CFThree                   Et
CH (Et) S (O)2CH2CH2CFThree                   Pr-n
CH (Et) S (O)2CH2CH2CFThree                   Pr-i
CH (Et) S (O)2CH2CH2CFThree                   Pr-c
CH (Et) S (O)2CH2CH2CFThree                   Bu-n
CH (Et) S (O)2CH2CH2CFThree                   Bu-i
CH (Et) S (O)2CH2CH2CFThree                   Bu-c
CH (Et) S (O)2CH2CH2CFThree                   Bu-s
CH (Et) S (O)2CH2CH2CFThree                   Bu-t
CH (Et) S (O)2CH2CH2CFThree                   Pen-n
CH (Et) S (O)2CH2CH2CFThree                   Pen-c
CH (Et) S (O)2CH2CH2CFThree                   Hex-n
CH (Et) S (O)2CH2CH2CFThree                   Hex-c
CH (Et) S (O)2CH2CH2CFThree                   CH2Pr-c
CH (Et) S (O)2CH2CH2CFThree                   CH2Bu-c
CH (Et) S (O)2CH2CH2CFThree                   CH2Pen-c
CH (Et) S (O)2CH2CH2CFThree                   CH2Hex-c
CH (Et) S (O)2CH2CH2CFThree                   CH2CH = CH2
CH (Et) S (O)2CH2CH2CFThree                   CH2CH = C (Cl)2
CH (Et) S (O)2CH2CH2CFThree                   CH2C≡CH
CH (Et) S (O)2CH2CH2CFThree                   CH2CN
CH (Et) S (O)2CH2CH2CFThree                   CH2CFThree
CH (Et) S (O)2CH2CH2CFThree                   CH2OMe
CH (Et) S (O)2CH2CH2CFThree                   CH2OCFThree
CH (Et) S (O)2CH2CH2CFThree                   CH2SMe
CH (Et) S (O)2CH2CH2CFThree                   CH2S (O) Me
CH (Et) S (O)2CH2CH2CFThree                   CH2S (O)2Me
CH (Et) S (O)2CH2CH2CFThree                   CH2SCFThree
CH (Et) S (O)2CH2CH2CFThree                   CH2S (O) CFThree
CH (Et) S (O)2CH2CH2CFThree                   CH2S (O)2CFThree
CH (Et) S (O)2CH2CH2CFThree                   CH2CH (OMe)2
CH (Et) S (O)2CH2CH2CFThree                   CH2CH (SMe)2
CH (Et) S (O)2CH2CH2CFThree                   CH2C (O) Me
CH (Et) S (O)2CH2CH2CFThree                   CH2C (O) CFThree
CH (Et) S (O)2CH2CH2CFThree                   CH2C (O) OMe
CH (Et) S (O)2CH2CH2CFThree                   CH2(D1-32a)
CH (Et) S (O)2CH2CH2CFThree                   CH2(D1-33a)
CH (Et) S (O)2CH2CH2CFThree                   CH2(D1-34a)
CH (Et) S (O)2CH2CH2CFThree                   CH2(D1-37a)
CH (Et) S (O)2CH2CH2CFThree                   CH2(D1-81a)
CH (Et) S (O)2CH2CH2CFThree                   CH2(D1-82a)
CH (Et) S (O)2CH2CH2CFThree                   CH2(D1-84a)
CH (Et) S (O)2CH2CH2CFThree                   CH2(D1-85a)
CH (Et) S (O)2CH2CH2CFThree                   CH2(D1-87a)
CH (Et) S (O)2CH2CH2CFThree                   CH2(D1-92a)
CH (Et) S (O)2CH2CH2CFThree                   CH2(D1-93a)
CH (Et) S (O)2CH2CH2CFThree                   CH2(D1-95a)
CH (Et) S (O)2CH2CH2CFThree                   CH2(D1-96a)
CH (Et) S (O)2CH2CH2CFThree                   CH2(D1-98a)
CH (Et) S (O)2CH2CH2CFThree                   CH2(D1-108a)
CH (Et) S (O)2CH2CH2CFThree                   CH2(D1-108b, Z = 2-Cl)
CH (Et) S (O)2CH2CH2CFThree                   CH2(D1-108b, Z = 3-Me)
CH (Et) S (O)2CH2CH2CFThree                   CH2(D1-108b, Z = 4-OMe)
CH (Et) S (O)2CH2CH2CFThree                   CH2(D1-108b, Z = 2-SMe)
CH (Et) S (O)2CH2CH2CFThree                   CH2(D1-108b, Z = 3-CFThree)
CH (Et) S (O)2CH2CH2CFThree                   CH2(D1-108b, Z = 4-OCFThree)
CH (Et) S (O)2CH2CH2CFThree                   CH2(D1-108b, Z = 2-SCFThree)
CH (Et) S (O)2CH2CH2CFThree                   CH2CH2CN
CH (Et) S (O)2CH2CH2CFThree                   CH2CH2CFThree
CH (Et) S (O)2CH2CH2CFThree                   CH2CH2OMe
CH (Et) S (O)2CH2CH2CFThree                   CH2CH2SMe
CH (Et) S (O)2CH2CH2CFThree                   CH2CH2S (O) Me
CH (Et) S (O)2CH2CH2CFThree                   CH2CH2S (O)2Me
CH (Et) S (O)2CH2CH2CFThree                   D1-32a
CH (Et) S (O)2CH2CH2CFThree                   D1-33a
CH (Et) S (O)2CH2CH2CFThree                   D1-34a
CH (Et) S (O)2CH2CH2CFThree                   D1-37a
CH (Et) S (O)2CH2CH2CFThree                   D1-81a
CH (Et) S (O)2CH2CH2CFThree                   D1-82a
CH (Et) S (O)2CH2CH2CFThree                   D1-84a
CH (Et) S (O)2CH2CH2CFThree                   D1-85a
CH (Et) S (O)2CH2CH2CFThree                   D1-87a
CH (Et) S (O)2CH2CH2CFThree                   D1-92a
CH (Et) S (O)2CH2CH2CFThree                   D1-93a
CH (Et) S (O)2CH2CH2CFThree                   D1-95a
CH (Et) S (O)2CH2CH2CFThree                   D1-96a
CH (Et) S (O)2CH2CH2CFThree                   D1-98a
CH (Et) S (O)2CH2CH2CFThree                   D1-108a
CH (Et) S (O)2CH2CH2CFThree                   D1-108b (Z = 2-Cl)
CH (Et) S (O)2CH2CH2CFThree                   D1-108b (Z = 3-Me)
CH (Et) S (O)2CH2CH2CFThree                   D1-108b (Z = 4-OMe)
CH (Et) S (O)2CH2CH2CFThree                   D1-108b (Z = 2-SMe)
CH (Et) S (O)2CH2CH2CFThree                   D1-108b (Z = 3-CFThree)
CH (Et) S (O)2CH2CH2CFThree                   D1-108b (Z = 4-OCFThree)
CH (Et) S (O)2CH2CH2CFThree                   D1-108b (Z = 2-SCFThree)
CH (Et) S (O)2CH2CH2CFThree                   C (O) Me
CH (Et) S (O)2CH2CH2CFThree                   C (O) CFThree
CH (Et) S (O)2CH2CH2CFThree                   C (O) OMe
CH2SCH2(D1-103a) Me
CH2SCH2(D1-103a) Et
CH2SCH2(D1-103a) Pr-n
CH2SCH2(D1-103a) Pr-i
CH2SCH2(D1-103a) Pr-c
CH2SCH2(D1-103a) Bu-n
CH2SCH2(D1-103a) Bu-i
CH2SCH2(D1-103a) Bu-c
CH2SCH2(D1-103a) Bu-s
CH2SCH2(D1-103a) Bu-t
CH2SCH2(D1-103a) Pen-n
CH2SCH2(D1-103a) Pen-c
CH2SCH2(D1-103a) Hex-n
CH2SCH2(D1-103a) Hex-c
CH2SCH2(D1-103a) CH2Pr-c
CH2SCH2(D1-103a) CH2Bu-c
CH2SCH2(D1-103a) CH2Pen-c
CH2SCH2(D1-103a) CH2Hex-c
CH2SCH2(D1-103a) CH2CH = CH2
CH2SCH2(D1-103a) CH2CH = C (Cl)2
CH2SCH2(D1-103a) CH2C≡CH
CH2SCH2(D1-103a) CH2CN
CH2SCH2(D1-103a) CH2CFThree
CH2SCH2(D1-103a) CH2OMe
CH2SCH2(D1-103a) CH2OCFThree
CH2SCH2(D1-103a) CH2SMe
CH2SCH2(D1-103a) CH2S (O) Me
CH2SCH2(D1-103a) CH2S (O)2Me
CH2SCH2(D1-103a) CH2SCFThree
CH2SCH2(D1-103a) CH2S (O) CFThree
CH2SCH2(D1-103a) CH2S (O)2CFThree
CH2SCH2(D1-103a) CH2CH (OMe)2
CH2SCH2(D1-103a) CH2CH (SMe)2
CH2SCH2(D1-103a) CH2C (O) Me
CH2SCH2(D1-103a) CH2C (O) CFThree
CH2SCH2(D1-103a) CH2C (O) OMe
CH2SCH2(D1-103a) CH2(D1-32a)
CH2SCH2(D1-103a) CH2(D1-33a)
CH2SCH2(D1-103a) CH2(D1-34a)
CH2SCH2(D1-103a) CH2(D1-37a)
CH2SCH2(D1-103a) CH2(D1-81a)
CH2SCH2(D1-103a) CH2(D1-82a)
CH2SCH2(D1-103a) CH2(D1-84a)
CH2SCH2(D1-103a) CH2(D1-85a)
CH2SCH2(D1-103a) CH2(D1-87a)
CH2SCH2(D1-103a) CH2(D1-92a)
CH2SCH2(D1-103a) CH2(D1-93a)
CH2SCH2(D1-103a) CH2(D1-95a)
CH2SCH2(D1-103a) CH2(D1-96a)
CH2SCH2(D1-103a) CH2(D1-98a)
CH2SCH2(D1-103a) CH2(D1-108a)
CH2SCH2(D1-103a) CH2(D1-108b, Z = 2-Cl)
CH2SCH2(D1-103a) CH2(D1-108b, Z = 3-Me)
CH2SCH2(D1-103a) CH2(D1-108b, Z = 4-OMe)
CH2SCH2(D1-103a) CH2(D1-108b, Z = 2-SMe)
CH2SCH2(D1-103a) CH2(D1-108b, Z = 3-CFThree)
CH2SCH2(D1-103a) CH2(D1-108b, Z = 4-OCFThree)
CH2SCH2(D1-103a) CH2(D1-108b, Z = 2-SCFThree)
CH2SCH2(D1-103a) CH2CH2CN
CH2SCH2(D1-103a) CH2CH2CFThree
CH2SCH2(D1-103a) CH2CH2OMe
CH2SCH2(D1-103a) CH2CH2SMe
CH2SCH2(D1-103a) CH2CH2S (O) Me
CH2SCH2(D1-103a) CH2CH2S (O)2Me
CH2SCH2(D1-103a) D1-32a
CH2SCH2(D1-103a) D1-33a
CH2SCH2(D1-103a) D1-34a
CH2SCH2(D1-103a) D1-37a
CH2SCH2(D1-103a) D1-81a
CH2SCH2(D1-103a) D1-82a
CH2SCH2(D1-103a) D1-84a
CH2SCH2(D1-103a) D1-85a
CH2SCH2(D1-103a) D1-87a
CH2SCH2(D1-103a) D1-92a
CH2SCH2(D1-103a) D1-93a
CH2SCH2(D1-103a) D1-95a
CH2SCH2(D1-103a) D1-96a
CH2SCH2(D1-103a) D1-98a
CH2SCH2(D1-103a) D1-108a
CH2SCH2(D1-103a) D1-108b (Z = 2-Cl)
CH2SCH2(D1-103a) D1-108b (Z = 3-Me)
CH2SCH2(D1-103a) D1-108b (Z = 4-OMe)
CH2SCH2(D1-103a) D1-108b (Z = 2-SMe)
CH2SCH2(D1-103a) D1-108b (Z = 3-CFThree)
CH2SCH2(D1-103a) D1-108b (Z = 4-OCFThree)
CH2SCH2(D1-103a) D1-108b (Z = 2-SCFThree)
CH2SCH2(D1-103a) C (O) Me
CH2SCH2(D1-103a) C (O) CFThree
CH2SCH2(D1-103a) C (O) OMe
CH2S (O) CH2(D1-103a) Me
CH2S (O) CH2(D1-103a) Et
CH2S (O) CH2(D1-103a) Pr-n
CH2S (O) CH2(D1-103a) Pr-i
CH2S (O) CH2(D1-103a) Pr-c
CH2S (O) CH2(D1-103a) Bu-n
CH2S (O) CH2(D1-103a) Bu-i
CH2S (O) CH2(D1-103a) Bu-c
CH2S (O) CH2(D1-103a) Bu-s
CH2S (O) CH2(D1-103a) Bu-t
CH2S (O) CH2(D1-103a) Pen-n
CH2S (O) CH2(D1-103a) Pen-c
CH2S (O) CH2(D1-103a) Hex-n
CH2S (O) CH2(D1-103a) Hex-c
CH2S (O) CH2(D1-103a) CH2Pr-c
CH2S (O) CH2(D1-103a) CH2Bu-c
CH2S (O) CH2(D1-103a) CH2Pen-c
CH2S (O) CH2(D1-103a) CH2Hex-c
CH2S (O) CH2(D1-103a) CH2CH = CH2
CH2S (O) CH2(D1-103a) CH2CH = C (Cl)2
CH2S (O) CH2(D1-103a) CH2C≡CH
CH2S (O) CH2(D1-103a) CH2CN
CH2S (O) CH2(D1-103a) CH2CFThree
CH2S (O) CH2(D1-103a) CH2OMe
CH2S (O) CH2(D1-103a) CH2OCFThree
CH2S (O) CH2(D1-103a) CH2SMe
CH2S (O) CH2(D1-103a) CH2S (O) Me
CH2S (O) CH2(D1-103a) CH2S (O)2Me
CH2S (O) CH2(D1-103a) CH2SCFThree
CH2S (O) CH2(D1-103a) CH2S (O) CFThree
CH2S (O) CH2(D1-103a) CH2S (O)2CFThree
CH2S (O) CH2(D1-103a) CH2CH (OMe)2
CH2S (O) CH2(D1-103a) CH2CH (SMe)2
CH2S (O) CH2(D1-103a) CH2C (O) Me
CH2S (O) CH2(D1-103a) CH2C (O) CFThree
CH2S (O) CH2(D1-103a) CH2C (O) OMe
CH2S (O) CH2(D1-103a) CH2(D1-32a)
CH2S (O) CH2(D1-103a) CH2(D1-33a)
CH2S (O) CH2(D1-103a) CH2(D1-34a)
CH2S (O) CH2(D1-103a) CH2(D1-37a)
CH2S (O) CH2(D1-103a) CH2(D1-81a)
CH2S (O) CH2(D1-103a) CH2(D1-82a)
CH2S (O) CH2(D1-103a) CH2(D1-84a)
CH2S (O) CH2(D1-103a) CH2(D1-85a)
CH2S (O) CH2(D1-103a) CH2(D1-87a)
CH2S (O) CH2(D1-103a) CH2(D1-92a)
CH2S (O) CH2(D1-103a) CH2(D1-93a)
CH2S (O) CH2(D1-103a) CH2(D1-95a)
CH2S (O) CH2(D1-103a) CH2(D1-96a)
CH2S (O) CH2(D1-103a) CH2(D1-98a)
CH2S (O) CH2(D1-103a) CH2(D1-108a)
CH2S (O) CH2(D1-103a) CH2(D1-108b, Z = 2-Cl)
CH2S (O) CH2(D1-103a) CH2(D1-108b, Z = 3-Me)
CH2S (O) CH2(D1-103a) CH2(D1-108b, Z = 4-OMe)
CH2S (O) CH2(D1-103a) CH2(D1-108b, Z = 2-SMe)
CH2S (O) CH2(D1-103a) CH2(D1-108b, Z = 3-CFThree)
CH2S (O) CH2(D1-103a) CH2(D1-108b, Z = 4-OCFThree)
CH2S (O) CH2(D1-103a) CH2(D1-108b, Z = 2-SCFThree)
CH2S (O) CH2(D1-103a) CH2CH2CN
CH2S (O) CH2(D1-103a) CH2CH2CFThree
CH2S (O) CH2(D1-103a) CH2CH2OMe
CH2S (O) CH2(D1-103a) CH2CH2SMe
CH2S (O) CH2(D1-103a) CH2CH2S (O) Me
CH2S (O) CH2(D1-103a) CH2CH2S (O)2Me
CH2S (O) CH2(D1-103a) D1-32a
CH2S (O) CH2(D1-103a) D1-33a
CH2S (O) CH2(D1-103a) D1-34a
CH2S (O) CH2(D1-103a) D1-37a
CH2S (O) CH2(D1-103a) D1-81a
CH2S (O) CH2(D1-103a) D1-82a
CH2S (O) CH2(D1-103a) D1-84a
CH2S (O) CH2(D1-103a) D1-85a
CH2S (O) CH2(D1-103a) D1-87a
CH2S (O) CH2(D1-103a) D1-92a
CH2S (O) CH2(D1-103a) D1-93a
CH2S (O) CH2(D1-103a) D1-95a
CH2S (O) CH2(D1-103a) D1-96a
CH2S (O) CH2(D1-103a) D1-98a
CH2S (O) CH2(D1-103a) D1-108a
CH2S (O) CH2(D1-103a) D1-108b (Z = 2-Cl)
CH2S (O) CH2(D1-103a) D1-108b (Z = 3-Me)
CH2S (O) CH2(D1-103a) D1-108b (Z = 4-OMe)
CH2S (O) CH2(D1-103a) D1-108b (Z = 2-SMe)
CH2S (O) CH2(D1-103a) D1-108b (Z = 3-CFThree)
CH2S (O) CH2(D1-103a) D1-108b (Z = 4-OCFThree)
CH2S (O) CH2(D1-103a) D1-108b (Z = 2-SCFThree)
CH2S (O) CH2(D1-103a) C (O) Me
CH2S (O) CH2(D1-103a) C (O) CFThree
CH2S (O) CH2(D1-103a) C (O) OMe
CH2S (O)2CH2(D1-103a) Me
CH2S (O)2CH2(D1-103a) Et
CH2S (O)2CH2(D1-103a) Pr-n
CH2S (O)2CH2(D1-103a) Pr-i
CH2S (O)2CH2(D1-103a) Pr-c
CH2S (O)2CH2(D1-103a) Bu-n
CH2S (O)2CH2(D1-103a) Bu-i
CH2S (O)2CH2(D1-103a) Bu-c
CH2S (O)2CH2(D1-103a) Bu-s
CH2S (O)2CH2(D1-103a) Bu-t
CH2S (O)2CH2(D1-103a) Pen-n
CH2S (O)2CH2(D1-103a) Pen-c
CH2S (O)2CH2(D1-103a) Hex-n
CH2S (O)2CH2(D1-103a) Hex-c
CH2S (O)2CH2(D1-103a) CH2Pr-c
CH2S (O)2CH2(D1-103a) CH2Bu-c
CH2S (O)2CH2(D1-103a) CH2Pen-c
CH2S (O)2CH2(D1-103a) CH2Hex-c
CH2S (O)2CH2(D1-103a) CH2CH = CH2
CH2S (O)2CH2(D1-103a) CH2CH = C (Cl)2
CH2S (O)2CH2(D1-103a) CH2C≡CH
CH2S (O)2CH2(D1-103a) CH2CN
CH2S (O)2CH2(D1-103a) CH2CFThree
CH2S (O)2CH2(D1-103a) CH2OMe
CH2S (O)2CH2(D1-103a) CH2OCFThree
CH2S (O)2CH2(D1-103a) CH2SMe
CH2S (O)2CH2(D1-103a) CH2S (O) Me
CH2S (O)2CH2(D1-103a) CH2S (O)2Me
CH2S (O)2CH2(D1-103a) CH2SCFThree
CH2S (O)2CH2(D1-103a) CH2S (O) CFThree
CH2S (O)2CH2(D1-103a) CH2S (O)2CFThree
CH2S (O)2CH2(D1-103a) CH2CH (OMe)2
CH2S (O)2CH2(D1-103a) CH2CH (SMe)2
CH2S (O)2CH2(D1-103a) CH2C (O) Me
CH2S (O)2CH2(D1-103a) CH2C (O) CFThree
CH2S (O)2CH2(D1-103a) CH2C (O) OMe
CH2S (O)2CH2(D1-103a) CH2(D1-32a)
CH2S (O)2CH2(D1-103a) CH2(D1-33a)
CH2S (O)2CH2(D1-103a) CH2(D1-34a)
CH2S (O)2CH2(D1-103a) CH2(D1-37a)
CH2S (O)2CH2(D1-103a) CH2(D1-81a)
CH2S (O)2CH2(D1-103a) CH2(D1-82a)
CH2S (O)2CH2(D1-103a) CH2(D1-84a)
CH2S (O)2CH2(D1-103a) CH2(D1-85a)
CH2S (O)2CH2(D1-103a) CH2(D1-87a)
CH2S (O)2CH2(D1-103a) CH2(D1-92a)
CH2S (O)2CH2(D1-103a) CH2(D1-93a)
CH2S (O)2CH2(D1-103a) CH2(D1-95a)
CH2S (O)2CH2(D1-103a) CH2(D1-96a)
CH2S (O)2CH2(D1-103a) CH2(D1-98a)
CH2S (O)2CH2(D1-103a) CH2(D1-108a)
CH2S (O)2CH2(D1-103a) CH2(D1-108b, Z = 2-Cl)
CH2S (O)2CH2(D1-103a) CH2(D1-108b, Z = 3-Me)
CH2S (O)2CH2(D1-103a) CH2(D1-108b, Z = 4-OMe)
CH2S (O)2CH2(D1-103a) CH2(D1-108b, Z = 2-SMe)
CH2S (O)2CH2(D1-103a) CH2(D1-108b, Z = 3-CFThree)
CH2S (O)2CH2(D1-103a) CH2(D1-108b, Z = 4-OCFThree)
CH2S (O)2CH2(D1-103a) CH2(D1-108b, Z = 2-SCFThree)
CH2S (O)2CH2(D1-103a) CH2CH2CN
CH2S (O)2CH2(D1-103a) CH2CH2CFThree
CH2S (O)2CH2(D1-103a) CH2CH2OMe
CH2S (O)2CH2(D1-103a) CH2CH2SMe
CH2S (O)2CH2(D1-103a) CH2CH2S (O) Me
CH2S (O)2CH2(D1-103a) CH2CH2S (O)2Me
CH2S (O)2CH2(D1-103a) D1-32a
CH2S (O)2CH2(D1-103a) D1-33a
CH2S (O)2CH2(D1-103a) D1-34a
CH2S (O)2CH2(D1-103a) D1-37a
CH2S (O)2CH2(D1-103a) D1-81a
CH2S (O)2CH2(D1-103a) D1-82a
CH2S (O)2CH2(D1-103a) D1-84a
CH2S (O)2CH2(D1-103a) D1-85a
CH2S (O)2CH2(D1-103a) D1-87a
CH2S (O)2CH2(D1-103a) D1-92a
CH2S (O)2CH2(D1-103a) D1-93a
CH2S (O)2CH2(D1-103a) D1-95a
CH2S (O)2CH2(D1-103a) D1-96a
CH2S (O)2CH2(D1-103a) D1-98a
CH2S (O)2CH2(D1-103a) D1-108a
CH2S (O)2CH2(D1-103a) D1-108b (Z = 2-Cl)
CH2S (O)2CH2(D1-103a) D1-108b (Z = 3-Me)
CH2S (O)2CH2(D1-103a) D1-108b (Z = 4-OMe)
CH2S (O)2CH2(D1-103a) D1-108b (Z = 2-SMe)
CH2S (O)2CH2(D1-103a) D1-108b (Z = 3-CFThree)
CH2S (O)2CH2(D1-103a) D1-108b (Z = 4-OCFThree)
CH2S (O)2CH2(D1-103a) D1-108b (Z = 2-SCFThree)
CH2S (O)2CH2(D1-103a) C (O) Me
CH2S (O)2CH2(D1-103a) C (O) CFThree
CH2S (O)2CH2(D1-103a) C (O) OMe
CH (Me) SCH2(D1-103a) Me
CH (Me) SCH2(D1-103a) Et
CH (Me) SCH2(D1-103a) Pr-n
CH (Me) SCH2(D1-103a) Pr-i
CH (Me) SCH2(D1-103a) Pr-c
CH (Me) SCH2(D1-103a) Bu-n
CH (Me) SCH2(D1-103a) Bu-i
CH (Me) SCH2(D1-103a) Bu-c
CH (Me) SCH2(D1-103a) Bu-s
CH (Me) SCH2(D1-103a) Bu-t
CH (Me) SCH2(D1-103a) Pen-n
CH (Me) SCH2(D1-103a) Pen-c
CH (Me) SCH2(D1-103a) Hex-n
CH (Me) SCH2(D1-103a) Hex-c
CH (Me) SCH2(D1-103a) CH2Pr-c
CH (Me) SCH2(D1-103a) CH2Bu-c
CH (Me) SCH2(D1-103a) CH2Pen-c
CH (Me) SCH2(D1-103a) CH2Hex-c
CH (Me) SCH2(D1-103a) CH2CH = CH2
CH (Me) SCH2(D1-103a) CH2CH = C (Cl)2
CH (Me) SCH2(D1-103a) CH2C≡CH
CH (Me) SCH2(D1-103a) CH2CN
CH (Me) SCH2(D1-103a) CH2CFThree
CH (Me) SCH2(D1-103a) CH2OMe
CH (Me) SCH2(D1-103a) CH2OCFThree
CH (Me) SCH2(D1-103a) CH2SMe
CH (Me) SCH2(D1-103a) CH2S (O) Me
CH (Me) SCH2(D1-103a) CH2S (O)2Me
CH (Me) SCH2(D1-103a) CH2SCFThree
CH (Me) SCH2(D1-103a) CH2S (O) CFThree
CH (Me) SCH2(D1-103a) CH2S (O)2CFThree
CH (Me) SCH2(D1-103a) CH2CH (OMe)2
CH (Me) SCH2(D1-103a) CH2CH (SMe)2
CH (Me) SCH2(D1-103a) CH2C (O) Me
CH (Me) SCH2(D1-103a) CH2C (O) CFThree
CH (Me) SCH2(D1-103a) CH2C (O) OMe
CH (Me) SCH2(D1-103a) CH2(D1-32a)
CH (Me) SCH2(D1-103a) CH2(D1-33a)
CH (Me) SCH2(D1-103a) CH2(D1-34a)
CH (Me) SCH2(D1-103a) CH2(D1-37a)
CH (Me) SCH2(D1-103a) CH2(D1-81a)
CH (Me) SCH2(D1-103a) CH2(D1-82a)
CH (Me) SCH2(D1-103a) CH2(D1-84a)
CH (Me) SCH2(D1-103a) CH2(D1-85a)
CH (Me) SCH2(D1-103a) CH2(D1-87a)
CH (Me) SCH2(D1-103a) CH2(D1-92a)
CH (Me) SCH2(D1-103a) CH2(D1-93a)
CH (Me) SCH2(D1-103a) CH2(D1-95a)
CH (Me) SCH2(D1-103a) CH2(D1-96a)
CH (Me) SCH2(D1-103a) CH2(D1-98a)
CH (Me) SCH2(D1-103a) CH2(D1-108a)
CH (Me) SCH2(D1-103a) CH2(D1-108b, Z = 2-Cl)
CH (Me) SCH2(D1-103a) CH2(D1-108b, Z = 3-Me)
CH (Me) SCH2(D1-103a) CH2(D1-108b, Z = 4-OMe)
CH (Me) SCH2(D1-103a) CH2(D1-108b, Z = 2-SMe)
CH (Me) SCH2(D1-103a) CH2(D1-108b, Z = 3-CFThree)
CH (Me) SCH2(D1-103a) CH2(D1-108b, Z = 4-OCFThree)
CH (Me) SCH2(D1-103a) CH2(D1-108b, Z = 2-SCFThree)
CH (Me) SCH2(D1-103a) CH2CH2CN
CH (Me) SCH2(D1-103a) CH2CH2CFThree
CH (Me) SCH2(D1-103a) CH2CH2OMe
CH (Me) SCH2(D1-103a) CH2CH2SMe
CH (Me) SCH2(D1-103a) CH2CH2S (O) Me
CH (Me) SCH2(D1-103a) CH2CH2S (O)2Me
CH (Me) SCH2(D1-103a) D1-32a
CH (Me) SCH2(D1-103a) D1-33a
CH (Me) SCH2(D1-103a) D1-34a
CH (Me) SCH2(D1-103a) D1-37a
CH (Me) SCH2(D1-103a) D1-81a
CH (Me) SCH2(D1-103a) D1-82a
CH (Me) SCH2(D1-103a) D1-84a
CH (Me) SCH2(D1-103a) D1-85a
CH (Me) SCH2(D1-103a) D1-87a
CH (Me) SCH2(D1-103a) D1-92a
CH (Me) SCH2(D1-103a) D1-93a
CH (Me) SCH2(D1-103a) D1-95a
CH (Me) SCH2(D1-103a) D1-96a
CH (Me) SCH2(D1-103a) D1-98a
CH (Me) SCH2(D1-103a) D1-108a
CH (Me) SCH2(D1-103a) D1-108b (Z = 2-Cl)
CH (Me) SCH2(D1-103a) D1-108b (Z = 3-Me)
CH (Me) SCH2(D1-103a) D1-108b (Z = 4-OMe)
CH (Me) SCH2(D1-103a) D1-108b (Z = 2-SMe)
CH (Me) SCH2(D1-103a) D1-108b (Z = 3-CFThree)
CH (Me) SCH2(D1-103a) D1-108b (Z = 4-OCFThree)
CH (Me) SCH2(D1-103a) D1-108b (Z = 2-SCFThree)
CH (Me) SCH2(D1-103a) C (O) Me
CH (Me) SCH2(D1-103a) C (O) CFThree
CH (Me) SCH2(D1-103a) C (O) OMe
CH (Me) S (O) CH2(D1-103a) Me
CH (Me) S (O) CH2(D1-103a) Et
CH (Me) S (O) CH2(D1-103a) Pr-n
CH (Me) S (O) CH2(D1-103a) Pr-i
CH (Me) S (O) CH2(D1-103a) Pr-c
CH (Me) S (O) CH2(D1-103a) Bu-n
CH (Me) S (O) CH2(D1-103a) Bu-i
CH (Me) S (O) CH2(D1-103a) Bu-c
CH (Me) S (O) CH2(D1-103a) Bu-s
CH (Me) S (O) CH2(D1-103a) Bu-t
CH (Me) S (O) CH2(D1-103a) Pen-n
CH (Me) S (O) CH2(D1-103a) Pen-c
CH (Me) S (O) CH2(D1-103a) Hex-n
CH (Me) S (O) CH2(D1-103a) Hex-c
CH (Me) S (O) CH2(D1-103a) CH2Pr-c
CH (Me) S (O) CH2(D1-103a) CH2Bu-c
CH (Me) S (O) CH2(D1-103a) CH2Pen-c
CH (Me) S (O) CH2(D1-103a) CH2Hex-c
CH (Me) S (O) CH2(D1-103a) CH2CH = CH2
CH (Me) S (O) CH2(D1-103a) CH2CH = C (Cl)2
CH (Me) S (O) CH2(D1-103a) CH2C≡CH
CH (Me) S (O) CH2(D1-103a) CH2CN
CH (Me) S (O) CH2(D1-103a) CH2CFThree
CH (Me) S (O) CH2(D1-103a) CH2OMe
CH (Me) S (O) CH2(D1-103a) CH2OCFThree
CH (Me) S (O) CH2(D1-103a) CH2SMe
CH (Me) S (O) CH2(D1-103a) CH2S (O) Me
CH (Me) S (O) CH2(D1-103a) CH2S (O)2Me
CH (Me) S (O) CH2(D1-103a) CH2SCFThree
CH (Me) S (O) CH2(D1-103a) CH2S (O) CFThree
CH (Me) S (O) CH2(D1-103a) CH2S (O)2CFThree
CH (Me) S (O) CH2(D1-103a) CH2CH (OMe)2
CH (Me) S (O) CH2(D1-103a) CH2CH (SMe)2
CH (Me) S (O) CH2(D1-103a) CH2C (O) Me
CH (Me) S (O) CH2(D1-103a) CH2C (O) CFThree
CH (Me) S (O) CH2(D1-103a) CH2C (O) OMe
CH (Me) S (O) CH2(D1-103a) CH2(D1-32a)
CH (Me) S (O) CH2(D1-103a) CH2(D1-33a)
CH (Me) S (O) CH2(D1-103a) CH2(D1-34a)
CH (Me) S (O) CH2(D1-103a) CH2(D1-37a)
CH (Me) S (O) CH2(D1-103a) CH2(D1-81a)
CH (Me) S (O) CH2(D1-103a) CH2(D1-82a)
CH (Me) S (O) CH2(D1-103a) CH2(D1-84a)
CH (Me) S (O) CH2(D1-103a) CH2(D1-85a)
CH (Me) S (O) CH2(D1-103a) CH2(D1-87a)
CH (Me) S (O) CH2(D1-103a) CH2(D1-92a)
CH (Me) S (O) CH2(D1-103a) CH2(D1-93a)
CH (Me) S (O) CH2(D1-103a) CH2(D1-95a)
CH (Me) S (O) CH2(D1-103a) CH2(D1-96a)
CH (Me) S (O) CH2(D1-103a) CH2(D1-98a)
CH (Me) S (O) CH2(D1-103a) CH2(D1-108a)
CH (Me) S (O) CH2(D1-103a) CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O) CH2(D1-103a) CH2(D1-108b, Z = 3-Me)
CH (Me) S (O) CH2(D1-103a) CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O) CH2(D1-103a) CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O) CH2(D1-103a) CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O) CH2(D1-103a) CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O) CH2(D1-103a) CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O) CH2(D1-103a) CH2CH2CN
CH (Me) S (O) CH2(D1-103a) CH2CH2CFThree
CH (Me) S (O) CH2(D1-103a) CH2CH2OMe
CH (Me) S (O) CH2(D1-103a) CH2CH2SMe
CH (Me) S (O) CH2(D1-103a) CH2CH2S (O) Me
CH (Me) S (O) CH2(D1-103a) CH2CH2S (O)2Me
CH (Me) S (O) CH2(D1-103a) D1-32a
CH (Me) S (O) CH2(D1-103a) D1-33a
CH (Me) S (O) CH2(D1-103a) D1-34a
CH (Me) S (O) CH2(D1-103a) D1-37a
CH (Me) S (O) CH2(D1-103a) D1-81a
CH (Me) S (O) CH2(D1-103a) D1-82a
CH (Me) S (O) CH2(D1-103a) D1-84a
CH (Me) S (O) CH2(D1-103a) D1-85a
CH (Me) S (O) CH2(D1-103a) D1-87a
CH (Me) S (O) CH2(D1-103a) D1-92a
CH (Me) S (O) CH2(D1-103a) D1-93a
CH (Me) S (O) CH2(D1-103a) D1-95a
CH (Me) S (O) CH2(D1-103a) D1-96a
CH (Me) S (O) CH2(D1-103a) D1-98a
CH (Me) S (O) CH2(D1-103a) D1-108a
CH (Me) S (O) CH2(D1-103a) D1-108b (Z = 2-Cl)
CH (Me) S (O) CH2(D1-103a) D1-108b (Z = 3-Me)
CH (Me) S (O) CH2(D1-103a) D1-108b (Z = 4-OMe)
CH (Me) S (O) CH2(D1-103a) D1-108b (Z = 2-SMe)
CH (Me) S (O) CH2(D1-103a) D1-108b (Z = 3-CFThree)
CH (Me) S (O) CH2(D1-103a) D1-108b (Z = 4-OCFThree)
CH (Me) S (O) CH2(D1-103a) D1-108b (Z = 2-SCFThree)
CH (Me) S (O) CH2(D1-103a) C (O) Me
CH (Me) S (O) CH2(D1-103a) C (O) CFThree
CH (Me) S (O) CH2(D1-103a) C (O) OMe
CH (Me) S (O)2CH2(D1-103a) Me
CH (Me) S (O)2CH2(D1-103a) Et
CH (Me) S (O)2CH2(D1-103a) Pr-n
CH (Me) S (O)2CH2(D1-103a) Pr-i
CH (Me) S (O)2CH2(D1-103a) Pr-c
CH (Me) S (O)2CH2(D1-103a) Bu-n
CH (Me) S (O)2CH2(D1-103a) Bu-i
CH (Me) S (O)2CH2(D1-103a) Bu-c
CH (Me) S (O)2CH2(D1-103a) Bu-s
CH (Me) S (O)2CH2(D1-103a) Bu-t
CH (Me) S (O)2CH2(D1-103a) Pen-n
CH (Me) S (O)2CH2(D1-103a) Pen-c
CH (Me) S (O)2CH2(D1-103a) Hex-n
CH (Me) S (O)2CH2(D1-103a) Hex-c
CH (Me) S (O)2CH2(D1-103a) CH2Pr-c
CH (Me) S (O)2CH2(D1-103a) CH2Bu-c
CH (Me) S (O)2CH2(D1-103a) CH2Pen-c
CH (Me) S (O)2CH2(D1-103a) CH2Hex-c
CH (Me) S (O)2CH2(D1-103a) CH2CH = CH2
CH (Me) S (O)2CH2(D1-103a) CH2CH = C (Cl)2
CH (Me) S (O)2CH2(D1-103a) CH2C≡CH
CH (Me) S (O)2CH2(D1-103a) CH2CN
CH (Me) S (O)2CH2(D1-103a) CH2CFThree
CH (Me) S (O)2CH2(D1-103a) CH2OMe
CH (Me) S (O)2CH2(D1-103a) CH2OCFThree
CH (Me) S (O)2CH2(D1-103a) CH2SMe
CH (Me) S (O)2CH2(D1-103a) CH2S (O) Me
CH (Me) S (O)2CH2(D1-103a) CH2S (O)2Me
CH (Me) S (O)2CH2(D1-103a) CH2SCFThree
CH (Me) S (O)2CH2(D1-103a) CH2S (O) CFThree
CH (Me) S (O)2CH2(D1-103a) CH2S (O)2CFThree
CH (Me) S (O)2CH2(D1-103a) CH2CH (OMe)2
CH (Me) S (O)2CH2(D1-103a) CH2CH (SMe)2
CH (Me) S (O)2CH2(D1-103a) CH2C (O) Me
CH (Me) S (O)2CH2(D1-103a) CH2C (O) CFThree
CH (Me) S (O)2CH2(D1-103a) CH2C (O) OMe
CH (Me) S (O)2CH2(D1-103a) CH2(D1-32a)
CH (Me) S (O)2CH2(D1-103a) CH2(D1-33a)
CH (Me) S (O)2CH2(D1-103a) CH2(D1-34a)
CH (Me) S (O)2CH2(D1-103a) CH2(D1-37a)
CH (Me) S (O)2CH2(D1-103a) CH2(D1-81a)
CH (Me) S (O)2CH2(D1-103a) CH2(D1-82a)
CH (Me) S (O)2CH2(D1-103a) CH2(D1-84a)
CH (Me) S (O)2CH2(D1-103a) CH2(D1-85a)
CH (Me) S (O)2CH2(D1-103a) CH2(D1-87a)
CH (Me) S (O)2CH2(D1-103a) CH2(D1-92a)
CH (Me) S (O)2CH2(D1-103a) CH2(D1-93a)
CH (Me) S (O)2CH2(D1-103a) CH2(D1-95a)
CH (Me) S (O)2CH2(D1-103a) CH2(D1-96a)
CH (Me) S (O)2CH2(D1-103a) CH2(D1-98a)
CH (Me) S (O)2CH2(D1-103a) CH2(D1-108a)
CH (Me) S (O)2CH2(D1-103a) CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O)2CH2(D1-103a) CH2(D1-108b, Z = 3-Me)
CH (Me) S (O)2CH2(D1-103a) CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O)2CH2(D1-103a) CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O)2CH2(D1-103a) CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O)2CH2(D1-103a) CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O)2CH2(D1-103a) CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O)2CH2(D1-103a) CH2CH2CN
CH (Me) S (O)2CH2(D1-103a) CH2CH2CFThree
CH (Me) S (O)2CH2(D1-103a) CH2CH2OMe
CH (Me) S (O)2CH2(D1-103a) CH2CH2SMe
CH (Me) S (O)2CH2(D1-103a) CH2CH2S (O) Me
CH (Me) S (O)2CH2(D1-103a) CH2CH2S (O)2Me
CH (Me) S (O)2CH2(D1-103a) D1-32a
CH (Me) S (O)2CH2(D1-103a) D1-33a
CH (Me) S (O)2CH2(D1-103a) D1-34a
CH (Me) S (O)2CH2(D1-103a) D1-37a
CH (Me) S (O)2CH2(D1-103a) D1-81a
CH (Me) S (O)2CH2(D1-103a) D1-82a
CH (Me) S (O)2CH2(D1-103a) D1-84a
CH (Me) S (O)2CH2(D1-103a) D1-85a
CH (Me) S (O)2CH2(D1-103a) D1-87a
CH (Me) S (O)2CH2(D1-103a) D1-92a
CH (Me) S (O)2CH2(D1-103a) D1-93a
CH (Me) S (O)2CH2(D1-103a) D1-95a
CH (Me) S (O)2CH2(D1-103a) D1-96a
CH (Me) S (O)2CH2(D1-103a) D1-98a
CH (Me) S (O)2CH2(D1-103a) D1-108a
CH (Me) S (O)2CH2(D1-103a) D1-108b (Z = 2-Cl)
CH (Me) S (O)2CH2(D1-103a) D1-108b (Z = 3-Me)
CH (Me) S (O)2CH2(D1-103a) D1-108b (Z = 4-OMe)
CH (Me) S (O)2CH2(D1-103a) D1-108b (Z = 2-SMe)
CH (Me) S (O)2CH2(D1-103a) D1-108b (Z = 3-CFThree)
CH (Me) S (O)2CH2(D1-103a) D1-108b (Z = 4-OCFThree)
CH (Me) S (O)2CH2(D1-103a) D1-108b (Z = 2-SCFThree)
CH (Me) S (O)2CH2(D1-103a) C (O) Me
CH (Me) S (O)2CH2(D1-103a) C (O) CFThree
CH (Me) S (O)2CH2(D1-103a) C (O) OMe
CH (Et) SCH2(D1-103a) Me
CH (Et) SCH2(D1-103a) Et
CH (Et) SCH2(D1-103a) Pr-n
CH (Et) SCH2(D1-103a) Pr-i
CH (Et) SCH2(D1-103a) Pr-c
CH (Et) SCH2(D1-103a) Bu-n
CH (Et) SCH2(D1-103a) Bu-i
CH (Et) SCH2(D1-103a) Bu-c
CH (Et) SCH2(D1-103a) Bu-s
CH (Et) SCH2(D1-103a) Bu-t
CH (Et) SCH2(D1-103a) Pen-n
CH (Et) SCH2(D1-103a) Pen-c
CH (Et) SCH2(D1-103a) Hex-n
CH (Et) SCH2(D1-103a) Hex-c
CH (Et) SCH2(D1-103a) CH2Pr-c
CH (Et) SCH2(D1-103a) CH2Bu-c
CH (Et) SCH2(D1-103a) CH2Pen-c
CH (Et) SCH2(D1-103a) CH2Hex-c
CH (Et) SCH2(D1-103a) CH2CH = CH2
CH (Et) SCH2(D1-103a) CH2CH = C (Cl)2
CH (Et) SCH2(D1-103a) CH2C≡CH
CH (Et) SCH2(D1-103a) CH2CN
CH (Et) SCH2(D1-103a) CH2CFThree
CH (Et) SCH2(D1-103a) CH2OMe
CH (Et) SCH2(D1-103a) CH2OCFThree
CH (Et) SCH2(D1-103a) CH2SMe
CH (Et) SCH2(D1-103a) CH2S (O) Me
CH (Et) SCH2(D1-103a) CH2S (O)2Me
CH (Et) SCH2(D1-103a) CH2SCFThree
CH (Et) SCH2(D1-103a) CH2S (O) CFThree
CH (Et) SCH2(D1-103a) CH2S (O)2CFThree
CH (Et) SCH2(D1-103a) CH2CH (OMe)2
CH (Et) SCH2(D1-103a) CH2CH (SMe)2
CH (Et) SCH2(D1-103a) CH2C (O) Me
CH (Et) SCH2(D1-103a) CH2C (O) CFThree
CH (Et) SCH2(D1-103a) CH2C (O) OMe
CH (Et) SCH2(D1-103a) CH2(D1-32a)
CH (Et) SCH2(D1-103a) CH2(D1-33a)
CH (Et) SCH2(D1-103a) CH2(D1-34a)
CH (Et) SCH2(D1-103a) CH2(D1-37a)
CH (Et) SCH2(D1-103a) CH2(D1-81a)
CH (Et) SCH2(D1-103a) CH2(D1-82a)
CH (Et) SCH2(D1-103a) CH2(D1-84a)
CH (Et) SCH2(D1-103a) CH2(D1-85a)
CH (Et) SCH2(D1-103a) CH2(D1-87a)
CH (Et) SCH2(D1-103a) CH2(D1-92a)
CH (Et) SCH2(D1-103a) CH2(D1-93a)
CH (Et) SCH2(D1-103a) CH2(D1-95a)
CH (Et) SCH2(D1-103a) CH2(D1-96a)
CH (Et) SCH2(D1-103a) CH2(D1-98a)
CH (Et) SCH2(D1-103a) CH2(D1-108a)
CH (Et) SCH2(D1-103a) CH2(D1-108b, Z = 2-Cl)
CH (Et) SCH2(D1-103a) CH2(D1-108b, Z = 3-Me)
CH (Et) SCH2(D1-103a) CH2(D1-108b, Z = 4-OMe)
CH (Et) SCH2(D1-103a) CH2(D1-108b, Z = 2-SMe)
CH (Et) SCH2(D1-103a) CH2(D1-108b, Z = 3-CFThree)
CH (Et) SCH2(D1-103a) CH2(D1-108b, Z = 4-OCFThree)
CH (Et) SCH2(D1-103a) CH2(D1-108b, Z = 2-SCFThree)
CH (Et) SCH2(D1-103a) CH2CH2CN
CH (Et) SCH2(D1-103a) CH2CH2CFThree
CH (Et) SCH2(D1-103a) CH2CH2OMe
CH (Et) SCH2(D1-103a) CH2CH2SMe
CH (Et) SCH2(D1-103a) CH2CH2S (O) Me
CH (Et) SCH2(D1-103a) CH2CH2S (O)2Me
CH (Et) SCH2(D1-103a) D1-32a
CH (Et) SCH2(D1-103a) D1-33a
CH (Et) SCH2(D1-103a) D1-34a
CH (Et) SCH2(D1-103a) D1-37a
CH (Et) SCH2(D1-103a) D1-81a
CH (Et) SCH2(D1-103a) D1-82a
CH (Et) SCH2(D1-103a) D1-84a
CH (Et) SCH2(D1-103a) D1-85a
CH (Et) SCH2(D1-103a) D1-87a
CH (Et) SCH2(D1-103a) D1-92a
CH (Et) SCH2(D1-103a) D1-93a
CH (Et) SCH2(D1-103a) D1-95a
CH (Et) SCH2(D1-103a) D1-96a
CH (Et) SCH2(D1-103a) D1-98a
CH (Et) SCH2(D1-103a) D1-108a
CH (Et) SCH2(D1-103a) D1-108b (Z = 2-Cl)
CH (Et) SCH2(D1-103a) D1-108b (Z = 3-Me)
CH (Et) SCH2(D1-103a) D1-108b (Z = 4-OMe)
CH (Et) SCH2(D1-103a) D1-108b (Z = 2-SMe)
CH (Et) SCH2(D1-103a) D1-108b (Z = 3-CFThree)
CH (Et) SCH2(D1-103a) D1-108b (Z = 4-OCFThree)
CH (Et) SCH2(D1-103a) D1-108b (Z = 2-SCFThree)
CH (Et) SCH2(D1-103a) C (O) Me
CH (Et) SCH2(D1-103a) C (O) CFThree
CH (Et) SCH2(D1-103a) C (O) OMe
CH (Et) S (O) CH2(D1-103a) Me
CH (Et) S (O) CH2(D1-103a) Et
CH (Et) S (O) CH2(D1-103a) Pr-n
CH (Et) S (O) CH2(D1-103a) Pr-i
CH (Et) S (O) CH2(D1-103a) Pr-c
CH (Et) S (O) CH2(D1-103a) Bu-n
CH (Et) S (O) CH2(D1-103a) Bu-i
CH (Et) S (O) CH2(D1-103a) Bu-c
CH (Et) S (O) CH2(D1-103a) Bu-s
CH (Et) S (O) CH2(D1-103a) Bu-t
CH (Et) S (O) CH2(D1-103a) Pen-n
CH (Et) S (O) CH2(D1-103a) Pen-c
CH (Et) S (O) CH2(D1-103a) Hex-n
CH (Et) S (O) CH2(D1-103a) Hex-c
CH (Et) S (O) CH2(D1-103a) CH2Pr-c
CH (Et) S (O) CH2(D1-103a) CH2Bu-c
CH (Et) S (O) CH2(D1-103a) CH2Pen-c
CH (Et) S (O) CH2(D1-103a) CH2Hex-c
CH (Et) S (O) CH2(D1-103a) CH2CH = CH2
CH (Et) S (O) CH2(D1-103a) CH2CH = C (Cl)2
CH (Et) S (O) CH2(D1-103a) CH2C≡CH
CH (Et) S (O) CH2(D1-103a) CH2CN
CH (Et) S (O) CH2(D1-103a) CH2CFThree
CH (Et) S (O) CH2(D1-103a) CH2OMe
CH (Et) S (O) CH2(D1-103a) CH2OCFThree
CH (Et) S (O) CH2(D1-103a) CH2SMe
CH (Et) S (O) CH2(D1-103a) CH2S (O) Me
CH (Et) S (O) CH2(D1-103a) CH2S (O)2Me
CH (Et) S (O) CH2(D1-103a) CH2SCFThree
CH (Et) S (O) CH2(D1-103a) CH2S (O) CFThree
CH (Et) S (O) CH2(D1-103a) CH2S (O)2CFThree
CH (Et) S (O) CH2(D1-103a) CH2CH (OMe)2
CH (Et) S (O) CH2(D1-103a) CH2CH (SMe)2
CH (Et) S (O) CH2(D1-103a) CH2C (O) Me
CH (Et) S (O) CH2(D1-103a) CH2C (O) CFThree
CH (Et) S (O) CH2(D1-103a) CH2C (O) OMe
CH (Et) S (O) CH2(D1-103a) CH2(D1-32a)
CH (Et) S (O) CH2(D1-103a) CH2(D1-33a)
CH (Et) S (O) CH2(D1-103a) CH2(D1-34a)
CH (Et) S (O) CH2(D1-103a) CH2(D1-37a)
CH (Et) S (O) CH2(D1-103a) CH2(D1-81a)
CH (Et) S (O) CH2(D1-103a) CH2(D1-82a)
CH (Et) S (O) CH2(D1-103a) CH2(D1-84a)
CH (Et) S (O) CH2(D1-103a) CH2(D1-85a)
CH (Et) S (O) CH2(D1-103a) CH2(D1-87a)
CH (Et) S (O) CH2(D1-103a) CH2(D1-92a)
CH (Et) S (O) CH2(D1-103a) CH2(D1-93a)
CH (Et) S (O) CH2(D1-103a) CH2(D1-95a)
CH (Et) S (O) CH2(D1-103a) CH2(D1-96a)
CH (Et) S (O) CH2(D1-103a) CH2(D1-98a)
CH (Et) S (O) CH2(D1-103a) CH2(D1-108a)
CH (Et) S (O) CH2(D1-103a) CH2(D1-108b, Z = 2-Cl)
CH (Et) S (O) CH2(D1-103a) CH2(D1-108b, Z = 3-Me)
CH (Et) S (O) CH2(D1-103a) CH2(D1-108b, Z = 4-OMe)
CH (Et) S (O) CH2(D1-103a) CH2(D1-108b, Z = 2-SMe)
CH (Et) S (O) CH2(D1-103a) CH2(D1-108b, Z = 3-CFThree)
CH (Et) S (O) CH2(D1-103a) CH2(D1-108b, Z = 4-OCFThree)
CH (Et) S (O) CH2(D1-103a) CH2(D1-108b, Z = 2-SCFThree)
CH (Et) S (O) CH2(D1-103a) CH2CH2CN
CH (Et) S (O) CH2(D1-103a) CH2CH2CFThree
CH (Et) S (O) CH2(D1-103a) CH2CH2OMe
CH (Et) S (O) CH2(D1-103a) CH2CH2SMe
CH (Et) S (O) CH2(D1-103a) CH2CH2S (O) Me
CH (Et) S (O) CH2(D1-103a) CH2CH2S (O)2Me
CH (Et) S (O) CH2(D1-103a) D1-32a
CH (Et) S (O) CH2(D1-103a) D1-33a
CH (Et) S (O) CH2(D1-103a) D1-34a
CH (Et) S (O) CH2(D1-103a) D1-37a
CH (Et) S (O) CH2(D1-103a) D1-81a
CH (Et) S (O) CH2(D1-103a) D1-82a
CH (Et) S (O) CH2(D1-103a) D1-84a
CH (Et) S (O) CH2(D1-103a) D1-85a
CH (Et) S (O) CH2(D1-103a) D1-87a
CH (Et) S (O) CH2(D1-103a) D1-92a
CH (Et) S (O) CH2(D1-103a) D1-93a
CH (Et) S (O) CH2(D1-103a) D1-95a
CH (Et) S (O) CH2(D1-103a) D1-96a
CH (Et) S (O) CH2(D1-103a) D1-98a
CH (Et) S (O) CH2(D1-103a) D1-108a
CH (Et) S (O) CH2(D1-103a) D1-108b (Z = 2-Cl)
CH (Et) S (O) CH2(D1-103a) D1-108b (Z = 3-Me)
CH (Et) S (O) CH2(D1-103a) D1-108b (Z = 4-OMe)
CH (Et) S (O) CH2(D1-103a) D1-108b (Z = 2-SMe)
CH (Et) S (O) CH2(D1-103a) D1-108b (Z = 3-CFThree)
CH (Et) S (O) CH2(D1-103a) D1-108b (Z = 4-OCFThree)
CH (Et) S (O) CH2(D1-103a) D1-108b (Z = 2-SCFThree)
CH (Et) S (O) CH2(D1-103a) C (O) Me
CH (Et) S (O) CH2(D1-103a) C (O) CFThree
CH (Et) S (O) CH2(D1-103a) C (O) OMe
CH (Et) S (O)2CH2(D1-103a) Me
CH (Et) S (O)2CH2(D1-103a) Et
CH (Et) S (O)2CH2(D1-103a) Pr-n
CH (Et) S (O)2CH2(D1-103a) Pr-i
CH (Et) S (O)2CH2(D1-103a) Pr-c
CH (Et) S (O)2CH2(D1-103a) Bu-n
CH (Et) S (O)2CH2(D1-103a) Bu-i
CH (Et) S (O)2CH2(D1-103a) Bu-c
CH (Et) S (O)2CH2(D1-103a) Bu-s
CH (Et) S (O)2CH2(D1-103a) Bu-t
CH (Et) S (O)2CH2(D1-103a) Pen-n
CH (Et) S (O)2CH2(D1-103a) Pen-c
CH (Et) S (O)2CH2(D1-103a) Hex-n
CH (Et) S (O)2CH2(D1-103a) Hex-c
CH (Et) S (O)2CH2(D1-103a) CH2Pr-c
CH (Et) S (O)2CH2(D1-103a) CH2Bu-c
CH (Et) S (O)2CH2(D1-103a) CH2Pen-c
CH (Et) S (O)2CH2(D1-103a) CH2Hex-c
CH (Et) S (O)2CH2(D1-103a) CH2CH = CH2
CH (Et) S (O)2CH2(D1-103a) CH2CH = C (Cl)2
CH (Et) S (O)2CH2(D1-103a) CH2C≡CH
CH (Et) S (O)2CH2(D1-103a) CH2CN
CH (Et) S (O)2CH2(D1-103a) CH2CFThree
CH (Et) S (O)2CH2(D1-103a) CH2OMe
CH (Et) S (O)2CH2(D1-103a) CH2OCFThree
CH (Et) S (O)2CH2(D1-103a) CH2SMe
CH (Et) S (O)2CH2(D1-103a) CH2S (O) Me
CH (Et) S (O)2CH2(D1-103a) CH2S (O)2Me
CH (Et) S (O)2CH2(D1-103a) CH2SCFThree
CH (Et) S (O)2CH2(D1-103a) CH2S (O) CFThree
CH (Et) S (O)2CH2(D1-103a) CH2S (O)2CFThree
CH (Et) S (O)2CH2(D1-103a) CH2CH (OMe)2
CH (Et) S (O)2CH2(D1-103a) CH2CH (SMe)2
CH (Et) S (O)2CH2(D1-103a) CH2C (O) Me
CH (Et) S (O)2CH2(D1-103a) CH2C (O) CFThree
CH (Et) S (O)2CH2(D1-103a) CH2C (O) OMe
CH (Et) S (O)2CH2(D1-103a) CH2(D1-32a)
CH (Et) S (O)2CH2(D1-103a) CH2(D1-33a)
CH (Et) S (O)2CH2(D1-103a) CH2(D1-34a)
CH (Et) S (O)2CH2(D1-103a) CH2(D1-37a)
CH (Et) S (O)2CH2(D1-103a) CH2(D1-81a)
CH (Et) S (O)2CH2(D1-103a) CH2(D1-82a)
CH (Et) S (O)2CH2(D1-103a) CH2(D1-84a)
CH (Et) S (O)2CH2(D1-103a) CH2(D1-85a)
CH (Et) S (O)2CH2(D1-103a) CH2(D1-87a)
CH (Et) S (O)2CH2(D1-103a) CH2(D1-92a)
CH (Et) S (O)2CH2(D1-103a) CH2(D1-93a)
CH (Et) S (O)2CH2(D1-103a) CH2(D1-95a)
CH (Et) S (O)2CH2(D1-103a) CH2(D1-96a)
CH (Et) S (O)2CH2(D1-103a) CH2(D1-98a)
CH (Et) S (O)2CH2(D1-103a) CH2(D1-108a)
CH (Et) S (O)2CH2(D1-103a) CH2(D1-108b, Z = 2-Cl)
CH (Et) S (O)2CH2(D1-103a) CH2(D1-108b, Z = 3-Me)
CH (Et) S (O)2CH2(D1-103a) CH2(D1-108b, Z = 4-OMe)
CH (Et) S (O)2CH2(D1-103a) CH2(D1-108b, Z = 2-SMe)
CH (Et) S (O)2CH2(D1-103a) CH2(D1-108b, Z = 3-CFThree)
CH (Et) S (O)2CH2(D1-103a) CH2(D1-108b, Z = 4-OCFThree)
CH (Et) S (O)2CH2(D1-103a) CH2(D1-108b, Z = 2-SCFThree)
CH (Et) S (O)2CH2(D1-103a) CH2CH2CN
CH (Et) S (O)2CH2(D1-103a) CH2CH2CFThree
CH (Et) S (O)2CH2(D1-103a) CH2CH2OMe
CH (Et) S (O)2CH2(D1-103a) CH2CH2SMe
CH (Et) S (O)2CH2(D1-103a) CH2CH2S (O) Me
CH (Et) S (O)2CH2(D1-103a) CH2CH2S (O)2Me
CH (Et) S (O)2CH2(D1-103a) D1-32a
CH (Et) S (O)2CH2(D1-103a) D1-33a
CH (Et) S (O)2CH2(D1-103a) D1-34a
CH (Et) S (O)2CH2(D1-103a) D1-37a
CH (Et) S (O)2CH2(D1-103a) D1-81a
CH (Et) S (O)2CH2(D1-103a) D1-82a
CH (Et) S (O)2CH2(D1-103a) D1-84a
CH (Et) S (O)2CH2(D1-103a) D1-85a
CH (Et) S (O)2CH2(D1-103a) D1-87a
CH (Et) S (O)2CH2(D1-103a) D1-92a
CH (Et) S (O)2CH2(D1-103a) D1-93a
CH (Et) S (O)2CH2(D1-103a) D1-95a
CH (Et) S (O)2CH2(D1-103a) D1-96a
CH (Et) S (O)2CH2(D1-103a) D1-98a
CH (Et) S (O)2CH2(D1-103a) D1-108a
CH (Et) S (O)2CH2(D1-103a) D1-108b (Z = 2-Cl)
CH (Et) S (O)2CH2(D1-103a) D1-108b (Z = 3-Me)
CH (Et) S (O)2CH2(D1-103a) D1-108b (Z = 4-OMe)
CH (Et) S (O)2CH2(D1-103a) D1-108b (Z = 2-SMe)
CH (Et) S (O)2CH2(D1-103a) D1-108b (Z = 3-CFThree)
CH (Et) S (O)2CH2(D1-103a) D1-108b (Z = 4-OCFThree)
CH (Et) S (O)2CH2(D1-103a) D1-108b (Z = 2-SCFThree)
CH (Et) S (O)2CH2(D1-103a) C (O) Me
CH (Et) S (O)2CH2(D1-103a) C (O) CFThree
CH (Et) S (O)2CH2(D1-103a) C (O) OMe
CH2SCH2CH = CH2                         Me
CH2SCH2CH = CH2                         Et
CH2SCH2CH = CH2                         Pr-n
CH2SCH2CH = CH2                         Pr-i
CH2SCH2CH = CH2                         Pr-c
CH2SCH2CH = CH2                         Bu-n
CH2SCH2CH = CH2                         Bu-i
CH2SCH2CH = CH2                         Bu-c
CH2SCH2CH = CH2                         Bu-s
CH2SCH2CH = CH2                         Bu-t
CH2SCH2CH = CH2                         Pen-n
CH2SCH2CH = CH2                         Pen-c
CH2SCH2CH = CH2                         Hex-n
CH2SCH2CH = CH2                         Hex-c
CH2SCH2CH = CH2                         CH2Pr-c
CH2SCH2CH = CH2                         CH2Bu-c
CH2SCH2CH = CH2                         CH2Pen-c
CH2SCH2CH = CH2                         CH2Hex-c
CH2SCH2CH = CH2                         CH2CH = CH2
CH2SCH2CH = CH2                         CH2CH = C (Cl)2
CH2SCH2CH = CH2                         CH2C≡CH
CH2SCH2CH = CH2                         CH2CN
CH2SCH2CH = CH2                         CH2CFThree
CH2SCH2CH = CH2                         CH2OMe
CH2SCH2CH = CH2                         CH2OCFThree
CH2SCH2CH = CH2                         CH2SMe
CH2SCH2CH = CH2                         CH2S (O) Me
CH2SCH2CH = CH2                         CH2S (O)2Me
CH2SCH2CH = CH2                         CH2SCFThree
CH2SCH2CH = CH2                         CH2S (O) CFThree
CH2SCH2CH = CH2                         CH2S (O)2CFThree
CH2SCH2CH = CH2                         CH2CH (OMe)2
CH2SCH2CH = CH2                         CH2CH (SMe)2
CH2SCH2CH = CH2                         CH2C (O) Me
CH2SCH2CH = CH2                         CH2C (O) CFThree
CH2SCH2CH = CH2                         CH2C (O) OMe
CH2SCH2CH = CH2                         CH2(D1-32a)
CH2SCH2CH = CH2                         CH2(D1-33a)
CH2SCH2CH = CH2                         CH2(D1-34a)
CH2SCH2CH = CH2                         CH2(D1-37a)
CH2SCH2CH = CH2                         CH2(D1-81a)
CH2SCH2CH = CH2                         CH2(D1-82a)
CH2SCH2CH = CH2                         CH2(D1-84a)
CH2SCH2CH = CH2                         CH2(D1-85a)
CH2SCH2CH = CH2                         CH2(D1-87a)
CH2SCH2CH = CH2                         CH2(D1-92a)
CH2SCH2CH = CH2                         CH2(D1-93a)
CH2SCH2CH = CH2                         CH2(D1-95a)
CH2SCH2CH = CH2                         CH2(D1-96a)
CH2SCH2CH = CH2                         CH2(D1-98a)
CH2SCH2CH = CH2                         CH2(D1-108a)
CH2SCH2CH = CH2                         CH2(D1-108b, Z = 2-Cl)
CH2SCH2CH = CH2                         CH2(D1-108b, Z = 3-Me)
CH2SCH2CH = CH2                         CH2(D1-108b, Z = 4-OMe)
CH2SCH2CH = CH2                         CH2(D1-108b, Z = 2-SMe)
CH2SCH2CH = CH2                         CH2(D1-108b, Z = 3-CFThree)
CH2SCH2CH = CH2                         CH2(D1-108b, Z = 4-OCFThree)
CH2SCH2CH = CH2                         CH2(D1-108b, Z = 2-SCFThree)
CH2SCH2CH = CH2                         CH2CH2CN
CH2SCH2CH = CH2                         CH2CH2CFThree
CH2SCH2CH = CH2                         CH2CH2OMe
CH2SCH2CH = CH2                         CH2CH2SMe
CH2SCH2CH = CH2                         CH2CH2S (O) Me
CH2SCH2CH = CH2                         CH2CH2S (O)2Me
CH2SCH2CH = CH2                         D1-32a
CH2SCH2CH = CH2                         D1-33a
CH2SCH2CH = CH2                         D1-34a
CH2SCH2CH = CH2                         D1-37a
CH2SCH2CH = CH2                         D1-81a
CH2SCH2CH = CH2                         D1-82a
CH2SCH2CH = CH2                         D1-84a
CH2SCH2CH = CH2                         D1-85a
CH2SCH2CH = CH2                         D1-87a
CH2SCH2CH = CH2                         D1-92a
CH2SCH2CH = CH2                         D1-93a
CH2SCH2CH = CH2                         D1-95a
CH2SCH2CH = CH2                         D1-96a
CH2SCH2CH = CH2                         D1-98a
CH2SCH2CH = CH2                         D1-108a
CH2SCH2CH = CH2                         D1-108b (Z = 2-Cl)
CH2SCH2CH = CH2                         D1-108b (Z = 3-Me)
CH2SCH2CH = CH2                         D1-108b (Z = 4-OMe)
CH2SCH2CH = CH2                         D1-108b (Z = 2-SMe)
CH2SCH2CH = CH2                         D1-108b (Z = 3-CFThree)
CH2SCH2CH = CH2                         D1-108b (Z = 4-OCFThree)
CH2SCH2CH = CH2                         D1-108b (Z = 2-SCFThree)
CH2SCH2CH = CH2                         C (O) Me
CH2SCH2CH = CH2                         C (O) CFThree
CH2SCH2CH = CH2                         C (O) OMe
CH2S (O) CH2CH = CH2                      Me
CH2S (O) CH2CH = CH2                      Et
CH2S (O) CH2CH = CH2                      Pr-n
CH2S (O) CH2CH = CH2                      Pr-i
CH2S (O) CH2CH = CH2                      Pr-c
CH2S (O) CH2CH = CH2                      Bu-n
CH2S (O) CH2CH = CH2                      Bu-i
CH2S (O) CH2CH = CH2                      Bu-c
CH2S (O) CH2CH = CH2                      Bu-s
CH2S (O) CH2CH = CH2                      Bu-t
CH2S (O) CH2CH = CH2                      Pen-n
CH2S (O) CH2CH = CH2                      Pen-c
CH2S (O) CH2CH = CH2                      Hex-n
CH2S (O) CH2CH = CH2                      Hex-c
CH2S (O) CH2CH = CH2                      CH2Pr-c
CH2S (O) CH2CH = CH2                      CH2Bu-c
CH2S (O) CH2CH = CH2                      CH2Pen-c
CH2S (O) CH2CH = CH2                      CH2Hex-c
CH2S (O) CH2CH = CH2                      CH2CH = CH2
CH2S (O) CH2CH = CH2                      CH2CH = C (Cl)2
CH2S (O) CH2CH = CH2                      CH2C≡CH
CH2S (O) CH2CH = CH2                      CH2CN
CH2S (O) CH2CH = CH2                      CH2CFThree
CH2S (O) CH2CH = CH2                      CH2OMe
CH2S (O) CH2CH = CH2                      CH2OCFThree
CH2S (O) CH2CH = CH2                      CH2SMe
CH2S (O) CH2CH = CH2                      CH2S (O) Me
CH2S (O) CH2CH = CH2                      CH2S (O)2Me
CH2S (O) CH2CH = CH2                      CH2SCFThree
CH2S (O) CH2CH = CH2                      CH2S (O) CFThree
CH2S (O) CH2CH = CH2                      CH2S (O)2CFThree
CH2S (O) CH2CH = CH2                      CH2CH (OMe)2
CH2S (O) CH2CH = CH2                      CH2CH (SMe)2
CH2S (O) CH2CH = CH2                      CH2C (O) Me
CH2S (O) CH2CH = CH2                      CH2C (O) CFThree
CH2S (O) CH2CH = CH2                      CH2C (O) OMe
CH2S (O) CH2CH = CH2                      CH2(D1-32a)
CH2S (O) CH2CH = CH2                      CH2(D1-33a)
CH2S (O) CH2CH = CH2                      CH2(D1-34a)
CH2S (O) CH2CH = CH2                      CH2(D1-37a)
CH2S (O) CH2CH = CH2                      CH2(D1-81a)
CH2S (O) CH2CH = CH2                      CH2(D1-82a)
CH2S (O) CH2CH = CH2                      CH2(D1-84a)
CH2S (O) CH2CH = CH2                      CH2(D1-85a)
CH2S (O) CH2CH = CH2                      CH2(D1-87a)
CH2S (O) CH2CH = CH2                      CH2(D1-92a)
CH2S (O) CH2CH = CH2                      CH2(D1-93a)
CH2S (O) CH2CH = CH2                      CH2(D1-95a)
CH2S (O) CH2CH = CH2                      CH2(D1-96a)
CH2S (O) CH2CH = CH2                      CH2(D1-98a)
CH2S (O) CH2CH = CH2                      CH2(D1-108a)
CH2S (O) CH2CH = CH2                      CH2(D1-108b, Z = 2-Cl)
CH2S (O) CH2CH = CH2                      CH2(D1-108b, Z = 3-Me)
CH2S (O) CH2CH = CH2                      CH2(D1-108b, Z = 4-OMe)
CH2S (O) CH2CH = CH2                      CH2(D1-108b, Z = 2-SMe)
CH2S (O) CH2CH = CH2                      CH2(D1-108b, Z = 3-CFThree)
CH2S (O) CH2CH = CH2                      CH2(D1-108b, Z = 4-OCFThree)
CH2S (O) CH2CH = CH2                      CH2(D1-108b, Z = 2-SCFThree)
CH2S (O) CH2CH = CH2                      CH2CH2CN
CH2S (O) CH2CH = CH2                      CH2CH2CFThree
CH2S (O) CH2CH = CH2                      CH2CH2OMe
CH2S (O) CH2CH = CH2                      CH2CH2SMe
CH2S (O) CH2CH = CH2                      CH2CH2S (O) Me
CH2S (O) CH2CH = CH2                      CH2CH2S (O)2Me
CH2S (O) CH2CH = CH2                      D1-32a
CH2S (O) CH2CH = CH2                      D1-33a
CH2S (O) CH2CH = CH2                      D1-34a
CH2S (O) CH2CH = CH2                      D1-37a
CH2S (O) CH2CH = CH2                      D1-81a
CH2S (O) CH2CH = CH2                      D1-82a
CH2S (O) CH2CH = CH2                      D1-84a
CH2S (O) CH2CH = CH2                      D1-85a
CH2S (O) CH2CH = CH2                      D1-87a
CH2S (O) CH2CH = CH2                      D1-92a
CH2S (O) CH2CH = CH2                      D1-93a
CH2S (O) CH2CH = CH2                      D1-95a
CH2S (O) CH2CH = CH2                      D1-96a
CH2S (O) CH2CH = CH2                      D1-98a
CH2S (O) CH2CH = CH2                      D1-108a
CH2S (O) CH2CH = CH2                      D1-108b (Z = 2-Cl)
CH2S (O) CH2CH = CH2                      D1-108b (Z = 3-Me)
CH2S (O) CH2CH = CH2                      D1-108b (Z = 4-OMe)
CH2S (O) CH2CH = CH2                      D1-108b (Z = 2-SMe)
CH2S (O) CH2CH = CH2                      D1-108b (Z = 3-CFThree)
CH2S (O) CH2CH = CH2                      D1-108b (Z = 4-OCFThree)
CH2S (O) CH2CH = CH2                      D1-108b (Z = 2-SCFThree)
CH2S (O) CH2CH = CH2                      C (O) Me
CH2S (O) CH2CH = CH2                      C (O) CFThree
CH2S (O) CH2CH = CH2                      C (O) OMe
CH2S (O)2CH2CH = CH2                     Me
CH2S (O)2CH2CH = CH2                     Et
CH2S (O)2CH2CH = CH2                     Pr-n
CH2S (O)2CH2CH = CH2                     Pr-i
CH2S (O)2CH2CH = CH2                     Pr-c
CH2S (O)2CH2CH = CH2                     Bu-n
CH2S (O)2CH2CH = CH2                     Bu-i
CH2S (O)2CH2CH = CH2                     Bu-c
CH2S (O)2CH2CH = CH2                     Bu-s
CH2S (O)2CH2CH = CH2                     Bu-t
CH2S (O)2CH2CH = CH2                     Pen-n
CH2S (O)2CH2CH = CH2                     Pen-c
CH2S (O)2CH2CH = CH2                     Hex-n
CH2S (O)2CH2CH = CH2                     Hex-c
CH2S (O)2CH2CH = CH2                     CH2Pr-c
CH2S (O)2CH2CH = CH2                     CH2Bu-c
CH2S (O)2CH2CH = CH2                     CH2Pen-c
CH2S (O)2CH2CH = CH2                     CH2Hex-c
CH2S (O)2CH2CH = CH2                     CH2CH = CH2
CH2S (O)2CH2CH = CH2                     CH2CH = C (Cl)2
CH2S (O)2CH2CH = CH2                     CH2C≡CH
CH2S (O)2CH2CH = CH2                     CH2CN
CH2S (O)2CH2CH = CH2                     CH2CFThree
CH2S (O)2CH2CH = CH2                     CH2OMe
CH2S (O)2CH2CH = CH2                     CH2OCFThree
CH2S (O)2CH2CH = CH2                     CH2SMe
CH2S (O)2CH2CH = CH2                     CH2S (O) Me
CH2S (O)2CH2CH = CH2                     CH2S (O)2Me
CH2S (O)2CH2CH = CH2                     CH2SCFThree
CH2S (O)2CH2CH = CH2                     CH2S (O) CFThree
CH2S (O)2CH2CH = CH2                     CH2S (O)2CFThree
CH2S (O)2CH2CH = CH2                     CH2CH (OMe)2
CH2S (O)2CH2CH = CH2                     CH2CH (SMe)2
CH2S (O)2CH2CH = CH2                     CH2C (O) Me
CH2S (O)2CH2CH = CH2                     CH2C (O) CFThree
CH2S (O)2CH2CH = CH2                     CH2C (O) OMe
CH2S (O)2CH2CH = CH2                     CH2(D1-32a)
CH2S (O)2CH2CH = CH2                     CH2(D1-33a)
CH2S (O)2CH2CH = CH2                     CH2(D1-34a)
CH2S (O)2CH2CH = CH2                     CH2(D1-37a)
CH2S (O)2CH2CH = CH2                     CH2(D1-81a)
CH2S (O)2CH2CH = CH2                     CH2(D1-82a)
CH2S (O)2CH2CH = CH2                     CH2(D1-84a)
CH2S (O)2CH2CH = CH2                     CH2(D1-85a)
CH2S (O)2CH2CH = CH2                     CH2(D1-87a)
CH2S (O)2CH2CH = CH2                     CH2(D1-92a)
CH2S (O)2CH2CH = CH2                     CH2(D1-93a)
CH2S (O)2CH2CH = CH2                     CH2(D1-95a)
CH2S (O)2CH2CH = CH2                     CH2(D1-96a)
CH2S (O)2CH2CH = CH2                     CH2(D1-98a)
CH2S (O)2CH2CH = CH2                     CH2(D1-108a)
CH2S (O)2CH2CH = CH2                     CH2(D1-108b, Z = 2-Cl)
CH2S (O)2CH2CH = CH2                     CH2(D1-108b, Z = 3-Me)
CH2S (O)2CH2CH = CH2                     CH2(D1-108b, Z = 4-OMe)
CH2S (O)2CH2CH = CH2                     CH2(D1-108b, Z = 2-SMe)
CH2S (O)2CH2CH = CH2                     CH2(D1-108b, Z = 3-CFThree)
CH2S (O)2CH2CH = CH2                     CH2(D1-108b, Z = 4-OCFThree)
CH2S (O)2CH2CH = CH2                     CH2(D1-108b, Z = 2-SCFThree)
CH2S (O)2CH2CH = CH2                     CH2CH2CN
CH2S (O)2CH2CH = CH2                     CH2CH2CFThree
CH2S (O)2CH2CH = CH2                     CH2CH2OMe
CH2S (O)2CH2CH = CH2                     CH2CH2SMe
CH2S (O)2CH2CH = CH2                     CH2CH2S (O) Me
CH2S (O)2CH2CH = CH2                     CH2CH2S (O)2Me
CH2S (O)2CH2CH = CH2                     D1-32a
CH2S (O)2CH2CH = CH2                     D1-33a
CH2S (O)2CH2CH = CH2                     D1-34a
CH2S (O)2CH2CH = CH2                     D1-37a
CH2S (O)2CH2CH = CH2                     D1-81a
CH2S (O)2CH2CH = CH2                     D1-82a
CH2S (O)2CH2CH = CH2                     D1-84a
CH2S (O)2CH2CH = CH2                     D1-85a
CH2S (O)2CH2CH = CH2                     D1-87a
CH2S (O)2CH2CH = CH2                     D1-92a
CH2S (O)2CH2CH = CH2                     D1-93a
CH2S (O)2CH2CH = CH2                     D1-95a
CH2S (O)2CH2CH = CH2                     D1-96a
CH2S (O)2CH2CH = CH2                     D1-98a
CH2S (O)2CH2CH = CH2                     D1-108a
CH2S (O)2CH2CH = CH2                     D1-108b (Z = 2-Cl)
CH2S (O)2CH2CH = CH2                     D1-108b (Z = 3-Me)
CH2S (O)2CH2CH = CH2                     D1-108b (Z = 4-OMe)
CH2S (O)2CH2CH = CH2                     D1-108b (Z = 2-SMe)
CH2S (O)2CH2CH = CH2                     D1-108b (Z = 3-CFThree)
CH2S (O)2CH2CH = CH2                     D1-108b (Z = 4-OCFThree)
CH2S (O)2CH2CH = CH2                     D1-108b (Z = 2-SCFThree)
CH2S (O)2CH2CH = CH2                     C (O) Me
CH2S (O)2CH2CH = CH2                     C (O) CFThree
CH2S (O)2CH2CH = CH2                     C (O) OMe
CH (Me) SCH2CH = CH2                      Me
CH (Me) SCH2CH = CH2                      Et
CH (Me) SCH2CH = CH2                      Pr-n
CH (Me) SCH2CH = CH2                      Pr-i
CH (Me) SCH2CH = CH2                      Pr-c
CH (Me) SCH2CH = CH2                      Bu-n
CH (Me) SCH2CH = CH2                      Bu-i
CH (Me) SCH2CH = CH2                      Bu-c
CH (Me) SCH2CH = CH2                      Bu-s
CH (Me) SCH2CH = CH2                      Bu-t
CH (Me) SCH2CH = CH2                      Pen-n
CH (Me) SCH2CH = CH2                      Pen-c
CH (Me) SCH2CH = CH2                      Hex-n
CH (Me) SCH2CH = CH2                      Hex-c
CH (Me) SCH2CH = CH2                      CH2Pr-c
CH (Me) SCH2CH = CH2                      CH2Bu-c
CH (Me) SCH2CH = CH2                      CH2Pen-c
CH (Me) SCH2CH = CH2                      CH2Hex-c
CH (Me) SCH2CH = CH2                      CH2CH = CH2
CH (Me) SCH2CH = CH2                      CH2CH = C (Cl)2
CH (Me) SCH2CH = CH2                      CH2C≡CH
CH (Me) SCH2CH = CH2                      CH2CN
CH (Me) SCH2CH = CH2                      CH2CFThree
CH (Me) SCH2CH = CH2                      CH2OMe
CH (Me) SCH2CH = CH2                      CH2OCFThree
CH (Me) SCH2CH = CH2                      CH2SMe
CH (Me) SCH2CH = CH2                      CH2S (O) Me
CH (Me) SCH2CH = CH2                      CH2S (O)2Me
CH (Me) SCH2CH = CH2                      CH2SCFThree
CH (Me) SCH2CH = CH2                      CH2S (O) CFThree
CH (Me) SCH2CH = CH2                      CH2S (O)2CFThree
CH (Me) SCH2CH = CH2                      CH2CH (OMe)2
CH (Me) SCH2CH = CH2                      CH2CH (SMe)2
CH (Me) SCH2CH = CH2                      CH2C (O) Me
CH (Me) SCH2CH = CH2                      CH2C (O) CFThree
CH (Me) SCH2CH = CH2                      CH2C (O) OMe
CH (Me) SCH2CH = CH2                      CH2(D1-32a)
CH (Me) SCH2CH = CH2                      CH2(D1-33a)
CH (Me) SCH2CH = CH2                      CH2(D1-34a)
CH (Me) SCH2CH = CH2                      CH2(D1-37a)
CH (Me) SCH2CH = CH2                      CH2(D1-81a)
CH (Me) SCH2CH = CH2                      CH2(D1-82a)
CH (Me) SCH2CH = CH2                      CH2(D1-84a)
CH (Me) SCH2CH = CH2                      CH2(D1-85a)
CH (Me) SCH2CH = CH2                      CH2(D1-87a)
CH (Me) SCH2CH = CH2                      CH2(D1-92a)
CH (Me) SCH2CH = CH2                      CH2(D1-93a)
CH (Me) SCH2CH = CH2                      CH2(D1-95a)
CH (Me) SCH2CH = CH2                      CH2(D1-96a)
CH (Me) SCH2CH = CH2                      CH2(D1-98a)
CH (Me) SCH2CH = CH2                      CH2(D1-108a)
CH (Me) SCH2CH = CH2                      CH2(D1-108b, Z = 2-Cl)
CH (Me) SCH2CH = CH2                      CH2(D1-108b, Z = 3-Me)
CH (Me) SCH2CH = CH2                      CH2(D1-108b, Z = 4-OMe)
CH (Me) SCH2CH = CH2                      CH2(D1-108b, Z = 2-SMe)
CH (Me) SCH2CH = CH2                      CH2(D1-108b, Z = 3-CFThree)
CH (Me) SCH2CH = CH2                      CH2(D1-108b, Z = 4-OCFThree)
CH (Me) SCH2CH = CH2                      CH2(D1-108b, Z = 2-SCFThree)
CH (Me) SCH2CH = CH2                      CH2CH2CN
CH (Me) SCH2CH = CH2                      CH2CH2CFThree
CH (Me) SCH2CH = CH2                      CH2CH2OMe
CH (Me) SCH2CH = CH2                      CH2CH2SMe
CH (Me) SCH2CH = CH2                      CH2CH2S (O) Me
CH (Me) SCH2CH = CH2                      CH2CH2S (O)2Me
CH (Me) SCH2CH = CH2                      D1-32a
CH (Me) SCH2CH = CH2                      D1-33a
CH (Me) SCH2CH = CH2                      D1-34a
CH (Me) SCH2CH = CH2                      D1-37a
CH (Me) SCH2CH = CH2                      D1-81a
CH (Me) SCH2CH = CH2                      D1-82a
CH (Me) SCH2CH = CH2                      D1-84a
CH (Me) SCH2CH = CH2                      D1-85a
CH (Me) SCH2CH = CH2                      D1-87a
CH (Me) SCH2CH = CH2                      D1-92a
CH (Me) SCH2CH = CH2                      D1-93a
CH (Me) SCH2CH = CH2                      D1-95a
CH (Me) SCH2CH = CH2                      D1-96a
CH (Me) SCH2CH = CH2                      D1-98a
CH (Me) SCH2CH = CH2                      D1-108a
CH (Me) SCH2CH = CH2                      D1-108b (Z = 2-Cl)
CH (Me) SCH2CH = CH2                      D1-108b (Z = 3-Me)
CH (Me) SCH2CH = CH2                      D1-108b (Z = 4-OMe)
CH (Me) SCH2CH = CH2                      D1-108b (Z = 2-SMe)
CH (Me) SCH2CH = CH2                      D1-108b (Z = 3-CFThree)
CH (Me) SCH2CH = CH2                      D1-108b (Z = 4-OCFThree)
CH (Me) SCH2CH = CH2                      D1-108b (Z = 2-SCFThree)
CH (Me) SCH2CH = CH2                      C (O) Me
CH (Me) SCH2CH = CH2                      C (O) CFThree
CH (Me) SCH2CH = CH2                      C (O) OMe
CH (Me) S (O) CH2CH = CH2                   Me
CH (Me) S (O) CH2CH = CH2                   Et
CH (Me) S (O) CH2CH = CH2                   Pr-n
CH (Me) S (O) CH2CH = CH2                   Pr-i
CH (Me) S (O) CH2CH = CH2                   Pr-c
CH (Me) S (O) CH2CH = CH2                   Bu-n
CH (Me) S (O) CH2CH = CH2                   Bu-i
CH (Me) S (O) CH2CH = CH2                   Bu-c
CH (Me) S (O) CH2CH = CH2                   Bu-s
CH (Me) S (O) CH2CH = CH2                   Bu-t
CH (Me) S (O) CH2CH = CH2                   Pen-n
CH (Me) S (O) CH2CH = CH2                   Pen-c
CH (Me) S (O) CH2CH = CH2                   Hex-n
CH (Me) S (O) CH2CH = CH2                   Hex-c
CH (Me) S (O) CH2CH = CH2                   CH2Pr-c
CH (Me) S (O) CH2CH = CH2                   CH2Bu-c
CH (Me) S (O) CH2CH = CH2                   CH2Pen-c
CH (Me) S (O) CH2CH = CH2                   CH2Hex-c
CH (Me) S (O) CH2CH = CH2                   CH2CH = CH2
CH (Me) S (O) CH2CH = CH2                   CH2CH = C (Cl)2
CH (Me) S (O) CH2CH = CH2                   CH2C≡CH
CH (Me) S (O) CH2CH = CH2                   CH2CN
CH (Me) S (O) CH2CH = CH2                   CH2CFThree
CH (Me) S (O) CH2CH = CH2                   CH2OMe
CH (Me) S (O) CH2CH = CH2                   CH2OCFThree
CH (Me) S (O) CH2CH = CH2                   CH2SMe
CH (Me) S (O) CH2CH = CH2                   CH2S (O) Me
CH (Me) S (O) CH2CH = CH2                   CH2S (O)2Me
CH (Me) S (O) CH2CH = CH2                   CH2SCFThree
CH (Me) S (O) CH2CH = CH2                   CH2S (O) CFThree
CH (Me) S (O) CH2CH = CH2                   CH2S (O)2CFThree
CH (Me) S (O) CH2CH = CH2                   CH2CH (OMe)2
CH (Me) S (O) CH2CH = CH2                   CH2CH (SMe)2
CH (Me) S (O) CH2CH = CH2                   CH2C (O) Me
CH (Me) S (O) CH2CH = CH2                   CH2C (O) CFThree
CH (Me) S (O) CH2CH = CH2                   CH2C (O) OMe
CH (Me) S (O) CH2CH = CH2                   CH2(D1-32a)
CH (Me) S (O) CH2CH = CH2                   CH2(D1-33a)
CH (Me) S (O) CH2CH = CH2                   CH2(D1-34a)
CH (Me) S (O) CH2CH = CH2                   CH2(D1-37a)
CH (Me) S (O) CH2CH = CH2                   CH2(D1-81a)
CH (Me) S (O) CH2CH = CH2                   CH2(D1-82a)
CH (Me) S (O) CH2CH = CH2                   CH2(D1-84a)
CH (Me) S (O) CH2CH = CH2                   CH2(D1-85a)
CH (Me) S (O) CH2CH = CH2                   CH2(D1-87a)
CH (Me) S (O) CH2CH = CH2                   CH2(D1-92a)
CH (Me) S (O) CH2CH = CH2                   CH2(D1-93a)
CH (Me) S (O) CH2CH = CH2                   CH2(D1-95a)
CH (Me) S (O) CH2CH = CH2                   CH2(D1-96a)
CH (Me) S (O) CH2CH = CH2                   CH2(D1-98a)
CH (Me) S (O) CH2CH = CH2                   CH2(D1-108a)
CH (Me) S (O) CH2CH = CH2                   CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O) CH2CH = CH2                   CH2(D1-108b, Z = 3-Me)
CH (Me) S (O) CH2CH = CH2                   CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O) CH2CH = CH2                   CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O) CH2CH = CH2                   CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O) CH2CH = CH2                   CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O) CH2CH = CH2                   CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O) CH2CH = CH2                   CH2CH2CN
CH (Me) S (O) CH2CH = CH2                   CH2CH2CFThree
CH (Me) S (O) CH2CH = CH2                   CH2CH2OMe
CH (Me) S (O) CH2CH = CH2                   CH2CH2SMe
CH (Me) S (O) CH2CH = CH2                   CH2CH2S (O) Me
CH (Me) S (O) CH2CH = CH2                   CH2CH2S (O)2Me
CH (Me) S (O) CH2CH = CH2                   D1-32a
CH (Me) S (O) CH2CH = CH2                   D1-33a
CH (Me) S (O) CH2CH = CH2                   D1-34a
CH (Me) S (O) CH2CH = CH2                   D1-37a
CH (Me) S (O) CH2CH = CH2                   D1-81a
CH (Me) S (O) CH2CH = CH2                   D1-82a
CH (Me) S (O) CH2CH = CH2                   D1-84a
CH (Me) S (O) CH2CH = CH2                   D1-85a
CH (Me) S (O) CH2CH = CH2                   D1-87a
CH (Me) S (O) CH2CH = CH2                   D1-92a
CH (Me) S (O) CH2CH = CH2                   D1-93a
CH (Me) S (O) CH2CH = CH2                   D1-95a
CH (Me) S (O) CH2CH = CH2                   D1-96a
CH (Me) S (O) CH2CH = CH2                   D1-98a
CH (Me) S (O) CH2CH = CH2                   D1-108a
CH (Me) S (O) CH2CH = CH2                   D1-108b (Z = 2-Cl)
CH (Me) S (O) CH2CH = CH2                   D1-108b (Z = 3-Me)
CH (Me) S (O) CH2CH = CH2                   D1-108b (Z = 4-OMe)
CH (Me) S (O) CH2CH = CH2                   D1-108b (Z = 2-SMe)
CH (Me) S (O) CH2CH = CH2                   D1-108b (Z = 3-CFThree)
CH (Me) S (O) CH2CH = CH2                   D1-108b (Z = 4-OCFThree)
CH (Me) S (O) CH2CH = CH2                   D1-108b (Z = 2-SCFThree)
CH (Me) S (O) CH2CH = CH2                   C (O) Me
CH (Me) S (O) CH2CH = CH2                   C (O) CFThree
CH (Me) S (O) CH2CH = CH2                   C (O) OMe
CH (Me) S (O)2CH2CH = CH2                   Me
CH (Me) S (O)2CH2CH = CH2                   Et
CH (Me) S (O)2CH2CH = CH2                   Pr-n
CH (Me) S (O)2CH2CH = CH2                   Pr-i
CH (Me) S (O)2CH2CH = CH2                   Pr-c
CH (Me) S (O)2CH2CH = CH2                   Bu-n
CH (Me) S (O)2CH2CH = CH2                   Bu-i
CH (Me) S (O)2CH2CH = CH2                   Bu-c
CH (Me) S (O)2CH2CH = CH2                   Bu-s
CH (Me) S (O)2CH2CH = CH2                   Bu-t
CH (Me) S (O)2CH2CH = CH2                   Pen-n
CH (Me) S (O)2CH2CH = CH2                   Pen-c
CH (Me) S (O)2CH2CH = CH2                   Hex-n
CH (Me) S (O)2CH2CH = CH2                   Hex-c
CH (Me) S (O)2CH2CH = CH2                   CH2Pr-c
CH (Me) S (O)2CH2CH = CH2                   CH2Bu-c
CH (Me) S (O)2CH2CH = CH2                   CH2Pen-c
CH (Me) S (O)2CH2CH = CH2                   CH2Hex-c
CH (Me) S (O)2CH2CH = CH2                   CH2CH = CH2
CH (Me) S (O)2CH2CH = CH2                   CH2CH = C (Cl)2
CH (Me) S (O)2CH2CH = CH2                   CH2C≡CH
CH (Me) S (O)2CH2CH = CH2                   CH2CN
CH (Me) S (O)2CH2CH = CH2                   CH2CFThree
CH (Me) S (O)2CH2CH = CH2                   CH2OMe
CH (Me) S (O)2CH2CH = CH2                   CH2OCFThree
CH (Me) S (O)2CH2CH = CH2                   CH2SMe
CH (Me) S (O)2CH2CH = CH2                   CH2S (O) Me
CH (Me) S (O)2CH2CH = CH2                   CH2S (O)2Me
CH (Me) S (O)2CH2CH = CH2                   CH2SCFThree
CH (Me) S (O)2CH2CH = CH2                   CH2S (O) CFThree
CH (Me) S (O)2CH2CH = CH2                   CH2S (O)2CFThree
CH (Me) S (O)2CH2CH = CH2                   CH2CH (OMe)2
CH (Me) S (O)2CH2CH = CH2                   CH2CH (SMe)2
CH (Me) S (O)2CH2CH = CH2                   CH2C (O) Me
CH (Me) S (O)2CH2CH = CH2                   CH2C (O) CFThree
CH (Me) S (O)2CH2CH = CH2                   CH2C (O) OMe
CH (Me) S (O)2CH2CH = CH2                   CH2(D1-32a)
CH (Me) S (O)2CH2CH = CH2                   CH2(D1-33a)
CH (Me) S (O)2CH2CH = CH2                   CH2(D1-34a)
CH (Me) S (O)2CH2CH = CH2                   CH2(D1-37a)
CH (Me) S (O)2CH2CH = CH2                   CH2(D1-81a)
CH (Me) S (O)2CH2CH = CH2                   CH2(D1-82a)
CH (Me) S (O)2CH2CH = CH2                   CH2(D1-84a)
CH (Me) S (O)2CH2CH = CH2                   CH2(D1-85a)
CH (Me) S (O)2CH2CH = CH2                   CH2(D1-87a)
CH (Me) S (O)2CH2CH = CH2                   CH2(D1-92a)
CH (Me) S (O)2CH2CH = CH2                   CH2(D1-93a)
CH (Me) S (O)2CH2CH = CH2                   CH2(D1-95a)
CH (Me) S (O)2CH2CH = CH2                   CH2(D1-96a)
CH (Me) S (O)2CH2CH = CH2                   CH2(D1-98a)
CH (Me) S (O)2CH2CH = CH2                   CH2(D1-108a)
CH (Me) S (O)2CH2CH = CH2                   CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O)2CH2CH = CH2                   CH2(D1-108b, Z = 3-Me)
CH (Me) S (O)2CH2CH = CH2                   CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O)2CH2CH = CH2                   CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O)2CH2CH = CH2                   CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O)2CH2CH = CH2                   CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O)2CH2CH = CH2                   CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O)2CH2CH = CH2                   CH2CH2CN
CH (Me) S (O)2CH2CH = CH2                   CH2CH2CFThree
CH (Me) S (O)2CH2CH = CH2                   CH2CH2OMe
CH (Me) S (O)2CH2CH = CH2                   CH2CH2SMe
CH (Me) S (O)2CH2CH = CH2                   CH2CH2S (O) Me
CH (Me) S (O)2CH2CH = CH2                   CH2CH2S (O)2Me
CH (Me) S (O)2CH2CH = CH2                   D1-32a
CH (Me) S (O)2CH2CH = CH2                   D1-33a
CH (Me) S (O)2CH2CH = CH2                   D1-34a
CH (Me) S (O)2CH2CH = CH2                   D1-37a
CH (Me) S (O)2CH2CH = CH2                   D1-81a
CH (Me) S (O)2CH2CH = CH2                   D1-82a
CH (Me) S (O)2CH2CH = CH2                   D1-84a
CH (Me) S (O)2CH2CH = CH2                   D1-85a
CH (Me) S (O)2CH2CH = CH2                   D1-87a
CH (Me) S (O)2CH2CH = CH2                   D1-92a
CH (Me) S (O)2CH2CH = CH2                   D1-93a
CH (Me) S (O)2CH2CH = CH2                   D1-95a
CH (Me) S (O)2CH2CH = CH2                   D1-96a
CH (Me) S (O)2CH2CH = CH2                   D1-98a
CH (Me) S (O)2CH2CH = CH2                   D1-108a
CH (Me) S (O)2CH2CH = CH2                   D1-108b (Z = 2-Cl)
CH (Me) S (O)2CH2CH = CH2                   D1-108b (Z = 3-Me)
CH (Me) S (O)2CH2CH = CH2                   D1-108b (Z = 4-OMe)
CH (Me) S (O)2CH2CH = CH2                   D1-108b (Z = 2-SMe)
CH (Me) S (O)2CH2CH = CH2                   D1-108b (Z = 3-CFThree)
CH (Me) S (O)2CH2CH = CH2                   D1-108b (Z = 4-OCFThree)
CH (Me) S (O)2CH2CH = CH2                   D1-108b (Z = 2-SCFThree)
CH (Me) S (O)2CH2CH = CH2                   C (O) Me
CH (Me) S (O)2CH2CH = CH2                   C (O) CFThree
CH (Me) S (O)2CH2CH = CH2                   C (O) OMe
CH (Et) SCH2CH = CH2                      Me
CH (Et) SCH2CH = CH2                      Et
CH (Et) SCH2CH = CH2                      Pr-n
CH (Et) SCH2CH = CH2                      Pr-i
CH (Et) SCH2CH = CH2                      Pr-c
CH (Et) SCH2CH = CH2                      Bu-n
CH (Et) SCH2CH = CH2                      Bu-i
CH (Et) SCH2CH = CH2                      Bu-c
CH (Et) SCH2CH = CH2                      Bu-s
CH (Et) SCH2CH = CH2                      Bu-t
CH (Et) SCH2CH = CH2                      Pen-n
CH (Et) SCH2CH = CH2                      Pen-c
CH (Et) SCH2CH = CH2                      Hex-n
CH (Et) SCH2CH = CH2                      Hex-c
CH (Et) SCH2CH = CH2                      CH2Pr-c
CH (Et) SCH2CH = CH2                      CH2Bu-c
CH (Et) SCH2CH = CH2                      CH2Pen-c
CH (Et) SCH2CH = CH2                      CH2Hex-c
CH (Et) SCH2CH = CH2                      CH2CH = CH2
CH (Et) SCH2CH = CH2                      CH2CH = C (Cl)2
CH (Et) SCH2CH = CH2                      CH2C≡CH
CH (Et) SCH2CH = CH2                      CH2CN
CH (Et) SCH2CH = CH2                      CH2CFThree
CH (Et) SCH2CH = CH2                      CH2OMe
CH (Et) SCH2CH = CH2                      CH2OCFThree
CH (Et) SCH2CH = CH2                      CH2SMe
CH (Et) SCH2CH = CH2                      CH2S (O) Me
CH (Et) SCH2CH = CH2                      CH2S (O)2Me
CH (Et) SCH2CH = CH2                      CH2SCFThree
CH (Et) SCH2CH = CH2                      CH2S (O) CFThree
CH (Et) SCH2CH = CH2                      CH2S (O)2CFThree
CH (Et) SCH2CH = CH2                      CH2CH (OMe)2
CH (Et) SCH2CH = CH2                      CH2CH (SMe)2
CH (Et) SCH2CH = CH2                      CH2C (O) Me
CH (Et) SCH2CH = CH2                      CH2C (O) CFThree
CH (Et) SCH2CH = CH2                      CH2C (O) OMe
CH (Et) SCH2CH = CH2                      CH2(D1-32a)
CH (Et) SCH2CH = CH2                      CH2(D1-33a)
CH (Et) SCH2CH = CH2                      CH2(D1-34a)
CH (Et) SCH2CH = CH2                      CH2(D1-37a)
CH (Et) SCH2CH = CH2                      CH2(D1-81a)
CH (Et) SCH2CH = CH2                      CH2(D1-82a)
CH (Et) SCH2CH = CH2                      CH2(D1-84a)
CH (Et) SCH2CH = CH2                      CH2(D1-85a)
CH (Et) SCH2CH = CH2                      CH2(D1-87a)
CH (Et) SCH2CH = CH2                      CH2(D1-92a)
CH (Et) SCH2CH = CH2                      CH2(D1-93a)
CH (Et) SCH2CH = CH2                      CH2(D1-95a)
CH (Et) SCH2CH = CH2                      CH2(D1-96a)
CH (Et) SCH2CH = CH2                      CH2(D1-98a)
CH (Et) SCH2CH = CH2                      CH2(D1-108a)
CH (Et) SCH2CH = CH2                      CH2(D1-108b, Z = 2-Cl)
CH (Et) SCH2CH = CH2                      CH2(D1-108b, Z = 3-Me)
CH (Et) SCH2CH = CH2                      CH2(D1-108b, Z = 4-OMe)
CH (Et) SCH2CH = CH2                      CH2(D1-108b, Z = 2-SMe)
CH (Et) SCH2CH = CH2                      CH2(D1-108b, Z = 3-CFThree)
CH (Et) SCH2CH = CH2                      CH2(D1-108b, Z = 4-OCFThree)
CH (Et) SCH2CH = CH2                      CH2(D1-108b, Z = 2-SCFThree)
CH (Et) SCH2CH = CH2                      CH2CH2CN
CH (Et) SCH2CH = CH2                      CH2CH2CFThree
CH (Et) SCH2CH = CH2                      CH2CH2OMe
CH (Et) SCH2CH = CH2                      CH2CH2SMe
CH (Et) SCH2CH = CH2                      CH2CH2S (O) Me
CH (Et) SCH2CH = CH2                      CH2CH2S (O)2Me
CH (Et) SCH2CH = CH2                      D1-32a
CH (Et) SCH2CH = CH2                      D1-33a
CH (Et) SCH2CH = CH2                      D1-34a
CH (Et) SCH2CH = CH2                      D1-37a
CH (Et) SCH2CH = CH2                      D1-81a
CH (Et) SCH2CH = CH2                      D1-82a
CH (Et) SCH2CH = CH2                      D1-84a
CH (Et) SCH2CH = CH2                      D1-85a
CH (Et) SCH2CH = CH2                      D1-87a
CH (Et) SCH2CH = CH2                      D1-92a
CH (Et) SCH2CH = CH2                      D1-93a
CH (Et) SCH2CH = CH2                      D1-95a
CH (Et) SCH2CH = CH2                      D1-96a
CH (Et) SCH2CH = CH2                      D1-98a
CH (Et) SCH2CH = CH2                      D1-108a
CH (Et) SCH2CH = CH2                      D1-108b (Z = 2-Cl)
CH (Et) SCH2CH = CH2                      D1-108b (Z = 3-Me)
CH (Et) SCH2CH = CH2                      D1-108b (Z = 4-OMe)
CH (Et) SCH2CH = CH2                      D1-108b (Z = 2-SMe)
CH (Et) SCH2CH = CH2                      D1-108b (Z = 3-CFThree)
CH (Et) SCH2CH = CH2                      D1-108b (Z = 4-OCFThree)
CH (Et) SCH2CH = CH2                      D1-108b (Z = 2-SCFThree)
CH (Et) SCH2CH = CH2                      C (O) Me
CH (Et) SCH2CH = CH2                      C (O) CFThree
CH (Et) SCH2CH = CH2                      C (O) OMe
CH (Et) S (O) CH2CH = CH2                   Me
CH (Et) S (O) CH2CH = CH2                   Et
CH (Et) S (O) CH2CH = CH2                   Pr-n
CH (Et) S (O) CH2CH = CH2                   Pr-i
CH (Et) S (O) CH2CH = CH2                   Pr-c
CH (Et) S (O) CH2CH = CH2                   Bu-n
CH (Et) S (O) CH2CH = CH2                   Bu-i
CH (Et) S (O) CH2CH = CH2                   Bu-c
CH (Et) S (O) CH2CH = CH2                   Bu-s
CH (Et) S (O) CH2CH = CH2                   Bu-t
CH (Et) S (O) CH2CH = CH2                   Pen-n
CH (Et) S (O) CH2CH = CH2                   Pen-c
CH (Et) S (O) CH2CH = CH2                   Hex-n
CH (Et) S (O) CH2CH = CH2                   Hex-c
CH (Et) S (O) CH2CH = CH2                   CH2Pr-c
CH (Et) S (O) CH2CH = CH2                   CH2Bu-c
CH (Et) S (O) CH2CH = CH2                   CH2Pen-c
CH (Et) S (O) CH2CH = CH2                   CH2Hex-c
CH (Et) S (O) CH2CH = CH2                   CH2CH = CH2
CH (Et) S (O) CH2CH = CH2                   CH2CH = C (Cl)2
CH (Et) S (O) CH2CH = CH2                   CH2C≡CH
CH (Et) S (O) CH2CH = CH2                   CH2CN
CH (Et) S (O) CH2CH = CH2                   CH2CFThree
CH (Et) S (O) CH2CH = CH2                   CH2OMe
CH (Et) S (O) CH2CH = CH2                   CH2OCFThree
CH (Et) S (O) CH2CH = CH2                   CH2SMe
CH (Et) S (O) CH2CH = CH2                   CH2S (O) Me
CH (Et) S (O) CH2CH = CH2                   CH2S (O)2Me
CH (Et) S (O) CH2CH = CH2                   CH2SCFThree
CH (Et) S (O) CH2CH = CH2                   CH2S (O) CFThree
CH (Et) S (O) CH2CH = CH2                   CH2S (O)2CFThree
CH (Et) S (O) CH2CH = CH2                   CH2CH (OMe)2
CH (Et) S (O) CH2CH = CH2                   CH2CH (SMe)2
CH (Et) S (O) CH2CH = CH2                   CH2C (O) Me
CH (Et) S (O) CH2CH = CH2                   CH2C (O) CFThree
CH (Et) S (O) CH2CH = CH2                   CH2C (O) OMe
CH (Et) S (O) CH2CH = CH2                   CH2(D1-32a)
CH (Et) S (O) CH2CH = CH2                   CH2(D1-33a)
CH (Et) S (O) CH2CH = CH2                   CH2(D1-34a)
CH (Et) S (O) CH2CH = CH2                   CH2(D1-37a)
CH (Et) S (O) CH2CH = CH2                   CH2(D1-81a)
CH (Et) S (O) CH2CH = CH2                   CH2(D1-82a)
CH (Et) S (O) CH2CH = CH2                   CH2(D1-84a)
CH (Et) S (O) CH2CH = CH2                   CH2(D1-85a)
CH (Et) S (O) CH2CH = CH2                   CH2(D1-87a)
CH (Et) S (O) CH2CH = CH2                   CH2(D1-92a)
CH (Et) S (O) CH2CH = CH2                   CH2(D1-93a)
CH (Et) S (O) CH2CH = CH2                   CH2(D1-95a)
CH (Et) S (O) CH2CH = CH2                   CH2(D1-96a)
CH (Et) S (O) CH2CH = CH2                   CH2(D1-98a)
CH (Et) S (O) CH2CH = CH2                   CH2(D1-108a)
CH (Et) S (O) CH2CH = CH2                   CH2(D1-108b, Z = 2-Cl)
CH (Et) S (O) CH2CH = CH2                   CH2(D1-108b, Z = 3-Me)
CH (Et) S (O) CH2CH = CH2                   CH2(D1-108b, Z = 4-OMe)
CH (Et) S (O) CH2CH = CH2                   CH2(D1-108b, Z = 2-SMe)
CH (Et) S (O) CH2CH = CH2                   CH2(D1-108b, Z = 3-CFThree)
CH (Et) S (O) CH2CH = CH2                   CH2(D1-108b, Z = 4-OCFThree)
CH (Et) S (O) CH2CH = CH2                   CH2(D1-108b, Z = 2-SCFThree)
CH (Et) S (O) CH2CH = CH2                   CH2CH2CN
CH (Et) S (O) CH2CH = CH2                   CH2CH2CFThree
CH (Et) S (O) CH2CH = CH2                   CH2CH2OMe
CH (Et) S (O) CH2CH = CH2                   CH2CH2SMe
CH (Et) S (O) CH2CH = CH2                   CH2CH2S (O) Me
CH (Et) S (O) CH2CH = CH2                   CH2CH2S (O)2Me
CH (Et) S (O) CH2CH = CH2                   D1-32a
CH (Et) S (O) CH2CH = CH2                   D1-33a
CH (Et) S (O) CH2CH = CH2                   D1-34a
CH (Et) S (O) CH2CH = CH2                   D1-37a
CH (Et) S (O) CH2CH = CH2                   D1-81a
CH (Et) S (O) CH2CH = CH2                   D1-82a
CH (Et) S (O) CH2CH = CH2                   D1-84a
CH (Et) S (O) CH2CH = CH2                   D1-85a
CH (Et) S (O) CH2CH = CH2                   D1-87a
CH (Et) S (O) CH2CH = CH2                   D1-92a
CH (Et) S (O) CH2CH = CH2                   D1-93a
CH (Et) S (O) CH2CH = CH2                   D1-95a
CH (Et) S (O) CH2CH = CH2                   D1-96a
CH (Et) S (O) CH2CH = CH2                   D1-98a
CH (Et) S (O) CH2CH = CH2                   D1-108a
CH (Et) S (O) CH2CH = CH2                   D1-108b (Z = 2-Cl)
CH (Et) S (O) CH2CH = CH2                   D1-108b (Z = 3-Me)
CH (Et) S (O) CH2CH = CH2                   D1-108b (Z = 4-OMe)
CH (Et) S (O) CH2CH = CH2                   D1-108b (Z = 2-SMe)
CH (Et) S (O) CH2CH = CH2                   D1-108b (Z = 3-CFThree)
CH (Et) S (O) CH2CH = CH2                   D1-108b (Z = 4-OCFThree)
CH (Et) S (O) CH2CH = CH2                   D1-108b (Z = 2-SCFThree)
CH (Et) S (O) CH2CH = CH2                   C (O) Me
CH (Et) S (O) CH2CH = CH2                   C (O) CFThree
CH (Et) S (O) CH2CH = CH2                   C (O) OMe
CH (Et) S (O)2CH2CH = CH2                   Me
CH (Et) S (O)2CH2CH = CH2                   Et
CH (Et) S (O)2CH2CH = CH2                   Pr-n
CH (Et) S (O)2CH2CH = CH2                   Pr-i
CH (Et) S (O)2CH2CH = CH2                   Pr-c
CH (Et) S (O)2CH2CH = CH2                   Bu-n
CH (Et) S (O)2CH2CH = CH2                   Bu-i
CH (Et) S (O)2CH2CH = CH2                   Bu-c
CH (Et) S (O)2CH2CH = CH2                   Bu-s
CH (Et) S (O)2CH2CH = CH2                   Bu-t
CH (Et) S (O)2CH2CH = CH2                   Pen-n
CH (Et) S (O)2CH2CH = CH2                   Pen-c
CH (Et) S (O)2CH2CH = CH2                   Hex-n
CH (Et) S (O)2CH2CH = CH2                   Hex-c
CH (Et) S (O)2CH2CH = CH2                   CH2Pr-c
CH (Et) S (O)2CH2CH = CH2                   CH2Bu-c
CH (Et) S (O)2CH2CH = CH2                   CH2Pen-c
CH (Et) S (O)2CH2CH = CH2                   CH2Hex-c
CH (Et) S (O)2CH2CH = CH2                   CH2CH = CH2
CH (Et) S (O)2CH2CH = CH2                   CH2CH = C (Cl)2
CH (Et) S (O)2CH2CH = CH2                   CH2C≡CH
CH (Et) S (O)2CH2CH = CH2                   CH2CN
CH (Et) S (O)2CH2CH = CH2                   CH2CFThree
CH (Et) S (O)2CH2CH = CH2                   CH2OMe
CH (Et) S (O)2CH2CH = CH2                   CH2OCFThree
CH (Et) S (O)2CH2CH = CH2                   CH2SMe
CH (Et) S (O)2CH2CH = CH2                   CH2S (O) Me
CH (Et) S (O)2CH2CH = CH2                   CH2S (O)2Me
CH (Et) S (O)2CH2CH = CH2                   CH2SCFThree
CH (Et) S (O)2CH2CH = CH2                   CH2S (O) CFThree
CH (Et) S (O)2CH2CH = CH2                   CH2S (O)2CFThree
CH (Et) S (O)2CH2CH = CH2                   CH2CH (OMe)2
CH (Et) S (O)2CH2CH = CH2                   CH2CH (SMe)2
CH (Et) S (O)2CH2CH = CH2                   CH2C (O) Me
CH (Et) S (O)2CH2CH = CH2                   CH2C (O) CFThree
CH (Et) S (O)2CH2CH = CH2                   CH2C (O) OMe
CH (Et) S (O)2CH2CH = CH2                   CH2(D1-32a)
CH (Et) S (O)2CH2CH = CH2                   CH2(D1-33a)
CH (Et) S (O)2CH2CH = CH2                   CH2(D1-34a)
CH (Et) S (O)2CH2CH = CH2                   CH2(D1-37a)
CH (Et) S (O)2CH2CH = CH2                   CH2(D1-81a)
CH (Et) S (O)2CH2CH = CH2                   CH2(D1-82a)
CH (Et) S (O)2CH2CH = CH2                   CH2(D1-84a)
CH (Et) S (O)2CH2CH = CH2                   CH2(D1-85a)
CH (Et) S (O)2CH2CH = CH2                   CH2(D1-87a)
CH (Et) S (O)2CH2CH = CH2                   CH2(D1-92a)
CH (Et) S (O)2CH2CH = CH2                   CH2(D1-93a)
CH (Et) S (O)2CH2CH = CH2                   CH2(D1-95a)
CH (Et) S (O)2CH2CH = CH2                   CH2(D1-96a)
CH (Et) S (O)2CH2CH = CH2                   CH2(D1-98a)
CH (Et) S (O)2CH2CH = CH2                   CH2(D1-108a)
CH (Et) S (O)2CH2CH = CH2                   CH2(D1-108b, Z = 2-Cl)
CH (Et) S (O)2CH2CH = CH2                   CH2(D1-108b, Z = 3-Me)
CH (Et) S (O)2CH2CH = CH2                   CH2(D1-108b, Z = 4-OMe)
CH (Et) S (O)2CH2CH = CH2                   CH2(D1-108b, Z = 2-SMe)
CH (Et) S (O)2CH2CH = CH2                   CH2(D1-108b, Z = 3-CFThree)
CH (Et) S (O)2CH2CH = CH2                   CH2(D1-108b, Z = 4-OCFThree)
CH (Et) S (O)2CH2CH = CH2                   CH2(D1-108b, Z = 2-SCFThree)
CH (Et) S (O)2CH2CH = CH2                   CH2CH2CN
CH (Et) S (O)2CH2CH = CH2                   CH2CH2CFThree
CH (Et) S (O)2CH2CH = CH2                   CH2CH2OMe
CH (Et) S (O)2CH2CH = CH2                   CH2CH2SMe
CH (Et) S (O)2CH2CH = CH2                   CH2CH2S (O) Me
CH (Et) S (O)2CH2CH = CH2                   CH2CH2S (O)2Me
CH (Et) S (O)2CH2CH = CH2                   D1-32a
CH (Et) S (O)2CH2CH = CH2                   D1-33a
CH (Et) S (O)2CH2CH = CH2                   D1-34a
CH (Et) S (O)2CH2CH = CH2                   D1-37a
CH (Et) S (O)2CH2CH = CH2                   D1-81a
CH (Et) S (O)2CH2CH = CH2                   D1-82a
CH (Et) S (O)2CH2CH = CH2                   D1-84a
CH (Et) S (O)2CH2CH = CH2                   D1-85a
CH (Et) S (O)2CH2CH = CH2                   D1-87a
CH (Et) S (O)2CH2CH = CH2                   D1-92a
CH (Et) S (O)2CH2CH = CH2                   D1-93a
CH (Et) S (O)2CH2CH = CH2                   D1-95a
CH (Et) S (O)2CH2CH = CH2                   D1-96a
CH (Et) S (O)2CH2CH = CH2                   D1-98a
CH (Et) S (O)2CH2CH = CH2                   D1-108a
CH (Et) S (O)2CH2CH = CH2                   D1-108b (Z = 2-Cl)
CH (Et) S (O)2CH2CH = CH2                   D1-108b (Z = 3-Me)
CH (Et) S (O)2CH2CH = CH2                   D1-108b (Z = 4-OMe)
CH (Et) S (O)2CH2CH = CH2                   D1-108b (Z = 2-SMe)
CH (Et) S (O)2CH2CH = CH2                   D1-108b (Z = 3-CFThree)
CH (Et) S (O)2CH2CH = CH2                   D1-108b (Z = 4-OCFThree)
CH (Et) S (O)2CH2CH = CH2                   D1-108b (Z = 2-SCFThree)
CH (Et) S (O)2CH2CH = CH2                   C (O) Me
CH (Et) S (O)2CH2CH = CH2                   C (O) CFThree
CH (Et) S (O)2CH2CH = CH2                   C (O) OMe
CH2SCH2CH2OMe Me
CH2SCH2CH2OMe Et
CH2SCH2CH2OMe Pr-n
CH2SCH2CH2OMe Pr-i
CH2SCH2CH2OMe Pr-c
CH2SCH2CH2OMe Bu-n
CH2SCH2CH2OMe Bu-i
CH2SCH2CH2OMe Bu-c
CH2SCH2CH2OMe Bu-s
CH2SCH2CH2OMe Bu-t
CH2SCH2CH2OMe Pen-n
CH2SCH2CH2OMe Pen-c
CH2SCH2CH2OMe Hex-n
CH2SCH2CH2OMe Hex-c
CH2SCH2CH2OMe CH2Pr-c
CH2SCH2CH2OMe CH2Bu-c
CH2SCH2CH2OMe CH2Pen-c
CH2SCH2CH2OMe CH2Hex-c
CH2SCH2CH2OMe CH2CH = CH2
CH2SCH2CH2OMe CH2CH = C (Cl)2
CH2SCH2CH2OMe CH2C≡CH
CH2SCH2CH2OMe CH2CN
CH2SCH2CH2OMe CH2CFThree
CH2SCH2CH2OMe CH2OMe
CH2SCH2CH2OMe CH2OCFThree
CH2SCH2CH2OMe CH2SMe
CH2SCH2CH2OMe CH2S (O) Me
CH2SCH2CH2OMe CH2S (O)2Me
CH2SCH2CH2OMe CH2SCFThree
CH2SCH2CH2OMe CH2S (O) CFThree
CH2SCH2CH2OMe CH2S (O)2CFThree
CH2SCH2CH2OMe CH2CH (OMe)2
CH2SCH2CH2OMe CH2CH (SMe)2
CH2SCH2CH2OMe CH2C (O) Me
CH2SCH2CH2OMe CH2C (O) CFThree
CH2SCH2CH2OMe CH2C (O) OMe
CH2SCH2CH2OMe CH2(D1-32a)
CH2SCH2CH2OMe CH2(D1-33a)
CH2SCH2CH2OMe CH2(D1-34a)
CH2SCH2CH2OMe CH2(D1-37a)
CH2SCH2CH2OMe CH2(D1-81a)
CH2SCH2CH2OMe CH2(D1-82a)
CH2SCH2CH2OMe CH2(D1-84a)
CH2SCH2CH2OMe CH2(D1-85a)
CH2SCH2CH2OMe CH2(D1-87a)
CH2SCH2CH2OMe CH2(D1-92a)
CH2SCH2CH2OMe CH2(D1-93a)
CH2SCH2CH2OMe CH2(D1-95a)
CH2SCH2CH2OMe CH2(D1-96a)
CH2SCH2CH2OMe CH2(D1-98a)
CH2SCH2CH2OMe CH2(D1-108a)
CH2SCH2CH2OMe CH2(D1-108b, Z = 2-Cl)
CH2SCH2CH2OMe CH2(D1-108b, Z = 3-Me)
CH2SCH2CH2OMe CH2(D1-108b, Z = 4-OMe)
CH2SCH2CH2OMe CH2(D1-108b, Z = 2-SMe)
CH2SCH2CH2OMe CH2(D1-108b, Z = 3-CFThree)
CH2SCH2CH2OMe CH2(D1-108b, Z = 4-OCFThree)
CH2SCH2CH2OMe CH2(D1-108b, Z = 2-SCFThree)
CH2SCH2CH2OMe CH2CH2CN
CH2SCH2CH2OMe CH2CH2CFThree
CH2SCH2CH2OMe CH2CH2OMe
CH2SCH2CH2OMe CH2CH2SMe
CH2SCH2CH2OMe CH2CH2S (O) Me
CH2SCH2CH2OMe CH2CH2S (O)2Me
CH2SCH2CH2OMe D1-32a
CH2SCH2CH2OMe D1-33a
CH2SCH2CH2OMe D1-34a
CH2SCH2CH2OMe D1-37a
CH2SCH2CH2OMe D1-81a
CH2SCH2CH2OMe D1-82a
CH2SCH2CH2OMe D1-84a
CH2SCH2CH2OMe D1-85a
CH2SCH2CH2OMe D1-87a
CH2SCH2CH2OMe D1-92a
CH2SCH2CH2OMe D1-93a
CH2SCH2CH2OMe D1-95a
CH2SCH2CH2OMe D1-96a
CH2SCH2CH2OMe D1-98a
CH2SCH2CH2OMe D1-108a
CH2SCH2CH2OMe D1-108b (Z = 2-Cl)
CH2SCH2CH2OMe D1-108b (Z = 3-Me)
CH2SCH2CH2OMe D1-108b (Z = 4-OMe)
CH2SCH2CH2OMe D1-108b (Z = 2-SMe)
CH2SCH2CH2OMe D1-108b (Z = 3-CFThree)
CH2SCH2CH2OMe D1-108b (Z = 4-OCFThree)
CH2SCH2CH2OMe D1-108b (Z = 2-SCFThree)
CH2SCH2CH2OMe C (O) Me
CH2SCH2CH2OMe C (O) CFThree
CH2SCH2CH2OMe C (O) OMe
CH2S (O) CH2CH2OMe Me
CH2S (O) CH2CH2OMe Et
CH2S (O) CH2CH2OMe Pr-n
CH2S (O) CH2CH2OMe Pr-i
CH2S (O) CH2CH2OMe Pr-c
CH2S (O) CH2CH2OMe Bu-n
CH2S (O) CH2CH2OMe Bu-i
CH2S (O) CH2CH2OMe Bu-c
CH2S (O) CH2CH2OMe Bu-s
CH2S (O) CH2CH2OMe Bu-t
CH2S (O) CH2CH2OMe Pen-n
CH2S (O) CH2CH2OMe Pen-c
CH2S (O) CH2CH2OMe Hex-n
CH2S (O) CH2CH2OMe Hex-c
CH2S (O) CH2CH2OMe CH2Pr-c
CH2S (O) CH2CH2OMe CH2Bu-c
CH2S (O) CH2CH2OMe CH2Pen-c
CH2S (O) CH2CH2OMe CH2Hex-c
CH2S (O) CH2CH2OMe CH2CH = CH2
CH2S (O) CH2CH2OMe CH2CH = C (Cl)2
CH2S (O) CH2CH2OMe CH2C≡CH
CH2S (O) CH2CH2OMe CH2CN
CH2S (O) CH2CH2OMe CH2CFThree
CH2S (O) CH2CH2OMe CH2OMe
CH2S (O) CH2CH2OMe CH2OCFThree
CH2S (O) CH2CH2OMe CH2SMe
CH2S (O) CH2CH2OMe CH2S (O) Me
CH2S (O) CH2CH2OMe CH2S (O)2Me
CH2S (O) CH2CH2OMe CH2SCFThree
CH2S (O) CH2CH2OMe CH2S (O) CFThree
CH2S (O) CH2CH2OMe CH2S (O)2CFThree
CH2S (O) CH2CH2OMe CH2CH (OMe)2
CH2S (O) CH2CH2OMe CH2CH (SMe)2
CH2S (O) CH2CH2OMe CH2C (O) Me
CH2S (O) CH2CH2OMe CH2C (O) CFThree
CH2S (O) CH2CH2OMe CH2C (O) OMe
CH2S (O) CH2CH2OMe CH2(D1-32a)
CH2S (O) CH2CH2OMe CH2(D1-33a)
CH2S (O) CH2CH2OMe CH2(D1-34a)
CH2S (O) CH2CH2OMe CH2(D1-37a)
CH2S (O) CH2CH2OMe CH2(D1-81a)
CH2S (O) CH2CH2OMe CH2(D1-82a)
CH2S (O) CH2CH2OMe CH2(D1-84a)
CH2S (O) CH2CH2OMe CH2(D1-85a)
CH2S (O) CH2CH2OMe CH2(D1-87a)
CH2S (O) CH2CH2OMe CH2(D1-92a)
CH2S (O) CH2CH2OMe CH2(D1-93a)
CH2S (O) CH2CH2OMe CH2(D1-95a)
CH2S (O) CH2CH2OMe CH2(D1-96a)
CH2S (O) CH2CH2OMe CH2(D1-98a)
CH2S (O) CH2CH2OMe CH2(D1-108a)
CH2S (O) CH2CH2OMe CH2(D1-108b, Z = 2-Cl)
CH2S (O) CH2CH2OMe CH2(D1-108b, Z = 3-Me)
CH2S (O) CH2CH2OMe CH2(D1-108b, Z = 4-OMe)
CH2S (O) CH2CH2OMe CH2(D1-108b, Z = 2-SMe)
CH2S (O) CH2CH2OMe CH2(D1-108b, Z = 3-CFThree)
CH2S (O) CH2CH2OMe CH2(D1-108b, Z = 4-OCFThree)
CH2S (O) CH2CH2OMe CH2(D1-108b, Z = 2-SCFThree)
CH2S (O) CH2CH2OMe CH2CH2CN
CH2S (O) CH2CH2OMe CH2CH2CFThree
CH2S (O) CH2CH2OMe CH2CH2OMe
CH2S (O) CH2CH2OMe CH2CH2SMe
CH2S (O) CH2CH2OMe CH2CH2S (O) Me
CH2S (O) CH2CH2OMe CH2CH2S (O)2Me
CH2S (O) CH2CH2OMe D1-32a
CH2S (O) CH2CH2OMe D1-33a
CH2S (O) CH2CH2OMe D1-34a
CH2S (O) CH2CH2OMe D1-37a
CH2S (O) CH2CH2OMe D1-81a
CH2S (O) CH2CH2OMe D1-82a
CH2S (O) CH2CH2OMe D1-84a
CH2S (O) CH2CH2OMe D1-85a
CH2S (O) CH2CH2OMe D1-87a
CH2S (O) CH2CH2OMe D1-92a
CH2S (O) CH2CH2OMe D1-93a
CH2S (O) CH2CH2OMe D1-95a
CH2S (O) CH2CH2OMe D1-96a
CH2S (O) CH2CH2OMe D1-98a
CH2S (O) CH2CH2OMe D1-108a
CH2S (O) CH2CH2OMe D1-108b (Z = 2-Cl)
CH2S (O) CH2CH2OMe D1-108b (Z = 3-Me)
CH2S (O) CH2CH2OMe D1-108b (Z = 4-OMe)
CH2S (O) CH2CH2OMe D1-108b (Z = 2-SMe)
CH2S (O) CH2CH2OMe D1-108b (Z = 3-CFThree)
CH2S (O) CH2CH2OMe D1-108b (Z = 4-OCFThree)
CH2S (O) CH2CH2OMe D1-108b (Z = 2-SCFThree)
CH2S (O) CH2CH2OMe C (O) Me
CH2S (O) CH2CH2OMe C (O) CFThree
CH2S (O) CH2CH2OMe C (O) OMe
CH2S (O)2CH2CH2OMe Me
CH2S (O)2CH2CH2OMe Et
CH2S (O)2CH2CH2OMe Pr-n
CH2S (O)2CH2CH2OMe Pr-i
CH2S (O)2CH2CH2OMe Pr-c
CH2S (O)2CH2CH2OMe Bu-n
CH2S (O)2CH2CH2OMe Bu-i
CH2S (O)2CH2CH2OMe Bu-c
CH2S (O)2CH2CH2OMe Bu-s
CH2S (O)2CH2CH2OMe Bu-t
CH2S (O)2CH2CH2OMe Pen-n
CH2S (O)2CH2CH2OMe Pen-c
CH2S (O)2CH2CH2OMe Hex-n
CH2S (O)2CH2CH2OMe Hex-c
CH2S (O)2CH2CH2OMe CH2Pr-c
CH2S (O)2CH2CH2OMe CH2Bu-c
CH2S (O)2CH2CH2OMe CH2Pen-c
CH2S (O)2CH2CH2OMe CH2Hex-c
CH2S (O)2CH2CH2OMe CH2CH = CH2
CH2S (O)2CH2CH2OMe CH2CH = C (Cl)2
CH2S (O)2CH2CH2OMe CH2C≡CH
CH2S (O)2CH2CH2OMe CH2CN
CH2S (O)2CH2CH2OMe CH2CFThree
CH2S (O)2CH2CH2OMe CH2OMe
CH2S (O)2CH2CH2OMe CH2OCFThree
CH2S (O)2CH2CH2OMe CH2SMe
CH2S (O)2CH2CH2OMe CH2S (O) Me
CH2S (O)2CH2CH2OMe CH2S (O)2Me
CH2S (O)2CH2CH2OMe CH2SCFThree
CH2S (O)2CH2CH2OMe CH2S (O) CFThree
CH2S (O)2CH2CH2OMe CH2S (O)2CFThree
CH2S (O)2CH2CH2OMe CH2CH (OMe)2
CH2S (O)2CH2CH2OMe CH2CH (SMe)2
CH2S (O)2CH2CH2OMe CH2C (O) Me
CH2S (O)2CH2CH2OMe CH2C (O) CFThree
CH2S (O)2CH2CH2OMe CH2C (O) OMe
CH2S (O)2CH2CH2OMe CH2(D1-32a)
CH2S (O)2CH2CH2OMe CH2(D1-33a)
CH2S (O)2CH2CH2OMe CH2(D1-34a)
CH2S (O)2CH2CH2OMe CH2(D1-37a)
CH2S (O)2CH2CH2OMe CH2(D1-81a)
CH2S (O)2CH2CH2OMe CH2(D1-82a)
CH2S (O)2CH2CH2OMe CH2(D1-84a)
CH2S (O)2CH2CH2OMe CH2(D1-85a)
CH2S (O)2CH2CH2OMe CH2(D1-87a)
CH2S (O)2CH2CH2OMe CH2(D1-92a)
CH2S (O)2CH2CH2OMe CH2(D1-93a)
CH2S (O)2CH2CH2OMe CH2(D1-95a)
CH2S (O)2CH2CH2OMe CH2(D1-96a)
CH2S (O)2CH2CH2OMe CH2(D1-98a)
CH2S (O)2CH2CH2OMe CH2(D1-108a)
CH2S (O)2CH2CH2OMe CH2(D1-108b, Z = 2-Cl)
CH2S (O)2CH2CH2OMe CH2(D1-108b, Z = 3-Me)
CH2S (O)2CH2CH2OMe CH2(D1-108b, Z = 4-OMe)
CH2S (O)2CH2CH2OMe CH2(D1-108b, Z = 2-SMe)
CH2S (O)2CH2CH2OMe CH2(D1-108b, Z = 3-CFThree)
CH2S (O)2CH2CH2OMe CH2(D1-108b, Z = 4-OCFThree)
CH2S (O)2CH2CH2OMe CH2(D1-108b, Z = 2-SCFThree)
CH2S (O)2CH2CH2OMe CH2CH2CN
CH2S (O)2CH2CH2OMe CH2CH2CFThree
CH2S (O)2CH2CH2OMe CH2CH2OMe
CH2S (O)2CH2CH2OMe CH2CH2SMe
CH2S (O)2CH2CH2OMe CH2CH2S (O) Me
CH2S (O)2CH2CH2OMe CH2CH2S (O)2Me
CH2S (O)2CH2CH2OMe D1-32a
CH2S (O)2CH2CH2OMe D1-33a
CH2S (O)2CH2CH2OMe D1-34a
CH2S (O)2CH2CH2OMe D1-37a
CH2S (O)2CH2CH2OMe D1-81a
CH2S (O)2CH2CH2OMe D1-82a
CH2S (O)2CH2CH2OMe D1-84a
CH2S (O)2CH2CH2OMe D1-85a
CH2S (O)2CH2CH2OMe D1-87a
CH2S (O)2CH2CH2OMe D1-92a
CH2S (O)2CH2CH2OMe D1-93a
CH2S (O)2CH2CH2OMe D1-95a
CH2S (O)2CH2CH2OMe D1-96a
CH2S (O)2CH2CH2OMe D1-98a
CH2S (O)2CH2CH2OMe D1-108a
CH2S (O)2CH2CH2OMe D1-108b (Z = 2-Cl)
CH2S (O)2CH2CH2OMe D1-108b (Z = 3-Me)
CH2S (O)2CH2CH2OMe D1-108b (Z = 4-OMe)
CH2S (O)2CH2CH2OMe D1-108b (Z = 2-SMe)
CH2S (O)2CH2CH2OMe D1-108b (Z = 3-CFThree)
CH2S (O)2CH2CH2OMe D1-108b (Z = 4-OCFThree)
CH2S (O)2CH2CH2OMe D1-108b (Z = 2-SCFThree)
CH2S (O)2CH2CH2OMe C (O) Me
CH2S (O)2CH2CH2OMe C (O) CFThree
CH2S (O)2CH2CH2OMe C (O) OMe
CH (Me) SCH2CH2OMe Me
CH (Me) SCH2CH2OMe Et
CH (Me) SCH2CH2OMe Pr-n
CH (Me) SCH2CH2OMe Pr-i
CH (Me) SCH2CH2OMe Pr-c
CH (Me) SCH2CH2OMe Bu-n
CH (Me) SCH2CH2OMe Bu-i
CH (Me) SCH2CH2OMe Bu-c
CH (Me) SCH2CH2OMe Bu-s
CH (Me) SCH2CH2OMe Bu-t
CH (Me) SCH2CH2OMe Pen-n
CH (Me) SCH2CH2OMe Pen-c
CH (Me) SCH2CH2OMe Hex-n
CH (Me) SCH2CH2OMe Hex-c
CH (Me) SCH2CH2OMe CH2Pr-c
CH (Me) SCH2CH2OMe CH2Bu-c
CH (Me) SCH2CH2OMe CH2Pen-c
CH (Me) SCH2CH2OMe CH2Hex-c
CH (Me) SCH2CH2OMe CH2CH = CH2
CH (Me) SCH2CH2OMe CH2CH = C (Cl)2
CH (Me) SCH2CH2OMe CH2C≡CH
CH (Me) SCH2CH2OMe CH2CN
CH (Me) SCH2CH2OMe CH2CFThree
CH (Me) SCH2CH2OMe CH2OMe
CH (Me) SCH2CH2OMe CH2OCFThree
CH (Me) SCH2CH2OMe CH2SMe
CH (Me) SCH2CH2OMe CH2S (O) Me
CH (Me) SCH2CH2OMe CH2S (O)2Me
CH (Me) SCH2CH2OMe CH2SCFThree
CH (Me) SCH2CH2OMe CH2S (O) CFThree
CH (Me) SCH2CH2OMe CH2S (O)2CFThree
CH (Me) SCH2CH2OMe CH2CH (OMe)2
CH (Me) SCH2CH2OMe CH2CH (SMe)2
CH (Me) SCH2CH2OMe CH2C (O) Me
CH (Me) SCH2CH2OMe CH2C (O) CFThree
CH (Me) SCH2CH2OMe CH2C (O) OMe
CH (Me) SCH2CH2OMe CH2(D1-32a)
CH (Me) SCH2CH2OMe CH2(D1-33a)
CH (Me) SCH2CH2OMe CH2(D1-34a)
CH (Me) SCH2CH2OMe CH2(D1-37a)
CH (Me) SCH2CH2OMe CH2(D1-81a)
CH (Me) SCH2CH2OMe CH2(D1-82a)
CH (Me) SCH2CH2OMe CH2(D1-84a)
CH (Me) SCH2CH2OMe CH2(D1-85a)
CH (Me) SCH2CH2OMe CH2(D1-87a)
CH (Me) SCH2CH2OMe CH2(D1-92a)
CH (Me) SCH2CH2OMe CH2(D1-93a)
CH (Me) SCH2CH2OMe CH2(D1-95a)
CH (Me) SCH2CH2OMe CH2(D1-96a)
CH (Me) SCH2CH2OMe CH2(D1-98a)
CH (Me) SCH2CH2OMe CH2(D1-108a)
CH (Me) SCH2CH2OMe CH2(D1-108b, Z = 2-Cl)
CH (Me) SCH2CH2OMe CH2(D1-108b, Z = 3-Me)
CH (Me) SCH2CH2OMe CH2(D1-108b, Z = 4-OMe)
CH (Me) SCH2CH2OMe CH2(D1-108b, Z = 2-SMe)
CH (Me) SCH2CH2OMe CH2(D1-108b, Z = 3-CFThree)
CH (Me) SCH2CH2OMe CH2(D1-108b, Z = 4-OCFThree)
CH (Me) SCH2CH2OMe CH2(D1-108b, Z = 2-SCFThree)
CH (Me) SCH2CH2OMe CH2CH2CN
CH (Me) SCH2CH2OMe CH2CH2CFThree
CH (Me) SCH2CH2OMe CH2CH2OMe
CH (Me) SCH2CH2OMe CH2CH2SMe
CH (Me) SCH2CH2OMe CH2CH2S (O) Me
CH (Me) SCH2CH2OMe CH2CH2S (O)2Me
CH (Me) SCH2CH2OMe D1-32a
CH (Me) SCH2CH2OMe D1-33a
CH (Me) SCH2CH2OMe D1-34a
CH (Me) SCH2CH2OMe D1-37a
CH (Me) SCH2CH2OMe D1-81a
CH (Me) SCH2CH2OMe D1-82a
CH (Me) SCH2CH2OMe D1-84a
CH (Me) SCH2CH2OMe D1-85a
CH (Me) SCH2CH2OMe D1-87a
CH (Me) SCH2CH2OMe D1-92a
CH (Me) SCH2CH2OMe D1-93a
CH (Me) SCH2CH2OMe D1-95a
CH (Me) SCH2CH2OMe D1-96a
CH (Me) SCH2CH2OMe D1-98a
CH (Me) SCH2CH2OMe D1-108a
CH (Me) SCH2CH2OMe D1-108b (Z = 2-Cl)
CH (Me) SCH2CH2OMe D1-108b (Z = 3-Me)
CH (Me) SCH2CH2OMe D1-108b (Z = 4-OMe)
CH (Me) SCH2CH2OMe D1-108b (Z = 2-SMe)
CH (Me) SCH2CH2OMe D1-108b (Z = 3-CFThree)
CH (Me) SCH2CH2OMe D1-108b (Z = 4-OCFThree)
CH (Me) SCH2CH2OMe D1-108b (Z = 2-SCFThree)
CH (Me) SCH2CH2OMe C (O) Me
CH (Me) SCH2CH2OMe C (O) CFThree
CH (Me) SCH2CH2OMe C (O) OMe
CH (Me) S (O) CH2CH2OMe Me
CH (Me) S (O) CH2CH2OMe Et
CH (Me) S (O) CH2CH2OMe Pr-n
CH (Me) S (O) CH2CH2OMe Pr-i
CH (Me) S (O) CH2CH2OMe Pr-c
CH (Me) S (O) CH2CH2OMe Bu-n
CH (Me) S (O) CH2CH2OMe Bu-i
CH (Me) S (O) CH2CH2OMe Bu-c
CH (Me) S (O) CH2CH2OMe Bu-s
CH (Me) S (O) CH2CH2OMe Bu-t
CH (Me) S (O) CH2CH2OMe Pen-n
CH (Me) S (O) CH2CH2OMe Pen-c
CH (Me) S (O) CH2CH2OMe Hex-n
CH (Me) S (O) CH2CH2OMe Hex-c
CH (Me) S (O) CH2CH2OMe CH2Pr-c
CH (Me) S (O) CH2CH2OMe CH2Bu-c
CH (Me) S (O) CH2CH2OMe CH2Pen-c
CH (Me) S (O) CH2CH2OMe CH2Hex-c
CH (Me) S (O) CH2CH2OMe CH2CH = CH2
CH (Me) S (O) CH2CH2OMe CH2CH = C (Cl)2
CH (Me) S (O) CH2CH2OMe CH2C≡CH
CH (Me) S (O) CH2CH2OMe CH2CN
CH (Me) S (O) CH2CH2OMe CH2CFThree
CH (Me) S (O) CH2CH2OMe CH2OMe
CH (Me) S (O) CH2CH2OMe CH2OCFThree
CH (Me) S (O) CH2CH2OMe CH2SMe
CH (Me) S (O) CH2CH2OMe CH2S (O) Me
CH (Me) S (O) CH2CH2OMe CH2S (O)2Me
CH (Me) S (O) CH2CH2OMe CH2SCFThree
CH (Me) S (O) CH2CH2OMe CH2S (O) CFThree
CH (Me) S (O) CH2CH2OMe CH2S (O)2CFThree
CH (Me) S (O) CH2CH2OMe CH2CH (OMe)2
CH (Me) S (O) CH2CH2OMe CH2CH (SMe)2
CH (Me) S (O) CH2CH2OMe CH2C (O) Me
CH (Me) S (O) CH2CH2OMe CH2C (O) CFThree
CH (Me) S (O) CH2CH2OMe CH2C (O) OMe
CH (Me) S (O) CH2CH2OMe CH2(D1-32a)
CH (Me) S (O) CH2CH2OMe CH2(D1-33a)
CH (Me) S (O) CH2CH2OMe CH2(D1-34a)
CH (Me) S (O) CH2CH2OMe CH2(D1-37a)
CH (Me) S (O) CH2CH2OMe CH2(D1-81a)
CH (Me) S (O) CH2CH2OMe CH2(D1-82a)
CH (Me) S (O) CH2CH2OMe CH2(D1-84a)
CH (Me) S (O) CH2CH2OMe CH2(D1-85a)
CH (Me) S (O) CH2CH2OMe CH2(D1-87a)
CH (Me) S (O) CH2CH2OMe CH2(D1-92a)
CH (Me) S (O) CH2CH2OMe CH2(D1-93a)
CH (Me) S (O) CH2CH2OMe CH2(D1-95a)
CH (Me) S (O) CH2CH2OMe CH2(D1-96a)
CH (Me) S (O) CH2CH2OMe CH2(D1-98a)
CH (Me) S (O) CH2CH2OMe CH2(D1-108a)
CH (Me) S (O) CH2CH2OMe CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O) CH2CH2OMe CH2(D1-108b, Z = 3-Me)
CH (Me) S (O) CH2CH2OMe CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O) CH2CH2OMe CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O) CH2CH2OMe CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O) CH2CH2OMe CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O) CH2CH2OMe CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O) CH2CH2OMe CH2CH2CN
CH (Me) S (O) CH2CH2OMe CH2CH2CFThree
CH (Me) S (O) CH2CH2OMe CH2CH2OMe
CH (Me) S (O) CH2CH2OMe CH2CH2SMe
CH (Me) S (O) CH2CH2OMe CH2CH2S (O) Me
CH (Me) S (O) CH2CH2OMe CH2CH2S (O)2Me
CH (Me) S (O) CH2CH2OMe D1-32a
CH (Me) S (O) CH2CH2OMe D1-33a
CH (Me) S (O) CH2CH2OMe D1-34a
CH (Me) S (O) CH2CH2OMe D1-37a
CH (Me) S (O) CH2CH2OMe D1-81a
CH (Me) S (O) CH2CH2OMe D1-82a
CH (Me) S (O) CH2CH2OMe D1-84a
CH (Me) S (O) CH2CH2OMe D1-85a
CH (Me) S (O) CH2CH2OMe D1-87a
CH (Me) S (O) CH2CH2OMe D1-92a
CH (Me) S (O) CH2CH2OMe D1-93a
CH (Me) S (O) CH2CH2OMe D1-95a
CH (Me) S (O) CH2CH2OMe D1-96a
CH (Me) S (O) CH2CH2OMe D1-98a
CH (Me) S (O) CH2CH2OMe D1-108a
CH (Me) S (O) CH2CH2OMe D1-108b (Z = 2-Cl)
CH (Me) S (O) CH2CH2OMe D1-108b (Z = 3-Me)
CH (Me) S (O) CH2CH2OMe D1-108b (Z = 4-OMe)
CH (Me) S (O) CH2CH2OMe D1-108b (Z = 2-SMe)
CH (Me) S (O) CH2CH2OMe D1-108b (Z = 3-CFThree)
CH (Me) S (O) CH2CH2OMe D1-108b (Z = 4-OCFThree)
CH (Me) S (O) CH2CH2OMe D1-108b (Z = 2-SCFThree)
CH (Me) S (O) CH2CH2OMe C (O) Me
CH (Me) S (O) CH2CH2OMe C (O) CFThree
CH (Me) S (O) CH2CH2OMe C (O) OMe
CH (Me) S (O)2CH2CH2OMe Me
CH (Me) S (O)2CH2CH2OMe Et
CH (Me) S (O)2CH2CH2OMe Pr-n
CH (Me) S (O)2CH2CH2OMe Pr-i
CH (Me) S (O)2CH2CH2OMe Pr-c
CH (Me) S (O)2CH2CH2OMe Bu-n
CH (Me) S (O)2CH2CH2OMe Bu-i
CH (Me) S (O)2CH2CH2OMe Bu-c
CH (Me) S (O)2CH2CH2OMe Bu-s
CH (Me) S (O)2CH2CH2OMe Bu-t
CH (Me) S (O)2CH2CH2OMe Pen-n
CH (Me) S (O)2CH2CH2OMe Pen-c
CH (Me) S (O)2CH2CH2OMe Hex-n
CH (Me) S (O)2CH2CH2OMe Hex-c
CH (Me) S (O)2CH2CH2OMe CH2Pr-c
CH (Me) S (O)2CH2CH2OMe CH2Bu-c
CH (Me) S (O)2CH2CH2OMe CH2Pen-c
CH (Me) S (O)2CH2CH2OMe CH2Hex-c
CH (Me) S (O)2CH2CH2OMe CH2CH = CH2
CH (Me) S (O)2CH2CH2OMe CH2CH = C (Cl)2
CH (Me) S (O)2CH2CH2OMe CH2C≡CH
CH (Me) S (O)2CH2CH2OMe CH2CN
CH (Me) S (O)2CH2CH2OMe CH2CFThree
CH (Me) S (O)2CH2CH2OMe CH2OMe
CH (Me) S (O)2CH2CH2OMe CH2OCFThree
CH (Me) S (O)2CH2CH2OMe CH2SMe
CH (Me) S (O)2CH2CH2OMe CH2S (O) Me
CH (Me) S (O)2CH2CH2OMe CH2S (O)2Me
CH (Me) S (O)2CH2CH2OMe CH2SCFThree
CH (Me) S (O)2CH2CH2OMe CH2S (O) CFThree
CH (Me) S (O)2CH2CH2OMe CH2S (O)2CFThree
CH (Me) S (O)2CH2CH2OMe CH2CH (OMe)2
CH (Me) S (O)2CH2CH2OMe CH2CH (SMe)2
CH (Me) S (O)2CH2CH2OMe CH2C (O) Me
CH (Me) S (O)2CH2CH2OMe CH2C (O) CFThree
CH (Me) S (O)2CH2CH2OMe CH2C (O) OMe
CH (Me) S (O)2CH2CH2OMe CH2(D1-32a)
CH (Me) S (O)2CH2CH2OMe CH2(D1-33a)
CH (Me) S (O)2CH2CH2OMe CH2(D1-34a)
CH (Me) S (O)2CH2CH2OMe CH2(D1-37a)
CH (Me) S (O)2CH2CH2OMe CH2(D1-81a)
CH (Me) S (O)2CH2CH2OMe CH2(D1-82a)
CH (Me) S (O)2CH2CH2OMe CH2(D1-84a)
CH (Me) S (O)2CH2CH2OMe CH2(D1-85a)
CH (Me) S (O)2CH2CH2OMe CH2(D1-87a)
CH (Me) S (O)2CH2CH2OMe CH2(D1-92a)
CH (Me) S (O)2CH2CH2OMe CH2(D1-93a)
CH (Me) S (O)2CH2CH2OMe CH2(D1-95a)
CH (Me) S (O)2CH2CH2OMe CH2(D1-96a)
CH (Me) S (O)2CH2CH2OMe CH2(D1-98a)
CH (Me) S (O)2CH2CH2OMe CH2(D1-108a)
CH (Me) S (O)2CH2CH2OMe CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O)2CH2CH2OMe CH2(D1-108b, Z = 3-Me)
CH (Me) S (O)2CH2CH2OMe CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O)2CH2CH2OMe CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O)2CH2CH2OMe CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O)2CH2CH2OMe CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O)2CH2CH2OMe CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O)2CH2CH2OMe CH2CH2CN
CH (Me) S (O)2CH2CH2OMe CH2CH2CFThree
CH (Me) S (O)2CH2CH2OMe CH2CH2OMe
CH (Me) S (O)2CH2CH2OMe CH2CH2SMe
CH (Me) S (O)2CH2CH2OMe CH2CH2S (O) Me
CH (Me) S (O)2CH2CH2OMe CH2CH2S (O)2Me
CH (Me) S (O)2CH2CH2OMe D1-32a
CH (Me) S (O)2CH2CH2OMe D1-33a
CH (Me) S (O)2CH2CH2OMe D1-34a
CH (Me) S (O)2CH2CH2OMe D1-37a
CH (Me) S (O)2CH2CH2OMe D1-81a
CH (Me) S (O)2CH2CH2OMe D1-82a
CH (Me) S (O)2CH2CH2OMe D1-84a
CH (Me) S (O)2CH2CH2OMe D1-85a
CH (Me) S (O)2CH2CH2OMe D1-87a
CH (Me) S (O)2CH2CH2OMe D1-92a
CH (Me) S (O)2CH2CH2OMe D1-93a
CH (Me) S (O)2CH2CH2OMe D1-95a
CH (Me) S (O)2CH2CH2OMe D1-96a
CH (Me) S (O)2CH2CH2OMe D1-98a
CH (Me) S (O)2CH2CH2OMe D1-108a
CH (Me) S (O)2CH2CH2OMe D1-108b (Z = 2-Cl)
CH (Me) S (O)2CH2CH2OMe D1-108b (Z = 3-Me)
CH (Me) S (O)2CH2CH2OMe D1-108b (Z = 4-OMe)
CH (Me) S (O)2CH2CH2OMe D1-108b (Z = 2-SMe)
CH (Me) S (O)2CH2CH2OMe D1-108b (Z = 3-CFThree)
CH (Me) S (O)2CH2CH2OMe D1-108b (Z = 4-OCFThree)
CH (Me) S (O)2CH2CH2OMe D1-108b (Z = 2-SCFThree)
CH (Me) S (O)2CH2CH2OMe C (O) Me
CH (Me) S (O)2CH2CH2OMe C (O) CFThree
CH (Me) S (O)2CH2CH2OMe C (O) OMe
CH (Et) SCH2CH2OMe Me
CH (Et) SCH2CH2OMe Et
CH (Et) SCH2CH2OMe Pr-n
CH (Et) SCH2CH2OMe Pr-i
CH (Et) SCH2CH2OMe Pr-c
CH (Et) SCH2CH2OMe Bu-n
CH (Et) SCH2CH2OMe Bu-i
CH (Et) SCH2CH2OMe Bu-c
CH (Et) SCH2CH2OMe Bu-s
CH (Et) SCH2CH2OMe Bu-t
CH (Et) SCH2CH2OMe Pen-n
CH (Et) SCH2CH2OMe Pen-c
CH (Et) SCH2CH2OMe Hex-n
CH (Et) SCH2CH2OMe Hex-c
CH (Et) SCH2CH2OMe CH2Pr-c
CH (Et) SCH2CH2OMe CH2Bu-c
CH (Et) SCH2CH2OMe CH2Pen-c
CH (Et) SCH2CH2OMe CH2Hex-c
CH (Et) SCH2CH2OMe CH2CH = CH2
CH (Et) SCH2CH2OMe CH2CH = C (Cl)2
CH (Et) SCH2CH2OMe CH2C≡CH
CH (Et) SCH2CH2OMe CH2CN
CH (Et) SCH2CH2OMe CH2CFThree
CH (Et) SCH2CH2OMe CH2OMe
CH (Et) SCH2CH2OMe CH2OCFThree
CH (Et) SCH2CH2OMe CH2SMe
CH (Et) SCH2CH2OMe CH2S (O) Me
CH (Et) SCH2CH2OMe CH2S (O)2Me
CH (Et) SCH2CH2OMe CH2SCFThree
CH (Et) SCH2CH2OMe CH2S (O) CFThree
CH (Et) SCH2CH2OMe CH2S (O)2CFThree
CH (Et) SCH2CH2OMe CH2CH (OMe)2
CH (Et) SCH2CH2OMe CH2CH (SMe)2
CH (Et) SCH2CH2OMe CH2C (O) Me
CH (Et) SCH2CH2OMe CH2C (O) CFThree
CH (Et) SCH2CH2OMe CH2C (O) OMe
CH (Et) SCH2CH2OMe CH2(D1-32a)
CH (Et) SCH2CH2OMe CH2(D1-33a)
CH (Et) SCH2CH2OMe CH2(D1-34a)
CH (Et) SCH2CH2OMe CH2(D1-37a)
CH (Et) SCH2CH2OMe CH2(D1-81a)
CH (Et) SCH2CH2OMe CH2(D1-82a)
CH (Et) SCH2CH2OMe CH2(D1-84a)
CH (Et) SCH2CH2OMe CH2(D1-85a)
CH (Et) SCH2CH2OMe CH2(D1-87a)
CH (Et) SCH2CH2OMe CH2(D1-92a)
CH (Et) SCH2CH2OMe CH2(D1-93a)
CH (Et) SCH2CH2OMe CH2(D1-95a)
CH (Et) SCH2CH2OMe CH2(D1-96a)
CH (Et) SCH2CH2OMe CH2(D1-98a)
CH (Et) SCH2CH2OMe CH2(D1-108a)
CH (Et) SCH2CH2OMe CH2(D1-108b, Z = 2-Cl)
CH (Et) SCH2CH2OMe CH2(D1-108b, Z = 3-Me)
CH (Et) SCH2CH2OMe CH2(D1-108b, Z = 4-OMe)
CH (Et) SCH2CH2OMe CH2(D1-108b, Z = 2-SMe)
CH (Et) SCH2CH2OMe CH2(D1-108b, Z = 3-CFThree)
CH (Et) SCH2CH2OMe CH2(D1-108b, Z = 4-OCFThree)
CH (Et) SCH2CH2OMe CH2(D1-108b, Z = 2-SCFThree)
CH (Et) SCH2CH2OMe CH2CH2CN
CH (Et) SCH2CH2OMe CH2CH2CFThree
CH (Et) SCH2CH2OMe CH2CH2OMe
CH (Et) SCH2CH2OMe CH2CH2SMe
CH (Et) SCH2CH2OMe CH2CH2S (O) Me
CH (Et) SCH2CH2OMe CH2CH2S (O)2Me
CH (Et) SCH2CH2OMe D1-32a
CH (Et) SCH2CH2OMe D1-33a
CH (Et) SCH2CH2OMe D1-34a
CH (Et) SCH2CH2OMe D1-37a
CH (Et) SCH2CH2OMe D1-81a
CH (Et) SCH2CH2OMe D1-82a
CH (Et) SCH2CH2OMe D1-84a
CH (Et) SCH2CH2OMe D1-85a
CH (Et) SCH2CH2OMe D1-87a
CH (Et) SCH2CH2OMe D1-92a
CH (Et) SCH2CH2OMe D1-93a
CH (Et) SCH2CH2OMe D1-95a
CH (Et) SCH2CH2OMe D1-96a
CH (Et) SCH2CH2OMe D1-98a
CH (Et) SCH2CH2OMe D1-108a
CH (Et) SCH2CH2OMe D1-108b (Z = 2-Cl)
CH (Et) SCH2CH2OMe D1-108b (Z = 3-Me)
CH (Et) SCH2CH2OMe D1-108b (Z = 4-OMe)
CH (Et) SCH2CH2OMe D1-108b (Z = 2-SMe)
CH (Et) SCH2CH2OMe D1-108b (Z = 3-CFThree)
CH (Et) SCH2CH2OMe D1-108b (Z = 4-OCFThree)
CH (Et) SCH2CH2OMe D1-108b (Z = 2-SCFThree)
CH (Et) SCH2CH2OMe C (O) Me
CH (Et) SCH2CH2OMe C (O) CFThree
CH (Et) SCH2CH2OMe C (O) OMe
CH (Et) S (O) CH2CH2OMe Me
CH (Et) S (O) CH2CH2OMe Et
CH (Et) S (O) CH2CH2OMe Pr-n
CH (Et) S (O) CH2CH2OMe Pr-i
CH (Et) S (O) CH2CH2OMe Pr-c
CH (Et) S (O) CH2CH2OMe Bu-n
CH (Et) S (O) CH2CH2OMe Bu-i
CH (Et) S (O) CH2CH2OMe Bu-c
CH (Et) S (O) CH2CH2OMe Bu-s
CH (Et) S (O) CH2CH2OMe Bu-t
CH (Et) S (O) CH2CH2OMe Pen-n
CH (Et) S (O) CH2CH2OMe Pen-c
CH (Et) S (O) CH2CH2OMe Hex-n
CH (Et) S (O) CH2CH2OMe Hex-c
CH (Et) S (O) CH2CH2OMe CH2Pr-c
CH (Et) S (O) CH2CH2OMe CH2Bu-c
CH (Et) S (O) CH2CH2OMe CH2Pen-c
CH (Et) S (O) CH2CH2OMe CH2Hex-c
CH (Et) S (O) CH2CH2OMe CH2CH = CH2
CH (Et) S (O) CH2CH2OMe CH2CH = C (Cl)2
CH (Et) S (O) CH2CH2OMe CH2C≡CH
CH (Et) S (O) CH2CH2OMe CH2CN
CH (Et) S (O) CH2CH2OMe CH2CFThree
CH (Et) S (O) CH2CH2OMe CH2OMe
CH (Et) S (O) CH2CH2OMe CH2OCFThree
CH (Et) S (O) CH2CH2OMe CH2SMe
CH (Et) S (O) CH2CH2OMe CH2S (O) Me
CH (Et) S (O) CH2CH2OMe CH2S (O)2Me
CH (Et) S (O) CH2CH2OMe CH2SCFThree
CH (Et) S (O) CH2CH2OMe CH2S (O) CFThree
CH (Et) S (O) CH2CH2OMe CH2S (O)2CFThree
CH (Et) S (O) CH2CH2OMe CH2CH (OMe)2
CH (Et) S (O) CH2CH2OMe CH2CH (SMe)2
CH (Et) S (O) CH2CH2OMe CH2C (O) Me
CH (Et) S (O) CH2CH2OMe CH2C (O) CFThree
CH (Et) S (O) CH2CH2OMe CH2C (O) OMe
CH (Et) S (O) CH2CH2OMe CH2(D1-32a)
CH (Et) S (O) CH2CH2OMe CH2(D1-33a)
CH (Et) S (O) CH2CH2OMe CH2(D1-34a)
CH (Et) S (O) CH2CH2OMe CH2(D1-37a)
CH (Et) S (O) CH2CH2OMe CH2(D1-81a)
CH (Et) S (O) CH2CH2OMe CH2(D1-82a)
CH (Et) S (O) CH2CH2OMe CH2(D1-84a)
CH (Et) S (O) CH2CH2OMe CH2(D1-85a)
CH (Et) S (O) CH2CH2OMe CH2(D1-87a)
CH (Et) S (O) CH2CH2OMe CH2(D1-92a)
CH (Et) S (O) CH2CH2OMe CH2(D1-93a)
CH (Et) S (O) CH2CH2OMe CH2(D1-95a)
CH (Et) S (O) CH2CH2OMe CH2(D1-96a)
CH (Et) S (O) CH2CH2OMe CH2(D1-98a)
CH (Et) S (O) CH2CH2OMe CH2(D1-108a)
CH (Et) S (O) CH2CH2OMe CH2(D1-108b, Z = 2-Cl)
CH (Et) S (O) CH2CH2OMe CH2(D1-108b, Z = 3-Me)
CH (Et) S (O) CH2CH2OMe CH2(D1-108b, Z = 4-OMe)
CH (Et) S (O) CH2CH2OMe CH2(D1-108b, Z = 2-SMe)
CH (Et) S (O) CH2CH2OMe CH2(D1-108b, Z = 3-CFThree)
CH (Et) S (O) CH2CH2OMe CH2(D1-108b, Z = 4-OCFThree)
CH (Et) S (O) CH2CH2OMe CH2(D1-108b, Z = 2-SCFThree)
CH (Et) S (O) CH2CH2OMe CH2CH2CN
CH (Et) S (O) CH2CH2OMe CH2CH2CFThree
CH (Et) S (O) CH2CH2OMe CH2CH2OMe
CH (Et) S (O) CH2CH2OMe CH2CH2SMe
CH (Et) S (O) CH2CH2OMe CH2CH2S (O) Me
CH (Et) S (O) CH2CH2OMe CH2CH2S (O)2Me
CH (Et) S (O) CH2CH2OMe D1-32a
CH (Et) S (O) CH2CH2OMe D1-33a
CH (Et) S (O) CH2CH2OMe D1-34a
CH (Et) S (O) CH2CH2OMe D1-37a
CH (Et) S (O) CH2CH2OMe D1-81a
CH (Et) S (O) CH2CH2OMe D1-82a
CH (Et) S (O) CH2CH2OMe D1-84a
CH (Et) S (O) CH2CH2OMe D1-85a
CH (Et) S (O) CH2CH2OMe D1-87a
CH (Et) S (O) CH2CH2OMe D1-92a
CH (Et) S (O) CH2CH2OMe D1-93a
CH (Et) S (O) CH2CH2OMe D1-95a
CH (Et) S (O) CH2CH2OMe D1-96a
CH (Et) S (O) CH2CH2OMe D1-98a
CH (Et) S (O) CH2CH2OMe D1-108a
CH (Et) S (O) CH2CH2OMe D1-108b (Z = 2-Cl)
CH (Et) S (O) CH2CH2OMe D1-108b (Z = 3-Me)
CH (Et) S (O) CH2CH2OMe D1-108b (Z = 4-OMe)
CH (Et) S (O) CH2CH2OMe D1-108b (Z = 2-SMe)
CH (Et) S (O) CH2CH2OMe D1-108b (Z = 3-CFThree)
CH (Et) S (O) CH2CH2OMe D1-108b (Z = 4-OCFThree)
CH (Et) S (O) CH2CH2OMe D1-108b (Z = 2-SCFThree)
CH (Et) S (O) CH2CH2OMe C (O) Me
CH (Et) S (O) CH2CH2OMe C (O) CFThree
CH (Et) S (O) CH2CH2OMe C (O) OMe
CH (Et) S (O)2CH2CH2OMe Me
CH (Et) S (O)2CH2CH2OMe Et
CH (Et) S (O)2CH2CH2OMe Pr-n
CH (Et) S (O)2CH2CH2OMe Pr-i
CH (Et) S (O)2CH2CH2OMe Pr-c
CH (Et) S (O)2CH2CH2OMe Bu-n
CH (Et) S (O)2CH2CH2OMe Bu-i
CH (Et) S (O)2CH2CH2OMe Bu-c
CH (Et) S (O)2CH2CH2OMe Bu-s
CH (Et) S (O)2CH2CH2OMe Bu-t
CH (Et) S (O)2CH2CH2OMe Pen-n
CH (Et) S (O)2CH2CH2OMe Pen-c
CH (Et) S (O)2CH2CH2OMe Hex-n
CH (Et) S (O)2CH2CH2OMe Hex-c
CH (Et) S (O)2CH2CH2OMe CH2Pr-c
CH (Et) S (O)2CH2CH2OMe CH2Bu-c
CH (Et) S (O)2CH2CH2OMe CH2Pen-c
CH (Et) S (O)2CH2CH2OMe CH2Hex-c
CH (Et) S (O)2CH2CH2OMe CH2CH = CH2
CH (Et) S (O)2CH2CH2OMe CH2CH = C (Cl)2
CH (Et) S (O)2CH2CH2OMe CH2C≡CH
CH (Et) S (O)2CH2CH2OMe CH2CN
CH (Et) S (O)2CH2CH2OMe CH2CFThree
CH (Et) S (O)2CH2CH2OMe CH2OMe
CH (Et) S (O)2CH2CH2OMe CH2OCFThree
CH (Et) S (O)2CH2CH2OMe CH2SMe
CH (Et) S (O)2CH2CH2OMe CH2S (O) Me
CH (Et) S (O)2CH2CH2OMe CH2S (O)2Me
CH (Et) S (O)2CH2CH2OMe CH2SCFThree
CH (Et) S (O)2CH2CH2OMe CH2S (O) CFThree
CH (Et) S (O)2CH2CH2OMe CH2S (O)2CFThree
CH (Et) S (O)2CH2CH2OMe CH2CH (OMe)2
CH (Et) S (O)2CH2CH2OMe CH2CH (SMe)2
CH (Et) S (O)2CH2CH2OMe CH2C (O) Me
CH (Et) S (O)2CH2CH2OMe CH2C (O) CFThree
CH (Et) S (O)2CH2CH2OMe CH2C (O) OMe
CH (Et) S (O)2CH2CH2OMe CH2(D1-32a)
CH (Et) S (O)2CH2CH2OMe CH2(D1-33a)
CH (Et) S (O)2CH2CH2OMe CH2(D1-34a)
CH (Et) S (O)2CH2CH2OMe CH2(D1-37a)
CH (Et) S (O)2CH2CH2OMe CH2(D1-81a)
CH (Et) S (O)2CH2CH2OMe CH2(D1-82a)
CH (Et) S (O)2CH2CH2OMe CH2(D1-84a)
CH (Et) S (O)2CH2CH2OMe CH2(D1-85a)
CH (Et) S (O)2CH2CH2OMe CH2(D1-87a)
CH (Et) S (O)2CH2CH2OMe CH2(D1-92a)
CH (Et) S (O)2CH2CH2OMe CH2(D1-93a)
CH (Et) S (O)2CH2CH2OMe CH2(D1-95a)
CH (Et) S (O)2CH2CH2OMe CH2(D1-96a)
CH (Et) S (O)2CH2CH2OMe CH2(D1-98a)
CH (Et) S (O)2CH2CH2OMe CH2(D1-108a)
CH (Et) S (O)2CH2CH2OMe CH2(D1-108b, Z = 2-Cl)
CH (Et) S (O)2CH2CH2OMe CH2(D1-108b, Z = 3-Me)
CH (Et) S (O)2CH2CH2OMe CH2(D1-108b, Z = 4-OMe)
CH (Et) S (O)2CH2CH2OMe CH2(D1-108b, Z = 2-SMe)
CH (Et) S (O)2CH2CH2OMe CH2(D1-108b, Z = 3-CFThree)
CH (Et) S (O)2CH2CH2OMe CH2(D1-108b, Z = 4-OCFThree)
CH (Et) S (O)2CH2CH2OMe CH2(D1-108b, Z = 2-SCFThree)
CH (Et) S (O)2CH2CH2OMe CH2CH2CN
CH (Et) S (O)2CH2CH2OMe CH2CH2CFThree
CH (Et) S (O)2CH2CH2OMe CH2CH2OMe
CH (Et) S (O)2CH2CH2OMe CH2CH2SMe
CH (Et) S (O)2CH2CH2OMe CH2CH2S (O) Me
CH (Et) S (O)2CH2CH2OMe CH2CH2S (O)2Me
CH (Et) S (O)2CH2CH2OMe D1-32a
CH (Et) S (O)2CH2CH2OMe D1-33a
CH (Et) S (O)2CH2CH2OMe D1-34a
CH (Et) S (O)2CH2CH2OMe D1-37a
CH (Et) S (O)2CH2CH2OMe D1-81a
CH (Et) S (O)2CH2CH2OMe D1-82a
CH (Et) S (O)2CH2CH2OMe D1-84a
CH (Et) S (O)2CH2CH2OMe D1-85a
CH (Et) S (O)2CH2CH2OMe D1-87a
CH (Et) S (O)2CH2CH2OMe D1-92a
CH (Et) S (O)2CH2CH2OMe D1-93a
CH (Et) S (O)2CH2CH2OMe D1-95a
CH (Et) S (O)2CH2CH2OMe D1-96a
CH (Et) S (O)2CH2CH2OMe D1-98a
CH (Et) S (O)2CH2CH2OMe D1-108a
CH (Et) S (O)2CH2CH2OMe D1-108b (Z = 2-Cl)
CH (Et) S (O)2CH2CH2OMe D1-108b (Z = 3-Me)
CH (Et) S (O)2CH2CH2OMe D1-108b (Z = 4-OMe)
CH (Et) S (O)2CH2CH2OMe D1-108b (Z = 2-SMe)
CH (Et) S (O)2CH2CH2OMe D1-108b (Z = 3-CFThree)
CH (Et) S (O)2CH2CH2OMe D1-108b (Z = 4-OCFThree)
CH (Et) S (O)2CH2CH2OMe D1-108b (Z = 2-SCFThree)
CH (Et) S (O)2CH2CH2OMe C (O) Me
CH (Et) S (O)2CH2CH2OMe C (O) CFThree
CH (Et) S (O)2CH2CH2OMe C (O) OMe
CH2SCH2CH2OEt Me
CH2SCH2CH2OEt Et
CH2SCH2CH2OEt Pr-n
CH2SCH2CH2OEt Pr-i
CH2SCH2CH2OEt Pr-c
CH2SCH2CH2OEt Bu-n
CH2SCH2CH2OEt Bu-i
CH2SCH2CH2OEt Bu-c
CH2SCH2CH2OEt Bu-s
CH2SCH2CH2OEt Bu-t
CH2SCH2CH2OEt Pen-n
CH2SCH2CH2OEt Pen-c
CH2SCH2CH2OEt Hex-n
CH2SCH2CH2OEt Hex-c
CH2SCH2CH2OEt CH2Pr-c
CH2SCH2CH2OEt CH2Bu-c
CH2SCH2CH2OEt CH2Pen-c
CH2SCH2CH2OEt CH2Hex-c
CH2SCH2CH2OEt CH2CH = CH2
CH2SCH2CH2OEt CH2CH = C (Cl)2
CH2SCH2CH2OEt CH2C≡CH
CH2SCH2CH2OEt CH2CN
CH2SCH2CH2OEt CH2CFThree
CH2SCH2CH2OEt CH2OMe
CH2SCH2CH2OEt CH2OCFThree
CH2SCH2CH2OEt CH2SMe
CH2SCH2CH2OEt CH2S (O) Me
CH2SCH2CH2OEt CH2S (O)2Me
CH2SCH2CH2OEt CH2SCFThree
CH2SCH2CH2OEt CH2S (O) CFThree
CH2SCH2CH2OEt CH2S (O)2CFThree
CH2SCH2CH2OEt CH2CH (OMe)2
CH2SCH2CH2OEt CH2CH (SMe)2
CH2SCH2CH2OEt CH2C (O) Me
CH2SCH2CH2OEt CH2C (O) CFThree
CH2SCH2CH2OEt CH2C (O) OMe
CH2SCH2CH2OEt CH2(D1-32a)
CH2SCH2CH2OEt CH2(D1-33a)
CH2SCH2CH2OEt CH2(D1-34a)
CH2SCH2CH2OEt CH2(D1-37a)
CH2SCH2CH2OEt CH2(D1-81a)
CH2SCH2CH2OEt CH2(D1-82a)
CH2SCH2CH2OEt CH2(D1-84a)
CH2SCH2CH2OEt CH2(D1-85a)
CH2SCH2CH2OEt CH2(D1-87a)
CH2SCH2CH2OEt CH2(D1-92a)
CH2SCH2CH2OEt CH2(D1-93a)
CH2SCH2CH2OEt CH2(D1-95a)
CH2SCH2CH2OEt CH2(D1-96a)
CH2SCH2CH2OEt CH2(D1-98a)
CH2SCH2CH2OEt CH2(D1-108a)
CH2SCH2CH2OEt CH2(D1-108b, Z = 2-Cl)
CH2SCH2CH2OEt CH2(D1-108b, Z = 3-Me)
CH2SCH2CH2OEt CH2(D1-108b, Z = 4-OEt)
CH2SCH2CH2OEt CH2(D1-108b, Z = 2-SMe)
CH2SCH2CH2OEt CH2(D1-108b, Z = 3-CFThree)
CH2SCH2CH2OEt CH2(D1-108b, Z = 4-OCFThree)
CH2SCH2CH2OEt CH2(D1-108b, Z = 2-SCFThree)
CH2SCH2CH2OEt CH2CH2CN
CH2SCH2CH2OEt CH2CH2CFThree
CH2SCH2CH2OEt CH2CH2OEt
CH2SCH2CH2OEt CH2CH2SMe
CH2SCH2CH2OEt CH2CH2S (O) Me
CH2SCH2CH2OEt CH2CH2S (O)2Me
CH2SCH2CH2OEt D1-32a
CH2SCH2CH2OEt D1-33a
CH2SCH2CH2OEt D1-34a
CH2SCH2CH2OEt D1-37a
CH2SCH2CH2OEt D1-81a
CH2SCH2CH2OEt D1-82a
CH2SCH2CH2OEt D1-84a
CH2SCH2CH2OEt D1-85a
CH2SCH2CH2OEt D1-87a
CH2SCH2CH2OEt D1-92a
CH2SCH2CH2OEt D1-93a
CH2SCH2CH2OEt D1-95a
CH2SCH2CH2OEt D1-96a
CH2SCH2CH2OEt D1-98a
CH2SCH2CH2OEt D1-108a
CH2SCH2CH2OEt D1-108b (Z = 2-Cl)
CH2SCH2CH2OEt D1-108b (Z = 3-Me)
CH2SCH2CH2OEt D1-108b (Z = 4-OEt)
CH2SCH2CH2OEt D1-108b (Z = 2-SMe)
CH2SCH2CH2OEt D1-108b (Z = 3-CFThree)
CH2SCH2CH2OEt D1-108b (Z = 4-OCFThree)
CH2SCH2CH2OEt D1-108b (Z = 2-SCFThree)
CH2SCH2CH2OEt C (O) Me
CH2SCH2CH2OEt C (O) CFThree
CH2SCH2CH2OEt C (O) OEt
CH2S (O) CH2CH2OEt Me
CH2S (O) CH2CH2OEt Et
CH2S (O) CH2CH2OEt Pr-n
CH2S (O) CH2CH2OEt Pr-i
CH2S (O) CH2CH2OEt Pr-c
CH2S (O) CH2CH2OEt Bu-n
CH2S (O) CH2CH2OEt Bu-i
CH2S (O) CH2CH2OEt Bu-c
CH2S (O) CH2CH2OEt Bu-s
CH2S (O) CH2CH2OEt Bu-t
CH2S (O) CH2CH2OEt Pen-n
CH2S (O) CH2CH2OEt Pen-c
CH2S (O) CH2CH2OEt Hex-n
CH2S (O) CH2CH2OEt Hex-c
CH2S (O) CH2CH2OEt CH2Pr-c
CH2S (O) CH2CH2OEt CH2Bu-c
CH2S (O) CH2CH2OEt CH2Pen-c
CH2S (O) CH2CH2OEt CH2Hex-c
CH2S (O) CH2CH2OEt CH2CH = CH2
CH2S (O) CH2CH2OEt CH2CH = C (Cl)2
CH2S (O) CH2CH2OEt CH2C≡CH
CH2S (O) CH2CH2OEt CH2CN
CH2S (O) CH2CH2OEt CH2CFThree
CH2S (O) CH2CH2OEt CH2OEt
CH2S (O) CH2CH2OEt CH2OCFThree
CH2S (O) CH2CH2OEt CH2SMe
CH2S (O) CH2CH2OEt CH2S (O) Me
CH2S (O) CH2CH2OEt CH2S (O)2Me
CH2S (O) CH2CH2OEt CH2SCFThree
CH2S (O) CH2CH2OEt CH2S (O) CFThree
CH2S (O) CH2CH2OEt CH2S (O)2CFThree
CH2S (O) CH2CH2OEt CH2CH (OEt)2
CH2S (O) CH2CH2OEt CH2CH (SMe)2
CH2S (O) CH2CH2OEt CH2C (O) Me
CH2S (O) CH2CH2OEt CH2C (O) CFThree
CH2S (O) CH2CH2OEt CH2C (O) OEt
CH2S (O) CH2CH2OEt CH2(D1-32a)
CH2S (O) CH2CH2OEt CH2(D1-33a)
CH2S (O) CH2CH2OEt CH2(D1-34a)
CH2S (O) CH2CH2OEt CH2(D1-37a)
CH2S (O) CH2CH2OEt CH2(D1-81a)
CH2S (O) CH2CH2OEt CH2(D1-82a)
CH2S (O) CH2CH2OEt CH2(D1-84a)
CH2S (O) CH2CH2OEt CH2(D1-85a)
CH2S (O) CH2CH2OEt CH2(D1-87a)
CH2S (O) CH2CH2OEt CH2(D1-92a)
CH2S (O) CH2CH2OEt CH2(D1-93a)
CH2S (O) CH2CH2OEt CH2(D1-95a)
CH2S (O) CH2CH2OEt CH2(D1-96a)
CH2S (O) CH2CH2OEt CH2(D1-98a)
CH2S (O) CH2CH2OEt CH2(D1-108a)
CH2S (O) CH2CH2OEt CH2(D1-108b, Z = 2-Cl)
CH2S (O) CH2CH2OEt CH2(D1-108b, Z = 3-Me)
CH2S (O) CH2CH2OEt CH2(D1-108b, Z = 4-OEt)
CH2S (O) CH2CH2OEt CH2(D1-108b, Z = 2-SMe)
CH2S (O) CH2CH2OEt CH2(D1-108b, Z = 3-CFThree)
CH2S (O) CH2CH2OEt CH2(D1-108b, Z = 4-OCFThree)
CH2S (O) CH2CH2OEt CH2(D1-108b, Z = 2-SCFThree)
CH2S (O) CH2CH2OEt CH2CH2CN
CH2S (O) CH2CH2OEt CH2CH2CFThree
CH2S (O) CH2CH2OEt CH2CH2OEt
CH2S (O) CH2CH2OEt CH2CH2SMe
CH2S (O) CH2CH2OEt CH2CH2S (O) Me
CH2S (O) CH2CH2OEt CH2CH2S (O)2Me
CH2S (O) CH2CH2OEt D1-32a
CH2S (O) CH2CH2OEt D1-33a
CH2S (O) CH2CH2OEt D1-34a
CH2S (O) CH2CH2OEt D1-37a
CH2S (O) CH2CH2OEt D1-81a
CH2S (O) CH2CH2OEt D1-82a
CH2S (O) CH2CH2OEt D1-84a
CH2S (O) CH2CH2OEt D1-85a
CH2S (O) CH2CH2OEt D1-87a
CH2S (O) CH2CH2OEt D1-92a
CH2S (O) CH2CH2OEt D1-93a
CH2S (O) CH2CH2OEt D1-95a
CH2S (O) CH2CH2OEt D1-96a
CH2S (O) CH2CH2OEt D1-98a
CH2S (O) CH2CH2OEt D1-108a
CH2S (O) CH2CH2OEt D1-108b (Z = 2-Cl)
CH2S (O) CH2CH2OEt D1-108b (Z = 3-Me)
CH2S (O) CH2CH2OEt D1-108b (Z = 4-OEt)
CH2S (O) CH2CH2OEt D1-108b (Z = 2-SMe)
CH2S (O) CH2CH2OEt D1-108b (Z = 3-CFThree)
CH2S (O) CH2CH2OEt D1-108b (Z = 4-OCFThree)
CH2S (O) CH2CH2OEt D1-108b (Z = 2-SCFThree)
CH2S (O) CH2CH2OEt C (O) Me
CH2S (O) CH2CH2OEt C (O) CFThree
CH2S (O) CH2CH2OEt C (O) OEt
CH2S (O)2CH2CH2OEt Me
CH2S (O)2CH2CH2OEt Et
CH2S (O)2CH2CH2OEt Pr-n
CH2S (O)2CH2CH2OEt Pr-i
CH2S (O)2CH2CH2OEt Pr-c
CH2S (O)2CH2CH2OEt Bu-n
CH2S (O)2CH2CH2OEt Bu-i
CH2S (O)2CH2CH2OEt Bu-c
CH2S (O)2CH2CH2OEt Bu-s
CH2S (O)2CH2CH2OEt Bu-t
CH2S (O)2CH2CH2OEt Pen-n
CH2S (O)2CH2CH2OEt Pen-c
CH2S (O)2CH2CH2OEt Hex-n
CH2S (O)2CH2CH2OEt Hex-c
CH2S (O)2CH2CH2OEt CH2Pr-c
CH2S (O)2CH2CH2OEt CH2Bu-c
CH2S (O)2CH2CH2OEt CH2Pen-c
CH2S (O)2CH2CH2OEt CH2Hex-c
CH2S (O)2CH2CH2OEt CH2CH = CH2
CH2S (O)2CH2CH2OEt CH2CH = C (Cl)2
CH2S (O)2CH2CH2OEt CH2C≡CH
CH2S (O)2CH2CH2OEt CH2CN
CH2S (O)2CH2CH2OEt CH2CFThree
CH2S (O)2CH2CH2OEt CH2OEt
CH2S (O)2CH2CH2OEt CH2OCFThree
CH2S (O)2CH2CH2OEt CH2SMe
CH2S (O)2CH2CH2OEt CH2S (O) Me
CH2S (O)2CH2CH2OEt CH2S (O)2Me
CH2S (O)2CH2CH2OEt CH2SCFThree
CH2S (O)2CH2CH2OEt CH2S (O) CFThree
CH2S (O)2CH2CH2OEt CH2S (O)2CFThree
CH2S (O)2CH2CH2OEt CH2CH (OEt)2
CH2S (O)2CH2CH2OEt CH2CH (SMe)2
CH2S (O)2CH2CH2OEt CH2C (O) Me
CH2S (O)2CH2CH2OEt CH2C (O) CFThree
CH2S (O)2CH2CH2OEt CH2C (O) OEt
CH2S (O)2CH2CH2OEt CH2(D1-32a)
CH2S (O)2CH2CH2OEt CH2(D1-33a)
CH2S (O)2CH2CH2OEt CH2(D1-34a)
CH2S (O)2CH2CH2OEt CH2(D1-37a)
CH2S (O)2CH2CH2OEt CH2(D1-81a)
CH2S (O)2CH2CH2OEt CH2(D1-82a)
CH2S (O)2CH2CH2OEt CH2(D1-84a)
CH2S (O)2CH2CH2OEt CH2(D1-85a)
CH2S (O)2CH2CH2OEt CH2(D1-87a)
CH2S (O)2CH2CH2OEt CH2(D1-92a)
CH2S (O)2CH2CH2OEt CH2(D1-93a)
CH2S (O)2CH2CH2OEt CH2(D1-95a)
CH2S (O)2CH2CH2OEt CH2(D1-96a)
CH2S (O)2CH2CH2OEt CH2(D1-98a)
CH2S (O)2CH2CH2OEt CH2(D1-108a)
CH2S (O)2CH2CH2OEt CH2(D1-108b, Z = 2-Cl)
CH2S (O)2CH2CH2OEt CH2(D1-108b, Z = 3-Me)
CH2S (O)2CH2CH2OEt CH2(D1-108b, Z = 4-OEt)
CH2S (O)2CH2CH2OEt CH2(D1-108b, Z = 2-SMe)
CH2S (O)2CH2CH2OEt CH2(D1-108b, Z = 3-CFThree)
CH2S (O)2CH2CH2OEt CH2(D1-108b, Z = 4-OCFThree)
CH2S (O)2CH2CH2OEt CH2(D1-108b, Z = 2-SCFThree)
CH2S (O)2CH2CH2OEt CH2CH2CN
CH2S (O)2CH2CH2OEt CH2CH2CFThree
CH2S (O)2CH2CH2OEt CH2CH2OEt
CH2S (O)2CH2CH2OEt CH2CH2SMe
CH2S (O)2CH2CH2OEt CH2CH2S (O) Me
CH2S (O)2CH2CH2OEt CH2CH2S (O)2Me
CH2S (O)2CH2CH2OEt D1-32a
CH2S (O)2CH2CH2OEt D1-33a
CH2S (O)2CH2CH2OEt D1-34a
CH2S (O)2CH2CH2OEt D1-37a
CH2S (O)2CH2CH2OEt D1-81a
CH2S (O)2CH2CH2OEt D1-82a
CH2S (O)2CH2CH2OEt D1-84a
CH2S (O)2CH2CH2OEt D1-85a
CH2S (O)2CH2CH2OEt D1-87a
CH2S (O)2CH2CH2OEt D1-92a
CH2S (O)2CH2CH2OEt D1-93a
CH2S (O)2CH2CH2OEt D1-95a
CH2S (O)2CH2CH2OEt D1-96a
CH2S (O)2CH2CH2OEt D1-98a
CH2S (O)2CH2CH2OEt D1-108a
CH2S (O)2CH2CH2OEt D1-108b (Z = 2-Cl)
CH2S (O)2CH2CH2OEt D1-108b (Z = 3-Me)
CH2S (O)2CH2CH2OEt D1-108b (Z = 4-OEt)
CH2S (O)2CH2CH2OEt D1-108b (Z = 2-SMe)
CH2S (O)2CH2CH2OEt D1-108b (Z = 3-CFThree)
CH2S (O)2CH2CH2OEt D1-108b (Z = 4-OCFThree)
CH2S (O)2CH2CH2OEt D1-108b (Z = 2-SCFThree)
CH2S (O)2CH2CH2OEt C (O) Me
CH2S (O)2CH2CH2OEt C (O) CFThree
CH2S (O)2CH2CH2OEt C (O) OEt
CH (Me) SCH2CH2OEt Me
CH (Me) SCH2CH2OEt Et
CH (Me) SCH2CH2OEt Pr-n
CH (Me) SCH2CH2OEt Pr-i
CH (Me) SCH2CH2OEt Pr-c
CH (Me) SCH2CH2OEt Bu-n
CH (Me) SCH2CH2OEt Bu-i
CH (Me) SCH2CH2OEt Bu-c
CH (Me) SCH2CH2OEt Bu-s
CH (Me) SCH2CH2OEt Bu-t
CH (Me) SCH2CH2OEt Pen-n
CH (Me) SCH2CH2OEt Pen-c
CH (Me) SCH2CH2OEt Hex-n
CH (Me) SCH2CH2OEt Hex-c
CH (Me) SCH2CH2OEt CH2Pr-c
CH (Me) SCH2CH2OEt CH2Bu-c
CH (Me) SCH2CH2OEt CH2Pen-c
CH (Me) SCH2CH2OEt CH2Hex-c
CH (Me) SCH2CH2OEt CH2CH = CH2
CH (Me) SCH2CH2OEt CH2CH = C (Cl)2
CH (Me) SCH2CH2OEt CH2C≡CH
CH (Me) SCH2CH2OEt CH2CN
CH (Me) SCH2CH2OEt CH2CFThree
CH (Me) SCH2CH2OEt CH2OEt
CH (Me) SCH2CH2OEt CH2OCFThree
CH (Me) SCH2CH2OEt CH2SMe
CH (Me) SCH2CH2OEt CH2S (O) Me
CH (Me) SCH2CH2OEt CH2S (O)2Me
CH (Me) SCH2CH2OEt CH2SCFThree
CH (Me) SCH2CH2OEt CH2S (O) CFThree
CH (Me) SCH2CH2OEt CH2S (O)2CFThree
CH (Me) SCH2CH2OEt CH2CH (OEt)2
CH (Me) SCH2CH2OEt CH2CH (SMe)2
CH (Me) SCH2CH2OEt CH2C (O) Me
CH (Me) SCH2CH2OEt CH2C (O) CFThree
CH (Me) SCH2CH2OEt CH2C (O) OEt
CH (Me) SCH2CH2OEt CH2(D1-32a)
CH (Me) SCH2CH2OEt CH2(D1-33a)
CH (Me) SCH2CH2OEt CH2(D1-34a)
CH (Me) SCH2CH2OEt CH2(D1-37a)
CH (Me) SCH2CH2OEt CH2(D1-81a)
CH (Me) SCH2CH2OEt CH2(D1-82a)
CH (Me) SCH2CH2OEt CH2(D1-84a)
CH (Me) SCH2CH2OEt CH2(D1-85a)
CH (Me) SCH2CH2OEt CH2(D1-87a)
CH (Me) SCH2CH2OEt CH2(D1-92a)
CH (Me) SCH2CH2OEt CH2(D1-93a)
CH (Me) SCH2CH2OEt CH2(D1-95a)
CH (Me) SCH2CH2OEt CH2(D1-96a)
CH (Me) SCH2CH2OEt CH2(D1-98a)
CH (Me) SCH2CH2OEt CH2(D1-108a)
CH (Me) SCH2CH2OEt CH2(D1-108b, Z = 2-Cl)
CH (Me) SCH2CH2OEt CH2(D1-108b, Z = 3-Me)
CH (Me) SCH2CH2OEt CH2(D1-108b, Z = 4-OEt)
CH (Me) SCH2CH2OEt CH2(D1-108b, Z = 2-SMe)
CH (Me) SCH2CH2OEt CH2(D1-108b, Z = 3-CFThree)
CH (Me) SCH2CH2OEt CH2(D1-108b, Z = 4-OCFThree)
CH (Me) SCH2CH2OEt CH2(D1-108b, Z = 2-SCFThree)
CH (Me) SCH2CH2OEt CH2CH2CN
CH (Me) SCH2CH2OEt CH2CH2CFThree
CH (Me) SCH2CH2OEt CH2CH2OEt
CH (Me) SCH2CH2OEt CH2CH2SMe
CH (Me) SCH2CH2OEt CH2CH2S (O) Me
CH (Me) SCH2CH2OEt CH2CH2S (O)2Me
CH (Me) SCH2CH2OEt D1-32a
CH (Me) SCH2CH2OEt D1-33a
CH (Me) SCH2CH2OEt D1-34a
CH (Me) SCH2CH2OEt D1-37a
CH (Me) SCH2CH2OEt D1-81a
CH (Me) SCH2CH2OEt D1-82a
CH (Me) SCH2CH2OEt D1-84a
CH (Me) SCH2CH2OEt D1-85a
CH (Me) SCH2CH2OEt D1-87a
CH (Me) SCH2CH2OEt D1-92a
CH (Me) SCH2CH2OEt D1-93a
CH (Me) SCH2CH2OEt D1-95a
CH (Me) SCH2CH2OEt D1-96a
CH (Me) SCH2CH2OEt D1-98a
CH (Me) SCH2CH2OEt D1-108a
CH (Me) SCH2CH2OEt D1-108b (Z = 2-Cl)
CH (Me) SCH2CH2OEt D1-108b (Z = 3-Me)
CH (Me) SCH2CH2OEt D1-108b (Z = 4-OEt)
CH (Me) SCH2CH2OEt D1-108b (Z = 2-SMe)
CH (Me) SCH2CH2OEt D1-108b (Z = 3-CFThree)
CH (Me) SCH2CH2OEt D1-108b (Z = 4-OCFThree)
CH (Me) SCH2CH2OEt D1-108b (Z = 2-SCFThree)
CH (Me) SCH2CH2OEt C (O) Me
CH (Me) SCH2CH2OEt C (O) CFThree
CH (Me) SCH2CH2OEt C (O) OEt
CH (Me) S (O) CH2CH2OEt Me
CH (Me) S (O) CH2CH2OEt Et
CH (Me) S (O) CH2CH2OEt Pr-n
CH (Me) S (O) CH2CH2OEt Pr-i
CH (Me) S (O) CH2CH2OEt Pr-c
CH (Me) S (O) CH2CH2OEt Bu-n
CH (Me) S (O) CH2CH2OEt Bu-i
CH (Me) S (O) CH2CH2OEt Bu-c
CH (Me) S (O) CH2CH2OEt Bu-s
CH (Me) S (O) CH2CH2OEt Bu-t
CH (Me) S (O) CH2CH2OEt Pen-n
CH (Me) S (O) CH2CH2OEt Pen-c
CH (Me) S (O) CH2CH2OEt Hex-n
CH (Me) S (O) CH2CH2OEt Hex-c
CH (Me) S (O) CH2CH2OEt CH2Pr-c
CH (Me) S (O) CH2CH2OEt CH2Bu-c
CH (Me) S (O) CH2CH2OEt CH2Pen-c
CH (Me) S (O) CH2CH2OEt CH2Hex-c
CH (Me) S (O) CH2CH2OEt CH2CH = CH2
CH (Me) S (O) CH2CH2OEt CH2CH = C (Cl)2
CH (Me) S (O) CH2CH2OEt CH2C≡CH
CH (Me) S (O) CH2CH2OEt CH2CN
CH (Me) S (O) CH2CH2OEt CH2CFThree
CH (Me) S (O) CH2CH2OEt CH2OEt
CH (Me) S (O) CH2CH2OEt CH2OCFThree
CH (Me) S (O) CH2CH2OEt CH2SMe
CH (Me) S (O) CH2CH2OEt CH2S (O) Me
CH (Me) S (O) CH2CH2OEt CH2S (O)2Me
CH (Me) S (O) CH2CH2OEt CH2SCFThree
CH (Me) S (O) CH2CH2OEt CH2S (O) CFThree
CH (Me) S (O) CH2CH2OEt CH2S (O)2CFThree
CH (Me) S (O) CH2CH2OEt CH2CH (OEt)2
CH (Me) S (O) CH2CH2OEt CH2CH (SMe)2
CH (Me) S (O) CH2CH2OEt CH2C (O) Me
CH (Me) S (O) CH2CH2OEt CH2C (O) CFThree
CH (Me) S (O) CH2CH2OEt CH2C (O) OEt
CH (Me) S (O) CH2CH2OEt CH2(D1-32a)
CH (Me) S (O) CH2CH2OEt CH2(D1-33a)
CH (Me) S (O) CH2CH2OEt CH2(D1-34a)
CH (Me) S (O) CH2CH2OEt CH2(D1-37a)
CH (Me) S (O) CH2CH2OEt CH2(D1-81a)
CH (Me) S (O) CH2CH2OEt CH2(D1-82a)
CH (Me) S (O) CH2CH2OEt CH2(D1-84a)
CH (Me) S (O) CH2CH2OEt CH2(D1-85a)
CH (Me) S (O) CH2CH2OEt CH2(D1-87a)
CH (Me) S (O) CH2CH2OEt CH2(D1-92a)
CH (Me) S (O) CH2CH2OEt CH2(D1-93a)
CH (Me) S (O) CH2CH2OEt CH2(D1-95a)
CH (Me) S (O) CH2CH2OEt CH2(D1-96a)
CH (Me) S (O) CH2CH2OEt CH2(D1-98a)
CH (Me) S (O) CH2CH2OEt CH2(D1-108a)
CH (Me) S (O) CH2CH2OEt CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O) CH2CH2OEt CH2(D1-108b, Z = 3-Me)
CH (Me) S (O) CH2CH2OEt CH2(D1-108b, Z = 4-OEt)
CH (Me) S (O) CH2CH2OEt CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O) CH2CH2OEt CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O) CH2CH2OEt CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O) CH2CH2OEt CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O) CH2CH2OEt CH2CH2CN
CH (Me) S (O) CH2CH2OEt CH2CH2CFThree
CH (Me) S (O) CH2CH2OEt CH2CH2OEt
CH (Me) S (O) CH2CH2OEt CH2CH2SMe
CH (Me) S (O) CH2CH2OEt CH2CH2S (O) Me
CH (Me) S (O) CH2CH2OEt CH2CH2S (O)2Me
CH (Me) S (O) CH2CH2OEt D1-32a
CH (Me) S (O) CH2CH2OEt D1-33a
CH (Me) S (O) CH2CH2OEt D1-34a
CH (Me) S (O) CH2CH2OEt D1-37a
CH (Me) S (O) CH2CH2OEt D1-81a
CH (Me) S (O) CH2CH2OEt D1-82a
CH (Me) S (O) CH2CH2OEt D1-84a
CH (Me) S (O) CH2CH2OEt D1-85a
CH (Me) S (O) CH2CH2OEt D1-87a
CH (Me) S (O) CH2CH2OEt D1-92a
CH (Me) S (O) CH2CH2OEt D1-93a
CH (Me) S (O) CH2CH2OEt D1-95a
CH (Me) S (O) CH2CH2OEt D1-96a
CH (Me) S (O) CH2CH2OEt D1-98a
CH (Me) S (O) CH2CH2OEt D1-108a
CH (Me) S (O) CH2CH2OEt D1-108b (Z = 2-Cl)
CH (Me) S (O) CH2CH2OEt D1-108b (Z = 3-Me)
CH (Me) S (O) CH2CH2OEt D1-108b (Z = 4-OEt)
CH (Me) S (O) CH2CH2OEt D1-108b (Z = 2-SMe)
CH (Me) S (O) CH2CH2OEt D1-108b (Z = 3-CFThree)
CH (Me) S (O) CH2CH2OEt D1-108b (Z = 4-OCFThree)
CH (Me) S (O) CH2CH2OEt D1-108b (Z = 2-SCFThree)
CH (Me) S (O) CH2CH2OEt C (O) Me
CH (Me) S (O) CH2CH2OEt C (O) CFThree
CH (Me) S (O) CH2CH2OEt C (O) OEt
CH (Me) S (O)2CH2CH2OEt Me
CH (Me) S (O)2CH2CH2OEt Et
CH (Me) S (O)2CH2CH2OEt Pr-n
CH (Me) S (O)2CH2CH2OEt Pr-i
CH (Me) S (O)2CH2CH2OEt Pr-c
CH (Me) S (O)2CH2CH2OEt Bu-n
CH (Me) S (O)2CH2CH2OEt Bu-i
CH (Me) S (O)2CH2CH2OEt Bu-c
CH (Me) S (O)2CH2CH2OEt Bu-s
CH (Me) S (O)2CH2CH2OEt Bu-t
CH (Me) S (O)2CH2CH2OEt Pen-n
CH (Me) S (O)2CH2CH2OEt Pen-c
CH (Me) S (O)2CH2CH2OEt Hex-n
CH (Me) S (O)2CH2CH2OEt Hex-c
CH (Me) S (O)2CH2CH2OEt CH2Pr-c
CH (Me) S (O)2CH2CH2OEt CH2Bu-c
CH (Me) S (O)2CH2CH2OEt CH2Pen-c
CH (Me) S (O)2CH2CH2OEt CH2Hex-c
CH (Me) S (O)2CH2CH2OEt CH2CH = CH2
CH (Me) S (O)2CH2CH2OEt CH2CH = C (Cl)2
CH (Me) S (O)2CH2CH2OEt CH2C≡CH
CH (Me) S (O)2CH2CH2OEt CH2CN
CH (Me) S (O)2CH2CH2OEt CH2CFThree
CH (Me) S (O)2CH2CH2OEt CH2OEt
CH (Me) S (O)2CH2CH2OEt CH2OCFThree
CH (Me) S (O)2CH2CH2OEt CH2SMe
CH (Me) S (O)2CH2CH2OEt CH2S (O) Me
CH (Me) S (O)2CH2CH2OEt CH2S (O)2Me
CH (Me) S (O)2CH2CH2OEt CH2SCFThree
CH (Me) S (O)2CH2CH2OEt CH2S (O) CFThree
CH (Me) S (O)2CH2CH2OEt CH2S (O)2CFThree
CH (Me) S (O)2CH2CH2OEt CH2CH (OEt)2
CH (Me) S (O)2CH2CH2OEt CH2CH (SMe)2
CH (Me) S (O)2CH2CH2OEt CH2C (O) Me
CH (Me) S (O)2CH2CH2OEt CH2C (O) CFThree
CH (Me) S (O)2CH2CH2OEt CH2C (O) OEt
CH (Me) S (O)2CH2CH2OEt CH2(D1-32a)
CH (Me) S (O)2CH2CH2OEt CH2(D1-33a)
CH (Me) S (O)2CH2CH2OEt CH2(D1-34a)
CH (Me) S (O)2CH2CH2OEt CH2(D1-37a)
CH (Me) S (O)2CH2CH2OEt CH2(D1-81a)
CH (Me) S (O)2CH2CH2OEt CH2(D1-82a)
CH (Me) S (O)2CH2CH2OEt CH2(D1-84a)
CH (Me) S (O)2CH2CH2OEt CH2(D1-85a)
CH (Me) S (O)2CH2CH2OEt CH2(D1-87a)
CH (Me) S (O)2CH2CH2OEt CH2(D1-92a)
CH (Me) S (O)2CH2CH2OEt CH2(D1-93a)
CH (Me) S (O)2CH2CH2OEt CH2(D1-95a)
CH (Me) S (O)2CH2CH2OEt CH2(D1-96a)
CH (Me) S (O)2CH2CH2OEt CH2(D1-98a)
CH (Me) S (O)2CH2CH2OEt CH2(D1-108a)
CH (Me) S (O)2CH2CH2OEt CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O)2CH2CH2OEt CH2(D1-108b, Z = 3-Me)
CH (Me) S (O)2CH2CH2OEt CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O)2CH2CH2OEt CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O)2CH2CH2OEt CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O)2CH2CH2OEt CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O)2CH2CH2OEt CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O)2CH2CH2OEt CH2CH2CN
CH (Me) S (O)2CH2CH2OEt CH2CH2CFThree
CH (Me) S (O)2CH2CH2OEt CH2CH2OMe
CH (Me) S (O)2CH2CH2OEt CH2CH2SMe
CH (Me) S (O)2CH2CH2OEt CH2CH2S (O) Me
CH (Me) S (O)2CH2CH2OEt CH2CH2S (O)2Me
CH (Me) S (O)2CH2CH2OEt D1-32a
CH (Me) S (O)2CH2CH2OEt D1-33a
CH (Me) S (O)2CH2CH2OEt D1-34a
CH (Me) S (O)2CH2CH2OEt D1-37a
CH (Me) S (O)2CH2CH2OEt D1-81a
CH (Me) S (O)2CH2CH2OEt D1-82a
CH (Me) S (O)2CH2CH2OEt D1-84a
CH (Me) S (O)2CH2CH2OEt D1-85a
CH (Me) S (O)2CH2CH2OEt D1-87a
CH (Me) S (O)2CH2CH2OEt D1-92a
CH (Me) S (O)2CH2CH2OEt D1-93a
CH (Me) S (O)2CH2CH2OEt D1-95a
CH (Me) S (O)2CH2CH2OEt D1-96a
CH (Me) S (O)2CH2CH2OEt D1-98a
CH (Me) S (O)2CH2CH2OEt D1-108a
CH (Me) S (O)2CH2CH2OEt D1-108b (Z = 2-Cl)
CH (Me) S (O)2CH2CH2OEt D1-108b (Z = 3-Me)
CH (Me) S (O)2CH2CH2OEt D1-108b (Z = 4-OMe)
CH (Me) S (O)2CH2CH2OEt D1-108b (Z = 2-SMe)
CH (Me) S (O)2CH2CH2OEt D1-108b (Z = 3-CFThree)
CH (Me) S (O)2CH2CH2OEt D1-108b (Z = 4-OCFThree)
CH (Me) S (O)2CH2CH2OEt D1-108b (Z = 2-SCFThree)
CH (Me) S (O)2CH2CH2OEt C (O) Me
CH (Me) S (O)2CH2CH2OEt C (O) CFThree
CH (Me) S (O)2CH2CH2OEt C (O) OEt
CH (Et) SCH2CH2OEt Me
CH (Et) SCH2CH2OEt Et
CH (Et) SCH2CH2OEt Pr-n
CH (Et) SCH2CH2OEt Pr-i
CH (Et) SCH2CH2OEt Pr-c
CH (Et) SCH2CH2OEt Bu-n
CH (Et) SCH2CH2OEt Bu-i
CH (Et) SCH2CH2OEt Bu-c
CH (Et) SCH2CH2OEt Bu-s
CH (Et) SCH2CH2OEt Bu-t
CH (Et) SCH2CH2OEt Pen-n
CH (Et) SCH2CH2OEt Pen-c
CH (Et) SCH2CH2OEt Hex-n
CH (Et) SCH2CH2OEt Hex-c
CH (Et) SCH2CH2OEt CH2Pr-c
CH (Et) SCH2CH2OEt CH2Bu-c
CH (Et) SCH2CH2OEt CH2Pen-c
CH (Et) SCH2CH2OEt CH2Hex-c
CH (Et) SCH2CH2OEt CH2CH = CH2
CH (Et) SCH2CH2OEt CH2CH = C (Cl)2
CH (Et) SCH2CH2OEt CH2C≡CH
CH (Et) SCH2CH2OEt CH2CN
CH (Et) SCH2CH2OEt CH2CFThree
CH (Et) SCH2CH2OEt CH2OMe
CH (Et) SCH2CH2OEt CH2OCFThree
CH (Et) SCH2CH2OEt CH2SMe
CH (Et) SCH2CH2OEt CH2S (O) Me
CH (Et) SCH2CH2OEt CH2S (O)2Me
CH (Et) SCH2CH2OEt CH2SCFThree
CH (Et) SCH2CH2OEt CH2S (O) CFThree
CH (Et) SCH2CH2OEt CH2S (O)2CFThree
CH (Et) SCH2CH2OEt CH2CH (OMe)2
CH (Et) SCH2CH2OEt CH2CH (SMe)2
CH (Et) SCH2CH2OEt CH2C (O) Me
CH (Et) SCH2CH2OEt CH2C (O) CFThree
CH (Et) SCH2CH2OEt CH2C (O) OMe
CH (Et) SCH2CH2OEt CH2(D1-32a)
CH (Et) SCH2CH2OEt CH2(D1-33a)
CH (Et) SCH2CH2OEt CH2(D1-34a)
CH (Et) SCH2CH2OEt CH2(D1-37a)
CH (Et) SCH2CH2OEt CH2(D1-81a)
CH (Et) SCH2CH2OEt CH2(D1-82a)
CH (Et) SCH2CH2OEt CH2(D1-84a)
CH (Et) SCH2CH2OEt CH2(D1-85a)
CH (Et) SCH2CH2OEt CH2(D1-87a)
CH (Et) SCH2CH2OEt CH2(D1-92a)
CH (Et) SCH2CH2OEt CH2(D1-93a)
CH (Et) SCH2CH2OEt CH2(D1-95a)
CH (Et) SCH2CH2OEt CH2(D1-96a)
CH (Et) SCH2CH2OEt CH2(D1-98a)
CH (Et) SCH2CH2OEt CH2(D1-108a)
CH (Et) SCH2CH2OEt CH2(D1-108b, Z = 2-Cl)
CH (Et) SCH2CH2OEt CH2(D1-108b, Z = 3-Me)
CH (Et) SCH2CH2OEt CH2(D1-108b, Z = 4-OMe)
CH (Et) SCH2CH2OEt CH2(D1-108b, Z = 2-SMe)
CH (Et) SCH2CH2OEt CH2(D1-108b, Z = 3-CFThree)
CH (Et) SCH2CH2OEt CH2(D1-108b, Z = 4-OCFThree)
CH (Et) SCH2CH2OEt CH2(D1-108b, Z = 2-SCFThree)
CH (Et) SCH2CH2OEt CH2CH2CN
CH (Et) SCH2CH2OEt CH2CH2CFThree
CH (Et) SCH2CH2OEt CH2CH2OMe
CH (Et) SCH2CH2OEt CH2CH2SMe
CH (Et) SCH2CH2OEt CH2CH2S (O) Me
CH (Et) SCH2CH2OEt CH2CH2S (O)2Me
CH (Et) SCH2CH2OEt D1-32a
CH (Et) SCH2CH2OEt D1-33a
CH (Et) SCH2CH2OEt D1-34a
CH (Et) SCH2CH2OEt D1-37a
CH (Et) SCH2CH2OEt D1-81a
CH (Et) SCH2CH2OEt D1-82a
CH (Et) SCH2CH2OEt D1-84a
CH (Et) SCH2CH2OEt D1-85a
CH (Et) SCH2CH2OEt D1-87a
CH (Et) SCH2CH2OEt D1-92a
CH (Et) SCH2CH2OEt D1-93a
CH (Et) SCH2CH2OEt D1-95a
CH (Et) SCH2CH2OEt D1-96a
CH (Et) SCH2CH2OEt D1-98a
CH (Et) SCH2CH2OEt D1-108a
CH (Et) SCH2CH2OEt D1-108b (Z = 2-Cl)
CH (Et) SCH2CH2OEt D1-108b (Z = 3-Me)
CH (Et) SCH2CH2OEt D1-108b (Z = 4-OMe)
CH (Et) SCH2CH2OEt D1-108b (Z = 2-SMe)
CH (Et) SCH2CH2OEt D1-108b (Z = 3-CFThree)
CH (Et) SCH2CH2OEt D1-108b (Z = 4-OCFThree)
CH (Et) SCH2CH2OEt D1-108b (Z = 2-SCFThree)
CH (Et) SCH2CH2OEt C (O) Me
CH (Et) SCH2CH2OEt C (O) CFThree
CH (Et) SCH2CH2OEt C (O) OMe
CH (Et) S (O) CH2CH2OEt Me
CH (Et) S (O) CH2CH2OEt Et
CH (Et) S (O) CH2CH2OEt Pr-n
CH (Et) S (O) CH2CH2OEt Pr-i
CH (Et) S (O) CH2CH2OEt Pr-c
CH (Et) S (O) CH2CH2OEt Bu-n
CH (Et) S (O) CH2CH2OEt Bu-i
CH (Et) S (O) CH2CH2OEt Bu-c
CH (Et) S (O) CH2CH2OEt Bu-s
CH (Et) S (O) CH2CH2OEt Bu-t
CH (Et) S (O) CH2CH2OEt Pen-n
CH (Et) S (O) CH2CH2OEt Pen-c
CH (Et) S (O) CH2CH2OEt Hex-n
CH (Et) S (O) CH2CH2OEt Hex-c
CH (Et) S (O) CH2CH2OEt CH2Pr-c
CH (Et) S (O) CH2CH2OEt CH2Bu-c
CH (Et) S (O) CH2CH2OEt CH2Pen-c
CH (Et) S (O) CH2CH2OEt CH2Hex-c
CH (Et) S (O) CH2CH2OEt CH2CH = CH2
CH (Et) S (O) CH2CH2OEt CH2CH = C (Cl)2
CH (Et) S (O) CH2CH2OEt CH2C≡CH
CH (Et) S (O) CH2CH2OEt CH2CN
CH (Et) S (O) CH2CH2OEt CH2CFThree
CH (Et) S (O) CH2CH2OEt CH2OMe
CH (Et) S (O) CH2CH2OEt CH2OCFThree
CH (Et) S (O) CH2CH2OEt CH2SMe
CH (Et) S (O) CH2CH2OEt CH2S (O) Me
CH (Et) S (O) CH2CH2OEt CH2S (O)2Me
CH (Et) S (O) CH2CH2OEt CH2SCFThree
CH (Et) S (O) CH2CH2OEt CH2S (O) CFThree
CH (Et) S (O) CH2CH2OEt CH2S (O)2CFThree
CH (Et) S (O) CH2CH2OEt CH2CH (OMe)2
CH (Et) S (O) CH2CH2OEt CH2CH (SMe)2
CH (Et) S (O) CH2CH2OEt CH2C (O) Me
CH (Et) S (O) CH2CH2OEt CH2C (O) CFThree
CH (Et) S (O) CH2CH2OEt CH2C (O) OMe
CH (Et) S (O) CH2CH2OEt CH2(D1-32a)
CH (Et) S (O) CH2CH2OEt CH2(D1-33a)
CH (Et) S (O) CH2CH2OEt CH2(D1-34a)
CH (Et) S (O) CH2CH2OEt CH2(D1-37a)
CH (Et) S (O) CH2CH2OEt CH2(D1-81a)
CH (Et) S (O) CH2CH2OEt CH2(D1-82a)
CH (Et) S (O) CH2CH2OEt CH2(D1-84a)
CH (Et) S (O) CH2CH2OEt CH2(D1-85a)
CH (Et) S (O) CH2CH2OEt CH2(D1-87a)
CH (Et) S (O) CH2CH2OEt CH2(D1-92a)
CH (Et) S (O) CH2CH2OEt CH2(D1-93a)
CH (Et) S (O) CH2CH2OEt CH2(D1-95a)
CH (Et) S (O) CH2CH2OEt CH2(D1-96a)
CH (Et) S (O) CH2CH2OEt CH2(D1-98a)
CH (Et) S (O) CH2CH2OEt CH2(D1-108a)
CH (Et) S (O) CH2CH2OEt CH2(D1-108b, Z = 2-Cl)
CH (Et) S (O) CH2CH2OEt CH2(D1-108b, Z = 3-Me)
CH (Et) S (O) CH2CH2OEt CH2(D1-108b, Z = 4-OMe)
CH (Et) S (O) CH2CH2OEt CH2(D1-108b, Z = 2-SMe)
CH (Et) S (O) CH2CH2OEt CH2(D1-108b, Z = 3-CFThree)
CH (Et) S (O) CH2CH2OEt CH2(D1-108b, Z = 4-OCFThree)
CH (Et) S (O) CH2CH2OEt CH2(D1-108b, Z = 2-SCFThree)
CH (Et) S (O) CH2CH2OEt CH2CH2CN
CH (Et) S (O) CH2CH2OEt CH2CH2CFThree
CH (Et) S (O) CH2CH2OEt CH2CH2OMe
CH (Et) S (O) CH2CH2OEt CH2CH2SMe
CH (Et) S (O) CH2CH2OEt CH2CH2S (O) Me
CH (Et) S (O) CH2CH2OEt CH2CH2S (O)2Me
CH (Et) S (O) CH2CH2OEt D1-32a
CH (Et) S (O) CH2CH2OEt D1-33a
CH (Et) S (O) CH2CH2OEt D1-34a
CH (Et) S (O) CH2CH2OEt D1-37a
CH (Et) S (O) CH2CH2OEt D1-81a
CH (Et) S (O) CH2CH2OEt D1-82a
CH (Et) S (O) CH2CH2OEt D1-84a
CH (Et) S (O) CH2CH2OEt D1-85a
CH (Et) S (O) CH2CH2OEt D1-87a
CH (Et) S (O) CH2CH2OEt D1-92a
CH (Et) S (O) CH2CH2OEt D1-93a
CH (Et) S (O) CH2CH2OEt D1-95a
CH (Et) S (O) CH2CH2OEt D1-96a
CH (Et) S (O) CH2CH2OEt D1-98a
CH (Et) S (O) CH2CH2OEt D1-108a
CH (Et) S (O) CH2CH2OEt D1-108b (Z = 2-Cl)
CH (Et) S (O) CH2CH2OEt D1-108b (Z = 3-Me)
CH (Et) S (O) CH2CH2OEt D1-108b (Z = 4-OMe)
CH (Et) S (O) CH2CH2OEt D1-108b (Z = 2-SMe)
CH (Et) S (O) CH2CH2OEt D1-108b (Z = 3-CFThree)
CH (Et) S (O) CH2CH2OEt D1-108b (Z = 4-OCFThree)
CH (Et) S (O) CH2CH2OEt D1-108b (Z = 2-SCFThree)
CH (Et) S (O) CH2CH2OEt C (O) Me
CH (Et) S (O) CH2CH2OEt C (O) CFThree
CH (Et) S (O) CH2CH2OEt C (O) OMe
CH (Et) S (O)2CH2CH2OEt Me
CH (Et) S (O)2CH2CH2OEt Et
CH (Et) S (O)2CH2CH2OEt Pr-n
CH (Et) S (O)2CH2CH2OEt Pr-i
CH (Et) S (O)2CH2CH2OEt Pr-c
CH (Et) S (O)2CH2CH2OEt Bu-n
CH (Et) S (O)2CH2CH2OEt Bu-i
CH (Et) S (O)2CH2CH2OEt Bu-c
CH (Et) S (O)2CH2CH2OEt Bu-s
CH (Et) S (O)2CH2CH2OEt Bu-t
CH (Et) S (O)2CH2CH2OEt Pen-n
CH (Et) S (O)2CH2CH2OEt Pen-c
CH (Et) S (O)2CH2CH2OEt Hex-n
CH (Et) S (O)2CH2CH2OEt Hex-c
CH (Et) S (O)2CH2CH2OEt CH2Pr-c
CH (Et) S (O)2CH2CH2OEt CH2Bu-c
CH (Et) S (O)2CH2CH2OEt CH2Pen-c
CH (Et) S (O)2CH2CH2OEt CH2Hex-c
CH (Et) S (O)2CH2CH2OEt CH2CH = CH2
CH (Et) S (O)2CH2CH2OEt CH2CH = C (Cl)2
CH (Et) S (O)2CH2CH2OEt CH2C≡CH
CH (Et) S (O)2CH2CH2OEt CH2CN
CH (Et) S (O)2CH2CH2OEt CH2CFThree
CH (Et) S (O)2CH2CH2OEt CH2OMe
CH (Et) S (O)2CH2CH2OEt CH2OCFThree
CH (Et) S (O)2CH2CH2OEt CH2SMe
CH (Et) S (O)2CH2CH2OEt CH2S (O) Me
CH (Et) S (O)2CH2CH2OEt CH2S (O)2Me
CH (Et) S (O)2CH2CH2OEt CH2SCFThree
CH (Et) S (O)2CH2CH2OEt CH2S (O) CFThree
CH (Et) S (O)2CH2CH2OEt CH2S (O)2CFThree
CH (Et) S (O)2CH2CH2OEt CH2CH (OMe)2
CH (Et) S (O)2CH2CH2OEt CH2CH (SMe)2
CH (Et) S (O)2CH2CH2OEt CH2C (O) Me
CH (Et) S (O)2CH2CH2OEt CH2C (O) CFThree
CH (Et) S (O)2CH2CH2OEt CH2C (O) OMe
CH (Et) S (O)2CH2CH2OEt CH2(D1-32a)
CH (Et) S (O)2CH2CH2OEt CH2(D1-33a)
CH (Et) S (O)2CH2CH2OEt CH2(D1-34a)
CH (Et) S (O)2CH2CH2OEt CH2(D1-37a)
CH (Et) S (O)2CH2CH2OEt CH2(D1-81a)
CH (Et) S (O)2CH2CH2OEt CH2(D1-82a)
CH (Et) S (O)2CH2CH2OEt CH2(D1-84a)
CH (Et) S (O)2CH2CH2OEt CH2(D1-85a)
CH (Et) S (O)2CH2CH2OEt CH2(D1-87a)
CH (Et) S (O)2CH2CH2OEt CH2(D1-92a)
CH (Et) S (O)2CH2CH2OEt CH2(D1-93a)
CH (Et) S (O)2CH2CH2OEt CH2(D1-95a)
CH (Et) S (O)2CH2CH2OEt CH2(D1-96a)
CH (Et) S (O)2CH2CH2OEt CH2(D1-98a)
CH (Et) S (O)2CH2CH2OEt CH2(D1-108a)
CH (Et) S (O)2CH2CH2OEt CH2(D1-108b, Z = 2-Cl)
CH (Et) S (O)2CH2CH2OEt CH2(D1-108b, Z = 3-Me)
CH (Et) S (O)2CH2CH2OEt CH2(D1-108b, Z = 4-OEt)
CH (Et) S (O)2CH2CH2OEt CH2(D1-108b, Z = 2-SMe)
CH (Et) S (O)2CH2CH2OEt CH2(D1-108b, Z = 3-CFThree)
CH (Et) S (O)2CH2CH2OEt CH2(D1-108b, Z = 4-OCFThree)
CH (Et) S (O)2CH2CH2OEt CH2(D1-108b, Z = 2-SCFThree)
CH (Et) S (O)2CH2CH2OEt CH2CH2CN
CH (Et) S (O)2CH2CH2OEt CH2CH2CFThree
CH (Et) S (O)2CH2CH2OEt CH2CH2OMe
CH (Et) S (O)2CH2CH2OEt CH2CH2SMe
CH (Et) S (O)2CH2CH2OEt CH2CH2S (O) Me
CH (Et) S (O)2CH2CH2OEt CH2CH2S (O)2Me
CH (Et) S (O)2CH2CH2OEt D1-32a
CH (Et) S (O)2CH2CH2OEt D1-33a
CH (Et) S (O)2CH2CH2OEt D1-34a
CH (Et) S (O)2CH2CH2OEt D1-37a
CH (Et) S (O)2CH2CH2OEt D1-81a
CH (Et) S (O)2CH2CH2OEt D1-82a
CH (Et) S (O)2CH2CH2OEt D1-84a
CH (Et) S (O)2CH2CH2OEt D1-85a
CH (Et) S (O)2CH2CH2OEt D1-87a
CH (Et) S (O)2CH2CH2OEt D1-92a
CH (Et) S (O)2CH2CH2OEt D1-93a
CH (Et) S (O)2CH2CH2OEt D1-95a
CH (Et) S (O)2CH2CH2OEt D1-96a
CH (Et) S (O)2CH2CH2OEt D1-98a
CH (Et) S (O)2CH2CH2OEt D1-108a
CH (Et) S (O)2CH2CH2OEt D1-108b (Z = 2-Cl)
CH (Et) S (O)2CH2CH2OEt D1-108b (Z = 3-Me)
CH (Et) S (O)2CH2CH2OEt D1-108b (Z = 4-OMe)
CH (Et) S (O)2CH2CH2OEt D1-108b (Z = 2-SMe)
CH (Et) S (O)2CH2CH2OEt D1-108b (Z = 3-CFThree)
CH (Et) S (O)2CH2CH2OEt D1-108b (Z = 4-OCFThree)
CH (Et) S (O)2CH2CH2OEt D1-108b (Z = 2-SCFThree)
CH (Et) S (O)2CH2CH2OEt C (O) Me
CH (Et) S (O)2CH2CH2OEt C (O) CFThree
CH (Et) S (O)2CH2CH2OEt C (O) OMe
CH2SCH2(D1-32a) Me
CH2SCH2(D1-32a) Et
CH2SCH2(D1-32a) Pr-n
CH2SCH2(D1-32a) Pr-i
CH2SCH2(D1-32a) Pr-c
CH2SCH2(D1-32a) Bu-n
CH2SCH2(D1-32a) Bu-i
CH2SCH2(D1-32a) Bu-c
CH2SCH2(D1-32a) Bu-s
CH2SCH2(D1-32a) Bu-t
CH2SCH2(D1-32a) Pen-n
CH2SCH2(D1-32a) Pen-c
CH2SCH2(D1-32a) Hex-n
CH2SCH2(D1-32a) Hex-c
CH2SCH2(D1-32a) CH2Pr-c
CH2SCH2(D1-32a) CH2Bu-c
CH2SCH2(D1-32a) CH2Pen-c
CH2SCH2(D1-32a) CH2Hex-c
CH2SCH2(D1-32a) CH2CH = CH2
CH2SCH2(D1-32a) CH2CH = C (Cl)2
CH2SCH2(D1-32a) CH2C≡CH
CH2SCH2(D1-32a) CH2CN
CH2SCH2(D1-32a) CH2CFThree
CH2SCH2(D1-32a) CH2OMe
CH2SCH2(D1-32a) CH2OCFThree
CH2SCH2(D1-32a) CH2SMe
CH2SCH2(D1-32a) CH2S (O) Me
CH2SCH2(D1-32a) CH2S (O)2Me
CH2SCH2(D1-32a) CH2SCFThree
CH2SCH2(D1-32a) CH2S (O) CFThree
CH2SCH2(D1-32a) CH2S (O)2CFThree
CH2SCH2(D1-32a) CH2CH (OMe)2
CH2SCH2(D1-32a) CH2CH (SMe)2
CH2SCH2(D1-32a) CH2C (O) Me
CH2SCH2(D1-32a) CH2C (O) CFThree
CH2SCH2(D1-32a) CH2C (O) OMe
CH2SCH2(D1-32a) CH2(D1-32a)
CH2SCH2(D1-32a) CH2(D1-33a)
CH2SCH2(D1-32a) CH2(D1-34a)
CH2SCH2(D1-32a) CH2(D1-37a)
CH2SCH2(D1-32a) CH2(D1-81a)
CH2SCH2(D1-32a) CH2(D1-82a)
CH2SCH2(D1-32a) CH2(D1-84a)
CH2SCH2(D1-32a) CH2(D1-85a)
CH2SCH2(D1-32a) CH2(D1-87a)
CH2SCH2(D1-32a) CH2(D1-92a)
CH2SCH2(D1-32a) CH2(D1-93a)
CH2SCH2(D1-32a) CH2(D1-95a)
CH2SCH2(D1-32a) CH2(D1-96a)
CH2SCH2(D1-32a) CH2(D1-98a)
CH2SCH2(D1-32a) CH2(D1-108a)
CH2SCH2(D1-32a) CH2(D1-108b, Z = 2-Cl)
CH2SCH2(D1-32a) CH2(D1-108b, Z = 3-Me)
CH2SCH2(D1-32a) CH2(D1-108b, Z = 4-OMe)
CH2SCH2(D1-32a) CH2(D1-108b, Z = 2-SMe)
CH2SCH2(D1-32a) CH2(D1-108b, Z = 3-CFThree)
CH2SCH2(D1-32a) CH2(D1-108b, Z = 4-OCFThree)
CH2SCH2(D1-32a) CH2(D1-108b, Z = 2-SCFThree)
CH2SCH2(D1-32a) CH2CH2CN
CH2SCH2(D1-32a) CH2CH2CFThree
CH2SCH2(D1-32a) CH2CH2OMe
CH2SCH2(D1-32a) CH2CH2SMe
CH2SCH2(D1-32a) CH2CH2S (O) Me
CH2SCH2(D1-32a) CH2CH2S (O)2Me
CH2SCH2(D1-32a) D1-32a
CH2SCH2(D1-32a) D1-33a
CH2SCH2(D1-32a) D1-34a
CH2SCH2(D1-32a) D1-37a
CH2SCH2(D1-32a) D1-81a
CH2SCH2(D1-32a) D1-82a
CH2SCH2(D1-32a) D1-84a
CH2SCH2(D1-32a) D1-85a
CH2SCH2(D1-32a) D1-87a
CH2SCH2(D1-32a) D1-92a
CH2SCH2(D1-32a) D1-93a
CH2SCH2(D1-32a) D1-95a
CH2SCH2(D1-32a) D1-96a
CH2SCH2(D1-32a) D1-98a
CH2SCH2(D1-32a) D1-108a
CH2SCH2(D1-32a) D1-108b (Z = 2-Cl)
CH2SCH2(D1-32a) D1-108b (Z = 3-Me)
CH2SCH2(D1-32a) D1-108b (Z = 4-OMe)
CH2SCH2(D1-32a) D1-108b (Z = 2-SMe)
CH2SCH2(D1-32a) D1-108b (Z = 3-CFThree)
CH2SCH2(D1-32a) D1-108b (Z = 4-OCFThree)
CH2SCH2(D1-32a) D1-108b (Z = 2-SCFThree)
CH2SCH2(D1-32a) C (O) Me
CH2SCH2(D1-32a) C (O) CFThree
CH2SCH2(D1-32a) C (O) OMe
CH2S (O) CH2(D1-32a) Me
CH2S (O) CH2(D1-32a) Et
CH2S (O) CH2(D1-32a) Pr-n
CH2S (O) CH2(D1-32a) Pr-i
CH2S (O) CH2(D1-32a) Pr-c
CH2S (O) CH2(D1-32a) Bu-n
CH2S (O) CH2(D1-32a) Bu-i
CH2S (O) CH2(D1-32a) Bu-c
CH2S (O) CH2(D1-32a) Bu-s
CH2S (O) CH2(D1-32a) Bu-t
CH2S (O) CH2(D1-32a) Pen-n
CH2S (O) CH2(D1-32a) Pen-c
CH2S (O) CH2(D1-32a) Hex-n
CH2S (O) CH2(D1-32a) Hex-c
CH2S (O) CH2(D1-32a) CH2Pr-c
CH2S (O) CH2(D1-32a) CH2Bu-c
CH2S (O) CH2(D1-32a) CH2Pen-c
CH2S (O) CH2(D1-32a) CH2Hex-c
CH2S (O) CH2(D1-32a) CH2CH = CH2
CH2S (O) CH2(D1-32a) CH2CH = C (Cl)2
CH2S (O) CH2(D1-32a) CH2C≡CH
CH2S (O) CH2(D1-32a) CH2CN
CH2S (O) CH2(D1-32a) CH2CFThree
CH2S (O) CH2(D1-32a) CH2OMe
CH2S (O) CH2(D1-32a) CH2OCFThree
CH2S (O) CH2(D1-32a) CH2SMe
CH2S (O) CH2(D1-32a) CH2S (O) Me
CH2S (O) CH2(D1-32a) CH2S (O)2Me
CH2S (O) CH2(D1-32a) CH2SCFThree
CH2S (O) CH2(D1-32a) CH2S (O) CFThree
CH2S (O) CH2(D1-32a) CH2S (O)2CFThree
CH2S (O) CH2(D1-32a) CH2CH (OMe)2
CH2S (O) CH2(D1-32a) CH2CH (SMe)2
CH2S (O) CH2(D1-32a) CH2C (O) Me
CH2S (O) CH2(D1-32a) CH2C (O) CFThree
CH2S (O) CH2(D1-32a) CH2C (O) OMe
CH2S (O) CH2(D1-32a) CH2(D1-32a)
CH2S (O) CH2(D1-32a) CH2(D1-33a)
CH2S (O) CH2(D1-32a) CH2(D1-34a)
CH2S (O) CH2(D1-32a) CH2(D1-37a)
CH2S (O) CH2(D1-32a) CH2(D1-81a)
CH2S (O) CH2(D1-32a) CH2(D1-82a)
CH2S (O) CH2(D1-32a) CH2(D1-84a)
CH2S (O) CH2(D1-32a) CH2(D1-85a)
CH2S (O) CH2(D1-32a) CH2(D1-87a)
CH2S (O) CH2(D1-32a) CH2(D1-92a)
CH2S (O) CH2(D1-32a) CH2(D1-93a)
CH2S (O) CH2(D1-32a) CH2(D1-95a)
CH2S (O) CH2(D1-32a) CH2(D1-96a)
CH2S (O) CH2(D1-32a) CH2(D1-98a)
CH2S (O) CH2(D1-32a) CH2(D1-108a)
CH2S (O) CH2(D1-32a) CH2(D1-108b, Z = 2-Cl)
CH2S (O) CH2(D1-32a) CH2(D1-108b, Z = 3-Me)
CH2S (O) CH2(D1-32a) CH2(D1-108b, Z = 4-OMe)
CH2S (O) CH2(D1-32a) CH2(D1-108b, Z = 2-SMe)
CH2S (O) CH2(D1-32a) CH2(D1-108b, Z = 3-CFThree)
CH2S (O) CH2(D1-32a) CH2(D1-108b, Z = 4-OCFThree)
CH2S (O) CH2(D1-32a) CH2(D1-108b, Z = 2-SCFThree)
CH2S (O) CH2(D1-32a) CH2CH2CN
CH2S (O) CH2(D1-32a) CH2CH2CFThree
CH2S (O) CH2(D1-32a) CH2CH2OMe
CH2S (O) CH2(D1-32a) CH2CH2SMe
CH2S (O) CH2(D1-32a) CH2CH2S (O) Me
CH2S (O) CH2(D1-32a) CH2CH2S (O)2Me
CH2S (O) CH2(D1-32a) D1-32a
CH2S (O) CH2(D1-32a) D1-33a
CH2S (O) CH2(D1-32a) D1-34a
CH2S (O) CH2(D1-32a) D1-37a
CH2S (O) CH2(D1-32a) D1-81a
CH2S (O) CH2(D1-32a) D1-82a
CH2S (O) CH2(D1-32a) D1-84a
CH2S (O) CH2(D1-32a) D1-85a
CH2S (O) CH2(D1-32a) D1-87a
CH2S (O) CH2(D1-32a) D1-92a
CH2S (O) CH2(D1-32a) D1-93a
CH2S (O) CH2(D1-32a) D1-95a
CH2S (O) CH2(D1-32a) D1-96a
CH2S (O) CH2(D1-32a) D1-98a
CH2S (O) CH2(D1-32a) D1-108a
CH2S (O) CH2(D1-32a) D1-108b (Z = 2-Cl)
CH2S (O) CH2(D1-32a) D1-108b (Z = 3-Me)
CH2S (O) CH2(D1-32a) D1-108b (Z = 4-OMe)
CH2S (O) CH2(D1-32a) D1-108b (Z = 2-SMe)
CH2S (O) CH2(D1-32a) D1-108b (Z = 3-CFThree)
CH2S (O) CH2(D1-32a) D1-108b (Z = 4-OCFThree)
CH2S (O) CH2(D1-32a) D1-108b (Z = 2-SCFThree)
CH2S (O) CH2(D1-32a) C (O) Me
CH2S (O) CH2(D1-32a) C (O) CFThree
CH2S (O) CH2(D1-32a) C (O) OMe
CH2S (O)2CH2(D1-32a) Me
CH2S (O)2CH2(D1-32a) Et
CH2S (O)2CH2(D1-32a) Pr-n
CH2S (O)2CH2(D1-32a) Pr-i
CH2S (O)2CH2(D1-32a) Pr-c
CH2S (O)2CH2(D1-32a) Bu-n
CH2S (O)2CH2(D1-32a) Bu-i
CH2S (O)2CH2(D1-32a) Bu-c
CH2S (O)2CH2(D1-32a) Bu-s
CH2S (O)2CH2(D1-32a) Bu-t
CH2S (O)2CH2(D1-32a) Pen-n
CH2S (O)2CH2(D1-32a) Pen-c
CH2S (O)2CH2(D1-32a) Hex-n
CH2S (O)2CH2(D1-32a) Hex-c
CH2S (O)2CH2(D1-32a) CH2Pr-c
CH2S (O)2CH2(D1-32a) CH2Bu-c
CH2S (O)2CH2(D1-32a) CH2Pen-c
CH2S (O)2CH2(D1-32a) CH2Hex-c
CH2S (O)2CH2(D1-32a) CH2CH = CH2
CH2S (O)2CH2(D1-32a) CH2CH = C (Cl)2
CH2S (O)2CH2(D1-32a) CH2C≡CH
CH2S (O)2CH2(D1-32a) CH2CN
CH2S (O)2CH2(D1-32a) CH2CFThree
CH2S (O)2CH2(D1-32a) CH2OMe
CH2S (O)2CH2(D1-32a) CH2OCFThree
CH2S (O)2CH2(D1-32a) CH2SMe
CH2S (O)2CH2(D1-32a) CH2S (O) Me
CH2S (O)2CH2(D1-32a) CH2S (O)2Me
CH2S (O)2CH2(D1-32a) CH2SCFThree
CH2S (O)2CH2(D1-32a) CH2S (O) CFThree
CH2S (O)2CH2(D1-32a) CH2S (O)2CFThree
CH2S (O)2CH2(D1-32a) CH2CH (OMe)2
CH2S (O)2CH2(D1-32a) CH2CH (SMe)2
CH2S (O)2CH2(D1-32a) CH2C (O) Me
CH2S (O)2CH2(D1-32a) CH2C (O) CFThree
CH2S (O)2CH2(D1-32a) CH2C (O) OMe
CH2S (O)2CH2(D1-32a) CH2(D1-32a)
CH2S (O)2CH2(D1-32a) CH2(D1-33a)
CH2S (O)2CH2(D1-32a) CH2(D1-34a)
CH2S (O)2CH2(D1-32a) CH2(D1-37a)
CH2S (O)2CH2(D1-32a) CH2(D1-81a)
CH2S (O)2CH2(D1-32a) CH2(D1-82a)
CH2S (O)2CH2(D1-32a) CH2(D1-84a)
CH2S (O)2CH2(D1-32a) CH2(D1-85a)
CH2S (O)2CH2(D1-32a) CH2(D1-87a)
CH2S (O)2CH2(D1-32a) CH2(D1-92a)
CH2S (O)2CH2(D1-32a) CH2(D1-93a)
CH2S (O)2CH2(D1-32a) CH2(D1-95a)
CH2S (O)2CH2(D1-32a) CH2(D1-96a)
CH2S (O)2CH2(D1-32a) CH2(D1-98a)
CH2S (O)2CH2(D1-32a) CH2(D1-108a)
CH2S (O)2CH2(D1-32a) CH2(D1-108b, Z = 2-Cl)
CH2S (O)2CH2(D1-32a) CH2(D1-108b, Z = 3-Me)
CH2S (O)2CH2(D1-32a) CH2(D1-108b, Z = 4-OMe)
CH2S (O)2CH2(D1-32a) CH2(D1-108b, Z = 2-SMe)
CH2S (O)2CH2(D1-32a) CH2(D1-108b, Z = 3-CFThree)
CH2S (O)2CH2(D1-32a) CH2(D1-108b, Z = 4-OCFThree)
CH2S (O)2CH2(D1-32a) CH2(D1-108b, Z = 2-SCFThree)
CH2S (O)2CH2(D1-32a) CH2CH2CN
CH2S (O)2CH2(D1-32a) CH2CH2CFThree
CH2S (O)2CH2(D1-32a) CH2CH2OMe
CH2S (O)2CH2(D1-32a) CH2CH2SMe
CH2S (O)2CH2(D1-32a) CH2CH2S (O) Me
CH2S (O)2CH2(D1-32a) CH2CH2S (O)2Me
CH2S (O)2CH2(D1-32a) D1-32a
CH2S (O)2CH2(D1-32a) D1-33a
CH2S (O)2CH2(D1-32a) D1-34a
CH2S (O)2CH2(D1-32a) D1-37a
CH2S (O)2CH2(D1-32a) D1-81a
CH2S (O)2CH2(D1-32a) D1-82a
CH2S (O)2CH2(D1-32a) D1-84a
CH2S (O)2CH2(D1-32a) D1-85a
CH2S (O)2CH2(D1-32a) D1-87a
CH2S (O)2CH2(D1-32a) D1-92a
CH2S (O)2CH2(D1-32a) D1-93a
CH2S (O)2CH2(D1-32a) D1-95a
CH2S (O)2CH2(D1-32a) D1-96a
CH2S (O)2CH2(D1-32a) D1-98a
CH2S (O)2CH2(D1-32a) D1-108a
CH2S (O)2CH2(D1-32a) D1-108b (Z = 2-Cl)
CH2S (O)2CH2(D1-32a) D1-108b (Z = 3-Me)
CH2S (O)2CH2(D1-32a) D1-108b (Z = 4-OMe)
CH2S (O)2CH2(D1-32a) D1-108b (Z = 2-SMe)
CH2S (O)2CH2(D1-32a) D1-108b (Z = 3-CFThree)
CH2S (O)2CH2(D1-32a) D1-108b (Z = 4-OCFThree)
CH2S (O)2CH2(D1-32a) D1-108b (Z = 2-SCFThree)
CH2S (O)2CH2(D1-32a) C (O) Me
CH2S (O)2CH2(D1-32a) C (O) CFThree
CH2S (O)2CH2(D1-32a) C (O) OMe
CH (Me) SCH2(D1-32a) Me
CH (Me) SCH2(D1-32a) Et
CH (Me) SCH2(D1-32a) Pr-n
CH (Me) SCH2(D1-32a) Pr-i
CH (Me) SCH2(D1-32a) Pr-c
CH (Me) SCH2(D1-32a) Bu-n
CH (Me) SCH2(D1-32a) Bu-i
CH (Me) SCH2(D1-32a) Bu-c
CH (Me) SCH2(D1-32a) Bu-s
CH (Me) SCH2(D1-32a) Bu-t
CH (Me) SCH2(D1-32a) Pen-n
CH (Me) SCH2(D1-32a) Pen-c
CH (Me) SCH2(D1-32a) Hex-n
CH (Me) SCH2(D1-32a) Hex-c
CH (Me) SCH2(D1-32a) CH2Pr-c
CH (Me) SCH2(D1-32a) CH2Bu-c
CH (Me) SCH2(D1-32a) CH2Pen-c
CH (Me) SCH2(D1-32a) CH2Hex-c
CH (Me) SCH2(D1-32a) CH2CH = CH2
CH (Me) SCH2(D1-32a) CH2CH = C (Cl)2
CH (Me) SCH2(D1-32a) CH2C≡CH
CH (Me) SCH2(D1-32a) CH2CN
CH (Me) SCH2(D1-32a) CH2CFThree
CH (Me) SCH2(D1-32a) CH2OMe
CH (Me) SCH2(D1-32a) CH2OCFThree
CH (Me) SCH2(D1-32a) CH2SMe
CH (Me) SCH2(D1-32a) CH2S (O) Me
CH (Me) SCH2(D1-32a) CH2S (O)2Me
CH (Me) SCH2(D1-32a) CH2SCFThree
CH (Me) SCH2(D1-32a) CH2S (O) CFThree
CH (Me) SCH2(D1-32a) CH2S (O)2CFThree
CH (Me) SCH2(D1-32a) CH2CH (OMe)2
CH (Me) SCH2(D1-32a) CH2CH (SMe)2
CH (Me) SCH2(D1-32a) CH2C (O) Me
CH (Me) SCH2(D1-32a) CH2C (O) CFThree
CH (Me) SCH2(D1-32a) CH2C (O) OMe
CH (Me) SCH2(D1-32a) CH2(D1-32a)
CH (Me) SCH2(D1-32a) CH2(D1-33a)
CH (Me) SCH2(D1-32a) CH2(D1-34a)
CH (Me) SCH2(D1-32a) CH2(D1-37a)
CH (Me) SCH2(D1-32a) CH2(D1-81a)
CH (Me) SCH2(D1-32a) CH2(D1-82a)
CH (Me) SCH2(D1-32a) CH2(D1-84a)
CH (Me) SCH2(D1-32a) CH2(D1-85a)
CH (Me) SCH2(D1-32a) CH2(D1-87a)
CH (Me) SCH2(D1-32a) CH2(D1-92a)
CH (Me) SCH2(D1-32a) CH2(D1-93a)
CH (Me) SCH2(D1-32a) CH2(D1-95a)
CH (Me) SCH2(D1-32a) CH2(D1-96a)
CH (Me) SCH2(D1-32a) CH2(D1-98a)
CH (Me) SCH2(D1-32a) CH2(D1-108a)
CH (Me) SCH2(D1-32a) CH2(D1-108b, Z = 2-Cl)
CH (Me) SCH2(D1-32a) CH2(D1-108b, Z = 3-Me)
CH (Me) SCH2(D1-32a) CH2(D1-108b, Z = 4-OMe)
CH (Me) SCH2(D1-32a) CH2(D1-108b, Z = 2-SMe)
CH (Me) SCH2(D1-32a) CH2(D1-108b, Z = 3-CFThree)
CH (Me) SCH2(D1-32a) CH2(D1-108b, Z = 4-OCFThree)
CH (Me) SCH2(D1-32a) CH2(D1-108b, Z = 2-SCFThree)
CH (Me) SCH2(D1-32a) CH2CH2CN
CH (Me) SCH2(D1-32a) CH2CH2CFThree
CH (Me) SCH2(D1-32a) CH2CH2OMe
CH (Me) SCH2(D1-32a) CH2CH2SMe
CH (Me) SCH2(D1-32a) CH2CH2S (O) Me
CH (Me) SCH2(D1-32a) CH2CH2S (O)2Me
CH (Me) SCH2(D1-32a) D1-32a
CH (Me) SCH2(D1-32a) D1-33a
CH (Me) SCH2(D1-32a) D1-34a
CH (Me) SCH2(D1-32a) D1-37a
CH (Me) SCH2(D1-32a) D1-81a
CH (Me) SCH2(D1-32a) D1-82a
CH (Me) SCH2(D1-32a) D1-84a
CH (Me) SCH2(D1-32a) D1-85a
CH (Me) SCH2(D1-32a) D1-87a
CH (Me) SCH2(D1-32a) D1-92a
CH (Me) SCH2(D1-32a) D1-93a
CH (Me) SCH2(D1-32a) D1-95a
CH (Me) SCH2(D1-32a) D1-96a
CH (Me) SCH2(D1-32a) D1-98a
CH (Me) SCH2(D1-32a) D1-108a
CH (Me) SCH2(D1-32a) D1-108b (Z = 2-Cl)
CH (Me) SCH2(D1-32a) D1-108b (Z = 3-Me)
CH (Me) SCH2(D1-32a) D1-108b (Z = 4-OMe)
CH (Me) SCH2(D1-32a) D1-108b (Z = 2-SMe)
CH (Me) SCH2(D1-32a) D1-108b (Z = 3-CFThree)
CH (Me) SCH2(D1-32a) D1-108b (Z = 4-OCFThree)
CH (Me) SCH2(D1-32a) D1-108b (Z = 2-SCFThree)
CH (Me) SCH2(D1-32a) C (O) Me
CH (Me) SCH2(D1-32a) C (O) CFThree
CH (Me) SCH2(D1-32a) C (O) OMe
CH (Me) S (O) CH2(D1-32a) Me
CH (Me) S (O) CH2(D1-32a) Et
CH (Me) S (O) CH2(D1-32a) Pr-n
CH (Me) S (O) CH2(D1-32a) Pr-i
CH (Me) S (O) CH2(D1-32a) Pr-c
CH (Me) S (O) CH2(D1-32a) Bu-n
CH (Me) S (O) CH2(D1-32a) Bu-i
CH (Me) S (O) CH2(D1-32a) Bu-c
CH (Me) S (O) CH2(D1-32a) Bu-s
CH (Me) S (O) CH2(D1-32a) Bu-t
CH (Me) S (O) CH2(D1-32a) Pen-n
CH (Me) S (O) CH2(D1-32a) Pen-c
CH (Me) S (O) CH2(D1-32a) Hex-n
CH (Me) S (O) CH2(D1-32a) Hex-c
CH (Me) S (O) CH2(D1-32a) CH2Pr-c
CH (Me) S (O) CH2(D1-32a) CH2Bu-c
CH (Me) S (O) CH2(D1-32a) CH2Pen-c
CH (Me) S (O) CH2(D1-32a) CH2Hex-c
CH (Me) S (O) CH2(D1-32a) CH2CH = CH2
CH (Me) S (O) CH2(D1-32a) CH2CH = C (Cl)2
CH (Me) S (O) CH2(D1-32a) CH2C≡CH
CH (Me) S (O) CH2(D1-32a) CH2CN
CH (Me) S (O) CH2(D1-32a) CH2CFThree
CH (Me) S (O) CH2(D1-32a) CH2OMe
CH (Me) S (O) CH2(D1-32a) CH2OCFThree
CH (Me) S (O) CH2(D1-32a) CH2SMe
CH (Me) S (O) CH2(D1-32a) CH2S (O) Me
CH (Me) S (O) CH2(D1-32a) CH2S (O)2Me
CH (Me) S (O) CH2(D1-32a) CH2SCFThree
CH (Me) S (O) CH2(D1-32a) CH2S (O) CFThree
CH (Me) S (O) CH2(D1-32a) CH2S (O)2CFThree
CH (Me) S (O) CH2(D1-32a) CH2CH (OMe)2
CH (Me) S (O) CH2(D1-32a) CH2CH (SMe)2
CH (Me) S (O) CH2(D1-32a) CH2C (O) Me
CH (Me) S (O) CH2(D1-32a) CH2C (O) CFThree
CH (Me) S (O) CH2(D1-32a) CH2C (O) OMe
CH (Me) S (O) CH2(D1-32a) CH2(D1-32a)
CH (Me) S (O) CH2(D1-32a) CH2(D1-33a)
CH (Me) S (O) CH2(D1-32a) CH2(D1-34a)
CH (Me) S (O) CH2(D1-32a) CH2(D1-37a)
CH (Me) S (O) CH2(D1-32a) CH2(D1-81a)
CH (Me) S (O) CH2(D1-32a) CH2(D1-82a)
CH (Me) S (O) CH2(D1-32a) CH2(D1-84a)
CH (Me) S (O) CH2(D1-32a) CH2(D1-85a)
CH (Me) S (O) CH2(D1-32a) CH2(D1-87a)
CH (Me) S (O) CH2(D1-32a) CH2(D1-92a)
CH (Me) S (O) CH2(D1-32a) CH2(D1-93a)
CH (Me) S (O) CH2(D1-32a) CH2(D1-95a)
CH (Me) S (O) CH2(D1-32a) CH2(D1-96a)
CH (Me) S (O) CH2(D1-32a) CH2(D1-98a)
CH (Me) S (O) CH2(D1-32a) CH2(D1-108a)
CH (Me) S (O) CH2(D1-32a) CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O) CH2(D1-32a) CH2(D1-108b, Z = 3-Me)
CH (Me) S (O) CH2(D1-32a) CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O) CH2(D1-32a) CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O) CH2(D1-32a) CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O) CH2(D1-32a) CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O) CH2(D1-32a) CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O) CH2(D1-32a) CH2CH2CN
CH (Me) S (O) CH2(D1-32a) CH2CH2CFThree
CH (Me) S (O) CH2(D1-32a) CH2CH2OMe
CH (Me) S (O) CH2(D1-32a) CH2CH2SMe
CH (Me) S (O) CH2(D1-32a) CH2CH2S (O) Me
CH (Me) S (O) CH2(D1-32a) CH2CH2S (O)2Me
CH (Me) S (O) CH2(D1-32a) D1-32a
CH (Me) S (O) CH2(D1-32a) D1-33a
CH (Me) S (O) CH2(D1-32a) D1-34a
CH (Me) S (O) CH2(D1-32a) D1-37a
CH (Me) S (O) CH2(D1-32a) D1-81a
CH (Me) S (O) CH2(D1-32a) D1-82a
CH (Me) S (O) CH2(D1-32a) D1-84a
CH (Me) S (O) CH2(D1-32a) D1-85a
CH (Me) S (O) CH2(D1-32a) D1-87a
CH (Me) S (O) CH2(D1-32a) D1-92a
CH (Me) S (O) CH2(D1-32a) D1-93a
CH (Me) S (O) CH2(D1-32a) D1-95a
CH (Me) S (O) CH2(D1-32a) D1-96a
CH (Me) S (O) CH2(D1-32a) D1-98a
CH (Me) S (O) CH2(D1-32a) D1-108a
CH (Me) S (O) CH2(D1-32a) D1-108b (Z = 2-Cl)
CH (Me) S (O) CH2(D1-32a) D1-108b (Z = 3-Me)
CH (Me) S (O) CH2(D1-32a) D1-108b (Z = 4-OMe)
CH (Me) S (O) CH2(D1-32a) D1-108b (Z = 2-SMe)
CH (Me) S (O) CH2(D1-32a) D1-108b (Z = 3-CFThree)
CH (Me) S (O) CH2(D1-32a) D1-108b (Z = 4-OCFThree)
CH (Me) S (O) CH2(D1-32a) D1-108b (Z = 2-SCFThree)
CH (Me) S (O) CH2(D1-32a) C (O) Me
CH (Me) S (O) CH2(D1-32a) C (O) CFThree
CH (Me) S (O) CH2(D1-32a) C (O) OMe
CH (Me) S (O)2CH2(D1-32a) Me
CH (Me) S (O)2CH2(D1-32a) Et
CH (Me) S (O)2CH2(D1-32a) Pr-n
CH (Me) S (O)2CH2(D1-32a) Pr-i
CH (Me) S (O)2CH2(D1-32a) Pr-c
CH (Me) S (O)2CH2(D1-32a) Bu-n
CH (Me) S (O)2CH2(D1-32a) Bu-i
CH (Me) S (O)2CH2(D1-32a) Bu-c
CH (Me) S (O)2CH2(D1-32a) Bu-s
CH (Me) S (O)2CH2(D1-32a) Bu-t
CH (Me) S (O)2CH2(D1-32a) Pen-n
CH (Me) S (O)2CH2(D1-32a) Pen-c
CH (Me) S (O)2CH2(D1-32a) Hex-n
CH (Me) S (O)2CH2(D1-32a) Hex-c
CH (Me) S (O)2CH2(D1-32a) CH2Pr-c
CH (Me) S (O)2CH2(D1-32a) CH2Bu-c
CH (Me) S (O)2CH2(D1-32a) CH2Pen-c
CH (Me) S (O)2CH2(D1-32a) CH2Hex-c
CH (Me) S (O)2CH2(D1-32a) CH2CH = CH2
CH (Me) S (O)2CH2(D1-32a) CH2CH = C (Cl)2
CH (Me) S (O)2CH2(D1-32a) CH2C≡CH
CH (Me) S (O)2CH2(D1-32a) CH2CN
CH (Me) S (O)2CH2(D1-32a) CH2CFThree
CH (Me) S (O)2CH2(D1-32a) CH2OMe
CH (Me) S (O)2CH2(D1-32a) CH2OCFThree
CH (Me) S (O)2CH2(D1-32a) CH2SMe
CH (Me) S (O)2CH2(D1-32a) CH2S (O) Me
CH (Me) S (O)2CH2(D1-32a) CH2S (O)2Me
CH (Me) S (O)2CH2(D1-32a) CH2SCFThree
CH (Me) S (O)2CH2(D1-32a) CH2S (O) CFThree
CH (Me) S (O)2CH2(D1-32a) CH2S (O)2CFThree
CH (Me) S (O)2CH2(D1-32a) CH2CH (OMe)2
CH (Me) S (O)2CH2(D1-32a) CH2CH (SMe)2
CH (Me) S (O)2CH2(D1-32a) CH2C (O) Me
CH (Me) S (O)2CH2(D1-32a) CH2C (O) CFThree
CH (Me) S (O)2CH2(D1-32a) CH2C (O) OMe
CH (Me) S (O)2CH2(D1-32a) CH2(D1-32a)
CH (Me) S (O)2CH2(D1-32a) CH2(D1-33a)
CH (Me) S (O)2CH2(D1-32a) CH2(D1-34a)
CH (Me) S (O)2CH2(D1-32a) CH2(D1-37a)
CH (Me) S (O)2CH2(D1-32a) CH2(D1-81a)
CH (Me) S (O)2CH2(D1-32a) CH2(D1-82a)
CH (Me) S (O)2CH2(D1-32a) CH2(D1-84a)
CH (Me) S (O)2CH2(D1-32a) CH2(D1-85a)
CH (Me) S (O)2CH2(D1-32a) CH2(D1-87a)
CH (Me) S (O)2CH2(D1-32a) CH2(D1-92a)
CH (Me) S (O)2CH2(D1-32a) CH2(D1-93a)
CH (Me) S (O)2CH2(D1-32a) CH2(D1-95a)
CH (Me) S (O)2CH2(D1-32a) CH2(D1-96a)
CH (Me) S (O)2CH2(D1-32a) CH2(D1-98a)
CH (Me) S (O)2CH2(D1-32a) CH2(D1-108a)
CH (Me) S (O)2CH2(D1-32a) CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O)2CH2(D1-32a) CH2(D1-108b, Z = 3-Me)
CH (Me) S (O)2CH2(D1-32a) CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O)2CH2(D1-32a) CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O)2CH2(D1-32a) CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O)2CH2(D1-32a) CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O)2CH2(D1-32a) CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O)2CH2(D1-32a) CH2CH2CN
CH (Me) S (O)2CH2(D1-32a) CH2CH2CFThree
CH (Me) S (O)2CH2(D1-32a) CH2CH2OMe
CH (Me) S (O)2CH2(D1-32a) CH2CH2SMe
CH (Me) S (O)2CH2(D1-32a) CH2CH2S (O) Me
CH (Me) S (O)2CH2(D1-32a) CH2CH2S (O)2Me
CH (Me) S (O)2CH2(D1-32a) D1-32a
CH (Me) S (O)2CH2(D1-32a) D1-33a
CH (Me) S (O)2CH2(D1-32a) D1-34a
CH (Me) S (O)2CH2(D1-32a) D1-37a
CH (Me) S (O)2CH2(D1-32a) D1-81a
CH (Me) S (O)2CH2(D1-32a) D1-82a
CH (Me) S (O)2CH2(D1-32a) D1-84a
CH (Me) S (O)2CH2(D1-32a) D1-85a
CH (Me) S (O)2CH2(D1-32a) D1-87a
CH (Me) S (O)2CH2(D1-32a) D1-92a
CH (Me) S (O)2CH2(D1-32a) D1-93a
CH (Me) S (O)2CH2(D1-32a) D1-95a
CH (Me) S (O)2CH2(D1-32a) D1-96a
CH (Me) S (O)2CH2(D1-32a) D1-98a
CH (Me) S (O)2CH2(D1-32a) D1-108a
CH (Me) S (O)2CH2(D1-32a) D1-108b (Z = 2-Cl)
CH (Me) S (O)2CH2(D1-32a) D1-108b (Z = 3-Me)
CH (Me) S (O)2CH2(D1-32a) D1-108b (Z = 4-OMe)
CH (Me) S (O)2CH2(D1-32a) D1-108b (Z = 2-SMe)
CH (Me) S (O)2CH2(D1-32a) D1-108b (Z = 3-CFThree)
CH (Me) S (O)2CH2(D1-32a) D1-108b (Z = 4-OCFThree)
CH (Me) S (O)2CH2(D1-32a) D1-108b (Z = 2-SCFThree)
CH (Me) S (O)2CH2(D1-32a) C (O) Me
CH (Me) S (O)2CH2(D1-32a) C (O) CFThree
CH (Me) S (O)2CH2(D1-32a) C (O) OMe
CH (Et) SCH2(D1-32a) Me
CH (Et) SCH2(D1-32a) Et
CH (Et) SCH2(D1-32a) Pr-n
CH (Et) SCH2(D1-32a) Pr-i
CH (Et) SCH2(D1-32a) Pr-c
CH (Et) SCH2(D1-32a) Bu-n
CH (Et) SCH2(D1-32a) Bu-i
CH (Et) SCH2(D1-32a) Bu-c
CH (Et) SCH2(D1-32a) Bu-s
CH (Et) SCH2(D1-32a) Bu-t
CH (Et) SCH2(D1-32a) Pen-n
CH (Et) SCH2(D1-32a) Pen-c
CH (Et) SCH2(D1-32a) Hex-n
CH (Et) SCH2(D1-32a) Hex-c
CH (Et) SCH2(D1-32a) CH2Pr-c
CH (Et) SCH2(D1-32a) CH2Bu-c
CH (Et) SCH2(D1-32a) CH2Pen-c
CH (Et) SCH2(D1-32a) CH2Hex-c
CH (Et) SCH2(D1-32a) CH2CH = CH2
CH (Et) SCH2(D1-32a) CH2CH = C (Cl)2
CH (Et) SCH2(D1-32a) CH2C≡CH
CH (Et) SCH2(D1-32a) CH2CN
CH (Et) SCH2(D1-32a) CH2CFThree
CH (Et) SCH2(D1-32a) CH2OMe
CH (Et) SCH2(D1-32a) CH2OCFThree
CH (Et) SCH2(D1-32a) CH2SMe
CH (Et) SCH2(D1-32a) CH2S (O) Me
CH (Et) SCH2(D1-32a) CH2S (O)2Me
CH (Et) SCH2(D1-32a) CH2SCFThree
CH (Et) SCH2(D1-32a) CH2S (O) CFThree
CH (Et) SCH2(D1-32a) CH2S (O)2CFThree
CH (Et) SCH2(D1-32a) CH2CH (OMe)2
CH (Et) SCH2(D1-32a) CH2CH (SMe)2
CH (Et) SCH2(D1-32a) CH2C (O) Me
CH (Et) SCH2(D1-32a) CH2C (O) CFThree
CH (Et) SCH2(D1-32a) CH2C (O) OMe
CH (Et) SCH2(D1-32a) CH2(D1-32a)
CH (Et) SCH2(D1-32a) CH2(D1-33a)
CH (Et) SCH2(D1-32a) CH2(D1-34a)
CH (Et) SCH2(D1-32a) CH2(D1-37a)
CH (Et) SCH2(D1-32a) CH2(D1-81a)
CH (Et) SCH2(D1-32a) CH2(D1-82a)
CH (Et) SCH2(D1-32a) CH2(D1-84a)
CH (Et) SCH2(D1-32a) CH2(D1-85a)
CH (Et) SCH2(D1-32a) CH2(D1-87a)
CH (Et) SCH2(D1-32a) CH2(D1-92a)
CH (Et) SCH2(D1-32a) CH2(D1-93a)
CH (Et) SCH2(D1-32a) CH2(D1-95a)
CH (Et) SCH2(D1-32a) CH2(D1-96a)
CH (Et) SCH2(D1-32a) CH2(D1-98a)
CH (Et) SCH2(D1-32a) CH2(D1-108a)
CH (Et) SCH2(D1-32a) CH2(D1-108b, Z = 2-Cl)
CH (Et) SCH2(D1-32a) CH2(D1-108b, Z = 3-Me)
CH (Et) SCH2(D1-32a) CH2(D1-108b, Z = 4-OMe)
CH (Et) SCH2(D1-32a) CH2(D1-108b, Z = 2-SMe)
CH (Et) SCH2(D1-32a) CH2(D1-108b, Z = 3-CFThree)
CH (Et) SCH2(D1-32a) CH2(D1-108b, Z = 4-OCFThree)
CH (Et) SCH2(D1-32a) CH2(D1-108b, Z = 2-SCFThree)
CH (Et) SCH2(D1-32a) CH2CH2CN
CH (Et) SCH2(D1-32a) CH2CH2CFThree
CH (Et) SCH2(D1-32a) CH2CH2OMe
CH (Et) SCH2(D1-32a) CH2CH2SMe
CH (Et) SCH2(D1-32a) CH2CH2S (O) Me
CH (Et) SCH2(D1-32a) CH2CH2S (O)2Me
CH (Et) SCH2(D1-32a) D1-32a
CH (Et) SCH2(D1-32a) D1-33a
CH (Et) SCH2(D1-32a) D1-34a
CH (Et) SCH2(D1-32a) D1-37a
CH (Et) SCH2(D1-32a) D1-81a
CH (Et) SCH2(D1-32a) D1-82a
CH (Et) SCH2(D1-32a) D1-84a
CH (Et) SCH2(D1-32a) D1-85a
CH (Et) SCH2(D1-32a) D1-87a
CH (Et) SCH2(D1-32a) D1-92a
CH (Et) SCH2(D1-32a) D1-93a
CH (Et) SCH2(D1-32a) D1-95a
CH (Et) SCH2(D1-32a) D1-96a
CH (Et) SCH2(D1-32a) D1-98a
CH (Et) SCH2(D1-32a) D1-108a
CH (Et) SCH2(D1-32a) D1-108b (Z = 2-Cl)
CH (Et) SCH2(D1-32a) D1-108b (Z = 3-Me)
CH (Et) SCH2(D1-32a) D1-108b (Z = 4-OMe)
CH (Et) SCH2(D1-32a) D1-108b (Z = 2-SMe)
CH (Et) SCH2(D1-32a) D1-108b (Z = 3-CFThree)
CH (Et) SCH2(D1-32a) D1-108b (Z = 4-OCFThree)
CH (Et) SCH2(D1-32a) D1-108b (Z = 2-SCFThree)
CH (Et) SCH2(D1-32a) C (O) Me
CH (Et) SCH2(D1-32a) C (O) CFThree
CH (Et) SCH2(D1-32a) C (O) OMe
CH (Et) S (O) CH2(D1-32a) Me
CH (Et) S (O) CH2(D1-32a) Et
CH (Et) S (O) CH2(D1-32a) Pr-n
CH (Et) S (O) CH2(D1-32a) Pr-i
CH (Et) S (O) CH2(D1-32a) Pr-c
CH (Et) S (O) CH2(D1-32a) Bu-n
CH (Et) S (O) CH2(D1-32a) Bu-i
CH (Et) S (O) CH2(D1-32a) Bu-c
CH (Et) S (O) CH2(D1-32a) Bu-s
CH (Et) S (O) CH2(D1-32a) Bu-t
CH (Et) S (O) CH2(D1-32a) Pen-n
CH (Et) S (O) CH2(D1-32a) Pen-c
CH (Et) S (O) CH2(D1-32a) Hex-n
CH (Et) S (O) CH2(D1-32a) Hex-c
CH (Et) S (O) CH2(D1-32a) CH2Pr-c
CH (Et) S (O) CH2(D1-32a) CH2Bu-c
CH (Et) S (O) CH2(D1-32a) CH2Pen-c
CH (Et) S (O) CH2(D1-32a) CH2Hex-c
CH (Et) S (O) CH2(D1-32a) CH2CH = CH2
CH (Et) S (O) CH2(D1-32a) CH2CH = C (Cl)2
CH (Et) S (O) CH2(D1-32a) CH2C≡CH
CH (Et) S (O) CH2(D1-32a) CH2CN
CH (Et) S (O) CH2(D1-32a) CH2CFThree
CH (Et) S (O) CH2(D1-32a) CH2OMe
CH (Et) S (O) CH2(D1-32a) CH2OCFThree
CH (Et) S (O) CH2(D1-32a) CH2SMe
CH (Et) S (O) CH2(D1-32a) CH2S (O) Me
CH (Et) S (O) CH2(D1-32a) CH2S (O)2Me
CH (Et) S (O) CH2(D1-32a) CH2SCFThree
CH (Et) S (O) CH2(D1-32a) CH2S (O) CFThree
CH (Et) S (O) CH2(D1-32a) CH2S (O)2CFThree
CH (Et) S (O) CH2(D1-32a) CH2CH (OMe)2
CH (Et) S (O) CH2(D1-32a) CH2CH (SMe)2
CH (Et) S (O) CH2(D1-32a) CH2C (O) Me
CH (Et) S (O) CH2(D1-32a) CH2C (O) CFThree
CH (Et) S (O) CH2(D1-32a) CH2C (O) OMe
CH (Et) S (O) CH2(D1-32a) CH2(D1-32a)
CH (Et) S (O) CH2(D1-32a) CH2(D1-33a)
CH (Et) S (O) CH2(D1-32a) CH2(D1-34a)
CH (Et) S (O) CH2(D1-32a) CH2(D1-37a)
CH (Et) S (O) CH2(D1-32a) CH2(D1-81a)
CH (Et) S (O) CH2(D1-32a) CH2(D1-82a)
CH (Et) S (O) CH2(D1-32a) CH2(D1-84a)
CH (Et) S (O) CH2(D1-32a) CH2(D1-85a)
CH (Et) S (O) CH2(D1-32a) CH2(D1-87a)
CH (Et) S (O) CH2(D1-32a) CH2(D1-92a)
CH (Et) S (O) CH2(D1-32a) CH2(D1-93a)
CH (Et) S (O) CH2(D1-32a) CH2(D1-95a)
CH (Et) S (O) CH2(D1-32a) CH2(D1-96a)
CH (Et) S (O) CH2(D1-32a) CH2(D1-98a)
CH (Et) S (O) CH2(D1-32a) CH2(D1-108a)
CH (Et) S (O) CH2(D1-32a) CH2(D1-108b, Z = 2-Cl)
CH (Et) S (O) CH2(D1-32a) CH2(D1-108b, Z = 3-Me)
CH (Et) S (O) CH2(D1-32a) CH2(D1-108b, Z = 4-OMe)
CH (Et) S (O) CH2(D1-32a) CH2(D1-108b, Z = 2-SMe)
CH (Et) S (O) CH2(D1-32a) CH2(D1-108b, Z = 3-CFThree)
CH (Et) S (O) CH2(D1-32a) CH2(D1-108b, Z = 4-OCFThree)
CH (Et) S (O) CH2(D1-32a) CH2(D1-108b, Z = 2-SCFThree)
CH (Et) S (O) CH2(D1-32a) CH2CH2CN
CH (Et) S (O) CH2(D1-32a) CH2CH2CFThree
CH (Et) S (O) CH2(D1-32a) CH2CH2OMe
CH (Et) S (O) CH2(D1-32a) CH2CH2SMe
CH (Et) S (O) CH2(D1-32a) CH2CH2S (O) Me
CH (Et) S (O) CH2(D1-32a) CH2CH2S (O)2Me
CH (Et) S (O) CH2(D1-32a) D1-32a
CH (Et) S (O) CH2(D1-32a) D1-33a
CH (Et) S (O) CH2(D1-32a) D1-34a
CH (Et) S (O) CH2(D1-32a) D1-37a
CH (Et) S (O) CH2(D1-32a) D1-81a
CH (Et) S (O) CH2(D1-32a) D1-82a
CH (Et) S (O) CH2(D1-32a) D1-84a
CH (Et) S (O) CH2(D1-32a) D1-85a
CH (Et) S (O) CH2(D1-32a) D1-87a
CH (Et) S (O) CH2(D1-32a) D1-92a
CH (Et) S (O) CH2(D1-32a) D1-93a
CH (Et) S (O) CH2(D1-32a) D1-95a
CH (Et) S (O) CH2(D1-32a) D1-96a
CH (Et) S (O) CH2(D1-32a) D1-98a
CH (Et) S (O) CH2(D1-32a) D1-108a
CH (Et) S (O) CH2(D1-32a) D1-108b (Z = 2-Cl)
CH (Et) S (O) CH2(D1-32a) D1-108b (Z = 3-Me)
CH (Et) S (O) CH2(D1-32a) D1-108b (Z = 4-OMe)
CH (Et) S (O) CH2(D1-32a) D1-108b (Z = 2-SMe)
CH (Et) S (O) CH2(D1-32a) D1-108b (Z = 3-CFThree)
CH (Et) S (O) CH2(D1-32a) D1-108b (Z = 4-OCFThree)
CH (Et) S (O) CH2(D1-32a) D1-108b (Z = 2-SCFThree)
CH (Et) S (O) CH2(D1-32a) C (O) Me
CH (Et) S (O) CH2(D1-32a) C (O) CFThree
CH (Et) S (O) CH2(D1-32a) C (O) OMe
CH (Et) S (O)2CH2(D1-32a) Me
CH (Et) S (O)2CH2(D1-32a) Et
CH (Et) S (O)2CH2(D1-32a) Pr-n
CH (Et) S (O)2CH2(D1-32a) Pr-i
CH (Et) S (O)2CH2(D1-32a) Pr-c
CH (Et) S (O)2CH2(D1-32a) Bu-n
CH (Et) S (O)2CH2(D1-32a) Bu-i
CH (Et) S (O)2CH2(D1-32a) Bu-c
CH (Et) S (O)2CH2(D1-32a) Bu-s
CH (Et) S (O)2CH2(D1-32a) Bu-t
CH (Et) S (O)2CH2(D1-32a) Pen-n
CH (Et) S (O)2CH2(D1-32a) Pen-c
CH (Et) S (O)2CH2(D1-32a) Hex-n
CH (Et) S (O)2CH2(D1-32a) Hex-c
CH (Et) S (O)2CH2(D1-32a) CH2Pr-c
CH (Et) S (O)2CH2(D1-32a) CH2Bu-c
CH (Et) S (O)2CH2(D1-32a) CH2Pen-c
CH (Et) S (O)2CH2(D1-32a) CH2Hex-c
CH (Et) S (O)2CH2(D1-32a) CH2CH = CH2
CH (Et) S (O)2CH2(D1-32a) CH2CH = C (Cl)2
CH (Et) S (O)2CH2(D1-32a) CH2C≡CH
CH (Et) S (O)2CH2(D1-32a) CH2CN
CH (Et) S (O)2CH2(D1-32a) CH2CFThree
CH (Et) S (O)2CH2(D1-32a) CH2OMe
CH (Et) S (O)2CH2(D1-32a) CH2OCFThree
CH (Et) S (O)2CH2(D1-32a) CH2SMe
CH (Et) S (O)2CH2(D1-32a) CH2S (O) Me
CH (Et) S (O)2CH2(D1-32a) CH2S (O)2Me
CH (Et) S (O)2CH2(D1-32a) CH2SCFThree
CH (Et) S (O)2CH2(D1-32a) CH2S (O) CFThree
CH (Et) S (O)2CH2(D1-32a) CH2S (O)2CFThree
CH (Et) S (O)2CH2(D1-32a) CH2CH (OMe)2
CH (Et) S (O)2CH2(D1-32a) CH2CH (SMe)2
CH (Et) S (O)2CH2(D1-32a) CH2C (O) Me
CH (Et) S (O)2CH2(D1-32a) CH2C (O) CFThree
CH (Et) S (O)2CH2(D1-32a) CH2C (O) OMe
CH (Et) S (O)2CH2(D1-32a) CH2(D1-32a)
CH (Et) S (O)2CH2(D1-32a) CH2(D1-33a)
CH (Et) S (O)2CH2(D1-32a) CH2(D1-34a)
CH (Et) S (O)2CH2(D1-32a) CH2(D1-37a)
CH (Et) S (O)2CH2(D1-32a) CH2(D1-81a)
CH (Et) S (O)2CH2(D1-32a) CH2(D1-82a)
CH (Et) S (O)2CH2(D1-32a) CH2(D1-84a)
CH (Et) S (O)2CH2(D1-32a) CH2(D1-85a)
CH (Et) S (O)2CH2(D1-32a) CH2(D1-87a)
CH (Et) S (O)2CH2(D1-32a) CH2(D1-92a)
CH (Et) S (O)2CH2(D1-32a) CH2(D1-93a)
CH (Et) S (O)2CH2(D1-32a) CH2(D1-95a)
CH (Et) S (O)2CH2(D1-32a) CH2(D1-96a)
CH (Et) S (O)2CH2(D1-32a) CH2(D1-98a)
CH (Et) S (O)2CH2(D1-32a) CH2(D1-108a)
CH (Et) S (O)2CH2(D1-32a) CH2(D1-108b, Z = 2-Cl)
CH (Et) S (O)2CH2(D1-32a) CH2(D1-108b, Z = 3-Me)
CH (Et) S (O)2CH2(D1-32a) CH2(D1-108b, Z = 4-OMe)
CH (Et) S (O)2CH2(D1-32a) CH2(D1-108b, Z = 2-SMe)
CH (Et) S (O)2CH2(D1-32a) CH2(D1-108b, Z = 3-CFThree)
CH (Et) S (O)2CH2(D1-32a) CH2(D1-108b, Z = 4-OCFThree)
CH (Et) S (O)2CH2(D1-32a) CH2(D1-108b, Z = 2-SCFThree)
CH (Et) S (O)2CH2(D1-32a) CH2CH2CN
CH (Et) S (O)2CH2(D1-32a) CH2CH2CFThree
CH (Et) S (O)2CH2(D1-32a) CH2CH2OMe
CH (Et) S (O)2CH2(D1-32a) CH2CH2SMe
CH (Et) S (O)2CH2(D1-32a) CH2CH2S (O) Me
CH (Et) S (O)2CH2(D1-32a) CH2CH2S (O)2Me
CH (Et) S (O)2CH2(D1-32a) D1-32a
CH (Et) S (O)2CH2(D1-32a) D1-33a
CH (Et) S (O)2CH2(D1-32a) D1-34a
CH (Et) S (O)2CH2(D1-32a) D1-37a
CH (Et) S (O)2CH2(D1-32a) D1-81a
CH (Et) S (O)2CH2(D1-32a) D1-82a
CH (Et) S (O)2CH2(D1-32a) D1-84a
CH (Et) S (O)2CH2(D1-32a) D1-85a
CH (Et) S (O)2CH2(D1-32a) D1-87a
CH (Et) S (O)2CH2(D1-32a) D1-92a
CH (Et) S (O)2CH2(D1-32a) D1-93a
CH (Et) S (O)2CH2(D1-32a) D1-95a
CH (Et) S (O)2CH2(D1-32a) D1-96a
CH (Et) S (O)2CH2(D1-32a) D1-98a
CH (Et) S (O)2CH2(D1-32a) D1-108a
CH (Et) S (O)2CH2(D1-32a) D1-108b (Z = 2-Cl)
CH (Et) S (O)2CH2(D1-32a) D1-108b (Z = 3-Me)
CH (Et) S (O)2CH2(D1-32a) D1-108b (Z = 4-OMe)
CH (Et) S (O)2CH2(D1-32a) D1-108b (Z = 2-SMe)
CH (Et) S (O)2CH2(D1-32a) D1-108b (Z = 3-CFThree)
CH (Et) S (O)2CH2(D1-32a) D1-108b (Z = 4-OCFThree)
CH (Et) S (O)2CH2(D1-32a) D1-108b (Z = 2-SCFThree)
CH (Et) S (O)2CH2(D1-32a) C (O) Me
CH (Et) S (O)2CH2(D1-32a) C (O) CFThree
CH2SCH2(D1-33a) Me
CH2SCH2(D1-33a) Et
CH2SCH2(D1-33a) Pr-n
CH2SCH2(D1-33a) Pr-i
CH2SCH2(D1-33a) Pr-c
CH2SCH2(D1-33a) Bu-n
CH2SCH2(D1-33a) Bu-i
CH2SCH2(D1-33a) Bu-c
CH2SCH2(D1-33a) Bu-s
CH2SCH2(D1-33a) Bu-t
CH2SCH2(D1-33a) Pen-n
CH2SCH2(D1-33a) Pen-c
CH2SCH2(D1-33a) Hex-n
CH2SCH2(D1-33a) Hex-c
CH2SCH2(D1-33a) CH2Pr-c
CH2SCH2(D1-33a) CH2Bu-c
CH2SCH2(D1-33a) CH2Pen-c
CH2SCH2(D1-33a) CH2Hex-c
CH2SCH2(D1-33a) CH2CH = CH2
CH2SCH2(D1-33a) CH2CH = C (Cl)2
CH2SCH2(D1-33a) CH2C≡CH
CH2SCH2(D1-33a) CH2CN
CH2SCH2(D1-33a) CH2CFThree
CH2SCH2(D1-33a) CH2OMe
CH2SCH2(D1-33a) CH2OCFThree
CH2SCH2(D1-33a) CH2SMe
CH2SCH2(D1-33a) CH2S (O) Me
CH2SCH2(D1-33a) CH2S (O)2Me
CH2SCH2(D1-33a) CH2SCFThree
CH2SCH2(D1-33a) CH2S (O) CFThree
CH2SCH2(D1-33a) CH2S (O)2CFThree
CH2SCH2(D1-33a) CH2CH (OMe)2
CH2SCH2(D1-33a) CH2CH (SMe)2
CH2SCH2(D1-33a) CH2C (O) Me
CH2SCH2(D1-33a) CH2C (O) CFThree
CH2SCH2(D1-33a) CH2C (O) OMe
CH2SCH2(D1-33a) CH2(D1-32a)
CH2SCH2(D1-33a) CH2(D1-33a)
CH2SCH2(D1-33a) CH2(D1-34a)
CH2SCH2(D1-33a) CH2(D1-37a)
CH2SCH2(D1-33a) CH2(D1-81a)
CH2SCH2(D1-33a) CH2(D1-82a)
CH2SCH2(D1-33a) CH2(D1-84a)
CH2SCH2(D1-33a) CH2(D1-85a)
CH2SCH2(D1-33a) CH2(D1-87a)
CH2SCH2(D1-33a) CH2(D1-92a)
CH2SCH2(D1-33a) CH2(D1-93a)
CH2SCH2(D1-33a) CH2(D1-95a)
CH2SCH2(D1-33a) CH2(D1-96a)
CH2SCH2(D1-33a) CH2(D1-98a)
CH2SCH2(D1-33a) CH2(D1-108a)
CH2SCH2(D1-33a) CH2(D1-108b, Z = 2-Cl)
CH2SCH2(D1-33a) CH2(D1-108b, Z = 3-Me)
CH2SCH2(D1-33a) CH2(D1-108b, Z = 4-OMe)
CH2SCH2(D1-33a) CH2(D1-108b, Z = 2-SMe)
CH2SCH2(D1-33a) CH2(D1-108b, Z = 3-CFThree)
CH2SCH2(D1-33a) CH2(D1-108b, Z = 4-OCFThree)
CH2SCH2(D1-33a) CH2(D1-108b, Z = 2-SCFThree)
CH2SCH2(D1-33a) CH2CH2CN
CH2SCH2(D1-33a) CH2CH2CFThree
CH2SCH2(D1-33a) CH2CH2OMe
CH2SCH2(D1-33a) CH2CH2SMe
CH2SCH2(D1-33a) CH2CH2S (O) Me
CH2SCH2(D1-33a) CH2CH2S (O)2Me
CH2SCH2(D1-33a) D1-32a
CH2SCH2(D1-33a) D1-33a
CH2SCH2(D1-33a) D1-34a
CH2SCH2(D1-33a) D1-37a
CH2SCH2(D1-33a) D1-81a
CH2SCH2(D1-33a) D1-82a
CH2SCH2(D1-33a) D1-84a
CH2SCH2(D1-33a) D1-85a
CH2SCH2(D1-33a) D1-87a
CH2SCH2(D1-33a) D1-92a
CH2SCH2(D1-33a) D1-93a
CH2SCH2(D1-33a) D1-95a
CH2SCH2(D1-33a) D1-96a
CH2SCH2(D1-33a) D1-98a
CH2SCH2(D1-33a) D1-108a
CH2SCH2(D1-33a) D1-108b (Z = 2-Cl)
CH2SCH2(D1-33a) D1-108b (Z = 3-Me)
CH2SCH2(D1-33a) D1-108b (Z = 4-OMe)
CH2SCH2(D1-33a) D1-108b (Z = 2-SMe)
CH2SCH2(D1-33a) D1-108b (Z = 3-CFThree)
CH2SCH2(D1-33a) D1-108b (Z = 4-OCFThree)
CH2SCH2(D1-33a) D1-108b (Z = 2-SCFThree)
CH2SCH2(D1-33a) C (O) Me
CH2SCH2(D1-33a) C (O) CFThree
CH2SCH2(D1-33a) C (O) OMe
CH2S (O) CH2(D1-33a) Me
CH2S (O) CH2(D1-33a) Et
CH2S (O) CH2(D1-33a) Pr-n
CH2S (O) CH2(D1-33a) Pr-i
CH2S (O) CH2(D1-33a) Pr-c
CH2S (O) CH2(D1-33a) Bu-n
CH2S (O) CH2(D1-33a) Bu-i
CH2S (O) CH2(D1-33a) Bu-c
CH2S (O) CH2(D1-33a) Bu-s
CH2S (O) CH2(D1-33a) Bu-t
CH2S (O) CH2(D1-33a) Pen-n
CH2S (O) CH2(D1-33a) Pen-c
CH2S (O) CH2(D1-33a) Hex-n
CH2S (O) CH2(D1-33a) Hex-c
CH2S (O) CH2(D1-33a) CH2Pr-c
CH2S (O) CH2(D1-33a) CH2Bu-c
CH2S (O) CH2(D1-33a) CH2Pen-c
CH2S (O) CH2(D1-33a) CH2Hex-c
CH2S (O) CH2(D1-33a) CH2CH = CH2
CH2S (O) CH2(D1-33a) CH2CH = C (Cl)2
CH2S (O) CH2(D1-33a) CH2C≡CH
CH2S (O) CH2(D1-33a) CH2CN
CH2S (O) CH2(D1-33a) CH2CFThree
CH2S (O) CH2(D1-33a) CH2OMe
CH2S (O) CH2(D1-33a) CH2OCFThree
CH2S (O) CH2(D1-33a) CH2SMe
CH2S (O) CH2(D1-33a) CH2S (O) Me
CH2S (O) CH2(D1-33a) CH2S (O)2Me
CH2S (O) CH2(D1-33a) CH2SCFThree
CH2S (O) CH2(D1-33a) CH2S (O) CFThree
CH2S (O) CH2(D1-33a) CH2S (O)2CFThree
CH2S (O) CH2(D1-33a) CH2CH (OMe)2
CH2S (O) CH2(D1-33a) CH2CH (SMe)2
CH2S (O) CH2(D1-33a) CH2C (O) Me
CH2S (O) CH2(D1-33a) CH2C (O) CFThree
CH2S (O) CH2(D1-33a) CH2C (O) OMe
CH2S (O) CH2(D1-33a) CH2(D1-32a)
CH2S (O) CH2(D1-33a) CH2(D1-33a)
CH2S (O) CH2(D1-33a) CH2(D1-34a)
CH2S (O) CH2(D1-33a) CH2(D1-37a)
CH2S (O) CH2(D1-33a) CH2(D1-81a)
CH2S (O) CH2(D1-33a) CH2(D1-82a)
CH2S (O) CH2(D1-33a) CH2(D1-84a)
CH2S (O) CH2(D1-33a) CH2(D1-85a)
CH2S (O) CH2(D1-33a) CH2(D1-87a)
CH2S (O) CH2(D1-33a) CH2(D1-92a)
CH2S (O) CH2(D1-33a) CH2(D1-93a)
CH2S (O) CH2(D1-33a) CH2(D1-95a)
CH2S (O) CH2(D1-33a) CH2(D1-96a)
CH2S (O) CH2(D1-33a) CH2(D1-98a)
CH2S (O) CH2(D1-33a) CH2(D1-108a)
CH2S (O) CH2(D1-33a) CH2(D1-108b, Z = 2-Cl)
CH2S (O) CH2(D1-33a) CH2(D1-108b, Z = 3-Me)
CH2S (O) CH2(D1-33a) CH2(D1-108b, Z = 4-OMe)
CH2S (O) CH2(D1-33a) CH2(D1-108b, Z = 2-SMe)
CH2S (O) CH2(D1-33a) CH2(D1-108b, Z = 3-CFThree)
CH2S (O) CH2(D1-33a) CH2(D1-108b, Z = 4-OCFThree)
CH2S (O) CH2(D1-33a) CH2(D1-108b, Z = 2-SCFThree)
CH2S (O) CH2(D1-33a) CH2CH2CN
CH2S (O) CH2(D1-33a) CH2CH2CFThree
CH2S (O) CH2(D1-33a) CH2CH2OMe
CH2S (O) CH2(D1-33a) CH2CH2SMe
CH2S (O) CH2(D1-33a) CH2CH2S (O) Me
CH2S (O) CH2(D1-33a) CH2CH2S (O)2Me
CH2S (O) CH2(D1-33a) D1-32a
CH2S (O) CH2(D1-33a) D1-33a
CH2S (O) CH2(D1-33a) D1-34a
CH2S (O) CH2(D1-33a) D1-37a
CH2S (O) CH2(D1-33a) D1-81a
CH2S (O) CH2(D1-33a) D1-82a
CH2S (O) CH2(D1-33a) D1-84a
CH2S (O) CH2(D1-33a) D1-85a
CH2S (O) CH2(D1-33a) D1-87a
CH2S (O) CH2(D1-33a) D1-92a
CH2S (O) CH2(D1-33a) D1-93a
CH2S (O) CH2(D1-33a) D1-95a
CH2S (O) CH2(D1-33a) D1-96a
CH2S (O) CH2(D1-33a) D1-98a
CH2S (O) CH2(D1-33a) D1-108a
CH2S (O) CH2(D1-33a) D1-108b (Z = 2-Cl)
CH2S (O) CH2(D1-33a) D1-108b (Z = 3-Me)
CH2S (O) CH2(D1-33a) D1-108b (Z = 4-OMe)
CH2S (O) CH2(D1-33a) D1-108b (Z = 2-SMe)
CH2S (O) CH2(D1-33a) D1-108b (Z = 3-CFThree)
CH2S (O) CH2(D1-33a) D1-108b (Z = 4-OCFThree)
CH2S (O) CH2(D1-33a) D1-108b (Z = 2-SCFThree)
CH2S (O) CH2(D1-33a) C (O) Me
CH2S (O) CH2(D1-33a) C (O) CFThree
CH2S (O) CH2(D1-33a) C (O) OMe
CH2S (O)2CH2(D1-33a) Me
CH2S (O)2CH2(D1-33a) Et
CH2S (O)2CH2(D1-33a) Pr-n
CH2S (O)2CH2(D1-33a) Pr-i
CH2S (O)2CH2(D1-33a) Pr-c
CH2S (O)2CH2(D1-33a) Bu-n
CH2S (O)2CH2(D1-33a) Bu-i
CH2S (O)2CH2(D1-33a) Bu-c
CH2S (O)2CH2(D1-33a) Bu-s
CH2S (O)2CH2(D1-33a) Bu-t
CH2S (O)2CH2(D1-33a) Pen-n
CH2S (O)2CH2(D1-33a) Pen-c
CH2S (O)2CH2(D1-33a) Hex-n
CH2S (O)2CH2(D1-33a) Hex-c
CH2S (O)2CH2(D1-33a) CH2Pr-c
CH2S (O)2CH2(D1-33a) CH2Bu-c
CH2S (O)2CH2(D1-33a) CH2Pen-c
CH2S (O)2CH2(D1-33a) CH2Hex-c
CH2S (O)2CH2(D1-33a) CH2CH = CH2
CH2S (O)2CH2(D1-33a) CH2CH = C (Cl)2
CH2S (O)2CH2(D1-33a) CH2C≡CH
CH2S (O)2CH2(D1-33a) CH2CN
CH2S (O)2CH2(D1-33a) CH2CFThree
CH2S (O)2CH2(D1-33a) CH2OMe
CH2S (O)2CH2(D1-33a) CH2OCFThree
CH2S (O)2CH2(D1-33a) CH2SMe
CH2S (O)2CH2(D1-33a) CH2S (O) Me
CH2S (O)2CH2(D1-33a) CH2S (O)2Me
CH2S (O)2CH2(D1-33a) CH2SCFThree
CH2S (O)2CH2(D1-33a) CH2S (O) CFThree
CH2S (O)2CH2(D1-33a) CH2S (O)2CFThree
CH2S (O)2CH2(D1-33a) CH2CH (OMe)2
CH2S (O)2CH2(D1-33a) CH2CH (SMe)2
CH2S (O)2CH2(D1-33a) CH2C (O) Me
CH2S (O)2CH2(D1-33a) CH2C (O) CFThree
CH2S (O)2CH2(D1-33a) CH2C (O) OMe
CH2S (O)2CH2(D1-33a) CH2(D1-32a)
CH2S (O)2CH2(D1-33a) CH2(D1-33a)
CH2S (O)2CH2(D1-33a) CH2(D1-34a)
CH2S (O)2CH2(D1-33a) CH2(D1-37a)
CH2S (O)2CH2(D1-33a) CH2(D1-81a)
CH2S (O)2CH2(D1-33a) CH2(D1-82a)
CH2S (O)2CH2(D1-33a) CH2(D1-84a)
CH2S (O)2CH2(D1-33a) CH2(D1-85a)
CH2S (O)2CH2(D1-33a) CH2(D1-87a)
CH2S (O)2CH2(D1-33a) CH2(D1-92a)
CH2S (O)2CH2(D1-33a) CH2(D1-93a)
CH2S (O)2CH2(D1-33a) CH2(D1-95a)
CH2S (O)2CH2(D1-33a) CH2(D1-96a)
CH2S (O)2CH2(D1-33a) CH2(D1-98a)
CH2S (O)2CH2(D1-33a) CH2(D1-108a)
CH2S (O)2CH2(D1-33a) CH2(D1-108b, Z = 2-Cl)
CH2S (O)2CH2(D1-33a) CH2(D1-108b, Z = 3-Me)
CH2S (O)2CH2(D1-33a) CH2(D1-108b, Z = 4-OMe)
CH2S (O)2CH2(D1-33a) CH2(D1-108b, Z = 2-SMe)
CH2S (O)2CH2(D1-33a) CH2(D1-108b, Z = 3-CFThree)
CH2S (O)2CH2(D1-33a) CH2(D1-108b, Z = 4-OCFThree)
CH2S (O)2CH2(D1-33a) CH2(D1-108b, Z = 2-SCFThree)
CH2S (O)2CH2(D1-33a) CH2CH2CN
CH2S (O)2CH2(D1-33a) CH2CH2CFThree
CH2S (O)2CH2(D1-33a) CH2CH2OMe
CH2S (O)2CH2(D1-33a) CH2CH2SMe
CH2S (O)2CH2(D1-33a) CH2CH2S (O) Me
CH2S (O)2CH2(D1-33a) CH2CH2S (O)2Me
CH2S (O)2CH2(D1-33a) D1-32a
CH2S (O)2CH2(D1-33a) D1-33a
CH2S (O)2CH2(D1-33a) D1-34a
CH2S (O)2CH2(D1-33a) D1-37a
CH2S (O)2CH2(D1-33a) D1-81a
CH2S (O)2CH2(D1-33a) D1-82a
CH2S (O)2CH2(D1-33a) D1-84a
CH2S (O)2CH2(D1-33a) D1-85a
CH2S (O)2CH2(D1-33a) D1-87a
CH2S (O)2CH2(D1-33a) D1-92a
CH2S (O)2CH2(D1-33a) D1-93a
CH2S (O)2CH2(D1-33a) D1-95a
CH2S (O)2CH2(D1-33a) D1-96a
CH2S (O)2CH2(D1-33a) D1-98a
CH2S (O)2CH2(D1-33a) D1-108a
CH2S (O)2CH2(D1-33a) D1-108b (Z = 2-Cl)
CH2S (O)2CH2(D1-33a) D1-108b (Z = 3-Me)
CH2S (O)2CH2(D1-33a) D1-108b (Z = 4-OMe)
CH2S (O)2CH2(D1-33a) D1-108b (Z = 2-SMe)
CH2S (O)2CH2(D1-33a) D1-108b (Z = 3-CFThree)
CH2S (O)2CH2(D1-33a) D1-108b (Z = 4-OCFThree)
CH2S (O)2CH2(D1-33a) D1-108b (Z = 2-SCFThree)
CH2S (O)2CH2(D1-33a) C (O) Me
CH2S (O)2CH2(D1-33a) C (O) CFThree
CH2S (O)2CH2(D1-33a) C (O) OMe
CH (Me) SCH2(D1-33a) Me
CH (Me) SCH2(D1-33a) Et
CH (Me) SCH2(D1-33a) Pr-n
CH (Me) SCH2(D1-33a) Pr-i
CH (Me) SCH2(D1-33a) Pr-c
CH (Me) SCH2(D1-33a) Bu-n
CH (Me) SCH2(D1-33a) Bu-i
CH (Me) SCH2(D1-33a) Bu-c
CH (Me) SCH2(D1-33a) Bu-s
CH (Me) SCH2(D1-33a) Bu-t
CH (Me) SCH2(D1-33a) Pen-n
CH (Me) SCH2(D1-33a) Pen-c
CH (Me) SCH2(D1-33a) Hex-n
CH (Me) SCH2(D1-33a) Hex-c
CH (Me) SCH2(D1-33a) CH2Pr-c
CH (Me) SCH2(D1-33a) CH2Bu-c
CH (Me) SCH2(D1-33a) CH2Pen-c
CH (Me) SCH2(D1-33a) CH2Hex-c
CH (Me) SCH2(D1-33a) CH2CH = CH2
CH (Me) SCH2(D1-33a) CH2CH = C (Cl)2
CH (Me) SCH2(D1-33a) CH2C≡CH
CH (Me) SCH2(D1-33a) CH2CN
CH (Me) SCH2(D1-33a) CH2CFThree
CH (Me) SCH2(D1-33a) CH2OMe
CH (Me) SCH2(D1-33a) CH2OCFThree
CH (Me) SCH2(D1-33a) CH2SMe
CH (Me) SCH2(D1-33a) CH2S (O) Me
CH (Me) SCH2(D1-33a) CH2S (O)2Me
CH (Me) SCH2(D1-33a) CH2SCFThree
CH (Me) SCH2(D1-33a) CH2S (O) CFThree
CH (Me) SCH2(D1-33a) CH2S (O)2CFThree
CH (Me) SCH2(D1-33a) CH2CH (OMe)2
CH (Me) SCH2(D1-33a) CH2CH (SMe)2
CH (Me) SCH2(D1-33a) CH2C (O) Me
CH (Me) SCH2(D1-33a) CH2C (O) CFThree
CH (Me) SCH2(D1-33a) CH2C (O) OMe
CH (Me) SCH2(D1-33a) CH2(D1-32a)
CH (Me) SCH2(D1-33a) CH2(D1-33a)
CH (Me) SCH2(D1-33a) CH2(D1-34a)
CH (Me) SCH2(D1-33a) CH2(D1-37a)
CH (Me) SCH2(D1-33a) CH2(D1-81a)
CH (Me) SCH2(D1-33a) CH2(D1-82a)
CH (Me) SCH2(D1-33a) CH2(D1-84a)
CH (Me) SCH2(D1-33a) CH2(D1-85a)
CH (Me) SCH2(D1-33a) CH2(D1-87a)
CH (Me) SCH2(D1-33a) CH2(D1-92a)
CH (Me) SCH2(D1-33a) CH2(D1-93a)
CH (Me) SCH2(D1-33a) CH2(D1-95a)
CH (Me) SCH2(D1-33a) CH2(D1-96a)
CH (Me) SCH2(D1-33a) CH2(D1-98a)
CH (Me) SCH2(D1-33a) CH2(D1-108a)
CH (Me) SCH2(D1-33a) CH2(D1-108b, Z = 2-Cl)
CH (Me) SCH2(D1-33a) CH2(D1-108b, Z = 3-Me)
CH (Me) SCH2(D1-33a) CH2(D1-108b, Z = 4-OMe)
CH (Me) SCH2(D1-33a) CH2(D1-108b, Z = 2-SMe)
CH (Me) SCH2(D1-33a) CH2(D1-108b, Z = 3-CFThree)
CH (Me) SCH2(D1-33a) CH2(D1-108b, Z = 4-OCFThree)
CH (Me) SCH2(D1-33a) CH2(D1-108b, Z = 2-SCFThree)
CH (Me) SCH2(D1-33a) CH2CH2CN
CH (Me) SCH2(D1-33a) CH2CH2CFThree
CH (Me) SCH2(D1-33a) CH2CH2OMe
CH (Me) SCH2(D1-33a) CH2CH2SMe
CH (Me) SCH2(D1-33a) CH2CH2S (O) Me
CH (Me) SCH2(D1-33a) CH2CH2S (O)2Me
CH (Me) SCH2(D1-33a) D1-32a
CH (Me) SCH2(D1-33a) D1-33a
CH (Me) SCH2(D1-33a) D1-34a
CH (Me) SCH2(D1-33a) D1-37a
CH (Me) SCH2(D1-33a) D1-81a
CH (Me) SCH2(D1-33a) D1-82a
CH (Me) SCH2(D1-33a) D1-84a
CH (Me) SCH2(D1-33a) D1-85a
CH (Me) SCH2(D1-33a) D1-87a
CH (Me) SCH2(D1-33a) D1-92a
CH (Me) SCH2(D1-33a) D1-93a
CH (Me) SCH2(D1-33a) D1-95a
CH (Me) SCH2(D1-33a) D1-96a
CH (Me) SCH2(D1-33a) D1-98a
CH (Me) SCH2(D1-33a) D1-108a
CH (Me) SCH2(D1-33a) D1-108b (Z = 2-Cl)
CH (Me) SCH2(D1-33a) D1-108b (Z = 3-Me)
CH (Me) SCH2(D1-33a) D1-108b (Z = 4-OMe)
CH (Me) SCH2(D1-33a) D1-108b (Z = 2-SMe)
CH (Me) SCH2(D1-33a) D1-108b (Z = 3-CFThree)
CH (Me) SCH2(D1-33a) D1-108b (Z = 4-OCFThree)
CH (Me) SCH2(D1-33a) D1-108b (Z = 2-SCFThree)
CH (Me) SCH2(D1-33a) C (O) Me
CH (Me) SCH2(D1-33a) C (O) CFThree
CH (Me) SCH2(D1-33a) C (O) OMe
CH (Me) S (O) CH2(D1-33a) Me
CH (Me) S (O) CH2(D1-33a) Et
CH (Me) S (O) CH2(D1-33a) Pr-n
CH (Me) S (O) CH2(D1-33a) Pr-i
CH (Me) S (O) CH2(D1-33a) Pr-c
CH (Me) S (O) CH2(D1-33a) Bu-n
CH (Me) S (O) CH2(D1-33a) Bu-i
CH (Me) S (O) CH2(D1-33a) Bu-c
CH (Me) S (O) CH2(D1-33a) Bu-s
CH (Me) S (O) CH2(D1-33a) Bu-t
CH (Me) S (O) CH2(D1-33a) Pen-n
CH (Me) S (O) CH2(D1-33a) Pen-c
CH (Me) S (O) CH2(D1-33a) Hex-n
CH (Me) S (O) CH2(D1-33a) Hex-c
CH (Me) S (O) CH2(D1-33a) CH2Pr-c
CH (Me) S (O) CH2(D1-33a) CH2Bu-c
CH (Me) S (O) CH2(D1-33a) CH2Pen-c
CH (Me) S (O) CH2(D1-33a) CH2Hex-c
CH (Me) S (O) CH2(D1-33a) CH2CH = CH2
CH (Me) S (O) CH2(D1-33a) CH2CH = C (Cl)2
CH (Me) S (O) CH2(D1-33a) CH2C≡CH
CH (Me) S (O) CH2(D1-33a) CH2CN
CH (Me) S (O) CH2(D1-33a) CH2CFThree
CH (Me) S (O) CH2(D1-33a) CH2OMe
CH (Me) S (O) CH2(D1-33a) CH2OCFThree
CH (Me) S (O) CH2(D1-33a) CH2SMe
CH (Me) S (O) CH2(D1-33a) CH2S (O) Me
CH (Me) S (O) CH2(D1-33a) CH2S (O)2Me
CH (Me) S (O) CH2(D1-33a) CH2SCFThree
CH (Me) S (O) CH2(D1-33a) CH2S (O) CFThree
CH (Me) S (O) CH2(D1-33a) CH2S (O)2CFThree
CH (Me) S (O) CH2(D1-33a) CH2CH (OMe)2
CH (Me) S (O) CH2(D1-33a) CH2CH (SMe)2
CH (Me) S (O) CH2(D1-33a) CH2C (O) Me
CH (Me) S (O) CH2(D1-33a) CH2C (O) CFThree
CH (Me) S (O) CH2(D1-33a) CH2C (O) OMe
CH (Me) S (O) CH2(D1-33a) CH2(D1-32a)
CH (Me) S (O) CH2(D1-33a) CH2(D1-33a)
CH (Me) S (O) CH2(D1-33a) CH2(D1-34a)
CH (Me) S (O) CH2(D1-33a) CH2(D1-37a)
CH (Me) S (O) CH2(D1-33a) CH2(D1-81a)
CH (Me) S (O) CH2(D1-33a) CH2(D1-82a)
CH (Me) S (O) CH2(D1-33a) CH2(D1-84a)
CH (Me) S (O) CH2(D1-33a) CH2(D1-85a)
CH (Me) S (O) CH2(D1-33a) CH2(D1-87a)
CH (Me) S (O) CH2(D1-33a) CH2(D1-92a)
CH (Me) S (O) CH2(D1-33a) CH2(D1-93a)
CH (Me) S (O) CH2(D1-33a) CH2(D1-95a)
CH (Me) S (O) CH2(D1-33a) CH2(D1-96a)
CH (Me) S (O) CH2(D1-33a) CH2(D1-98a)
CH (Me) S (O) CH2(D1-33a) CH2(D1-108a)
CH (Me) S (O) CH2(D1-33a) CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O) CH2(D1-33a) CH2(D1-108b, Z = 3-Me)
CH (Me) S (O) CH2(D1-33a) CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O) CH2(D1-33a) CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O) CH2(D1-33a) CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O) CH2(D1-33a) CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O) CH2(D1-33a) CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O) CH2(D1-33a) CH2CH2CN
CH (Me) S (O) CH2(D1-33a) CH2CH2CFThree
CH (Me) S (O) CH2(D1-33a) CH2CH2OMe
CH (Me) S (O) CH2(D1-33a) CH2CH2SMe
CH (Me) S (O) CH2(D1-33a) CH2CH2S (O) Me
CH (Me) S (O) CH2(D1-33a) CH2CH2S (O)2Me
CH (Me) S (O) CH2(D1-33a) D1-32a
CH (Me) S (O) CH2(D1-33a) D1-33a
CH (Me) S (O) CH2(D1-33a) D1-34a
CH (Me) S (O) CH2(D1-33a) D1-37a
CH (Me) S (O) CH2(D1-33a) D1-81a
CH (Me) S (O) CH2(D1-33a) D1-82a
CH (Me) S (O) CH2(D1-33a) D1-84a
CH (Me) S (O) CH2(D1-33a) D1-85a
CH (Me) S (O) CH2(D1-33a) D1-87a
CH (Me) S (O) CH2(D1-33a) D1-92a
CH (Me) S (O) CH2(D1-33a) D1-93a
CH (Me) S (O) CH2(D1-33a) D1-95a
CH (Me) S (O) CH2(D1-33a) D1-96a
CH (Me) S (O) CH2(D1-33a) D1-98a
CH (Me) S (O) CH2(D1-33a) D1-108a
CH (Me) S (O) CH2(D1-33a) D1-108b (Z = 2-Cl)
CH (Me) S (O) CH2(D1-33a) D1-108b (Z = 3-Me)
CH (Me) S (O) CH2(D1-33a) D1-108b (Z = 4-OMe)
CH (Me) S (O) CH2(D1-33a) D1-108b (Z = 2-SMe)
CH (Me) S (O) CH2(D1-33a) D1-108b (Z = 3-CFThree)
CH (Me) S (O) CH2(D1-33a) D1-108b (Z = 4-OCFThree)
CH (Me) S (O) CH2(D1-33a) D1-108b (Z = 2-SCFThree)
CH (Me) S (O) CH2(D1-33a) C (O) Me
CH (Me) S (O) CH2(D1-33a) C (O) CFThree
CH (Me) S (O) CH2(D1-33a) C (O) OMe
CH (Me) S (O)2CH2(D1-33a) Me
CH (Me) S (O)2CH2(D1-33a) Et
CH (Me) S (O)2CH2(D1-33a) Pr-n
CH (Me) S (O)2CH2(D1-33a) Pr-i
CH (Me) S (O)2CH2(D1-33a) Pr-c
CH (Me) S (O)2CH2(D1-33a) Bu-n
CH (Me) S (O)2CH2(D1-33a) Bu-i
CH (Me) S (O)2CH2(D1-33a) Bu-c
CH (Me) S (O)2CH2(D1-33a) Bu-s
CH (Me) S (O)2CH2(D1-33a) Bu-t
CH (Me) S (O)2CH2(D1-33a) Pen-n
CH (Me) S (O)2CH2(D1-33a) Pen-c
CH (Me) S (O)2CH2(D1-33a) Hex-n
CH (Me) S (O)2CH2(D1-33a) Hex-c
CH (Me) S (O)2CH2(D1-33a) CH2Pr-c
CH (Me) S (O)2CH2(D1-33a) CH2Bu-c
CH (Me) S (O)2CH2(D1-33a) CH2Pen-c
CH (Me) S (O)2CH2(D1-33a) CH2Hex-c
CH (Me) S (O)2CH2(D1-33a) CH2CH = CH2
CH (Me) S (O)2CH2(D1-33a) CH2CH = C (Cl)2
CH (Me) S (O)2CH2(D1-33a) CH2C≡CH
CH (Me) S (O)2CH2(D1-33a) CH2CN
CH (Me) S (O)2CH2(D1-33a) CH2CFThree
CH (Me) S (O)2CH2(D1-33a) CH2OMe
CH (Me) S (O)2CH2(D1-33a) CH2OCFThree
CH (Me) S (O)2CH2(D1-33a) CH2SMe
CH (Me) S (O)2CH2(D1-33a) CH2S (O) Me
CH (Me) S (O)2CH2(D1-33a) CH2S (O)2Me
CH (Me) S (O)2CH2(D1-33a) CH2SCFThree
CH (Me) S (O)2CH2(D1-33a) CH2S (O) CFThree
CH (Me) S (O)2CH2(D1-33a) CH2S (O)2CFThree
CH (Me) S (O)2CH2(D1-33a) CH2CH (OMe)2
CH (Me) S (O)2CH2(D1-33a) CH2CH (SMe)2
CH (Me) S (O)2CH2(D1-33a) CH2C (O) Me
CH (Me) S (O)2CH2(D1-33a) CH2C (O) CFThree
CH (Me) S (O)2CH2(D1-33a) CH2C (O) OMe
CH (Me) S (O)2CH2(D1-33a) CH2(D1-32a)
CH (Me) S (O)2CH2(D1-33a) CH2(D1-33a)
CH (Me) S (O)2CH2(D1-33a) CH2(D1-34a)
CH (Me) S (O)2CH2(D1-33a) CH2(D1-37a)
CH (Me) S (O)2CH2(D1-33a) CH2(D1-81a)
CH (Me) S (O)2CH2(D1-33a) CH2(D1-82a)
CH (Me) S (O)2CH2(D1-33a) CH2(D1-84a)
CH (Me) S (O)2CH2(D1-33a) CH2(D1-85a)
CH (Me) S (O)2CH2(D1-33a) CH2(D1-87a)
CH (Me) S (O)2CH2(D1-33a) CH2(D1-92a)
CH (Me) S (O)2CH2(D1-33a) CH2(D1-93a)
CH (Me) S (O)2CH2(D1-33a) CH2(D1-95a)
CH (Me) S (O)2CH2(D1-33a) CH2(D1-96a)
CH (Me) S (O)2CH2(D1-33a) CH2(D1-98a)
CH (Me) S (O)2CH2(D1-33a) CH2(D1-108a)
CH (Me) S (O)2CH2(D1-33a) CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O)2CH2(D1-33a) CH2(D1-108b, Z = 3-Me)
CH (Me) S (O)2CH2(D1-33a) CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O)2CH2(D1-33a) CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O)2CH2(D1-33a) CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O)2CH2(D1-33a) CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O)2CH2(D1-33a) CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O)2CH2(D1-33a) CH2CH2CN
CH (Me) S (O)2CH2(D1-33a) CH2CH2CFThree
CH (Me) S (O)2CH2(D1-33a) CH2CH2OMe
CH (Me) S (O)2CH2(D1-33a) CH2CH2SMe
CH (Me) S (O)2CH2(D1-33a) CH2CH2S (O) Me
CH (Me) S (O)2CH2(D1-33a) CH2CH2S (O)2Me
CH (Me) S (O)2CH2(D1-33a) D1-32a
CH (Me) S (O)2CH2(D1-33a) D1-33a
CH (Me) S (O)2CH2(D1-33a) D1-34a
CH (Me) S (O)2CH2(D1-33a) D1-37a
CH (Me) S (O)2CH2(D1-33a) D1-81a
CH (Me) S (O)2CH2(D1-33a) D1-82a
CH (Me) S (O)2CH2(D1-33a) D1-84a
CH (Me) S (O)2CH2(D1-33a) D1-85a
CH (Me) S (O)2CH2(D1-33a) D1-87a
CH (Me) S (O)2CH2(D1-33a) D1-92a
CH (Me) S (O)2CH2(D1-33a) D1-93a
CH (Me) S (O)2CH2(D1-33a) D1-95a
CH (Me) S (O)2CH2(D1-33a) D1-96a
CH (Me) S (O)2CH2(D1-33a) D1-98a
CH (Me) S (O)2CH2(D1-33a) D1-108a
CH (Me) S (O)2CH2(D1-33a) D1-108b (Z = 2-Cl)
CH (Me) S (O)2CH2(D1-33a) D1-108b (Z = 3-Me)
CH (Me) S (O)2CH2(D1-33a) D1-108b (Z = 4-OMe)
CH (Me) S (O)2CH2(D1-33a) D1-108b (Z = 2-SMe)
CH (Me) S (O)2CH2(D1-33a) D1-108b (Z = 3-CFThree)
CH (Me) S (O)2CH2(D1-33a) D1-108b (Z = 4-OCFThree)
CH (Me) S (O)2CH2(D1-33a) D1-108b (Z = 2-SCFThree)
CH (Me) S (O)2CH2(D1-33a) C (O) Me
CH (Me) S (O)2CH2(D1-33a) C (O) CFThree
CH (Me) S (O)2CH2(D1-33a) C (O) OMe
CH (Et) SCH2(D1-33a) Me
CH (Et) SCH2(D1-33a) Et
CH (Et) SCH2(D1-33a) Pr-n
CH (Et) SCH2(D1-33a) Pr-i
CH (Et) SCH2(D1-33a) Pr-c
CH (Et) SCH2(D1-33a) Bu-n
CH (Et) SCH2(D1-33a) Bu-i
CH (Et) SCH2(D1-33a) Bu-c
CH (Et) SCH2(D1-33a) Bu-s
CH (Et) SCH2(D1-33a) Bu-t
CH (Et) SCH2(D1-33a) Pen-n
CH (Et) SCH2(D1-33a) Pen-c
CH (Et) SCH2(D1-33a) Hex-n
CH (Et) SCH2(D1-33a) Hex-c
CH (Et) SCH2(D1-33a) CH2Pr-c
CH (Et) SCH2(D1-33a) CH2Bu-c
CH (Et) SCH2(D1-33a) CH2Pen-c
CH (Et) SCH2(D1-33a) CH2Hex-c
CH (Et) SCH2(D1-33a) CH2CH = CH2
CH (Et) SCH2(D1-33a) CH2CH = C (Cl)2
CH (Et) SCH2(D1-33a) CH2C≡CH
CH (Et) SCH2(D1-33a) CH2CN
CH (Et) SCH2(D1-33a) CH2CFThree
CH (Et) SCH2(D1-33a) CH2OMe
CH (Et) SCH2(D1-33a) CH2OCFThree
CH (Et) SCH2(D1-33a) CH2SMe
CH (Et) SCH2(D1-33a) CH2S (O) Me
CH (Et) SCH2(D1-33a) CH2S (O)2Me
CH (Et) SCH2(D1-33a) CH2SCFThree
CH (Et) SCH2(D1-33a) CH2S (O) CFThree
CH (Et) SCH2(D1-33a) CH2S (O)2CFThree
CH (Et) SCH2(D1-33a) CH2CH (OMe)2
CH (Et) SCH2(D1-33a) CH2CH (SMe)2
CH (Et) SCH2(D1-33a) CH2C (O) Me
CH (Et) SCH2(D1-33a) CH2C (O) CFThree
CH (Et) SCH2(D1-33a) CH2C (O) OMe
CH (Et) SCH2(D1-33a) CH2(D1-32a)
CH (Et) SCH2(D1-33a) CH2(D1-33a)
CH (Et) SCH2(D1-33a) CH2(D1-34a)
CH (Et) SCH2(D1-33a) CH2(D1-37a)
CH (Et) SCH2(D1-33a) CH2(D1-81a)
CH (Et) SCH2(D1-33a) CH2(D1-82a)
CH (Et) SCH2(D1-33a) CH2(D1-84a)
CH (Et) SCH2(D1-33a) CH2(D1-85a)
CH (Et) SCH2(D1-33a) CH2(D1-87a)
CH (Et) SCH2(D1-33a) CH2(D1-92a)
CH (Et) SCH2(D1-33a) CH2(D1-93a)
CH (Et) SCH2(D1-33a) CH2(D1-95a)
CH (Et) SCH2(D1-33a) CH2(D1-96a)
CH (Et) SCH2(D1-33a) CH2(D1-98a)
CH (Et) SCH2(D1-33a) CH2(D1-108a)
CH (Et) SCH2(D1-33a) CH2(D1-108b, Z = 2-Cl)
CH (Et) SCH2(D1-33a) CH2(D1-108b, Z = 3-Me)
CH (Et) SCH2(D1-33a) CH2(D1-108b, Z = 4-OMe)
CH (Et) SCH2(D1-33a) CH2(D1-108b, Z = 2-SMe)
CH (Et) SCH2(D1-33a) CH2(D1-108b, Z = 3-CFThree)
CH (Et) SCH2(D1-33a) CH2(D1-108b, Z = 4-OCFThree)
CH (Et) SCH2(D1-33a) CH2(D1-108b, Z = 2-SCFThree)
CH (Et) SCH2(D1-33a) CH2CH2CN
CH (Et) SCH2(D1-33a) CH2CH2CFThree
CH (Et) SCH2(D1-33a) CH2CH2OMe
CH (Et) SCH2(D1-33a) CH2CH2SMe
CH (Et) SCH2(D1-33a) CH2CH2S (O) Me
CH (Et) SCH2(D1-33a) CH2CH2S (O)2Me
CH (Et) SCH2(D1-33a) D1-32a
CH (Et) SCH2(D1-33a) D1-33a
CH (Et) SCH2(D1-33a) D1-34a
CH (Et) SCH2(D1-33a) D1-37a
CH (Et) SCH2(D1-33a) D1-81a
CH (Et) SCH2(D1-33a) D1-82a
CH (Et) SCH2(D1-33a) D1-84a
CH (Et) SCH2(D1-33a) D1-85a
CH (Et) SCH2(D1-33a) D1-87a
CH (Et) SCH2(D1-33a) D1-92a
CH (Et) SCH2(D1-33a) D1-93a
CH (Et) SCH2(D1-33a) D1-95a
CH (Et) SCH2(D1-33a) D1-96a
CH (Et) SCH2(D1-33a) D1-98a
CH (Et) SCH2(D1-33a) D1-108a
CH (Et) SCH2(D1-33a) D1-108b (Z = 2-Cl)
CH (Et) SCH2(D1-33a) D1-108b (Z = 3-Me)
CH (Et) SCH2(D1-33a) D1-108b (Z = 4-OMe)
CH (Et) SCH2(D1-33a) D1-108b (Z = 2-SMe)
CH (Et) SCH2(D1-33a) D1-108b (Z = 3-CFThree)
CH (Et) SCH2(D1-33a) D1-108b (Z = 4-OCFThree)
CH (Et) SCH2(D1-33a) D1-108b (Z = 2-SCFThree)
CH (Et) SCH2(D1-33a) C (O) Me
CH (Et) SCH2(D1-33a) C (O) CFThree
CH (Et) SCH2(D1-33a) C (O) OMe
CH (Et) S (O) CH2(D1-33a) Me
CH (Et) S (O) CH2(D1-33a) Et
CH (Et) S (O) CH2(D1-33a) Pr-n
CH (Et) S (O) CH2(D1-33a) Pr-i
CH (Et) S (O) CH2(D1-33a) Pr-c
CH (Et) S (O) CH2(D1-33a) Bu-n
CH (Et) S (O) CH2(D1-33a) Bu-i
CH (Et) S (O) CH2(D1-33a) Bu-c
CH (Et) S (O) CH2(D1-33a) Bu-s
CH (Et) S (O) CH2(D1-33a) Bu-t
CH (Et) S (O) CH2(D1-33a) Pen-n
CH (Et) S (O) CH2(D1-33a) Pen-c
CH (Et) S (O) CH2(D1-33a) Hex-n
CH (Et) S (O) CH2(D1-33a) Hex-c
CH (Et) S (O) CH2(D1-33a) CH2Pr-c
CH (Et) S (O) CH2(D1-33a) CH2Bu-c
CH (Et) S (O) CH2(D1-33a) CH2Pen-c
CH (Et) S (O) CH2(D1-33a) CH2Hex-c
CH (Et) S (O) CH2(D1-33a) CH2CH = CH2
CH (Et) S (O) CH2(D1-33a) CH2CH = C (Cl)2
CH (Et) S (O) CH2(D1-33a) CH2C≡CH
CH (Et) S (O) CH2(D1-33a) CH2CN
CH (Et) S (O) CH2(D1-33a) CH2CFThree
CH (Et) S (O) CH2(D1-33a) CH2OMe
CH (Et) S (O) CH2(D1-33a) CH2OCFThree
CH (Et) S (O) CH2(D1-33a) CH2SMe
CH (Et) S (O) CH2(D1-33a) CH2S (O) Me
CH (Et) S (O) CH2(D1-33a) CH2S (O)2Me
CH (Et) S (O) CH2(D1-33a) CH2SCFThree
CH (Et) S (O) CH2(D1-33a) CH2S (O) CFThree
CH (Et) S (O) CH2(D1-33a) CH2S (O)2CFThree
CH (Et) S (O) CH2(D1-33a) CH2CH (OMe)2
CH (Et) S (O) CH2(D1-33a) CH2CH (SMe)2
CH (Et) S (O) CH2(D1-33a) CH2C (O) Me
CH (Et) S (O) CH2(D1-33a) CH2C (O) CFThree
CH (Et) S (O) CH2(D1-33a) CH2C (O) OMe
CH (Et) S (O) CH2(D1-33a) CH2(D1-32a)
CH (Et) S (O) CH2(D1-33a) CH2(D1-33a)
CH (Et) S (O) CH2(D1-33a) CH2(D1-34a)
CH (Et) S (O) CH2(D1-33a) CH2(D1-37a)
CH (Et) S (O) CH2(D1-33a) CH2(D1-81a)
CH (Et) S (O) CH2(D1-33a) CH2(D1-82a)
CH (Et) S (O) CH2(D1-33a) CH2(D1-84a)
CH (Et) S (O) CH2(D1-33a) CH2(D1-85a)
CH (Et) S (O) CH2(D1-33a) CH2(D1-87a)
CH (Et) S (O) CH2(D1-33a) CH2(D1-92a)
CH (Et) S (O) CH2(D1-33a) CH2(D1-93a)
CH (Et) S (O) CH2(D1-33a) CH2(D1-95a)
CH (Et) S (O) CH2(D1-33a) CH2(D1-96a)
CH (Et) S (O) CH2(D1-33a) CH2(D1-98a)
CH (Et) S (O) CH2(D1-33a) CH2(D1-108a)
CH (Et) S (O) CH2(D1-33a) CH2(D1-108b, Z = 2-Cl)
CH (Et) S (O) CH2(D1-33a) CH2(D1-108b, Z = 3-Me)
CH (Et) S (O) CH2(D1-33a) CH2(D1-108b, Z = 4-OMe)
CH (Et) S (O) CH2(D1-33a) CH2(D1-108b, Z = 2-SMe)
CH (Et) S (O) CH2(D1-33a) CH2(D1-108b, Z = 3-CFThree)
CH (Et) S (O) CH2(D1-33a) CH2(D1-108b, Z = 4-OCFThree)
CH (Et) S (O) CH2(D1-33a) CH2(D1-108b, Z = 2-SCFThree)
CH (Et) S (O) CH2(D1-33a) CH2CH2CN
CH (Et) S (O) CH2(D1-33a) CH2CH2CFThree
CH (Et) S (O) CH2(D1-33a) CH2CH2OMe
CH (Et) S (O) CH2(D1-33a) CH2CH2SMe
CH (Et) S (O) CH2(D1-33a) CH2CH2S (O) Me
CH (Et) S (O) CH2(D1-33a) CH2CH2S (O)2Me
CH (Et) S (O) CH2(D1-33a) D1-32a
CH (Et) S (O) CH2(D1-33a) D1-33a
CH (Et) S (O) CH2(D1-33a) D1-34a
CH (Et) S (O) CH2(D1-33a) D1-37a
CH (Et) S (O) CH2(D1-33a) D1-81a
CH (Et) S (O) CH2(D1-33a) D1-82a
CH (Et) S (O) CH2(D1-33a) D1-84a
CH (Et) S (O) CH2(D1-33a) D1-85a
CH (Et) S (O) CH2(D1-33a) D1-87a
CH (Et) S (O) CH2(D1-33a) D1-92a
CH (Et) S (O) CH2(D1-33a) D1-93a
CH (Et) S (O) CH2(D1-33a) D1-95a
CH (Et) S (O) CH2(D1-33a) D1-96a
CH (Et) S (O) CH2(D1-33a) D1-98a
CH (Et) S (O) CH2(D1-33a) D1-108a
CH (Et) S (O) CH2(D1-33a) D1-108b (Z = 2-Cl)
CH (Et) S (O) CH2(D1-33a) D1-108b (Z = 3-Me)
CH (Et) S (O) CH2(D1-33a) D1-108b (Z = 4-OMe)
CH (Et) S (O) CH2(D1-33a) D1-108b (Z = 2-SMe)
CH (Et) S (O) CH2(D1-33a) D1-108b (Z = 3-CFThree)
CH (Et) S (O) CH2(D1-33a) D1-108b (Z = 4-OCFThree)
CH (Et) S (O) CH2(D1-33a) D1-108b (Z = 2-SCFThree)
CH (Et) S (O) CH2(D1-33a) C (O) Me
CH (Et) S (O) CH2(D1-33a) C (O) CFThree
CH (Et) S (O) CH2(D1-33a) C (O) OMe
CH (Et) S (O)2CH2(D1-33a) Me
CH (Et) S (O)2CH2(D1-33a) Et
CH (Et) S (O)2CH2(D1-33a) Pr-n
CH (Et) S (O)2CH2(D1-33a) Pr-i
CH (Et) S (O)2CH2(D1-33a) Pr-c
CH (Et) S (O)2CH2(D1-33a) Bu-n
CH (Et) S (O)2CH2(D1-33a) Bu-i
CH (Et) S (O)2CH2(D1-33a) Bu-c
CH (Et) S (O)2CH2(D1-33a) Bu-s
CH (Et) S (O)2CH2(D1-33a) Bu-t
CH (Et) S (O)2CH2(D1-33a) Pen-n
CH (Et) S (O)2CH2(D1-33a) Pen-c
CH (Et) S (O)2CH2(D1-33a) Hex-n
CH (Et) S (O)2CH2(D1-33a) Hex-c
CH (Et) S (O)2CH2(D1-33a) CH2Pr-c
CH (Et) S (O)2CH2(D1-33a) CH2Bu-c
CH (Et) S (O)2CH2(D1-33a) CH2Pen-c
CH (Et) S (O)2CH2(D1-33a) CH2Hex-c
CH (Et) S (O)2CH2(D1-33a) CH2CH = CH2
CH (Et) S (O)2CH2(D1-33a) CH2CH = C (Cl)2
CH (Et) S (O)2CH2(D1-33a) CH2C≡CH
CH (Et) S (O)2CH2(D1-33a) CH2CN
CH (Et) S (O)2CH2(D1-33a) CH2CFThree
CH (Et) S (O)2CH2(D1-33a) CH2OMe
CH (Et) S (O)2CH2(D1-33a) CH2OCFThree
CH (Et) S (O)2CH2(D1-33a) CH2SMe
CH (Et) S (O)2CH2(D1-33a) CH2S (O) Me
CH (Et) S (O)2CH2(D1-33a) CH2S (O)2Me
CH (Et) S (O)2CH2(D1-33a) CH2SCFThree
CH (Et) S (O)2CH2(D1-33a) CH2S (O) CFThree
CH (Et) S (O)2CH2(D1-33a) CH2S (O)2CFThree
CH (Et) S (O)2CH2(D1-33a) CH2CH (OMe)2
CH (Et) S (O)2CH2(D1-33a) CH2CH (SMe)2
CH (Et) S (O)2CH2(D1-33a) CH2C (O) Me
CH (Et) S (O)2CH2(D1-33a) CH2C (O) CFThree
CH (Et) S (O)2CH2(D1-33a) CH2C (O) OMe
CH (Et) S (O)2CH2(D1-33a) CH2(D1-32a)
CH (Et) S (O)2CH2(D1-33a) CH2(D1-33a)
CH (Et) S (O)2CH2(D1-33a) CH2(D1-34a)
CH (Et) S (O)2CH2(D1-33a) CH2(D1-37a)
CH (Et) S (O)2CH2(D1-33a) CH2(D1-81a)
CH (Et) S (O)2CH2(D1-33a) CH2(D1-82a)
CH (Et) S (O)2CH2(D1-33a) CH2(D1-84a)
CH (Et) S (O)2CH2(D1-33a) CH2(D1-85a)
CH (Et) S (O)2CH2(D1-33a) CH2(D1-87a)
CH (Et) S (O)2CH2(D1-33a) CH2(D1-92a)
CH (Et) S (O)2CH2(D1-33a) CH2(D1-93a)
CH (Et) S (O)2CH2(D1-33a) CH2(D1-95a)
CH (Et) S (O)2CH2(D1-33a) CH2(D1-96a)
CH (Et) S (O)2CH2(D1-33a) CH2(D1-98a)
CH (Et) S (O)2CH2(D1-33a) CH2(D1-108a)
CH (Et) S (O)2CH2(D1-33a) CH2(D1-108b, Z = 2-Cl)
CH (Et) S (O)2CH2(D1-33a) CH2(D1-108b, Z = 3-Me)
CH (Et) S (O)2CH2(D1-33a) CH2(D1-108b, Z = 4-OMe)
CH (Et) S (O)2CH2(D1-33a) CH2(D1-108b, Z = 2-SMe)
CH (Et) S (O)2CH2(D1-33a) CH2(D1-108b, Z = 3-CFThree)
CH (Et) S (O)2CH2(D1-33a) CH2(D1-108b, Z = 4-OCFThree)
CH (Et) S (O)2CH2(D1-33a) CH2(D1-108b, Z = 2-SCFThree)
CH (Et) S (O)2CH2(D1-33a) CH2CH2CN
CH (Et) S (O)2CH2(D1-33a) CH2CH2CFThree
CH (Et) S (O)2CH2(D1-33a) CH2CH2OMe
CH (Et) S (O)2CH2(D1-33a) CH2CH2SMe
CH (Et) S (O)2CH2(D1-33a) CH2CH2S (O) Me
CH (Et) S (O)2CH2(D1-33a) CH2CH2S (O)2Me
CH (Et) S (O)2CH2(D1-33a) D1-32a
CH (Et) S (O)2CH2(D1-33a) D1-33a
CH (Et) S (O)2CH2(D1-33a) D1-34a
CH (Et) S (O)2CH2(D1-33a) D1-37a
CH (Et) S (O)2CH2(D1-33a) D1-81a
CH (Et) S (O)2CH2(D1-33a) D1-82a
CH (Et) S (O)2CH2(D1-33a) D1-84a
CH (Et) S (O)2CH2(D1-33a) D1-85a
CH (Et) S (O)2CH2(D1-33a) D1-87a
CH (Et) S (O)2CH2(D1-33a) D1-92a
CH (Et) S (O)2CH2(D1-33a) D1-93a
CH (Et) S (O)2CH2(D1-33a) D1-95a
CH (Et) S (O)2CH2(D1-33a) D1-96a
CH (Et) S (O)2CH2(D1-33a) D1-98a
CH (Et) S (O)2CH2(D1-33a) D1-108a
CH (Et) S (O)2CH2(D1-33a) D1-108b (Z = 2-Cl)
CH (Et) S (O)2CH2(D1-33a) D1-108b (Z = 3-Me)
CH (Et) S (O)2CH2(D1-33a) D1-108b (Z = 4-OMe)
CH (Et) S (O)2CH2(D1-33a) D1-108b (Z = 2-SMe)
CH (Et) S (O)2CH2(D1-33a) D1-108b (Z = 3-CFThree)
CH (Et) S (O)2CH2(D1-33a) D1-108b (Z = 4-OCFThree)
CH (Et) S (O)2CH2(D1-33a) D1-108b (Z = 2-SCFThree)
CH (Et) S (O)2CH2(D1-33a) C (O) Me
CH (Et) S (O)2CH2(D1-33a) C (O) CFThree
CH (Et) S (O)2CH2(D1-33a) C (O) OMe
CH2SCH2(D1-34a) Me
CH2SCH2(D1-34a) Et
CH2SCH2(D1-34a) Pr-n
CH2SCH2(D1-34a) Pr-i
CH2SCH2(D1-34a) Pr-c
CH2SCH2(D1-34a) Bu-n
CH2SCH2(D1-34a) Bu-i
CH2SCH2(D1-34a) Bu-c
CH2SCH2(D1-34a) Bu-s
CH2SCH2(D1-34a) Bu-t
CH2SCH2(D1-34a) Pen-n
CH2SCH2(D1-34a) Pen-c
CH2SCH2(D1-34a) Hex-n
CH2SCH2(D1-34a) Hex-c
CH2SCH2(D1-34a) CH2Pr-c
CH2SCH2(D1-34a) CH2Bu-c
CH2SCH2(D1-34a) CH2Pen-c
CH2SCH2(D1-34a) CH2Hex-c
CH2SCH2(D1-34a) CH2CH = CH2
CH2SCH2(D1-34a) CH2CH = C (Cl)2
CH2SCH2(D1-34a) CH2C≡CH
CH2SCH2(D1-34a) CH2CN
CH2SCH2(D1-34a) CH2CFThree
CH2SCH2(D1-34a) CH2OMe
CH2SCH2(D1-34a) CH2OCFThree
CH2SCH2(D1-34a) CH2SMe
CH2SCH2(D1-34a) CH2S (O) Me
CH2SCH2(D1-34a) CH2S (O)2Me
CH2SCH2(D1-34a) CH2SCFThree
CH2SCH2(D1-34a) CH2S (O) CFThree
CH2SCH2(D1-34a) CH2S (O)2CFThree
CH2SCH2(D1-34a) CH2CH (OMe)2
CH2SCH2(D1-34a) CH2CH (SMe)2
CH2SCH2(D1-34a) CH2C (O) Me
CH2SCH2(D1-34a) CH2C (O) CFThree
CH2SCH2(D1-34a) CH2C (O) OMe
CH2SCH2(D1-34a) CH2(D1-32a)
CH2SCH2(D1-34a) CH2(D1-33a)
CH2SCH2(D1-34a) CH2(D1-34a)
CH2SCH2(D1-34a) CH2(D1-37a)
CH2SCH2(D1-34a) CH2(D1-81a)
CH2SCH2(D1-34a) CH2(D1-82a)
CH2SCH2(D1-34a) CH2(D1-84a)
CH2SCH2(D1-34a) CH2(D1-85a)
CH2SCH2(D1-34a) CH2(D1-87a)
CH2SCH2(D1-34a) CH2(D1-92a)
CH2SCH2(D1-34a) CH2(D1-93a)
CH2SCH2(D1-34a) CH2(D1-95a)
CH2SCH2(D1-34a) CH2(D1-96a)
CH2SCH2(D1-34a) CH2(D1-98a)
CH2SCH2(D1-34a) CH2(D1-108a)
CH2SCH2(D1-34a) CH2(D1-108b, Z = 2-Cl)
CH2SCH2(D1-34a) CH2(D1-108b, Z = 3-Me)
CH2SCH2(D1-34a) CH2(D1-108b, Z = 4-OMe)
CH2SCH2(D1-34a) CH2(D1-108b, Z = 2-SMe)
CH2SCH2(D1-34a) CH2(D1-108b, Z = 3-CFThree)
CH2SCH2(D1-34a) CH2(D1-108b, Z = 4-OCFThree)
CH2SCH2(D1-34a) CH2(D1-108b, Z = 2-SCFThree)
CH2SCH2(D1-34a) CH2CH2CN
CH2SCH2(D1-34a) CH2CH2CFThree
CH2SCH2(D1-34a) CH2CH2OMe
CH2SCH2(D1-34a) CH2CH2SMe
CH2SCH2(D1-34a) CH2CH2S (O) Me
CH2SCH2(D1-34a) CH2CH2S (O)2Me
CH2SCH2(D1-34a) D1-32a
CH2SCH2(D1-34a) D1-33a
CH2SCH2(D1-34a) D1-34a
CH2SCH2(D1-34a) D1-37a
CH2SCH2(D1-34a) D1-81a
CH2SCH2(D1-34a) D1-82a
CH2SCH2(D1-34a) D1-84a
CH2SCH2(D1-34a) D1-85a
CH2SCH2(D1-34a) D1-87a
CH2SCH2(D1-34a) D1-92a
CH2SCH2(D1-34a) D1-93a
CH2SCH2(D1-34a) D1-95a
CH2SCH2(D1-34a) D1-96a
CH2SCH2(D1-34a) D1-98a
CH2SCH2(D1-34a) D1-108a
CH2SCH2(D1-34a) D1-108b (Z = 2-Cl)
CH2SCH2(D1-34a) D1-108b (Z = 3-Me)
CH2SCH2(D1-34a) D1-108b (Z = 4-OMe)
CH2SCH2(D1-34a) D1-108b (Z = 2-SMe)
CH2SCH2(D1-34a) D1-108b (Z = 3-CFThree)
CH2SCH2(D1-34a) D1-108b (Z = 4-OCFThree)
CH2SCH2(D1-34a) D1-108b (Z = 2-SCFThree)
CH2SCH2(D1-34a) C (O) Me
CH2SCH2(D1-34a) C (O) CFThree
CH2SCH2(D1-34a) C (O) OMe
CH2S (O) CH2(D1-34a) Me
CH2S (O) CH2(D1-34a) Et
CH2S (O) CH2(D1-34a) Pr-n
CH2S (O) CH2(D1-34a) Pr-i
CH2S (O) CH2(D1-34a) Pr-c
CH2S (O) CH2(D1-34a) Bu-n
CH2S (O) CH2(D1-34a) Bu-i
CH2S (O) CH2(D1-34a) Bu-c
CH2S (O) CH2(D1-34a) Bu-s
CH2S (O) CH2(D1-34a) Bu-t
CH2S (O) CH2(D1-34a) Pen-n
CH2S (O) CH2(D1-34a) Pen-c
CH2S (O) CH2(D1-34a) Hex-n
CH2S (O) CH2(D1-34a) Hex-c
CH2S (O) CH2(D1-34a) CH2Pr-c
CH2S (O) CH2(D1-34a) CH2Bu-c
CH2S (O) CH2(D1-34a) CH2Pen-c
CH2S (O) CH2(D1-34a) CH2Hex-c
CH2S (O) CH2(D1-34a) CH2CH = CH2
CH2S (O) CH2(D1-34a) CH2CH = C (Cl)2
CH2S (O) CH2(D1-34a) CH2C≡CH
CH2S (O) CH2(D1-34a) CH2CN
CH2S (O) CH2(D1-34a) CH2CFThree
CH2S (O) CH2(D1-34a) CH2OMe
CH2S (O) CH2(D1-34a) CH2OCFThree
CH2S (O) CH2(D1-34a) CH2SMe
CH2S (O) CH2(D1-34a) CH2S (O) Me
CH2S (O) CH2(D1-34a) CH2S (O)2Me
CH2S (O) CH2(D1-34a) CH2SCFThree
CH2S (O) CH2(D1-34a) CH2S (O) CFThree
CH2S (O) CH2(D1-34a) CH2S (O)2CFThree
CH2S (O) CH2(D1-34a) CH2CH (OMe)2
CH2S (O) CH2(D1-34a) CH2CH (SMe)2
CH2S (O) CH2(D1-34a) CH2C (O) Me
CH2S (O) CH2(D1-34a) CH2C (O) CFThree
CH2S (O) CH2(D1-34a) CH2C (O) OMe
CH2S (O) CH2(D1-34a) CH2(D1-32a)
CH2S (O) CH2(D1-34a) CH2(D1-33a)
CH2S (O) CH2(D1-34a) CH2(D1-34a)
CH2S (O) CH2(D1-34a) CH2(D1-37a)
CH2S (O) CH2(D1-34a) CH2(D1-81a)
CH2S (O) CH2(D1-34a) CH2(D1-82a)
CH2S (O) CH2(D1-34a) CH2(D1-84a)
CH2S (O) CH2(D1-34a) CH2(D1-85a)
CH2S (O) CH2(D1-34a) CH2(D1-87a)
CH2S (O) CH2(D1-34a) CH2(D1-92a)
CH2S (O) CH2(D1-34a) CH2(D1-93a)
CH2S (O) CH2(D1-34a) CH2(D1-95a)
CH2S (O) CH2(D1-34a) CH2(D1-96a)
CH2S (O) CH2(D1-34a) CH2(D1-98a)
CH2S (O) CH2(D1-34a) CH2(D1-108a)
CH2S (O) CH2(D1-34a) CH2(D1-108b, Z = 2-Cl)
CH2S (O) CH2(D1-34a) CH2(D1-108b, Z = 3-Me)
CH2S (O) CH2(D1-34a) CH2(D1-108b, Z = 4-OMe)
CH2S (O) CH2(D1-34a) CH2(D1-108b, Z = 2-SMe)
CH2S (O) CH2(D1-34a) CH2(D1-108b, Z = 3-CFThree)
CH2S (O) CH2(D1-34a) CH2(D1-108b, Z = 4-OCFThree)
CH2S (O) CH2(D1-34a) CH2(D1-108b, Z = 2-SCFThree)
CH2S (O) CH2(D1-34a) CH2CH2CN
CH2S (O) CH2(D1-34a) CH2CH2CFThree
CH2S (O) CH2(D1-34a) CH2CH2OMe
CH2S (O) CH2(D1-34a) CH2CH2SMe
CH2S (O) CH2(D1-34a) CH2CH2S (O) Me
CH2S (O) CH2(D1-34a) CH2CH2S (O)2Me
CH2S (O) CH2(D1-34a) D1-32a
CH2S (O) CH2(D1-34a) D1-33a
CH2S (O) CH2(D1-34a) D1-34a
CH2S (O) CH2(D1-34a) D1-37a
CH2S (O) CH2(D1-34a) D1-81a
CH2S (O) CH2(D1-34a) D1-82a
CH2S (O) CH2(D1-34a) D1-84a
CH2S (O) CH2(D1-34a) D1-85a
CH2S (O) CH2(D1-34a) D1-87a
CH2S (O) CH2(D1-34a) D1-92a
CH2S (O) CH2(D1-34a) D1-93a
CH2S (O) CH2(D1-34a) D1-95a
CH2S (O) CH2(D1-34a) D1-96a
CH2S (O) CH2(D1-34a) D1-98a
CH2S (O) CH2(D1-34a) D1-108a
CH2S (O) CH2(D1-34a) D1-108b (Z = 2-Cl)
CH2S (O) CH2(D1-34a) D1-108b (Z = 3-Me)
CH2S (O) CH2(D1-34a) D1-108b (Z = 4-OMe)
CH2S (O) CH2(D1-34a) D1-108b (Z = 2-SMe)
CH2S (O) CH2(D1-34a) D1-108b (Z = 3-CFThree)
CH2S (O) CH2(D1-34a) D1-108b (Z = 4-OCFThree)
CH2S (O) CH2(D1-34a) D1-108b (Z = 2-SCFThree)
CH2S (O) CH2(D1-34a) C (O) Me
CH2S (O) CH2(D1-34a) C (O) CFThree
CH2S (O) CH2(D1-34a) C (O) OMe
CH2S (O)2CH2(D1-34a) Me
CH2S (O)2CH2(D1-34a) Et
CH2S (O)2CH2(D1-34a) Pr-n
CH2S (O)2CH2(D1-34a) Pr-i
CH2S (O)2CH2(D1-34a) Pr-c
CH2S (O)2CH2(D1-34a) Bu-n
CH2S (O)2CH2(D1-34a) Bu-i
CH2S (O)2CH2(D1-34a) Bu-c
CH2S (O)2CH2(D1-34a) Bu-s
CH2S (O)2CH2(D1-34a) Bu-t
CH2S (O)2CH2(D1-34a) Pen-n
CH2S (O)2CH2(D1-34a) Pen-c
CH2S (O)2CH2(D1-34a) Hex-n
CH2S (O)2CH2(D1-34a) Hex-c
CH2S (O)2CH2(D1-34a) CH2Pr-c
CH2S (O)2CH2(D1-34a) CH2Bu-c
CH2S (O)2CH2(D1-34a) CH2Pen-c
CH2S (O)2CH2(D1-34a) CH2Hex-c
CH2S (O)2CH2(D1-34a) CH2CH = CH2
CH2S (O)2CH2(D1-34a) CH2CH = C (Cl)2
CH2S (O)2CH2(D1-34a) CH2C≡CH
CH2S (O)2CH2(D1-34a) CH2CN
CH2S (O)2CH2(D1-34a) CH2CFThree
CH2S (O)2CH2(D1-34a) CH2OMe
CH2S (O)2CH2(D1-34a) CH2OCFThree
CH2S (O)2CH2(D1-34a) CH2SMe
CH2S (O)2CH2(D1-34a) CH2S (O) Me
CH2S (O)2CH2(D1-34a) CH2S (O)2Me
CH2S (O)2CH2(D1-34a) CH2SCFThree
CH2S (O)2CH2(D1-34a) CH2S (O) CFThree
CH2S (O)2CH2(D1-34a) CH2S (O)2CFThree
CH2S (O)2CH2(D1-34a) CH2CH (OMe)2
CH2S (O)2CH2(D1-34a) CH2CH (SMe)2
CH2S (O)2CH2(D1-34a) CH2C (O) Me
CH2S (O)2CH2(D1-34a) CH2C (O) CFThree
CH2S (O)2CH2(D1-34a) CH2C (O) OMe
CH2S (O)2CH2(D1-34a) CH2(D1-32a)
CH2S (O)2CH2(D1-34a) CH2(D1-33a)
CH2S (O)2CH2(D1-34a) CH2(D1-34a)
CH2S (O)2CH2(D1-34a) CH2(D1-37a)
CH2S (O)2CH2(D1-34a) CH2(D1-81a)
CH2S (O)2CH2(D1-34a) CH2(D1-82a)
CH2S (O)2CH2(D1-34a) CH2(D1-84a)
CH2S (O)2CH2(D1-34a) CH2(D1-85a)
CH2S (O)2CH2(D1-34a) CH2(D1-87a)
CH2S (O)2CH2(D1-34a) CH2(D1-92a)
CH2S (O)2CH2(D1-34a) CH2(D1-93a)
CH2S (O)2CH2(D1-34a) CH2(D1-95a)
CH2S (O)2CH2(D1-34a) CH2(D1-96a)
CH2S (O)2CH2(D1-34a) CH2(D1-98a)
CH2S (O)2CH2(D1-34a) CH2(D1-108a)
CH2S (O)2CH2(D1-34a) CH2(D1-108b, Z = 2-Cl)
CH2S (O)2CH2(D1-34a) CH2(D1-108b, Z = 3-Me)
CH2S (O)2CH2(D1-34a) CH2(D1-108b, Z = 4-OMe)
CH2S (O)2CH2(D1-34a) CH2(D1-108b, Z = 2-SMe)
CH2S (O)2CH2(D1-34a) CH2(D1-108b, Z = 3-CFThree)
CH2S (O)2CH2(D1-34a) CH2(D1-108b, Z = 4-OCFThree)
CH2S (O)2CH2(D1-34a) CH2(D1-108b, Z = 2-SCFThree)
CH2S (O)2CH2(D1-34a) CH2CH2CN
CH2S (O)2CH2(D1-34a) CH2CH2CFThree
CH2S (O)2CH2(D1-34a) CH2CH2OMe
CH2S (O)2CH2(D1-34a) CH2CH2SMe
CH2S (O)2CH2(D1-34a) CH2CH2S (O) Me
CH2S (O)2CH2(D1-34a) CH2CH2S (O)2Me
CH2S (O)2CH2(D1-34a) D1-32a
CH2S (O)2CH2(D1-34a) D1-33a
CH2S (O)2CH2(D1-34a) D1-34a
CH2S (O)2CH2(D1-34a) D1-37a
CH2S (O)2CH2(D1-34a) D1-81a
CH2S (O)2CH2(D1-34a) D1-82a
CH2S (O)2CH2(D1-34a) D1-84a
CH2S (O)2CH2(D1-34a) D1-85a
CH2S (O)2CH2(D1-34a) D1-87a
CH2S (O)2CH2(D1-34a) D1-92a
CH2S (O)2CH2(D1-34a) D1-93a
CH2S (O)2CH2(D1-34a) D1-95a
CH2S (O)2CH2(D1-34a) D1-96a
CH2S (O)2CH2(D1-34a) D1-98a
CH2S (O)2CH2(D1-34a) D1-108a
CH2S (O)2CH2(D1-34a) D1-108b (Z = 2-Cl)
CH2S (O)2CH2(D1-34a) D1-108b (Z = 3-Me)
CH2S (O)2CH2(D1-34a) D1-108b (Z = 4-OMe)
CH2S (O)2CH2(D1-34a) D1-108b (Z = 2-SMe)
CH2S (O)2CH2(D1-34a) D1-108b (Z = 3-CFThree)
CH2S (O)2CH2(D1-34a) D1-108b (Z = 4-OCFThree)
CH2S (O)2CH2(D1-34a) D1-108b (Z = 2-SCFThree)
CH2S (O)2CH2(D1-34a) C (O) Me
CH2S (O)2CH2(D1-34a) C (O) CFThree
CH2S (O)2CH2(D1-34a) C (O) OMe
CH (Me) SCH2(D1-34a) Me
CH (Me) SCH2(D1-34a) Et
CH (Me) SCH2(D1-34a) Pr-n
CH (Me) SCH2(D1-34a) Pr-i
CH (Me) SCH2(D1-34a) Pr-c
CH (Me) SCH2(D1-34a) Bu-n
CH (Me) SCH2(D1-34a) Bu-i
CH (Me) SCH2(D1-34a) Bu-c
CH (Me) SCH2(D1-34a) Bu-s
CH (Me) SCH2(D1-34a) Bu-t
CH (Me) SCH2(D1-34a) Pen-n
CH (Me) SCH2(D1-34a) Pen-c
CH (Me) SCH2(D1-34a) Hex-n
CH (Me) SCH2(D1-34a) Hex-c
CH (Me) SCH2(D1-34a) CH2Pr-c
CH (Me) SCH2(D1-34a) CH2Bu-c
CH (Me) SCH2(D1-34a) CH2Pen-c
CH (Me) SCH2(D1-34a) CH2Hex-c
CH (Me) SCH2(D1-34a) CH2CH = CH2
CH (Me) SCH2(D1-34a) CH2CH = C (Cl)2
CH (Me) SCH2(D1-34a) CH2C≡CH
CH (Me) SCH2(D1-34a) CH2CN
CH (Me) SCH2(D1-34a) CH2CFThree
CH (Me) SCH2(D1-34a) CH2OMe
CH (Me) SCH2(D1-34a) CH2OCFThree
CH (Me) SCH2(D1-34a) CH2SMe
CH (Me) SCH2(D1-34a) CH2S (O) Me
CH (Me) SCH2(D1-34a) CH2S (O)2Me
CH (Me) SCH2(D1-34a) CH2SCFThree
CH (Me) SCH2(D1-34a) CH2S (O) CFThree
CH (Me) SCH2(D1-34a) CH2S (O)2CFThree
CH (Me) SCH2(D1-34a) CH2CH (OMe)2
CH (Me) SCH2(D1-34a) CH2CH (SMe)2
CH (Me) SCH2(D1-34a) CH2C (O) Me
CH (Me) SCH2(D1-34a) CH2C (O) CFThree
CH (Me) SCH2(D1-34a) CH2C (O) OMe
CH (Me) SCH2(D1-34a) CH2(D1-32a)
CH (Me) SCH2(D1-34a) CH2(D1-33a)
CH (Me) SCH2(D1-34a) CH2(D1-34a)
CH (Me) SCH2(D1-34a) CH2(D1-37a)
CH (Me) SCH2(D1-34a) CH2(D1-81a)
CH (Me) SCH2(D1-34a) CH2(D1-82a)
CH (Me) SCH2(D1-34a) CH2(D1-84a)
CH (Me) SCH2(D1-34a) CH2(D1-85a)
CH (Me) SCH2(D1-34a) CH2(D1-87a)
CH (Me) SCH2(D1-34a) CH2(D1-92a)
CH (Me) SCH2(D1-34a) CH2(D1-93a)
CH (Me) SCH2(D1-34a) CH2(D1-95a)
CH (Me) SCH2(D1-34a) CH2(D1-96a)
CH (Me) SCH2(D1-34a) CH2(D1-98a)
CH (Me) SCH2(D1-34a) CH2(D1-108a)
CH (Me) SCH2(D1-34a) CH2(D1-108b, Z = 2-Cl)
CH (Me) SCH2(D1-34a) CH2(D1-108b, Z = 3-Me)
CH (Me) SCH2(D1-34a) CH2(D1-108b, Z = 4-OMe)
CH (Me) SCH2(D1-34a) CH2(D1-108b, Z = 2-SMe)
CH (Me) SCH2(D1-34a) CH2(D1-108b, Z = 3-CFThree)
CH (Me) SCH2(D1-34a) CH2(D1-108b, Z = 4-OCFThree)
CH (Me) SCH2(D1-34a) CH2(D1-108b, Z = 2-SCFThree)
CH (Me) SCH2(D1-34a) CH2CH2CN
CH (Me) SCH2(D1-34a) CH2CH2CFThree
CH (Me) SCH2(D1-34a) CH2CH2OMe
CH (Me) SCH2(D1-34a) CH2CH2SMe
CH (Me) SCH2(D1-34a) CH2CH2S (O) Me
CH (Me) SCH2(D1-34a) CH2CH2S (O)2Me
CH (Me) SCH2(D1-34a) D1-32a
CH (Me) SCH2(D1-34a) D1-33a
CH (Me) SCH2(D1-34a) D1-34a
CH (Me) SCH2(D1-34a) D1-37a
CH (Me) SCH2(D1-34a) D1-81a
CH (Me) SCH2(D1-34a) D1-82a
CH (Me) SCH2(D1-34a) D1-84a
CH (Me) SCH2(D1-34a) D1-85a
CH (Me) SCH2(D1-34a) D1-87a
CH (Me) SCH2(D1-34a) D1-92a
CH (Me) SCH2(D1-34a) D1-93a
CH (Me) SCH2(D1-34a) D1-95a
CH (Me) SCH2(D1-34a) D1-96a
CH (Me) SCH2(D1-34a) D1-98a
CH (Me) SCH2(D1-34a) D1-108a
CH (Me) SCH2(D1-34a) D1-108b (Z = 2-Cl)
CH (Me) SCH2(D1-34a) D1-108b (Z = 3-Me)
CH (Me) SCH2(D1-34a) D1-108b (Z = 4-OMe)
CH (Me) SCH2(D1-34a) D1-108b (Z = 2-SMe)
CH (Me) SCH2(D1-34a) D1-108b (Z = 3-CFThree)
CH (Me) SCH2(D1-34a) D1-108b (Z = 4-OCFThree)
CH (Me) SCH2(D1-34a) D1-108b (Z = 2-SCFThree)
CH (Me) SCH2(D1-34a) C (O) Me
CH (Me) SCH2(D1-34a) C (O) CFThree
CH (Me) SCH2(D1-34a) C (O) OMe
CH (Me) S (O) CH2(D1-34a) Me
CH (Me) S (O) CH2(D1-34a) Et
CH (Me) S (O) CH2(D1-34a) Pr-n
CH (Me) S (O) CH2(D1-34a) Pr-i
CH (Me) S (O) CH2(D1-34a) Pr-c
CH (Me) S (O) CH2(D1-34a) Bu-n
CH (Me) S (O) CH2(D1-34a) Bu-i
CH (Me) S (O) CH2(D1-34a) Bu-c
CH (Me) S (O) CH2(D1-34a) Bu-s
CH (Me) S (O) CH2(D1-34a) Bu-t
CH (Me) S (O) CH2(D1-34a) Pen-n
CH (Me) S (O) CH2(D1-34a) Pen-c
CH (Me) S (O) CH2(D1-34a) Hex-n
CH (Me) S (O) CH2(D1-34a) Hex-c
CH (Me) S (O) CH2(D1-34a) CH2Pr-c
CH (Me) S (O) CH2(D1-34a) CH2Bu-c
CH (Me) S (O) CH2(D1-34a) CH2Pen-c
CH (Me) S (O) CH2(D1-34a) CH2Hex-c
CH (Me) S (O) CH2(D1-34a) CH2CH = CH2
CH (Me) S (O) CH2(D1-34a) CH2CH = C (Cl)2
CH (Me) S (O) CH2(D1-34a) CH2C≡CH
CH (Me) S (O) CH2(D1-34a) CH2CN
CH (Me) S (O) CH2(D1-34a) CH2CFThree
CH (Me) S (O) CH2(D1-34a) CH2OMe
CH (Me) S (O) CH2(D1-34a) CH2OCFThree
CH (Me) S (O) CH2(D1-34a) CH2SMe
CH (Me) S (O) CH2(D1-34a) CH2S (O) Me
CH (Me) S (O) CH2(D1-34a) CH2S (O)2Me
CH (Me) S (O) CH2(D1-34a) CH2SCFThree
CH (Me) S (O) CH2(D1-34a) CH2S (O) CFThree
CH (Me) S (O) CH2(D1-34a) CH2S (O)2CFThree
CH (Me) S (O) CH2(D1-34a) CH2CH (OMe)2
CH (Me) S (O) CH2(D1-34a) CH2CH (SMe)2
CH (Me) S (O) CH2(D1-34a) CH2C (O) Me
CH (Me) S (O) CH2(D1-34a) CH2C (O) CFThree
CH (Me) S (O) CH2(D1-34a) CH2C (O) OMe
CH (Me) S (O) CH2(D1-34a) CH2(D1-32a)
CH (Me) S (O) CH2(D1-34a) CH2(D1-33a)
CH (Me) S (O) CH2(D1-34a) CH2(D1-34a)
CH (Me) S (O) CH2(D1-34a) CH2(D1-37a)
CH (Me) S (O) CH2(D1-34a) CH2(D1-81a)
CH (Me) S (O) CH2(D1-34a) CH2(D1-82a)
CH (Me) S (O) CH2(D1-34a) CH2(D1-84a)
CH (Me) S (O) CH2(D1-34a) CH2(D1-85a)
CH (Me) S (O) CH2(D1-34a) CH2(D1-87a)
CH (Me) S (O) CH2(D1-34a) CH2(D1-92a)
CH (Me) S (O) CH2(D1-34a) CH2(D1-93a)
CH (Me) S (O) CH2(D1-34a) CH2(D1-95a)
CH (Me) S (O) CH2(D1-34a) CH2(D1-96a)
CH (Me) S (O) CH2(D1-34a) CH2(D1-98a)
CH (Me) S (O) CH2(D1-34a) CH2(D1-108a)
CH (Me) S (O) CH2(D1-34a) CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O) CH2(D1-34a) CH2(D1-108b, Z = 3-Me)
CH (Me) S (O) CH2(D1-34a) CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O) CH2(D1-34a) CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O) CH2(D1-34a) CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O) CH2(D1-34a) CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O) CH2(D1-34a) CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O) CH2(D1-34a) CH2CH2CN
CH (Me) S (O) CH2(D1-34a) CH2CH2CFThree
CH (Me) S (O) CH2(D1-34a) CH2CH2OMe
CH (Me) S (O) CH2(D1-34a) CH2CH2SMe
CH (Me) S (O) CH2(D1-34a) CH2CH2S (O) Me
CH (Me) S (O) CH2(D1-34a) CH2CH2S (O)2Me
CH (Me) S (O) CH2(D1-34a) D1-32a
CH (Me) S (O) CH2(D1-34a) D1-33a
CH (Me) S (O) CH2(D1-34a) D1-34a
CH (Me) S (O) CH2(D1-34a) D1-37a
CH (Me) S (O) CH2(D1-34a) D1-81a
CH (Me) S (O) CH2(D1-34a) D1-82a
CH (Me) S (O) CH2(D1-34a) D1-84a
CH (Me) S (O) CH2(D1-34a) D1-85a
CH (Me) S (O) CH2(D1-34a) D1-87a
CH (Me) S (O) CH2(D1-34a) D1-92a
CH (Me) S (O) CH2(D1-34a) D1-93a
CH (Me) S (O) CH2(D1-34a) D1-95a
CH (Me) S (O) CH2(D1-34a) D1-96a
CH (Me) S (O) CH2(D1-34a) D1-98a
CH (Me) S (O) CH2(D1-34a) D1-108a
CH (Me) S (O) CH2(D1-34a) D1-108b (Z = 2-Cl)
CH (Me) S (O) CH2(D1-34a) D1-108b (Z = 3-Me)
CH (Me) S (O) CH2(D1-34a) D1-108b (Z = 4-OMe)
CH (Me) S (O) CH2(D1-34a) D1-108b (Z = 2-SMe)
CH (Me) S (O) CH2(D1-34a) D1-108b (Z = 3-CFThree)
CH (Me) S (O) CH2(D1-34a) D1-108b (Z = 4-OCFThree)
CH (Me) S (O) CH2(D1-34a) D1-108b (Z = 2-SCFThree)
CH (Me) S (O) CH2(D1-34a) C (O) Me
CH (Me) S (O) CH2(D1-34a) C (O) CFThree
CH (Me) S (O) CH2(D1-34a) C (O) OMe
CH (Me) S (O)2CH2(D1-34a) Me
CH (Me) S (O)2CH2(D1-34a) Et
CH (Me) S (O)2CH2(D1-34a) Pr-n
CH (Me) S (O)2CH2(D1-34a) Pr-i
CH (Me) S (O)2CH2(D1-34a) Pr-c
CH (Me) S (O)2CH2(D1-34a) Bu-n
CH (Me) S (O)2CH2(D1-34a) Bu-i
CH (Me) S (O)2CH2(D1-34a) Bu-c
CH (Me) S (O)2CH2(D1-34a) Bu-s
CH (Me) S (O)2CH2(D1-34a) Bu-t
CH (Me) S (O)2CH2(D1-34a) Pen-n
CH (Me) S (O)2CH2(D1-34a) Pen-c
CH (Me) S (O)2CH2(D1-34a) Hex-n
CH (Me) S (O)2CH2(D1-34a) Hex-c
CH (Me) S (O)2CH2(D1-34a) CH2Pr-c
CH (Me) S (O)2CH2(D1-34a) CH2Bu-c
CH (Me) S (O)2CH2(D1-34a) CH2Pen-c
CH (Me) S (O)2CH2(D1-34a) CH2Hex-c
CH (Me) S (O)2CH2(D1-34a) CH2CH = CH2
CH (Me) S (O)2CH2(D1-34a) CH2CH = C (Cl)2
CH (Me) S (O)2CH2(D1-34a) CH2C≡CH
CH (Me) S (O)2CH2(D1-34a) CH2CN
CH (Me) S (O)2CH2(D1-34a) CH2CFThree
CH (Me) S (O)2CH2(D1-34a) CH2OMe
CH (Me) S (O)2CH2(D1-34a) CH2OCFThree
CH (Me) S (O)2CH2(D1-34a) CH2SMe
CH (Me) S (O)2CH2(D1-34a) CH2S (O) Me
CH (Me) S (O)2CH2(D1-34a) CH2S (O)2Me
CH (Me) S (O)2CH2(D1-34a) CH2SCFThree
CH (Me) S (O)2CH2(D1-34a) CH2S (O) CFThree
CH (Me) S (O)2CH2(D1-34a) CH2S (O)2CFThree
CH (Me) S (O)2CH2(D1-34a) CH2CH (OMe)2
CH (Me) S (O)2CH2(D1-34a) CH2CH (SMe)2
CH (Me) S (O)2CH2(D1-34a) CH2C (O) Me
CH (Me) S (O)2CH2(D1-34a) CH2C (O) CFThree
CH (Me) S (O)2CH2(D1-34a) CH2C (O) OMe
CH (Me) S (O)2CH2(D1-34a) CH2(D1-32a)
CH (Me) S (O)2CH2(D1-34a) CH2(D1-33a)
CH (Me) S (O)2CH2(D1-34a) CH2(D1-34a)
CH (Me) S (O)2CH2(D1-34a) CH2(D1-37a)
CH (Me) S (O)2CH2(D1-34a) CH2(D1-81a)
CH (Me) S (O)2CH2(D1-34a) CH2(D1-82a)
CH (Me) S (O)2CH2(D1-34a) CH2(D1-84a)
CH (Me) S (O)2CH2(D1-34a) CH2(D1-85a)
CH (Me) S (O)2CH2(D1-34a) CH2(D1-87a)
CH (Me) S (O)2CH2(D1-34a) CH2(D1-92a)
CH (Me) S (O)2CH2(D1-34a) CH2(D1-93a)
CH (Me) S (O)2CH2(D1-34a) CH2(D1-95a)
CH (Me) S (O)2CH2(D1-34a) CH2(D1-96a)
CH (Me) S (O)2CH2(D1-34a) CH2(D1-98a)
CH (Me) S (O)2CH2(D1-34a) CH2(D1-108a)
CH (Me) S (O)2CH2(D1-34a) CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O)2CH2(D1-34a) CH2(D1-108b, Z = 3-Me)
CH (Me) S (O)2CH2(D1-34a) CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O)2CH2(D1-34a) CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O)2CH2(D1-34a) CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O)2CH2(D1-34a) CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O)2CH2(D1-34a) CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O)2CH2(D1-34a) CH2CH2CN
CH (Me) S (O)2CH2(D1-34a) CH2CH2CFThree
CH (Me) S (O)2CH2(D1-34a) CH2CH2OMe
CH (Me) S (O)2CH2(D1-34a) CH2CH2SMe
CH (Me) S (O)2CH2(D1-34a) CH2CH2S (O) Me
CH (Me) S (O)2CH2(D1-34a) CH2CH2S (O)2Me
CH (Me) S (O)2CH2(D1-34a) D1-32a
CH (Me) S (O)2CH2(D1-34a) D1-33a
CH (Me) S (O)2CH2(D1-34a) D1-34a
CH (Me) S (O)2CH2(D1-34a) D1-37a
CH (Me) S (O)2CH2(D1-34a) D1-81a
CH (Me) S (O)2CH2(D1-34a) D1-82a
CH (Me) S (O)2CH2(D1-34a) D1-84a
CH (Me) S (O)2CH2(D1-34a) D1-85a
CH (Me) S (O)2CH2(D1-34a) D1-87a
CH (Me) S (O)2CH2(D1-34a) D1-92a
CH (Me) S (O)2CH2(D1-34a) D1-93a
CH (Me) S (O)2CH2(D1-34a) D1-95a
CH (Me) S (O)2CH2(D1-34a) D1-96a
CH (Me) S (O)2CH2(D1-34a) D1-98a
CH (Me) S (O)2CH2(D1-34a) D1-108a
CH (Me) S (O)2CH2(D1-34a) D1-108b (Z = 2-Cl)
CH (Me) S (O)2CH2(D1-34a) D1-108b (Z = 3-Me)
CH (Me) S (O)2CH2(D1-34a) D1-108b (Z = 4-OMe)
CH (Me) S (O)2CH2(D1-34a) D1-108b (Z = 2-SMe)
CH (Me) S (O)2CH2(D1-34a) D1-108b (Z = 3-CFThree)
CH (Me) S (O)2CH2(D1-34a) D1-108b (Z = 4-OCFThree)
CH (Me) S (O)2CH2(D1-34a) D1-108b (Z = 2-SCFThree)
CH (Me) S (O)2CH2(D1-34a) C (O) Me
CH (Me) S (O)2CH2(D1-34a) C (O) CFThree
CH (Me) S (O)2CH2(D1-34a) C (O) OMe
CH (Et) SCH2(D1-34a) Me
CH (Et) SCH2(D1-34a) Et
CH (Et) SCH2(D1-34a) Pr-n
CH (Et) SCH2(D1-34a) Pr-i
CH (Et) SCH2(D1-34a) Pr-c
CH (Et) SCH2(D1-34a) Bu-n
CH (Et) SCH2(D1-34a) Bu-i
CH (Et) SCH2(D1-34a) Bu-c
CH (Et) SCH2(D1-34a) Bu-s
CH (Et) SCH2(D1-34a) Bu-t
CH (Et) SCH2(D1-34a) Pen-n
CH (Et) SCH2(D1-34a) Pen-c
CH (Et) SCH2(D1-34a) Hex-n
CH (Et) SCH2(D1-34a) Hex-c
CH (Et) SCH2(D1-34a) CH2Pr-c
CH (Et) SCH2(D1-34a) CH2Bu-c
CH (Et) SCH2(D1-34a) CH2Pen-c
CH (Et) SCH2(D1-34a) CH2Hex-c
CH (Et) SCH2(D1-34a) CH2CH = CH2
CH (Et) SCH2(D1-34a) CH2CH = C (Cl)2
CH (Et) SCH2(D1-34a) CH2C≡CH
CH (Et) SCH2(D1-34a) CH2CN
CH (Et) SCH2(D1-34a) CH2CFThree
CH (Et) SCH2(D1-34a) CH2OMe
CH (Et) SCH2(D1-34a) CH2OCFThree
CH (Et) SCH2(D1-34a) CH2SMe
CH (Et) SCH2(D1-34a) CH2S (O) Me
CH (Et) SCH2(D1-34a) CH2S (O)2Me
CH (Et) SCH2(D1-34a) CH2SCFThree
CH (Et) SCH2(D1-34a) CH2S (O) CFThree
CH (Et) SCH2(D1-34a) CH2S (O)2CFThree
CH (Et) SCH2(D1-34a) CH2CH (OMe)2
CH (Et) SCH2(D1-34a) CH2CH (SMe)2
CH (Et) SCH2(D1-34a) CH2C (O) Me
CH (Et) SCH2(D1-34a) CH2C (O) CFThree
CH (Et) SCH2(D1-34a) CH2C (O) OMe
CH (Et) SCH2(D1-34a) CH2(D1-32a)
CH (Et) SCH2(D1-34a) CH2(D1-33a)
CH (Et) SCH2(D1-34a) CH2(D1-34a)
CH (Et) SCH2(D1-34a) CH2(D1-37a)
CH (Et) SCH2(D1-34a) CH2(D1-81a)
CH (Et) SCH2(D1-34a) CH2(D1-82a)
CH (Et) SCH2(D1-34a) CH2(D1-84a)
CH (Et) SCH2(D1-34a) CH2(D1-85a)
CH (Et) SCH2(D1-34a) CH2(D1-87a)
CH (Et) SCH2(D1-34a) CH2(D1-92a)
CH (Et) SCH2(D1-34a) CH2(D1-93a)
CH (Et) SCH2(D1-34a) CH2(D1-95a)
CH (Et) SCH2(D1-34a) CH2(D1-96a)
CH (Et) SCH2(D1-34a) CH2(D1-98a)
CH (Et) SCH2(D1-34a) CH2(D1-108a)
CH (Et) SCH2(D1-34a) CH2(D1-108b, Z = 2-Cl)
CH (Et) SCH2(D1-34a) CH2(D1-108b, Z = 3-Me)
CH (Et) SCH2(D1-34a) CH2(D1-108b, Z = 4-OMe)
CH (Et) SCH2(D1-34a) CH2(D1-108b, Z = 2-SMe)
CH (Et) SCH2(D1-34a) CH2(D1-108b, Z = 3-CFThree)
CH (Et) SCH2(D1-34a) CH2(D1-108b, Z = 4-OCFThree)
CH (Et) SCH2(D1-34a) CH2(D1-108b, Z = 2-SCFThree)
CH (Et) SCH2(D1-34a) CH2CH2CN
CH (Et) SCH2(D1-34a) CH2CH2CFThree
CH (Et) SCH2(D1-34a) CH2CH2OMe
CH (Et) SCH2(D1-34a) CH2CH2SMe
CH (Et) SCH2(D1-34a) CH2CH2S (O) Me
CH (Et) SCH2(D1-34a) CH2CH2S (O)2Me
CH (Et) SCH2(D1-34a) D1-32a
CH (Et) SCH2(D1-34a) D1-33a
CH (Et) SCH2(D1-34a) D1-34a
CH (Et) SCH2(D1-34a) D1-37a
CH (Et) SCH2(D1-34a) D1-81a
CH (Et) SCH2(D1-34a) D1-82a
CH (Et) SCH2(D1-34a) D1-84a
CH (Et) SCH2(D1-34a) D1-85a
CH (Et) SCH2(D1-34a) D1-87a
CH (Et) SCH2(D1-34a) D1-92a
CH (Et) SCH2(D1-34a) D1-93a
CH (Et) SCH2(D1-34a) D1-95a
CH (Et) SCH2(D1-34a) D1-96a
CH (Et) SCH2(D1-34a) D1-98a
CH (Et) SCH2(D1-34a) D1-108a
CH (Et) SCH2(D1-34a) D1-108b (Z = 2-Cl)
CH (Et) SCH2(D1-34a) D1-108b (Z = 3-Me)
CH (Et) SCH2(D1-34a) D1-108b (Z = 4-OMe)
CH (Et) SCH2(D1-34a) D1-108b (Z = 2-SMe)
CH (Et) SCH2(D1-34a) D1-108b (Z = 3-CFThree)
CH (Et) SCH2(D1-34a) D1-108b (Z = 4-OCFThree)
CH (Et) SCH2(D1-34a) D1-108b (Z = 2-SCFThree)
CH (Et) SCH2(D1-34a) C (O) Me
CH (Et) SCH2(D1-34a) C (O) CFThree
CH (Et) SCH2(D1-34a) C (O) OMe
CH (Et) S (O) CH2(D1-34a) Me
CH (Et) S (O) CH2(D1-34a) Et
CH (Et) S (O) CH2(D1-34a) Pr-n
CH (Et) S (O) CH2(D1-34a) Pr-i
CH (Et) S (O) CH2(D1-34a) Pr-c
CH (Et) S (O) CH2(D1-34a) Bu-n
CH (Et) S (O) CH2(D1-34a) Bu-i
CH (Et) S (O) CH2(D1-34a) Bu-c
CH (Et) S (O) CH2(D1-34a) Bu-s
CH (Et) S (O) CH2(D1-34a) Bu-t
CH (Et) S (O) CH2(D1-34a) Pen-n
CH (Et) S (O) CH2(D1-34a) Pen-c
CH (Et) S (O) CH2(D1-34a) Hex-n
CH (Et) S (O) CH2(D1-34a) Hex-c
CH (Et) S (O) CH2(D1-34a) CH2Pr-c
CH (Et) S (O) CH2(D1-34a) CH2Bu-c
CH (Et) S (O) CH2(D1-34a) CH2Pen-c
CH (Et) S (O) CH2(D1-34a) CH2Hex-c
CH (Et) S (O) CH2(D1-34a) CH2CH = CH2
CH (Et) S (O) CH2(D1-34a) CH2CH = C (Cl)2
CH (Et) S (O) CH2(D1-34a) CH2C≡CH
CH (Et) S (O) CH2(D1-34a) CH2CN
CH (Et) S (O) CH2(D1-34a) CH2CFThree
CH (Et) S (O) CH2(D1-34a) CH2OMe
CH (Et) S (O) CH2(D1-34a) CH2OCFThree
CH (Et) S (O) CH2(D1-34a) CH2SMe
CH (Et) S (O) CH2(D1-34a) CH2S (O) Me
CH (Et) S (O) CH2(D1-34a) CH2S (O)2Me
CH (Et) S (O) CH2(D1-34a) CH2SCFThree
CH (Et) S (O) CH2(D1-34a) CH2S (O) CFThree
CH (Et) S (O) CH2(D1-34a) CH2S (O)2CFThree
CH (Et) S (O) CH2(D1-34a) CH2CH (OMe)2
CH (Et) S (O) CH2(D1-34a) CH2CH (SMe)2
CH (Et) S (O) CH2(D1-34a) CH2C (O) Me
CH (Et) S (O) CH2(D1-34a) CH2C (O) CFThree
CH (Et) S (O) CH2(D1-34a) CH2C (O) OMe
CH (Et) S (O) CH2(D1-34a) CH2(D1-32a)
CH (Et) S (O) CH2(D1-34a) CH2(D1-33a)
CH (Et) S (O) CH2(D1-34a) CH2(D1-34a)
CH (Et) S (O) CH2(D1-34a) CH2(D1-37a)
CH (Et) S (O) CH2(D1-34a) CH2(D1-81a)
CH (Et) S (O) CH2(D1-34a) CH2(D1-82a)
CH (Et) S (O) CH2(D1-34a) CH2(D1-84a)
CH (Et) S (O) CH2(D1-34a) CH2(D1-85a)
CH (Et) S (O) CH2(D1-34a) CH2(D1-87a)
CH (Et) S (O) CH2(D1-34a) CH2(D1-92a)
CH (Et) S (O) CH2(D1-34a) CH2(D1-93a)
CH (Et) S (O) CH2(D1-34a) CH2(D1-95a)
CH (Et) S (O) CH2(D1-34a) CH2(D1-96a)
CH (Et) S (O) CH2(D1-34a) CH2(D1-98a)
CH (Et) S (O) CH2(D1-34a) CH2(D1-108a)
CH (Et) S (O) CH2(D1-34a) CH2(D1-108b, Z = 2-Cl)
CH (Et) S (O) CH2(D1-34a) CH2(D1-108b, Z = 3-Me)
CH (Et) S (O) CH2(D1-34a) CH2(D1-108b, Z = 4-OMe)
CH (Et) S (O) CH2(D1-34a) CH2(D1-108b, Z = 2-SMe)
CH (Et) S (O) CH2(D1-34a) CH2(D1-108b, Z = 3-CFThree)
CH (Et) S (O) CH2(D1-34a) CH2(D1-108b, Z = 4-OCFThree)
CH (Et) S (O) CH2(D1-34a) CH2(D1-108b, Z = 2-SCFThree)
CH (Et) S (O) CH2(D1-34a) CH2CH2CN
CH (Et) S (O) CH2(D1-34a) CH2CH2CFThree
CH (Et) S (O) CH2(D1-34a) CH2CH2OMe
CH (Et) S (O) CH2(D1-34a) CH2CH2SMe
CH (Et) S (O) CH2(D1-34a) CH2CH2S (O) Me
CH (Et) S (O) CH2(D1-34a) CH2CH2S (O)2Me
CH (Et) S (O) CH2(D1-34a) D1-32a
CH (Et) S (O) CH2(D1-34a) D1-33a
CH (Et) S (O) CH2(D1-34a) D1-34a
CH (Et) S (O) CH2(D1-34a) D1-37a
CH (Et) S (O) CH2(D1-34a) D1-81a
CH (Et) S (O) CH2(D1-34a) D1-82a
CH (Et) S (O) CH2(D1-34a) D1-84a
CH (Et) S (O) CH2(D1-34a) D1-85a
CH (Et) S (O) CH2(D1-34a) D1-87a
CH (Et) S (O) CH2(D1-34a) D1-92a
CH (Et) S (O) CH2(D1-34a) D1-93a
CH (Et) S (O) CH2(D1-34a) D1-95a
CH (Et) S (O) CH2(D1-34a) D1-96a
CH (Et) S (O) CH2(D1-34a) D1-98a
CH (Et) S (O) CH2(D1-34a) D1-108a
CH (Et) S (O) CH2(D1-34a) D1-108b (Z = 2-Cl)
CH (Et) S (O) CH2(D1-34a) D1-108b (Z = 3-Me)
CH (Et) S (O) CH2(D1-34a) D1-108b (Z = 4-OMe)
CH (Et) S (O) CH2(D1-34a) D1-108b (Z = 2-SMe)
CH (Et) S (O) CH2(D1-34a) D1-108b (Z = 3-CFThree)
CH (Et) S (O) CH2(D1-34a) D1-108b (Z = 4-OCFThree)
CH (Et) S (O) CH2(D1-34a) D1-108b (Z = 2-SCFThree)
CH (Et) S (O) CH2(D1-34a) C (O) Me
CH (Et) S (O) CH2(D1-34a) C (O) CFThree
CH (Et) S (O) CH2(D1-34a) C (O) OMe
CH (Et) S (O)2CH2(D1-34a) Me
CH (Et) S (O)2CH2(D1-34a) Et
CH (Et) S (O)2CH2(D1-34a) Pr-n
CH (Et) S (O)2CH2(D1-34a) Pr-i
CH (Et) S (O)2CH2(D1-34a) Pr-c
CH (Et) S (O)2CH2(D1-34a) Bu-n
CH (Et) S (O)2CH2(D1-34a) Bu-i
CH (Et) S (O)2CH2(D1-34a) Bu-c
CH (Et) S (O)2CH2(D1-34a) Bu-s
CH (Et) S (O)2CH2(D1-34a) Bu-t
CH (Et) S (O)2CH2(D1-34a) Pen-n
CH (Et) S (O)2CH2(D1-34a) Pen-c
CH (Et) S (O)2CH2(D1-34a) Hex-n
CH (Et) S (O)2CH2(D1-34a) Hex-c
CH (Et) S (O)2CH2(D1-34a) CH2Pr-c
CH (Et) S (O)2CH2(D1-34a) CH2Bu-c
CH (Et) S (O)2CH2(D1-34a) CH2Pen-c
CH (Et) S (O)2CH2(D1-34a) CH2Hex-c
CH (Et) S (O)2CH2(D1-34a) CH2CH = CH2
CH (Et) S (O)2CH2(D1-34a) CH2CH = C (Cl)2
CH (Et) S (O)2CH2(D1-34a) CH2C≡CH
CH (Et) S (O)2CH2(D1-34a) CH2CN
CH (Et) S (O)2CH2(D1-34a) CH2CFThree
CH (Et) S (O)2CH2(D1-34a) CH2OMe
CH (Et) S (O)2CH2(D1-34a) CH2OCFThree
CH (Et) S (O)2CH2(D1-34a) CH2SMe
CH (Et) S (O)2CH2(D1-34a) CH2S (O) Me
CH (Et) S (O)2CH2(D1-34a) CH2S (O)2Me
CH (Et) S (O)2CH2(D1-34a) CH2SCFThree
CH (Et) S (O)2CH2(D1-34a) CH2S (O) CFThree
CH (Et) S (O)2CH2(D1-34a) CH2S (O)2CFThree
CH (Et) S (O)2CH2(D1-34a) CH2CH (OMe)2
CH (Et) S (O)2CH2(D1-34a) CH2CH (SMe)2
CH (Et) S (O)2CH2(D1-34a) CH2C (O) Me
CH (Et) S (O)2CH2(D1-34a) CH2C (O) CFThree
CH (Et) S (O)2CH2(D1-34a) CH2C (O) OMe
CH (Et) S (O)2CH2(D1-34a) CH2(D1-32a)
CH (Et) S (O)2CH2(D1-34a) CH2(D1-33a)
CH (Et) S (O)2CH2(D1-34a) CH2(D1-34a)
CH (Et) S (O)2CH2(D1-34a) CH2(D1-37a)
CH (Et) S (O)2CH2(D1-34a) CH2(D1-81a)
CH (Et) S (O)2CH2(D1-34a) CH2(D1-82a)
CH (Et) S (O)2CH2(D1-34a) CH2(D1-84a)
CH (Et) S (O)2CH2(D1-34a) CH2(D1-85a)
CH (Et) S (O)2CH2(D1-34a) CH2(D1-87a)
CH (Et) S (O)2CH2(D1-34a) CH2(D1-92a)
CH (Et) S (O)2CH2(D1-34a) CH2(D1-93a)
CH (Et) S (O)2CH2(D1-34a) CH2(D1-95a)
CH (Et) S (O)2CH2(D1-34a) CH2(D1-96a)
CH (Et) S (O)2CH2(D1-34a) CH2(D1-98a)
CH (Et) S (O)2CH2(D1-34a) CH2(D1-108a)
CH (Et) S (O)2CH2(D1-34a) CH2(D1-108b, Z = 2-Cl)
CH (Et) S (O)2CH2(D1-34a) CH2(D1-108b, Z = 3-Me)
CH (Et) S (O)2CH2(D1-34a) CH2(D1-108b, Z = 4-OMe)
CH (Et) S (O)2CH2(D1-34a) CH2(D1-108b, Z = 2-SMe)
CH (Et) S (O)2CH2(D1-34a) CH2(D1-108b, Z = 3-CFThree)
CH (Et) S (O)2CH2(D1-34a) CH2(D1-108b, Z = 4-OCFThree)
CH (Et) S (O)2CH2(D1-34a) CH2(D1-108b, Z = 2-SCFThree)
CH (Et) S (O)2CH2(D1-34a) CH2CH2CN
CH (Et) S (O)2CH2(D1-34a) CH2CH2CFThree
CH (Et) S (O)2CH2(D1-34a) CH2CH2OMe
CH (Et) S (O)2CH2(D1-34a) CH2CH2SMe
CH (Et) S (O)2CH2(D1-34a) CH2CH2S (O) Me
CH (Et) S (O)2CH2(D1-34a) CH2CH2S (O)2Me
CH (Et) S (O)2CH2(D1-34a) D1-32a
CH (Et) S (O)2CH2(D1-34a) D1-33a
CH (Et) S (O)2CH2(D1-34a) D1-34a
CH (Et) S (O)2CH2(D1-34a) D1-37a
CH (Et) S (O)2CH2(D1-34a) D1-81a
CH (Et) S (O)2CH2(D1-34a) D1-82a
CH (Et) S (O)2CH2(D1-34a) D1-84a
CH (Et) S (O)2CH2(D1-34a) D1-85a
CH (Et) S (O)2CH2(D1-34a) D1-87a
CH (Et) S (O)2CH2(D1-34a) D1-92a
CH (Et) S (O)2CH2(D1-34a) D1-93a
CH (Et) S (O)2CH2(D1-34a) D1-95a
CH (Et) S (O)2CH2(D1-34a) D1-96a
CH (Et) S (O)2CH2(D1-34a) D1-98a
CH (Et) S (O)2CH2(D1-34a) D1-108a
CH (Et) S (O)2CH2(D1-34a) D1-108b (Z = 2-Cl)
CH (Et) S (O)2CH2(D1-34a) D1-108b (Z = 3-Me)
CH (Et) S (O)2CH2(D1-34a) D1-108b (Z = 4-OMe)
CH (Et) S (O)2CH2(D1-34a) D1-108b (Z = 2-SMe)
CH (Et) S (O)2CH2(D1-34a) D1-108b (Z = 3-CFThree)
CH (Et) S (O)2CH2(D1-34a) D1-108b (Z = 4-OCFThree)
CH (Et) S (O)2CH2(D1-34a) D1-108b (Z = 2-SCFThree)
CH (Et) S (O)2CH2(D1-34a) C (O) Me
CH (Et) S (O)2CH2(D1-34a) C (O) CFThree
CH (Et) S (O)2CH2(D1-34a) C (O) OMe
CH2S {D1-32b (X1= 5-CFThree)} Me
CH2S {D1-32b (X1= 5-CFThree)} Et
CH2S {D1-32b (X1= 5-CFThree)} Pr-n
CH2S {D1-32b (X1= 5-CFThree)} Pr-i
CH2S {D1-32b (X1= 5-CFThree)} Pr-c
CH2S {D1-32b (X1= 5-CFThree)} Bu-n
CH2S {D1-32b (X1= 5-CFThree)} Bu-i
CH2S {D1-32b (X1= 5-CFThree)} Bu-c
CH2S {D1-32b (X1= 5-CFThree)} Bu-s
CH2S {D1-32b (X1= 5-CFThree)} Bu-t
CH2S {D1-32b (X1= 5-CFThree)} Pen-n
CH2S {D1-32b (X1= 5-CFThree)} Pen-c
CH2S {D1-32b (X1= 5-CFThree)} Hex-n
CH2S {D1-32b (X1= 5-CFThree)} Hex-c
CH2S {D1-32b (X1= 5-CFThree)} CH2Pr-c
CH2S {D1-32b (X1= 5-CFThree)} CH2Bu-c
CH2S {D1-32b (X1= 5-CFThree)} CH2Pen-c
CH2S {D1-32b (X1= 5-CFThree)} CH2Hex-c
CH2S {D1-32b (X1= 5-CFThree)} CH2CH = CH2
CH2S {D1-32b (X1= 5-CFThree)} CH2CH = C (Cl)2
CH2S {D1-32b (X1= 5-CFThree)} CH2C≡CH
CH2S {D1-32b (X1= 5-CFThree)} CH2CN
CH2S {D1-32b (X1= 5-CFThree)} CH2CFThree
CH2S {D1-32b (X1= 5-CFThree)} CH2OMe
CH2S {D1-32b (X1= 5-CFThree)} CH2OCFThree
CH2S {D1-32b (X1= 5-CFThree)} CH2SMe
CH2S {D1-32b (X1= 5-CFThree)} CH2S (O) Me
CH2S {D1-32b (X1= 5-CFThree)} CH2S (O)2Me
CH2S {D1-32b (X1= 5-CFThree)} CH2SCFThree
CH2S {D1-32b (X1= 5-CFThree)} CH2S (O) CFThree
CH2S {D1-32b (X1= 5-CFThree)} CH2S (O)2CFThree
CH2S {D1-32b (X1= 5-CFThree)} CH2CH (OMe)2
CH2S {D1-32b (X1= 5-CFThree)} CH2CH (SMe)2
CH2S {D1-32b (X1= 5-CFThree)} CH2C (O) Me
CH2S {D1-32b (X1= 5-CFThree)} CH2C (O) CFThree
CH2S {D1-32b (X1= 5-CFThree)} CH2C (O) OMe
CH2S {D1-32b (X1= 5-CFThree)} CH2(D1-32a)
CH2S {D1-32b (X1= 5-CFThree)} CH2(D1-33a)
CH2S {D1-32b (X1= 5-CFThree)} CH2(D1-34a)
CH2S {D1-32b (X1= 5-CFThree)} CH2(D1-37a)
CH2S {D1-32b (X1= 5-CFThree)} CH2(D1-81a)
CH2S {D1-32b (X1= 5-CFThree)} CH2(D1-82a)
CH2S {D1-32b (X1= 5-CFThree)} CH2(D1-84a)
CH2S {D1-32b (X1= 5-CFThree)} CH2(D1-85a)
CH2S {D1-32b (X1= 5-CFThree)} CH2(D1-87a)
CH2S {D1-32b (X1= 5-CFThree)} CH2(D1-92a)
CH2S {D1-32b (X1= 5-CFThree)} CH2(D1-93a)
CH2S {D1-32b (X1= 5-CFThree)} CH2(D1-95a)
CH2S {D1-32b (X1= 5-CFThree)} CH2(D1-96a)
CH2S {D1-32b (X1= 5-CFThree)} CH2(D1-98a)
CH2S {D1-32b (X1= 5-CFThree)} CH2(D1-108a)
CH2S {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-Cl)
CH2S {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 3-Me)
CH2S {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 4-OMe)
CH2S {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-SMe)
CH2S {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 3-CFThree)
CH2S {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 4-OCFThree)
CH2S {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-SCFThree)
CH2S {D1-32b (X1= 5-CFThree)} CH2CH2CN
CH2S {D1-32b (X1= 5-CFThree)} CH2CH2CFThree
CH2S {D1-32b (X1= 5-CFThree)} CH2CH2OMe
CH2S {D1-32b (X1= 5-CFThree)} CH2CH2SMe
CH2S {D1-32b (X1= 5-CFThree)} CH2CH2S (O) Me
CH2S {D1-32b (X1= 5-CFThree)} CH2CH2S (O)2Me
CH2S {D1-32b (X1= 5-CFThree)} D1-32a
CH2S {D1-32b (X1= 5-CFThree)} D1-33a
CH2S {D1-32b (X1= 5-CFThree)} D1-34a
CH2S {D1-32b (X1= 5-CFThree)} D1-37a
CH2S {D1-32b (X1= 5-CFThree)} D1-81a
CH2S {D1-32b (X1= 5-CFThree)} D1-82a
CH2S {D1-32b (X1= 5-CFThree)} D1-84a
CH2S {D1-32b (X1= 5-CFThree)} D1-85a
CH2S {D1-32b (X1= 5-CFThree)} D1-87a
CH2S {D1-32b (X1= 5-CFThree)} D1-92a
CH2S {D1-32b (X1= 5-CFThree)} D1-93a
CH2S {D1-32b (X1= 5-CFThree)} D1-95a
CH2S {D1-32b (X1= 5-CFThree)} D1-96a
CH2S {D1-32b (X1= 5-CFThree)} D1-98a
CH2S {D1-32b (X1= 5-CFThree)} D1-108a
CH2S {D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-Cl)
CH2S {D1-32b (X1= 5-CFThree)} D1-108b (Z = 3-Me)
CH2S {D1-32b (X1= 5-CFThree)} D1-108b (Z = 4-OMe)
CH2S {D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-SMe)
CH2S {D1-32b (X1= 5-CFThree)} D1-108b (Z = 3-CFThree)
CH2S {D1-32b (X1= 5-CFThree)} D1-108b (Z = 4-OCFThree)
CH2S {D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-SCFThree)
CH2S {D1-32b (X1= 5-CFThree)} C (O) Me
CH2S {D1-32b (X1= 5-CFThree)} C (O) CFThree
CH2S {D1-32b (X1= 5-CFThree)} C (O) OMe
CH2S (O) {D1-32b (X1= 5-CFThree)} Me
CH2S (O) {D1-32b (X1= 5-CFThree)} Et
CH2S (O) {D1-32b (X1= 5-CFThree)} Pr-n
CH2S (O) {D1-32b (X1= 5-CFThree)} Pr-i
CH2S (O) {D1-32b (X1= 5-CFThree)} Pr-c
CH2S (O) {D1-32b (X1= 5-CFThree)} Bu-n
CH2S (O) {D1-32b (X1= 5-CFThree)} Bu-i
CH2S (O) {D1-32b (X1= 5-CFThree)} Bu-c
CH2S (O) {D1-32b (X1= 5-CFThree)} Bu-s
CH2S (O) {D1-32b (X1= 5-CFThree)} Bu-t
CH2S (O) {D1-32b (X1= 5-CFThree)} Pen-n
CH2S (O) {D1-32b (X1= 5-CFThree)} Pen-c
CH2S (O) {D1-32b (X1= 5-CFThree)} Hex-n
CH2S (O) {D1-32b (X1= 5-CFThree)} Hex-c
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2Pr-c
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2Bu-c
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2Pen-c
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2Hex-c
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2CH = CH2
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2CH = C (Cl)2
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2C≡CH
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2CN
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2CFThree
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2OMe
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2OCFThree
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2SMe
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2S (O) Me
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2S (O)2Me
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2SCFThree
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2S (O) CFThree
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2S (O)2CFThree
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2CH (OMe)2
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2CH (SMe)2
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2C (O) Me
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2C (O) CFThree
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2C (O) OMe
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-32a)
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-33a)
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-34a)
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-37a)
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-81a)
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-82a)
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-84a)
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-85a)
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-87a)
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-92a)
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-93a)
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-95a)
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-96a)
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-98a)
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108a)
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-Cl)
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 3-Me)
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 4-OMe)
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-SMe)
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 3-CFThree)
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 4-OCFThree)
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-SCFThree)
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2CH2CN
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2CH2CFThree
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2CH2OMe
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2CH2SMe
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2CH2S (O) Me
CH2S (O) {D1-32b (X1= 5-CFThree)} CH2CH2S (O)2Me
CH2S (O) {D1-32b (X1= 5-CFThree)} D1-32a
CH2S (O) {D1-32b (X1= 5-CFThree)} D1-33a
CH2S (O) {D1-32b (X1= 5-CFThree)} D1-34a
CH2S (O) {D1-32b (X1= 5-CFThree)} D1-37a
CH2S (O) {D1-32b (X1= 5-CFThree)} D1-81a
CH2S (O) {D1-32b (X1= 5-CFThree)} D1-82a
CH2S (O) {D1-32b (X1= 5-CFThree)} D1-84a
CH2S (O) {D1-32b (X1= 5-CFThree)} D1-85a
CH2S (O) {D1-32b (X1= 5-CFThree)} D1-87a
CH2S (O) {D1-32b (X1= 5-CFThree)} D1-92a
CH2S (O) {D1-32b (X1= 5-CFThree)} D1-93a
CH2S (O) {D1-32b (X1= 5-CFThree)} D1-95a
CH2S (O) {D1-32b (X1= 5-CFThree)} D1-96a
CH2S (O) {D1-32b (X1= 5-CFThree)} D1-98a
CH2S (O) {D1-32b (X1= 5-CFThree)} D1-108a
CH2S (O) {D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-Cl)
CH2S (O) {D1-32b (X1= 5-CFThree)} D1-108b (Z = 3-Me)
CH2S (O) {D1-32b (X1= 5-CFThree)} D1-108b (Z = 4-OMe)
CH2S (O) {D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-SMe)
CH2S (O) {D1-32b (X1= 5-CFThree)} D1-108b (Z = 3-CFThree)
CH2S (O) {D1-32b (X1= 5-CFThree)} D1-108b (Z = 4-OCFThree)
CH2S (O) {D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-SCFThree)
CH2S (O) {D1-32b (X1= 5-CFThree)} C (O) Me
CH2S (O) {D1-32b (X1= 5-CFThree)} C (O) CFThree
CH2S (O) {D1-32b (X1= 5-CFThree)} C (O) OMe
CH2S (O)2{D1-32b (X1= 5-CFThree)} Me
CH2S (O)2{D1-32b (X1= 5-CFThree)} Et
CH2S (O)2{D1-32b (X1= 5-CFThree)} Pr-n
CH2S (O)2{D1-32b (X1= 5-CFThree)} Pr-i
CH2S (O)2{D1-32b (X1= 5-CFThree)} Pr-c
CH2S (O)2{D1-32b (X1= 5-CFThree)} Bu-n
CH2S (O)2{D1-32b (X1= 5-CFThree)} Bu-i
CH2S (O)2{D1-32b (X1= 5-CFThree)} Bu-c
CH2S (O)2{D1-32b (X1= 5-CFThree)} Bu-s
CH2S (O)2{D1-32b (X1= 5-CFThree)} Bu-t
CH2S (O)2{D1-32b (X1= 5-CFThree)} Pen-n
CH2S (O)2{D1-32b (X1= 5-CFThree)} Pen-c
CH2S (O)2{D1-32b (X1= 5-CFThree)} Hex-n
CH2S (O)2{D1-32b (X1= 5-CFThree)} Hex-c
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2Pr-c
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2Bu-c
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2Pen-c
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2Hex-c
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2CH = CH2
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2CH = C (Cl)2
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2C≡CH
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2CN
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2CFThree
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2OMe
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2OCFThree
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2SMe
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2S (O) Me
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2S (O)2Me
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2SCFThree
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2S (O) CFThree
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2S (O)2CFThree
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2CH (OMe)2
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2CH (SMe)2
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2C (O) Me
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2C (O) CFThree
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2C (O) OMe
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-32a)
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-33a)
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-34a)
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-37a)
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-81a)
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-82a)
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-84a)
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-85a)
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-87a)
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-92a)
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-93a)
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-95a)
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-96a)
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-98a)
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108a)
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-Cl)
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 3-Me)
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 4-OMe)
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-SMe)
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 3-CFThree)
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 4-OCFThree)
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-SCFThree)
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2CH2CN
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2CH2CFThree
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2CH2OMe
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2CH2SMe
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2CH2S (O) Me
CH2S (O)2{D1-32b (X1= 5-CFThree)} CH2CH2S (O)2Me
CH2S (O)2{D1-32b (X1= 5-CFThree)} D1-32a
CH2S (O)2{D1-32b (X1= 5-CFThree)} D1-33a
CH2S (O)2{D1-32b (X1= 5-CFThree)} D1-34a
CH2S (O)2{D1-32b (X1= 5-CFThree)} D1-37a
CH2S (O)2{D1-32b (X1= 5-CFThree)} D1-81a
CH2S (O)2{D1-32b (X1= 5-CFThree)} D1-82a
CH2S (O)2{D1-32b (X1= 5-CFThree)} D1-84a
CH2S (O)2{D1-32b (X1= 5-CFThree)} D1-85a
CH2S (O)2{D1-32b (X1= 5-CFThree)} D1-87a
CH2S (O)2{D1-32b (X1= 5-CFThree)} D1-92a
CH2S (O)2{D1-32b (X1= 5-CFThree)} D1-93a
CH2S (O)2{D1-32b (X1= 5-CFThree)} D1-95a
CH2S (O)2{D1-32b (X1= 5-CFThree)} D1-96a
CH2S (O)2{D1-32b (X1= 5-CFThree)} D1-98a
CH2S (O)2{D1-32b (X1= 5-CFThree)} D1-108a
CH2S (O)2{D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-Cl)
CH2S (O)2{D1-32b (X1= 5-CFThree)} D1-108b (Z = 3-Me)
CH2S (O)2{D1-32b (X1= 5-CFThree)} D1-108b (Z = 4-OMe)
CH2S (O)2{D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-SMe)
CH2S (O)2{D1-32b (X1= 5-CFThree)} D1-108b (Z = 3-CFThree)
CH2S (O)2{D1-32b (X1= 5-CFThree)} D1-108b (Z = 4-OCFThree)
CH2S (O)2{D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-SCFThree)
CH2S (O)2{D1-32b (X1= 5-CFThree)} C (O) Me
CH2S (O)2{D1-32b (X1= 5-CFThree)} C (O) CFThree
CH2S (O)2{D1-32b (X1= 5-CFThree)} C (O) OMe
CH (Me) S {D1-32b (X1= 5-CFThree)} Me
CH (Me) S {D1-32b (X1= 5-CFThree)} Et
CH (Me) S {D1-32b (X1= 5-CFThree)} Pr-n
CH (Me) S {D1-32b (X1= 5-CFThree)} Pr-i
CH (Me) S {D1-32b (X1= 5-CFThree)} Pr-c
CH (Me) S {D1-32b (X1= 5-CFThree)} Bu-n
CH (Me) S {D1-32b (X1= 5-CFThree)} Bu-i
CH (Me) S {D1-32b (X1= 5-CFThree)} Bu-c
CH (Me) S {D1-32b (X1= 5-CFThree)} Bu-s
CH (Me) S {D1-32b (X1= 5-CFThree)} Bu-t
CH (Me) S {D1-32b (X1= 5-CFThree)} Pen-n
CH (Me) S {D1-32b (X1= 5-CFThree)} Pen-c
CH (Me) S {D1-32b (X1= 5-CFThree)} Hex-n
CH (Me) S {D1-32b (X1= 5-CFThree)} Hex-c
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2Pr-c
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2Bu-c
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2Pen-c
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2Hex-c
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2CH = CH2
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2CH = C (Cl)2
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2C≡CH
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2CN
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2CFThree
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2OMe
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2OCFThree
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2SMe
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2S (O) Me
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2S (O)2Me
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2SCFThree
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2S (O) CFThree
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2S (O)2CFThree
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2CH (OMe)2
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2CH (SMe)2
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2C (O) Me
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2C (O) CFThree
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2C (O) OMe
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2(D1-32a)
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2(D1-33a)
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2(D1-34a)
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2(D1-37a)
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2(D1-81a)
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2(D1-82a)
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2(D1-84a)
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2(D1-85a)
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2(D1-87a)
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2(D1-92a)
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2(D1-93a)
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2(D1-95a)
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2(D1-96a)
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2(D1-98a)
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2(D1-108a)
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-Cl)
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 3-Me)
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 4-OMe)
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-SMe)
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 3-CFThree)
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2CH2CN
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2CH2CFThree
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2CH2OMe
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2CH2SMe
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2CH2S (O) Me
CH (Me) S {D1-32b (X1= 5-CFThree)} CH2CH2S (O)2Me
CH (Me) S {D1-32b (X1= 5-CFThree)} D1-32a
CH (Me) S {D1-32b (X1= 5-CFThree)} D1-33a
CH (Me) S {D1-32b (X1= 5-CFThree)} D1-34a
CH (Me) S {D1-32b (X1= 5-CFThree)} D1-37a
CH (Me) S {D1-32b (X1= 5-CFThree)} D1-81a
CH (Me) S {D1-32b (X1= 5-CFThree)} D1-82a
CH (Me) S {D1-32b (X1= 5-CFThree)} D1-84a
CH (Me) S {D1-32b (X1= 5-CFThree)} D1-85a
CH (Me) S {D1-32b (X1= 5-CFThree)} D1-87a
CH (Me) S {D1-32b (X1= 5-CFThree)} D1-92a
CH (Me) S {D1-32b (X1= 5-CFThree)} D1-93a
CH (Me) S {D1-32b (X1= 5-CFThree)} D1-95a
CH (Me) S {D1-32b (X1= 5-CFThree)} D1-96a
CH (Me) S {D1-32b (X1= 5-CFThree)} D1-98a
CH (Me) S {D1-32b (X1= 5-CFThree)} D1-108a
CH (Me) S {D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-Cl)
CH (Me) S {D1-32b (X1= 5-CFThree)} D1-108b (Z = 3-Me)
CH (Me) S {D1-32b (X1= 5-CFThree)} D1-108b (Z = 4-OMe)
CH (Me) S {D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-SMe)
CH (Me) S {D1-32b (X1= 5-CFThree)} D1-108b (Z = 3-CFThree)
CH (Me) S {D1-32b (X1= 5-CFThree)} D1-108b (Z = 4-OCFThree)
CH (Me) S {D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-SCFThree)
CH (Me) S {D1-32b (X1= 5-CFThree)} C (O) Me
CH (Me) S {D1-32b (X1= 5-CFThree)} C (O) CFThree
CH (Me) S {D1-32b (X1= 5-CFThree)} C (O) OMe
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} Me
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} Et
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} Pr-n
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} Pr-i
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} Pr-c
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} Bu-n
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} Bu-i
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} Bu-c
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} Bu-s
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} Bu-t
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} Pen-n
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} Pen-c
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} Hex-n
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} Hex-c
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2Pr-c
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2Bu-c
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2Pen-c
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2Hex-c
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2CH = CH2
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2CH = C (Cl)2
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2C≡CH
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2CN
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2CFThree
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2OMe
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2OCFThree
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2SMe
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2S (O) Me
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2S (O)2Me
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2SCFThree
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2S (O) CFThree
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2S (O)2CFThree
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2CH (OMe)2
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2CH (SMe)2
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2C (O) Me
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2C (O) CFThree
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2C (O) OMe
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-32a)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-33a)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-34a)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-37a)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-81a)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-82a)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-84a)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-85a)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-87a)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-92a)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-93a)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-95a)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-96a)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-98a)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108a)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 3-Me)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2CH2CN
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2CH2CFThree
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2CH2OMe
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2CH2SMe
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2CH2S (O) Me
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} CH2CH2S (O)2Me
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} D1-32a
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} D1-33a
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} D1-34a
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} D1-37a
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} D1-81a
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} D1-82a
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} D1-84a
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} D1-85a
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} D1-87a
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} D1-92a
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} D1-93a
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} D1-95a
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} D1-96a
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} D1-98a
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} D1-108a
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-Cl)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} D1-108b (Z = 3-Me)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} D1-108b (Z = 4-OMe)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-SMe)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} D1-108b (Z = 3-CFThree)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} D1-108b (Z = 4-OCFThree)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-SCFThree)
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} C (O) Me
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} C (O) CFThree
CH (Me) S (O) {D1-32b (X1= 5-CFThree)} C (O) OMe
CH (Me) S (O)2{D1-32b (X1= 5-CF3)} Me
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} Et
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} Pr-n
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} Pr-i
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} Pr-c
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} Bu-n
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} Bu-i
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} Bu-c
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} Bu-s
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} Bu-t
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} Pen-n
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} Pen-c
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} Hex-n
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} Hex-c
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2Pr-c
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2Bu-c
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2Pen-c
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2Hex-c
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2CH = CH2
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2CH = C (Cl)2
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2C≡CH
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2CN
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2CFThree
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2OMe
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2OCFThree
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2SMe
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2S (O) Me
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2S (O)2Me
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2SCFThree
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2S (O) CFThree
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2S (O)2CFThree
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2CH (OMe)2
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2CH (SMe)2
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2C (O) Me
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2C (O) CFThree
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2C (O) OMe
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-32a)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-33a)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-34a)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-37a)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-81a)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-82a)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-84a)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-85a)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-87a)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-92a)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-93a)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-95a)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-96a)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-98a)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108a)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 3-Me)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2CH2CN
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2CH2CFThree
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2CH2OMe
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2CH2SMe
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2CH2S (O) Me
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} CH2CH2S (O)2Me
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} D1-32a
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} D1-33a
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} D1-34a
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} D1-37a
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} D1-81a
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} D1-82a
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} D1-84a
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} D1-85a
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} D1-87a
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} D1-92a
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} D1-93a
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} D1-95a
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} D1-96a
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} D1-98a
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} D1-108a
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-Cl)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} D1-108b (Z = 3-Me)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} D1-108b (Z = 4-OMe)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-SMe)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} D1-108b (Z = 3-CFThree)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} D1-108b (Z = 4-OCFThree)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-SCFThree)
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} C (O) Me
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} C (O) CFThree
CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} C (O) OMe
CH (Et) S {D1-32b (X1= 5-CFThree)} Me
CH (Et) S {D1-32b (X1= 5-CFThree)} Et
CH (Et) S {D1-32b (X1= 5-CFThree)} Pr-n
CH (Et) S {D1-32b (X1= 5-CFThree)} Pr-i
CH (Et) S {D1-32b (X1= 5-CFThree)} Pr-c
CH (Et) S {D1-32b (X1= 5-CFThree)} Bu-n
CH (Et) S {D1-32b (X1= 5-CFThree)} Bu-i
CH (Et) S {D1-32b (X1= 5-CFThree)} Bu-c
CH (Et) S {D1-32b (X1= 5-CFThree)} Bu-s
CH (Et) S {D1-32b (X1= 5-CFThree)} Bu-t
CH (Et) S {D1-32b (X1= 5-CFThree)} Pen-n
CH (Et) S {D1-32b (X1= 5-CFThree)} Pen-c
CH (Et) S {D1-32b (X1= 5-CFThree)} Hex-n
CH (Et) S {D1-32b (X1= 5-CFThree)} Hex-c
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2Pr-c
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2Bu-c
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2Pen-c
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2Hex-c
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2CH = CH2
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2CH = C (Cl)2
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2C≡CH
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2CN
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2CFThree
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2OMe
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2OCFThree
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2SMe
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2S (O) Me
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2S (O)2Me
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2SCFThree
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2S (O) CFThree
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2S (O)2CFThree
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2CH (OMe)2
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2CH (SMe)2
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2C (O) Me
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2C (O) CFThree
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2C (O) OMe
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2(D1-32a)
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2(D1-33a)
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2(D1-34a)
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2(D1-37a)
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2(D1-81a)
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2(D1-82a)
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2(D1-84a)
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2(D1-85a)
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2(D1-87a)
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2(D1-92a)
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2(D1-93a)
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2(D1-95a)
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2(D1-96a)
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2(D1-98a)
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2(D1-108a)
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-Cl)
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 3-Me)
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 4-OMe)
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-SMe)
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 3-CFThree)
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 4-OCFThree)
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-SCFThree)
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2CH2CN
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2CH2CFThree
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2CH2OMe
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2CH2SMe
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2CH2S (O) Me
CH (Et) S {D1-32b (X1= 5-CFThree)} CH2CH2S (O)2Me
CH (Et) S {D1-32b (X1= 5-CFThree)} D1-32a
CH (Et) S {D1-32b (X1= 5-CFThree)} D1-33a
CH (Et) S {D1-32b (X1= 5-CFThree)} D1-34a
CH (Et) S {D1-32b (X1= 5-CFThree)} D1-37a
CH (Et) S {D1-32b (X1= 5-CFThree)} D1-81a
CH (Et) S {D1-32b (X1= 5-CFThree)} D1-82a
CH (Et) S {D1-32b (X1= 5-CFThree)} D1-84a
CH (Et) S {D1-32b (X1= 5-CFThree)} D1-85a
CH (Et) S {D1-32b (X1= 5-CFThree)} D1-87a
CH (Et) S {D1-32b (X1= 5-CFThree)} D1-92a
CH (Et) S {D1-32b (X1= 5-CFThree)} D1-93a
CH (Et) S {D1-32b (X1= 5-CFThree)} D1-95a
CH (Et) S {D1-32b (X1= 5-CFThree)} D1-96a
CH (Et) S {D1-32b (X1= 5-CFThree)} D1-98a
CH (Et) S {D1-32b (X1= 5-CFThree)} D1-108a
CH (Et) S {D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-Cl)
CH (Et) S {D1-32b (X1= 5-CFThree)} D1-108b (Z = 3-Me)
CH (Et) S {D1-32b (X1= 5-CFThree)} D1-108b (Z = 4-OMe)
CH (Et) S {D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-SMe)
CH (Et) S {D1-32b (X1= 5-CFThree)} D1-108b (Z = 3-CFThree)
CH (Et) S {D1-32b (X1= 5-CFThree)} D1-108b (Z = 4-OCFThree)
CH (Et) S {D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-SCFThree)
CH (Et) S {D1-32b (X1= 5-CFThree)} C (O) Me
CH (Et) S {D1-32b (X1= 5-CFThree)} C (O) CFThree
CH (Et) S {D1-32b (X1= 5-CFThree)} C (O) OMe
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} Me
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} Et
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} Pr-n
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} Pr-i
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} Pr-c
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} Bu-n
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} Bu-i
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} Bu-c
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} Bu-s
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} Bu-t
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} Pen-n
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} Pen-c
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} Hex-n
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} Hex-c
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2Pr-c
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2Bu-c
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2Pen-c
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2Hex-c
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2CH = CH2
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2CH = C (Cl)2
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2C≡CH
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2CN
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2CFThree
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2OMe
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2OCFThree
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2SMe
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2S (O) Me
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2S (O)2Me
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2SCFThree
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2S (O) CFThree
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2S (O)2CFThree
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2CH (OMe)2
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2CH (SMe)2
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2C (O) Me
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2C (O) CFThree
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2C (O) OMe
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-32a)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-33a)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-34a)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-37a)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-81a)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-82a)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-84a)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-85a)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-87a)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-92a)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-93a)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-95a)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-96a)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-98a)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108a)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-Cl)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 3-Me)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 4-OMe)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-SMe)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 3-CFThree)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 4-OCFThree)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-SCFThree)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2CH2CN
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2CH2CFThree
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2CH2OMe
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2CH2SMe
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2CH2S (O) Me
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} CH2CH2S (O)2Me
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} D1-32a
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} D1-33a
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} D1-34a
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} D1-37a
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} D1-81a
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} D1-82a
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} D1-84a
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} D1-85a
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} D1-87a
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} D1-92a
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} D1-93a
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} D1-95a
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} D1-96a
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} D1-98a
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} D1-108a
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-Cl)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} D1-108b (Z = 3-Me)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} D1-108b (Z = 4-OMe)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-SMe)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} D1-108b (Z = 3-CFThree)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} D1-108b (Z = 4-OCFThree)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-SCFThree)
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} C (O) Me
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} C (O) CFThree
CH (Et) S (O) {D1-32b (X1= 5-CFThree)} C (O) OMe
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} Me
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} Et
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} Pr-n
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} Pr-i
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} Pr-c
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} Bu-n
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} Bu-i
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} Bu-c
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} Bu-s
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} Bu-t
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} Pen-n
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} Pen-c
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} Hex-n
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} Hex-c
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2Pr-c
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2Bu-c
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2Pen-c
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2Hex-c
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2CH = CH2
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2CH = C (Cl)2
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2C≡CH
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2CN
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2CFThree
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2OMe
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2OCFThree
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2SMe
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2S (O) Me
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2S (O)2Me
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2SCFThree
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2S (O) CFThree
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2S (O)2CFThree
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2CH (OMe)2
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2CH (SMe)2
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2C (O) Me
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2C (O) CFThree
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2C (O) OMe
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-32a)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-33a)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-34a)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-37a)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-81a)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-82a)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-84a)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-85a)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-87a)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-92a)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-93a)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-95a)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-96a)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-98a)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108a)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-Cl)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 3-Me)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 4-OMe)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-SMe)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 3-CFThree)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 4-OCFThree)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2(D1-108b, Z = 2-SCFThree)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2CH2CN
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2CH2CFThree
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2CH2OMe
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2CH2SMe
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2CH2S (O) Me
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} CH2CH2S (O)2Me
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} D1-32a
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} D1-33a
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} D1-34a
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} D1-37a
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} D1-81a
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} D1-82a
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} D1-84a
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} D1-85a
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} D1-87a
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} D1-92a
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} D1-93a
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} D1-95a
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} D1-96a
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} D1-98a
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} D1-108a
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-Cl)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} D1-108b (Z = 3-Me)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} D1-108b (Z = 4-OMe)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-SMe)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} D1-108b (Z = 3-CFThree)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} D1-108b (Z = 4-OCFThree)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} D1-108b (Z = 2-SCFThree)
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} C (O) Me
CH (Et) S (O)2{D1-32b (X1= 5-CFThree)} C (O) CFThree
CH2SCH2C≡CH Me
CH2SCH2C≡CH Et
CH2SCH2C≡CH Pr-n
CH2SCH2C≡CH Pr-i
CH2SCH2C≡CH Pr-c
CH2SCH2C≡CH Bu-n
CH2SCH2C≡CH Bu-i
CH2SCH2C≡CH Bu-c
CH2SCH2C≡CH Bu-s
CH2SCH2C≡CH Bu-t
CH2SCH2C≡CH Pen-n
CH2SCH2C≡CH Pen-c
CH2SCH2C≡CH Hex-n
CH2SCH2C≡CH Hex-c
CH2SCH2C≡CH CH2Pr-c
CH2SCH2C≡CH CH2Bu-c
CH2SCH2C≡CH CH2Pen-c
CH2SCH2C≡CH CH2Hex-c
CH2SCH2C≡CH CH2CH = CH2
CH2SCH2C≡CH CH2CH = C (Cl)2
CH2SCH2C≡CH CH2C≡CH
CH2SCH2C≡CH CH2CN
CH2SCH2C≡CH CH2CFThree
CH2SCH2C≡CH CH2OMe
CH2SCH2C≡CH CH2OCFThree
CH2SCH2C≡CH CH2SMe
CH2SCH2C≡CH CH2S (O) Me
CH2SCH2C≡CH CH2S (O)2Me
CH2SCH2C≡CH CH2SCFThree
CH2SCH2C≡CH CH2S (O) CFThree
CH2SCH2C≡CH CH2S (O)2CFThree
CH2SCH2C≡CH CH2CH (OMe)2
CH2SCH2C≡CH CH2CH (SMe)2
CH2SCH2C≡CH CH2C (O) Me
CH2SCH2C≡CH CH2C (O) CFThree
CH2SCH2C≡CH CH2C (O) OMe
CH2SCH2C≡CH CH2(D1-32a)
CH2SCH2C≡CH CH2(D1-33a)
CH2SCH2C≡CH CH2(D1-34a)
CH2SCH2C≡CH CH2(D1-37a)
CH2SCH2C≡CH CH2(D1-81a)
CH2SCH2C≡CH CH2(D1-82a)
CH2SCH2C≡CH CH2(D1-84a)
CH2SCH2C≡CH CH2(D1-85a)
CH2SCH2C≡CH CH2(D1-87a)
CH2SCH2C≡CH CH2(D1-92a)
CH2SCH2C≡CH CH2(D1-93a)
CH2SCH2C≡CH CH2(D1-95a)
CH2SCH2C≡CH CH2(D1-96a)
CH2SCH2C≡CH CH2(D1-98a)
CH2SCH2C≡CH CH2(D1-108a)
CH2SCH2C≡CH CH2(D1-108b, Z = 2-Cl)
CH2SCH2C≡CH CH2(D1-108b, Z = 3-Me)
CH2SCH2C≡CH CH2(D1-108b, Z = 4-OMe)
CH2SCH2C≡CH CH2(D1-108b, Z = 2-SMe)
CH2SCH2C≡CH CH2(D1-108b, Z = 3-CFThree)
CH2SCH2C≡CH CH2(D1-108b, Z = 4-OCFThree)
CH2SCH2C≡CH CH2(D1-108b, Z = 2-SCFThree)
CH2SCH2C≡CH CH2CH2CN
CH2SCH2C≡CH CH2CH2CFThree
CH2SCH2C≡CH CH2CH2OMe
CH2SCH2C≡CH CH2CH2SMe
CH2SCH2C≡CH CH2CH2S (O) Me
CH2SCH2C≡CH CH2CH2S (O)2Me
CH2SCH2C≡CH D1-32a
CH2SCH2C≡CH D1-33a
CH2SCH2C≡CH D1-34a
CH2SCH2C≡CH D1-37a
CH2SCH2C≡CH D1-81a
CH2SCH2C≡CH D1-82a
CH2SCH2C≡CH D1-84a
CH2SCH2C≡CH D1-85a
CH2SCH2C≡CH D1-87a
CH2SCH2C≡CH D1-92a
CH2SCH2C≡CH D1-93a
CH2SCH2C≡CH D1-95a
CH2SCH2C≡CH D1-96a
CH2SCH2C≡CH D1-98a
CH2SCH2C≡CH D1-108a
CH2SCH2C≡CH D1-108b (Z = 2-Cl)
CH2SCH2C≡CH D1-108b (Z = 3-Me)
CH2SCH2C≡CH D1-108b (Z = 4-OMe)
CH2SCH2C≡CH D1-108b (Z = 2-SMe)
CH2SCH2C≡CH D1-108b (Z = 3-CFThree)
CH2SCH2C≡CH D1-108b (Z = 4-OCFThree)
CH2SCH2C≡CH D1-108b (Z = 2-SCFThree)
CH2SCH2C≡CH C (O) Me
CH2SCH2C≡CH C (O) CFThree
CH2SCH2C≡CH C (O) OMe
CH2S (O) CH2C≡CH Me
CH2S (O) CH2C≡CH Et
CH2S (O) CH2C≡CH Pr-n
CH2S (O) CH2C≡CH Pr-i
CH2S (O) CH2C≡CH Pr-c
CH2S (O) CH2C≡CH Bu-n
CH2S (O) CH2C≡CH Bu-i
CH2S (O) CH2C≡CH Bu-c
CH2S (O) CH2C≡CH Bu-s
CH2S (O) CH2C≡CH Bu-t
CH2S (O) CH2C≡CH Pen-n
CH2S (O) CH2C≡CH Pen-c
CH2S (O) CH2C≡CH Hex-n
CH2S (O) CH2C≡CH Hex-c
CH2S (O) CH2C≡CH CH2Pr-c
CH2S (O) CH2C≡CH CH2Bu-c
CH2S (O) CH2C≡CH CH2Pen-c
CH2S (O) CH2C≡CH CH2Hex-c
CH2S (O) CH2C≡CH CH2CH = CH2
CH2S (O) CH2C≡CH CH2CH = C (Cl)2
CH2S (O) CH2C≡CH CH2C≡CH
CH2S (O) CH2C≡CH CH2CN
CH2S (O) CH2C≡CH CH2CFThree
CH2S (O) CH2C≡CH CH2OMe
CH2S (O) CH2C≡CH CH2OCFThree
CH2S (O) CH2C≡CH CH2SMe
CH2S (O) CH2C≡CH CH2S (O) Me
CH2S (O) CH2C≡CH CH2S (O)2Me
CH2S (O) CH2C≡CH CH2SCFThree
CH2S (O) CH2C≡CH CH2S (O) CFThree
CH2S (O) CH2C≡CH CH2S (O)2CFThree
CH2S (O) CH2C≡CH CH2CH (OMe)2
CH2S (O) CH2C≡CH CH2CH (SMe)2
CH2S (O) CH2C≡CH CH2C (O) Me
CH2S (O) CH2C≡CH CH2C (O) CFThree
CH2S (O) CH2C≡CH CH2C (O) OMe
CH2S (O) CH2C≡CH CH2(D1-32a)
CH2S (O) CH2C≡CH CH2(D1-33a)
CH2S (O) CH2C≡CH CH2(D1-34a)
CH2S (O) CH2C≡CH CH2(D1-37a)
CH2S (O) CH2C≡CH CH2(D1-81a)
CH2S (O) CH2C≡CH CH2(D1-82a)
CH2S (O) CH2C≡CH CH2(D1-84a)
CH2S (O) CH2C≡CH CH2(D1-85a)
CH2S (O) CH2C≡CH CH2(D1-87a)
CH2S (O) CH2C≡CH CH2(D1-92a)
CH2S (O) CH2C≡CH CH2(D1-93a)
CH2S (O) CH2C≡CH CH2(D1-95a)
CH2S (O) CH2C≡CH CH2(D1-96a)
CH2S (O) CH2C≡CH CH2(D1-98a)
CH2S (O) CH2C≡CH CH2(D1-108a)
CH2S (O) CH2C≡CH CH2(D1-108b, Z = 2-Cl)
CH2S (O) CH2C≡CH CH2(D1-108b, Z = 3-Me)
CH2S (O) CH2C≡CH CH2(D1-108b, Z = 4-OMe)
CH2S (O) CH2C≡CH CH2(D1-108b, Z = 2-SMe)
CH2S (O) CH2C≡CH CH2(D1-108b, Z = 3-CFThree)
CH2S (O) CH2C≡CH CH2(D1-108b, Z = 4-OCFThree)
CH2S (O) CH2C≡CH CH2(D1-108b, Z = 2-SCFThree)
CH2S (O) CH2C≡CH CH2CH2CN
CH2S (O) CH2C≡CH CH2CH2CFThree
CH2S (O) CH2C≡CH CH2CH2OMe
CH2S (O) CH2C≡CH CH2CH2SMe
CH2S (O) CH2C≡CH CH2CH2S (O) Me
CH2S (O) CH2C≡CH CH2CH2S (O)2Me
CH2S (O) CH2C≡CH D1-32a
CH2S (O) CH2C≡CH D1-33a
CH2S (O) CH2C≡CH D1-34a
CH2S (O) CH2C≡CH D1-37a
CH2S (O) CH2C≡CH D1-81a
CH2S (O) CH2C≡CH D1-82a
CH2S (O) CH2C≡CH D1-84a
CH2S (O) CH2C≡CH D1-85a
CH2S (O) CH2C≡CH D1-87a
CH2S (O) CH2C≡CH D1-92a
CH2S (O) CH2C≡CH D1-93a
CH2S (O) CH2C≡CH D1-95a
CH2S (O) CH2C≡CH D1-96a
CH2S (O) CH2C≡CH D1-98a
CH2S (O) CH2C≡CH D1-108a
CH2S (O) CH2C≡CH D1-108b (Z = 2-Cl)
CH2S (O) CH2C≡CH D1-108b (Z = 3-Me)
CH2S (O) CH2C≡CH D1-108b (Z = 4-OMe)
CH2S (O) CH2C≡CH D1-108b (Z = 2-SMe)
CH2S (O) CH2C≡CH D1-108b (Z = 3-CFThree)
CH2S (O) CH2C≡CH D1-108b (Z = 4-OCFThree)
CH2S (O) CH2C≡CH D1-108b (Z = 2-SCFThree)
CH2S (O) CH2C≡CH C (O) Me
CH2S (O) CH2C≡CH C (O) CFThree
CH2S (O) CH2C≡CH C (O) OMe
CH2S (O)2CH2C≡CH Me
CH2S (O)2CH2C≡CH Et
CH2S (O)2CH2C≡CH Pr-n
CH2S (O)2CH2C≡CH Pr-i
CH2S (O)2CH2C≡CH Pr-c
CH2S (O)2CH2C≡CH Bu-n
CH2S (O)2CH2C≡CH Bu-i
CH2S (O)2CH2C≡CH Bu-c
CH2S (O)2CH2C≡CH Bu-s
CH2S (O)2CH2C≡CH Bu-t
CH2S (O)2CH2C≡CH Pen-n
CH2S (O)2CH2C≡CH Pen-c
CH2S (O)2CH2C≡CH Hex-n
CH2S (O)2CH2C≡CH Hex-c
CH2S (O)2CH2C≡CH CH2Pr-c
CH2S (O)2CH2C≡CH CH2Bu-c
CH2S (O)2CH2C≡CH CH2Pen-c
CH2S (O)2CH2C≡CH CH2Hex-c
CH2S (O)2CH2C≡CH CH2CH = CH2
CH2S (O)2CH2C≡CH CH2CH = C (Cl)2
CH2S (O)2CH2C≡CH CH2C≡CH
CH2S (O)2CH2C≡CH CH2CN
CH2S (O)2CH2C≡CH CH2CFThree
CH2S (O)2CH2C≡CH CH2OMe
CH2S (O)2CH2C≡CH CH2OCFThree
CH2S (O)2CH2C≡CH CH2SMe
CH2S (O)2CH2C≡CH CH2S (O) Me
CH2S (O)2CH2C≡CH CH2S (O)2Me
CH2S (O)2CH2C≡CH CH2SCFThree
CH2S (O)2CH2C≡CH CH2S (O) CFThree
CH2S (O)2CH2C≡CH CH2S (O)2CFThree
CH2S (O)2CH2C≡CH CH2CH (OMe)2
CH2S (O)2CH2C≡CH CH2CH (SMe)2
CH2S (O)2CH2C≡CH CH2C (O) Me
CH2S (O)2CH2C≡CH CH2C (O) CFThree
CH2S (O)2CH2C≡CH CH2C (O) OMe
CH2S (O)2CH2C≡CH CH2(D1-32a)
CH2S (O)2CH2C≡CH CH2(D1-33a)
CH2S (O)2CH2C≡CH CH2(D1-34a)
CH2S (O)2CH2C≡CH CH2(D1-37a)
CH2S (O)2CH2C≡CH CH2(D1-81a)
CH2S (O)2CH2C≡CH CH2(D1-82a)
CH2S (O)2CH2C≡CH CH2(D1-84a)
CH2S (O)2CH2C≡CH CH2(D1-85a)
CH2S (O)2CH2C≡CH CH2(D1-87a)
CH2S (O)2CH2C≡CH CH2(D1-92a)
CH2S (O)2CH2C≡CH CH2(D1-93a)
CH2S (O)2CH2C≡CH CH2(D1-95a)
CH2S (O)2CH2C≡CH CH2(D1-96a)
CH2S (O)2CH2C≡CH CH2(D1-98a)
CH2S (O)2CH2C≡CH CH2(D1-108a)
CH2S (O)2CH2C≡CH CH2(D1-108b, Z = 2-Cl)
CH2S (O)2CH2C≡CH CH2(D1-108b, Z = 3-Me)
CH2S (O)2CH2C≡CH CH2(D1-108b, Z = 4-OMe)
CH2S (O)2CH2C≡CH CH2(D1-108b, Z = 2-SMe)
CH2S (O)2CH2C≡CH CH2(D1-108b, Z = 3-CFThree)
CH2S (O)2CH2C≡CH CH2(D1-108b, Z = 4-OCFThree)
CH2S (O)2CH2C≡CH CH2(D1-108b, Z = 2-SCFThree)
CH2S (O)2CH2C≡CH CH2CH2CN
CH2S (O)2CH2C≡CH CH2CH2CFThree
CH2S (O)2CH2C≡CH CH2CH2OMe
CH2S (O)2CH2C≡CH CH2CH2SMe
CH2S (O)2CH2C≡CH CH2CH2S (O) Me
CH2S (O)2CH2C≡CH CH2CH2S (O)2Me
CH2S (O)2CH2C≡CH D1-32a
CH2S (O)2CH2C≡CH D1-33a
CH2S (O)2CH2C≡CH D1-34a
CH2S (O)2CH2C≡CH D1-37a
CH2S (O)2CH2C≡CH D1-81a
CH2S (O)2CH2C≡CH D1-82a
CH2S (O)2CH2C≡CH D1-84a
CH2S (O)2CH2C≡CH D1-85a
CH2S (O)2CH2C≡CH D1-87a
CH2S (O)2CH2C≡CH D1-92a
CH2S (O)2CH2C≡CH D1-93a
CH2S (O)2CH2C≡CH D1-95a
CH2S (O)2CH2C≡CH D1-96a
CH2S (O)2CH2C≡CH D1-98a
CH2S (O)2CH2C≡CH D1-108a
CH2S (O)2CH2C≡CH D1-108b (Z = 2-Cl)
CH2S (O)2CH2C≡CH D1-108b (Z = 3-Me)
CH2S (O)2CH2C≡CH D1-108b (Z = 4-OMe)
CH2S (O)2CH2C≡CH D1-108b (Z = 2-SMe)
CH2S (O)2CH2C≡CH D1-108b (Z = 3-CFThree)
CH2S (O)2CH2C≡CH D1-108b (Z = 4-OCFThree)
CH2S (O)2CH2C≡CH D1-108b (Z = 2-SCFThree)
CH2S (O)2CH2C≡CH C (O) Me
CH2S (O)2CH2C≡CH C (O) CFThree
CH2S (O)2CH2C≡CH C (O) OMe
CH (Me) SCH2C≡CH Me
CH (Me) SCH2C≡CH Et
CH (Me) SCH2C≡CH Pr-n
CH (Me) SCH2C≡CH Pr-i
CH (Me) SCH2C≡CH Pr-c
CH (Me) SCH2C≡CH Bu-n
CH (Me) SCH2C≡CH Bu-i
CH (Me) SCH2C≡CH Bu-c
CH (Me) SCH2C≡CH Bu-s
CH (Me) SCH2C≡CH Bu-t
CH (Me) SCH2C≡CH Pen-n
CH (Me) SCH2C≡CH Pen-c
CH (Me) SCH2C≡CH Hex-n
CH (Me) SCH2C≡CH Hex-c
CH (Me) SCH2C≡CH CH2Pr-c
CH (Me) SCH2C≡CH CH2Bu-c
CH (Me) SCH2C≡CH CH2Pen-c
CH (Me) SCH2C≡CH CH2Hex-c
CH (Me) SCH2C≡CH CH2CH = CH2
CH (Me) SCH2C≡CH CH2CH = C (Cl)2
CH (Me) SCH2C≡CH CH2C≡CH
CH (Me) SCH2C≡CH CH2CN
CH (Me) SCH2C≡CH CH2CFThree
CH (Me) SCH2C≡CH CH2OMe
CH (Me) SCH2C≡CH CH2OCFThree
CH (Me) SCH2C≡CH CH2SMe
CH (Me) SCH2C≡CH CH2S (O) Me
CH (Me) SCH2C≡CH CH2S (O)2Me
CH (Me) SCH2C≡CH CH2SCFThree
CH (Me) SCH2C≡CH CH2S (O) CFThree
CH (Me) SCH2C≡CH CH2S (O)2CFThree
CH (Me) SCH2C≡CH CH2CH (OMe)2
CH (Me) SCH2C≡CH CH2CH (SMe)2
CH (Me) SCH2C≡CH CH2C (O) Me
CH (Me) SCH2C≡CH CH2C (O) CFThree
CH (Me) SCH2C≡CH CH2C (O) OMe
CH (Me) SCH2C≡CH CH2(D1-32a)
CH (Me) SCH2C≡CH CH2(D1-33a)
CH (Me) SCH2C≡CH CH2(D1-34a)
CH (Me) SCH2C≡CH CH2(D1-37a)
CH (Me) SCH2C≡CH CH2(D1-81a)
CH (Me) SCH2C≡CH CH2(D1-82a)
CH (Me) SCH2C≡CH CH2(D1-84a)
CH (Me) SCH2C≡CH CH2(D1-85a)
CH (Me) SCH2C≡CH CH2(D1-87a)
CH (Me) SCH2C≡CH CH2(D1-92a)
CH (Me) SCH2C≡CH CH2(D1-93a)
CH (Me) SCH2C≡CH CH2(D1-95a)
CH (Me) SCH2C≡CH CH2(D1-96a)
CH (Me) SCH2C≡CH CH2(D1-98a)
CH (Me) SCH2C≡CH CH2(D1-108a)
CH (Me) SCH2C≡CH CH2(D1-108b, Z = 2-Cl)
CH (Me) SCH2C≡CH CH2(D1-108b, Z = 3-Me)
CH (Me) SCH2C≡CH CH2(D1-108b, Z = 4-OMe)
CH (Me) SCH2C≡CH CH2(D1-108b, Z = 2-SMe)
CH (Me) SCH2C≡CH CH2(D1-108b, Z = 3-CFThree)
CH (Me) SCH2C≡CH CH2(D1-108b, Z = 4-OCFThree)
CH (Me) SCH2C≡CH CH2(D1-108b, Z = 2-SCFThree)
CH (Me) SCH2C≡CH CH2CH2CN
CH (Me) SCH2C≡CH CH2CH2CFThree
CH (Me) SCH2C≡CH CH2CH2OMe
CH (Me) SCH2C≡CH CH2CH2SMe
CH (Me) SCH2C≡CH CH2CH2S (O) Me
CH (Me) SCH2C≡CH CH2CH2S (O)2Me
CH (Me) SCH2C≡CH D1-32a
CH (Me) SCH2C≡CH D1-33a
CH (Me) SCH2C≡CH D1-34a
CH (Me) SCH2C≡CH D1-37a
CH (Me) SCH2C≡CH D1-81a
CH (Me) SCH2C≡CH D1-82a
CH (Me) SCH2C≡CH D1-84a
CH (Me) SCH2C≡CH D1-85a
CH (Me) SCH2C≡CH D1-87a
CH (Me) SCH2C≡CH D1-92a
CH (Me) SCH2C≡CH D1-93a
CH (Me) SCH2C≡CH D1-95a
CH (Me) SCH2C≡CH D1-96a
CH (Me) SCH2C≡CH D1-98a
CH (Me) SCH2C≡CH D1-108a
CH (Me) SCH2C≡CH D1-108b (Z = 2-Cl)
CH (Me) SCH2C≡CH D1-108b (Z = 3-Me)
CH (Me) SCH2C≡CH D1-108b (Z = 4-OMe)
CH (Me) SCH2C≡CH D1-108b (Z = 2-SMe)
CH (Me) SCH2C≡CH D1-108b (Z = 3-CFThree)
CH (Me) SCH2C≡CH D1-108b (Z = 4-OCFThree)
CH (Me) SCH2C≡CH D1-108b (Z = 2-SCFThree)
CH (Me) SCH2C≡CH C (O) Me
CH (Me) SCH2C≡CH C (O) CFThree
CH (Me) SCH2C≡CH C (O) OMe
CH (Me) S (O) CH2C≡CH Me
CH (Me) S (O) CH2C≡CH Et
CH (Me) S (O) CH2C≡CH Pr-n
CH (Me) S (O) CH2C≡CH Pr-i
CH (Me) S (O) CH2C≡CH Pr-c
CH (Me) S (O) CH2C≡CH Bu-n
CH (Me) S (O) CH2C≡CH Bu-i
CH (Me) S (O) CH2C≡CH Bu-c
CH (Me) S (O) CH2C≡CH Bu-s
CH (Me) S (O) CH2C≡CH Bu-t
CH (Me) S (O) CH2C≡CH Pen-n
CH (Me) S (O) CH2C≡CH Pen-c
CH (Me) S (O) CH2C≡CH Hex-n
CH (Me) S (O) CH2C≡CH Hex-c
CH (Me) S (O) CH2C≡CH CH2Pr-c
CH (Me) S (O) CH2C≡CH CH2Bu-c
CH (Me) S (O) CH2C≡CH CH2Pen-c
CH (Me) S (O) CH2C≡CH CH2Hex-c
CH (Me) S (O) CH2C≡CH CH2CH = CH2
CH (Me) S (O) CH2C≡CH CH2CH = C (Cl)2
CH (Me) S (O) CH2C≡CH CH2C≡CH
CH (Me) S (O) CH2C≡CH CH2CN
CH (Me) S (O) CH2C≡CH CH2CFThree
CH (Me) S (O) CH2C≡CH CH2OMe
CH (Me) S (O) CH2C≡CH CH2OCFThree
CH (Me) S (O) CH2C≡CH CH2SMe
CH (Me) S (O) CH2C≡CH CH2S (O) Me
CH (Me) S (O) CH2C≡CH CH2S (O)2Me
CH (Me) S (O) CH2C≡CH CH2SCFThree
CH (Me) S (O) CH2C≡CH CH2S (O) CFThree
CH (Me) S (O) CH2C≡CH CH2S (O)2CFThree
CH (Me) S (O) CH2C≡CH CH2CH (OMe)2
CH (Me) S (O) CH2C≡CH CH2CH (SMe)2
CH (Me) S (O) CH2C≡CH CH2C (O) Me
CH (Me) S (O) CH2C≡CH CH2C (O) CFThree
CH (Me) S (O) CH2C≡CH CH2C (O) OMe
CH (Me) S (O) CH2C≡CH CH2(D1-32a)
CH (Me) S (O) CH2C≡CH CH2(D1-33a)
CH (Me) S (O) CH2C≡CH CH2(D1-34a)
CH (Me) S (O) CH2C≡CH CH2(D1-37a)
CH (Me) S (O) CH2C≡CH CH2(D1-81a)
CH (Me) S (O) CH2C≡CH CH2(D1-82a)
CH (Me) S (O) CH2C≡CH CH2(D1-84a)
CH (Me) S (O) CH2C≡CH CH2(D1-85a)
CH (Me) S (O) CH2C≡CH CH2(D1-87a)
CH (Me) S (O) CH2C≡CH CH2(D1-92a)
CH (Me) S (O) CH2C≡CH CH2(D1-93a)
CH (Me) S (O) CH2C≡CH CH2(D1-95a)
CH (Me) S (O) CH2C≡CH CH2(D1-96a)
CH (Me) S (O) CH2C≡CH CH2(D1-98a)
CH (Me) S (O) CH2C≡CH CH2(D1-108a)
CH (Me) S (O) CH2C≡CH CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O) CH2C≡CH CH2(D1-108b, Z = 3-Me)
CH (Me) S (O) CH2C≡CH CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O) CH2C≡CH CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O) CH2C≡CH CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O) CH2C≡CH CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O) CH2C≡CH CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O) CH2C≡CH CH2CH2CN
CH (Me) S (O) CH2C≡CH CH2CH2CFThree
CH (Me) S (O) CH2C≡CH CH2CH2OMe
CH (Me) S (O) CH2C≡CH CH2CH2SMe
CH (Me) S (O) CH2C≡CH CH2CH2S (O) Me
CH (Me) S (O) CH2C≡CH CH2CH2S (O)2Me
CH (Me) S (O) CH2C≡CH D1-32a
CH (Me) S (O) CH2C≡CH D1-33a
CH (Me) S (O) CH2C≡CH D1-34a
CH (Me) S (O) CH2C≡CH D1-37a
CH (Me) S (O) CH2C≡CH D1-81a
CH (Me) S (O) CH2C≡CH D1-82a
CH (Me) S (O) CH2C≡CH D1-84a
CH (Me) S (O) CH2C≡CH D1-85a
CH (Me) S (O) CH2C≡CH D1-87a
CH (Me) S (O) CH2C≡CH D1-92a
CH (Me) S (O) CH2C≡CH D1-93a
CH (Me) S (O) CH2C≡CH D1-95a
CH (Me) S (O) CH2C≡CH D1-96a
CH (Me) S (O) CH2C≡CH D1-98a
CH (Me) S (O) CH2C≡CH D1-108a
CH (Me) S (O) CH2C≡CH D1-108b (Z = 2-Cl)
CH (Me) S (O) CH2C≡CH D1-108b (Z = 3-Me)
CH (Me) S (O) CH2C≡CH D1-108b (Z = 4-OMe)
CH (Me) S (O) CH2C≡CH D1-108b (Z = 2-SMe)
CH (Me) S (O) CH2C≡CH D1-108b (Z = 3-CFThree)
CH (Me) S (O) CH2C≡CH D1-108b (Z = 4-OCFThree)
CH (Me) S (O) CH2C≡CH D1-108b (Z = 2-SCFThree)
CH (Me) S (O) CH2C≡CH C (O) Me
CH (Me) S (O) CH2C≡CH C (O) CFThree
CH (Me) S (O) CH2C≡CH C (O) OMe
CH (Me) S (O)2CH2C≡CH Me
CH (Me) S (O)2CH2C≡CH Et
CH (Me) S (O)2CH2C≡CH Pr-n
CH (Me) S (O)2CH2C≡CH Pr-i
CH (Me) S (O)2CH2C≡CH Pr-c
CH (Me) S (O)2CH2C≡CH Bu-n
CH (Me) S (O)2CH2C≡CH Bu-i
CH (Me) S (O)2CH2C≡CH Bu-c
CH (Me) S (O)2CH2C≡CH Bu-s
CH (Me) S (O)2CH2C≡CH Bu-t
CH (Me) S (O)2CH2C≡CH Pen-n
CH (Me) S (O)2CH2C≡CH Pen-c
CH (Me) S (O)2CH2C≡CH Hex-n
CH (Me) S (O)2CH2C≡CH Hex-c
CH (Me) S (O)2CH2C≡CH CH2Pr-c
CH (Me) S (O)2CH2C≡CH CH2Bu-c
CH (Me) S (O)2CH2C≡CH CH2Pen-c
CH (Me) S (O)2CH2C≡CH CH2Hex-c
CH (Me) S (O)2CH2C≡CH CH2CH = CH2
CH (Me) S (O)2CH2C≡CH CH2CH = C (Cl)2
CH (Me) S (O)2CH2C≡CH CH2C≡CH
CH (Me) S (O)2CH2C≡CH CH2CN
CH (Me) S (O)2CH2C≡CH CH2CFThree
CH (Me) S (O)2CH2C≡CH CH2OMe
CH (Me) S (O)2CH2C≡CH CH2OCFThree
CH (Me) S (O)2CH2C≡CH CH2SMe
CH (Me) S (O)2CH2C≡CH CH2S (O) Me
CH (Me) S (O)2CH2C≡CH CH2S (O)2Me
CH (Me) S (O)2CH2C≡CH CH2SCFThree
CH (Me) S (O)2CH2C≡CH CH2S (O) CFThree
CH (Me) S (O)2CH2C≡CH CH2S (O)2CFThree
CH (Me) S (O)2CH2C≡CH CH2CH (OMe)2
CH (Me) S (O)2CH2C≡CH CH2CH (SMe)2
CH (Me) S (O)2CH2C≡CH CH2C (O) Me
CH (Me) S (O)2CH2C≡CH CH2C (O) CFThree
CH (Me) S (O)2CH2C≡CH CH2C (O) OMe
CH (Me) S (O)2CH2C≡CH CH2(D1-32a)
CH (Me) S (O)2CH2C≡CH CH2(D1-33a)
CH (Me) S (O)2CH2C≡CH CH2(D1-34a)
CH (Me) S (O)2CH2C≡CH CH2(D1-37a)
CH (Me) S (O)2CH2C≡CH CH2(D1-81a)
CH (Me) S (O)2CH2C≡CH CH2(D1-82a)
CH (Me) S (O)2CH2C≡CH CH2(D1-84a)
CH (Me) S (O)2CH2C≡CH CH2(D1-85a)
CH (Me) S (O)2CH2C≡CH CH2(D1-87a)
CH (Me) S (O)2CH2C≡CH CH2(D1-92a)
CH (Me) S (O)2CH2C≡CH CH2(D1-93a)
CH (Me) S (O)2CH2C≡CH CH2(D1-95a)
CH (Me) S (O)2CH2C≡CH CH2(D1-96a)
CH (Me) S (O)2CH2C≡CH CH2(D1-98a)
CH (Me) S (O)2CH2C≡CH CH2(D1-108a)
CH (Me) S (O)2CH2C≡CH CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O)2CH2C≡CH CH2(D1-108b, Z = 3-Me)
CH (Me) S (O)2CH2C≡CH CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O)2CH2C≡CH CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O)2CH2C≡CH CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O)2CH2C≡CH CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O)2CH2C≡CH CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O)2CH2C≡CH CH2CH2CN
CH (Me) S (O)2CH2C≡CH CH2CH2CFThree
CH (Me) S (O)2CH2C≡CH CH2CH2OMe
CH (Me) S (O)2CH2C≡CH CH2CH2SMe
CH (Me) S (O)2CH2C≡CH CH2CH2S (O) Me
CH (Me) S (O)2CH2C≡CH CH2CH2S (O)2Me
CH (Me) S (O)2CH2C≡CH D1-32a
CH (Me) S (O)2CH2C≡CH D1-33a
CH (Me) S (O)2CH2C≡CH D1-34a
CH (Me) S (O)2CH2C≡CH D1-37a
CH (Me) S (O)2CH2C≡CH D1-81a
CH (Me) S (O)2CH2C≡CH D1-82a
CH (Me) S (O)2CH2C≡CH D1-84a
CH (Me) S (O)2CH2C≡CH D1-85a
CH (Me) S (O)2CH2C≡CH D1-87a
CH (Me) S (O)2CH2C≡CH D1-92a
CH (Me) S (O)2CH2C≡CH D1-93a
CH (Me) S (O)2CH2C≡CH D1-95a
CH (Me) S (O)2CH2C≡CH D1-96a
CH (Me) S (O)2CH2C≡CH D1-98a
CH (Me) S (O)2CH2C≡CH D1-108a
CH (Me) S (O)2CH2C≡CH D1-108b (Z = 2-Cl)
CH (Me) S (O)2CH2C≡CH D1-108b (Z = 3-Me)
CH (Me) S (O)2CH2C≡CH D1-108b (Z = 4-OMe)
CH (Me) S (O)2CH2C≡CH D1-108b (Z = 2-SMe)
CH (Me) S (O)2CH2C≡CH D1-108b (Z = 3-CFThree)
CH (Me) S (O)2CH2C≡CH D1-108b (Z = 4-OCFThree)
CH (Me) S (O)2CH2C≡CH D1-108b (Z = 2-SCFThree)
CH (Me) S (O)2CH2C≡CH C (O) Me
CH (Me) S (O)2CH2C≡CH C (O) CFThree
CH (Me) S (O)2CH2C≡CH C (O) OMe
CH (Et) SCH2C≡CH Me
CH (Et) SCH2C≡CH Et
CH (Et) SCH2C≡CH Pr-n
CH (Et) SCH2C≡CH Pr-i
CH (Et) SCH2C≡CH Pr-c
CH (Et) SCH2C≡CH Bu-n
CH (Et) SCH2C≡CH Bu-i
CH (Et) SCH2C≡CH Bu-c
CH (Et) SCH2C≡CH Bu-s
CH (Et) SCH2C≡CH Bu-t
CH (Et) SCH2C≡CH Pen-n
CH (Et) SCH2C≡CH Pen-c
CH (Et) SCH2C≡CH Hex-n
CH (Et) SCH2C≡CH Hex-c
CH (Et) SCH2C≡CH CH2Pr-c
CH (Et) SCH2C≡CH CH2Bu-c
CH (Et) SCH2C≡CH CH2Pen-c
CH (Et) SCH2C≡CH CH2Hex-c
CH (Et) SCH2C≡CH CH2CH = CH2
CH (Et) SCH2C≡CH CH2CH = C (Cl)2
CH (Et) SCH2C≡CH CH2C≡CH
CH (Et) SCH2C≡CH CH2CN
CH (Et) SCH2C≡CH CH2CFThree
CH (Et) SCH2C≡CH CH2OMe
CH (Et) SCH2C≡CH CH2OCFThree
CH (Et) SCH2C≡CH CH2SMe
CH (Et) SCH2C≡CH CH2S (O) Me
CH (Et) SCH2C≡CH CH2S (O)2Me
CH (Et) SCH2C≡CH CH2SCFThree
CH (Et) SCH2C≡CH CH2S (O) CFThree
CH (Et) SCH2C≡CH CH2S (O)2CFThree
CH (Et) SCH2C≡CH CH2CH (OMe)2
CH (Et) SCH2C≡CH CH2CH (SMe)2
CH (Et) SCH2C≡CH CH2C (O) Me
CH (Et) SCH2C≡CH CH2C (O) CFThree
CH (Et) SCH2C≡CH CH2C (O) OMe
CH (Et) SCH2C≡CH CH2(D1-32a)
CH (Et) SCH2C≡CH CH2(D1-33a)
CH (Et) SCH2C≡CH CH2(D1-34a)
CH (Et) SCH2C≡CH CH2(D1-37a)
CH (Et) SCH2C≡CH CH2(D1-81a)
CH (Et) SCH2C≡CH CH2(D1-82a)
CH (Et) SCH2C≡CH CH2(D1-84a)
CH (Et) SCH2C≡CH CH2(D1-85a)
CH (Et) SCH2C≡CH CH2(D1-87a)
CH (Et) SCH2C≡CH CH2(D1-92a)
CH (Et) SCH2C≡CH CH2(D1-93a)
CH (Et) SCH2C≡CH CH2(D1-95a)
CH (Et) SCH2C≡CH CH2(D1-96a)
CH (Et) SCH2C≡CH CH2(D1-98a)
CH (Et) SCH2C≡CH CH2(D1-108a)
CH (Et) SCH2C≡CH CH2(D1-108b, Z = 2-Cl)
CH (Et) SCH2C≡CH CH2(D1-108b, Z = 3-Me)
CH (Et) SCH2C≡CH CH2(D1-108b, Z = 4-OMe)
CH (Et) SCH2C≡CH CH2(D1-108b, Z = 2-SMe)
CH (Et) SCH2C≡CH CH2(D1-108b, Z = 3-CFThree)
CH (Et) SCH2C≡CH CH2(D1-108b, Z = 4-OCFThree)
CH (Et) SCH2C≡CH CH2(D1-108b, Z = 2-SCFThree)
CH (Et) SCH2C≡CH CH2CH2CN
CH (Et) SCH2C≡CH CH2CH2CFThree
CH (Et) SCH2C≡CH CH2CH2OMe
CH (Et) SCH2C≡CH CH2CH2SMe
CH (Et) SCH2C≡CH CH2CH2S (O) Me
CH (Et) SCH2C≡CH CH2CH2S (O)2Me
CH (Et) SCH2C≡CH D1-32a
CH (Et) SCH2C≡CH D1-33a
CH (Et) SCH2C≡CH D1-34a
CH (Et) SCH2C≡CH D1-37a
CH (Et) SCH2C≡CH D1-81a
CH (Et) SCH2C≡CH D1-82a
CH (Et) SCH2C≡CH D1-84a
CH (Et) SCH2C≡CH D1-85a
CH (Et) SCH2C≡CH D1-87a
CH (Et) SCH2C≡CH D1-92a
CH (Et) SCH2C≡CH D1-93a
CH (Et) SCH2C≡CH D1-95a
CH (Et) SCH2C≡CH D1-96a
CH (Et) SCH2C≡CH D1-98a
CH (Et) SCH2C≡CH D1-108a
CH (Et) SCH2C≡CH D1-108b (Z = 2-Cl)
CH (Et) SCH2C≡CH D1-108b (Z = 3-Me)
CH (Et) SCH2C≡CH D1-108b (Z = 4-OMe)
CH (Et) SCH2C≡CH D1-108b (Z = 2-SMe)
CH (Et) SCH2C≡CH D1-108b (Z = 3-CFThree)
CH (Et) SCH2C≡CH D1-108b (Z = 4-OCFThree)
CH (Et) SCH2C≡CH D1-108b (Z = 2-SCFThree)
CH (Et) SCH2C≡CH C (O) Me
CH (Et) SCH2C≡CH C (O) CFThree
CH (Et) SCH2C≡CH C (O) OMe
CH (Et) S (O) CH2C≡CH Me
CH (Et) S (O) CH2C≡CH Et
CH (Et) S (O) CH2C≡CH Pr-n
CH (Et) S (O) CH2C≡CH Pr-i
CH (Et) S (O) CH2C≡CH Pr-c
CH (Et) S (O) CH2C≡CH Bu-n
CH (Et) S (O) CH2C≡CH Bu-i
CH (Et) S (O) CH2C≡CH Bu-c
CH (Et) S (O) CH2C≡CH Bu-s
CH (Et) S (O) CH2C≡CH Bu-t
CH (Et) S (O) CH2C≡CH Pen-n
CH (Et) S (O) CH2C≡CH Pen-c
CH (Et) S (O) CH2C≡CH Hex-n
CH (Et) S (O) CH2C≡CH Hex-c
CH (Et) S (O) CH2C≡CH CH2Pr-c
CH (Et) S (O) CH2C≡CH CH2Bu-c
CH (Et) S (O) CH2C≡CH CH2Pen-c
CH (Et) S (O) CH2C≡CH CH2Hex-c
CH (Et) S (O) CH2C≡CH CH2CH = CH2
CH (Et) S (O) CH2C≡CH CH2CH = C (Cl)2
CH (Et) S (O) CH2C≡CH CH2C≡CH
CH (Et) S (O) CH2C≡CH CH2CN
CH (Et) S (O) CH2C≡CH CH2CFThree
CH (Et) S (O) CH2C≡CH CH2OMe
CH (Et) S (O) CH2C≡CH CH2OCFThree
CH (Et) S (O) CH2C≡CH CH2SMe
CH (Et) S (O) CH2C≡CH CH2S (O) Me
CH (Et) S (O) CH2C≡CH CH2S (O)2Me
CH (Et) S (O) CH2C≡CH CH2SCFThree
CH (Et) S (O) CH2C≡CH CH2S (O) CFThree
CH (Et) S (O) CH2C≡CH CH2S (O)2CFThree
CH (Et) S (O) CH2C≡CH CH2CH (OMe)2
CH (Et) S (O) CH2C≡CH CH2CH (SMe)2
CH (Et) S (O) CH2C≡CH CH2C (O) Me
CH (Et) S (O) CH2C≡CH CH2C (O) CFThree
CH (Et) S (O) CH2C≡CH CH2C (O) OMe
CH (Et) S (O) CH2C≡CH CH2(D1-32a)
CH (Et) S (O) CH2C≡CH CH2(D1-33a)
CH (Et) S (O) CH2C≡CH CH2(D1-34a)
CH (Et) S (O) CH2C≡CH CH2(D1-37a)
CH (Et) S (O) CH2C≡CH CH2(D1-81a)
CH (Et) S (O) CH2C≡CH CH2(D1-82a)
CH (Et) S (O) CH2C≡CH CH2(D1-84a)
CH (Et) S (O) CH2C≡CH CH2(D1-85a)
CH (Et) S (O) CH2C≡CH CH2(D1-87a)
CH (Et) S (O) CH2C≡CH CH2(D1-92a)
CH (Et) S (O) CH2C≡CH CH2(D1-93a)
CH (Et) S (O) CH2C≡CH CH2(D1-95a)
CH (Et) S (O) CH2C≡CH CH2(D1-96a)
CH (Et) S (O) CH2C≡CH CH2(D1-98a)
CH (Et) S (O) CH2C≡CH CH2(D1-108a)
CH (Et) S (O) CH2C≡CH CH2(D1-108b, Z = 2-Cl)
CH (Et) S (O) CH2C≡CH CH2(D1-108b, Z = 3-Me)
CH (Et) S (O) CH2C≡CH CH2(D1-108b, Z = 4-OMe)
CH (Et) S (O) CH2C≡CH CH2(D1-108b, Z = 2-SMe)
CH (Et) S (O) CH2C≡CH CH2(D1-108b, Z = 3-CFThree)
CH (Et) S (O) CH2C≡CH CH2(D1-108b, Z = 4-OCFThree)
CH (Et) S (O) CH2C≡CH CH2(D1-108b, Z = 2-SCFThree)
CH (Et) S (O) CH2C≡CH CH2CH2CN
CH (Et) S (O) CH2C≡CH CH2CH2CFThree
CH (Et) S (O) CH2C≡CH CH2CH2OMe
CH (Et) S (O) CH2C≡CH CH2CH2SMe
CH (Et) S (O) CH2C≡CH CH2CH2S (O) Me
CH (Et) S (O) CH2C≡CH CH2CH2S (O)2Me
CH (Et) S (O) CH2C≡CH D1-32a
CH (Et) S (O) CH2C≡CH D1-33a
CH (Et) S (O) CH2C≡CH D1-34a
CH (Et) S (O) CH2C≡CH D1-37a
CH (Et) S (O) CH2C≡CH D1-81a
CH (Et) S (O) CH2C≡CH D1-82a
CH (Et) S (O) CH2C≡CH D1-84a
CH (Et) S (O) CH2C≡CH D1-85a
CH (Et) S (O) CH2C≡CH D1-87a
CH (Et) S (O) CH2C≡CH D1-92a
CH (Et) S (O) CH2C≡CH D1-93a
CH (Et) S (O) CH2C≡CH D1-95a
CH (Et) S (O) CH2C≡CH D1-96a
CH (Et) S (O) CH2C≡CH D1-98a
CH (Et) S (O) CH2C≡CH D1-108a
CH (Et) S (O) CH2C≡CH D1-108b (Z = 2-Cl)
CH (Et) S (O) CH2C≡CH D1-108b (Z = 3-Me)
CH (Et) S (O) CH2C≡CH D1-108b (Z = 4-OMe)
CH (Et) S (O) CH2C≡CH D1-108b (Z = 2-SMe)
CH (Et) S (O) CH2C≡CH D1-108b (Z = 3-CFThree)
CH (Et) S (O) CH2C≡CH D1-108b (Z = 4-OCFThree)
CH (Et) S (O) CH2C≡CH D1-108b (Z = 2-SCFThree)
CH (Et) S (O) CH2C≡CH C (O) Me
CH (Et) S (O) CH2C≡CH C (O) CFThree
CH (Et) S (O) CH2C≡CH C (O) OMe
CH (Et) S (O)2CH2C≡CH Me
CH (Et) S (O)2CH2C≡CH Et
CH (Et) S (O)2CH2C≡CH Pr-n
CH (Et) S (O)2CH2C≡CH Pr-i
CH (Et) S (O)2CH2C≡CH Pr-c
CH (Et) S (O)2CH2C≡CH Bu-n
CH (Et) S (O)2CH2C≡CH Bu-i
CH (Et) S (O)2CH2C≡CH Bu-c
CH (Et) S (O)2CH2C≡CH Bu-s
CH (Et) S (O)2CH2C≡CH Bu-t
CH (Et) S (O)2CH2C≡CH Pen-n
CH (Et) S (O)2CH2C≡CH Pen-c
CH (Et) S (O)2CH2C≡CH Hex-n
CH (Et) S (O)2CH2C≡CH Hex-c
CH (Et) S (O)2CH2C≡CH CH2Pr-c
CH (Et) S (O)2CH2C≡CH CH2Bu-c
CH (Et) S (O)2CH2C≡CH CH2Pen-c
CH (Et) S (O)2CH2C≡CH CH2Hex-c
CH (Et) S (O)2CH2C≡CH CH2CH = CH2
CH (Et) S (O)2CH2C≡CH CH2CH = C (Cl)2
CH (Et) S (O)2CH2C≡CH CH2C≡CH
CH (Et) S (O)2CH2C≡CH CH2CN
CH (Et) S (O)2CH2C≡CH CH2CFThree
CH (Et) S (O)2CH2C≡CH CH2OMe
CH (Et) S (O)2CH2C≡CH CH2OCFThree
CH (Et) S (O)2CH2C≡CH CH2SMe
CH (Et) S (O)2CH2C≡CH CH2S (O) Me
CH (Et) S (O)2CH2C≡CH CH2S (O)2Me
CH (Et) S (O)2CH2C≡CH CH2SCFThree
CH (Et) S (O)2CH2C≡CH CH2S (O) CFThree
CH (Et) S (O)2CH2C≡CH CH2S (O)2CFThree
CH (Et) S (O)2CH2C≡CH CH2CH (OMe)2
CH (Et) S (O)2CH2C≡CH CH2CH (SMe)2
CH (Et) S (O)2CH2C≡CH CH2C (O) Me
CH (Et) S (O)2CH2C≡CH CH2C (O) CFThree
CH (Et) S (O)2CH2C≡CH CH2C (O) OMe
CH (Et) S (O)2CH2C≡CH CH2(D1-32a)
CH (Et) S (O)2CH2C≡CH CH2(D1-33a)
CH (Et) S (O)2CH2C≡CH CH2(D1-34a)
CH (Et) S (O)2CH2C≡CH CH2(D1-37a)
CH (Et) S (O)2CH2C≡CH CH2(D1-81a)
CH (Et) S (O)2CH2C≡CH CH2(D1-82a)
CH (Et) S (O)2CH2C≡CH CH2(D1-84a)
CH (Et) S (O)2CH2C≡CH CH2(D1-85a)
CH (Et) S (O)2CH2C≡CH CH2(D1-87a)
CH (Et) S (O)2CH2C≡CH CH2(D1-92a)
CH (Et) S (O)2CH2C≡CH CH2(D1-93a)
CH (Et) S (O)2CH2C≡CH CH2(D1-95a)
CH (Et) S (O)2CH2C≡CH CH2(D1-96a)
CH (Et) S (O)2CH2C≡CH CH2(D1-98a)
CH (Et) S (O)2CH2C≡CH CH2(D1-108a)
CH (Et) S (O)2CH2C≡CH CH2(D1-108b, Z = 2-Cl)
CH (Et) S (O)2CH2C≡CH CH2(D1-108b, Z = 3-Me)
CH (Et) S (O)2CH2C≡CH CH2(D1-108b, Z = 4-OMe)
CH (Et) S (O)2CH2C≡CH CH2(D1-108b, Z = 2-SMe)
CH (Et) S (O)2CH2C≡CH CH2(D1-108b, Z = 3-CFThree)
CH (Et) S (O)2CH2C≡CH CH2(D1-108b, Z = 4-OCFThree)
CH (Et) S (O)2CH2C≡CH CH2(D1-108b, Z = 2-SCFThree)
CH (Et) S (O)2CH2C≡CH CH2CH2CN
CH (Et) S (O)2CH2C≡CH CH2CH2CFThree
CH (Et) S (O)2CH2C≡CH CH2CH2OMe
CH (Et) S (O)2CH2C≡CH CH2CH2SMe
CH (Et) S (O)2CH2C≡CH CH2CH2S (O) Me
CH (Et) S (O)2CH2C≡CH CH2CH2S (O)2Me
CH (Et) S (O)2CH2C≡CH D1-32a
CH (Et) S (O)2CH2C≡CH D1-33a
CH (Et) S (O)2CH2C≡CH D1-34a
CH (Et) S (O)2CH2C≡CH D1-37a
CH (Et) S (O)2CH2C≡CH D1-81a
CH (Et) S (O)2CH2C≡CH D1-82a
CH (Et) S (O)2CH2C≡CH D1-84a
CH (Et) S (O)2CH2C≡CH D1-85a
CH (Et) S (O)2CH2C≡CH D1-87a
CH (Et) S (O)2CH2C≡CH D1-92a
CH (Et) S (O)2CH2C≡CH D1-93a
CH (Et) S (O)2CH2C≡CH D1-95a
CH (Et) S (O)2CH2C≡CH D1-96a
CH (Et) S (O)2CH2C≡CH D1-98a
CH (Et) S (O)2CH2C≡CH D1-108a
CH (Et) S (O)2CH2C≡CH D1-108b (Z = 2-Cl)
CH (Et) S (O)2CH2C≡CH D1-108b (Z = 3-Me)
CH (Et) S (O)2CH2C≡CH D1-108b (Z = 4-OMe)
CH (Et) S (O)2CH2C≡CH D1-108b (Z = 2-SMe)
CH (Et) S (O)2CH2C≡CH D1-108b (Z = 3-CFThree)
CH (Et) S (O)2CH2C≡CH D1-108b (Z = 4-OCFThree)
CH (Et) S (O)2CH2C≡CH D1-108b (Z = 2-SCFThree)
CH (Et) S (O)2CH2C≡CH C (O) Me
CH (Et) S (O)2CH2C≡CH C (O) CFThree
CH (Et) S (O)2CH2C≡CH C (O) OMe
Me Me
Et Me
Pr-n Me
Pr-i Me
Bu-n Me
Bu-i Me
Bu-t Me
Pen-n Me
Hex-n Me
CH (Et) Cl Me
CH2{D1-7b (3-CFThree)} Me
CH (CN) Ph Me
SMe Me
SEt Me
SPr-n Me
SPr-i Me
SBu-n Me
SBu-i Me
SBu-t Me
SPen-n Me
SHex-n Me
SPr-c Me
SBu-c Me
SPen-c Me
SHex-c Me
SCH2CH = CH2                            Me
SCH2C Three CH Me
SCF2H Me
SCFThree                                 Me
SCF2Cl Me
SCH2CFThree                              Me
S (D1-108c) Me
CH2OH Me
CH2OMe Me
CH2OEt Me
CH2OPr-n Me
CH2OPr-i Me
CH2OBu-n Me
CH2OBu-i Me
CH2OBu-s Me
CH2OBu-t Me
CH2OPen-n Me
CH2OHex-n Me
CH2O (D1-104c) Me
CH (Me) OH Me
CH (Me) OMe Me
CH (Me) OEt Me
CH (Me) OPr-n Me
CH (Me) OPr-i Me
CH (Me) OBu-n Me
CH (Me) OBu-i Me
CH (Me) OBu-s Me
CH (Me) OBu-t Me
CH (Me) OPen-n Me
CH (Me) OHex-n Me
CH (Me) O (D1-104c) Me
CH (Et) OH Me
CH (Et) OMe Me
CH (Et) OEt Me
CH (Et) OPr-n Me
CH (Et) OPr-i Me
CH (Et) OBu-n Me
CH (Et) OBu-i Me
CH (Et) OBu-s Me
CH (Et) OBu-t Me
CH (Et) OPen-n Me
CH (Et) OHex-n Me
CH (Et) O (D1-104c) Me
CH (n-Pr) OH Me
CH (n-Pr) OMe Me
CH (n-Pr) OEt Me
CH (n-Pr) O (D1-104c) Me
CH (i-Pr) OH Me
CH (i-Pr) OMe Me
CH (i-Pr) OEt Me
CH (i-Pr) O (D1-104c) Me
CH (n-Bu) OH Me
CH (n-Bu) OMe Me
CH (n-Bu) OEt Me
CH (n-Bu) O (D1-104c) Me
C (Me)2OH Me
C (Me)2OMe Me
C (Me)2OEt Me
C (Me)2O (D1-104c) Me
CH2CH2OH Me
CH2CH2OMe Me
CH2CH2OEt Me
CH2CH2O (D1-104c) Me
CH (Me) CH2OH Me
CH (Me) CH2OMe Me
CH (Me) CH2OEt Me
CH (Me) CH2O (D1-104c) Me
CH (Et) CH2OH Me
CH (Et) CH2OMe Me
CH (Et) CH2OEt Me
CH (Et) CH2O (D1-104c) Me
CH (n-Pr) CH2OH Me
CH (n-Pr) CH2OMe Me
CH (n-Pr) CH2OEt Me
CH (n-Pr) CH2O (D1-104c) Me
CH (i-Pr) CH2OH Me
CH (i-Pr) CH2OMe Me
CH (i-Pr) CH2OEt Me
CH (i-Pr) CH2O (D1-104c) Me
CH (n-Bu) CH2OH Me
CH (n-Bu) CH2OMe Me
CH (n-Bu) CH2OEt Me
CH (n-Bu) CH2O (D1-104c) Me
C (Me)2CH2OH Me
C (Me)2CH2OMe Me
C (Me)2CH2OEt Me
C (Me)2CH2O (D1-104c) Me
CH2SH Me
CH2SMe Me
CH2SEt Me
CH2SPr-n Me
CH2SPr-i Me
CH2SBu-n Me
CH2SBu-i Me
CH2SBu-t Me
CH2SPen-n Me
CH2SHex-n Me
CH2SPr-c Me
CH2SBu-c Me
CH2SPen-c Me
CH2SHex-c Me
CH2SCH2CH = CH2                         Me
CH2SCH2C Three CH Me
CH2SCF2H Me
CH2SCFThree                               Me
CH2SCF2Cl Me
CH2SCH2CFThree                            Me
CH2S {D1-108c} Me
CH2S (O) Me Me
CH2S (O) Et Me
CH2S (O) Pr-n Me
CH2S (O) Pr-i Me
CH2S (O) Bu-n Me
CH2S (O) Bu-i Me
CH2S (O) Bu-t Me
CH2S (O) Pen-n Me
CH2S (O) Hex-n Me
CH2S (O) Pr-c Me
CH2S (O) Bu-c Me
CH2S (O) Pen-c Me
CH2S (O) Hex-c Me
CH2S (O) CH2CH = CH2                      Me
CH2S (O) CH2C Three CH Me
CH2S (O) CF2H Me
CH2S (O) CFThree                            Me
CH2S (O) CF2Cl Me
CH2S (O) CH2CFThree                         Me
CH2S (O) {D1-108c} Me
CH2S (O)2Me Me
CH2S (O)2Et Me
CH2S (O)2Pr-n Me
CH2S (O)2Pr-i Me
CH2S (O)2Bu-n Me
CH2S (O)2Bu-i Me
CH2S (O)2Bu-t Me
CH2S (O)2Pen-n Me
CH2S (O)2Hex-n Me
CH2S (O)2Pr-c Me
CH2S (O)2Bu-c Me
CH2S (O)2Pen-c Me
CH2S (O)2Hex-c Me
CH2S (O)2CH2CH = CH2                      Me
CH2S (O)2CH2C Three CH Me
CH2S (O)2CF2H Me
CH2S (O)2CFThree                           Me
CH2S (O)2CF2Cl Me
CH2S (O)2CH2CFThree                         Me
CH2S (O)2{D1-108c} Me
CH (Me) SH Me
CH (Me) SMe Me
CH (Me) SEt Me
CH (Me) SPr-n Me
CH (Me) SPr-i Me
CH (Me) SBu-n Me
CH (Me) SBu-i Me
CH (Me) SBu-t Me
CH (Me) SPen-n Me
CH (Me) SHex-n Me
CH (Me) SPr-c Me
CH (Me) SBu-c Me
CH (Me) SPen-c Me
CH (Me) SHex-c Me
CH (Me) SCH2CH = CH2                      Me
CH (Me) SCH2C Three CH Me
CH (Me) SCF2H Me
CH (Me) SCFThree                            Me
CH (Me) SCF2Cl Me
CH (Me) SCH2CFThree                          Me
CH (Me) S {D1-108c} Me
CH (Me) S (O) Me Me
CH (Me) S (O) Et Me
CH (Me) S (O) Pr-n Me
CH (Me) S (O) Pr-i Me
CH (Me) S (O) Bu-n Me
CH (Me) S (O) Bu-i Me
CH (Me) S (O) Bu-t Me
CH (Me) S (O) Pen-n Me
CH (Me) S (O) Hex-n Me
CH (Me) S (O) Pr-c Me
CH (Me) S (O) Bu-c Me
CH (Me) S (O) Pen-c Me
CH (Me) S (O) Hex-c Me
CH (Me) S (O) CH2CH = CH2                    Me
CH (Me) S (O) CH2C Three CH Me
CH (Me) S (O) CF2H Me
CH (Me) S (O) CFThree                         Me
CH (Me) S (O) CF2Cl Me
CH (Me) S (O) CH2CFThree                      Me
CH (Me) S (O) {D1-108c} Me
CH (Me) S (O)2Me Me
CH (Me) S (O)2Et Me
CH (Me) S (O)2Pr-n Me
CH (Me) S (O)2Pr-i Me
CH (Me) S (O)2Bu-n Me
CH (Me) S (O)2Bu-i Me
CH (Me) S (O)2Bu-t Me
CH (Me) S (O)2Pen-n Me
CH (Me) S (O)2Hex-n Me
CH (Me) S (O)2Pr-c Me
CH (Me) S (O)2Bu-c Me
CH (Me) S (O)2Pen-c Me
CH (Me) S (O)2Hex-c Me
CH (Me) S (O)2CH2CH = CH2                   Me
CH (Me) S (O)2CH2C Three CH Me
CH (Me) S (O)2CF2H Me
CH (Me) S (O)2CFThree                        Me
CH (Me) S (O)2CF2Cl Me
CH (Me) S (O)2CH2CFThree                      Me
CH (Me) S (O)2{D1-108c} Me
CH (Et) SH Me
CH (Et) SMe Me
CH (Et) SEt Me
CH (Et) SPr-n Me
CH (Et) SPr-i Me
CH (Et) SBu-n Me
CH (Et) SBu-i Me
CH (Et) SBu-t Me
CH (Et) SPen-n Me
CH (Et) SHex-n Me
CH (Et) SPr-c Me
CH (Et) SBu-c Me
CH (Et) SPen-c Me
CH (Et) SHex-c Me
CH (Et) SCH2CH = CH2                      Me
CH (Et) SCH2C Three CH Me
CH (Et) SCF2H Me
CH (Et) SCFThree                            Me
CH (Et) SCF2Cl Me
CH (Et) SCH2CFThree                          Me
CH (Et) S {D1-108c} Me
CH (Et) S (O) Me Me
CH (Et) S (O) Et Me
CH (Et) S (O) Pr-n Me
CH (Et) S (O) Pr-i Me
CH (Et) S (O) Bu-n Me
CH (Et) S (O) Bu-i Me
CH (Et) S (O) Bu-t Me
CH (Et) S (O) Pen-n Me
CH (Et) S (O) Hex-n Me
CH (Et) S (O) Pr-c Me
CH (Et) S (O) Bu-c Me
CH (Et) S (O) Pen-c Me
CH (Et) S (O) Hex-c Me
CH (Et) S (O) CH2CH = CH2                    Me
CH (Et) S (O) CH2C Three CH Me
CH (Et) S (O) CF2H Me
CH (Et) S (O) CFThree                         Me
CH (Et) S (O) CF2Cl Me
CH (Et) S (O) CH2CFThree                      Me
CH (Et) S (O) {D1-108c} Me
CH (Et) S (O)2Me Me
CH (Et) S (O)2Et Me
CH (Et) S (O)2Pr-n Me
CH (Et) S (O)2Pr-i Me
CH (Et) S (O)2Bu-n Me
CH (Et) S (O)2Bu-i Me
CH (Et) S (O)2Bu-t Me
CH (Et) S (O)2Pen-n Me
CH (Et) S (O)2Hex-n Me
CH (Et) S (O)2Pr-c Me
CH (Et) S (O)2Bu-c Me
CH (Et) S (O)2Pen-c Me
CH (Et) S (O)2Hex-c Me
CH (Et) S (O)2CH2CH = CH2                   Me
CH (Et) S (O)2CH2C Three CH Me
CH (Et) S (O)2CF2H Me
CH (Et) S (O)2CFThree                        Me
CH (Et) S (O)2CF2Cl Me
CH (Et) S (O)2CH2CFThree                      Me
CH (Et) S (O)2{D1-108c} Me
CH (n-Pr) SH Me
CH (n-Pr) SMe Me
CH (n-Pr) SEt Me
CH (n-Pr) SPr-n Me
CH (n-Pr) SPr-i Me
CH (n-Pr) SBu-n Me
CH (n-Pr) SBu-i Me
CH (n-Pr) SBu-t Me
CH (n-Pr) SPen-n Me
CH (n-Pr) SHex-n Me
CH (n-Pr) SPr-c Me
CH (n-Pr) SBu-c Me
CH (n-Pr) SPen-c Me
CH (n-Pr) SHex-c Me
CH (n-Pr) SCH2CH = CH2                      Me
CH (n-Pr) SCH2C Three CH Me
CH (n-Pr) SCF2H Me
CH (n-Pr) SCFThree                            Me
CH (n-Pr) SCF2Cl Me
CH (n-Pr) SCH2CFThree                          Me
CH (n-Pr) S {D1-108c} Me
CH (n-Pr) S (O) Me Me
CH (n-Pr) S (O) Et Me
CH (n-Pr) S (O) Pr-n Me
CH (n-Pr) S (O) Pr-i Me
CH (n-Pr) S (O) Bu-n Me
CH (n-Pr) S (O) Bu-i Me
CH (n-Pr) S (O) Bu-t Me
CH (n-Pr) S (O) Pen-n Me
CH (n-Pr) S (O) Hex-n Me
CH (n-Pr) S (O) Pr-c Me
CH (n-Pr) S (O) Bu-c Me
CH (n-Pr) S (O) Pen-c Me
CH (n-Pr) S (O) Hex-c Me
CH (n-Pr) S (O) CH2CH = CH2                    Me
CH (n-Pr) S (O) CH2C Three CH Me
CH (n-Pr) S (O) CF2H Me
CH (n-Pr) S (O) CFThree                         Me
CH (n-Pr) S (O) CF2Cl Me
CH (n-Pr) S (O) CH2CFThree                      Me
CH (n-Pr) S (O) {D1-108c} Me
CH (n-Pr) S (O)2Me Me
CH (n-Pr) S (O)2Et Me
CH (n-Pr) S (O)2Pr-n Me
CH (n-Pr) S (O)2Pr-i Me
CH (n-Pr) S (O)2Bu-n Me
CH (n-Pr) S (O)2Bu-i Me
CH (n-Pr) S (O)2Bu-t Me
CH (n-Pr) S (O)2Pen-n Me
CH (n-Pr) S (O)2Hex-n Me
CH (n-Pr) S (O)2Pr-c Me
CH (n-Pr) S (O)2Bu-c Me
CH (n-Pr) S (O)2Pen-c Me
CH (n-Pr) S (O)2Hex-c Me
CH (n-Pr) S (O)2CH2CH = CH2                   Me
CH (n-Pr) S (O)2CH2C Three CH Me
CH (n-Pr) S (O)2CF2H Me
CH (n-Pr) S (O)2CFThree                        Me
CH (n-Pr) S (O)2CF2Cl Me
CH (n-Pr) S (O)2CH2CFThree                      Me
CH (n-Pr) S (O)2{D1-108c} Me
CH (i-Pr) SH Me
CH (i-Pr) SMe Me
CH (i-Pr) SEt Me
CH (i-Pr) SPr-n Me
CH (i-Pr) SPr-i Me
CH (i-Pr) SBu-n Me
CH (i-Pr) SBu-i Me
CH (i-Pr) SBu-t Me
CH (i-Pr) SPen-n Me
CH (i-Pr) SHex-n Me
CH (i-Pr) SPr-c Me
CH (i-Pr) SBu-c Me
CH (i-Pr) SPen-c Me
CH (i-Pr) SHex-c Me
CH (i-Pr) SCH2CH = CH2                      Me
CH (i-Pr) SCH2C Three CH Me
CH (i-Pr) SCF2H Me
CH (i-Pr) SCFThree                            Me
CH (i-Pr) SCF2Cl Me
CH (i-Pr) SCH2CFThree                          Me
CH (i-Pr) S {D1-108c} Me
CH (i-Pr) S (O) Me Me
CH (i-Pr) S (O) Et Me
CH (i-Pr) S (O) Pr-n Me
CH (i-Pr) S (O) Pr-i Me
CH (i-Pr) S (O) Bu-n Me
CH (i-Pr) S (O) Bu-i Me
CH (i-Pr) S (O) Bu-t Me
CH (i-Pr) S (O) Pen-n Me
CH (i-Pr) S (O) Hex-n Me
CH (i-Pr) S (O) Pr-c Me
CH (i-Pr) S (O) Bu-c Me
CH (i-Pr) S (O) Pen-c Me
CH (i-Pr) S (O) Hex-c Me
CH (i-Pr) S (O) CH2CH = CH2                    Me
CH (i-Pr) S (O) CH2C Three CH Me
CH (i-Pr) S (O) CF2H Me
CH (i-Pr) S (O) CFThree                         Me
CH (i-Pr) S (O) CF2Cl Me
CH (i-Pr) S (O) CH2CFThree                      Me
CH (i-Pr) S (O) {D1-108c} Me
CH (i-Pr) S (O)2Me Me
CH (i-Pr) S (O)2Et Me
CH (i-Pr) S (O)2Pr-n Me
CH (i-Pr) S (O)2Pr-i Me
CH (i-Pr) S (O)2Bu-n Me
CH (i-Pr) S (O)2Bu-i Me
CH (i-Pr) S (O)2Bu-t Me
CH (i-Pr) S (O)2Pen-n Me
CH (i-Pr) S (O)2Hex-n Me
CH (i-Pr) S (O)2Pr-c Me
CH (i-Pr) S (O)2Bu-c Me
CH (i-Pr) S (O)2Pen-c Me
CH (i-Pr) S (O)2Hex-c Me
CH (i-Pr) S (O)2CH2CH = CH2                   Me
CH (i-Pr) S (O)2CH2C Three CH Me
CH (i-Pr) S (O)2CF2H Me
CH (i-Pr) S (O)2CFThree                        Me
CH (i-Pr) S (O)2CF2Cl Me
CH (i-Pr) S (O)2CH2CFThree                      Me
CH (i-Pr) S (O)2{D1-108c} Me
CH (n-Bu) SH Me
CH (n-Bu) SMe Me
CH (n-Bu) SEt Me
CH (n-Bu) SPr-n Me
CH (n-Bu) SPr-i Me
CH (n-Bu) SBu-n Me
CH (n-Bu) SBu-i Me
CH (n-Bu) SBu-t Me
CH (n-Bu) SPen-n Me
CH (n-Bu) SHex-n Me
CH (n-Bu) SPr-c Me
CH (n-Bu) SBu-c Me
CH (n-Bu) SPen-c Me
CH (n-Bu) SHex-c Me
CH (n-Bu) SCH2CH = CH2                      Me
CH (n-Bu) SCH2C Three CH Me
CH (n-Bu) SCF2H Me
CH (n-Bu) SCFThree                            Me
CH (n-Bu) SCF2Cl Me
CH (n-Bu) SCH2CFThree                          Me
CH (n-Bu) S {D1-108c} Me
CH (n-Bu) S (O) Me Me
CH (n-Bu) S (O) Et Me
CH (n-Bu) S (O) Pr-n Me
CH (n-Bu) S (O) Pr-i Me
CH (n-Bu) S (O) Bu-n Me
CH (n-Bu) S (O) Bu-i Me
CH (n-Bu) S (O) Bu-t Me
CH (n-Bu) S (O) Pen-n Me
CH (n-Bu) S (O) Hex-n Me
CH (n-Bu) S (O) Pr-c Me
CH (n-Bu) S (O) Bu-c Me
CH (n-Bu) S (O) Pen-c Me
CH (n-Bu) S (O) Hex-c Me
CH (n-Bu) S (O) CH2CH = CH2                    Me
CH (n-Bu) S (O) CH2C Three CH Me
CH (n-Bu) S (O) CF2H Me
CH (n-Bu) S (O) CFThree                         Me
CH (n-Bu) S (O) CF2Cl Me
CH (n-Bu) S (O) CH2CFThree                      Me
CH (n-Bu) S (O) {D1-108c} Me
CH (n-Bu) S (O)2Me Me
CH (n-Bu) S (O)2Et Me
CH (n-Bu) S (O)2Pr-n Me
CH (n-Bu) S (O)2Pr-i Me
CH (n-Bu) S (O)2Bu-n Me
CH (n-Bu) S (O)2Bu-i Me
CH (n-Bu) S (O)2Bu-t Me
CH (n-Bu) S (O)2Pen-n Me
CH (n-Bu) S (O)2Hex-n Me
CH (n-Bu) S (O)2Pr-c Me
CH (n-Bu) S (O)2Bu-c Me
CH (n-Bu) S (O)2Pen-c Me
CH (n-Bu) S (O)2Hex-c Me
CH (n-Bu) S (O)2CH2CH = CH2                   Me
CH (n-Bu) S (O)2CH2C Three CH Me
CH (n-Bu) S (O)2CF2H Me
CH (n-Bu) S (O)2CFThree                        Me
CH (n-Bu) S (O)2CF2Cl Me
CH (n-Bu) S (O)2CH2CFThree                      Me
CH (n-Bu) S (O)2{D1-108c} Me
CH (CH2OMe) SH Me
CH (CH2OMe) SMe Me
CH (CH2OMe) SEt Me
CH (CH2OMe) SPr-n Me
CH (CH2OMe) SPr-i Me
CH (CH2OMe) SBu-n Me
CH (CH2OMe) SBu-i Me
CH (CH2OMe) SBu-t Me
CH (CH2OMe) SPen-n Me
CH (CH2OMe) SHex-n Me
CH (CH2OMe) SPr-c Me
CH (CH2OMe) SBu-c Me
CH (CH2OMe) SPen-c Me
CH (CH2OMe) SHex-c Me
CH (CH2OMe) SCH2CH = CH2                    Me
CH (CH2OMe) SCH2C Three CH Me
CH (CH2OMe) SCF2H Me
CH (CH2OMe) SCFThree                         Me
CH (CH2OMe) SCF2Cl Me
CH (CH2OMe) SCH2CFThree                       Me
CH (CH2OMe) S {D1-108c} Me
CH (CH2OMe) SCH2CH2CN Me
CH (CH2OMe) SCH2CH2CFThree                   Me
CH (CH2OMe) SCH2(D1-103a) Me
CH (CH2OMe) SCH2CH2OMe Me
CH (CH2OMe) SCH2CH2OEt Me
CH (CH2OMe) SCH2(D1-32a) Me
CH (CH2OMe) SCH2(D1-33a) Me
CH (CH2OMe) SCH2(D1-34a) Me
CH (CH2OMe) S {D1-32b (X1= 5-CFThree)} Me
CH (CH2OMe) SCH2(D1-81a) Me
CH (CH2OMe) SCH2(D1-82a) Me
CH (CH2OMe) SCH2(D1-84a) Me
CH (CH2OMe) SCH2(D1-85a) Me
CH (CH2OMe) SCH2(D1-87a) Me
CH (CH2OMe) SCH2(D1-95a) Me
CH (CH2OMe) SCH2(D1-96a) Me
CH (CH2OMe) SCH2(D1-98a) Me
CH (CH2OMe) SC (O) Me Me
CH (CH2OMe) SC (O) (D1-108a) Me
CH (CH2OMe) S (O) Me Me
CH (CH2OMe) S (O) Et Me
CH (CH2OMe) S (O) Pr-n Me
CH (CH2OMe) S (O) Pr-i Me
CH (CH2OMe) S (O) Bu-n Me
CH (CH2OMe) S (O) Bu-i Me
CH (CH2OMe) S (O) Bu-t Me
CH (CH2OMe) S (O) Pen-n Me
CH (CH2OMe) S (O) Hex-n Me
CH (CH2OMe) S (O) Pr-c Me
CH (CH2OMe) S (O) Bu-c Me
CH (CH2OMe) S (O) Pen-c Me
CH (CH2OMe) S (O) Hex-c Me
CH (CH2OMe) S (O) CH2CH = CH2                 Me
CH (CH2OMe) S (O) CH2C Three CH Me
CH (CH2OMe) S (O) CF2H Me
CH (CH2OMe) S (O) CFThree                      Me
CH (CH2OMe) S (O) CF2Cl Me
CH (CH2OMe) S (O) CH2CFThree                   Me
CH (CH2OMe) S (O) {D1-108c} Me
CH (CH2OMe) S (O) CH2CH2CN Me
CH (CH2OMe) S (O) CH2CH2CFThree                Me
CH (CH2OMe) S (O) CH2(D1-103a) Me
CH (CH2OMe) S (O) CH2CH2OMe Me
CH (CH2OMe) S (O) CH2CH2OEt Me
CH (CH2OMe) S (O) CH2(D1-32a) Me
CH (CH2OMe) S (O) CH2(D1-33a) Me
CH (CH2OMe) S (O) CH2(D1-34a) Me
CH (CH2OMe) S (O) {D1-32b (X1= 5-CFThree)} Me
CH (CH2OMe) S (O) CH2(D1-81a) Me
CH (CH2OMe) S (O) CH2(D1-82a) Me
CH (CH2OMe) S (O) CH2(D1-84a) Me
CH (CH2OMe) S (O) CH2(D1-85a) Me
CH (CH2OMe) S (O) CH2(D1-87a) Me
CH (CH2OMe) S (O) CH2(D1-95a) Me
CH (CH2OMe) S (O) CH2(D1-96a) Me
CH (CH2OMe) S (O) CH2(D1-98a) Me
CH (CH2OMe) S (O)2Me Me
CH (CH2OMe) S (O)2Et Me
CH (CH2OMe) S (O)2Pr-n Me
CH (CH2OMe) S (O)2Pr-i Me
CH (CH2OMe) S (O)2Bu-n Me
CH (CH2OMe) S (O)2Bu-i Me
CH (CH2OMe) S (O)2Bu-t Me
CH (CH2OMe) S (O)2Pen-n Me
CH (CH2OMe) S (O)2Hex-n Me
CH (CH2OMe) S (O)2Pr-c Me
CH (CH2OMe) S (O)2Bu-c Me
CH (CH2OMe) S (O)2Pen-c Me
CH (CH2OMe) S (O)2Hex-c Me
CH (CH2OMe) S (O)2CH2CH = CH2                 Me
CH (CH2OMe) S (O)2CH2C Three CH Me
CH (CH2OMe) S (O)2CF2H Me
CH (CH2OMe) S (O)2CFThree                      Me
CH (CH2OMe) S (O)2CF2Cl Me
CH (CH2OMe) S (O)2CH2CFThree                    Me
CH (CH2OMe) S (O)2{D1-108c} Me
CH (CH2OMe) S (O)2CH2CH2CN Me
CH (CH2OMe) S (O)2CH2CH2CFThree                Me
CH (CH2OMe) S (O)2CH2(D1-103a) Me
CH (CH2OMe) S (O)2CH2CH2OMe Me
CH (CH2OMe) S (O)2CH2CH2OEt Me
CH (CH2OMe) S (O)2CH2(D1-32a) Me
CH (CH2OMe) S (O)2CH2(D1-33a) Me
CH (CH2OMe) S (O)2CH2(D1-34a) Me
CH (CH2OMe) S (O)2{D1-32b (X1= 5-CFThree)} Me
CH (CH2OMe) S (O)2CH2(D1-81a) Me
CH (CH2OMe) S (O)2CH2(D1-82a) Me
CH (CH2OMe) S (O)2CH2(D1-84a) Me
CH (CH2OMe) S (O)2CH2(D1-85a) Me
CH (CH2OMe) S (O)2CH2(D1-87a) Me
CH (CH2OMe) S (O)2CH2(D1-95a) Me
CH (CH2OMe) S (O)2CH2(D1-96a) Me
CH (CH2OMe) S (O)2CH2(D1-98a) Me
CH (CH2CH = CH2SH Me
CH (CH2CH = CH2SMe Me
CH (CH2CH = CH2) SEt Me
CH (CH2CH = CH2SPr-n Me
CH (CH2CH = CH2SPr-i Me
CH (CH2CH = CH2) SBu-n Me
CH (CH2CH = CH2) SBu-i Me
CH (CH2CH = CH2) SBu-t Me
CH (CH2CH = CH2SPen-n Me
CH (CH2CH = CH2SHex-n Me
CH (CH2CH = CH2SPr-c Me
CH (CH2CH = CH2) SBu-c Me
CH (CH2CH = CH2SPen-c Me
CH (CH2CH = CH2SHex-c Me
CH (CH2CH = CH2) SCH2CH = CH2                  Me
CH (CH2CH = CH2) SCH2C Three CH Me
CH (CH2CH = CH2) SCF2H Me
CH (CH2CH = CH2) SCFThree                       Me
CH (CH2CH = CH2) SCF2Cl Me
CH (CH2CH = CH2) SCH2CFThree                     Me
CH (CH2CH = CH2) S {D1-108c} Me
CH (CH2CH = CH2) SCH2CH2CN Me
CH (CH2CH = CH2) SCH2CH2CFThree                   Me
CH (CH2CH = CH2) SCH2(D1-103a) Me
CH (CH2CH = CH2) SCH2CH2OMe Me
CH (CH2CH = CH2) SCH2CH2OEt Me
CH (CH2CH = CH2) SCH2(D1-32a) Me
CH (CH2CH = CH2) SCH2(D1-33a) Me
CH (CH2CH = CH2) SCH2(D1-34a) Me
CH (CH2CH = CH2) S {D1-32b (X1= 5-CFThree)} Me
CH (CH2CH = CH2) SCH2(D1-81a) Me
CH (CH2CH = CH2) SCH2(D1-82a) Me
CH (CH2CH = CH2) SCH2(D1-84a) Me
CH (CH2CH = CH2) SCH2(D1-85a) Me
CH (CH2CH = CH2) SCH2(D1-87a) Me
CH (CH2CH = CH2) SCH2(D1-95a) Me
CH (CH2CH = CH2) SCH2(D1-96a) Me
CH (CH2CH = CH2) SCH2(D1-98a) Me
CH (CH2CH = CH2) SC (O) Me Me
CH (CH2CH = CH2) SC (O) (D1-108a) Me
CH (CH2CH = CH2) S (O) Me Me
CH (CH2CH = CH2) S (O) Et Me
CH (CH2CH = CH2) S (O) Pr-n Me
CH (CH2CH = CH2) S (O) Pr-i Me
CH (CH2CH = CH2) S (O) Bu-n Me
CH (CH2CH = CH2) S (O) Bu-i Me
CH (CH2CH = CH2) S (O) Bu-t Me
CH (CH2CH = CH2) S (O) Pen-n Me
CH (CH2CH = CH2) S (O) Hex-n Me
CH (CH2CH = CH2) S (O) Pr-c Me
CH (CH2CH = CH2) S (O) Bu-c Me
CH (CH2CH = CH2) S (O) Pen-c Me
CH (CH2CH = CH2) S (O) Hex-c Me
CH (CH2CH = CH2) S (O) CH2CH = CH2               Me
CH (CH2CH = CH2) S (O) CH2C Three CH Me
CH (CH2CH = CH2) S (O) CF2H Me
CH (CH2CH = CH2) S (O) CFThree                    Me
CH (CH2CH = CH2) S (O) CF2Cl Me
CH (CH2CH = CH2) S (O) CH2CFThree                 Me
CH (CH2CH = CH2) S (O) {D1-108c} Me
CH (CH2CH = CH2) S (O) CH2CH2CN Me
CH (CH2CH = CH2) S (O) CH2CH2CFThree              Me
CH (CH2CH = CH2) S (O) CH2(D1-103a) Me
CH (CH2CH = CH2) S (O) CH2CH2OMe Me
CH (CH2CH = CH2) S (O) CH2CH2OEt Me
CH (CH2CH = CH2) S (O) CH2(D1-32a) Me
CH (CH2CH = CH2) S (O) CH2(D1-33a) Me
CH (CH2CH = CH2) S (O) CH2(D1-34a) Me
CH (CH2CH = CH2) S (O) {D1-32b (X1= 5-CFThree)} Me
CH (CH2CH = CH2) S (O) CH2(D1-81a) Me
CH (CH2CH = CH2) S (O) CH2(D1-82a) Me
CH (CH2CH = CH2) S (O) CH2(D1-84a) Me
CH (CH2CH = CH2) S (O) CH2(D1-85a) Me
CH (CH2CH = CH2) S (O) CH2(D1-87a) Me
CH (CH2CH = CH2) S (O) CH2(D1-95a) Me
CH (CH2CH = CH2) S (O) CH2(D1-96a) Me
CH (CH2CH = CH2) S (O) CH2(D1-98a) Me
CH (CH2CH = CH2) S (O)2Me Me
CH (CH2CH = CH2) S (O)2Et Me
CH (CH2CH = CH2) S (O)2Pr-n Me
CH (CH2CH = CH2) S (O)2Pr-i Me
CH (CH2CH = CH2) S (O)2Bu-n Me
CH (CH2CH = CH2) S (O)2Bu-i Me
CH (CH2CH = CH2) S (O)2Bu-t Me
CH (CH2CH = CH2) S (O)2Pen-n Me
CH (CH2CH = CH2) S (O)2Hex-n Me
CH (CH2CH = CH2) S (O)2Pr-c Me
CH (CH2CH = CH2) S (O)2Bu-c Me
CH (CH2CH = CH2) S (O)2Pen-c Me
CH (CH2CH = CH2) S (O)2Hex-c Me
CH (CH2CH = CH2) S (O)2CH2CH = CH2              Me
CH (CH2CH = CH2) S (O)2CH2C Three CH Me
CH (CH2CH = CH2) S (O)2CF2H Me
CH (CH2CH = CH2) S (O)2CFThree                    Me
CH (CH2CH = CH2) S (O)2CF2Cl Me
CH (CH2CH = CH2) S (O)2CH2CFThree                  Me
CH (CH2CH = CH2) S (O)2{D1-108c} Me
CH (CH2CH = CH2) S (O)2CH2CH2CN Me
CH (CH2CH = CH2) S (O)2CH2CH2CFThree              Me
CH (CH2CH = CH2) S (O)2CH2(D1-103a) Me
CH (CH2CH = CH2) S (O)2CH2CH2OMe Me
CH (CH2CH = CH2) S (O)2CH2CH2OEt Me
CH (CH2CH = CH2) S (O)2CH2(D1-32a) Me
CH (CH2CH = CH2) S (O)2CH2(D1-33a) Me
CH (CH2CH = CH2) S (O)2CH2(D1-34a) Me
CH (CH2CH = CH2) S (O)2{D1-32b (X1= 5-CFThree)} Me
CH (CH2CH = CH2) S (O)2CH2(D1-81a) Me
CH (CH2CH = CH2) S (O)2CH2(D1-82a) Me
CH (CH2CH = CH2) S (O)2CH2(D1-84a) Me
CH (CH2CH = CH2) S (O)2CH2(D1-85a) Me
CH (CH2CH = CH2) S (O)2CH2(D1-87a) Me
CH (CH2CH = CH2) S (O)2CH2(D1-95a) Me
CH (CH2CH = CH2) S (O)2CH2(D1-96a) Me
CH (CH2CH = CH2) S (O)2CH2(D1-98a) Me
CH (CH2C≡CH) SH Me
CH (CH2C≡CH) SMe Me
CH (CH2C≡CH) SEt Me
CH (CH2C≡CH) SPr-n Me
CH (CH2C≡CH) SPr-i Me
CH (CH2C≡CH) SBu-n Me
CH (CH2C≡CH) SBu-i Me
CH (CH2C≡CH) SBu-t Me
CH (CH2C≡CH) SPen-n Me
CH (CH2C≡CH) SHex-n Me
CH (CH2C≡CH) SPr-c Me
CH (CH2C≡CH) SBu-c Me
CH (CH2C≡CH) SPen-c Me
CH (CH2C≡CH) SHex-c Me
CH (CH2C≡CH) SCH2CH = CH2                   Me
CH (CH2C≡CH) SCH2C Three CH Me
CH (CH2C≡CH) SCF2H Me
CH (CH2C≡CH) SCFThree                        Me
CH (CH2C≡CH) SCF2Cl Me
CH (CH2C≡CH) SCH2CFThree                      Me
CH (CH2C≡CH) S {D1-108c} Me
CH (CH2C≡CH) SCH2CH2CN Me
CH (CH2C≡CH) SCH2CH2CFThree                   Me
CH (CH2C≡CH) SCH2(D1-103a) Me
CH (CH2C≡CH) SCH2CH2OMe Me
CH (CH2C≡CH) SCH2CH2OEt Me
CH (CH2C≡CH) SCH2(D1-32a) Me
CH (CH2C≡CH) SCH2(D1-33a) Me
CH (CH2C≡CH) SCH2(D1-34a) Me
CH (CH2C≡CH) S {D1-32b (X1= 5-CFThree)} Me
CH (CH2C≡CH) SCH2(D1-81a) Me
CH (CH2C≡CH) SCH2(D1-82a) Me
CH (CH2C≡CH) SCH2(D1-84a) Me
CH (CH2C≡CH) SCH2(D1-85a) Me
CH (CH2C≡CH) SCH2(D1-87a) Me
CH (CH2C≡CH) SCH2(D1-95a) Me
CH (CH2C≡CH) SCH2(D1-96a) Me
CH (CH2C≡CH) SCH2(D1-98a) Me
CH (CH2C≡CH) SC (O) Me Me
CH (CH2C≡CH) SC (O) (D1-108a) Me
CH (CH2C≡CH) S (O) Me Me
CH (CH2C≡CH) S (O) Et Me
CH (CH2C≡CH) S (O) Pr-n Me
CH (CH2C≡CH) S (O) Pr-i Me
CH (CH2C≡CH) S (O) Bu-n Me
CH (CH2C≡CH) S (O) Bu-i Me
CH (CH2C≡CH) S (O) Bu-t Me
CH (CH2C≡CH) S (O) Pen-n Me
CH (CH2C≡CH) S (O) Hex-n Me
CH (CH2C≡CH) S (O) Pr-c Me
CH (CH2C≡CH) S (O) Bu-c Me
CH (CH2C≡CH) S (O) Pen-c Me
CH (CH2C≡CH) S (O) Hex-c Me
CH (CH2C≡CH) S (O) CH2CH = CH2                Me
CH (CH2C≡CH) S (O) CH2C Three CH Me
CH (CH2C≡CH) S (O) CF2H Me
CH (CH2C≡CH) S (O) CFThree                     Me
CH (CH2C≡CH) S (O) CF2Cl Me
CH (CH2C≡CH) S (O) CH2CFThree                  Me
CH (CH2C≡CH) S (O) {D1-108c} Me
CH (CH2C≡CH) S (O) CH2CH2CN Me
CH (CH2C≡CH) S (O) CH2CH2CFThree               Me
CH (CH2C≡CH) S (O) CH2(D1-103a) Me
CH (CH2C≡CH) S (O) CH2CH2OMe Me
CH (CH2C≡CH) S (O) CH2CH2OEt Me
CH (CH2C≡CH) S (O) CH2(D1-32a) Me
CH (CH2C≡CH) S (O) CH2(D1-33a) Me
CH (CH2C≡CH) S (O) CH2(D1-34a) Me
CH (CH2C≡CH) S (O) {D1-32b (X1= 5-CFThree)} Me
CH (CH2C≡CH) S (O) CH2(D1-81a) Me
CH (CH2C≡CH) S (O) CH2(D1-82a) Me
CH (CH2C≡CH) S (O) CH2(D1-84a) Me
CH (CH2C≡CH) S (O) CH2(D1-85a) Me
CH (CH2C≡CH) S (O) CH2(D1-87a) Me
CH (CH2C≡CH) S (O) CH2(D1-95a) Me
CH (CH2C≡CH) S (O) CH2(D1-96a) Me
CH (CH2C≡CH) S (O) CH2(D1-98a) Me
CH (CH2C≡CH) S (O)2Me Me
CH (CH2C≡CH) S (O)2Et Me
CH (CH2C≡CH) S (O)2Pr-n Me
CH (CH2C≡CH) S (O)2Pr-i Me
CH (CH2C≡CH) S (O)2Bu-n Me
CH (CH2C≡CH) S (O)2Bu-i Me
CH (CH2C≡CH) S (O)2Bu-t Me
CH (CH2C≡CH) S (O)2Pen-n Me
CH (CH2C≡CH) S (O)2Hex-n Me
CH (CH2C≡CH) S (O)2Pr-c Me
CH (CH2C≡CH) S (O)2Bu-c Me
CH (CH2C≡CH) S (O)2Pen-c Me
CH (CH2C≡CH) S (O)2Hex-c Me
CH (CH2C≡CH) S (O)2CH2CH = CH2               Me
CH (CH2C≡CH) S (O)2CH2C Three CH Me
CH (CH2C≡CH) S (O)2CF2H Me
CH (CH2C≡CH) S (O)2CFThree                     Me
CH (CH2C≡CH) S (O)2CF2Cl Me
CH (CH2C≡CH) S (O)2CH2CFThree                   Me
CH (CH2C≡CH) S (O)2{D1-108c} Me
CH (CH2C≡CH) S (O)2CH2CH2CN Me
CH (CH2C≡CH) S (O)2CH2CH2CFThree               Me
CH (CH2C≡CH) S (O)2CH2(D1-103a) Me
CH (CH2C≡CH) S (O)2CH2CH2OMe Me
CH (CH2C≡CH) S (O)2CH2CH2OEt Me
CH (CH2C≡CH) S (O)2CH2(D1-32a) Me
CH (CH2C≡CH) S (O)2CH2(D1-33a) Me
CH (CH2C≡CH) S (O)2CH2(D1-34a) Me
CH (CH2C≡CH) S (O)2{D1-32b (X1= 5-CFThree)} Me
CH (CH2C≡CH) S (O)2CH2(D1-81a) Me
CH (CH2C≡CH) S (O)2CH2(D1-82a) Me
CH (CH2C≡CH) S (O)2CH2(D1-84a) Me
CH (CH2C≡CH) S (O)2CH2(D1-85a) Me
CH (CH2C≡CH) S (O)2CH2(D1-87a) Me
CH (CH2C≡CH) S (O)2CH2(D1-95a) Me
CH (CH2C≡CH) S (O)2CH2(D1-96a) Me
CH (CH2C≡CH) S (O)2CH2(D1-98a) Me
CH (CH2CN) SH Me
CH (CH2CN) SMe Me
CH (CH2CN) SEt Me
CH (CH2CN) SPr-n Me
CH (CH2CN) SPr-i Me
CH (CH2CN) SBu-n Me
CH (CH2CN) SBu-i Me
CH (CH2CN) SBu-t Me
CH (CH2CN) SPen-n Me
CH (CH2CN) SHex-n Me
CH (CH2CN) SPr-c Me
CH (CH2CN) SBu-c Me
CH (CH2CN) SPen-c Me
CH (CH2CN) SHex-c Me
CH (CH2CN) SCH2CH = CH2                      Me
CH (CH2CN) SCH2C Three CH Me
CH (CH2CN) SCF2H Me
CH (CH2CN) SCFThree                           Me
CH (CH2CN) SCF2Cl Me
CH (CH2CN) SCH2CFThree                         Me
CH (CH2CN) S {D1-108c} Me
CH (CH2CN) SCH2CH2CN Me
CH (CH2CN) SCH2CH2CFThree                     Me
CH (CH2CN) SCH2(D1-103a) Me
CH (CH2CN) SCH2CH2OMe Me
CH (CH2CN) SCH2CH2OEt Me
CH (CH2CN) SCH2(D1-32a) Me
CH (CH2CN) SCH2(D1-33a) Me
CH (CH2CN) SCH2(D1-34a) Me
CH (CH2CN) S {D1-32b (X1= 5-CFThree)} Me
CH (CH2CN) SCH2(D1-81a) Me
CH (CH2CN) SCH2(D1-82a) Me
CH (CH2CN) SCH2(D1-84a) Me
CH (CH2CN) SCH2(D1-85a) Me
CH (CH2CN) SCH2(D1-87a) Me
CH (CH2CN) SCH2(D1-95a) Me
CH (CH2CN) SCH2(D1-96a) Me
CH (CH2CN) SCH2(D1-98a) Me
CH (CH2CN) SC (O) Me Me
CH (CH2CN) SC (O) (D1-108a) Me
CH (CH2CN) S (O) Me Me
CH (CH2CN) S (O) Et Me
CH (CH2CN) S (O) Pr-n Me
CH (CH2CN) S (O) Pr-i Me
CH (CH2CN) S (O) Bu-n Me
CH (CH2CN) S (O) Bu-i Me
CH (CH2CN) S (O) Bu-t Me
CH (CH2CN) S (O) Pen-n Me
CH (CH2CN) S (O) Hex-n Me
CH (CH2CN) S (O) Pr-c Me
CH (CH2CN) S (O) Bu-c Me
CH (CH2CN) S (O) Pen-c Me
CH (CH2CN) S (O) Hex-c Me
CH (CH2CN) S (O) CH2CH = CH2                   Me
CH (CH2CN) S (O) CH2C Three CH Me
CH (CH2CN) S (O) CF2H Me
CH (CH2CN) S (O) CFThree                        Me
CH (CH2CN) S (O) CF2Cl Me
CH (CH2CN) S (O) CH2CFThree                    Me
CH (CH2CN) S (O) {D1-108c} Me
CH (CH2CN) S (O) CH2CH2CN Me
CH (CH2CN) S (O) CH2CH2CFThree                  Me
CH (CH2CN) S (O) CH2(D1-103a) Me
CH (CH2CN) S (O) CH2CH2OMe Me
CH (CH2CN) S (O) CH2CH2OEt Me
CH (CH2CN) S (O) CH2(D1-32a) Me
CH (CH2CN) S (O) CH2(D1-33a) Me
CH (CH2CN) S (O) CH2(D1-34a) Me
CH (CH2CN) S (O) {D1-32b (X1= 5-CFThree)} Me
CH (CH2CN) S (O) CH2(D1-81a) Me
CH (CH2CN) S (O) CH2(D1-82a) Me
CH (CH2CN) S (O) CH2(D1-84a) Me
CH (CH2CN) S (O) CH2(D1-85a) Me
CH (CH2CN) S (O) CH2(D1-87a) Me
CH (CH2CN) S (O) CH2(D1-95a) Me
CH (CH2CN) S (O) CH2(D1-96a) Me
CH (CH2CN) S (O) CH2(D1-98a) Me
CH (CH2CN) S (O)2Me Me
CH (CH2CN) S (O)2Et Me
CH (CH2CN) S (O)2Pr-n Me
CH (CH2CN) S (O)2Pr-i Me
CH (CH2CN) S (O)2Bu-n Me
CH (CH2CN) S (O)2Bu-i Me
CH (CH2CN) S (O)2Bu-t Me
CH (CH2CN) S (O)2Pen-n Me
CH (CH2CN) S (O)2Hex-n Me
CH (CH2CN) S (O)2Pr-c Me
CH (CH2CN) S (O)2Bu-c Me
CH (CH2CN) S (O)2Pen-c Me
CH (CH2CN) S (O)2Hex-c Me
CH (CH2CN) S (O)2CH2CH = CH2                  Me
CH (CH2CN) S (O)2CH2C Three CH Me
CH (CH2CN) S (O)2CF2H Me
CH (CH2CN) S (O)2CFThree                        Me
CH (CH2CN) S (O)2CF2Cl Me
CH (CH2CN) S (O)2CH2CFThree                     Me
CH (CH2CN) S (O)2{D1-108c} Me
CH (CH2CN) S (O)2CH2CH2CN Me
CH (CH2CN) S (O)2CH2CH2CFThree                 Me
CH (CH2CN) S (O)2CH2(D1-103a) Me
CH (CH2CN) S (O)2CH2CH2OMe Me
CH (CH2CN) S (O)2CH2CH2OEt Me
CH (CH2CN) S (O)2CH2(D1-32a) Me
CH (CH2CN) S (O)2CH2(D1-33a) Me
CH (CH2CN) S (O)2CH2(D1-34a) Me
CH (CH2CN) S (O)2{D1-32b (X1= 5-CFThree)} Me
CH (CH2CN) S (O)2CH2(D1-81a) Me
CH (CH2CN) S (O)2CH2(D1-82a) Me
CH (CH2CN) S (O)2CH2(D1-84a) Me
CH (CH2CN) S (O)2CH2(D1-85a) Me
CH (CH2CN) S (O)2CH2(D1-87a) Me
CH (CH2CN) S (O)2CH2(D1-95a) Me
CH (CH2CN) S (O)2CH2(D1-96a) Me
CH (CH2CN) S (O)2CH2(D1-98a) Me
CH (Me)2SH Me
CH (Me)2SMe Me
CH (Me)2SEt Me
CH (Me)2SPr-n Me
CH (Me)2SPr-i Me
CH (Me)2SBu-n Me
CH (Me)2SBu-i Me
CH (Me)2SBu-t Me
CH (Me)2SPen-n Me
CH (Me)2SHex-n Me
CH (Me)2SPr-c Me
CH (Me)2SBu-c Me
CH (Me)2SPen-c Me
CH (Me)2SHex-c Me
CH (Me)2SCH2CH = CH2                        Me
CH (Me)2SCH2C Three CH Me
CH (Me)2SCF2H Me
CH (Me)2SCFThree                             Me
CH (Me)2SCF2Cl Me
CH (Me)2SCH2CFThree                           Me
CH (Me)2S {D1-108c} Me
CH (Me)2SCH2CH2CN Me
CH (Me)2SCH2CH2CFThree                       Me
CH (Me)2SCH2(D1-103a) Me
CH (Me)2SCH2CH2OMe Me
CH (Me)2SCH2CH2OEt Me
CH (Me)2SCH2(D1-32a) Me
CH (Me)2SCH2(D1-33a) Me
CH (Me)2SCH2(D1-34a) Me
CH (Me)2S {D1-32b (X1= 5-CFThree)} Me
CH (Me)2SCH2(D1-81a) Me
CH (Me)2SCH2(D1-82a) Me
CH (Me)2SCH2(D1-84a) Me
CH (Me)2SCH2(D1-85a) Me
CH (Me)2SCH2(D1-87a) Me
CH (Me)2SCH2(D1-95a) Me
CH (Me)2SCH2(D1-96a) Me
CH (Me)2SCH2(D1-98a) Me
CH (Me)2SC (O) Me Me
CH (Me)2SC (O) (D1-108a) Me
CH (Me)2S (O) Me Me
CH (Me)2S (O) Et Me
CH (Me)2S (O) Pr-n Me
CH (Me)2S (O) Pr-i Me
CH (Me)2S (O) Bu-n Me
CH (Me)2S (O) Bu-i Me
CH (Me)2S (O) Bu-t Me
CH (Me)2S (O) Pen-n Me
CH (Me)2S (O) Hex-n Me
CH (Me)2S (O) Pr-c Me
CH (Me)2S (O) Bu-c Me
CH (Me)2S (O) Pen-c Me
CH (Me)2S (O) Hex-c Me
CH (Me)2S (O) CH2CH = CH2                     Me
CH (Me)2S (O) CH2C Three CH Me
CH (Me)2S (O) CF2H Me
CH (Me)2S (O) CFThree                          Me
CH (Me)2S (O) CF2Cl Me
CH (Me)2S (O) CH2CFThree                      Me
CH (Me)2S (O) {D1-108c} Me
CH (Me)2S (O) CH2CH2CN Me
CH (Me)2S (O) CH2CH2CFThree                      Me
CH (Me)2S (O) CH2(D1-103a) Me
CH (Me)2S (O) CH2CH2OMe Me
CH (Me)2S (O) CH2CH2OEt Me
CH (Me)2S (O) CH2(D1-32a) Me
CH (Me)2S (O) CH2(D1-33a) Me
CH (Me)2S (O) CH2(D1-34a) Me
CH (Me)2S (O) {D1-32b (X1= 5-CFThree)} Me
CH (Me)2S (O) CH2(D1-81a) Me
CH (Me)2S (O) CH2(D1-82a) Me
CH (Me)2S (O) CH2(D1-84a) Me
CH (Me)2S (O) CH2(D1-85a) Me
CH (Me)2S (O) CH2(D1-87a) Me
CH (Me)2S (O) CH2(D1-95a) Me
CH (Me)2S (O) CH2(D1-96a) Me
CH (Me)2S (O) CH2(D1-98a) Me
CH (Me)2S (O)2Me Me
CH (Me)2S (O)2Et Me
CH (Me)2S (O)2Pr-n Me
CH (Me)2S (O)2Pr-i Me
CH (Me)2S (O)2Bu-n Me
CH (Me)2S (O)2Bu-i Me
CH (Me)2S (O)2Bu-t Me
CH (Me)2S (O)2Pen-n Me
CH (Me)2S (O)2Hex-n Me
CH (Me)2S (O)2Pr-c Me
CH (Me)2S (O)2Bu-c Me
CH (Me)2S (O)2Pen-c Me
CH (Me)2S (O)2Hex-c Me
CH (Me)2S (O)2CH2CH = CH2                    Me
CH (Me)2S (O)2CH2C Three CH Me
CH (Me)2S (O)2CF2H Me
CH (Me)2S (O)2CFThree                          Me
CH (Me)2S (O)2CF2Cl Me
CH (Me)2S (O)2CH2CFThree                        Me
CH (Me)2S (O)2{D1-108c} Me
CH (Me)2S (O)2CH2CH2CN Me
CH (Me)2S (O)2CH2CH2CFThree                      Me
CH (Me)2S (O)2CH2(D1-103a) Me
CH (Me)2S (O)2CH2CH2OMe Me
CH (Me)2S (O)2CH2CH2OEt Me
CH (Me)2S (O)2CH2(D1-32a) Me
CH (Me)2S (O)2CH2(D1-33a) Me
CH (Me)2S (O)2CH2(D1-34a) Me
CH (Me)2S (O)2{D1-32b (X1= 5-CFThree)} Me
CH (Me)2S (O)2CH2(D1-81a) Me
CH (Me)2S (O)2CH2(D1-82a) Me
CH (Me)2S (O)2CH2(D1-84a) Me
CH (Me)2S (O)2CH2(D1-85a) Me
CH (Me)2S (O)2CH2(D1-87a) Me
CH (Me)2S (O)2CH2(D1-95a) Me
CH (Me)2S (O)2CH2(D1-96a) Me
CH (Me)2S (O)2CH2(D1-98a) Me
CH2CH2SH Me
CH2CH2SMe Me
CH2CH2SEt Me
CH2CH2SPr-n Me
CH2CH2SPr-i Me
CH2CH2SBu-n Me
CH2CH2SBu-i Me
CH2CH2SBu-t Me
CH2CH2SPen-n Me
CH2CH2SHex-n Me
CH2CH2SPr-c Me
CH2CH2SBu-c Me
CH2CH2SPen-c Me
CH2CH2SHex-c Me
CH2CH2SCH2CH = CH2                         Me
CH2CH2SCH2C Three CH Me
CH2CH2SCF2H Me
CH2CH2SCFThree                              Me
CH2CH2SCF2Cl Me
CH2CH2SCH2CFThree                            Me
CH2CH2S {D1-108c} Me
CH2CH2SCH2CH2CN Me
CH2CH2SCH2CH2CFThree                         Me
CH2CH2SCH2(D1-103a) Me
CH2CH2SCH2CH2OMe Me
CH2CH2SCH2CH2OEt Me
CH2CH2SCH2(D1-32a) Me
CH2CH2SCH2(D1-33a) Me
CH2CH2SCH2(D1-34a) Me
CH2CH2S {D1-32b (X1= 5-CFThree)} Me
CH2CH2SCH2(D1-81a) Me
CH2CH2SCH2(D1-82a) Me
CH2CH2SCH2(D1-84a) Me
CH2CH2SCH2(D1-85a) Me
CH2CH2SCH2(D1-87a) Me
CH2CH2SCH2(D1-95a) Me
CH2CH2SCH2(D1-96a) Me
CH2CH2SCH2(D1-98a) Me
CH2CH2SC (O) Me Me
CH2CH2SC (O) (D1-108a) Me
CH2CH2S (O) Me Me
CH2CH2S (O) Et Me
CH2CH2S (O) Pr-n Me
CH2CH2S (O) Pr-i Me
CH2CH2S (O) Bu-n Me
CH2CH2S (O) Bu-i Me
CH2CH2S (O) Bu-t Me
CH2CH2S (O) Pen-n Me
CH2CH2S (O) Hex-n Me
CH2CH2S (O) Pr-c Me
CH2CH2S (O) Bu-c Me
CH2CH2S (O) Pen-c Me
CH2CH2S (O) Hex-c Me
CH2CH2S (O) CH2CH = CH2                      Me
CH2CH2S (O) CH2C Three CH Me
CH2CH2S (O) CF2H Me
CH2CH2S (O) CFThree                           Me
CH2CH2S (O) CF2Cl Me
CH2CH2S (O) CH2CFThree                       Me
CH2CH2S (O) {D1-108c} Me
CH2CH2S (O) CH2CH2CN Me
CH2CH2S (O) CH2CH2CFThree                      Me
CH2CH2S (O) CH2(D1-103a) Me
CH2CH2S (O) CH2CH2OMe Me
CH2CH2S (O) CH2CH2OEt Me
CH2CH2S (O) CH2(D1-32a) Me
CH2CH2S (O) CH2(D1-33a) Me
CH2CH2S (O) CH2(D1-34a) Me
CH2CH2S (O) {D1-32b (X1= 5-CFThree)} Me
CH2CH2S (O) CH2(D1-81a) Me
CH2CH2S (O) CH2(D1-82a) Me
CH2CH2S (O) CH2(D1-84a) Me
CH2CH2S (O) CH2(D1-85a) Me
CH2CH2S (O) CH2(D1-87a) Me
CH2CH2S (O) CH2(D1-95a) Me
CH2CH2S (O) CH2(D1-96a) Me
CH2CH2S (O) CH2(D1-98a) Me
CH2CH2S (O)2Me Me
CH2CH2S (O)2Et Me
CH2CH2S (O)2Pr-n Me
CH2CH2S (O)2Pr-i Me
CH2CH2S (O)2Bu-n Me
CH2CH2S (O)2Bu-i Me
CH2CH2S (O)2Bu-t Me
CH2CH2S (O)2Pen-n Me
CH2CH2S (O)2Hex-n Me
CH2CH2S (O)2Pr-c Me
CH2CH2S (O)2Bu-c Me
CH2CH2S (O)2Pen-c Me
CH2CH2S (O)2Hex-c Me
CH2CH2S (O)2CH2CH = CH2                     Me
CH2CH2S (O)2CH2C Three CH Me
CH2CH2S (O)2CF2H Me
CH2CH2S (O)2CFThree                           Me
CH2CH2S (O)2CF2Cl Me
CH2CH2S (O)2CH2CFThree                         Me
CH2CH2S (O)2{D1-108c} Me
CH2CH2S (O)2CH2CH2CN Me
CH2CH2S (O)2CH2CH2CFThree                      Me
CH2CH2S (O)2CH2(D1-103a) Me
CH2CH2S (O)2CH2CH2OMe Me
CH2CH2S (O)2CH2CH2OEt Me
CH2CH2S (O)2CH2(D1-32a) Me
CH2CH2S (O)2CH2(D1-33a) Me
CH2CH2S (O)2CH2(D1-34a) Me
CH2CH2S (O)2{D1-32b (X1= 5-CFThree)} Me
CH2CH2S (O)2CH2(D1-81a) Me
CH2CH2S (O)2CH2(D1-82a) Me
CH2CH2S (O)2CH2(D1-84a) Me
CH2CH2S (O)2CH2(D1-85a) Me
CH2CH2S (O)2CH2(D1-87a) Me
CH2CH2S (O)2CH2(D1-95a) Me
CH2CH2S (O)2CH2(D1-96a) Me
CH2CH2S (O)2CH2(D1-98a) Me
CH (Me) CH2SH Me
CH (Me) CH2SMe Me
CH (Me) CH2SEt Me
CH (Me) CH2SPr-n Me
CH (Me) CH2SPr-i Me
CH (Me) CH2SBu-n Me
CH (Me) CH2SBu-i Me
CH (Me) CH2SBu-t Me
CH (Me) CH2SPen-n Me
CH (Me) CH2SHex-n Me
CH (Me) CH2SPr-c Me
CH (Me) CH2SBu-c Me
CH (Me) CH2SPen-c Me
CH (Me) CH2SHex-c Me
CH (Me) CH2SCH2CH = CH2                      Me
CH (Me) CH2SCH2C Three CH Me
CH (Me) CH2SCF2H Me
CH (Me) CH2SCFThree                           Me
CH (Me) CH2SCF2Cl Me
CH (Me) CH2SCH2CFThree                         Me
CH (Me) CH2S {D1-108c} Me
CH (Me) CH2SCH2CH2CN Me
CH (Me) CH2SCH2CH2CFThree                      Me
CH (Me) CH2SCH2(D1-103a) Me
CH (Me) CH2SCH2CH2OMe Me
CH (Me) CH2SCH2CH2OEt Me
CH (Me) CH2SCH2(D1-32a) Me
CH (Me) CH2SCH2(D1-33a) Me
CH (Me) CH2SCH2(D1-34a) Me
CH (Me) CH2S {D1-32b (X1= 5-CFThree)} Me
CH (Me) CH2SCH2(D1-81a) Me
CH (Me) CH2SCH2(D1-82a) Me
CH (Me) CH2SCH2(D1-84a) Me
CH (Me) CH2SCH2(D1-85a) Me
CH (Me) CH2SCH2(D1-87a) Me
CH (Me) CH2SCH2(D1-95a) Me
CH (Me) CH2SCH2(D1-96a) Me
CH (Me) CH2SCH2(D1-98a) Me
CH (Me) CH2SC (O) Me Me
CH (Me) CH2SC (O) (D1-108a) Me
CH (Me) CH2S (O) Me Me
CH (Me) CH2S (O) Et Me
CH (Me) CH2S (O) Pr-n Me
CH (Me) CH2S (O) Pr-i Me
CH (Me) CH2S (O) Bu-n Me
CH (Me) CH2S (O) Bu-i Me
CH (Me) CH2S (O) Bu-t Me
CH (Me) CH2S (O) Pen-n Me
CH (Me) CH2S (O) Hex-n Me
CH (Me) CH2S (O) Pr-c Me
CH (Me) CH2S (O) Bu-c Me
CH (Me) CH2S (O) Pen-c Me
CH (Me) CH2S (O) Hex-c Me
CH (Me) CH2S (O) CH2CH = CH2                   Me
CH (Me) CH2S (O) CH2C Three CH Me
CH (Me) CH2S (O) CF2H Me
CH (Me) CH2S (O) CFThree                        Me
CH (Me) CH2S (O) CF2Cl Me
CH (Me) CH2S (O) CH2CFThree                     Me
CH (Me) CH2S (O) {D1-108c} Me
CH (Me) CH2S (O) CH2CH2CN Me
CH (Me) CH2S (O) CH2CH2CFThree                   Me
CH (Me) CH2S (O) CH2(D1-103a) Me
CH (Me) CH2S (O) CH2CH2OMe Me
CH (Me) CH2S (O) CH2CH2OEt Me
CH (Me) CH2S (O) CH2(D1-32a) Me
CH (Me) CH2S (O) CH2(D1-33a) Me
CH (Me) CH2S (O) CH2(D1-34a) Me
CH (Me) CH2S (O) {D1-32b (X1= 5-CFThree)} Me
CH (Me) CH2S (O) CH2(D1-81a) Me
CH (Me) CH2S (O) CH2(D1-82a) Me
CH (Me) CH2S (O) CH2(D1-84a) Me
CH (Me) CH2S (O) CH2(D1-85a) Me
CH (Me) CH2S (O) CH2(D1-87a) Me
CH (Me) CH2S (O) CH2(D1-95a) Me
CH (Me) CH2S (O) CH2(D1-96a) Me
CH (Me) CH2S (O) CH2(D1-98a) Me
CH (Me) CH2S (O)2Me Me
CH (Me) CH2S (O)2Et Me
CH (Me) CH2S (O)2Pr-n Me
CH (Me) CH2S (O)2Pr-i Me
CH (Me) CH2S (O)2Bu-n Me
CH (Me) CH2S (O)2Bu-i Me
CH (Me) CH2S (O)2Bu-t Me
CH (Me) CH2S (O)2Pen-n Me
CH (Me) CH2S (O)2Hex-n Me
CH (Me) CH2S (O)2Pr-c Me
CH (Me) CH2S (O)2Bu-c Me
CH (Me) CH2S (O)2Pen-c Me
CH (Me) CH2S (O)2Hex-c Me
CH (Me) CH2S (O)2CH2CH = CH2                  Me
CH (Me) CH2S (O)2CH2C Three CH Me
CH (Me) CH2S (O)2CF2H Me
CH (Me) CH2S (O)2CFThree                        Me
CH (Me) CH2S (O)2CF2Cl Me
CH (Me) CH2S (O)2CH2CFThree                     Me
CH (Me) CH2S (O)2{D1-108c} Me
CH (Me) CH2S (O)2CH2CH2CN Me
CH (Me) CH2S (O)2CH2CH2CFThree                   Me
CH (Me) CH2S (O)2CH2(D1-103a) Me
CH (Me) CH2S (O)2CH2CH2OMe Me
CH (Me) CH2S (O)2CH2CH2OEt Me
CH (Me) CH2S (O)2CH2(D1-32a) Me
CH (Me) CH2S (O)2CH2(D1-33a) Me
CH (Me) CH2S (O)2CH2(D1-34a) Me
CH (Me) CH2S (O)2{D1-32b (X1= 5-CFThree)} Me
CH (Me) CH2S (O)2CH2(D1-81a) Me
CH (Me) CH2S (O)2CH2(D1-82a) Me
CH (Me) CH2S (O)2CH2(D1-84a) Me
CH (Me) CH2S (O)2CH2(D1-85a) Me
CH (Me) CH2S (O)2CH2(D1-87a) Me
CH (Me) CH2S (O)2CH2(D1-95a) Me
CH (Me) CH2S (O)2CH2(D1-96a) Me
CH (Me) CH2S (O)2CH2(D1-98a) Me
CH (Me) CH (Me) SH Me
CH (Me) CH (Me) SMe Me
CH (Me) CH (Me) SEt Me
CH (Me) CH (Me) SPr-n Me
CH (Me) CH (Me) SPr-i Me
CH (Me) CH (Me) SBu-n Me
CH (Me) CH (Me) SBu-i Me
CH (Me) CH (Me) SBu-t Me
CH (Me) CH (Me) SPen-n Me
CH (Me) CH (Me) SHex-n Me
CH (Me) CH (Me) SPr-c Me
CH (Me) CH (Me) SBu-c Me
CH (Me) CH (Me) SPen-c Me
CH (Me) CH (Me) SHex-c Me
CH (Me) CH (Me) SCH2CH = CH2                    Me
CH (Me) CH (Me) SCH2C Three CH Me
CH (Me) CH (Me) SCF2H Me
CH (Me) CH (Me) SCFThree                         Me
CH (Me) CH (Me) SCF2Cl Me
CH (Me) CH (Me) SCH2CFThree                       Me
CH (Me) CH (Me) S {D1-108c} Me
CH (Me) CH (Me) SCH2CH2CN Me
CH (Me) CH (Me) SCH2CH2CFThree                    Me
CH (Me) CH (Me) SCH2(D1-103a) Me
CH (Me) CH (Me) SCH2CH2OMe Me
CH (Me) CH (Me) SCH2CH2OEt Me
CH (Me) CH (Me) SCH2(D1-32a) Me
CH (Me) CH (Me) SCH2(D1-33a) Me
CH (Me) CH (Me) SCH2(D1-34a) Me
CH (Me) CH (Me) S {D1-32b (X1= 5-CFThree)} Me
CH (Me) CH (Me) SCH2(D1-81a) Me
CH (Me) CH (Me) SCH2(D1-82a) Me
CH (Me) CH (Me) SCH2(D1-84a) Me
CH (Me) CH (Me) SCH2(D1-85a) Me
CH (Me) CH (Me) SCH2(D1-87a) Me
CH (Me) CH (Me) SCH2(D1-95a) Me
CH (Me) CH (Me) SCH2(D1-96a) Me
CH (Me) CH (Me) SCH2(D1-98a) Me
CH (Me) CH (Me) SC (O) Me Me
CH (Me) CH (Me) SC (O) (D1-108a) Me
CH (Me) CH (Me) S (O) Me Me
CH (Me) CH (Me) S (O) Et Me
CH (Me) CH (Me) S (O) Pr-n Me
CH (Me) CH (Me) S (O) Pr-i Me
CH (Me) CH (Me) S (O) Bu-n Me
CH (Me) CH (Me) S (O) Bu-i Me
CH (Me) CH (Me) S (O) Bu-t Me
CH (Me) CH (Me) S (O) Pen-n Me
CH (Me) CH (Me) S (O) Hex-n Me
CH (Me) CH (Me) S (O) Pr-c Me
CH (Me) CH (Me) S (O) Bu-c Me
CH (Me) CH (Me) S (O) Pen-c Me
CH (Me) CH (Me) S (O) Hex-c Me
CH (Me) CH (Me) S (O) CH2CH = CH2                 Me
CH (Me) CH (Me) S (O) CH2C Three CH Me
CH (Me) CH (Me) S (O) CF2H Me
CH (Me) CH (Me) S (O) CFThree                      Me
CH (Me) CH (Me) S (O) CF2Cl Me
CH (Me) CH (Me) S (O) CH2CFThree                   Me
CH (Me) CH (Me) S (O) {D1-108c} Me
CH (Me) CH (Me) S (O) CH2CH2CN Me
CH (Me) CH (Me) S (O) CH2CH2CFThree                Me
CH (Me) CH (Me) S (O) CH2(D1-103a) Me
CH (Me) CH (Me) S (O) CH2CH2OMe Me
CH (Me) CH (Me) S (O) CH2CH2OEt Me
CH (Me) CH (Me) S (O) CH2(D1-32a) Me
CH (Me) CH (Me) S (O) CH2(D1-33a) Me
CH (Me) CH (Me) S (O) CH2(D1-34a) Me
CH (Me) CH (Me) S (O) {D1-32b (X1= 5-CFThree)} Me
CH (Me) CH (Me) S (O) CH2(D1-81a) Me
CH (Me) CH (Me) S (O) CH2(D1-82a) Me
CH (Me) CH (Me) S (O) CH2(D1-84a) Me
CH (Me) CH (Me) S (O) CH2(D1-85a) Me
CH (Me) CH (Me) S (O) CH2(D1-87a) Me
CH (Me) CH (Me) S (O) CH2(D1-95a) Me
CH (Me) CH (Me) S (O) CH2(D1-96a) Me
CH (Me) CH (Me) S (O) CH2(D1-98a) Me
CH (Me) CH (Me) S (O)2Me Me
CH (Me) CH (Me) S (O)2Et Me
CH (Me) CH (Me) S (O)2Pr-n Me
CH (Me) CH (Me) S (O)2Pr-i Me
CH (Me) CH (Me) S (O)2Bu-n Me
CH (Me) CH (Me) S (O)2Bu-i Me
CH (Me) CH (Me) S (O)2Bu-t Me
CH (Me) CH (Me) S (O)2Pen-n Me
CH (Me) CH (Me) S (O)2Hex-n Me
CH (Me) CH (Me) S (O)2Pr-c Me
CH (Me) CH (Me) S (O)2Bu-c Me
CH (Me) CH (Me) S (O)2Pen-c Me
CH (Me) CH (Me) S (O)2Hex-c Me
CH (Me) CH (Me) S (O)2CH2CH = CH2                Me
CH (Me) CH (Me) S (O)2CH2C Three CH Me
CH (Me) CH (Me) S (O)2CF2H Me
CH (Me) CH (Me) S (O)2CFThree                      Me
CH (Me) CH (Me) S (O)2CF2Cl Me
CH (Me) CH (Me) S (O)2CH2CFThree                   Me
CH (Me) CH (Me) S (O)2{D1-108c} Me
CH (Me) CH (Me) S (O)2CH2CH2CN Me
CH (Me) CH (Me) S (O)2CH2CH2CFThree                Me
CH (Me) CH (Me) S (O)2CH2(D1-103a) Me
CH (Me) CH (Me) S (O)2CH2CH2OMe Me
CH (Me) CH (Me) S (O)2CH2CH2OEt Me
CH (Me) CH (Me) S (O)2CH2(D1-32a) Me
CH (Me) CH (Me) S (O)2CH2(D1-33a) Me
CH (Me) CH (Me) S (O)2CH2(D1-34a) Me
CH (Me) CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} Me
CH (Me) CH (Me) S (O)2CH2(D1-81a) Me
CH (Me) CH (Me) S (O)2CH2(D1-82a) Me
CH (Me) CH (Me) S (O)2CH2(D1-84a) Me
CH (Me) CH (Me) S (O)2CH2(D1-85a) Me
CH (Me) CH (Me) S (O)2CH2(D1-87a) Me
CH (Me) CH (Me) S (O)2CH2(D1-95a) Me
CH (Me) CH (Me) S (O)2CH2(D1-96a) Me
CH (Me) CH (Me) S (O)2CH2(D1-98a) Me
CH2CH (Me) SH Me
CH2CH (Me) SMe Me
CH2CH (Me) SEt Me
CH2CH (Me) SPr-n Me
CH2CH (Me) SPr-i Me
CH2CH (Me) SBu-n Me
CH2CH (Me) SBu-i Me
CH2CH (Me) SBu-t Me
CH2CH (Me) SPen-n Me
CH2CH (Me) SHex-n Me
CH2CH (Me) SPr-c Me
CH2CH (Me) SBu-c Me
CH2CH (Me) SPen-c Me
CH2CH (Me) SHex-c Me
CH2CH (Me) SCH2CH = CH2                       Me
CH2CH (Me) SCH2C Three CH Me
CH2CH (Me) SCF2H Me
CH2CH (Me) SCFThree                            Me
CH2CH (Me) SCF2Cl Me
CH2CH (Me) SCH2CFThree                          Me
CH2CH (Me) S {D1-108c} Me
CH2CH (Me) SCH2CH2CN Me
CH2CH (Me) SCH2CH2CFThree                      Me
CH2CH (Me) SCH2(D1-103a) Me
CH2CH (Me) SCH2CH2OMe Me
CH2CH (Me) SCH2CH2OEt Me
CH2CH (Me) SCH2(D1-32a) Me
CH2CH (Me) SCH2(D1-33a) Me
CH2CH (Me) SCH2(D1-34a) Me
CH2CH (Me) S {D1-32b (X1= 5-CFThree)} Me
CH2CH (Me) SCH2(D1-81a) Me
CH2CH (Me) SCH2(D1-82a) Me
CH2CH (Me) SCH2(D1-84a) Me
CH2CH (Me) SCH2(D1-85a) Me
CH2CH (Me) SCH2(D1-87a) Me
CH2CH (Me) SCH2(D1-95a) Me
CH2CH (Me) SCH2(D1-96a) Me
CH2CH (Me) SCH2(D1-98a) Me
CH2CH (Me) SC (O) Me Me
CH2CH (Me) SC (O) (D1-108a) Me
CH2CH (Me) S (O) Me Me
CH2CH (Me) S (O) Et Me
CH2CH (Me) S (O) Pr-n Me
CH2CH (Me) S (O) Pr-i Me
CH2CH (Me) S (O) Bu-n Me
CH2CH (Me) S (O) Bu-i Me
CH2CH (Me) S (O) Bu-t Me
CH2CH (Me) S (O) Pen-n Me
CH2CH (Me) S (O) Hex-n Me
CH2CH (Me) S (O) Pr-c Me
CH2CH (Me) S (O) Bu-c Me
CH2CH (Me) S (O) Pen-c Me
CH2CH (Me) S (O) Hex-c Me
CH2CH (Me) S (O) CH2CH = CH2                    Me
CH2CH (Me) S (O) CH2C Three CH Me
CH2CH (Me) S (O) CF2H Me
CH2CH (Me) S (O) CFThree                        Me
CH2CH (Me) S (O) CF2Cl Me
CH2CH (Me) S (O) CH2CFThree                      Me
CH2CH (Me) S (O) {D1-108c} Me
CH2CH (Me) S (O) CH2CH2CN Me
CH2CH (Me) S (O) CH2CH2CFThree                    Me
CH2CH (Me) S (O) CH2(D1-103a) Me
CH2CH (Me) S (O) CH2CH2OMe Me
CH2CH (Me) S (O) CH2CH2OEt Me
CH2CH (Me) S (O) CH2(D1-32a) Me
CH2CH (Me) S (O) CH2(D1-33a) Me
CH2CH (Me) S (O) CH2(D1-34a) Me
CH2CH (Me) S (O) {D1-32b (X1= 5-CFThree)} Me
CH2CH (Me) S (O) CH2(D1-81a) Me
CH2CH (Me) S (O) CH2(D1-82a) Me
CH2CH (Me) S (O) CH2(D1-84a) Me
CH2CH (Me) S (O) CH2(D1-85a) Me
CH2CH (Me) S (O) CH2(D1-87a) Me
CH2CH (Me) S (O) CH2(D1-95a) Me
CH2CH (Me) S (O) CH2(D1-96a) Me
CH2CH (Me) S (O) CH2(D1-98a) Me
CH2CH (Me) S (O)2Me Me
CH2CH (Me) S (O)2Et Me
CH2CH (Me) S (O)2Pr-n Me
CH2CH (Me) S (O)2Pr-i Me
CH2CH (Me) S (O)2Bu-n Me
CH2CH (Me) S (O)2Bu-i Me
CH2CH (Me) S (O)2Bu-t Me
CH2CH (Me) S (O)2Pen-n Me
CH2CH (Me) S (O)2Hex-n Me
CH2CH (Me) S (O)2Pr-c Me
CH2CH (Me) S (O)2Bu-c Me
CH2CH (Me) S (O)2Pen-c Me
CH2CH (Me) S (O)2Hex-c Me
CH2CH (Me) S (O)2CH2CH = CH2                   Me
CH2CH (Me) S (O)2CH2C Three CH Me
CH2CH (Me) S (O)2CF2H Me
CH2CH (Me) S (O)2CFThree                         Me
CH2CH (Me) S (O)2CF2Cl Me
CH2CH (Me) S (O)2CH2CFThree                      Me
CH2CH (Me) S (O)2{D1-108c} Me
CH2CH (Me) S (O) 2CH2CH2CN Me
CH2CH (Me) S (O)2CH2CH2CFThree                    Me
CH2CH (Me) S (O)2CH2(D1-103a) Me
CH2CH (Me) S (O)2CH2CH2OMe Me
CH2CH (Me) S (O)2CH2CH2OEt Me
CH2CH (Me) S (O)2CH2(D1-32a) Me
CH2CH (Me) S (O)2CH2(D1-33a) Me
CH2CH (Me) S (O)2CH2(D1-34a) Me
CH2CH (Me) S (O)2{D1-32b (X1= 5-CFThree)} Me
CH2CH (Me) S (O)2CH2(D1-81a) Me
CH2CH (Me) S (O)2CH2(D1-82a) Me
CH2CH (Me) S (O)2CH2(D1-84a) Me
CH2CH (Me) S (O)2CH2(D1-85a) Me
CH2CH (Me) S (O)2CH2(D1-87a) Me
CH2CH (Me) S (O)2CH2(D1-95a) Me
CH2CH (Me) S (O)2CH2(D1-96a) Me
CH2CH (Me) S (O)2CH2(D1-98a) Me
C (O) OH Me
C (O) OMe Me
C (O) OEt Me
C (O) OPr-n Me
C (O) OPr-i Me
C (O) OBu-n Me
C (O) OBu-i Me
C (O) OBu-s Me
C (O) OBu-t Me
C (O) OPen-n Me
C (O) OHex-n Me
CHO Me
C (O) Me Me
C (O) Et Me
C (O) Pr-n Me
C (O) Pr-i Me
C (O) Bu-n Me
C (O) Bu-i Me
C (O) Bu-s Me
C (O) Bu-t Me
C (O) Pen-n Me
C (O) Hex-n Me
C (O) NHC (O) Me Me
C (O) NHMe Me
C (O) NHEt Me
C (O) NHPr-n Me
C (O) NHPr-i Me
C (O) NHBu-n Me
C (O) NHBu-i Me
C (O) NHBu-s Me
C (O) NHBu-t Me
C (O) NHPen-n Me
C (O) NHHex-n Me
CN Me
Ph Me
CH2Cl Me
CH2Br Me
CH2I Me
CH (Me) Cl Me
CH (Me) Br Me
CH (Me) I Me
CH (Et) Cl Me
CH (Et) Br Me
CH (Et) I Me
CH (n-Pr) Cl Me
CH (n-Pr) Br Me
CH (n-Pr) I Me
CH (i-Pr) Cl Me
CH (i-Pr) Br Me
CH (i-Pr) I Me
CH (n-Bu) Cl Me
CH (n-Bu) Br Me
CH (n-Bu) I Me
CH (CH2OMe) Cl Me
CH (CH2OMe) Br Me
CH (CH2OMe) I Me
CH (CH2CH = CH2) Cl Me
CH (CH2CH = CH2Br Me
CH (CH2CH = CH2) I Me
CH (CH2C3CH) Cl Me
CH (CH2C3CH) Br Me
CH (CH2C3CH) I Me
CH (Me) CH2Cl Me
CH (Me) CH2Br Me
CH (Me) CH2I Me
C (Me)2CH2Cl Me
C (Me)2CH2Br Me
C (Me)2CH2I Me
CH2SCH2(D1-81a) Me
CH2SCH2(D1-81a) Et
CH2SCH2(D1-81a) Pr-n
CH2SCH2(D1-81a) Pr-i
CH2SCH2(D1-81a) Pr-c
CH2SCH2(D1-81a) Bu-n
CH2SCH2(D1-81a) Bu-i
CH2SCH2(D1-81a) Bu-c
CH2SCH2(D1-81a) Bu-s
CH2SCH2(D1-81a) Bu-t
CH2SCH2(D1-81a) Pen-n
CH2SCH2(D1-81a) Pen-c
CH2SCH2(D1-81a) Hex-n
CH2SCH2(D1-81a) Hex-c
CH2SCH2(D1-81a) CH2Pr-c
CH2SCH2(D1-81a) CH2Bu-c
CH2SCH2(D1-81a) CH2Pen-c
CH2SCH2(D1-81a) CH2Hex-c
CH2SCH2(D1-81a) CH2CH = CH2
CH2SCH2(D1-81a) CH2CH = C (Cl)2
CH2SCH2(D1-81a) CH2C≡CH
CH2SCH2(D1-81a) CH2CN
CH2SCH2(D1-81a) CH2CFThree
CH2SCH2(D1-81a) CH2OMe
CH2SCH2(D1-81a) CH2OCFThree
CH2SCH2(D1-81a) CH2SMe
CH2SCH2(D1-81a) CH2S (O) Me
CH2SCH2(D1-81a) CH2S (O)2Me
CH2SCH2(D1-81a) CH2SCFThree
CH2SCH2(D1-81a) CH2S (O) CFThree
CH2SCH2(D1-81a) CH2S (O)2CFThree
CH2SCH2(D1-81a) CH2CH (OMe)2
CH2SCH2(D1-81a) CH2CH (SMe)2
CH2SCH2(D1-81a) CH2C (O) Me
CH2SCH2(D1-81a) CH2C (O) CFThree
CH2SCH2(D1-81a) CH2C (O) OMe
CH2SCH2(D1-81a) CH2(D1-32a)
CH2SCH2(D1-81a) CH2(D1-33a)
CH2SCH2(D1-81a) CH2(D1-34a)
CH2SCH2(D1-81a) CH2(D1-37a)
CH2SCH2(D1-81a) CH2(D1-81a)
CH2SCH2(D1-81a) CH2(D1-82a)
CH2SCH2(D1-81a) CH2(D1-84a)
CH2SCH2(D1-81a) CH2(D1-85a)
CH2SCH2(D1-81a) CH2(D1-87a)
CH2SCH2(D1-81a) CH2(D1-92a)
CH2SCH2(D1-81a) CH2(D1-93a)
CH2SCH2(D1-81a) CH2(D1-95a)
CH2SCH2(D1-81a) CH2(D1-96a)
CH2SCH2(D1-81a) CH2(D1-98a)
CH2SCH2(D1-81a) CH2(D1-108a)
CH2SCH2(D1-81a) CH2(D1-108b, Z = 2-Cl)
CH2SCH2(D1-81a) CH2(D1-108b, Z = 3-Me)
CH2SCH2(D1-81a) CH2(D1-108b, Z = 4-OMe)
CH2SCH2(D1-81a) CH2(D1-108b, Z = 2-SMe)
CH2SCH2(D1-81a) CH2(D1-108b, Z = 3-CFThree)
CH2SCH2(D1-81a) CH2(D1-108b, Z = 4-OCFThree)
CH2SCH2(D1-81a) CH2(D1-108b, Z = 2-SCFThree)
CH2SCH2(D1-81a) CH2CH2CN
CH2SCH2(D1-81a) CH2CH2CFThree
CH2SCH2(D1-81a) CH2CH2OMe
CH2SCH2(D1-81a) CH2CH2SMe
CH2SCH2(D1-81a) CH2CH2S (O) Me
CH2SCH2(D1-81a) CH2CH2S (O)2Me
CH2SCH2(D1-81a) D1-32a
CH2SCH2(D1-81a) D1-33a
CH2SCH2(D1-81a) D1-34a
CH2SCH2(D1-81a) D1-37a
CH2SCH2(D1-81a) D1-81a
CH2SCH2(D1-81a) D1-82a
CH2SCH2(D1-81a) D1-84a
CH2SCH2(D1-81a) D1-85a
CH2SCH2(D1-81a) D1-87a
CH2SCH2(D1-81a) D1-92a
CH2SCH2(D1-81a) D1-93a
CH2SCH2(D1-81a) D1-95a
CH2SCH2(D1-81a) D1-96a
CH2SCH2(D1-81a) D1-98a
CH2SCH2(D1-81a) D1-108a
CH2SCH2(D1-81a) D1-108b (Z = 2-Cl)
CH2SCH2(D1-81a) D1-108b (Z = 3-Me)
CH2SCH2(D1-81a) D1-108b (Z = 4-OMe)
CH2SCH2(D1-81a) D1-108b (Z = 2-SMe)
CH2SCH2(D1-81a) D1-108b (Z = 3-CFThree)
CH2SCH2(D1-81a) D1-108b (Z = 4-OCFThree)
CH2SCH2(D1-81a) D1-108b (Z = 2-SCFThree)
CH2SCH2(D1-81a) C (O) Me
CH2SCH2(D1-81a) C (O) CFThree
CH2SCH2(D1-81a) C (O) OMe
CH2S (O) CH2(D1-81a) Me
CH2S (O) CH2(D1-81a) Et
CH2S (O) CH2(D1-81a) Pr-n
CH2S (O) CH2(D1-81a) Pr-i
CH2S (O) CH2(D1-81a) Pr-c
CH2S (O) CH2(D1-81a) Bu-n
CH2S (O) CH2(D1-81a) Bu-i
CH2S (O) CH2(D1-81a) Bu-c
CH2S (O) CH2(D1-81a) Bu-s
CH2S (O) CH2(D1-81a) Bu-t
CH2S (O) CH2(D1-81a) Pen-n
CH2S (O) CH2(D1-81a) Pen-c
CH2S (O) CH2(D1-81a) Hex-n
CH2S (O) CH2(D1-81a) Hex-c
CH2S (O) CH2(D1-81a) CH2Pr-c
CH2S (O) CH2(D1-81a) CH2Bu-c
CH2S (O) CH2(D1-81a) CH2Pen-c
CH2S (O) CH2(D1-81a) CH2Hex-c
CH2S (O) CH2(D1-81a) CH2CH = CH2
CH2S (O) CH2(D1-81a) CH2CH = C (Cl)2
CH2S (O) CH2(D1-81a) CH2C≡CH
CH2S (O) CH2(D1-81a) CH2CN
CH2S (O) CH2(D1-81a) CH2CFThree
CH2S (O) CH2(D1-81a) CH2OMe
CH2S (O) CH2(D1-81a) CH2OCFThree
CH2S (O) CH2(D1-81a) CH2SMe
CH2S (O) CH2(D1-81a) CH2S (O) Me
CH2S (O) CH2(D1-81a) CH2S (O)2Me
CH2S (O) CH2(D1-81a) CH2SCFThree
CH2S (O) CH2(D1-81a) CH2S (O) CFThree
CH2S (O) CH2(D1-81a) CH2S (O)2CFThree
CH2S (O) CH2(D1-81a) CH2CH (OMe)2
CH2S (O) CH2(D1-81a) CH2CH (SMe)2
CH2S (O) CH2(D1-81a) CH2C (O) Me
CH2S (O) CH2(D1-81a) CH2C (O) CFThree
CH2S (O) CH2(D1-81a) CH2C (O) OMe
CH2S (O) CH2(D1-81a) CH2(D1-32a)
CH2S (O) CH2(D1-81a) CH2(D1-33a)
CH2S (O) CH2(D1-81a) CH2(D1-34a)
CH2S (O) CH2(D1-81a) CH2(D1-37a)
CH2S (O) CH2(D1-81a) CH2(D1-81a)
CH2S (O) CH2(D1-81a) CH2(D1-82a)
CH2S (O) CH2(D1-81a) CH2(D1-84a)
CH2S (O) CH2(D1-81a) CH2(D1-85a)
CH2S (O) CH2(D1-81a) CH2(D1-87a)
CH2S (O) CH2(D1-81a) CH2(D1-92a)
CH2S (O) CH2(D1-81a) CH2(D1-93a)
CH2S (O) CH2(D1-81a) CH2(D1-95a)
CH2S (O) CH2(D1-81a) CH2(D1-96a)
CH2S (O) CH2(D1-81a) CH2(D1-98a)
CH2S (O) CH2(D1-81a) CH2(D1-108a)
CH2S (O) CH2(D1-81a) CH2(D1-108b, Z = 2-Cl)
CH2S (O) CH2(D1-81a) CH2(D1-108b, Z = 3-Me)
CH2S (O) CH2(D1-81a) CH2(D1-108b, Z = 4-OMe)
CH2S (O) CH2(D1-81a) CH2(D1-108b, Z = 2-SMe)
CH2S (O) CH2(D1-81a) CH2(D1-108b, Z = 3-CFThree)
CH2S (O) CH2(D1-81a) CH2(D1-108b, Z = 4-OCFThree)
CH2S (O) CH2(D1-81a) CH2(D1-108b, Z = 2-SCFThree)
CH2S (O) CH2(D1-81a) CH2CH2CN
CH2S (O) CH2(D1-81a) CH2CH2CFThree
CH2S (O) CH2(D1-81a) CH2CH2OMe
CH2S (O) CH2(D1-81a) CH2CH2SMe
CH2S (O) CH2(D1-81a) CH2CH2S (O) Me
CH2S (O) CH2(D1-81a) CH2CH2S (O)2Me
CH2S (O) CH2(D1-81a) D1-32a
CH2S (O) CH2(D1-81a) D1-33a
CH2S (O) CH2(D1-81a) D1-34a
CH2S (O) CH2(D1-81a) D1-37a
CH2S (O) CH2(D1-81a) D1-81a
CH2S (O) CH2(D1-81a) D1-82a
CH2S (O) CH2(D1-81a) D1-84a
CH2S (O) CH2(D1-81a) D1-85a
CH2S (O) CH2(D1-81a) D1-87a
CH2S (O) CH2(D1-81a) D1-92a
CH2S (O) CH2(D1-81a) D1-93a
CH2S (O) CH2(D1-81a) D1-95a
CH2S (O) CH2(D1-81a) D1-96a
CH2S (O) CH2(D1-81a) D1-98a
CH2S (O) CH2(D1-81a) D1-108a
CH2S (O) CH2(D1-81a) D1-108b (Z = 2-Cl)
CH2S (O) CH2(D1-81a) D1-108b (Z = 3-Me)
CH2S (O) CH2(D1-81a) D1-108b (Z = 4-OMe)
CH2S (O) CH2(D1-81a) D1-108b (Z = 2-SMe)
CH2S (O) CH2(D1-81a) D1-108b (Z = 3-CFThree)
CH2S (O) CH2(D1-81a) D1-108b (Z = 4-OCFThree)
CH2S (O) CH2(D1-81a) D1-108b (Z = 2-SCFThree)
CH2S (O) CH2(D1-81a) C (O) Me
CH2S (O) CH2(D1-81a) C (O) CFThree
CH2S (O) CH2(D1-81a) C (O) OMe
CH2S (O)2CH2(D1-81a) Me
CH2S (O)2CH2(D1-81a) Et
CH2S (O)2CH2(D1-81a) Pr-n
CH2S (O)2CH2(D1-81a) Pr-i
CH2S (O)2CH2(D1-81a) Pr-c
CH2S (O)2CH2(D1-81a) Bu-n
CH2S (O)2CH2(D1-81a) Bu-i
CH2S (O)2CH2(D1-81a) Bu-c
CH2S (O)2CH2(D1-81a) Bu-s
CH2S (O)2CH2(D1-81a) Bu-t
CH2S (O)2CH2(D1-81a) Pen-n
CH2S (O)2CH2(D1-81a) Pen-c
CH2S (O)2CH2(D1-81a) Hex-n
CH2S (O)2CH2(D1-81a) Hex-c
CH2S (O)2CH2(D1-81a) CH2Pr-c
CH2S (O)2CH2(D1-81a) CH2Bu-c
CH2S (O)2CH2(D1-81a) CH2Pen-c
CH2S (O)2CH2(D1-81a) CH2Hex-c
CH2S (O)2CH2(D1-81a) CH2CH = CH2
CH2S (O)2CH2(D1-81a) CH2CH = C (Cl)2
CH2S (O)2CH2(D1-81a) CH2C≡CH
CH2S (O)2CH2(D1-81a) CH2CN
CH2S (O)2CH2(D1-81a) CH2CFThree
CH2S (O)2CH2(D1-81a) CH2OMe
CH2S (O)2CH2(D1-81a) CH2OCFThree
CH2S (O)2CH2(D1-81a) CH2SMe
CH2S (O)2CH2(D1-81a) CH2S (O) Me
CH2S (O)2CH2(D1-81a) CH2S (O)2Me
CH2S (O)2CH2(D1-81a) CH2SCFThree
CH2S (O)2CH2(D1-81a) CH2S (O) CFThree
CH2S (O)2CH2(D1-81a) CH2S (O)2CFThree
CH2S (O)2CH2(D1-81a) CH2CH (OMe)2
CH2S (O)2CH2(D1-81a) CH2CH (SMe)2
CH2S (O)2CH2(D1-81a) CH2C (O) Me
CH2S (O)2CH2(D1-81a) CH2C (O) CFThree
CH2S (O)2CH2(D1-81a) CH2C (O) OMe
CH2S (O)2CH2(D1-81a) CH2(D1-32a)
CH2S (O)2CH2(D1-81a) CH2(D1-33a)
CH2S (O)2CH2(D1-81a) CH2(D1-34a)
CH2S (O)2CH2(D1-81a) CH2(D1-37a)
CH2S (O)2CH2(D1-81a) CH2(D1-81a)
CH2S (O)2CH2(D1-81a) CH2(D1-82a)
CH2S (O)2CH2(D1-81a) CH2(D1-84a)
CH2S (O)2CH2(D1-81a) CH2(D1-85a)
CH2S (O)2CH2(D1-81a) CH2(D1-87a)
CH2S (O)2CH2(D1-81a) CH2(D1-92a)
CH2S (O)2CH2(D1-81a) CH2(D1-93a)
CH2S (O)2CH2(D1-81a) CH2(D1-95a)
CH2S (O)2CH2(D1-81a) CH2(D1-96a)
CH2S (O)2CH2(D1-81a) CH2(D1-98a)
CH2S (O)2CH2(D1-81a) CH2(D1-108a)
CH2S (O)2CH2(D1-81a) CH2(D1-108b, Z = 2-Cl)
CH2S (O)2CH2(D1-81a) CH2(D1-108b, Z = 3-Me)
CH2S (O)2CH2(D1-81a) CH2(D1-108b, Z = 4-OMe)
CH2S (O)2CH2(D1-81a) CH2(D1-108b, Z = 2-SMe)
CH2S (O)2CH2(D1-81a) CH2(D1-108b, Z = 3-CFThree)
CH2S (O)2CH2(D1-81a) CH2(D1-108b, Z = 4-OCFThree)
CH2S (O)2CH2(D1-81a) CH2(D1-108b, Z = 2-SCFThree)
CH2S (O)2CH2(D1-81a) CH2CH2CN
CH2S (O)2CH2(D1-81a) CH2CH2CFThree
CH2S (O)2CH2(D1-81a) CH2CH2OMe
CH2S (O)2CH2(D1-81a) CH2CH2SMe
CH2S (O)2CH2(D1-81a) CH2CH2S (O) Me
CH2S (O)2CH2(D1-81a) CH2CH2S (O)2Me
CH2S (O)2CH2(D1-81a) D1-32a
CH2S (O)2CH2(D1-81a) D1-33a
CH2S (O)2CH2(D1-81a) D1-34a
CH2S (O)2CH2(D1-81a) D1-37a
CH2S (O)2CH2(D1-81a) D1-81a
CH2S (O)2CH2(D1-81a) D1-82a
CH2S (O)2CH2(D1-81a) D1-84a
CH2S (O)2CH2(D1-81a) D1-85a
CH2S (O)2CH2(D1-81a) D1-87a
CH2S (O)2CH2(D1-81a) D1-92a
CH2S (O)2CH2(D1-81a) D1-93a
CH2S (O)2CH2(D1-81a) D1-95a
CH2S (O)2CH2(D1-81a) D1-96a
CH2S (O)2CH2(D1-81a) D1-98a
CH2S (O)2CH2(D1-81a) D1-108a
CH2S (O)2CH2(D1-81a) D1-108b (Z = 2-Cl)
CH2S (O)2CH2(D1-81a) D1-108b (Z = 3-Me)
CH2S (O)2CH2(D1-81a) D1-108b (Z = 4-OMe)
CH2S (O)2CH2(D1-81a) D1-108b (Z = 2-SMe)
CH2S (O)2CH2(D1-81a) D1-108b (Z = 3-CFThree)
CH2S (O)2CH2(D1-81a) D1-108b (Z = 4-OCFThree)
CH2S (O)2CH2(D1-81a) D1-108b (Z = 2-SCFThree)
CH2S (O)2CH2(D1-81a) C (O) Me
CH2S (O)2CH2(D1-81a) C (O) CFThree
CH2S (O)2CH2(D1-81a) C (O) OMe
CH (Me) SCH2(D1-81a) Me
CH (Me) SCH2(D1-81a) Et
CH (Me) SCH2(D1-81a) Pr-n
CH (Me) SCH2(D1-81a) Pr-i
CH (Me) SCH2(D1-81a) Pr-c
CH (Me) SCH2(D1-81a) Bu-n
CH (Me) SCH2(D1-81a) Bu-i
CH (Me) SCH2(D1-81a) Bu-c
CH (Me) SCH2(D1-81a) Bu-s
CH (Me) SCH2(D1-81a) Bu-t
CH (Me) SCH2(D1-81a) Pen-n
CH (Me) SCH2(D1-81a) Pen-c
CH (Me) SCH2(D1-81a) Hex-n
CH (Me) SCH2(D1-81a) Hex-c
CH (Me) SCH2(D1-81a) CH2Pr-c
CH (Me) SCH2(D1-81a) CH2Bu-c
CH (Me) SCH2(D1-81a) CH2Pen-c
CH (Me) SCH2(D1-81a) CH2Hex-c
CH (Me) SCH2(D1-81a) CH2CH = CH2
CH (Me) SCH2(D1-81a) CH2CH = C (Cl)2
CH (Me) SCH2(D1-81a) CH2C≡CH
CH (Me) SCH2(D1-81a) CH2CN
CH (Me) SCH2(D1-81a) CH2CFThree
CH (Me) SCH2(D1-81a) CH2OMe
CH (Me) SCH2(D1-81a) CH2OCFThree
CH (Me) SCH2(D1-81a) CH2SMe
CH (Me) SCH2(D1-81a) CH2S (O) Me
CH (Me) SCH2(D1-81a) CH2S (O)2Me
CH (Me) SCH2(D1-81a) CH2SCFThree
CH (Me) SCH2(D1-81a) CH2S (O) CFThree
CH (Me) SCH2(D1-81a) CH2S (O)2CFThree
CH (Me) SCH2(D1-81a) CH2CH (OMe)2
CH (Me) SCH2(D1-81a) CH2CH (SMe)2
CH (Me) SCH2(D1-81a) CH2C (O) Me
CH (Me) SCH2(D1-81a) CH2C (O) CFThree
CH (Me) SCH2(D1-81a) CH2C (O) OMe
CH (Me) SCH2(D1-81a) CH2(D1-32a)
CH (Me) SCH2(D1-81a) CH2(D1-33a)
CH (Me) SCH2(D1-81a) CH2(D1-34a)
CH (Me) SCH2(D1-81a) CH2(D1-37a)
CH (Me) SCH2(D1-81a) CH2(D1-81a)
CH (Me) SCH2(D1-81a) CH2(D1-82a)
CH (Me) SCH2(D1-81a) CH2(D1-84a)
CH (Me) SCH2(D1-81a) CH2(D1-85a)
CH (Me) SCH2(D1-81a) CH2(D1-87a)
CH (Me) SCH2(D1-81a) CH2(D1-92a)
CH (Me) SCH2(D1-81a) CH2(D1-93a)
CH (Me) SCH2(D1-81a) CH2(D1-95a)
CH (Me) SCH2(D1-81a) CH2(D1-96a)
CH (Me) SCH2(D1-81a) CH2(D1-98a)
CH (Me) SCH2(D1-81a) CH2(D1-108a)
CH (Me) SCH2(D1-81a) CH2(D1-108b, Z = 2-Cl)
CH (Me) SCH2(D1-81a) CH2(D1-108b, Z = 3-Me)
CH (Me) SCH2(D1-81a) CH2(D1-108b, Z = 4-OMe)
CH (Me) SCH2(D1-81a) CH2(D1-108b, Z = 2-SMe)
CH (Me) SCH2(D1-81a) CH2(D1-108b, Z = 3-CFThree)
CH (Me) SCH2(D1-81a) CH2(D1-108b, Z = 4-OCFThree)
CH (Me) SCH2(D1-81a) CH2(D1-108b, Z = 2-SCFThree)
CH (Me) SCH2(D1-81a) CH2CH2CN
CH (Me) SCH2(D1-81a) CH2CH2CFThree
CH (Me) SCH2(D1-81a) CH2CH2OMe
CH (Me) SCH2(D1-81a) CH2CH2SMe
CH (Me) SCH2(D1-81a) CH2CH2S (O) Me
CH (Me) SCH2(D1-81a) CH2CH2S (O)2Me
CH (Me) SCH2(D1-81a) D1-32a
CH (Me) SCH2(D1-81a) D1-33a
CH (Me) SCH2(D1-81a) D1-34a
CH (Me) SCH2(D1-81a) D1-37a
CH (Me) SCH2(D1-81a) D1-81a
CH (Me) SCH2(D1-81a) D1-82a
CH (Me) SCH2(D1-81a) D1-84a
CH (Me) SCH2(D1-81a) D1-85a
CH (Me) SCH2(D1-81a) D1-87a
CH (Me) SCH2(D1-81a) D1-92a
CH (Me) SCH2(D1-81a) D1-93a
CH (Me) SCH2(D1-81a) D1-95a
CH (Me) SCH2(D1-81a) D1-96a
CH (Me) SCH2(D1-81a) D1-98a
CH (Me) SCH2(D1-81a) D1-108a
CH (Me) SCH2(D1-81a) D1-108b (Z = 2-Cl)
CH (Me) SCH2(D1-81a) D1-108b (Z = 3-Me)
CH (Me) SCH2(D1-81a) D1-108b (Z = 4-OMe)
CH (Me) SCH2(D1-81a) D1-108b (Z = 2-SMe)
CH (Me) SCH2(D1-81a) D1-108b (Z = 3-CFThree)
CH (Me) SCH2(D1-81a) D1-108b (Z = 4-OCFThree)
CH (Me) SCH2(D1-81a) D1-108b (Z = 2-SCFThree)
CH (Me) SCH2(D1-81a) C (O) Me
CH (Me) SCH2(D1-81a) C (O) CFThree
CH (Me) SCH2(D1-81a) C (O) OMe
CH (Me) S (O) CH2(D1-81a) Me
CH (Me) S (O) CH2(D1-81a) Et
CH (Me) S (O) CH2(D1-81a) Pr-n
CH (Me) S (O) CH2(D1-81a) Pr-i
CH (Me) S (O) CH2(D1-81a) Pr-c
CH (Me) S (O) CH2(D1-81a) Bu-n
CH (Me) S (O) CH2(D1-81a) Bu-i
CH (Me) S (O) CH2(D1-81a) Bu-c
CH (Me) S (O) CH2(D1-81a) Bu-s
CH (Me) S (O) CH2(D1-81a) Bu-t
CH (Me) S (O) CH2(D1-81a) Pen-n
CH (Me) S (O) CH2(D1-81a) Pen-c
CH (Me) S (O) CH2(D1-81a) Hex-n
CH (Me) S (O) CH2(D1-81a) Hex-c
CH (Me) S (O) CH2(D1-81a) CH2Pr-c
CH (Me) S (O) CH2(D1-81a) CH2Bu-c
CH (Me) S (O) CH2(D1-81a) CH2Pen-c
CH (Me) S (O) CH2(D1-81a) CH2Hex-c
CH (Me) S (O) CH2(D1-81a) CH2CH = CH2
CH (Me) S (O) CH2(D1-81a) CH2CH = C (Cl)2
CH (Me) S (O) CH2(D1-81a) CH2C≡CH
CH (Me) S (O) CH2(D1-81a) CH2CN
CH (Me) S (O) CH2(D1-81a) CH2CFThree
CH (Me) S (O) CH2(D1-81a) CH2OMe
CH (Me) S (O) CH2(D1-81a) CH2OCFThree
CH (Me) S (O) CH2(D1-81a) CH2SMe
CH (Me) S (O) CH2(D1-81a) CH2S (O) Me
CH (Me) S (O) CH2(D1-81a) CH2S (O)2Me
CH (Me) S (O) CH2(D1-81a) CH2SCFThree
CH (Me) S (O) CH2(D1-81a) CH2S (O) CFThree
CH (Me) S (O) CH2(D1-81a) CH2S (O)2CFThree
CH (Me) S (O) CH2(D1-81a) CH2CH (OMe)2
CH (Me) S (O) CH2(D1-81a) CH2CH (SMe)2
CH (Me) S (O) CH2(D1-81a) CH2C (O) Me
CH (Me) S (O) CH2(D1-81a) CH2C (O) CFThree
CH (Me) S (O) CH2(D1-81a) CH2C (O) OMe
CH (Me) S (O) CH2(D1-81a) CH2(D1-32a)
CH (Me) S (O) CH2(D1-81a) CH2(D1-33a)
CH (Me) S (O) CH2(D1-81a) CH2(D1-34a)
CH (Me) S (O) CH2(D1-81a) CH2(D1-37a)
CH (Me) S (O) CH2(D1-81a) CH2(D1-81a)
CH (Me) S (O) CH2(D1-81a) CH2(D1-82a)
CH (Me) S (O) CH2(D1-81a) CH2(D1-84a)
CH (Me) S (O) CH2(D1-81a) CH2(D1-85a)
CH (Me) S (O) CH2(D1-81a) CH2(D1-87a)
CH (Me) S (O) CH2(D1-81a) CH2(D1-92a)
CH (Me) S (O) CH2(D1-81a) CH2(D1-93a)
CH (Me) S (O) CH2(D1-81a) CH2(D1-95a)
CH (Me) S (O) CH2(D1-81a) CH2(D1-96a)
CH (Me) S (O) CH2(D1-81a) CH2(D1-98a)
CH (Me) S (O) CH2(D1-81a) CH2(D1-108a)
CH (Me) S (O) CH2(D1-81a) CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O) CH2(D1-81a) CH2(D1-108b, Z = 3-Me)
CH (Me) S (O) CH2(D1-81a) CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O) CH2(D1-81a) CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O) CH2(D1-81a) CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O) CH2(D1-81a) CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O) CH2(D1-81a) CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O) CH2(D1-81a) CH2CH2CN
CH (Me) S (O) CH2(D1-81a) CH2CH2CFThree
CH (Me) S (O) CH2(D1-81a) CH2CH2OMe
CH (Me) S (O) CH2(D1-81a) CH2CH2SMe
CH (Me) S (O) CH2(D1-81a) CH2CH2S (O) Me
CH (Me) S (O) CH2(D1-81a) CH2CH2S (O)2Me
CH (Me) S (O) CH2(D1-81a) D1-32a
CH (Me) S (O) CH2(D1-81a) D1-33a
CH (Me) S (O) CH2(D1-81a) D1-34a
CH (Me) S (O) CH2(D1-81a) D1-37a
CH (Me) S (O) CH2(D1-81a) D1-81a
CH (Me) S (O) CH2(D1-81a) D1-82a
CH (Me) S (O) CH2(D1-81a) D1-84a
CH (Me) S (O) CH2(D1-81a) D1-85a
CH (Me) S (O) CH2(D1-81a) D1-87a
CH (Me) S (O) CH2(D1-81a) D1-92a
CH (Me) S (O) CH2(D1-81a) D1-93a
CH (Me) S (O) CH2(D1-81a) D1-95a
CH (Me) S (O) CH2(D1-81a) D1-96a
CH (Me) S (O) CH2(D1-81a) D1-98a
CH (Me) S (O) CH2(D1-81a) D1-108a
CH (Me) S (O) CH2(D1-81a) D1-108b (Z = 2-Cl)
CH (Me) S (O) CH2(D1-81a) D1-108b (Z = 3-Me)
CH (Me) S (O) CH2(D1-81a) D1-108b (Z = 4-OMe)
CH (Me) S (O) CH2(D1-81a) D1-108b (Z = 2-SMe)
CH (Me) S (O) CH2(D1-81a) D1-108b (Z = 3-CFThree)
CH (Me) S (O) CH2(D1-81a) D1-108b (Z = 4-OCFThree)
CH (Me) S (O) CH2(D1-81a) D1-108b (Z = 2-SCFThree)
CH (Me) S (O) CH2(D1-81a) C (O) Me
CH (Me) S (O) CH2(D1-81a) C (O) CFThree
CH (Me) S (O) CH2(D1-81a) C (O) OMe
CH (Me) S (O)2CH2(D1-81a) Me
CH (Me) S (O)2CH2(D1-81a) Et
CH (Me) S (O)2CH2(D1-81a) Pr-n
CH (Me) S (O)2CH2(D1-81a) Pr-i
CH (Me) S (O)2CH2(D1-81a) Pr-c
CH (Me) S (O)2CH2(D1-81a) Bu-n
CH (Me) S (O)2CH2(D1-81a) Bu-i
CH (Me) S (O)2CH2(D1-81a) Bu-c
CH (Me) S (O)2CH2(D1-81a) Bu-s
CH (Me) S (O)2CH2(D1-81a) Bu-t
CH (Me) S (O)2CH2(D1-81a) Pen-n
CH (Me) S (O)2CH2(D1-81a) Pen-c
CH (Me) S (O)2CH2(D1-81a) Hex-n
CH (Me) S (O)2CH2(D1-81a) Hex-c
CH (Me) S (O)2CH2(D1-81a) CH2Pr-c
CH (Me) S (O)2CH2(D1-81a) CH2Bu-c
CH (Me) S (O)2CH2(D1-81a) CH2Pen-c
CH (Me) S (O)2CH2(D1-81a) CH2Hex-c
CH (Me) S (O)2CH2(D1-81a) CH2CH = CH2
CH (Me) S (O)2CH2(D1-81a) CH2CH = C (Cl)2
CH (Me) S (O)2CH2(D1-81a) CH2C≡CH
CH (Me) S (O)2CH2(D1-81a) CH2CN
CH (Me) S (O)2CH2(D1-81a) CH2CFThree
CH (Me) S (O)2CH2(D1-81a) CH2OMe
CH (Me) S (O)2CH2(D1-81a) CH2OCFThree
CH (Me) S (O)2CH2(D1-81a) CH2SMe
CH (Me) S (O)2CH2(D1-81a) CH2S (O) Me
CH (Me) S (O)2CH2(D1-81a) CH2S (O)2Me
CH (Me) S (O)2CH2(D1-81a) CH2SCFThree
CH (Me) S (O)2CH2(D1-81a) CH2S (O) CFThree
CH (Me) S (O)2CH2(D1-81a) CH2S (O)2CFThree
CH (Me) S (O)2CH2(D1-81a) CH2CH (OMe)2
CH (Me) S (O)2CH2(D1-81a) CH2CH (SMe)2
CH (Me) S (O)2CH2(D1-81a) CH2C (O) Me
CH (Me) S (O)2CH2(D1-81a) CH2C (O) CFThree
CH (Me) S (O)2CH2(D1-81a) CH2C (O) OMe
CH (Me) S (O)2CH2(D1-81a) CH2(D1-32a)
CH (Me) S (O)2CH2(D1-81a) CH2(D1-33a)
CH (Me) S (O)2CH2(D1-81a) CH2(D1-34a)
CH (Me) S (O)2CH2(D1-81a) CH2(D1-37a)
CH (Me) S (O)2CH2(D1-81a) CH2(D1-81a)
CH (Me) S (O)2CH2(D1-81a) CH2(D1-82a)
CH (Me) S (O)2CH2(D1-81a) CH2(D1-84a)
CH (Me) S (O)2CH2(D1-81a) CH2(D1-85a)
CH (Me) S (O)2CH2(D1-81a) CH2(D1-87a)
CH (Me) S (O)2CH2(D1-81a) CH2(D1-92a)
CH (Me) S (O)2CH2(D1-81a) CH2(D1-93a)
CH (Me) S (O)2CH2(D1-81a) CH2(D1-95a)
CH (Me) S (O)2CH2(D1-81a) CH2(D1-96a)
CH (Me) S (O)2CH2(D1-81a) CH2(D1-98a)
CH (Me) S (O)2CH2(D1-81a) CH2(D1-108a)
CH (Me) S (O)2CH2(D1-81a) CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O)2CH2(D1-81a) CH2(D1-108b, Z = 3-Me)
CH (Me) S (O)2CH2(D1-81a) CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O)2CH2(D1-81a) CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O)2CH2(D1-81a) CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O)2CH2(D1-81a) CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O)2CH2(D1-81a) CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O)2CH2(D1-81a) CH2CH2CN
CH (Me) S (O)2CH2(D1-81a) CH2CH2CFThree
CH (Me) S (O)2CH2(D1-81a) CH2CH2OMe
CH (Me) S (O)2CH2(D1-81a) CH2CH2SMe
CH (Me) S (O)2CH2(D1-81a) CH2CH2S (O) Me
CH (Me) S (O)2CH2(D1-81a) CH2CH2S (O)2Me
CH (Me) S (O)2CH2(D1-81a) D1-32a
CH (Me) S (O)2CH2(D1-81a) D1-33a
CH (Me) S (O)2CH2(D1-81a) D1-34a
CH (Me) S (O)2CH2(D1-81a) D1-37a
CH (Me) S (O)2CH2(D1-81a) D1-81a
CH (Me) S (O)2CH2(D1-81a) D1-82a
CH (Me) S (O)2CH2(D1-81a) D1-84a
CH (Me) S (O)2CH2(D1-81a) D1-85a
CH (Me) S (O)2CH2(D1-81a) D1-87a
CH (Me) S (O)2CH2(D1-81a) D1-92a
CH (Me) S (O)2CH2(D1-81a) D1-93a
CH (Me) S (O)2CH2(D1-81a) D1-95a
CH (Me) S (O)2CH2(D1-81a) D1-96a
CH (Me) S (O)2CH2(D1-81a) D1-98a
CH (Me) S (O)2CH2(D1-81a) D1-108a
CH (Me) S (O)2CH2(D1-81a) D1-108b (Z = 2-Cl)
CH (Me) S (O)2CH2(D1-81a) D1-108b (Z = 3-Me)
CH (Me) S (O)2CH2(D1-81a) D1-108b (Z = 4-OMe)
CH (Me) S (O)2CH2(D1-81a) D1-108b (Z = 2-SMe)
CH (Me) S (O)2CH2(D1-81a) D1-108b (Z = 3-CFThree)
CH (Me) S (O)2CH2(D1-81a) D1-108b (Z = 4-OCFThree)
CH (Me) S (O)2CH2(D1-81a) D1-108b (Z = 2-SCFThree)
CH (Me) S (O)2CH2(D1-81a) C (O) Me
CH (Me) S (O)2CH2(D1-81a) C (O) CFThree
CH (Me) S (O)2CH2(D1-81a) C (O) OMe
CH2SCH2(D1-82a) Me
CH2SCH2(D1-82a) Et
CH2SCH2(D1-82a) Pr-n
CH2SCH2(D1-82a) Pr-i
CH2SCH2(D1-82a) Pr-c
CH2SCH2(D1-82a) Bu-n
CH2SCH2(D1-82a) Bu-i
CH2SCH2(D1-82a) Bu-c
CH2SCH2(D1-82a) Bu-s
CH2SCH2(D1-82a) Bu-t
CH2SCH2(D1-82a) Pen-n
CH2SCH2(D1-82a) Pen-c
CH2SCH2(D1-82a) Hex-n
CH2SCH2(D1-82a) Hex-c
CH2SCH2(D1-82a) CH2Pr-c
CH2SCH2(D1-82a) CH2Bu-c
CH2SCH2(D1-82a) CH2Pen-c
CH2SCH2(D1-82a) CH2Hex-c
CH2SCH2(D1-82a) CH2CH = CH2
CH2SCH2(D1-82a) CH2CH = C (Cl)2
CH2SCH2(D1-82a) CH2C≡CH
CH2SCH2(D1-82a) CH2CN
CH2SCH2(D1-82a) CH2CFThree
CH2SCH2(D1-82a) CH2OMe
CH2SCH2(D1-82a) CH2OCFThree
CH2SCH2(D1-82a) CH2SMe
CH2SCH2(D1-82a) CH2S (O) Me
CH2SCH2(D1-82a) CH2S (O)2Me
CH2SCH2(D1-82a) CH2SCFThree
CH2SCH2(D1-82a) CH2S (O) CFThree
CH2SCH2(D1-82a) CH2S (O)2CFThree
CH2SCH2(D1-82a) CH2CH (OMe)2
CH2SCH2(D1-82a) CH2CH (SMe)2
CH2SCH2(D1-82a) CH2C (O) Me
CH2SCH2(D1-82a) CH2C (O) CFThree
CH2SCH2(D1-82a) CH2C (O) OMe
CH2SCH2(D1-82a) CH2(D1-32a)
CH2SCH2(D1-82a) CH2(D1-33a)
CH2SCH2(D1-82a) CH2(D1-34a)
CH2SCH2(D1-82a) CH2(D1-37a)
CH2SCH2(D1-82a) CH2(D1-81a)
CH2SCH2(D1-82a) CH2(D1-82a)
CH2SCH2(D1-82a) CH2(D1-84a)
CH2SCH2(D1-82a) CH2(D1-85a)
CH2SCH2(D1-82a) CH2(D1-87a)
CH2SCH2(D1-82a) CH2(D1-92a)
CH2SCH2(D1-82a) CH2(D1-93a)
CH2SCH2(D1-82a) CH2(D1-95a)
CH2SCH2(D1-82a) CH2(D1-96a)
CH2SCH2(D1-82a) CH2(D1-98a)
CH2SCH2(D1-82a) CH2(D1-108a)
CH2SCH2(D1-82a) CH2(D1-108b, Z = 2-Cl)
CH2SCH2(D1-82a) CH2(D1-108b, Z = 3-Me)
CH2SCH2(D1-82a) CH2(D1-108b, Z = 4-OMe)
CH2SCH2(D1-82a) CH2(D1-108b, Z = 2-SMe)
CH2SCH2(D1-82a) CH2(D1-108b, Z = 3-CFThree)
CH2SCH2(D1-82a) CH2(D1-108b, Z = 4-OCFThree)
CH2SCH2(D1-82a) CH2(D1-108b, Z = 2-SCFThree)
CH2SCH2(D1-82a) CH2CH2CN
CH2SCH2(D1-82a) CH2CH2CFThree
CH2SCH2(D1-82a) CH2CH2OMe
CH2SCH2(D1-82a) CH2CH2SMe
CH2SCH2(D1-82a) CH2CH2S (O) Me
CH2SCH2(D1-82a) CH2CH2S (O)2Me
CH2SCH2(D1-82a) D1-32a
CH2SCH2(D1-82a) D1-33a
CH2SCH2(D1-82a) D1-34a
CH2SCH2(D1-82a) D1-37a
CH2SCH2(D1-82a) D1-81a
CH2SCH2(D1-82a) D1-82a
CH2SCH2(D1-82a) D1-84a
CH2SCH2(D1-82a) D1-85a
CH2SCH2(D1-82a) D1-87a
CH2SCH2(D1-82a) D1-92a
CH2SCH2(D1-82a) D1-93a
CH2SCH2(D1-82a) D1-95a
CH2SCH2(D1-82a) D1-96a
CH2SCH2(D1-82a) D1-98a
CH2SCH2(D1-82a) D1-108a
CH2SCH2(D1-82a) D1-108b (Z = 2-Cl)
CH2SCH2(D1-82a) D1-108b (Z = 3-Me)
CH2SCH2(D1-82a) D1-108b (Z = 4-OMe)
CH2SCH2(D1-82a) D1-108b (Z = 2-SMe)
CH2SCH2(D1-82a) D1-108b (Z = 3-CFThree)
CH2SCH2(D1-82a) D1-108b (Z = 4-OCFThree)
CH2SCH2(D1-82a) D1-108b (Z = 2-SCFThree)
CH2SCH2(D1-82a) C (O) Me
CH2SCH2(D1-82a) C (O) CFThree
CH2SCH2(D1-82a) C (O) OMe
CH2S (O) CH2(D1-82a) Me
CH2S (O) CH2(D1-82a) Et
CH2S (O) CH2(D1-82a) Pr-n
CH2S (O) CH2(D1-82a) Pr-i
CH2S (O) CH2(D1-82a) Pr-c
CH2S (O) CH2(D1-82a) Bu-n
CH2S (O) CH2(D1-82a) Bu-i
CH2S (O) CH2(D1-82a) Bu-c
CH2S (O) CH2(D1-82a) Bu-s
CH2S (O) CH2(D1-82a) Bu-t
CH2S (O) CH2(D1-82a) Pen-n
CH2S (O) CH2(D1-82a) Pen-c
CH2S (O) CH2(D1-82a) Hex-n
CH2S (O) CH2(D1-82a) Hex-c
CH2S (O) CH2(D1-82a) CH2Pr-c
CH2S (O) CH2(D1-82a) CH2Bu-c
CH2S (O) CH2(D1-82a) CH2Pen-c
CH2S (O) CH2(D1-82a) CH2Hex-c
CH2S (O) CH2(D1-82a) CH2CH = CH2
CH2S (O) CH2(D1-82a) CH2CH = C (Cl)2
CH2S (O) CH2(D1-82a) CH2C≡CH
CH2S (O) CH2(D1-82a) CH2CN
CH2S (O) CH2(D1-82a) CH2CFThree
CH2S (O) CH2(D1-82a) CH2OMe
CH2S (O) CH2(D1-82a) CH2OCFThree
CH2S (O) CH2(D1-82a) CH2SMe
CH2S (O) CH2(D1-82a) CH2S (O) Me
CH2S (O) CH2(D1-82a) CH2S (O)2Me
CH2S (O) CH2(D1-82a) CH2SCFThree
CH2S (O) CH2(D1-82a) CH2S (O) CFThree
CH2S (O) CH2(D1-82a) CH2S (O)2CFThree
CH2S (O) CH2(D1-82a) CH2CH (OMe)2
CH2S (O) CH2(D1-82a) CH2CH (SMe)2
CH2S (O) CH2(D1-82a) CH2C (O) Me
CH2S (O) CH2(D1-82a) CH2C (O) CFThree
CH2S (O) CH2(D1-82a) CH2C (O) OMe
CH2S (O) CH2(D1-82a) CH2(D1-32a)
CH2S (O) CH2(D1-82a) CH2(D1-33a)
CH2S (O) CH2(D1-82a) CH2(D1-34a)
CH2S (O) CH2(D1-82a) CH2(D1-37a)
CH2S (O) CH2(D1-82a) CH2(D1-81a)
CH2S (O) CH2(D1-82a) CH2(D1-82a)
CH2S (O) CH2(D1-82a) CH2(D1-84a)
CH2S (O) CH2(D1-82a) CH2(D1-85a)
CH2S (O) CH2(D1-82a) CH2(D1-87a)
CH2S (O) CH2(D1-82a) CH2(D1-92a)
CH2S (O) CH2(D1-82a) CH2(D1-93a)
CH2S (O) CH2(D1-82a) CH2(D1-95a)
CH2S (O) CH2(D1-82a) CH2(D1-96a)
CH2S (O) CH2(D1-82a) CH2(D1-98a)
CH2S (O) CH2(D1-82a) CH2(D1-108a)
CH2S (O) CH2(D1-82a) CH2(D1-108b, Z = 2-Cl)
CH2S (O) CH2(D1-82a) CH2(D1-108b, Z = 3-Me)
CH2S (O) CH2(D1-82a) CH2(D1-108b, Z = 4-OMe)
CH2S (O) CH2(D1-82a) CH2(D1-108b, Z = 2-SMe)
CH2S (O) CH2(D1-82a) CH2(D1-108b, Z = 3-CFThree)
CH2S (O) CH2(D1-82a) CH2(D1-108b, Z = 4-OCFThree)
CH2S (O) CH2(D1-82a) CH2(D1-108b, Z = 2-SCFThree)
CH2S (O) CH2(D1-82a) CH2CH2CN
CH2S (O) CH2(D1-82a) CH2CH2CFThree
CH2S (O) CH2(D1-82a) CH2CH2OMe
CH2S (O) CH2(D1-82a) CH2CH2SMe
CH2S (O) CH2(D1-82a) CH2CH2S (O) Me
CH2S (O) CH2(D1-82a) CH2CH2S (O)2Me
CH2S (O) CH2(D1-82a) D1-32a
CH2S (O) CH2(D1-82a) D1-33a
CH2S (O) CH2(D1-82a) D1-34a
CH2S (O) CH2(D1-82a) D1-37a
CH2S (O) CH2(D1-82a) D1-81a
CH2S (O) CH2(D1-82a) D1-82a
CH2S (O) CH2(D1-82a) D1-84a
CH2S (O) CH2(D1-82a) D1-85a
CH2S (O) CH2(D1-82a) D1-87a
CH2S (O) CH2(D1-82a) D1-92a
CH2S (O) CH2(D1-82a) D1-93a
CH2S (O) CH2(D1-82a) D1-95a
CH2S (O) CH2(D1-82a) D1-96a
CH2S (O) CH2(D1-82a) D1-98a
CH2S (O) CH2(D1-82a) D1-108a
CH2S (O) CH2(D1-82a) D1-108b (Z = 2-Cl)
CH2S (O) CH2(D1-82a) D1-108b (Z = 3-Me)
CH2S (O) CH2(D1-82a) D1-108b (Z = 4-OMe)
CH2S (O) CH2(D1-82a) D1-108b (Z = 2-SMe)
CH2S (O) CH2(D1-82a) D1-108b (Z = 3-CFThree)
CH2S (O) CH2(D1-82a) D1-108b (Z = 4-OCFThree)
CH2S (O) CH2(D1-82a) D1-108b (Z = 2-SCFThree)
CH2S (O) CH2(D1-82a) C (O) Me
CH2S (O) CH2(D1-82a) C (O) CFThree
CH2S (O) CH2(D1-82a) C (O) OMe
CH2S (O)2CH2(D1-82a) Me
CH2S (O)2CH2(D1-82a) Et
CH2S (O)2CH2(D1-82a) Pr-n
CH2S (O)2CH2(D1-82a) Pr-i
CH2S (O)2CH2(D1-82a) Pr-c
CH2S (O)2CH2(D1-82a) Bu-n
CH2S (O)2CH2(D1-82a) Bu-i
CH2S (O)2CH2(D1-82a) Bu-c
CH2S (O)2CH2(D1-82a) Bu-s
CH2S (O)2CH2(D1-82a) Bu-t
CH2S (O)2CH2(D1-82a) Pen-n
CH2S (O)2CH2(D1-82a) Pen-c
CH2S (O)2CH2(D1-82a) Hex-n
CH2S (O)2CH2(D1-82a) Hex-c
CH2S (O)2CH2(D1-82a) CH2Pr-c
CH2S (O)2CH2(D1-82a) CH2Bu-c
CH2S (O)2CH2(D1-82a) CH2Pen-c
CH2S (O)2CH2(D1-82a) CH2Hex-c
CH2S (O)2CH2(D1-82a) CH2CH = CH2
CH2S (O)2CH2(D1-82a) CH2CH = C (Cl)2
CH2S (O)2CH2(D1-82a) CH2C≡CH
CH2S (O)2CH2(D1-82a) CH2CN
CH2S (O)2CH2(D1-82a) CH2CFThree
CH2S (O)2CH2(D1-82a) CH2OMe
CH2S (O)2CH2(D1-82a) CH2OCFThree
CH2S (O)2CH2(D1-82a) CH2SMe
CH2S (O)2CH2(D1-82a) CH2S (O) Me
CH2S (O)2CH2(D1-82a) CH2S (O)2Me
CH2S (O)2CH2(D1-82a) CH2SCFThree
CH2S (O)2CH2(D1-82a) CH2S (O) CFThree
CH2S (O)2CH2(D1-82a) CH2S (O)2CFThree
CH2S (O)2CH2(D1-82a) CH2CH (OMe)2
CH2S (O)2CH2(D1-82a) CH2CH (SMe)2
CH2S (O)2CH2(D1-82a) CH2C (O) Me
CH2S (O)2CH2(D1-82a) CH2C (O) CFThree
CH2S (O)2CH2(D1-82a) CH2C (O) OMe
CH2S (O)2CH2(D1-82a) CH2(D1-32a)
CH2S (O)2CH2(D1-82a) CH2(D1-33a)
CH2S (O)2CH2(D1-82a) CH2(D1-34a)
CH2S (O)2CH2(D1-82a) CH2(D1-37a)
CH2S (O)2CH2(D1-82a) CH2(D1-81a)
CH2S (O)2CH2(D1-82a) CH2(D1-82a)
CH2S (O)2CH2(D1-82a) CH2(D1-84a)
CH2S (O)2CH2(D1-82a) CH2(D1-85a)
CH2S (O)2CH2(D1-82a) CH2(D1-87a)
CH2S (O)2CH2(D1-82a) CH2(D1-92a)
CH2S (O)2CH2(D1-82a) CH2(D1-93a)
CH2S (O)2CH2(D1-82a) CH2(D1-95a)
CH2S (O)2CH2(D1-82a) CH2(D1-96a)
CH2S (O)2CH2(D1-82a) CH2(D1-98a)
CH2S (O)2CH2(D1-82a) CH2(D1-108a)
CH2S (O)2CH2(D1-82a) CH2(D1-108b, Z = 2-Cl)
CH2S (O)2CH2(D1-82a) CH2(D1-108b, Z = 3-Me)
CH2S (O)2CH2(D1-82a) CH2(D1-108b, Z = 4-OMe)
CH2S (O)2CH2(D1-82a) CH2(D1-108b, Z = 2-SMe)
CH2S (O)2CH2(D1-82a) CH2(D1-108b, Z = 3-CFThree)
CH2S (O)2CH2(D1-82a) CH2(D1-108b, Z = 4-OCFThree)
CH2S (O)2CH2(D1-82a) CH2(D1-108b, Z = 2-SCFThree)
CH2S (O)2CH2(D1-82a) CH2CH2CN
CH2S (O)2CH2(D1-82a) CH2CH2CFThree
CH2S (O)2CH2(D1-82a) CH2CH2OMe
CH2S (O)2CH2(D1-82a) CH2CH2SMe
CH2S (O)2CH2(D1-82a) CH2CH2S (O) Me
CH2S (O)2CH2(D1-82a) CH2CH2S (O)2Me
CH2S (O)2CH2(D1-82a) D1-32a
CH2S (O)2CH2(D1-82a) D1-33a
CH2S (O)2CH2(D1-82a) D1-34a
CH2S (O)2CH2(D1-82a) D1-37a
CH2S (O)2CH2(D1-82a) D1-81a
CH2S (O)2CH2(D1-82a) D1-82a
CH2S (O)2CH2(D1-82a) D1-84a
CH2S (O)2CH2(D1-82a) D1-85a
CH2S (O)2CH2(D1-82a) D1-87a
CH2S (O)2CH2(D1-82a) D1-92a
CH2S (O)2CH2(D1-82a) D1-93a
CH2S (O)2CH2(D1-82a) D1-95a
CH2S (O)2CH2(D1-82a) D1-96a
CH2S (O)2CH2(D1-82a) D1-98a
CH2S (O)2CH2(D1-82a) D1-108a
CH2S (O)2CH2(D1-82a) D1-108b (Z = 2-Cl)
CH2S (O)2CH2(D1-82a) D1-108b (Z = 3-Me)
CH2S (O)2CH2(D1-82a) D1-108b (Z = 4-OMe)
CH2S (O)2CH2(D1-82a) D1-108b (Z = 2-SMe)
CH2S (O)2CH2(D1-82a) D1-108b (Z = 3-CFThree)
CH2S (O)2CH2(D1-82a) D1-108b (Z = 4-OCFThree)
CH2S (O)2CH2(D1-82a) D1-108b (Z = 2-SCFThree)
CH2S (O)2CH2(D1-82a) C (O) Me
CH2S (O)2CH2(D1-82a) C (O) CFThree
CH2S (O)2CH2(D1-82a) C (O) OMe
CH (Me) SCH2(D1-84a) Me
CH (Me) SCH2(D1-84a) Et
CH (Me) SCH2(D1-84a) Pr-n
CH (Me) SCH2(D1-84a) Pr-i
CH (Me) SCH2(D1-84a) Pr-c
CH (Me) SCH2(D1-84a) Bu-n
CH (Me) SCH2(D1-84a) Bu-i
CH (Me) SCH2(D1-84a) Bu-c
CH (Me) SCH2(D1-84a) Bu-s
CH (Me) SCH2(D1-84a) Bu-t
CH (Me) SCH2(D1-84a) Pen-n
CH (Me) SCH2(D1-84a) Pen-c
CH (Me) SCH2(D1-84a) Hex-n
CH (Me) SCH2(D1-84a) Hex-c
CH (Me) SCH2(D1-84a) CH2Pr-c
CH (Me) SCH2(D1-84a) CH2Bu-c
CH (Me) SCH2(D1-84a) CH2Pen-c
CH (Me) SCH2(D1-84a) CH2Hex-c
CH (Me) SCH2(D1-84a) CH2CH = CH2
CH (Me) SCH2(D1-84a) CH2CH = C (Cl)2
CH (Me) SCH2(D1-84a) CH2C≡CH
CH (Me) SCH2(D1-84a) CH2CN
CH (Me) SCH2(D1-84a) CH2CFThree
CH (Me) SCH2(D1-84a) CH2OMe
CH (Me) SCH2(D1-84a) CH2OCFThree
CH (Me) SCH2(D1-84a) CH2SMe
CH (Me) SCH2(D1-84a) CH2S (O) Me
CH (Me) SCH2(D1-84a) CH2S (O)2Me
CH (Me) SCH2(D1-84a) CH2SCFThree
CH (Me) SCH2(D1-84a) CH2S (O) CFThree
CH (Me) SCH2(D1-84a) CH2S (O)2CFThree
CH (Me) SCH2(D1-84a) CH2CH (OMe)2
CH (Me) SCH2(D1-84a) CH2CH (SMe)2
CH (Me) SCH2(D1-84a) CH2C (O) Me
CH (Me) SCH2(D1-84a) CH2C (O) CFThree
CH (Me) SCH2(D1-84a) CH2C (O) OMe
CH (Me) SCH2(D1-84a) CH2(D1-32a)
CH (Me) SCH2(D1-84a) CH2(D1-33a)
CH (Me) SCH2(D1-84a) CH2(D1-34a)
CH (Me) SCH2(D1-84a) CH2(D1-37a)
CH (Me) SCH2(D1-84a) CH2(D1-81a)
CH (Me) SCH2(D1-84a) CH2(D1-82a)
CH (Me) SCH2(D1-84a) CH2(D1-84a)
CH (Me) SCH2(D1-84a) CH2(D1-85a)
CH (Me) SCH2(D1-84a) CH2(D1-87a)
CH (Me) SCH2(D1-84a) CH2(D1-92a)
CH (Me) SCH2(D1-84a) CH2(D1-93a)
CH (Me) SCH2(D1-84a) CH2(D1-95a)
CH (Me) SCH2(D1-84a) CH2(D1-96a)
CH (Me) SCH2(D1-84a) CH2(D1-98a)
CH (Me) SCH2(D1-84a) CH2(D1-108a)
CH (Me) SCH2(D1-84a) CH2(D1-108b, Z = 2-Cl)
CH (Me) SCH2(D1-84a) CH2(D1-108b, Z = 3-Me)
CH (Me) SCH2(D1-84a) CH2(D1-108b, Z = 4-OMe)
CH (Me) SCH2(D1-84a) CH2(D1-108b, Z = 2-SMe)
CH (Me) SCH2(D1-84a) CH2(D1-108b, Z = 3-CFThree)
CH (Me) SCH2(D1-84a) CH2(D1-108b, Z = 4-OCFThree)
CH (Me) SCH2(D1-84a) CH2(D1-108b, Z = 2-SCFThree)
CH (Me) SCH2(D1-84a) CH2CH2CN
CH (Me) SCH2(D1-84a) CH2CH2CFThree
CH (Me) SCH2(D1-84a) CH2CH2OMe
CH (Me) SCH2(D1-84a) CH2CH2SMe
CH (Me) SCH2(D1-84a) CH2CH2S (O) Me
CH (Me) SCH2(D1-84a) CH2CH2S (O)2Me
CH (Me) SCH2(D1-84a) D1-32a
CH (Me) SCH2(D1-84a) D1-33a
CH (Me) SCH2(D1-84a) D1-34a
CH (Me) SCH2(D1-84a) D1-37a
CH (Me) SCH2(D1-84a) D1-81a
CH (Me) SCH2(D1-84a) D1-82a
CH (Me) SCH2(D1-84a) D1-84a
CH (Me) SCH2(D1-84a) D1-85a
CH (Me) SCH2(D1-84a) D1-87a
CH (Me) SCH2(D1-84a) D1-92a
CH (Me) SCH2(D1-84a) D1-93a
CH (Me) SCH2(D1-84a) D1-95a
CH (Me) SCH2(D1-84a) D1-96a
CH (Me) SCH2(D1-84a) D1-98a
CH (Me) SCH2(D1-84a) D1-108a
CH (Me) SCH2(D1-84a) D1-108b (Z = 2-Cl)
CH (Me) SCH2(D1-84a) D1-108b (Z = 3-Me)
CH (Me) SCH2(D1-84a) D1-108b (Z = 4-OMe)
CH (Me) SCH2(D1-84a) D1-108b (Z = 2-SMe)
CH (Me) SCH2(D1-84a) D1-108b (Z = 3-CFThree)
CH (Me) SCH2(D1-84a) D1-108b (Z = 4-OCFThree)
CH (Me) SCH2(D1-84a) D1-108b (Z = 2-SCFThree)
CH (Me) SCH2(D1-84a) C (O) Me
CH (Me) SCH2(D1-84a) C (O) CFThree
CH (Me) SCH2(D1-84a) C (O) OMe
CH (Me) S (O) CH2(D1-84a) Me
CH (Me) S (O) CH2(D1-84a) Et
CH (Me) S (O) CH2(D1-84a) Pr-n
CH (Me) S (O) CH2(D1-84a) Pr-i
CH (Me) S (O) CH2(D1-84a) Pr-c
CH (Me) S (O) CH2(D1-84a) Bu-n
CH (Me) S (O) CH2(D1-84a) Bu-i
CH (Me) S (O) CH2(D1-84a) Bu-c
CH (Me) S (O) CH2(D1-84a) Bu-s
CH (Me) S (O) CH2(D1-84a) Bu-t
CH (Me) S (O) CH2(D1-84a) Pen-n
CH (Me) S (O) CH2(D1-84a) Pen-c
CH (Me) S (O) CH2(D1-84a) Hex-n
CH (Me) S (O) CH2(D1-84a) Hex-c
CH (Me) S (O) CH2(D1-84a) CH2Pr-c
CH (Me) S (O) CH2(D1-84a) CH2Bu-c
CH (Me) S (O) CH2(D1-84a) CH2Pen-c
CH (Me) S (O) CH2(D1-84a) CH2Hex-c
CH (Me) S (O) CH2(D1-84a) CH2CH = CH2
CH (Me) S (O) CH2(D1-84a) CH2CH = C (Cl)2
CH (Me) S (O) CH2(D1-84a) CH2C≡CH
CH (Me) S (O) CH2(D1-84a) CH2CN
CH (Me) S (O) CH2(D1-84a) CH2CFThree
CH (Me) S (O) CH2(D1-84a) CH2OMe
CH (Me) S (O) CH2(D1-84a) CH2OCFThree
CH (Me) S (O) CH2(D1-84a) CH2SMe
CH (Me) S (O) CH2(D1-84a) CH2S (O) Me
CH (Me) S (O) CH2(D1-84a) CH2S (O)2Me
CH (Me) S (O) CH2(D1-84a) CH2SCFThree
CH (Me) S (O) CH2(D1-84a) CH2S (O) CFThree
CH (Me) S (O) CH2(D1-84a) CH2S (O)2CFThree
CH (Me) S (O) CH2(D1-84a) CH2CH (OMe)2
CH (Me) S (O) CH2(D1-84a) CH2CH (SMe)2
CH (Me) S (O) CH2(D1-84a) CH2C (O) Me
CH (Me) S (O) CH2(D1-84a) CH2C (O) CFThree
CH (Me) S (O) CH2(D1-84a) CH2C (O) OMe
CH (Me) S (O) CH2(D1-84a) CH2(D1-32a)
CH (Me) S (O) CH2(D1-84a) CH2(D1-33a)
CH (Me) S (O) CH2(D1-84a) CH2(D1-34a)
CH (Me) S (O) CH2(D1-84a) CH2(D1-37a)
CH (Me) S (O) CH2(D1-84a) CH2(D1-81a)
CH (Me) S (O) CH2(D1-84a) CH2(D1-82a)
CH (Me) S (O) CH2(D1-84a) CH2(D1-84a)
CH (Me) S (O) CH2(D1-84a) CH2(D1-85a)
CH (Me) S (O) CH2(D1-84a) CH2(D1-87a)
CH (Me) S (O) CH2(D1-84a) CH2(D1-92a)
CH (Me) S (O) CH2(D1-84a) CH2(D1-93a)
CH (Me) S (O) CH2(D1-84a) CH2(D1-95a)
CH (Me) S (O) CH2(D1-84a) CH2(D1-96a)
CH (Me) S (O) CH2(D1-84a) CH2(D1-98a)
CH (Me) S (O) CH2(D1-84a) CH2(D1-108a)
CH (Me) S (O) CH2(D1-84a) CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O) CH2(D1-84a) CH2(D1-108b, Z = 3-Me)
CH (Me) S (O) CH2(D1-84a) CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O) CH2(D1-84a) CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O) CH2(D1-84a) CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O) CH2(D1-84a) CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O) CH2(D1-84a) CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O) CH2(D1-84a) CH2CH2CN
CH (Me) S (O) CH2(D1-84a) CH2CH2CFThree
CH (Me) S (O) CH2(D1-84a) CH2CH2OMe
CH (Me) S (O) CH2(D1-84a) CH2CH2SMe
CH (Me) S (O) CH2(D1-84a) CH2CH2S (O) Me
CH (Me) S (O) CH2(D1-84a) CH2CH2S (O)2Me
CH (Me) S (O) CH2(D1-84a) D1-32a
CH (Me) S (O) CH2(D1-84a) D1-33a
CH (Me) S (O) CH2(D1-84a) D1-34a
CH (Me) S (O) CH2(D1-84a) D1-37a
CH (Me) S (O) CH2(D1-84a) D1-81a
CH (Me) S (O) CH2(D1-84a) D1-82a
CH (Me) S (O) CH2(D1-84a) D1-84a
CH (Me) S (O) CH2(D1-84a) D1-85a
CH (Me) S (O) CH2(D1-84a) D1-87a
CH (Me) S (O) CH2(D1-84a) D1-92a
CH (Me) S (O) CH2(D1-84a) D1-93a
CH (Me) S (O) CH2(D1-84a) D1-95a
CH (Me) S (O) CH2(D1-84a) D1-96a
CH (Me) S (O) CH2(D1-84a) D1-98a
CH (Me) S (O) CH2(D1-84a) D1-108a
CH (Me) S (O) CH2(D1-84a) D1-108b (Z = 2-Cl)
CH (Me) S (O) CH2(D1-84a) D1-108b (Z = 3-Me)
CH (Me) S (O) CH2(D1-84a) D1-108b (Z = 4-OMe)
CH (Me) S (O) CH2(D1-84a) D1-108b (Z = 2-SMe)
CH (Me) S (O) CH2(D1-84a) D1-108b (Z = 3-CFThree)
CH (Me) S (O) CH2(D1-84a) D1-108b (Z = 4-OCFThree)
CH (Me) S (O) CH2(D1-84a) D1-108b (Z = 2-SCFThree)
CH (Me) S (O) CH2(D1-84a) C (O) Me
CH (Me) S (O) CH2(D1-84a) C (O) CFThree
CH (Me) S (O) CH2(D1-84a) C (O) OMe
CH (Me) S (O)2CH2(D1-84a) Me
CH (Me) S (O)2CH2(D1-84a) Et
CH (Me) S (O)2CH2(D1-84a) Pr-n
CH (Me) S (O)2CH2(D1-84a) Pr-i
CH (Me) S (O)2CH2(D1-84a) Pr-c
CH (Me) S (O)2CH2(D1-84a) Bu-n
CH (Me) S (O)2CH2(D1-84a) Bu-i
CH (Me) S (O)2CH2(D1-84a) Bu-c
CH (Me) S (O)2CH2(D1-84a) Bu-s
CH (Me) S (O)2CH2(D1-84a) Bu-t
CH (Me) S (O)2CH2(D1-84a) Pen-n
CH (Me) S (O)2CH2(D1-84a) Pen-c
CH (Me) S (O)2CH2(D1-84a) Hex-n
CH (Me) S (O)2CH2(D1-84a) Hex-c
CH (Me) S (O)2CH2(D1-84a) CH2Pr-c
CH (Me) S (O)2CH2(D1-84a) CH2Bu-c
CH (Me) S (O)2CH2(D1-84a) CH2Pen-c
CH (Me) S (O)2CH2(D1-84a) CH2Hex-c
CH (Me) S (O)2CH2(D1-84a) CH2CH = CH2
CH (Me) S (O)2CH2(D1-84a) CH2CH = C (Cl)2
CH (Me) S (O)2CH2(D1-84a) CH2C≡CH
CH (Me) S (O)2CH2(D1-84a) CH2CN
CH (Me) S (O)2CH2(D1-84a) CH2CFThree
CH (Me) S (O)2CH2(D1-84a) CH2OMe
CH (Me) S (O)2CH2(D1-84a) CH2OCFThree
CH (Me) S (O)2CH2(D1-84a) CH2SMe
CH (Me) S (O)2CH2(D1-84a) CH2S (O) Me
CH (Me) S (O)2CH2(D1-84a) CH2S (O)2Me
CH (Me) S (O)2CH2(D1-84a) CH2SCFThree
CH (Me) S (O)2CH2(D1-84a) CH2S (O) CFThree
CH (Me) S (O)2CH2(D1-84a) CH2S (O)2CFThree
CH (Me) S (O)2CH2(D1-84a) CH2CH (OMe)2
CH (Me) S (O)2CH2(D1-84a) CH2CH (SMe)2
CH (Me) S (O)2CH2(D1-84a) CH2C (O) Me
CH (Me) S (O)2CH2(D1-84a) CH2C (O) CFThree
CH (Me) S (O)2CH2(D1-84a) CH2C (O) OMe
CH (Me) S (O)2CH2(D1-84a) CH2(D1-32a)
CH (Me) S (O)2CH2(D1-84a) CH2(D1-33a)
CH (Me) S (O)2CH2(D1-84a) CH2(D1-34a)
CH (Me) S (O)2CH2(D1-84a) CH2(D1-37a)
CH (Me) S (O)2CH2(D1-84a) CH2(D1-81a)
CH (Me) S (O)2CH2(D1-84a) CH2(D1-82a)
CH (Me) S (O)2CH2(D1-84a) CH2(D1-84a)
CH (Me) S (O)2CH2(D1-84a) CH2(D1-85a)
CH (Me) S (O)2CH2(D1-84a) CH2(D1-87a)
CH (Me) S (O)2CH2(D1-84a) CH2(D1-92a)
CH (Me) S (O)2CH2(D1-84a) CH2(D1-93a)
CH (Me) S (O)2CH2(D1-84a) CH2(D1-95a)
CH (Me) S (O)2CH2(D1-84a) CH2(D1-96a)
CH (Me) S (O)2CH2(D1-84a) CH2(D1-98a)
CH (Me) S (O)2CH2(D1-84a) CH2(D1-108a)
CH (Me) S (O)2CH2(D1-84a) CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O)2CH2(D1-84a) CH2(D1-108b, Z = 3-Me)
CH (Me) S (O)2CH2(D1-84a) CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O)2CH2(D1-84a) CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O)2CH2(D1-84a) CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O)2CH2(D1-84a) CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O)2CH2(D1-84a) CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O)2CH2(D1-84a) CH2CH2CN
CH (Me) S (O)2CH2(D1-84a) CH2CH2CFThree
CH (Me) S (O)2CH2(D1-84a) CH2CH2OMe
CH (Me) S (O)2CH2(D1-84a) CH2CH2SMe
CH (Me) S (O)2CH2(D1-84a) CH2CH2S (O) Me
CH (Me) S (O)2CH2(D1-84a) CH2CH2S (O)2Me
CH (Me) S (O)2CH2(D1-84a) D1-32a
CH (Me) S (O)2CH2(D1-84a) D1-33a
CH (Me) S (O)2CH2(D1-84a) D1-34a
CH (Me) S (O)2CH2(D1-84a) D1-37a
CH (Me) S (O)2CH2(D1-84a) D1-81a
CH (Me) S (O)2CH2(D1-84a) D1-82a
CH (Me) S (O)2CH2(D1-84a) D1-84a
CH (Me) S (O)2CH2(D1-84a) D1-85a
CH (Me) S (O)2CH2(D1-84a) D1-87a
CH (Me) S (O)2CH2(D1-84a) D1-92a
CH (Me) S (O)2CH2(D1-84a) D1-93a
CH (Me) S (O)2CH2(D1-84a) D1-95a
CH (Me) S (O)2CH2(D1-84a) D1-96a
CH (Me) S (O)2CH2(D1-84a) D1-98a
CH (Me) S (O)2CH2(D1-84a) D1-108a
CH (Me) S (O)2CH2(D1-84a) D1-108b (Z = 2-Cl)
CH (Me) S (O)2CH2(D1-84a) D1-108b (Z = 3-Me)
CH (Me) S (O)2CH2(D1-84a) D1-108b (Z = 4-OMe)
CH (Me) S (O)2CH2(D1-84a) D1-108b (Z = 2-SMe)
CH (Me) S (O)2CH2(D1-84a) D1-108b (Z = 3-CFThree)
CH (Me) S (O)2CH2(D1-84a) D1-108b (Z = 4-OCFThree)
CH (Me) S (O)2CH2(D1-84a) D1-108b (Z = 2-SCFThree)
CH (Me) S (O)2CH2(D1-84a) C (O) Me
CH (Me) S (O)2CH2(D1-84a) C (O) CFThree
CH (Me) S (O)2CH2(D1-84a) C (O) OMe
CH2SCH2(D1-85a) Me
CH2SCH2(D1-85a) Et
CH2SCH2(D1-85a) Pr-n
CH2SCH2(D1-85a) Pr-i
CH2SCH2(D1-85a) Pr-c
CH2SCH2(D1-85a) Bu-n
CH2SCH2(D1-85a) Bu-i
CH2SCH2(D1-85a) Bu-c
CH2SCH2(D1-85a) Bu-s
CH2SCH2(D1-85a) Bu-t
CH2SCH2(D1-85a) Pen-n
CH2SCH2(D1-85a) Pen-c
CH2SCH2(D1-85a) Hex-n
CH2SCH2(D1-85a) Hex-c
CH2SCH2(D1-85a) CH2Pr-c
CH2SCH2(D1-85a) CH2Bu-c
CH2SCH2(D1-85a) CH2Pen-c
CH2SCH2(D1-85a) CH2Hex-c
CH2SCH2(D1-85a) CH2CH = CH2
CH2SCH2(D1-85a) CH2CH = C (Cl)2
CH2SCH2(D1-85a) CH2C≡CH
CH2SCH2(D1-85a) CH2CN
CH2SCH2(D1-85a) CH2CFThree
CH2SCH2(D1-85a) CH2OMe
CH2SCH2(D1-85a) CH2OCFThree
CH2SCH2(D1-85a) CH2SMe
CH2SCH2(D1-85a) CH2S (O) Me
CH2SCH2(D1-85a) CH2S (O)2Me
CH2SCH2(D1-85a) CH2SCFThree
CH2SCH2(D1-85a) CH2S (O) CFThree
CH2SCH2(D1-85a) CH2S (O)2CFThree
CH2SCH2(D1-85a) CH2CH (OMe)2
CH2SCH2(D1-85a) CH2CH (SMe)2
CH2SCH2(D1-85a) CH2C (O) Me
CH2SCH2(D1-85a) CH2C (O) CFThree
CH2SCH2(D1-85a) CH2C (O) OMe
CH2SCH2(D1-85a) CH2(D1-32a)
CH2SCH2(D1-85a) CH2(D1-33a)
CH2SCH2(D1-85a) CH2(D1-34a)
CH2SCH2(D1-85a) CH2(D1-37a)
CH2SCH2(D1-85a) CH2(D1-81a)
CH2SCH2(D1-85a) CH2(D1-82a)
CH2SCH2(D1-85a) CH2(D1-84a)
CH2SCH2(D1-85a) CH2(D1-85a)
CH2SCH2(D1-85a) CH2(D1-87a)
CH2SCH2(D1-85a) CH2(D1-92a)
CH2SCH2(D1-85a) CH2(D1-93a)
CH2SCH2(D1-85a) CH2(D1-95a)
CH2SCH2(D1-85a) CH2(D1-96a)
CH2SCH2(D1-85a) CH2(D1-98a)
CH2SCH2(D1-85a) CH2(D1-108a)
CH2SCH2(D1-85a) CH2(D1-108b, Z = 2-Cl)
CH2SCH2(D1-85a) CH2(D1-108b, Z = 3-Me)
CH2SCH2(D1-85a) CH2(D1-108b, Z = 4-OMe)
CH2SCH2(D1-85a) CH2(D1-108b, Z = 2-SMe)
CH2SCH2(D1-85a) CH2(D1-108b, Z = 3-CFThree)
CH2SCH2(D1-85a) CH2(D1-108b, Z = 4-OCFThree)
CH2SCH2(D1-85a) CH2(D1-108b, Z = 2-SCFThree)
CH2SCH2(D1-85a) CH2CH2CN
CH2SCH2(D1-85a) CH2CH2CFThree
CH2SCH2(D1-85a) CH2CH2OMe
CH2SCH2(D1-85a) CH2CH2SMe
CH2SCH2(D1-85a) CH2CH2S (O) Me
CH2SCH2(D1-85a) CH2CH2S (O)2Me
CH2SCH2(D1-85a) D1-32a
CH2SCH2(D1-85a) D1-33a
CH2SCH2(D1-85a) D1-34a
CH2SCH2(D1-85a) D1-37a
CH2SCH2(D1-85a) D1-81a
CH2SCH2(D1-85a) D1-82a
CH2SCH2(D1-85a) D1-84a
CH2SCH2(D1-85a) D1-85a
CH2SCH2(D1-85a) D1-87a
CH2SCH2(D1-85a) D1-92a
CH2SCH2(D1-85a) D1-93a
CH2SCH2(D1-85a) D1-95a
CH2SCH2(D1-85a) D1-96a
CH2SCH2(D1-85a) D1-98a
CH2SCH2(D1-85a) D1-108a
CH2SCH2(D1-85a) D1-108b (Z = 2-Cl)
CH2SCH2(D1-85a) D1-108b (Z = 3-Me)
CH2SCH2(D1-85a) D1-108b (Z = 4-OMe)
CH2SCH2(D1-85a) D1-108b (Z = 2-SMe)
CH2SCH2(D1-85a) D1-108b (Z = 3-CFThree)
CH2SCH2(D1-85a) D1-108b (Z = 4-OCFThree)
CH2SCH2(D1-85a) D1-108b (Z = 2-SCFThree)
CH2SCH2(D1-85a) C (O) Me
CH2SCH2(D1-85a) C (O) CFThree
CH2SCH2(D1-85a) C (O) OMe
CH2S (O) CH2(D1-85a) Me
CH2S (O) CH2(D1-85a) Et
CH2S (O) CH2(D1-85a) Pr-n
CH2S (O) CH2(D1-85a) Pr-i
CH2S (O) CH2(D1-85a) Pr-c
CH2S (O) CH2(D1-85a) Bu-n
CH2S (O) CH2(D1-85a) Bu-i
CH2S (O) CH2(D1-85a) Bu-c
CH2S (O) CH2(D1-85a) Bu-s
CH2S (O) CH2(D1-85a) Bu-t
CH2S (O) CH2(D1-85a) Pen-n
CH2S (O) CH2(D1-85a) Pen-c
CH2S (O) CH2(D1-85a) Hex-n
CH2S (O) CH2(D1-85a) Hex-c
CH2S (O) CH2(D1-85a) CH2Pr-c
CH2S (O) CH2(D1-85a) CH2Bu-c
CH2S (O) CH2(D1-85a) CH2Pen-c
CH2S (O) CH2(D1-85a) CH2Hex-c
CH2S (O) CH2(D1-85a) CH2CH = CH2
CH2S (O) CH2(D1-85a) CH2CH = C (Cl)2
CH2S (O) CH2(D1-85a) CH2C≡CH
CH2S (O) CH2(D1-85a) CH2CN
CH2S (O) CH2(D1-85a) CH2CFThree
CH2S (O) CH2(D1-85a) CH2OMe
CH2S (O) CH2(D1-85a) CH2OCFThree
CH2S (O) CH2(D1-85a) CH2SMe
CH2S (O) CH2(D1-85a) CH2S (O) Me
CH2S (O) CH2(D1-85a) CH2S (O)2Me
CH2S (O) CH2(D1-85a) CH2SCFThree
CH2S (O) CH2(D1-85a) CH2S (O) CFThree
CH2S (O) CH2(D1-85a) CH2S (O)2CFThree
CH2S (O) CH2(D1-85a) CH2CH (OMe)2
CH2S (O) CH2(D1-85a) CH2CH (SMe)2
CH2S (O) CH2(D1-85a) CH2C (O) Me
CH2S (O) CH2(D1-85a) CH2C (O) CFThree
CH2S (O) CH2(D1-85a) CH2C (O) OMe
CH2S (O) CH2(D1-85a) CH2(D1-32a)
CH2S (O) CH2(D1-85a) CH2(D1-33a)
CH2S (O) CH2(D1-85a) CH2(D1-34a)
CH2S (O) CH2(D1-85a) CH2(D1-37a)
CH2S (O) CH2(D1-85a) CH2(D1-81a)
CH2S (O) CH2(D1-85a) CH2(D1-82a)
CH2S (O) CH2(D1-85a) CH2(D1-84a)
CH2S (O) CH2(D1-85a) CH2(D1-85a)
CH2S (O) CH2(D1-85a) CH2(D1-87a)
CH2S (O) CH2(D1-85a) CH2(D1-92a)
CH2S (O) CH2(D1-85a) CH2(D1-93a)
CH2S (O) CH2(D1-85a) CH2(D1-95a)
CH2S (O) CH2(D1-85a) CH2(D1-96a)
CH2S (O) CH2(D1-85a) CH2(D1-98a)
CH2S (O) CH2(D1-85a) CH2(D1-108a)
CH2S (O) CH2(D1-85a) CH2(D1-108b, Z = 2-Cl)
CH2S (O) CH2(D1-85a) CH2(D1-108b, Z = 3-Me)
CH2S (O) CH2(D1-85a) CH2(D1-108b, Z = 4-OMe)
CH2S (O) CH2(D1-85a) CH2(D1-108b, Z = 2-SMe)
CH2S (O) CH2(D1-85a) CH2(D1-108b, Z = 3-CFThree)
CH2S (O) CH2(D1-85a) CH2(D1-108b, Z = 4-OCFThree)
CH2S (O) CH2(D1-85a) CH2(D1-108b, Z = 2-SCFThree)
CH2S (O) CH2(D1-85a) CH2CH2CN
CH2S (O) CH2(D1-85a) CH2CH2CFThree
CH2S (O) CH2(D1-85a) CH2CH2OMe
CH2S (O) CH2(D1-85a) CH2CH2SMe
CH2S (O) CH2(D1-85a) CH2CH2S (O) Me
CH2S (O) CH2(D1-85a) CH2CH2S (O)2Me
CH2S (O) CH2(D1-85a) D1-32a
CH2S (O) CH2(D1-85a) D1-33a
CH2S (O) CH2(D1-85a) D1-34a
CH2S (O) CH2(D1-85a) D1-37a
CH2S (O) CH2(D1-85a) D1-81a
CH2S (O) CH2(D1-85a) D1-82a
CH2S (O) CH2(D1-85a) D1-84a
CH2S (O) CH2(D1-85a) D1-85a
CH2S (O) CH2(D1-85a) D1-87a
CH2S (O) CH2(D1-85a) D1-92a
CH2S (O) CH2(D1-85a) D1-93a
CH2S (O) CH2(D1-85a) D1-95a
CH2S (O) CH2(D1-85a) D1-96a
CH2S (O) CH2(D1-85a) D1-98a
CH2S (O) CH2(D1-85a) D1-108a
CH2S (O) CH2(D1-85a) D1-108b (Z = 2-Cl)
CH2S (O) CH2(D1-85a) D1-108b (Z = 3-Me)
CH2S (O) CH2(D1-85a) D1-108b (Z = 4-OMe)
CH2S (O) CH2(D1-85a) D1-108b (Z = 2-SMe)
CH2S (O) CH2(D1-85a) D1-108b (Z = 3-CFThree)
CH2S (O) CH2(D1-85a) D1-108b (Z = 4-OCFThree)
CH2S (O) CH2(D1-85a) D1-108b (Z = 2-SCFThree)
CH2S (O) CH2(D1-85a) C (O) Me
CH2S (O) CH2(D1-85a) C (O) CFThree
CH2S (O) CH2(D1-85a) C (O) OMe
CH2S (O)2CH2(D1-85a) Me
CH2S (O)2CH2(D1-85a) Et
CH2S (O)2CH2(D1-85a) Pr-n
CH2S (O)2CH2(D1-85a) Pr-i
CH2S (O)2CH2(D1-85a) Pr-c
CH2S (O)2CH2(D1-85a) Bu-n
CH2S (O)2CH2(D1-85a) Bu-i
CH2S (O)2CH2(D1-85a) Bu-c
CH2S (O)2CH2(D1-85a) Bu-s
CH2S (O)2CH2(D1-85a) Bu-t
CH2S (O)2CH2(D1-85a) Pen-n
CH2S (O)2CH2(D1-85a) Pen-c
CH2S (O)2CH2(D1-85a) Hex-n
CH2S (O)2CH2(D1-85a) Hex-c
CH2S (O)2CH2(D1-85a) CH2Pr-c
CH2S (O)2CH2(D1-85a) CH2Bu-c
CH2S (O)2CH2(D1-85a) CH2Pen-c
CH2S (O)2CH2(D1-85a) CH2Hex-c
CH2S (O)2CH2(D1-85a) CH2CH = CH2
CH2S (O)2CH2(D1-85a) CH2CH = C (Cl)2
CH2S (O)2CH2(D1-85a) CH2C≡CH
CH2S (O)2CH2(D1-85a) CH2CN
CH2S (O)2CH2(D1-85a) CH2CFThree
CH2S (O)2CH2(D1-85a) CH2OMe
CH2S (O)2CH2(D1-85a) CH2OCFThree
CH2S (O)2CH2(D1-85a) CH2SMe
CH2S (O)2CH2(D1-85a) CH2S (O) Me
CH2S (O)2CH2(D1-85a) CH2S (O)2Me
CH2S (O)2CH2(D1-85a) CH2SCFThree
CH2S (O)2CH2(D1-85a) CH2S (O) CFThree
CH2S (O)2CH2(D1-85a) CH2S (O)2CFThree
CH2S (O)2CH2(D1-85a) CH2CH (OMe)2
CH2S (O)2CH2(D1-85a) CH2CH (SMe)2
CH2S (O)2CH2(D1-85a) CH2C (O) Me
CH2S (O)2CH2(D1-85a) CH2C (O) CFThree
CH2S (O)2CH2(D1-85a) CH2C (O) OMe
CH2S (O)2CH2(D1-85a) CH2(D1-32a)
CH2S (O)2CH2(D1-85a) CH2(D1-33a)
CH2S (O)2CH2(D1-85a) CH2(D1-34a)
CH2S (O)2CH2(D1-85a) CH2(D1-37a)
CH2S (O)2CH2(D1-85a) CH2(D1-81a)
CH2S (O)2CH2(D1-85a) CH2(D1-82a)
CH2S (O)2CH2(D1-85a) CH2(D1-84a)
CH2S (O)2CH2(D1-85a) CH2(D1-85a)
CH2S (O)2CH2(D1-85a) CH2(D1-87a)
CH2S (O)2CH2(D1-85a) CH2(D1-92a)
CH2S (O)2CH2(D1-85a) CH2(D1-93a)
CH2S (O)2CH2(D1-85a) CH2(D1-95a)
CH2S (O)2CH2(D1-85a) CH2(D1-96a)
CH2S (O)2CH2(D1-85a) CH2(D1-98a)
CH2S (O)2CH2(D1-85a) CH2(D1-108a)
CH2S (O)2CH2(D1-85a) CH2(D1-108b, Z = 2-Cl)
CH2S (O)2CH2(D1-85a) CH2(D1-108b, Z = 3-Me)
CH2S (O)2CH2(D1-85a) CH2(D1-108b, Z = 4-OMe)
CH2S (O)2CH2(D1-85a) CH2(D1-108b, Z = 2-SMe)
CH2S (O)2CH2(D1-85a) CH2(D1-108b, Z = 3-CFThree)
CH2S (O)2CH2(D1-85a) CH2(D1-108b, Z = 4-OCFThree)
CH2S (O)2CH2(D1-85a) CH2(D1-108b, Z = 2-SCFThree)
CH2S (O)2CH2(D1-85a) CH2CH2CN
CH2S (O)2CH2(D1-85a) CH2CH2CFThree
CH2S (O)2CH2(D1-85a) CH2CH2OMe
CH2S (O)2CH2(D1-85a) CH2CH2SMe
CH2S (O)2CH2(D1-85a) CH2CH2S (O) Me
CH2S (O)2CH2(D1-85a) CH2CH2S (O)2Me
CH2S (O)2CH2(D1-85a) D1-32a
CH2S (O)2CH2(D1-85a) D1-33a
CH2S (O)2CH2(D1-85a) D1-34a
CH2S (O)2CH2(D1-85a) D1-37a
CH2S (O)2CH2(D1-85a) D1-81a
CH2S (O)2CH2(D1-85a) D1-82a
CH2S (O)2CH2(D1-85a) D1-84a
CH2S (O)2CH2(D1-85a) D1-85a
CH2S (O)2CH2(D1-85a) D1-87a
CH2S (O)2CH2(D1-85a) D1-92a
CH2S (O)2CH2(D1-85a) D1-93a
CH2S (O)2CH2(D1-85a) D1-95a
CH2S (O)2CH2(D1-85a) D1-96a
CH2S (O)2CH2(D1-85a) D1-98a
CH2S (O)2CH2(D1-85a) D1-108a
CH2S (O)2CH2(D1-85a) D1-108b (Z = 2-Cl)
CH2S (O)2CH2(D1-85a) D1-108b (Z = 3-Me)
CH2S (O)2CH2(D1-85a) D1-108b (Z = 4-OMe)
CH2S (O)2CH2(D1-85a) D1-108b (Z = 2-SMe)
CH2S (O)2CH2(D1-85a) D1-108b (Z = 3-CFThree)
CH2S (O)2CH2(D1-85a) D1-108b (Z = 4-OCFThree)
CH2S (O)2CH2(D1-85a) D1-108b (Z = 2-SCFThree)
CH2SCH2(D1-87a) Me
CH2SCH2(D1-87a) Et
CH2SCH2(D1-87a) Pr-n
CH2SCH2(D1-87a) Pr-i
CH2SCH2(D1-87a) Pr-c
CH2SCH2(D1-87a) Bu-n
CH2SCH2(D1-87a) Bu-i
CH2SCH2(D1-87a) Bu-c
CH2SCH2(D1-87a) Bu-s
CH2SCH2(D1-87a) Bu-t
CH2SCH2(D1-87a) Pen-n
CH2SCH2(D1-87a) Pen-c
CH2SCH2(D1-87a) Hex-n
CH2SCH2(D1-87a) Hex-c
CH2SCH2(D1-87a) CH2Pr-c
CH2SCH2(D1-87a) CH2Bu-c
CH2SCH2(D1-87a) CH2Pen-c
CH2SCH2(D1-87a) CH2Hex-c
CH2SCH2(D1-87a) CH2CH = CH2
CH2SCH2(D1-87a) CH2CH = C (Cl)2
CH2SCH2(D1-87a) CH2C≡CH
CH2SCH2(D1-87a) CH2CN
CH2SCH2(D1-87a) CH2CFThree
CH2SCH2(D1-87a) CH2OMe
CH2SCH2(D1-87a) CH2OCFThree
CH2SCH2(D1-87a) CH2SMe
CH2SCH2(D1-87a) CH2S (O) Me
CH2SCH2(D1-87a) CH2S (O)2Me
CH2SCH2(D1-87a) CH2SCFThree
CH2SCH2(D1-87a) CH2S (O) CFThree
CH2SCH2(D1-87a) CH2S (O)2CFThree
CH2SCH2(D1-87a) CH2CH (OMe)2
CH2SCH2(D1-87a) CH2CH (SMe)2
CH2SCH2(D1-87a) CH2C (O) Me
CH2SCH2(D1-87a) CH2C (O) CFThree
CH2SCH2(D1-87a) CH2C (O) OMe
CH2SCH2(D1-87a) CH2(D1-32a)
CH2SCH2(D1-87a) CH2(D1-33a)
CH2SCH2(D1-87a) CH2(D1-34a)
CH2SCH2(D1-87a) CH2(D1-37a)
CH2SCH2(D1-87a) CH2(D1-81a)
CH2SCH2(D1-87a) CH2(D1-82a)
CH2SCH2(D1-87a) CH2(D1-84a)
CH2SCH2(D1-87a) CH2(D1-85a)
CH2SCH2(D1-87a) CH2(D1-87a)
CH2SCH2(D1-87a) CH2(D1-92a)
CH2SCH2(D1-87a) CH2(D1-93a)
CH2SCH2(D1-87a) CH2(D1-95a)
CH2SCH2(D1-87a) CH2(D1-96a)
CH2SCH2(D1-87a) CH2(D1-98a)
CH2SCH2(D1-87a) CH2(D1-108a)
CH2SCH2(D1-87a) CH2(D1-108b, Z = 2-Cl)
CH2SCH2(D1-87a) CH2(D1-108b, Z = 3-Me)
CH2SCH2(D1-87a) CH2(D1-108b, Z = 4-OMe)
CH2SCH2(D1-87a) CH2(D1-108b, Z = 2-SMe)
CH2SCH2(D1-87a) CH2(D1-108b, Z = 3-CFThree)
CH2SCH2(D1-87a) CH2(D1-108b, Z = 4-OCFThree)
CH2SCH2(D1-87a) CH2(D1-108b, Z = 2-SCFThree)
CH2SCH2(D1-87a) CH2CH2CN
CH2SCH2(D1-87a) CH2CH2CFThree
CH2SCH2(D1-87a) CH2CH2OMe
CH2SCH2(D1-87a) CH2CH2SMe
CH2SCH2(D1-87a) CH2CH2S (O) Me
CH2SCH2(D1-87a) CH2CH2S (O)2Me
CH2SCH2(D1-87a) D1-32a
CH2SCH2(D1-87a) D1-33a
CH2SCH2(D1-87a) D1-34a
CH2SCH2(D1-87a) D1-37a
CH2SCH2(D1-87a) D1-81a
CH2SCH2(D1-87a) D1-82a
CH2SCH2(D1-87a) D1-84a
CH2SCH2(D1-87a) D1-85a
CH2SCH2(D1-87a) D1-87a
CH2SCH2(D1-87a) D1-92a
CH2SCH2(D1-87a) D1-93a
CH2SCH2(D1-87a) D1-95a
CH2SCH2(D1-87a) D1-96a
CH2SCH2(D1-87a) D1-98a
CH2SCH2(D1-87a) D1-108a
CH2SCH2(D1-87a) D1-108b (Z = 2-Cl)
CH2SCH2(D1-87a) D1-108b (Z = 3-Me)
CH2SCH2(D1-87a) D1-108b (Z = 4-OMe)
CH2SCH2(D1-87a) D1-108b (Z = 2-SMe)
CH2SCH2(D1-87a) D1-108b (Z = 3-CFThree)
CH2SCH2(D1-87a) D1-108b (Z = 4-OCFThree)
CH2SCH2(D1-87a) D1-108b (Z = 2-SCFThree)
CH2SCH2(D1-87a) C (O) Me
CH2SCH2(D1-87a) C (O) CFThree
CH2SCH2(D1-87a) C (O) OMe
CH2S (O) CH2(D1-87a) Me
CH2S (O) CH2(D1-87a) Et
CH2S (O) CH2(D1-87a) Pr-n
CH2S (O) CH2(D1-87a) Pr-i
CH2S (O) CH2(D1-87a) Pr-c
CH2S (O) CH2(D1-87a) Bu-n
CH2S (O) CH2(D1-87a) Bu-i
CH2S (O) CH2(D1-87a) Bu-c
CH2S (O) CH2(D1-87a) Bu-s
CH2S (O) CH2(D1-87a) Bu-t
CH2S (O) CH2(D1-87a) Pen-n
CH2S (O) CH2(D1-87a) Pen-c
CH2S (O) CH2(D1-87a) Hex-n
CH2S (O) CH2(D1-87a) Hex-c
CH2S (O) CH2(D1-87a) CH2Pr-c
CH2S (O) CH2(D1-87a) CH2Bu-c
CH2S (O) CH2(D1-87a) CH2Pen-c
CH2S (O) CH2(D1-87a) CH2Hex-c
CH2S (O) CH2(D1-87a) CH2CH = CH2
CH2S (O) CH2(D1-87a) CH2CH = C (Cl)2
CH2S (O) CH2(D1-87a) CH2C≡CH
CH2S (O) CH2(D1-87a) CH2CN
CH2S (O) CH2(D1-87a) CH2CFThree
CH2S (O) CH2(D1-87a) CH2OMe
CH2S (O) CH2(D1-87a) CH2OCFThree
CH2S (O) CH2(D1-87a) CH2SMe
CH2S (O) CH2(D1-87a) CH2S (O) Me
CH2S (O) CH2(D1-87a) CH2S (O)2Me
CH2S (O) CH2(D1-87a) CH2SCFThree
CH2S (O) CH2(D1-87a) CH2S (O) CFThree
CH2S (O) CH2(D1-87a) CH2S (O)2CFThree
CH2S (O) CH2(D1-87a) CH2CH (OMe)2
CH2S (O) CH2(D1-87a) CH2CH (SMe)2
CH2S (O) CH2(D1-87a) CH2C (O) Me
CH2S (O) CH2(D1-87a) CH2C (O) CFThree
CH2S (O) CH2(D1-87a) CH2C (O) OMe
CH2S (O) CH2(D1-87a) CH2(D1-32a)
CH2S (O) CH2(D1-87a) CH2(D1-33a)
CH2S (O) CH2(D1-87a) CH2(D1-34a)
CH2S (O) CH2(D1-87a) CH2(D1-37a)
CH2S (O) CH2(D1-87a) CH2(D1-81a)
CH2S (O) CH2(D1-87a) CH2(D1-82a)
CH2S (O) CH2(D1-87a) CH2(D1-84a)
CH2S (O) CH2(D1-87a) CH2(D1-85a)
CH2S (O) CH2(D1-87a) CH2(D1-87a)
CH2S (O) CH2(D1-87a) CH2(D1-92a)
CH2S (O) CH2(D1-87a) CH2(D1-93a)
CH2S (O) CH2(D1-87a) CH2(D1-95a)
CH2S (O) CH2(D1-87a) CH2(D1-96a)
CH2S (O) CH2(D1-87a) CH2(D1-98a)
CH2S (O) CH2(D1-87a) CH2(D1-108a)
CH2S (O) CH2(D1-87a) CH2(D1-108b, Z = 2-Cl)
CH2S (O) CH2(D1-87a) CH2(D1-108b, Z = 3-Me)
CH2S (O) CH2(D1-87a) CH2(D1-108b, Z = 4-OMe)
CH2S (O) CH2(D1-87a) CH2(D1-108b, Z = 2-SMe)
CH2S (O) CH2(D1-87a) CH2(D1-108b, Z = 3-CFThree)
CH2S (O) CH2(D1-87a) CH2(D1-108b, Z = 4-OCFThree)
CH2S (O) CH2(D1-87a) CH2(D1-108b, Z = 2-SCFThree)
CH2S (O) CH2(D1-87a) CH2CH2CN
CH2S (O) CH2(D1-87a) CH2CH2CFThree
CH2S (O) CH2(D1-87a) CH2CH2OMe
CH2S (O) CH2(D1-87a) CH2CH2SMe
CH2S (O) CH2(D1-87a) CH2CH2S (O) Me
CH2S (O) CH2(D1-87a) CH2CH2S (O)2Me
CH2S (O) CH2(D1-87a) D1-32a
CH2S (O) CH2(D1-87a) D1-33a
CH2S (O) CH2(D1-87a) D1-34a
CH2S (O) CH2(D1-87a) D1-37a
CH2S (O) CH2(D1-87a) D1-81a
CH2S (O) CH2(D1-87a) D1-82a
CH2S (O) CH2(D1-87a) D1-84a
CH2S (O) CH2(D1-87a) D1-85a
CH2S (O) CH2(D1-87a) D1-87a
CH2S (O) CH2(D1-87a) D1-92a
CH2S (O) CH2(D1-87a) D1-93a
CH2S (O) CH2(D1-87a) D1-95a
CH2S (O) CH2(D1-87a) D1-96a
CH2S (O) CH2(D1-87a) D1-98a
CH2S (O) CH2(D1-87a) D1-108a
CH2S (O) CH2(D1-87a) D1-108b (Z = 2-Cl)
CH2S (O) CH2(D1-87a) D1-108b (Z = 3-Me)
CH2S (O) CH2(D1-87a) D1-108b (Z = 4-OMe)
CH2S (O) CH2(D1-87a) D1-108b (Z = 2-SMe)
CH2S (O) CH2(D1-87a) D1-108b (Z = 3-CFThree)
CH2S (O) CH2(D1-87a) D1-108b (Z = 4-OCFThree)
CH2S (O) CH2(D1-87a) D1-108b (Z = 2-SCFThree)
CH2S (O) CH2(D1-87a) C (O) Me
CH2S (O) CH2(D1-87a) C (O) CFThree
CH2S (O) CH2(D1-87a) C (O) OMe
CH2S (O)2CH2(D1-87a) Me
CH2S (O)2CH2(D1-87a) Et
CH2S (O)2CH2(D1-87a) Pr-n
CH2S (O)2CH2(D1-87a) Pr-i
CH2S (O)2CH2(D1-87a) Pr-c
CH2S (O)2CH2(D1-87a) Bu-n
CH2S (O)2CH2(D1-87a) Bu-i
CH2S (O)2CH2(D1-87a) Bu-c
CH2S (O)2CH2(D1-87a) Bu-s
CH2S (O)2CH2(D1-87a) Bu-t
CH2S (O)2CH2(D1-87a) Pen-n
CH2S (O)2CH2(D1-87a) Pen-c
CH2S (O)2CH2(D1-87a) Hex-n
CH2S (O)2CH2(D1-87a) Hex-c
CH2S (O)2CH2(D1-87a) CH2Pr-c
CH2S (O)2CH2(D1-87a) CH2Bu-c
CH2S (O)2CH2(D1-87a) CH2Pen-c
CH2S (O)2CH2(D1-87a) CH2Hex-c
CH2S (O)2CH2(D1-87a) CH2CH = CH2
CH2S (O)2CH2(D1-87a) CH2CH = C (Cl)2
CH2S (O)2CH2(D1-87a) CH2C≡CH
CH2S (O)2CH2(D1-87a) CH2CN
CH2S (O)2CH2(D1-87a) CH2CFThree
CH2S (O)2CH2(D1-87a) CH2OMe
CH2S (O)2CH2(D1-87a) CH2OCFThree
CH2S (O)2CH2(D1-87a) CH2SMe
CH2S (O)2CH2(D1-87a) CH2S (O) Me
CH2S (O)2CH2(D1-87a) CH2S (O)2Me
CH2S (O)2CH2(D1-87a) CH2SCFThree
CH2S (O)2CH2(D1-87a) CH2S (O) CFThree
CH2S (O)2CH2(D1-87a) CH2S (O)2CFThree
CH2S (O)2CH2(D1-87a) CH2CH (OMe)2
CH2S (O)2CH2(D1-87a) CH2CH (SMe)2
CH2S (O)2CH2(D1-87a) CH2C (O) Me
CH2S (O)2CH2(D1-87a) CH2C (O) CFThree
CH2S (O)2CH2(D1-87a) CH2C (O) OMe
CH2S (O)2CH2(D1-87a) CH2(D1-32a)
CH2S (O)2CH2(D1-87a) CH2(D1-33a)
CH2S (O)2CH2(D1-87a) CH2(D1-34a)
CH2S (O)2CH2(D1-87a) CH2(D1-37a)
CH2S (O)2CH2(D1-87a) CH2(D1-81a)
CH2S (O)2CH2(D1-87a) CH2(D1-82a)
CH2S (O)2CH2(D1-87a) CH2(D1-84a)
CH2S (O)2CH2(D1-87a) CH2(D1-85a)
CH2S (O)2CH2(D1-87a) CH2(D1-87a)
CH2S (O)2CH2(D1-87a) CH2(D1-92a)
CH2S (O)2CH2(D1-87a) CH2(D1-93a)
CH2S (O)2CH2(D1-87a) CH2(D1-95a)
CH2S (O)2CH2(D1-87a) CH2(D1-96a)
CH2S (O)2CH2(D1-87a) CH2(D1-98a)
CH2S (O)2CH2(D1-87a) CH2(D1-108a)
CH2S (O)2CH2(D1-87a) CH2(D1-108b, Z = 2-Cl)
CH2S (O)2CH2(D1-87a) CH2(D1-108b, Z = 3-Me)
CH2S (O)2CH2(D1-87a) CH2(D1-108b, Z = 4-OMe)
CH2S (O)2CH2(D1-87a) CH2(D1-108b, Z = 2-SMe)
CH2S (O)2CH2(D1-87a) CH2(D1-108b, Z = 3-CFThree)
CH2S (O)2CH2(D1-87a) CH2(D1-108b, Z = 4-OCFThree)
CH2S (O)2CH2(D1-87a) CH2(D1-108b, Z = 2-SCFThree)
CH2S (O)2CH2(D1-87a) CH2CH2CN
CH2S (O)2CH2(D1-87a) CH2CH2CFThree
CH2S (O)2CH2(D1-87a) CH2CH2OMe
CH2S (O)2CH2(D1-87a) CH2CH2SMe
CH2S (O)2CH2(D1-87a) CH2CH2S (O) Me
CH2S (O)2CH2(D1-87a) CH2CH2S (O)2Me
CH2S (O)2CH2(D1-87a) D1-32a
CH2S (O)2CH2(D1-87a) D1-33a
CH2S (O)2CH2(D1-87a) D1-34a
CH2S (O)2CH2(D1-87a) D1-37a
CH2S (O)2CH2(D1-87a) D1-81a
CH2S (O)2CH2(D1-87a) D1-82a
CH2S (O)2CH2(D1-87a) D1-84a
CH2S (O)2CH2(D1-87a) D1-85a
CH2S (O)2CH2(D1-87a) D1-87a
CH2S (O)2CH2(D1-87a) D1-92a
CH2S (O)2CH2(D1-87a) D1-93a
CH2S (O)2CH2(D1-87a) D1-95a
CH2S (O)2CH2(D1-87a) D1-96a
CH2S (O)2CH2(D1-87a) D1-98a
CH2S (O)2CH2(D1-87a) D1-108a
CH2S (O)2CH2(D1-87a) D1-108b (Z = 2-Cl)
CH2S (O)2CH2(D1-87a) D1-108b (Z = 3-Me)
CH2S (O)2CH2(D1-87a) D1-108b (Z = 4-OMe)
CH2S (O)2CH2(D1-87a) D1-108b (Z = 2-SMe)
CH2S (O)2CH2(D1-87a) D1-108b (Z = 3-CFThree)
CH2S (O)2CH2(D1-87a) D1-108b (Z = 4-OCFThree)
CH2S (O)2CH2(D1-87a) D1-108b (Z = 2-SCFThree)
CH2SCH2(D1-95a) Me
CH2SCH2(D1-95a) Et
CH2SCH2(D1-95a) Pr-n
CH2SCH2(D1-95a) Pr-i
CH2SCH2(D1-95a) Pr-c
CH2SCH2(D1-95a) Bu-n
CH2SCH2(D1-95a) Bu-i
CH2SCH2(D1-95a) Bu-c
CH2SCH2(D1-95a) Bu-s
CH2SCH2(D1-95a) Bu-t
CH2SCH2(D1-95a) Pen-n
CH2SCH2(D1-95a) Pen-c
CH2SCH2(D1-95a) Hex-n
CH2SCH2(D1-95a) Hex-c
CH2SCH2(D1-95a) CH2Pr-c
CH2SCH2(D1-95a) CH2Bu-c
CH2SCH2(D1-95a) CH2Pen-c
CH2SCH2(D1-95a) CH2Hex-c
CH2SCH2(D1-95a) CH2CH = CH2
CH2SCH2(D1-95a) CH2CH = C (Cl)2
CH2SCH2(D1-95a) CH2C≡CH
CH2SCH2(D1-95a) CH2CN
CH2SCH2(D1-95a) CH2CFThree
CH2SCH2(D1-95a) CH2OMe
CH2SCH2(D1-95a) CH2OCFThree
CH2SCH2(D1-95a) CH2SMe
CH2SCH2(D1-95a) CH2S (O) Me
CH2SCH2(D1-95a) CH2S (O)2Me
CH2SCH2(D1-95a) CH2SCFThree
CH2SCH2(D1-95a) CH2S (O) CFThree
CH2SCH2(D1-95a) CH2S (O)2CFThree
CH2SCH2(D1-95a) CH2CH (OMe)2
CH2SCH2(D1-95a) CH2CH (SMe)2
CH2SCH2(D1-95a) CH2C (O) Me
CH2SCH2(D1-95a) CH2C (O) CFThree
CH2SCH2(D1-95a) CH2C (O) OMe
CH2SCH2(D1-95a) CH2(D1-32a)
CH2SCH2(D1-95a) CH2(D1-33a)
CH2SCH2(D1-95a) CH2(D1-34a)
CH2SCH2(D1-95a) CH2(D1-37a)
CH2SCH2(D1-95a) CH2(D1-81a)
CH2SCH2(D1-95a) CH2(D1-82a)
CH2SCH2(D1-95a) CH2(D1-84a)
CH2SCH2(D1-95a) CH2(D1-85a)
CH2SCH2(D1-95a) CH2(D1-87a)
CH2SCH2(D1-95a) CH2(D1-92a)
CH2SCH2(D1-95a) CH2(D1-93a)
CH2SCH2(D1-95a) CH2(D1-95a)
CH2SCH2(D1-95a) CH2(D1-96a)
CH2SCH2(D1-95a) CH2(D1-98a)
CH2SCH2(D1-95a) CH2(D1-108a)
CH2SCH2(D1-95a) CH2(D1-108b, Z = 2-Cl)
CH2SCH2(D1-95a) CH2(D1-108b, Z = 3-Me)
CH2SCH2(D1-95a) CH2(D1-108b, Z = 4-OMe)
CH2SCH2(D1-95a) CH2(D1-108b, Z = 2-SMe)
CH2SCH2(D1-95a) CH2(D1-108b, Z = 3-CFThree)
CH2SCH2(D1-95a) CH2(D1-108b, Z = 4-OCFThree)
CH2SCH2(D1-95a) CH2(D1-108b, Z = 2-SCFThree)
CH2SCH2(D1-95a) CH2CH2CN
CH2SCH2(D1-95a) CH2CH2CFThree
CH2SCH2(D1-95a) CH2CH2OMe
CH2SCH2(D1-95a) CH2CH2SMe
CH2SCH2(D1-95a) CH2CH2S (O) Me
CH2SCH2(D1-95a) CH2CH2S (O)2Me
CH2SCH2(D1-95a) D1-32a
CH2SCH2(D1-95a) D1-33a
CH2SCH2(D1-95a) D1-34a
CH2SCH2(D1-95a) D1-37a
CH2SCH2(D1-95a) D1-81a
CH2SCH2(D1-95a) D1-82a
CH2SCH2(D1-95a) D1-84a
CH2SCH2(D1-95a) D1-85a
CH2SCH2(D1-95a) D1-87a
CH2SCH2(D1-95a) D1-92a
CH2SCH2(D1-95a) D1-93a
CH2SCH2(D1-95a) D1-95a
CH2SCH2(D1-95a) D1-96a
CH2SCH2(D1-95a) D1-98a
CH2SCH2(D1-95a) D1-108a
CH2SCH2(D1-95a) D1-108b (Z = 2-Cl)
CH2SCH2(D1-95a) D1-108b (Z = 3-Me)
CH2SCH2(D1-95a) D1-108b (Z = 4-OMe)
CH2SCH2(D1-95a) D1-108b (Z = 2-SMe)
CH2SCH2(D1-95a) D1-108b (Z = 3-CFThree)
CH2SCH2(D1-95a) D1-108b (Z = 4-OCFThree)
CH2SCH2(D1-95a) D1-108b (Z = 2-SCFThree)
CH2SCH2(D1-95a) C (O) Me
CH2SCH2(D1-95a) C (O) CFThree
CH2SCH2(D1-95a) C (O) OMe
CH2S (O) CH2(D1-95a) Me
CH2S (O) CH2(D1-95a) Et
CH2S (O) CH2(D1-95a) Pr-n
CH2S (O) CH2(D1-95a) Pr-i
CH2S (O) CH2(D1-95a) Pr-c
CH2S (O) CH2(D1-95a) Bu-n
CH2S (O) CH2(D1-95a) Bu-i
CH2S (O) CH2(D1-95a) Bu-c
CH2S (O) CH2(D1-95a) Bu-s
CH2S (O) CH2(D1-95a) Bu-t
CH2S (O) CH2(D1-95a) Pen-n
CH2S (O) CH2(D1-95a) Pen-c
CH2S (O) CH2(D1-95a) Hex-n
CH2S (O) CH2(D1-95a) Hex-c
CH2S (O) CH2(D1-95a) CH2Pr-c
CH2S (O) CH2(D1-95a) CH2Bu-c
CH2S (O) CH2(D1-95a) CH2Pen-c
CH2S (O) CH2(D1-95a) CH2Hex-c
CH2S (O) CH2(D1-95a) CH2CH = CH2
CH2S (O) CH2(D1-95a) CH2CH = C (Cl)2
CH2S (O) CH2(D1-95a) CH2C≡CH
CH2S (O) CH2(D1-95a) CH2CN
CH2S (O) CH2(D1-95a) CH2CFThree
CH2S (O) CH2(D1-95a) CH2OMe
CH2S (O) CH2(D1-95a) CH2OCFThree
CH2S (O) CH2(D1-95a) CH2SMe
CH2S (O) CH2(D1-95a) CH2S (O) Me
CH2S (O) CH2(D1-95a) CH2S (O)2Me
CH2S (O) CH2(D1-95a) CH2SCFThree
CH2S (O) CH2(D1-95a) CH2S (O) CFThree
CH2S (O) CH2(D1-95a) CH2S (O)2CFThree
CH2S (O) CH2(D1-95a) CH2CH (OMe)2
CH2S (O) CH2(D1-95a) CH2CH (SMe)2
CH2S (O) CH2(D1-95a) CH2C (O) Me
CH2S (O) CH2(D1-95a) CH2C (O) CFThree
CH2S (O) CH2(D1-95a) CH2C (O) OMe
CH2S (O) CH2(D1-95a) CH2(D1-32a)
CH2S (O) CH2(D1-95a) CH2(D1-33a)
CH2S (O) CH2(D1-95a) CH2(D1-34a)
CH2S (O) CH2(D1-95a) CH2(D1-37a)
CH2S (O) CH2(D1-95a) CH2(D1-81a)
CH2S (O) CH2(D1-95a) CH2(D1-82a)
CH2S (O) CH2(D1-95a) CH2(D1-84a)
CH2S (O) CH2(D1-95a) CH2(D1-85a)
CH2S (O) CH2(D1-95a) CH2(D1-87a)
CH2S (O) CH2(D1-95a) CH2(D1-92a)
CH2S (O) CH2(D1-95a) CH2(D1-93a)
CH2S (O) CH2(D1-95a) CH2(D1-95a)
CH2S (O) CH2(D1-95a) CH2(D1-96a)
CH2S (O) CH2(D1-95a) CH2(D1-98a)
CH2S (O) CH2(D1-95a) CH2(D1-108a)
CH2S (O) CH2(D1-95a) CH2(D1-108b, Z = 2-Cl)
CH2S (O) CH2(D1-95a) CH2(D1-108b, Z = 3-Me)
CH2S (O) CH2(D1-95a) CH2(D1-108b, Z = 4-OMe)
CH2S (O) CH2(D1-95a) CH2(D1-108b, Z = 2-SMe)
CH2S (O) CH2(D1-95a) CH2(D1-108b, Z = 3-CFThree)
CH2S (O) CH2(D1-95a) CH2(D1-108b, Z = 4-OCFThree)
CH2S (O) CH2(D1-95a) CH2(D1-108b, Z = 2-SCFThree)
CH2S (O) CH2(D1-95a) CH2CH2CN
CH2S (O) CH2(D1-95a) CH2CH2CFThree
CH2S (O) CH2(D1-95a) CH2CH2OMe
CH2S (O) CH2(D1-95a) CH2CH2SMe
CH2S (O) CH2(D1-95a) CH2CH2S (O) Me
CH2S (O) CH2(D1-95a) CH2CH2S (O)2Me
CH2S (O) CH2(D1-95a) D1-32a
CH2S (O) CH2(D1-95a) D1-33a
CH2S (O) CH2(D1-95a) D1-34a
CH2S (O) CH2(D1-95a) D1-37a
CH2S (O) CH2(D1-95a) D1-81a
CH2S (O) CH2(D1-95a) D1-82a
CH2S (O) CH2(D1-95a) D1-84a
CH2S (O) CH2(D1-95a) D1-85a
CH2S (O) CH2(D1-95a) D1-87a
CH2S (O) CH2(D1-95a) D1-92a
CH2S (O) CH2(D1-95a) D1-93a
CH2S (O) CH2(D1-95a) D1-95a
CH2S (O) CH2(D1-95a) D1-96a
CH2S (O) CH2(D1-95a) D1-98a
CH2S (O) CH2(D1-95a) D1-108a
CH2S (O) CH2(D1-95a) D1-108b (Z = 2-Cl)
CH2S (O) CH2(D1-95a) D1-108b (Z = 3-Me)
CH2S (O) CH2(D1-95a) D1-108b (Z = 4-OMe)
CH2S (O) CH2(D1-95a) D1-108b (Z = 2-SMe)
CH2S (O) CH2(D1-95a) D1-108b (Z = 3-CFThree)
CH2S (O) CH2(D1-95a) D1-108b (Z = 4-OCFThree)
CH2S (O) CH2(D1-95a) D1-108b (Z = 2-SCFThree)
CH2S (O) CH2(D1-95a) C (O) Me
CH2S (O) CH2(D1-95a) C (O) CFThree
CH2S (O) CH2(D1-95a) C (O) OMe
CH2S (O)2CH2(D1-95a) Me
CH2S (O)2CH2(D1-95a) Et
CH2S (O)2CH2(D1-95a) Pr-n
CH2S (O)2CH2(D1-95a) Pr-i
CH2S (O)2CH2(D1-95a) Pr-c
CH2S (O)2CH2(D1-95a) Bu-n
CH2S (O)2CH2(D1-95a) Bu-i
CH2S (O)2CH2(D1-95a) Bu-c
CH2S (O)2CH2(D1-95a) Bu-s
CH2S (O)2CH2(D1-95a) Bu-t
CH2S (O)2CH2(D1-95a) Pen-n
CH2S (O)2CH2(D1-95a) Pen-c
CH2S (O)2CH2(D1-95a) Hex-n
CH2S (O)2CH2(D1-95a) Hex-c
CH2S (O)2CH2(D1-95a) CH2Pr-c
CH2S (O)2CH2(D1-95a) CH2Bu-c
CH2S (O)2CH2(D1-95a) CH2Pen-c
CH2S (O)2CH2(D1-95a) CH2Hex-c
CH2S (O)2CH2(D1-95a) CH2CH = CH2
CH2S (O)2CH2(D1-95a) CH2CH = C (Cl)2
CH2S (O)2CH2(D1-95a) CH2C≡CH
CH2S (O)2CH2(D1-95a) CH2CN
CH2S (O)2CH2(D1-95a) CH2CFThree
CH2S (O)2CH2(D1-95a) CH2OMe
CH2S (O)2CH2(D1-95a) CH2OCFThree
CH2S (O)2CH2(D1-95a) CH2SMe
CH2S (O)2CH2(D1-95a) CH2S (O) Me
CH2S (O)2CH2(D1-95a) CH2S (O)2Me
CH2S (O)2CH2(D1-95a) CH2SCFThree
CH2S (O)2CH2(D1-95a) CH2S (O) CFThree
CH2S (O)2CH2(D1-95a) CH2S (O)2CFThree
CH2S (O)2CH2(D1-95a) CH2CH (OMe)2
CH2S (O)2CH2(D1-95a) CH2CH (SMe)2
CH2S (O)2CH2(D1-95a) CH2C (O) Me
CH2S (O)2CH2(D1-95a) CH2C (O) CFThree
CH2S (O)2CH2(D1-95a) CH2C (O) OMe
CH2S (O)2CH2(D1-95a) CH2(D1-32a)
CH2S (O)2CH2(D1-95a) CH2(D1-33a)
CH2S (O)2CH2(D1-95a) CH2(D1-34a)
CH2S (O)2CH2(D1-95a) CH2(D1-37a)
CH2S (O)2CH2(D1-95a) CH2(D1-81a)
CH2S (O)2CH2(D1-95a) CH2(D1-82a)
CH2S (O)2CH2(D1-95a) CH2(D1-84a)
CH2S (O)2CH2(D1-95a) CH2(D1-85a)
CH2S (O)2CH2(D1-95a) CH2(D1-87a)
CH2S (O)2CH2(D1-95a) CH2(D1-92a)
CH2S (O)2CH2(D1-95a) CH2(D1-93a)
CH2S (O)2CH2(D1-95a) CH2(D1-95a)
CH2S (O)2CH2(D1-95a) CH2(D1-96a)
CH2S (O)2CH2(D1-95a) CH2(D1-98a)
CH2S (O)2CH2(D1-95a) CH2(D1-108a)
CH2S (O)2CH2(D1-95a) CH2(D1-108b, Z = 2-Cl)
CH2S (O)2CH2(D1-95a) CH2(D1-108b, Z = 3-Me)
CH2S (O)2CH2(D1-95a) CH2(D1-108b, Z = 4-OMe)
CH2S (O)2CH2(D1-95a) CH2(D1-108b, Z = 2-SMe)
CH2S (O)2CH2(D1-95a) CH2(D1-108b, Z = 3-CFThree)
CH2S (O)2CH2(D1-95a) CH2(D1-108b, Z = 4-OCFThree)
CH2S (O)2CH2(D1-95a) CH2(D1-108b, Z = 2-SCFThree)
CH2S (O)2CH2(D1-95a) CH2CH2CN
CH2S (O)2CH2(D1-95a) CH2CH2CFThree
CH2S (O)2CH2(D1-95a) CH2CH2OMe
CH2S (O)2CH2(D1-95a) CH2CH2SMe
CH2S (O)2CH2(D1-95a) CH2CH2S (O) Me
CH2S (O)2CH2(D1-95a) CH2CH2S (O)2Me
CH2S (O)2CH2(D1-95a) D1-32a
CH2S (O)2CH2(D1-95a) D1-33a
CH2S (O)2CH2(D1-95a) D1-34a
CH2S (O)2CH2(D1-95a) D1-37a
CH2S (O)2CH2(D1-95a) D1-81a
CH2S (O)2CH2(D1-95a) D1-82a
CH2S (O)2CH2(D1-95a) D1-84a
CH2S (O)2CH2(D1-95a) D1-85a
CH2S (O)2CH2(D1-95a) D1-87a
CH2S (O)2CH2(D1-95a) D1-92a
CH2S (O)2CH2(D1-95a) D1-93a
CH2S (O)2CH2(D1-95a) D1-95a
CH2S (O)2CH2(D1-95a) D1-96a
CH2S (O)2CH2(D1-95a) D1-98a
CH2S (O)2CH2(D1-95a) D1-108a
CH2S (O)2CH2(D1-95a) D1-108b (Z = 2-Cl)
CH2S (O)2CH2(D1-95a) D1-108b (Z = 3-Me)
CH2S (O)2CH2(D1-95a) D1-108b (Z = 4-OMe)
CH2S (O)2CH2(D1-95a) D1-108b (Z = 2-SMe)
CH2S (O)2CH2(D1-95a) D1-108b (Z = 3-CFThree)
CH2S (O)2CH2(D1-95a) D1-108b (Z = 4-OCFThree)
CH2S (O)2CH2(D1-95a) D1-108b (Z = 2-SCFThree)
CH2SCH2(D1-96a) Me
CH2SCH2(D1-96a) Et
CH2SCH2(D1-96a) Pr-n
CH2SCH2(D1-96a) Pr-i
CH2SCH2(D1-96a) Pr-c
CH2SCH2(D1-96a) Bu-n
CH2SCH2(D1-96a) Bu-i
CH2SCH2(D1-96a) Bu-c
CH2SCH2(D1-96a) Bu-s
CH2SCH2(D1-96a) Bu-t
CH2SCH2(D1-96a) Pen-n
CH2SCH2(D1-96a) Pen-c
CH2SCH2(D1-96a) Hex-n
CH2SCH2(D1-96a) Hex-c
CH2SCH2(D1-96a) CH2Pr-c
CH2SCH2(D1-96a) CH2Bu-c
CH2SCH2(D1-96a) CH2Pen-c
CH2SCH2(D1-96a) CH2Hex-c
CH2SCH2(D1-96a) CH2CH = CH2
CH2SCH2(D1-96a) CH2CH = C (Cl)2
CH2SCH2(D1-96a) CH2C≡CH
CH2SCH2(D1-96a) CH2CN
CH2SCH2(D1-96a) CH2CFThree
CH2SCH2(D1-96a) CH2OMe
CH2SCH2(D1-96a) CH2OCFThree
CH2SCH2(D1-96a) CH2SMe
CH2SCH2(D1-96a) CH2S (O) Me
CH2SCH2(D1-96a) CH2S (O)2Me
CH2SCH2(D1-96a) CH2SCFThree
CH2SCH2(D1-96a) CH2S (O) CFThree
CH2SCH2(D1-96a) CH2S (O)2CFThree
CH2SCH2(D1-96a) CH2CH (OMe)2
CH2SCH2(D1-96a) CH2CH (SMe)2
CH2SCH2(D1-96a) CH2C (O) Me
CH2SCH2(D1-96a) CH2C (O) CFThree
CH2SCH2(D1-96a) CH2C (O) OMe
CH2SCH2(D1-96a) CH2(D1-32a)
CH2SCH2(D1-96a) CH2(D1-33a)
CH2SCH2(D1-96a) CH2(D1-34a)
CH2SCH2(D1-96a) CH2(D1-37a)
CH2SCH2(D1-96a) CH2(D1-81a)
CH2SCH2(D1-96a) CH2(D1-82a)
CH2SCH2(D1-96a) CH2(D1-84a)
CH2SCH2(D1-96a) CH2(D1-85a)
CH2SCH2(D1-96a) CH2(D1-87a)
CH2SCH2(D1-96a) CH2(D1-92a)
CH2SCH2(D1-96a) CH2(D1-93a)
CH2SCH2(D1-96a) CH2(D1-95a)
CH2SCH2(D1-96a) CH2(D1-96a)
CH2SCH2(D1-96a) CH2(D1-98a)
CH2SCH2(D1-96a) CH2(D1-108a)
CH2SCH2(D1-96a) CH2(D1-108b, Z = 2-Cl)
CH2SCH2(D1-96a) CH2(D1-108b, Z = 3-Me)
CH2SCH2(D1-96a) CH2(D1-108b, Z = 4-OMe)
CH2SCH2(D1-96a) CH2(D1-108b, Z = 2-SMe)
CH2SCH2(D1-96a) CH2(D1-108b, Z = 3-CFThree)
CH2SCH2(D1-96a) CH2(D1-108b, Z = 4-OCFThree)
CH2SCH2(D1-96a) CH2(D1-108b, Z = 2-SCFThree)
CH2SCH2(D1-96a) CH2CH2CN
CH2SCH2(D1-96a) CH2CH2CFThree
CH2SCH2(D1-96a) CH2CH2OMe
CH2SCH2(D1-96a) CH2CH2SMe
CH2SCH2(D1-96a) CH2CH2S (O) Me
CH2SCH2(D1-96a) CH2CH2S (O)2Me
CH2SCH2(D1-96a) D1-32a
CH2SCH2(D1-96a) D1-33a
CH2SCH2(D1-96a) D1-34a
CH2SCH2(D1-96a) D1-37a
CH2SCH2(D1-96a) D1-81a
CH2SCH2(D1-96a) D1-82a
CH2SCH2(D1-96a) D1-84a
CH2SCH2(D1-96a) D1-85a
CH2SCH2(D1-96a) D1-87a
CH2SCH2(D1-96a) D1-92a
CH2SCH2(D1-96a) D1-93a
CH2SCH2(D1-96a) D1-95a
CH2SCH2(D1-96a) D1-96a
CH2SCH2(D1-96a) D1-98a
CH2SCH2(D1-96a) D1-108a
CH2SCH2(D1-96a) D1-108b (Z = 2-Cl)
CH2SCH2(D1-96a) D1-108b (Z = 3-Me)
CH2SCH2(D1-96a) D1-108b (Z = 4-OMe)
CH2SCH2(D1-96a) D1-108b (Z = 2-SMe)
CH2SCH2(D1-96a) D1-108b (Z = 3-CFThree)
CH2SCH2(D1-96a) D1-108b (Z = 4-OCFThree)
CH2SCH2(D1-96a) D1-108b (Z = 2-SCFThree)
CH2SCH2(D1-96a) C (O) Me
CH2SCH2(D1-96a) C (O) CFThree
CH2SCH2(D1-96a) C (O) OMe
CH2S (O) CH2(D1-96a) Me
CH2S (O) CH2(D1-96a) Et
CH2S (O) CH2(D1-96a) Pr-n
CH2S (O) CH2(D1-96a) Pr-i
CH2S (O) CH2(D1-96a) Pr-c
CH2S (O) CH2(D1-96a) Bu-n
CH2S (O) CH2(D1-96a) Bu-i
CH2S (O) CH2(D1-96a) Bu-c
CH2S (O) CH2(D1-96a) Bu-s
CH2S (O) CH2(D1-96a) Bu-t
CH2S (O) CH2(D1-96a) Pen-n
CH2S (O) CH2(D1-96a) Pen-c
CH2S (O) CH2(D1-96a) Hex-n
CH2S (O) CH2(D1-96a) Hex-c
CH2S (O) CH2(D1-96a) CH2Pr-c
CH2S (O) CH2(D1-96a) CH2Bu-c
CH2S (O) CH2(D1-96a) CH2Pen-c
CH2S (O) CH2(D1-96a) CH2Hex-c
CH2S (O) CH2(D1-96a) CH2CH = CH2
CH2S (O) CH2(D1-96a) CH2CH = C (Cl)2
CH2S (O) CH2(D1-96a) CH2C≡CH
CH2S (O) CH2(D1-96a) CH2CN
CH2S (O) CH2(D1-96a) CH2CFThree
CH2S (O) CH2(D1-96a) CH2OMe
CH2S (O) CH2(D1-96a) CH2OCFThree
CH2S (O) CH2(D1-96a) CH2SMe
CH2S (O) CH2(D1-96a) CH2S (O) Me
CH2S (O) CH2(D1-96a) CH2S (O)2Me
CH2S (O) CH2(D1-96a) CH2SCFThree
CH2S (O) CH2(D1-96a) CH2S (O) CFThree
CH2S (O) CH2(D1-96a) CH2S (O)2CFThree
CH2S (O) CH2(D1-96a) CH2CH (OMe)2
CH2S (O) CH2(D1-96a) CH2CH (SMe)2
CH2S (O) CH2(D1-96a) CH2C (O) Me
CH2S (O) CH2(D1-96a) CH2C (O) CFThree
CH2S (O) CH2(D1-96a) CH2C (O) OMe
CH2S (O) CH2(D1-96a) CH2(D1-32a)
CH2S (O) CH2(D1-96a) CH2(D1-33a)
CH2S (O) CH2(D1-96a) CH2(D1-34a)
CH2S (O) CH2(D1-96a) CH2(D1-37a)
CH2S (O) CH2(D1-96a) CH2(D1-81a)
CH2S (O) CH2(D1-96a) CH2(D1-82a)
CH2S (O) CH2(D1-96a) CH2(D1-84a)
CH2S (O) CH2(D1-96a) CH2(D1-85a)
CH2S (O) CH2(D1-96a) CH2(D1-87a)
CH2S (O) CH2(D1-96a) CH2(D1-92a)
CH2S (O) CH2(D1-96a) CH2(D1-93a)
CH2S (O) CH2(D1-96a) CH2(D1-95a)
CH2S (O) CH2(D1-96a) CH2(D1-96a)
CH2S (O) CH2(D1-96a) CH2(D1-98a)
CH2S (O) CH2(D1-96a) CH2(D1-108a)
CH2S (O) CH2(D1-96a) CH2(D1-108b, Z = 2-Cl)
CH2S (O) CH2(D1-96a) CH2(D1-108b, Z = 3-Me)
CH2S (O) CH2(D1-96a) CH2(D1-108b, Z = 4-OMe)
CH2S (O) CH2(D1-96a) CH2(D1-108b, Z = 2-SMe)
CH2S (O) CH2(D1-96a) CH2(D1-108b, Z = 3-CFThree)
CH2S (O) CH2(D1-96a) CH2(D1-108b, Z = 4-OCFThree)
CH2S (O) CH2(D1-96a) CH2(D1-108b, Z = 2-SCFThree)
CH2S (O) CH2(D1-96a) CH2CH2CN
CH2S (O) CH2(D1-96a) CH2CH2CFThree
CH2S (O) CH2(D1-96a) CH2CH2OMe
CH2S (O) CH2(D1-96a) CH2CH2SMe
CH2S (O) CH2(D1-96a) CH2CH2S (O) Me
CH2S (O) CH2(D1-96a) CH2CH2S (O)2Me
CH2S (O) CH2(D1-96a) D1-32a
CH2S (O) CH2(D1-96a) D1-33a
CH2S (O) CH2(D1-96a) D1-34a
CH2S (O) CH2(D1-96a) D1-37a
CH2S (O) CH2(D1-96a) D1-81a
CH2S (O) CH2(D1-96a) D1-82a
CH2S (O) CH2(D1-96a) D1-84a
CH2S (O) CH2(D1-96a) D1-85a
CH2S (O) CH2(D1-96a) D1-87a
CH2S (O) CH2(D1-96a) D1-92a
CH2S (O) CH2(D1-96a) D1-93a
CH2S (O) CH2(D1-96a) D1-95a
CH2S (O) CH2(D1-96a) D1-96a
CH2S (O) CH2(D1-96a) D1-98a
CH2S (O) CH2(D1-96a) D1-108a
CH2S (O) CH2(D1-96a) D1-108b (Z = 2-Cl)
CH2S (O) CH2(D1-96a) D1-108b (Z = 3-Me)
CH2S (O) CH2(D1-96a) D1-108b (Z = 4-OMe)
CH2S (O) CH2(D1-96a) D1-108b (Z = 2-SMe)
CH2S (O) CH2(D1-96a) D1-108b (Z = 3-CFThree)
CH2S (O) CH2(D1-96a) D1-108b (Z = 4-OCFThree)
CH2S (O) CH2(D1-96a) D1-108b (Z = 2-SCFThree)
CH2S (O) CH2(D1-96a) C (O) Me
CH2S (O) CH2(D1-96a) C (O) CFThree
CH2S (O) CH2(D1-96a) C (O) OMe
CH2S (O)2CH2(D1-96a) Me
CH2S (O)2CH2(D1-96a) Et
CH2S (O)2CH2(D1-96a) Pr-n
CH2S (O)2CH2(D1-96a) Pr-i
CH2S (O)2CH2(D1-96a) Pr-c
CH2S (O)2CH2(D1-96a) Bu-n
CH2S (O)2CH2(D1-96a) Bu-i
CH2S (O)2CH2(D1-96a) Bu-c
CH2S (O)2CH2(D1-96a) Bu-s
CH2S (O)2CH2(D1-96a) Bu-t
CH2S (O)2CH2(D1-96a) Pen-n
CH2S (O)2CH2(D1-96a) Pen-c
CH2S (O)2CH2(D1-96a) Hex-n
CH2S (O)2CH2(D1-96a) Hex-c
CH2S (O)2CH2(D1-96a) CH2Pr-c
CH2S (O)2CH2(D1-96a) CH2Bu-c
CH2S (O)2CH2(D1-96a) CH2Pen-c
CH2S (O)2CH2(D1-96a) CH2Hex-c
CH2S (O)2CH2(D1-96a) CH2CH = CH2
CH2S (O)2CH2(D1-96a) CH2CH = C (Cl)2
CH2S (O)2CH2(D1-96a) CH2C≡CH
CH2S (O)2CH2(D1-96a) CH2CN
CH2S (O)2CH2(D1-96a) CH2CFThree
CH2S (O)2CH2(D1-96a) CH2OMe
CH2S (O)2CH2(D1-96a) CH2OCFThree
CH2S (O)2CH2(D1-96a) CH2SMe
CH2S (O)2CH2(D1-96a) CH2S (O) Me
CH2S (O)2CH2(D1-96a) CH2S (O)2Me
CH2S (O)2CH2(D1-96a) CH2SCFThree
CH2S (O)2CH2(D1-96a) CH2S (O) CFThree
CH2S (O)2CH2(D1-96a) CH2S (O)2CFThree
CH2S (O)2CH2(D1-96a) CH2CH (OMe)2
CH2S (O)2CH2(D1-96a) CH2CH (SMe)2
CH2S (O)2CH2(D1-96a) CH2C (O) Me
CH2S (O)2CH2(D1-96a) CH2C (O) CFThree
CH2S (O)2CH2(D1-96a) CH2C (O) OMe
CH2S (O)2CH2(D1-96a) CH2(D1-32a)
CH2S (O)2CH2(D1-96a) CH2(D1-33a)
CH2S (O)2CH2(D1-96a) CH2(D1-34a)
CH2S (O)2CH2(D1-96a) CH2(D1-37a)
CH2S (O)2CH2(D1-96a) CH2(D1-81a)
CH2S (O)2CH2(D1-96a) CH2(D1-82a)
CH2S (O)2CH2(D1-96a) CH2(D1-84a)
CH2S (O)2CH2(D1-96a) CH2(D1-85a)
CH2S (O)2CH2(D1-96a) CH2(D1-87a)
CH2S (O)2CH2(D1-96a) CH2(D1-92a)
CH2S (O)2CH2(D1-96a) CH2(D1-93a)
CH2S (O)2CH2(D1-96a) CH2(D1-95a)
CH2S (O)2CH2(D1-96a) CH2(D1-96a)
CH2S (O)2CH2(D1-96a) CH2(D1-98a)
CH2S (O)2CH2(D1-96a) CH2(D1-108a)
CH2S (O)2CH2(D1-96a) CH2(D1-108b, Z = 2-Cl)
CH2S (O)2CH2(D1-96a) CH2(D1-108b, Z = 3-Me)
CH2S (O)2CH2(D1-96a) CH2(D1-108b, Z = 4-OMe)
CH2S (O)2CH2(D1-96a) CH2(D1-108b, Z = 2-SMe)
CH2S (O)2CH2(D1-96a) CH2(D1-108b, Z = 3-CFThree)
CH2S (O)2CH2(D1-96a) CH2(D1-108b, Z = 4-OCFThree)
CH2S (O)2CH2(D1-96a) CH2(D1-108b, Z = 2-SCFThree)
CH2S (O)2CH2(D1-96a) CH2CH2CN
CH2S (O)2CH2(D1-96a) CH2CH2CFThree
CH2S (O)2CH2(D1-96a) CH2CH2OMe
CH2S (O)2CH2(D1-96a) CH2CH2SMe
CH2S (O)2CH2(D1-96a) CH2CH2S (O) Me
CH2S (O)2CH2(D1-96a) CH2CH2S (O)2Me
CH2S (O)2CH2(D1-96a) D1-32a
CH2S (O)2CH2(D1-96a) D1-33a
CH2S (O)2CH2(D1-96a) D1-34a
CH2S (O)2CH2(D1-96a) D1-37a
CH2S (O)2CH2(D1-96a) D1-81a
CH2S (O)2CH2(D1-96a) D1-82a
CH2S (O)2CH2(D1-96a) D1-84a
CH2S (O)2CH2(D1-96a) D1-85a
CH2S (O)2CH2(D1-96a) D1-87a
CH2S (O)2CH2(D1-96a) D1-92a
CH2S (O)2CH2(D1-96a) D1-93a
CH2S (O)2CH2(D1-96a) D1-95a
CH2S (O)2CH2(D1-96a) D1-96a
CH2S (O)2CH2(D1-96a) D1-98a
CH2S (O)2CH2(D1-96a) D1-108a
CH2S (O)2CH2(D1-96a) D1-108b (Z = 2-Cl)
CH2S (O)2CH2(D1-96a) D1-108b (Z = 3-Me)
CH2S (O)2CH2(D1-96a) D1-108b (Z = 4-OMe)
CH2S (O)2CH2(D1-96a) D1-108b (Z = 2-SMe)
CH2S (O)2CH2(D1-96a) D1-108b (Z = 3-CFThree)
CH2S (O)2CH2(D1-96a) D1-108b (Z = 4-OCFThree)
CH2S (O)2CH2(D1-96a) D1-108b (Z = 2-SCFThree)
CH2SCH2(D1-98a) Me
CH2SCH2(D1-98a) Et
CH2SCH2(D1-98a) Pr-n
CH2SCH2(D1-98a) Pr-i
CH2SCH2(D1-98a) Pr-c
CH2SCH2(D1-98a) Bu-n
CH2SCH2(D1-98a) Bu-i
CH2SCH2(D1-98a) Bu-c
CH2SCH2(D1-98a) Bu-s
CH2SCH2(D1-98a) Bu-t
CH2SCH2(D1-98a) Pen-n
CH2SCH2(D1-98a) Pen-c
CH2SCH2(D1-98a) Hex-n
CH2SCH2(D1-98a) Hex-c
CH2SCH2(D1-98a) CH2Pr-c
CH2SCH2(D1-98a) CH2Bu-c
CH2SCH2(D1-98a) CH2Pen-c
CH2SCH2(D1-98a) CH2Hex-c
CH2SCH2(D1-98a) CH2CH = CH2
CH2SCH2(D1-98a) CH2CH = C (Cl)2
CH2SCH2(D1-98a) CH2C≡CH
CH2SCH2(D1-98a) CH2CN
CH2SCH2(D1-98a) CH2CFThree
CH2SCH2(D1-98a) CH2OMe
CH2SCH2(D1-98a) CH2OCFThree
CH2SCH2(D1-98a) CH2SMe
CH2SCH2(D1-98a) CH2S (O) Me
CH2SCH2(D1-98a) CH2S (O)2Me
CH2SCH2(D1-98a) CH2SCFThree
CH2SCH2(D1-98a) CH2S (O) CFThree
CH2SCH2(D1-98a) CH2S (O)2CFThree
CH2SCH2(D1-98a) CH2CH (OMe)2
CH2SCH2(D1-98a) CH2CH (SMe)2
CH2SCH2(D1-98a) CH2C (O) Me
CH2SCH2(D1-98a) CH2C (O) CFThree
CH2SCH2(D1-98a) CH2C (O) OMe
CH2SCH2(D1-98a) CH2(D1-32a)
CH2SCH2(D1-98a) CH2(D1-33a)
CH2SCH2(D1-98a) CH2(D1-34a)
CH2SCH2(D1-98a) CH2(D1-37a)
CH2SCH2(D1-98a) CH2(D1-81a)
CH2SCH2(D1-98a) CH2(D1-82a)
CH2SCH2(D1-98a) CH2(D1-84a)
CH2SCH2(D1-98a) CH2(D1-85a)
CH2SCH2(D1-98a) CH2(D1-87a)
CH2SCH2(D1-98a) CH2(D1-92a)
CH2SCH2(D1-98a) CH2(D1-93a)
CH2SCH2(D1-98a) CH2(D1-95a)
CH2SCH2(D1-98a) CH2(D1-96a)
CH2SCH2(D1-98a) CH2(D1-98a)
CH2SCH2(D1-98a) CH2(D1-108a)
CH2SCH2(D1-98a) CH2(D1-108b, Z = 2-Cl)
CH2SCH2(D1-98a) CH2(D1-108b, Z = 3-Me)
CH2SCH2(D1-98a) CH2(D1-108b, Z = 4-OMe)
CH2SCH2(D1-98a) CH2(D1-108b, Z = 2-SMe)
CH2SCH2(D1-98a) CH2(D1-108b, Z = 3-CFThree)
CH2SCH2(D1-98a) CH2(D1-108b, Z = 4-OCFThree)
CH2SCH2(D1-98a) CH2(D1-108b, Z = 2-SCFThree)
CH2SCH2(D1-98a) CH2CH2CN
CH2SCH2(D1-98a) CH2CH2CFThree
CH2SCH2(D1-98a) CH2CH2OMe
CH2SCH2(D1-98a) CH2CH2SMe
CH2SCH2(D1-98a) CH2CH2S (O) Me
CH2SCH2(D1-98a) CH2CH2S (O)2Me
CH2SCH2(D1-98a) D1-32a
CH2SCH2(D1-98a) D1-33a
CH2SCH2(D1-98a) D1-34a
CH2SCH2(D1-98a) D1-37a
CH2SCH2(D1-98a) D1-81a
CH2SCH2(D1-98a) D1-82a
CH2SCH2(D1-98a) D1-84a
CH2SCH2(D1-98a) D1-85a
CH2SCH2(D1-98a) D1-87a
CH2SCH2(D1-98a) D1-92a
CH2SCH2(D1-98a) D1-93a
CH2SCH2(D1-98a) D1-95a
CH2SCH2(D1-98a) D1-96a
CH2SCH2(D1-98a) D1-98a
CH2SCH2(D1-98a) D1-108a
CH2SCH2(D1-98a) D1-108b (Z = 2-Cl)
CH2SCH2(D1-98a) D1-108b (Z = 3-Me)
CH2SCH2(D1-98a) D1-108b (Z = 4-OMe)
CH2SCH2(D1-98a) D1-108b (Z = 2-SMe)
CH2SCH2(D1-98a) D1-108b (Z = 3-CFThree)
CH2SCH2(D1-98a) D1-108b (Z = 4-OCFThree)
CH2SCH2(D1-98a) D1-108b (Z = 2-SCFThree)
CH2SCH2(D1-98a) C (O) Me
CH2SCH2(D1-98a) C (O) CFThree
CH2SCH2(D1-98a) C (O) OMe
CH2S (O) CH2(D1-98a) Me
CH2S (O) CH2(D1-98a) Et
CH2S (O) CH2(D1-98a) Pr-n
CH2S (O) CH2(D1-98a) Pr-i
CH2S (O) CH2(D1-98a) Pr-c
CH2S (O) CH2(D1-98a) Bu-n
CH2S (O) CH2(D1-98a) Bu-i
CH2S (O) CH2(D1-98a) Bu-c
CH2S (O) CH2(D1-98a) Bu-s
CH2S (O) CH2(D1-98a) Bu-t
CH2S (O) CH2(D1-98a) Pen-n
CH2S (O) CH2(D1-98a) Pen-c
CH2S (O) CH2(D1-98a) Hex-n
CH2S (O) CH2(D1-98a) Hex-c
CH2S (O) CH2(D1-98a) CH2Pr-c
CH2S (O) CH2(D1-98a) CH2Bu-c
CH2S (O) CH2(D1-98a) CH2Pen-c
CH2S (O) CH2(D1-98a) CH2Hex-c
CH2S (O) CH2(D1-98a) CH2CH = CH2
CH2S (O) CH2(D1-98a) CH2CH = C (Cl)2
CH2S (O) CH2(D1-98a) CH2C≡CH
CH2S (O) CH2(D1-98a) CH2CN
CH2S (O) CH2(D1-98a) CH2CFThree
CH2S (O) CH2(D1-98a) CH2OMe
CH2S (O) CH2(D1-98a) CH2OCFThree
CH2S (O) CH2(D1-98a) CH2SMe
CH2S (O) CH2(D1-98a) CH2S (O) Me
CH2S (O) CH2(D1-98a) CH2S (O)2Me
CH2S (O) CH2(D1-98a) CH2SCFThree
CH2S (O) CH2(D1-98a) CH2S (O) CFThree
CH2S (O) CH2(D1-98a) CH2S (O)2CFThree
CH2S (O) CH2(D1-98a) CH2CH (OMe)2
CH2S (O) CH2(D1-98a) CH2CH (SMe)2
CH2S (O) CH2(D1-98a) CH2C (O) Me
CH2S (O) CH2(D1-98a) CH2C (O) CFThree
CH2S (O) CH2(D1-98a) CH2C (O) OMe
CH2S (O) CH2(D1-98a) CH2(D1-32a)
CH2S (O) CH2(D1-98a) CH2(D1-33a)
CH2S (O) CH2(D1-98a) CH2(D1-34a)
CH2S (O) CH2(D1-98a) CH2(D1-37a)
CH2S (O) CH2(D1-98a) CH2(D1-81a)
CH2S (O) CH2(D1-98a) CH2(D1-82a)
CH2S (O) CH2(D1-98a) CH2(D1-84a)
CH2S (O) CH2(D1-98a) CH2(D1-85a)
CH2S (O) CH2(D1-98a) CH2(D1-87a)
CH2S (O) CH2(D1-98a) CH2(D1-92a)
CH2S (O) CH2(D1-98a) CH2(D1-93a)
CH2S (O) CH2(D1-98a) CH2(D1-95a)
CH2S (O) CH2(D1-98a) CH2(D1-96a)
CH2S (O) CH2(D1-98a) CH2(D1-98a)
CH2S (O) CH2(D1-98a) CH2(D1-108a)
CH2S (O) CH2(D1-98a) CH2(D1-108b, Z = 2-Cl)
CH2S (O) CH2(D1-98a) CH2(D1-108b, Z = 3-Me)
CH2S (O) CH2(D1-98a) CH2(D1-108b, Z = 4-OMe)
CH2S (O) CH2(D1-98a) CH2(D1-108b, Z = 2-SMe)
CH2S (O) CH2(D1-98a) CH2(D1-108b, Z = 3-CFThree)
CH2S (O) CH2(D1-98a) CH2(D1-108b, Z = 4-OCFThree)
CH2S (O) CH2(D1-98a) CH2(D1-108b, Z = 2-SCFThree)
CH2S (O) CH2(D1-98a) CH2CH2CN
CH2S (O) CH2(D1-98a) CH2CH2CFThree
CH2S (O) CH2(D1-98a) CH2CH2OMe
CH2S (O) CH2(D1-98a) CH2CH2SMe
CH2S (O) CH2(D1-98a) CH2CH2S (O) Me
CH2S (O) CH2(D1-98a) CH2CH2S (O)2Me
CH2S (O) CH2(D1-98a) D1-32a
CH2S (O) CH2(D1-98a) D1-33a
CH2S (O) CH2(D1-98a) D1-34a
CH2S (O) CH2(D1-98a) D1-37a
CH2S (O) CH2(D1-98a) D1-81a
CH2S (O) CH2(D1-98a) D1-82a
CH2S (O) CH2(D1-98a) D1-84a
CH2S (O) CH2(D1-98a) D1-85a
CH2S (O) CH2(D1-98a) D1-87a
CH2S (O) CH2(D1-98a) D1-92a
CH2S (O) CH2(D1-98a) D1-93a
CH2S (O) CH2(D1-98a) D1-95a
CH2S (O) CH2(D1-98a) D1-96a
CH2S (O) CH2(D1-98a) D1-98a
CH2S (O) CH2(D1-98a) D1-108a
CH2S (O) CH2(D1-98a) D1-108b (Z = 2-Cl)
CH2S (O) CH2(D1-98a) D1-108b (Z = 3-Me)
CH2S (O) CH2(D1-98a) D1-108b (Z = 4-OMe)
CH2S (O) CH2(D1-98a) D1-108b (Z = 2-SMe)
CH2S (O) CH2(D1-98a) D1-108b (Z = 3-CFThree)
CH2S (O) CH2(D1-98a) D1-108b (Z = 4-OCFThree)
CH2S (O) CH2(D1-98a) D1-108b (Z = 2-SCFThree)
CH2S (O) CH2(D1-98a) C (O) Me
CH2S (O) CH2(D1-98a) C (O) CFThree
CH2S (O) CH2(D1-98a) C (O) OMe
CH2S (O)2CH2(D1-98a) Me
CH2S (O)2CH2(D1-98a) Et
CH2S (O)2CH2(D1-98a) Pr-n
CH2S (O)2CH2(D1-98a) Pr-i
CH2S (O)2CH2(D1-98a) Pr-c
CH2S (O)2CH2(D1-98a) Bu-n
CH2S (O)2CH2(D1-98a) Bu-i
CH2S (O)2CH2(D1-98a) Bu-c
CH2S (O)2CH2(D1-98a) Bu-s
CH2S (O)2CH2(D1-98a) Bu-t
CH2S (O)2CH2(D1-98a) Pen-n
CH2S (O)2CH2(D1-98a) Pen-c
CH2S (O)2CH2(D1-98a) Hex-n
CH2S (O)2CH2(D1-98a) Hex-c
CH2S (O)2CH2(D1-98a) CH2Pr-c
CH2S (O)2CH2(D1-98a) CH2Bu-c
CH2S (O)2CH2(D1-98a) CH2Pen-c
CH2S (O)2CH2(D1-98a) CH2Hex-c
CH2S (O)2CH2(D1-98a) CH2CH = CH2
CH2S (O)2CH2(D1-98a) CH2CH = C (Cl)2
CH2S (O)2CH2(D1-98a) CH2C≡CH
CH2S (O)2CH2(D1-98a) CH2CN
CH2S (O)2CH2(D1-98a) CH2CFThree
CH2S (O)2CH2(D1-98a) CH2OMe
CH2S (O)2CH2(D1-98a) CH2OCFThree
CH2S (O)2CH2(D1-98a) CH2SMe
CH2S (O)2CH2(D1-98a) CH2S (O) Me
CH2S (O)2CH2(D1-98a) CH2S (O)2Me
CH2S (O)2CH2(D1-98a) CH2SCFThree
CH2S (O)2CH2(D1-98a) CH2S (O) CFThree
CH2S (O)2CH2(D1-98a) CH2S (O)2CFThree
CH2S (O)2CH2(D1-98a) CH2CH (OMe)2
CH2S (O)2CH2(D1-98a) CH2CH (SMe)2
CH2S (O)2CH2(D1-98a) CH2C (O) Me
CH2S (O)2CH2(D1-98a) CH2C (O) CFThree
CH2S (O)2CH2(D1-98a) CH2C (O) OMe
CH2S (O)2CH2(D1-98a) CH2(D1-32a)
CH2S (O)2CH2(D1-98a) CH2(D1-33a)
CH2S (O)2CH2(D1-98a) CH2(D1-34a)
CH2S (O)2CH2(D1-98a) CH2(D1-37a)
CH2S (O)2CH2(D1-98a) CH2(D1-81a)
CH2S (O)2CH2(D1-98a) CH2(D1-82a)
CH2S (O)2CH2(D1-98a) CH2(D1-84a)
CH2S (O)2CH2(D1-98a) CH2(D1-85a)
CH2S (O)2CH2(D1-98a) CH2(D1-87a)
CH2S (O)2CH2(D1-98a) CH2(D1-92a)
CH2S (O)2CH2(D1-98a) CH2(D1-93a)
CH2S (O)2CH2(D1-98a) CH2(D1-95a)
CH2S (O)2CH2(D1-98a) CH2(D1-96a)
CH2S (O)2CH2(D1-98a) CH2(D1-98a)
CH2S (O)2CH2(D1-98a) CH2(D1-108a)
CH2S (O)2CH2(D1-98a) CH2(D1-108b, Z = 2-Cl)
CH2S (O)2CH2(D1-98a) CH2(D1-108b, Z = 3-Me)
CH2S (O)2CH2(D1-98a) CH2(D1-108b, Z = 4-OMe)
CH2S (O)2CH2(D1-98a) CH2(D1-108b, Z = 2-SMe)
CH2S (O)2CH2(D1-98a) CH2(D1-108b, Z = 3-CFThree)
CH2S (O)2CH2(D1-98a) CH2(D1-108b, Z = 4-OCFThree)
CH2S (O)2CH2(D1-98a) CH2(D1-108b, Z = 2-SCFThree)
CH2S (O)2CH2(D1-98a) CH2CH2CN
CH2S (O)2CH2(D1-98a) CH2CH2CFThree
CH2S (O)2CH2(D1-98a) CH2CH2OMe
CH2S (O)2CH2(D1-98a) CH2CH2SMe
CH2S (O)2CH2(D1-98a) CH2CH2S (O) Me
CH2S (O)2CH2(D1-98a) CH2CH2S (O)2Me
CH2S (O)2CH2(D1-98a) D1-32a
CH2S (O)2CH2(D1-98a) D1-33a
CH2S (O)2CH2(D1-98a) D1-34a
CH2S (O)2CH2(D1-98a) D1-37a
CH2S (O)2CH2(D1-98a) D1-81a
CH2S (O)2CH2(D1-98a) D1-82a
CH2S (O)2CH2(D1-98a) D1-84a
CH2S (O)2CH2(D1-98a) D1-85a
CH2S (O)2CH2(D1-98a) D1-87a
CH2S (O)2CH2(D1-98a) D1-92a
CH2S (O)2CH2(D1-98a) D1-93a
CH2S (O)2CH2(D1-98a) D1-95a
CH2S (O)2CH2(D1-98a) D1-96a
CH2S (O)2CH2(D1-98a) D1-98a
CH2S (O)2CH2(D1-98a) D1-108a
CH2S (O)2CH2(D1-98a) D1-108b (Z = 2-Cl)
CH2S (O)2CH2(D1-98a) D1-108b (Z = 3-Me)
CH2S (O)2CH2(D1-98a) D1-108b (Z = 4-OMe)
CH2S (O)2CH2(D1-98a) D1-108b (Z = 2-SMe)
CH2S (O)2CH2(D1-98a) D1-108b (Z = 3-CFThree)
CH2S (O)2CH2(D1-98a) D1-108b (Z = 4-OCFThree)
CH2S (O)2CH2(D1-98a) D1-108b (Z = 2-SCFThree)
CH2SH H
CH2SH Me
CH2SH Et
CH2SH Pr-n
CH2SH Pr-i
CH2SH Pr-c
CH2SH Bu-n
CH2SH Bu-i
CH2SH Bu-c
CH2SH Bu-s
CH2SH Bu-t
CH2SH Pen-n
CH2SH Pen-c
CH2SH Hex-n
CH2SH Hex-c
CH2SH CH2Pr-c
CH2SH CH2Bu-c
CH2SH CH2Pen-c
CH2SH CH2Hex-c
CH2SH CH2CH = CH2
CH2SH CH2CH = C (Cl)2
CH2SH CH2C≡CH
CH2SH CH2CN
CH2SH CH2CFThree
CH2SH CH2OMe
CH2SH CH2OCFThree
CH2SH CH2SMe
CH2SH CH2S (O) Me
CH2SH CH2S (O)2Me
CH2SH CH2SCFThree
CH2SH CH2S (O) CFThree
CH2SH CH2S (O)2CFThree
CH2SH CH2CH (OMe)2
CH2SH CH2CH (SMe)2
CH2SH CH2C (O) Me
CH2SH CH2C (O) CFThree
CH2SH CH2C (O) OMe
CH2SH CH2(D1-32a)
CH2SH CH2(D1-33a)
CH2SH CH2(D1-34a)
CH2SH CH2(D1-37a)
CH2SH CH2(D1-81a)
CH2SH CH2(D1-82a)
CH2SH CH2(D1-84a)
CH2SH CH2(D1-85a)
CH2SH CH2(D1-87a)
CH2SH CH2(D1-92a)
CH2SH CH2(D1-93a)
CH2SH CH2(D1-95a)
CH2SH CH2(D1-96a)
CH2SH CH2(D1-98a)
CH2SH CH2(D1-108a)
CH2SH CH2(D1-108b, Z = 2-Cl)
CH2SH CH2(D1-108b, Z = 3-Me)
CH2SH CH2(D1-108b, Z = 4-OMe)
CH2SH CH2(D1-108b, Z = 2-SMe)
CH2SH CH2(D1-108b, Z = 3-CFThree)
CH2SH CH2(D1-108b, Z = 4-OCFThree)
CH2SH CH2(D1-108b, Z = 2-SCFThree)
CH2SH CH2CH2CN
CH2SH CH2CH2CFThree
CH2SH CH2CH2OMe
CH2SH CH2CH2SMe
CH2SH CH2CH2S (O) Me
CH2SH CH2CH2S (O)2Me
CH2SH D1-32a
CH2SH D1-33a
CH2SH D1-34a
CH2SH D1-37a
CH2SH D1-81a
CH2SH D1-82a
CH2SH D1-84a
CH2SH D1-85a
CH2SH D1-87a
CH2SH D1-92a
CH2SH D1-93a
CH2SH D1-95a
CH2SH D1-96a
CH2SH D1-98a
CH2SH D1-108a
CH2SH D1-108b (Z = 2-Cl)
CH2SH D1-108b (Z = 3-Me)
CH2SH D1-108b (Z = 4-OMe)
CH2SH D1-108b (Z = 2-SMe)
CH2SH D1-108b (Z = 3-CFThree)
CH2SH D1-108b (Z = 4-OCFThree)
CH2SH D1-108b (Z = 2-SCFThree)
CH2SH C (O) Me
CH2SH C (O) CFThree
CH2SH C (O) OMe
CH (Me) SH H
CH (Me) SH Me
CH (Me) SH Et
CH (Me) SH Pr-n
CH (Me) SH Pr-i
CH (Me) SH Pr-c
CH (Me) SH Bu-n
CH (Me) SH Bu-i
CH (Me) SH Bu-c
CH (Me) SH Bu-s
CH (Me) SH Bu-t
CH (Me) SH Pen-n
CH (Me) SH Pen-c
CH (Me) SH Hex-n
CH (Me) SH Hex-c
CH (Me) SH CH2Pr-c
CH (Me) SH CH2Bu-c
CH (Me) SH CH2Pen-c
CH (Me) SH CH2Hex-c
CH (Me) SH CH2CH = CH2
CH (Me) SH CH2CH = C (Cl)2
CH (Me) SH CH2C≡CH
CH (Me) SH CH2CN
CH (Me) SH CH2CFThree
CH (Me) SH CH2OMe
CH (Me) SH CH2OCFThree
CH (Me) SH CH2SMe
CH (Me) SH CH2S (O) Me
CH (Me) SH CH2S (O)2Me
CH (Me) SH CH2SCFThree
CH (Me) SH CH2S (O) CFThree
CH (Me) SH CH2S (O)2CFThree
CH (Me) SH CH2CH (OMe)2
CH (Me) SH CH2CH (SMe)2
CH (Me) SH CH2C (O) Me
CH (Me) SH CH2C (O) CFThree
CH (Me) SH CH2C (O) OMe
CH (Me) SH CH2(D1-32a)
CH (Me) SH CH2(D1-33a)
CH (Me) SH CH2(D1-34a)
CH (Me) SH CH2(D1-37a)
CH (Me) SH CH2(D1-81a)
CH (Me) SH CH2(D1-82a)
CH (Me) SH CH2(D1-84a)
CH (Me) SH CH2(D1-85a)
CH (Me) SH CH2(D1-87a)
CH (Me) SH CH2(D1-92a)
CH (Me) SH CH2(D1-93a)
CH (Me) SH CH2(D1-95a)
CH (Me) SH CH2(D1-96a)
CH (Me) SH CH2(D1-98a)
CH (Me) SH CH2(D1-108a)
CH (Me) SH CH2(D1-108b, Z = 2-Cl)
CH (Me) SH CH2(D1-108b, Z = 3-Me)
CH (Me) SH CH2(D1-108b, Z = 4-OMe)
CH (Me) SH CH2(D1-108b, Z = 2-SMe)
CH (Me) SH CH2(D1-108b, Z = 3-CFThree)
CH (Me) SH CH2(D1-108b, Z = 4-OCFThree)
CH (Me) SH CH2(D1-108b, Z = 2-SCFThree)
CH (Me) SH CH2CH2CN
CH (Me) SH CH2CH2CFThree
CH (Me) SH CH2CH2OMe
CH (Me) SH CH2CH2SMe
CH (Me) SH CH2CH2S (O) Me
CH (Me) SH CH2CH2S (O)2Me
CH (Me) SH D1-32a
CH (Me) SH D1-33a
CH (Me) SH D1-34a
CH (Me) SH D1-37a
CH (Me) SH D1-81a
CH (Me) SH D1-82a
CH (Me) SH D1-84a
CH (Me) SH D1-85a
CH (Me) SH D1-87a
CH (Me) SH D1-92a
CH (Me) SH D1-93a
CH (Me) SH D1-95a
CH (Me) SH D1-96a
CH (Me) SH D1-98a
CH (Me) SH D1-108a
CH (Me) SH D1-108b (Z = 2-Cl)
CH (Me) SH D1-108b (Z = 3-Me)
CH (Me) SH D1-108b (Z = 4-OMe)
CH (Me) SH D1-108b (Z = 2-SMe)
CH (Me) SH D1-108b (Z = 3-CFThree)
CH (Me) SH D1-108b (Z = 4-OCFThree)
CH (Me) SH D1-108b (Z = 2-SCFThree)
CH (Me) SH C (O) Me
CH (Me) SH C (O) CFThree
CH (Me) SH C (O) OMe
CH (Et) SH H
CH (Et) SH Me
CH (Et) SH Et
CH (Et) SH Pr-n
CH (Et) SH Pr-i
CH (Et) SH Pr-c
CH (Et) SH Bu-n
CH (Et) SH Bu-i
CH (Et) SH Bu-c
CH (Et) SH Bu-s
CH (Et) SH Bu-t
CH (Et) SH Pen-n
CH (Et) SH Pen-c
CH (Et) SH Hex-n
CH (Et) SH Hex-c
CH (Et) SH CH2Pr-c
CH (Et) SH CH2Bu-c
CH (Et) SH CH2Pen-c
CH (Et) SH CH2Hex-c
CH (Et) SH CH2CH = CH2
CH (Et) SH CH2CH = C (Cl)2
CH (Et) SH CH2C≡CH
CH (Et) SH CH2CN
CH (Et) SH CH2CFThree
CH (Et) SH CH2OMe
CH (Et) SH CH2OCFThree
CH (Et) SH CH2SMe
CH (Et) SH CH2S (O) Me
CH (Et) SH CH2S (O)2Me
CH (Et) SH CH2SCFThree
CH (Et) SH CH2S (O) CFThree
CH (Et) SH CH2S (O)2CFThree
CH (Et) SH CH2CH (OMe)2
CH (Et) SH CH2CH (SMe)2
CH (Et) SH CH2C (O) Me
CH (Et) SH CH2C (O) CFThree
CH (Et) SH CH2C (O) OMe
CH (Et) SH CH2(D1-32a)
CH (Et) SH CH2(D1-33a)
CH (Et) SH CH2(D1-34a)
CH (Et) SH CH2(D1-37a)
CH (Et) SH CH2(D1-81a)
CH (Et) SH CH2(D1-82a)
CH (Et) SH CH2(D1-84a)
CH (Et) SH CH2(D1-85a)
CH (Et) SH CH2(D1-87a)
CH (Et) SH CH2(D1-92a)
CH (Et) SH CH2(D1-93a)
CH (Et) SH CH2(D1-95a)
CH (Et) SH CH2(D1-96a)
CH (Et) SH CH2(D1-98a)
CH (Et) SH CH2(D1-108a)
CH (Et) SH CH2(D1-108b, Z = 2-Cl)
CH (Et) SH CH2(D1-108b, Z = 3-Me)
CH (Et) SH CH2(D1-108b, Z = 4-OMe)
CH (Et) SH CH2(D1-108b, Z = 2-SMe)
CH (Et) SH CH2(D1-108b, Z = 3-CFThree)
CH (Et) SH CH2(D1-108b, Z = 4-OCFThree)
CH (Et) SH CH2(D1-108b, Z = 2-SCFThree)
CH (Et) SH CH2CH2CN
CH (Et) SH CH2CH2CFThree
CH (Et) SH CH2CH2OMe
CH (Et) SH CH2CH2SMe
CH (Et) SH CH2CH2S (O) Me
CH (Et) SH CH2CH2S (O)2Me
CH (Et) SH D1-32a
CH (Et) SH D1-33a
CH (Et) SH D1-34a
CH (Et) SH D1-37a
CH (Et) SH D1-81a
CH (Et) SH D1-82a
CH (Et) SH D1-84a
CH (Et) SH D1-85a
CH (Et) SH D1-87a
CH (Et) SH D1-92a
CH (Et) SH D1-93a
CH (Et) SH D1-95a
CH (Et) SH D1-96a
CH (Et) SH D1-98a
CH (Et) SH D1-108a
CH (Et) SH D1-108b (Z = 2-Cl)
CH (Et) SH D1-108b (Z = 3-Me)
CH (Et) SH D1-108b (Z = 4-OMe)
CH (Et) SH D1-108b (Z = 2-SMe)
CH (Et) SH D1-108b (Z = 3-CFThree)
CH (Et) SH D1-108b (Z = 4-OCFThree)
CH (Et) SH D1-108b (Z = 2-SCFThree)
CH (Et) SH C (O) Me
CH (Et) SH C (O) CFThree
CH (Et) SH C (O) OMe
CH2SC (O) Me H
CH2SC (O) Me Me
CH2SC (O) Me Et
CH2SC (O) Me Pr-n
CH2SC (O) Me Pr-i
CH2SC (O) Me Pr-c
CH2SC (O) Me Bu-n
CH2SC (O) Me Bu-i
CH2SC (O) Me Bu-c
CH2SC (O) Me Bu-s
CH2SC (O) Me Bu-t
CH2SC (O) Me Pen-n
CH2SC (O) Me Pen-c
CH2SC (O) Me Hex-n
CH2SC (O) Me Hex-c
CH2SC (O) Me CH2Pr-c
CH2SC (O) Me CH2Bu-c
CH2SC (O) Me CH2Pen-c
CH2SC (O) Me CH2Hex-c
CH2SC (O) Me CH2CH = CH2
CH2SC (O) Me CH2CH = C (Cl)2
CH2SC (O) Me CH2C≡CH
CH2SC (O) Me CH2CN
CH2SC (O) Me CH2CFThree
CH2SC (O) Me CH2OMe
CH2SC (O) Me CH2OCFThree
CH2SC (O) Me CH2SMe
CH2SC (O) Me CH2S (O) Me
CH2SC (O) Me CH2S (O)2Me
CH2SC (O) Me CH2SCFThree
CH2SC (O) Me CH2S (O) CFThree
CH2SC (O) Me CH2S (O)2CFThree
CH2SC (O) Me CH2CH (OMe)2
CH2SC (O) Me CH2CH (SMe)2
CH2SC (O) Me CH2C (O) Me
CH2SC (O) Me CH2C (O) CFThree
CH2SC (O) Me CH2C (O) OMe
CH2SC (O) Me CH2(D1-32a)
CH2SC (O) Me CH2(D1-33a)
CH2SC (O) Me CH2(D1-34a)
CH2SC (O) Me CH2(D1-37a)
CH2SC (O) Me CH2(D1-81a)
CH2SC (O) Me CH2(D1-82a)
CH2SC (O) Me CH2(D1-84a)
CH2SC (O) Me CH2(D1-85a)
CH2SC (O) Me CH2(D1-87a)
CH2SC (O) Me CH2(D1-92a)
CH2SC (O) Me CH2(D1-93a)
CH2SC (O) Me CH2(D1-95a)
CH2SC (O) Me CH2(D1-96a)
CH2SC (O) Me CH2(D1-98a)
CH2SC (O) Me CH2(D1-108a)
CH2SC (O) Me CH2(D1-108b, Z = 2-Cl)
CH2SC (O) Me CH2(D1-108b, Z = 3-Me)
CH2SC (O) Me CH2(D1-108b, Z = 4-OMe)
CH2SC (O) Me CH2(D1-108b, Z = 2-SMe)
CH2SC (O) Me CH2(D1-108b, Z = 3-CFThree)
CH2SC (O) Me CH2(D1-108b, Z = 4-OCFThree)
CH2SC (O) Me CH2(D1-108b, Z = 2-SCFThree)
CH2SC (O) Me CH2CH2CN
CH2SC (O) Me CH2CH2CFThree
CH2SC (O) Me CH2CH2OMe
CH2SC (O) Me CH2CH2SMe
CH2SC (O) Me CH2CH2S (O) Me
CH2SC (O) Me CH2CH2S (O)2Me
CH2SC (O) Me D1-32a
CH2SC (O) Me D1-33a
CH2SC (O) Me D1-34a
CH2SC (O) Me D1-37a
CH2SC (O) Me D1-81a
CH2SC (O) Me D1-82a
CH2SC (O) Me D1-84a
CH2SC (O) Me D1-85a
CH2SC (O) Me D1-87a
CH2SC (O) Me D1-92a
CH2SC (O) Me D1-93a
CH2SC (O) Me D1-95a
CH2SC (O) Me D1-96a
CH2SC (O) Me D1-98a
CH2SC (O) Me D1-108a
CH2SC (O) Me D1-108b (Z = 2-Cl)
CH2SC (O) Me D1-108b (Z = 3-Me)
CH2SC (O) Me D1-108b (Z = 4-OMe)
CH2SC (O) Me D1-108b (Z = 2-SMe)
CH2SC (O) Me D1-108b (Z = 3-CFThree)
CH2SC (O) Me D1-108b (Z = 4-OCFThree)
CH2SC (O) Me D1-108b (Z = 2-SCFThree)
CH2SC (O) Me C (O) Me
CH2SC (O) Me C (O) CFThree
CH2SC (O) Me C (O) OMe
CH (Me) SC (O) Me H
CH (Me) SC (O) Me Me
CH (Me) SC (O) Me Et
CH (Me) SC (O) Me Pr-n
CH (Me) SC (O) Me Pr-i
CH (Me) SC (O) Me Pr-c
CH (Me) SC (O) Me Bu-n
CH (Me) SC (O) Me Bu-i
CH (Me) SC (O) Me Bu-c
CH (Me) SC (O) Me Bu-s
CH (Me) SC (O) Me Bu-t
CH (Me) SC (O) Me Pen-n
CH (Me) SC (O) Me Pen-c
CH (Me) SC (O) Me Hex-n
CH (Me) SC (O) Me Hex-c
CH (Me) SC (O) Me CH2Pr-c
CH (Me) SC (O) Me CH2Bu-c
CH (Me) SC (O) Me CH2Pen-c
CH (Me) SC (O) Me CH2Hex-c
CH (Me) SC (O) Me CH2CH = CH2
CH (Me) SC (O) Me CH2CH = C (Cl)2
CH (Me) SC (O) Me CH2C≡CH
CH (Me) SC (O) Me CH2CN
CH (Me) SC (O) Me CH2CFThree
CH (Me) SC (O) Me CH2OMe
CH (Me) SC (O) Me CH2OCFThree
CH (Me) SC (O) Me CH2SMe
CH (Me) SC (O) Me CH2S (O) Me
CH (Me) SC (O) Me CH2S (O)2Me
CH (Me) SC (O) Me CH2SCFThree
CH (Me) SC (O) Me CH2S (O) CFThree
CH (Me) SC (O) Me CH2S (O)2CFThree
CH (Me) SC (O) Me CH2CH (OMe)2
CH (Me) SC (O) Me CH2CH (SMe)2
CH (Me) SC (O) Me CH2C (O) Me
CH (Me) SC (O) Me CH2C (O) CFThree
CH (Me) SC (O) Me CH2C (O) OMe
CH (Me) SC (O) Me CH2(D1-32a)
CH (Me) SC (O) Me CH2(D1-33a)
CH (Me) SC (O) Me CH2(D1-34a)
CH (Me) SC (O) Me CH2(D1-37a)
CH (Me) SC (O) Me CH2(D1-81a)
CH (Me) SC (O) Me CH2(D1-82a)
CH (Me) SC (O) Me CH2(D1-84a)
CH (Me) SC (O) Me CH2(D1-85a)
CH (Me) SC (O) Me CH2(D1-87a)
CH (Me) SC (O) Me CH2(D1-92a)
CH (Me) SC (O) Me CH2(D1-93a)
CH (Me) SC (O) Me CH2(D1-95a)
CH (Me) SC (O) Me CH2(D1-96a)
CH (Me) SC (O) Me CH2(D1-98a)
CH (Me) SC (O) Me CH2(D1-108a)
CH (Me) SC (O) Me CH2(D1-108b, Z = 2-Cl)
CH (Me) SC (O) Me CH2(D1-108b, Z = 3-Me)
CH (Me) SC (O) Me CH2(D1-108b, Z = 4-OMe)
CH (Me) SC (O) Me CH2(D1-108b, Z = 2-SMe)
CH (Me) SC (O) Me CH2(D1-108b, Z = 3-CFThree)
CH (Me) SC (O) Me CH2(D1-108b, Z = 4-OCFThree)
CH (Me) SC (O) Me CH2(D1-108b, Z = 2-SCFThree)
CH (Me) SC (O) Me CH2CH2CN
CH (Me) SC (O) Me CH2CH2CFThree
CH (Me) SC (O) Me CH2CH2OMe
CH (Me) SC (O) Me CH2CH2SMe
CH (Me) SC (O) Me CH2CH2S (O) Me
CH (Me) SC (O) Me CH2CH2S (O)2Me
CH (Me) SC (O) Me D1-32a
CH (Me) SC (O) Me D1-33a
CH (Me) SC (O) Me D1-34a
CH (Me) SC (O) Me D1-37a
CH (Me) SC (O) Me D1-81a
CH (Me) SC (O) Me D1-82a
CH (Me) SC (O) Me D1-84a
CH (Me) SC (O) Me D1-85a
CH (Me) SC (O) Me D1-87a
CH (Me) SC (O) Me D1-92a
CH (Me) SC (O) Me D1-93a
CH (Me) SC (O) Me D1-95a
CH (Me) SC (O) Me D1-96a
CH (Me) SC (O) Me D1-98a
CH (Me) SC (O) Me D1-108a
CH (Me) SC (O) Me D1-108b (Z = 2-Cl)
CH (Me) SC (O) Me D1-108b (Z = 3-Me)
CH (Me) SC (O) Me D1-108b (Z = 4-OMe)
CH (Me) SC (O) Me D1-108b (Z = 2-SMe)
CH (Me) SC (O) Me D1-108b (Z = 3-CFThree)
CH (Me) SC (O) Me D1-108b (Z = 4-OCFThree)
CH (Me) SC (O) Me D1-108b (Z = 2-SCFThree)
CH (Me) SC (O) Me C (O) Me
CH (Me) SC (O) Me C (O) CFThree
CH (Me) SC (O) Me C (O) OMe
CH (Et) SC (O) Me H
CH (Et) SC (O) Me Me
CH (Et) SC (O) Me Et
CH (Et) SC (O) Me Pr-n
CH (Et) SC (O) Me Pr-i
CH (Et) SC (O) Me Pr-c
CH (Et) SC (O) Me Bu-n
CH (Et) SC (O) Me Bu-i
CH (Et) SC (O) Me Bu-c
CH (Et) SC (O) Me Bu-s
CH (Et) SC (O) Me Bu-t
CH (Et) SC (O) Me Pen-n
CH (Et) SC (O) Me Pen-c
CH (Et) SC (O) Me Hex-n
CH (Et) SC (O) Me Hex-c
CH (Et) SC (O) Me CH2Pr-c
CH (Et) SC (O) Me CH2Bu-c
CH (Et) SC (O) Me CH2Pen-c
CH (Et) SC (O) Me CH2Hex-c
CH (Et) SC (O) Me CH2CH = CH2
CH (Et) SC (O) Me CH2CH = C (Cl)2
CH (Et) SC (O) Me CH2C≡CH
CH (Et) SC (O) Me CH2CN
CH (Et) SC (O) Me CH2CFThree
CH (Et) SC (O) Me CH2OMe
CH (Et) SC (O) Me CH2OCFThree
CH (Et) SC (O) Me CH2SMe
CH (Et) SC (O) Me CH2S (O) Me
CH (Et) SC (O) Me CH2S (O)2Me
CH (Et) SC (O) Me CH2SCFThree
CH (Et) SC (O) Me CH2S (O) CFThree
CH (Et) SC (O) Me CH2S (O)2CFThree
CH (Et) SC (O) Me CH2CH (OMe)2
CH (Et) SC (O) Me CH2CH (SMe)2
CH (Et) SC (O) Me CH2C (O) Me
CH (Et) SC (O) Me CH2C (O) CFThree
CH (Et) SC (O) Me CH2C (O) OMe
CH (Et) SC (O) Me CH2(D1-32a)
CH (Et) SC (O) Me CH2(D1-33a)
CH (Et) SC (O) Me CH2(D1-34a)
CH (Et) SC (O) Me CH2(D1-37a)
CH (Et) SC (O) Me CH2(D1-81a)
CH (Et) SC (O) Me CH2(D1-82a)
CH (Et) SC (O) Me CH2(D1-84a)
CH (Et) SC (O) Me CH2(D1-85a)
CH (Et) SC (O) Me CH2(D1-87a)
CH (Et) SC (O) Me CH2(D1-92a)
CH (Et) SC (O) Me CH2(D1-93a)
CH (Et) SC (O) Me CH2(D1-95a)
CH (Et) SC (O) Me CH2(D1-96a)
CH (Et) SC (O) Me CH2(D1-98a)
CH (Et) SC (O) Me CH2(D1-108a)
CH (Et) SC (O) Me CH2(D1-108b, Z = 2-Cl)
CH (Et) SC (O) Me CH2(D1-108b, Z = 3-Me)
CH (Et) SC (O) Me CH2(D1-108b, Z = 4-OMe)
CH (Et) SC (O) Me CH2(D1-108b, Z = 2-SMe)
CH (Et) SC (O) Me CH2(D1-108b, Z = 3-CFThree)
CH (Et) SC (O) Me CH2(D1-108b, Z = 4-OCFThree)
CH (Et) SC (O) Me CH2(D1-108b, Z = 2-SCFThree)
CH (Et) SC (O) Me CH2CH2CN
CH (Et) SC (O) Me CH2CH2CFThree
CH (Et) SC (O) Me CH2CH2OMe
CH (Et) SC (O) Me CH2CH2SMe
CH (Et) SC (O) Me CH2CH2S (O) Me
CH (Et) SC (O) Me CH2CH2S (O)2Me
CH (Et) SC (O) Me D1-32a
CH (Et) SC (O) Me D1-33a
CH (Et) SC (O) Me D1-34a
CH (Et) SC (O) Me D1-37a
CH (Et) SC (O) Me D1-81a
CH (Et) SC (O) Me D1-82a
CH (Et) SC (O) Me D1-84a
CH (Et) SC (O) Me D1-85a
CH (Et) SC (O) Me D1-87a
CH (Et) SC (O) Me D1-92a
CH (Et) SC (O) Me D1-93a
CH (Et) SC (O) Me D1-95a
CH (Et) SC (O) Me D1-96a
CH (Et) SC (O) Me D1-98a
CH (Et) SC (O) Me D1-108a
CH (Et) SC (O) Me D1-108b (Z = 2-Cl)
CH (Et) SC (O) Me D1-108b (Z = 3-Me)
CH (Et) SC (O) Me D1-108b (Z = 4-OMe)
CH (Et) SC (O) Me D1-108b (Z = 2-SMe)
CH (Et) SC (O) Me D1-108b (Z = 3-CFThree)
CH (Et) SC (O) Me D1-108b (Z = 4-OCFThree)
CH (Et) SC (O) Me D1-108b (Z = 2-SCFThree)
CH (Et) SC (O) Me C (O) Me
CH (Et) SC (O) Me C (O) CFThree
CH (Et) SC (O) Me C (O) OMe
CH2SC (O) (D1-108a) H
CH2SC (O) (D1-108a) Me
CH2SC (O) (D1-108a) Et
CH2SC (O) (D1-108a) Pr-n
CH2SC (O) (D1-108a) Pr-i
CH2SC (O) (D1-108a) Pr-c
CH2SC (O) (D1-108a) Bu-n
CH2SC (O) (D1-108a) Bu-i
CH2SC (O) (D1-108a) Bu-c
CH2SC (O) (D1-108a) Bu-s
CH2SC (O) (D1-108a) Bu-t
CH2SC (O) (D1-108a) Pen-n
CH2SC (O) (D1-108a) Pen-c
CH2SC (O) (D1-108a) Hex-n
CH2SC (O) (D1-108a) Hex-c
CH2SC (O) (D1-108a) CH2Pr-c
CH2SC (O) (D1-108a) CH2Bu-c
CH2SC (O) (D1-108a) CH2Pen-c
CH2SC (O) (D1-108a) CH2Hex-c
CH2SC (O) (D1-108a) CH2CH = CH2
CH2SC (O) (D1-108a) CH2CH = C (Cl)2
CH2SC (O) (D1-108a) CH2C≡CH
CH2SC (O) (D1-108a) CH2CN
CH2SC (O) (D1-108a) CH2CFThree
CH2SC (O) (D1-108a) CH2OMe
CH2SC (O) (D1-108a) CH2OCFThree
CH2SC (O) (D1-108a) CH2SMe
CH2SC (O) (D1-108a) CH2S (O) Me
CH2SC (O) (D1-108a) CH2S (O)2Me
CH2SC (O) (D1-108a) CH2SCFThree
CH2SC (O) (D1-108a) CH2S (O) CFThree
CH2SC (O) (D1-108a) CH2S (O)2CFThree
CH2SC (O) (D1-108a) CH2CH (OMe)2
CH2SC (O) (D1-108a) CH2CH (SMe)2
CH2SC (O) (D1-108a) CH2C (O) Me
CH2SC (O) (D1-108a) CH2C (O) CFThree
CH2SC (O) (D1-108a) CH2C (O) OMe
CH2SC (O) (D1-108a) CH2(D1-32a)
CH2SC (O) (D1-108a) CH2(D1-33a)
CH2SC (O) (D1-108a) CH2(D1-34a)
CH2SC (O) (D1-108a) CH2(D1-37a)
CH2SC (O) (D1-108a) CH2(D1-81a)
CH2SC (O) (D1-108a) CH2(D1-82a)
CH2SC (O) (D1-108a) CH2(D1-84a)
CH2SC (O) (D1-108a) CH2(D1-85a)
CH2SC (O) (D1-108a) CH2(D1-87a)
CH2SC (O) (D1-108a) CH2(D1-92a)
CH2SC (O) (D1-108a) CH2(D1-93a)
CH2SC (O) (D1-108a) CH2(D1-95a)
CH2SC (O) (D1-108a) CH2(D1-96a)
CH2SC (O) (D1-108a) CH2(D1-98a)
CH2SC (O) (D1-108a) CH2(D1-108a)
CH2SC (O) (D1-108a) CH2(D1-108b, Z = 2-Cl)
CH2SC (O) (D1-108a) CH2(D1-108b, Z = 3-Me)
CH2SC (O) (D1-108a) CH2(D1-108b, Z = 4-OMe)
CH2SC (O) (D1-108a) CH2(D1-108b, Z = 2-SMe)
CH2SC (O) (D1-108a) CH2(D1-108b, Z = 3-CFThree)
CH2SC (O) (D1-108a) CH2(D1-108b, Z = 4-OCFThree)
CH2SC (O) (D1-108a) CH2(D1-108b, Z = 2-SCFThree)
CH2SC (O) (D1-108a) CH2CH2CN
CH2SC (O) (D1-108a) CH2CH2CFThree
CH2SC (O) (D1-108a) CH2CH2OMe
CH2SC (O) (D1-108a) CH2CH2SMe
CH2SC (O) (D1-108a) CH2CH2S (O) Me
CH2SC (O) (D1-108a) CH2CH2S (O)2Me
CH2SC (O) (D1-108a) D1-32a
CH2SC (O) (D1-108a) D1-33a
CH2SC (O) (D1-108a) D1-34a
CH2SC (O) (D1-108a) D1-37a
CH2SC (O) (D1-108a) D1-81a
CH2SC (O) (D1-108a) D1-82a
CH2SC (O) (D1-108a) D1-84a
CH2SC (O) (D1-108a) D1-85a
CH2SC (O) (D1-108a) D1-87a
CH2SC (O) (D1-108a) D1-92a
CH2SC (O) (D1-108a) D1-93a
CH2SC (O) (D1-108a) D1-95a
CH2SC (O) (D1-108a) D1-96a
CH2SC (O) (D1-108a) D1-98a
CH2SC (O) (D1-108a) D1-108a
CH2SC (O) (D1-108a) D1-108b (Z = 2-Cl)
CH2SC (O) (D1-108a) D1-108b (Z = 3-Me)
CH2SC (O) (D1-108a) D1-108b (Z = 4-OMe)
CH2SC (O) (D1-108a) D1-108b (Z = 2-SMe)
CH2SC (O) (D1-108a) D1-108b (Z = 3-CFThree)
CH2SC (O) (D1-108a) D1-108b (Z = 4-OCFThree)
CH2SC (O) (D1-108a) D1-108b (Z = 2-SCFThree)
CH2SC (O) (D1-108a) C (O) Me
CH2SC (O) (D1-108a) C (O) CFThree
CH2SC (O) (D1-108a) C (O) OMe
CH (Me) SC (O) (D1-108a) H
CH (Me) SC (O) (D1-108a) Me
CH (Me) SC (O) (D1-108a) Et
CH (Me) SC (O) (D1-108a) Pr-n
CH (Me) SC (O) (D1-108a) Pr-i
CH (Me) SC (O) (D1-108a) Pr-c
CH (Me) SC (O) (D1-108a) Bu-n
CH (Me) SC (O) (D1-108a) Bu-i
CH (Me) SC (O) (D1-108a) Bu-c
CH (Me) SC (O) (D1-108a) Bu-s
CH (Me) SC (O) (D1-108a) Bu-t
CH (Me) SC (O) (D1-108a) Pen-n
CH (Me) SC (O) (D1-108a) Pen-c
CH (Me) SC (O) (D1-108a) Hex-n
CH (Me) SC (O) (D1-108a) Hex-c
CH (Me) SC (O) (D1-108a) CH2Pr-c
CH (Me) SC (O) (D1-108a) CH2Bu-c
CH (Me) SC (O) (D1-108a) CH2Pen-c
CH (Me) SC (O) (D1-108a) CH2Hex-c
CH (Me) SC (O) (D1-108a) CH2CH = CH2
CH (Me) SC (O) (D1-108a) CH2CH = C (Cl)2
CH (Me) SC (O) (D1-108a) CH2C≡CH
CH (Me) SC (O) (D1-108a) CH2CN
CH (Me) SC (O) (D1-108a) CH2CFThree
CH (Me) SC (O) (D1-108a) CH2OMe
CH (Me) SC (O) (D1-108a) CH2OCFThree
CH (Me) SC (O) (D1-108a) CH2SMe
CH (Me) SC (O) (D1-108a) CH2S (O) Me
CH (Me) SC (O) (D1-108a) CH2S (O)2Me
CH (Me) SC (O) (D1-108a) CH2SCFThree
CH (Me) SC (O) (D1-108a) CH2S (O) CFThree
CH (Me) SC (O) (D1-108a) CH2S (O)2CFThree
CH (Me) SC (O) (D1-108a) CH2CH (OMe)2
CH (Me) SC (O) (D1-108a) CH2CH (SMe)2
CH (Me) SC (O) (D1-108a) CH2C (O) Me
CH (Me) SC (O) (D1-108a) CH2C (O) CFThree
CH (Me) SC (O) (D1-108a) CH2C (O) OMe
CH (Me) SC (O) (D1-108a) CH2(D1-32a)
CH (Me) SC (O) (D1-108a) CH2(D1-33a)
CH (Me) SC (O) (D1-108a) CH2(D1-34a)
CH (Me) SC (O) (D1-108a) CH2(D1-37a)
CH (Me) SC (O) (D1-108a) CH2(D1-81a)
CH (Me) SC (O) (D1-108a) CH2(D1-82a)
CH (Me) SC (O) (D1-108a) CH2(D1-84a)
CH (Me) SC (O) (D1-108a) CH2(D1-85a)
CH (Me) SC (O) (D1-108a) CH2(D1-87a)
CH (Me) SC (O) (D1-108a) CH2(D1-92a)
CH (Me) SC (O) (D1-108a) CH2(D1-93a)
CH (Me) SC (O) (D1-108a) CH2(D1-95a)
CH (Me) SC (O) (D1-108a) CH2(D1-96a)
CH (Me) SC (O) (D1-108a) CH2(D1-98a)
CH (Me) SC (O) (D1-108a) CH2(D1-108a)
CH (Me) SC (O) (D1-108a) CH2(D1-108b, Z = 2-Cl)
CH (Me) SC (O) (D1-108a) CH2(D1-108b, Z = 3-Me)
CH (Me) SC (O) (D1-108a) CH2(D1-108b, Z = 4-OMe)
CH (Me) SC (O) (D1-108a) CH2(D1-108b, Z = 2-SMe)
CH (Me) SC (O) (D1-108a) CH2(D1-108b, Z = 3-CFThree)
CH (Me) SC (O) (D1-108a) CH2(D1-108b, Z = 4-OCFThree)
CH (Me) SC (O) (D1-108a) CH2(D1-108b, Z = 2-SCFThree)
CH (Me) SC (O) (D1-108a) CH2CH2CN
CH (Me) SC (O) (D1-108a) CH2CH2CFThree
CH (Me) SC (O) (D1-108a) CH2CH2OMe
CH (Me) SC (O) (D1-108a) CH2CH2SMe
CH (Me) SC (O) (D1-108a) CH2CH2S (O) Me
CH (Me) SC (O) (D1-108a) CH2CH2S (O)2Me
CH (Me) SC (O) (D1-108a) D1-32a
CH (Me) SC (O) (D1-108a) D1-33a
CH (Me) SC (O) (D1-108a) D1-34a
CH (Me) SC (O) (D1-108a) D1-37a
CH (Me) SC (O) (D1-108a) D1-81a
CH (Me) SC (O) (D1-108a) D1-82a
CH (Me) SC (O) (D1-108a) D1-84a
CH (Me) SC (O) (D1-108a) D1-85a
CH (Me) SC (O) (D1-108a) D1-87a
CH (Me) SC (O) (D1-108a) D1-92a
CH (Me) SC (O) (D1-108a) D1-93a
CH (Me) SC (O) (D1-108a) D1-95a
CH (Me) SC (O) (D1-108a) D1-96a
CH (Me) SC (O) (D1-108a) D1-98a
CH (Me) SC (O) (D1-108a) D1-108a
CH (Me) SC (O) (D1-108a) D1-108b (Z = 2-Cl)
CH (Me) SC (O) (D1-108a) D1-108b (Z = 3-Me)
CH (Me) SC (O) (D1-108a) D1-108b (Z = 4-OMe)
CH (Me) SC (O) (D1-108a) D1-108b (Z = 2-SMe)
CH (Me) SC (O) (D1-108a) D1-108b (Z = 3-CFThree)
CH (Me) SC (O) (D1-108a) D1-108b (Z = 4-OCFThree)
CH (Me) SC (O) (D1-108a) D1-108b (Z = 2-SCFThree)
CH (Me) SC (O) (D1-108a) C (O) Me
CH (Me) SC (O) (D1-108a) C (O) CFThree
CH (Me) SC (O) (D1-108a) C (O) OMe
CH (Et) SC (O) (D1-108a) H
CH (Et) SC (O) (D1-108a) Me
CH (Et) SC (O) (D1-108a) Et
CH (Et) SC (O) (D1-108a) Pr-n
CH (Et) SC (O) (D1-108a) Pr-i
CH (Et) SC (O) (D1-108a) Pr-c
CH (Et) SC (O) (D1-108a) Bu-n
CH (Et) SC (O) (D1-108a) Bu-i
CH (Et) SC (O) (D1-108a) Bu-c
CH (Et) SC (O) (D1-108a) Bu-s
CH (Et) SC (O) (D1-108a) Bu-t
CH (Et) SC (O) (D1-108a) Pen-n
CH (Et) SC (O) (D1-108a) Pen-c
CH (Et) SC (O) (D1-108a) Hex-n
CH (Et) SC (O) (D1-108a) Hex-c
CH (Et) SC (O) (D1-108a) CH2Pr-c
CH (Et) SC (O) (D1-108a) CH2Bu-c
CH (Et) SC (O) (D1-108a) CH2Pen-c
CH (Et) SC (O) (D1-108a) CH2Hex-c
CH (Et) SC (O) (D1-108a) CH2CH = CH2
CH (Et) SC (O) (D1-108a) CH2CH = C (Cl)2
CH (Et) SC (O) (D1-108a) CH2C≡CH
CH (Et) SC (O) (D1-108a) CH2CN
CH (Et) SC (O) (D1-108a) CH2CFThree
CH (Et) SC (O) (D1-108a) CH2OMe
CH (Et) SC (O) (D1-108a) CH2OCFThree
CH (Et) SC (O) (D1-108a) CH2SMe
CH (Et) SC (O) (D1-108a) CH2S (O) Me
CH (Et) SC (O) (D1-108a) CH2S (O)2Me
CH (Et) SC (O) (D1-108a) CH2SCFThree
CH (Et) SC (O) (D1-108a) CH2S (O) CFThree
CH (Et) SC (O) (D1-108a) CH2S (O)2CFThree
CH (Et) SC (O) (D1-108a) CH2CH (OMe)2
CH (Et) SC (O) (D1-108a) CH2CH (SMe)2
CH (Et) SC (O) (D1-108a) CH2C (O) Me
CH (Et) SC (O) (D1-108a) CH2C (O) CFThree
CH (Et) SC (O) (D1-108a) CH2C (O) OMe
CH (Et) SC (O) (D1-108a) CH2(D1-32a)
CH (Et) SC (O) (D1-108a) CH2(D1-33a)
CH (Et) SC (O) (D1-108a) CH2(D1-34a)
CH (Et) SC (O) (D1-108a) CH2(D1-37a)
CH (Et) SC (O) (D1-108a) CH2(D1-81a)
CH (Et) SC (O) (D1-108a) CH2(D1-82a)
CH (Et) SC (O) (D1-108a) CH2(D1-84a)
CH (Et) SC (O) (D1-108a) CH2(D1-85a)
CH (Et) SC (O) (D1-108a) CH2(D1-87a)
CH (Et) SC (O) (D1-108a) CH2(D1-92a)
CH (Et) SC (O) (D1-108a) CH2(D1-93a)
CH (Et) SC (O) (D1-108a) CH2(D1-95a)
CH (Et) SC (O) (D1-108a) CH2(D1-96a)
CH (Et) SC (O) (D1-108a) CH2(D1-98a)
CH (Et) SC (O) (D1-108a) CH2(D1-108a)
CH (Et) SC (O) (D1-108a) CH2(D1-108b, Z = 2-Cl)
CH (Et) SC (O) (D1-108a) CH2(D1-108b, Z = 3-Me)
CH (Et) SC (O) (D1-108a) CH2(D1-108b, Z = 4-OMe)
CH (Et) SC (O) (D1-108a) CH2(D1-108b, Z = 2-SMe)
CH (Et) SC (O) (D1-108a) CH2(D1-108b, Z = 3-CFThree)
CH (Et) SC (O) (D1-108a) CH2(D1-108b, Z = 4-OCFThree)
CH (Et) SC (O) (D1-108a) CH2(D1-108b, Z = 2-SCFThree)
CH (Et) SC (O) (D1-108a) CH2CH2CN
CH (Et) SC (O) (D1-108a) CH2CH2CFThree
CH (Et) SC (O) (D1-108a) CH2CH2OMe
CH (Et) SC (O) (D1-108a) CH2CH2SMe
CH (Et) SC (O) (D1-108a) CH2CH2S (O) Me
CH (Et) SC (O) (D1-108a) CH2CH2S (O)2Me
CH (Et) SC (O) (D1-108a) D1-32a
CH (Et) SC (O) (D1-108a) D1-33a
CH (Et) SC (O) (D1-108a) D1-34a
CH (Et) SC (O) (D1-108a) D1-37a
CH (Et) SC (O) (D1-108a) D1-81a
CH (Et) SC (O) (D1-108a) D1-82a
CH (Et) SC (O) (D1-108a) D1-84a
CH (Et) SC (O) (D1-108a) D1-85a
CH (Et) SC (O) (D1-108a) D1-87a
CH (Et) SC (O) (D1-108a) D1-92a
CH (Et) SC (O) (D1-108a) D1-93a
CH (Et) SC (O) (D1-108a) D1-95a
CH (Et) SC (O) (D1-108a) D1-96a
CH (Et) SC (O) (D1-108a) D1-98a
CH (Et) SC (O) (D1-108a) D1-108a
CH (Et) SC (O) (D1-108a) D1-108b (Z = 2-Cl)
CH (Et) SC (O) (D1-108a) D1-108b (Z = 3-Me)
CH (Et) SC (O) (D1-108a) D1-108b (Z = 4-OMe)
CH (Et) SC (O) (D1-108a) D1-108b (Z = 2-SMe)
CH (Et) SC (O) (D1-108a) D1-108b (Z = 3-CFThree)
CH (Et) SC (O) (D1-108a) D1-108b (Z = 4-OCFThree)
CH (Et) SC (O) (D1-108a) D1-108b (Z = 2-SCFThree)
CH (Et) SC (O) (D1-108a) C (O) Me
CH (Et) SC (O) (D1-108a) C (O) CFThree
CH (Et) SC (O) (D1-108a) C (O) OMe
Me H
Et H
Pr-n H
Pr-i H
Bu-n H
Bu-i H
Bu-t H
Pen-n H
Hex-n H
CH (Et) Cl H
CH2{D1-7b (3-CFThree)} H
CH (CN) Ph H
SMe H
SEt H
SPr-n H
SPr-i H
SBu-n H
SBu-i H
SBu-t H
SPen-n H
SHex-n H
SPr-c H
SBu-c H
SPen-c H
SHex-c H
SCH2CH = CH2                            H
SCH2C Three CH H
SCF2H H
SCFThree                                 H
SCF2Cl H
SCH2CFThree                              H
S (D1-108c) H
CH2OH H
CH2OMe H
CH2OEt H
CH2OPr-n H
CH2OPr-i H
CH2OBu-n H
CH2OBu-i H
CH2OBu-s H
CH2OBu-t H
CH2OPen-n H
CH2OHex-n H
CH2O (D1-104c) H
CH (Me) OH H
CH (Me) OMe H
CH (Me) OEt H
CH (Me) OPr-n H
CH (Me) OPr-i H
CH (Me) OBu-n H
CH (Me) OBu-i H
CH (Me) OBu-s H
CH (Me) OBu-t H
CH (Me) OPen-n H
CH (Me) OHex-n H
CH (Me) O (D1-104c) H
CH (Et) OH H
CH (Et) OMe H
CH (Et) OEt H
CH (Et) OPr-n H
CH (Et) OPr-i H
CH (Et) OBu-n H
CH (Et) OBu-i H
CH (Et) OBu-s H
CH (Et) OBu-t H
CH (Et) OPen-n H
CH (Et) OHex-n H
CH (Et) O (D1-104c) H
CH (n-Pr) OH H
CH (n-Pr) OMe H
CH (n-Pr) OEt H
CH (n-Pr) O (D1-104c) H
CH (i-Pr) OH H
CH (i-Pr) OMe H
CH (i-Pr) OEt H
CH (i-Pr) O (D1-104c) H
CH (n-Bu) OH H
CH (n-Bu) OMe H
CH (n-Bu) OEt H
CH (n-Bu) O (D1-104c) H
C (Me)2OH H
C (Me)2OMe H
C (Me)2OEt H
C (Me)2O (D1-104c) H
CH2CH2OH H
CH2CH2OMe H
CH2CH2OEt H
CH2CH2O (D1-104c) H
CH (Me) CH2OH H
CH (Me) CH2OMe H
CH (Me) CH2OEt H
CH (Me) CH2O (D1-104c) H
CH (Et) CH2OH H
CH (Et) CH2OMe H
CH (Et) CH2OEt H
CH (Et) CH2O (D1-104c) H
CH (n-Pr) CH2OH H
CH (n-Pr) CH2OMe H
CH (n-Pr) CH2OEt H
CH (n-Pr) CH2O (D1-104c) H
CH (i-Pr) CH2OH H
CH (i-Pr) CH2OMe H
CH (i-Pr) CH2OEt H
CH (i-Pr) CH2O (D1-104c) H
CH (n-Bu) CH2OH H
CH (n-Bu) CH2OMe H
CH (n-Bu) CH2OEt H
CH (n-Bu) CH2O (D1-104c) H
C (Me)2CH2OH H
C (Me)2CH2OMe H
C (Me)2CH2OEt H
C (Me)2CH2O (D1-104c) H
CH2SH H
CH2SMe H
CH2SEt H
CH2SPr-n H
CH2SPr-i H
CH2SBu-n H
CH2SBu-i H
CH2SBu-t H
CH2SPen-n H
CH2SHex-n H
CH2SPr-c H
CH2SBu-c H
CH2SPen-c H
CH2SHex-c H
CH2SCH2CH = CH2                         H
CH2SCH2C Three CH H
CH2SCF2H H
CH2SCFThree                               H
CH2SCF2Cl H
CH2SCH2CFThree                            H
CH2S {D1-108c} H
CH2S (O) Me H
CH2S (O) Et H
CH2S (O) Pr-n H
CH2S (O) Pr-i H
CH2S (O) Bu-n H
CH2S (O) Bu-i H
CH2S (O) Bu-t H
CH2S (O) Pen-n H
CH2S (O) Hex-n H
CH2S (O) Pr-c H
CH2S (O) Bu-c H
CH2S (O) Pen-c H
CH2S (O) Hex-c H
CH2S (O) CH2CH = CH2                      H
CH2S (O) CH2C Three CH H
CH2S (O) CF2H H
CH2S (O) CFThree                            H
CH2S (O) CF2Cl H
CH2S (O) CH2CFThree                         H
CH2S (O) {D1-108c} H
CH2S (O)2Me H
CH2S (O)2Et H
CH2S (O)2Pr-n H
CH2S (O)2Pr-i H
CH2S (O)2Bu-n H
CH2S (O)2Bu-i H
CH2S (O)2Bu-t H
CH2S (O)2Pen-n H
CH2S (O)2Hex-n H
CH2S (O)2Pr-c H
CH2S (O)2Bu-c H
CH2S (O)2Pen-c H
CH2S (O)2Hex-c H
CH2S (O)2CH2CH = CH2                      H
CH2S (O)2CH2C Three CH H
CH2S (O)2CF2H H
CH2S (O)2CFThree                           H
CH2S (O)2CF2Cl H
CH2S (O)2CH2CFThree                         H
CH2S (O)2{D1-108c} H
CH (Me) SH H
CH (Me) SMe H
CH (Me) SEt H
CH (Me) SPr-n H
CH (Me) SPr-i H
CH (Me) SBu-n H
CH (Me) SBu-i H
CH (Me) SBu-t H
CH (Me) SPen-n H
CH (Me) SHex-n H
CH (Me) SPr-c H
CH (Me) SBu-c H
CH (Me) SPen-c H
CH (Me) SHex-c H
CH (Me) SCH2CH = CH2                      H
CH (Me) SCH2C Three CH H
CH (Me) SCF2H H
CH (Me) SCFThree                            H
CH (Me) SCF2Cl H
CH (Me) SCH2CFThree                          H
CH (Me) S {D1-108c} H
CH (Me) S (O) Me H
CH (Me) S (O) Et H
CH (Me) S (O) Pr-n H
CH (Me) S (O) Pr-i H
CH (Me) S (O) Bu-n H
CH (Me) S (O) Bu-i H
CH (Me) S (O) Bu-t H
CH (Me) S (O) Pen-n H
CH (Me) S (O) Hex-n H
CH (Me) S (O) Pr-c H
CH (Me) S (O) Bu-c H
CH (Me) S (O) Pen-c H
CH (Me) S (O) Hex-c H
CH (Me) S (O) CH2CH = CH2                    H
CH (Me) S (O) CH2C Three CH H
CH (Me) S (O) CF2H H
CH (Me) S (O) CFThree                         H
CH (Me) S (O) CF2Cl H
CH (Me) S (O) CH2CFThree                      H
CH (Me) S (O) {D1-108c} H
CH (Me) S (O)2Me H
CH (Me) S (O)2Et H
CH (Me) S (O)2Pr-n H
CH (Me) S (O)2Pr-i H
CH (Me) S (O)2Bu-n H
CH (Me) S (O)2Bu-i H
CH (Me) S (O)2Bu-t H
CH (Me) S (O)2Pen-n H
CH (Me) S (O)2Hex-n H
CH (Me) S (O)2Pr-c H
CH (Me) S (O)2Bu-c H
CH (Me) S (O)2Pen-c H
CH (Me) S (O)2Hex-c H
CH (Me) S (O)2CH2CH = CH2                   H
CH (Me) S (O)2CH2C Three CH H
CH (Me) S (O)2CF2H H
CH (Me) S (O)2CFThree                        H
CH (Me) S (O)2CF2Cl H
CH (Me) S (O)2CH2CFThree                      H
CH (Me) S (O)2{D1-108c} H
CH (Et) SH H
CH (Et) SMe H
CH (Et) SEt H
CH (Et) SPr-n H
CH (Et) SPr-i H
CH (Et) SBu-n H
CH (Et) SBu-i H
CH (Et) SBu-t H
CH (Et) SPen-n H
CH (Et) SHex-n H
CH (Et) SPr-c H
CH (Et) SBu-c H
CH (Et) SPen-c H
CH (Et) SHex-c H
CH (Et) SCH2CH = CH2                      H
CH (Et) SCH2C Three CH H
CH (Et) SCF2H H
CH (Et) SCFThree                            H
CH (Et) SCF2Cl H
CH (Et) SCH2CFThree                          H
CH (Et) S {D1-108c} H
CH (Et) S (O) Me H
CH (Et) S (O) Et H
CH (Et) S (O) Pr-n H
CH (Et) S (O) Pr-i H
CH (Et) S (O) Bu-n H
CH (Et) S (O) Bu-i H
CH (Et) S (O) Bu-t H
CH (Et) S (O) Pen-n H
CH (Et) S (O) Hex-n H
CH (Et) S (O) Pr-c H
CH (Et) S (O) Bu-c H
CH (Et) S (O) Pen-c H
CH (Et) S (O) Hex-c H
CH (Et) S (O) CH2CH = CH2                    H
CH (Et) S (O) CH2C Three CH H
CH (Et) S (O) CF2H H
CH (Et) S (O) CFThree                         H
CH (Et) S (O) CF2Cl H
CH (Et) S (O) CH2CFThree                      H
CH (Et) S (O) {D1-108c} H
CH (Et) S (O)2Me H
CH (Et) S (O)2Et H
CH (Et) S (O)2Pr-n H
CH (Et) S (O)2Pr-i H
CH (Et) S (O)2Bu-n H
CH (Et) S (O)2Bu-i H
CH (Et) S (O)2Bu-t H
CH (Et) S (O)2Pen-n H
CH (Et) S (O)2Hex-n H
CH (Et) S (O)2Pr-c H
CH (Et) S (O)2Bu-c H
CH (Et) S (O)2Pen-c H
CH (Et) S (O)2Hex-c H
CH (Et) S (O)2CH2CH = CH2                   H
CH (Et) S (O)2CH2C Three CH H
CH (Et) S (O)2CF2H H
CH (Et) S (O)2CFThree                        H
CH (Et) S (O)2CF2Cl H
CH (Et) S (O)2CH2CFThree                      H
CH (Et) S (O)2{D1-108c} H
CH (n-Pr) SH H
CH (n-Pr) SMe H
CH (n-Pr) SEt H
CH (n-Pr) SPr-n H
CH (n-Pr) SPr-i H
CH (n-Pr) SBu-n H
CH (n-Pr) SBu-i H
CH (n-Pr) SBu-t H
CH (n-Pr) SPen-n H
CH (n-Pr) SHex-n H
CH (n-Pr) SPr-c H
CH (n-Pr) SBu-c H
CH (n-Pr) SPen-c H
CH (n-Pr) SHex-c H
CH (n-Pr) SCH2CH = CH2                      H
CH (n-Pr) SCH2C Three CH H
CH (n-Pr) SCF2H H
CH (n-Pr) SCFThree                            H
CH (n-Pr) SCF2Cl H
CH (n-Pr) SCH2CFThree                          H
CH (n-Pr) S {D1-108c} H
CH (n-Pr) S (O) Me H
CH (n-Pr) S (O) Et H
CH (n-Pr) S (O) Pr-n H
CH (n-Pr) S (O) Pr-i H
CH (n-Pr) S (O) Bu-n H
CH (n-Pr) S (O) Bu-i H
CH (n-Pr) S (O) Bu-t H
CH (n-Pr) S (O) Pen-n H
CH (n-Pr) S (O) Hex-n H
CH (n-Pr) S (O) Pr-c H
CH (n-Pr) S (O) Bu-c H
CH (n-Pr) S (O) Pen-c H
CH (n-Pr) S (O) Hex-c H
CH (n-Pr) S (O) CH2CH = CH2                    H
CH (n-Pr) S (O) CH2C Three CH H
CH (n-Pr) S (O) CF2H H
CH (n-Pr) S (O) CFThree                         H
CH (n-Pr) S (O) CF2Cl H
CH (n-Pr) S (O) CH2CFThree                      H
CH (n-Pr) S (O) {D1-108c} H
CH (n-Pr) S (O)2Me H
CH (n-Pr) S (O)2Et H
CH (n-Pr) S (O)2Pr-n H
CH (n-Pr) S (O)2Pr-i H
CH (n-Pr) S (O)2Bu-n H
CH (n-Pr) S (O)2Bu-i H
CH (n-Pr) S (O)2Bu-t H
CH (n-Pr) S (O)2Pen-n H
CH (n-Pr) S (O)2Hex-n H
CH (n-Pr) S (O)2Pr-c H
CH (n-Pr) S (O)2Bu-c H
CH (n-Pr) S (O)2Pen-c H
CH (n-Pr) S (O)2Hex-c H
CH (n-Pr) S (O)2CH2CH = CH2                   H
CH (n-Pr) S (O)2CH2C Three CH H
CH (n-Pr) S (O)2CF2H H
CH (n-Pr) S (O)2CFThree                        H
CH (n-Pr) S (O)2CF2Cl H
CH (n-Pr) S (O)2CH2CFThree                      H
CH (n-Pr) S (O)2{D1-108c} H
CH (i-Pr) SH H
CH (i-Pr) SMe H
CH (i-Pr) SEt H
CH (i-Pr) SPr-n H
CH (i-Pr) SPr-i H
CH (i-Pr) SBu-n H
CH (i-Pr) SBu-i H
CH (i-Pr) SBu-t H
CH (i-Pr) SPen-n H
CH (i-Pr) SHex-n H
CH (i-Pr) SPr-c H
CH (i-Pr) SBu-c H
CH (i-Pr) SPen-c H
CH (i-Pr) SHex-c H
CH (i-Pr) SCH2CH = CH2                      H
CH (i-Pr) SCH2C Three CH H
CH (i-Pr) SCF2H H
CH (i-Pr) SCFThree                            H
CH (i-Pr) SCF2Cl H
CH (i-Pr) SCH2CFThree                          H
CH (i-Pr) S {D1-108c} H
CH (i-Pr) S (O) Me H
CH (i-Pr) S (O) Et H
CH (i-Pr) S (O) Pr-n H
CH (i-Pr) S (O) Pr-i H
CH (i-Pr) S (O) Bu-n H
CH (i-Pr) S (O) Bu-i H
CH (i-Pr) S (O) Bu-t H
CH (i-Pr) S (O) Pen-n H
CH (i-Pr) S (O) Hex-n H
CH (i-Pr) S (O) Pr-c H
CH (i-Pr) S (O) Bu-c H
CH (i-Pr) S (O) Pen-c H
CH (i-Pr) S (O) Hex-c H
CH (i-Pr) S (O) CH2CH = CH2                    H
CH (i-Pr) S (O) CH2C Three CH H
CH (i-Pr) S (O) CF2H H
CH (i-Pr) S (O) CFThree                         H
CH (i-Pr) S (O) CF2Cl H
CH (i-Pr) S (O) CH2CFThree                      H
CH (i-Pr) S (O) {D1-108c} H
CH (i-Pr) S (O)2Me H
CH (i-Pr) S (O)2Et H
CH (i-Pr) S (O)2Pr-n H
CH (i-Pr) S (O)2Pr-i H
CH (i-Pr) S (O)2Bu-n H
CH (i-Pr) S (O)2Bu-i H
CH (i-Pr) S (O)2Bu-t H
CH (i-Pr) S (O)2Pen-n H
CH (i-Pr) S (O)2Hex-n H
CH (i-Pr) S (O)2Pr-c H
CH (i-Pr) S (O)2Bu-c H
CH (i-Pr) S (O)2Pen-c H
CH (i-Pr) S (O)2Hex-c H
CH (i-Pr) S (O)2CH2CH = CH2                   H
CH (i-Pr) S (O)2CH2C Three CH H
CH (i-Pr) S (O)2CF2H H
CH (i-Pr) S (O)2CFThree                        H
CH (i-Pr) S (O)2CF2Cl H
CH (i-Pr) S (O)2CH2CFThree                      H
CH (i-Pr) S (O)2{D1-108c} H
CH (n-Bu) SH H
CH (n-Bu) SMe H
CH (n-Bu) SEt H
CH (n-Bu) SPr-n H
CH (n-Bu) SPr-i H
CH (n-Bu) SBu-n H
CH (n-Bu) SBu-i H
CH (n-Bu) SBu-t H
CH (n-Bu) SPen-n H
CH (n-Bu) SHex-n H
CH (n-Bu) SPr-c H
CH (n-Bu) SBu-c H
CH (n-Bu) SPen-c H
CH (n-Bu) SHex-c H
CH (n-Bu) SCH2CH = CH2                      H
CH (n-Bu) SCH2C Three CH H
CH (n-Bu) SCF2H H
CH (n-Bu) SCFThree                            H
CH (n-Bu) SCF2Cl H
CH (n-Bu) SCH2CFThree                          H
CH (n-Bu) S {D1-108c} H
CH (n-Bu) S (O) Me H
CH (n-Bu) S (O) Et H
CH (n-Bu) S (O) Pr-n H
CH (n-Bu) S (O) Pr-i H
CH (n-Bu) S (O) Bu-n H
CH (n-Bu) S (O) Bu-i H
CH (n-Bu) S (O) Bu-t H
CH (n-Bu) S (O) Pen-n H
CH (n-Bu) S (O) Hex-n H
CH (n-Bu) S (O) Pr-c H
CH (n-Bu) S (O) Bu-c H
CH (n-Bu) S (O) Pen-c H
CH (n-Bu) S (O) Hex-c H
CH (n-Bu) S (O) CH2CH = CH2                    H
CH (n-Bu) S (O) CH2C Three CH H
CH (n-Bu) S (O) CF2H H
CH (n-Bu) S (O) CFThree                         H
CH (n-Bu) S (O) CF2Cl H
CH (n-Bu) S (O) CH2CFThree                      H
CH (n-Bu) S (O) {D1-108c} H
CH (n-Bu) S (O)2Me H
CH (n-Bu) S (O)2Et H
CH (n-Bu) S (O)2Pr-n H
CH (n-Bu) S (O)2Pr-i H
CH (n-Bu) S (O)2Bu-n H
CH (n-Bu) S (O)2Bu-i H
CH (n-Bu) S (O)2Bu-t H
CH (n-Bu) S (O)2Pen-n H
CH (n-Bu) S (O)2Hex-n H
CH (n-Bu) S (O)2Pr-c H
CH (n-Bu) S (O)2Bu-c H
CH (n-Bu) S (O)2Pen-c H
CH (n-Bu) S (O)2Hex-c H
CH (n-Bu) S (O)2CH2CH = CH2                   H
CH (n-Bu) S (O)2CH2C Three CH H
CH (n-Bu) S (O)2CF2H H
CH (n-Bu) S (O)2CFThree                        H
CH (n-Bu) S (O)2CF2Cl H
CH (n-Bu) S (O)2CH2CFThree                      H
CH (n-Bu) S (O)2{D1-108c} H
CH (CH2OMe) SH H
CH (CH2OMe) SMe H
CH (CH2OMe) SEt H
CH (CH2OMe) SPr-n H
CH (CH2OMe) SPr-i H
CH (CH2OMe) SBu-n H
CH (CH2OMe) SBu-i H
CH (CH2OMe) SBu-t H
CH (CH2OMe) SPen-n H
CH (CH2OMe) SHex-n H
CH (CH2OMe) SPr-c H
CH (CH2OMe) SBu-c H
CH (CH2OMe) SPen-c H
CH (CH2OMe) SHex-c H
CH (CH2OMe) SCH2CH = CH2                    H
CH (CH2OMe) SCH2C Three CH H
CH (CH2OMe) SCF2H H
CH (CH2OMe) SCFThree                         H
CH (CH2OMe) SCF2Cl H
CH (CH2OMe) SCH2CFThree                       H
CH (CH2OMe) S {D1-108c} H
CH (CH2OMe) S (O) Me H
CH (CH2OMe) S (O) Et H
CH (CH2OMe) S (O) Pr-n H
CH (CH2OMe) S (O) Pr-i H
CH (CH2OMe) S (O) Bu-n H
CH (CH2OMe) S (O) Bu-i H
CH (CH2OMe) S (O) Bu-t H
CH (CH2OMe) S (O) Pen-n H
CH (CH2OMe) S (O) Hex-n H
CH (CH2OMe) S (O) Pr-c H
CH (CH2OMe) S (O) Bu-c H
CH (CH2OMe) S (O) Pen-c H
CH (CH2OMe) S (O) Hex-c H
CH (CH2OMe) S (O) CH2CH = CH2                 H
CH (CH2OMe) S (O) CH2C Three CH H
CH (CH2OMe) S (O) CF2H H
CH (CH2OMe) S (O) CFThree                      H
CH (CH2OMe) S (O) CF2Cl H
CH (CH2OMe) S (O) CH2CFThree                   H
CH (CH2OMe) S (O) {D1-108c} H
CH (CH2OMe) S (O)2Me H
CH (CH2OMe) S (O)2Et H
CH (CH2OMe) S (O)2Pr-n H
CH (CH2OMe) S (O)2Pr-i H
CH (CH2OMe) S (O)2Bu-n H
CH (CH2OMe) S (O)2Bu-i H
CH (CH2OMe) S (O)2Bu-t H
CH (CH2OMe) S (O)2Pen-n H
CH (CH2OMe) S (O)2Hex-n H
CH (CH2OMe) S (O)2Pr-c H
CH (CH2OMe) S (O)2Bu-c H
CH (CH2OMe) S (O)2Pen-c H
CH (CH2OMe) S (O)2Hex-c H
CH (CH2OMe) S (O)2CH2CH = CH2                 H
CH (CH2OMe) S (O)2CH2C Three CH H
CH (CH2OMe) S (O)2CF2H H
CH (CH2OMe) S (O)2CFThree                      H
CH (CH2OMe) S (O)2CF2Cl H
CH (CH2OMe) S (O)2CH2CFThree                    H
CH (CH2OMe) S (O)2{D1-108c} H
CH (CH2CH = CH2) SH H
CH (CH2CH = CH2) SMe H
CH (CH2CH = CH2) SEt H
CH (CH2CH = CH2SPr-n H
CH (CH2CH = CH2SPr-i H
CH (CH2CH = CH2) SBu-n H
CH (CH2CH = CH2) SBu-i H
CH (CH2CH = CH2) SBu-t H
CH (CH2CH = CH2SPen-n H
CH (CH2CH = CH2) SHex-n H
CH (CH2CH = CH2SPr-c H
CH (CH2CH = CH2) SBu-c H
CH (CH2CH = CH2SPen-c H
CH (CH2CH = CH2) SHex-c H
CH (CH2CH = CH2) SCH2CH = CH2                  H
CH (CH2CH = CH2) SCH2C Three CH H
CH (CH2CH = CH2) SCF2H H
CH (CH2CH = CH2) SCFThree                       H
CH (CH2CH = CH2) SCF2Cl H
CH (CH2CH = CH2) SCH2CFThree                     H
CH (CH2CH = CH2) S {D1-108c} H
CH (CH2CH = CH2) S (O) Me H
CH (CH2CH = CH2) S (O) Et H
CH (CH2CH = CH2) S (O) Pr-n H
CH (CH2CH = CH2) S (O) Pr-i H
CH (CH2CH = CH2) S (O) Bu-n H
CH (CH2CH = CH2) S (O) Bu-i H
CH (CH2CH = CH2) S (O) Bu-t H
CH (CH2CH = CH2) S (O) Pen-n H
CH (CH2CH = CH2) S (O) Hex-n H
CH (CH2CH = CH2) S (O) Pr-c H
CH (CH2CH = CH2) S (O) Bu-c H
CH (CH2CH = CH2) S (O) Pen-c H
CH (CH2CH = CH2) S (O) Hex-c H
CH (CH2CH = CH2) S (O) CH2CH = CH2               H
CH (CH2CH = CH2) S (O) CH2C Three CH H
CH (CH2CH = CH2) S (O) CF2H H
CH (CH2CH = CH2) S (O) CFThree                    H
CH (CH2CH = CH2) S (O) CF2Cl H
CH (CH2CH = CH2) S (O) CH2CFThree                 H
CH (CH2CH = CH2) S (O) {D1-108c} H
CH (CH2CH = CH2) S (O)2Me H
CH (CH2CH = CH2) S (O)2Et H
CH (CH2CH = CH2) S (O)2Pr-n H
CH (CH2CH = CH2) S (O)2Pr-i H
CH (CH2CH = CH2) S (O)2Bu-n H
CH (CH2CH = CH2) S (O)2Bu-i H
CH (CH2CH = CH2) S (O)2Bu-t H
CH (CH2CH = CH2) S (O)2Pen-n H
CH (CH2CH = CH2) S (O)2Hex-n H
CH (CH2CH = CH2) S (O)2Pr-c H
CH (CH2CH = CH2) S (O)2Bu-c H
CH (CH2CH = CH2) S (O)2Pen-c H
CH (CH2CH = CH2) S (O)2Hex-c H
CH (CH2CH = CH2) S (O)2CH2CH = CH2              H
CH (CH2CH = CH2) S (O)2CH2C Three CH H
CH (CH2CH = CH2) S (O)2CF2H H
CH (CH2CH = CH2) S (O)2CFThree                    H
CH (CH2CH = CH2) S (O)2CF2Cl H
CH (CH2CH = CH2) S (O)2CH2CFThree                  H
CH (CH2CH = CH2) S (O)2{D1-108c} H
CH (CH2C≡CH) SH H
CH (CH2C≡CH) SMe H
CH (CH2C≡CH) SEt H
CH (CH2C≡CH) SPr-n H
CH (CH2C≡CH) SPr-i H
CH (CH2C≡CH) SBu-n H
CH (CH2C≡CH) SBu-i H
CH (CH2C≡CH) SBu-t H
CH (CH2C≡CH) SPen-n H
CH (CH2C≡CH) SHex-n H
CH (CH2C≡CH) SPr-c H
CH (CH2C≡CH) SBu-c H
CH (CH2C≡CH) SPen-c H
CH (CH2C≡CH) SHex-c H
CH (CH2C≡CH) SCH2CH = CH2                   H
CH (CH2C≡CH) SCH2C Three CH H
CH (CH2C≡CH) SCF2H H
CH (CH2C≡CH) SCFThree                        H
CH (CH2C≡CH) SCF2Cl H
CH (CH2C≡CH) SCH2CFThree                      H
CH (CH2C≡CH) S {D1-108c} H
CH (CH2C≡CH) S (O) Me H
CH (CH2C≡CH) S (O) Et H
CH (CH2C≡CH) S (O) Pr-n H
CH (CH2C≡CH) S (O) Pr-i H
CH (CH2C≡CH) S (O) Bu-n H
CH (CH2C≡CH) S (O) Bu-i H
CH (CH2C≡CH) S (O) Bu-t H
CH (CH2C≡CH) S (O) Pen-n H
CH (CH2C≡CH) S (O) Hex-n H
CH (CH2C≡CH) S (O) Pr-c H
CH (CH2C≡CH) S (O) Bu-c H
CH (CH2C≡CH) S (O) Pen-c H
CH (CH2C≡CH) S (O) Hex-c H
CH (CH2C≡CH) S (O) CH2CH = CH2                H
CH (CH2C≡CH) S (O) CH2C Three CH H
CH (CH2C≡CH) S (O) CF2H H
CH (CH2C≡CH) S (O) CFThree                     H
CH (CH2C≡CH) S (O) CF2Cl H
CH (CH2C≡CH) S (O) CH2CFThree                  H
CH (CH2C≡CH) S (O) {D1-108c} H
CH (CH2C≡CH) S (O)2Me H
CH (CH2C≡CH) S (O)2Et H
CH (CH2C≡CH) S (O)2Pr-n H
CH (CH2C≡CH) S (O)2Pr-i H
CH (CH2C≡CH) S (O)2Bu-n H
CH (CH2C≡CH) S (O)2Bu-i H
CH (CH2C≡CH) S (O)2Bu-t H
CH (CH2C≡CH) S (O)2Pen-n H
CH (CH2C≡CH) S (O)2Hex-n H
CH (CH2C≡CH) S (O)2Pr-c H
CH (CH2C≡CH) S (O)2Bu-c H
CH (CH2C≡CH) S (O)2Pen-c H
CH (CH2C≡CH) S (O)2Hex-c H
CH (CH2C≡CH) S (O)2CH2CH = CH2               H
CH (CH2C≡CH) S (O)2CH2C Three CH H
CH (CH2C≡CH) S (O)2CF2H H
CH (CH2C≡CH) S (O)2CFThree                     H
CH (CH2C≡CH) S (O)2CF2Cl H
CH (CH2C≡CH) S (O)2CH2CFThree                   H
CH (CH2C≡CH) S (O)2{D1-108c} H
CH (CH2CN) SH H
CH (CH2CN) SMe H
CH (CH2CN) SEt H
CH (CH2CN) SPr-n H
CH (CH2CN) SPr-i H
CH (CH2CN) SBu-n H
CH (CH2CN) SBu-i H
CH (CH2CN) SBu-t H
CH (CH2CN) SPen-n H
CH (CH2CN) SHex-n H
CH (CH2CN) SPr-c H
CH (CH2CN) SBu-c H
CH (CH2CN) SPen-c H
CH (CH2CN) SHex-c H
CH (CH2CN) SCH2CH = CH2                      H
CH (CH2CN) SCH2C Three CH H
CH (CH2CN) SCF2H H
CH (CH2CN) SCFThree                           H
CH (CH2CN) SCF2Cl H
CH (CH2CN) SCH2CFThree                         H
CH (CH2CN) S {D1-108c} H
CH (CH2CN) S (O) Me H
CH (CH2CN) S (O) Et H
CH (CH2CN) S (O) Pr-n H
CH (CH2CN) S (O) Pr-i H
CH (CH2CN) S (O) Bu-n H
CH (CH2CN) S (O) Bu-i H
CH (CH2CN) S (O) Bu-t H
CH (CH2CN) S (O) Pen-n H
CH (CH2CN) S (O) Hex-n H
CH (CH2CN) S (O) Pr-c H
CH (CH2CN) S (O) Bu-c H
CH (CH2CN) S (O) Pen-c H
CH (CH2CN) S (O) Hex-c H
CH (CH2CN) S (O) CH2CH = CH2                   H
CH (CH2CN) S (O) CH2C Three CH H
CH (CH2CN) S (O) CF2H H
CH (CH2CN) S (O) CFThree                        H
CH (CH2CN) S (O) CF2Cl H
CH (CH2CN) S (O) CH2CFThree                    H
CH (CH2CN) S (O) {D1-108c} H
CH (CH2CN) S (O)2Me H
CH (CH2CN) S (O)2Et H
CH (CH2CN) S (O)2Pr-n H
CH (CH2CN) S (O)2Pr-i H
CH (CH2CN) S (O)2Bu-n H
CH (CH2CN) S (O)2Bu-i H
CH (CH2CN) S (O)2Bu-t H
CH (CH2CN) S (O)2Pen-n H
CH (CH2CN) S (O)2Hex-n H
CH (CH2CN) S (O)2Pr-c H
CH (CH2CN) S (O)2Bu-c H
CH (CH2CN) S (O)2Pen-c H
CH (CH2CN) S (O)2Hex-c H
CH (CH2CN) S (O)2CH2CH = CH2                  H
CH (CH2CN) S (O)2CH2C Three CH H
CH (CH2CN) S (O)2CF2H H
CH (CH2CN) S (O)2CFThree                        H
CH (CH2CN) S (O)2CF2Cl H
CH (CH2CN) S (O)2CH2CFThree                      H
CH (CH2CN) S (O)2{D1-108c} H
CH (Me)2SH H
CH (Me)2SMe H
CH (Me)2SEt H
CH (Me)2SPr-n H
CH (Me)2SPr-i H
CH (Me)2SBu-n H
CH (Me)2SBu-i H
CH (Me)2SBu-t H
CH (Me)2SPen-n H
CH (Me)2SHex-n H
CH (Me)2SPr-c H
CH (Me)2SBu-c H
CH (Me)2SPen-c H
CH (Me)2SHex-c H
CH (Me)2SCH2CH = CH2                        H
CH (Me)2SCH2C Three CH H
CH (Me)2SCF2H H
CH (Me)2SCFThree                             H
CH (Me)2SCF2Cl H
CH (Me)2SCH2CFThree                           H
CH (Me)2S {D1-108c} H
CH (Me)2S (O) Me H
CH (Me)2S (O) Et H
CH (Me)2S (O) Pr-n H
CH (Me)2S (O) Pr-i H
CH (Me)2S (O) Bu-n H
CH (Me)2S (O) Bu-i H
CH (Me)2S (O) Bu-t H
CH (Me)2S (O) Pen-n H
CH (Me)2S (O) Hex-n H
CH (Me)2S (O) Pr-c H
CH (Me)2S (O) Bu-c H
CH (Me)2S (O) Pen-c H
CH (Me)2S (O) Hex-c H
CH (Me)2S (O) CH2CH = CH2                     H
CH (Me)2S (O) CH2C Three CH H
CH (Me)2S (O) CF2H H
CH (Me)2S (O) CFThree                          H
CH (Me)2S (O) CF2Cl H
CH (Me)2S (O) CH2CFThree                      H
CH (Me)2S (O) {D1-108c} H
CH (Me)2S (O)2Me H
CH (Me)2S (O)2Et H
CH (Me)2S (O)2Pr-n H
CH (Me)2S (O)2Pr-i H
CH (Me)2S (O)2Bu-n H
CH (Me)2S (O)2Bu-i H
CH (Me)2S (O)2Bu-t H
CH (Me)2S (O)2Pen-n H
CH (Me)2S (O)2Hex-n H
CH (Me)2S (O)2Pr-c H
CH (Me)2S (O)2Bu-c H
CH (Me)2S (O)2Pen-c H
CH (Me)2S (O)2Hex-c H
CH (Me)2S (O)2CH2CH = CH2                    H
CH (Me)2S (O)2CH2C Three CH H
CH (Me)2S (O)2CF2H H
CH (Me)2S (O)2CFThree                          H
CH (Me)2S (O)2CF2Cl H
CH (Me)2S (O)2CH2CFThree                        H
CH (Me)2S (O)2{D1-108c} H
CH2CH2SH H
CH2CH2SMe H
CH2CH2SEt H
CH2CH2SPr-n H
CH2CH2SPr-i H
CH2CH2SBu-n H
CH2CH2SBu-i H
CH2CH2SBu-t H
CH2CH2SPen-n H
CH2CH2SHex-n H
CH2CH2SPr-c H
CH2CH2SBu-c H
CH2CH2SPen-c H
CH2CH2SHex-c H
CH2CH2SCH2CH = CH2                         H
CH2CH2SCH2C Three CH H
CH2CH2SCF2H H
CH2CH2SCFThree                              H
CH2CH2SCF2Cl H
CH2CH2SCH2CFThree                            H
CH2CH2S {D1-108c} H
CH2CH2S (O) Me H
CH2CH2S (O) Et H
CH2CH2S (O) Pr-n H
CH2CH2S (O) Pr-i H
CH2CH2S (O) Bu-n H
CH2CH2S (O) Bu-i H
CH2CH2S (O) Bu-t H
CH2CH2S (O) Pen-n H
CH2CH2S (O) Hex-n H
CH2CH2S (O) Pr-c H
CH2CH2S (O) Bu-c H
CH2CH2S (O) Pen-c H
CH2CH2S (O) Hex-c H
CH2CH2S (O) CH2CH = CH2                      H
CH2CH2S (O) CH2C Three CH H
CH2CH2S (O) CF2H H
CH2CH2S (O) CFThree                           H
CH2CH2S (O) CF2Cl H
CH2CH2S (O) CH2CFThree                       H
CH2CH2S (O) {D1-108c} H
CH2CH2S (O)2Me H
CH2CH2S (O)2Et H
CH2CH2S (O)2Pr-n H
CH2CH2S (O)2Pr-i H
CH2CH2S (O)2Bu-n H
CH2CH2S (O)2Bu-i H
CH2CH2S (O)2Bu-t H
CH2CH2S (O)2Pen-n H
CH2CH2S (O)2Hex-n H
CH2CH2S (O)2Pr-c H
CH2CH2S (O)2Bu-c H
CH2CH2S (O)2Pen-c H
CH2CH2S (O)2Hex-c H
CH2CH2S (O)2CH2CH = CH2                     H
CH2CH2S (O)2CH2C Three CH H
CH2CH2S (O)2CF2H H
CH2CH2S (O)2CFThree                           H
CH2CH2S (O)2CF2Cl H
CH2CH2S (O)2CH2CFThree                         H
CH2CH2S (O)2{D1-108c} H
CH (Me) CH2SH H
CH (Me) CH2SMe H
CH (Me) CH2SEt H
CH (Me) CH2SPr-n H
CH (Me) CH2SPr-i H
CH (Me) CH2SBu-n H
CH (Me) CH2SBu-i H
CH (Me) CH2SBu-t H
CH (Me) CH2SPen-n H
CH (Me) CH2SHex-n H
CH (Me) CH2SPr-c H
CH (Me) CH2SBu-c H
CH (Me) CH2SPen-c H
CH (Me) CH2SHex-c H
CH (Me) CH2SCH2CH = CH2                      H
CH (Me) CH2SCH2C Three CH H
CH (Me) CH2SCF2H H
CH (Me) CH2SCFThree                           H
CH (Me) CH2SCF2Cl H
CH (Me) CH2SCH2CFThree                         H
CH (Me) CH2S {D1-108c} H
CH (Me) CH2S (O) Me H
CH (Me) CH2S (O) Et H
CH (Me) CH2S (O) Pr-n H
CH (Me) CH2S (O) Pr-i H
CH (Me) CH2S (O) Bu-n H
CH (Me) CH2S (O) Bu-i H
CH (Me) CH2S (O) Bu-t H
CH (Me) CH2S (O) Pen-n H
CH (Me) CH2S (O) Hex-n H
CH (Me) CH2S (O) Pr-c H
CH (Me) CH2S (O) Bu-c H
CH (Me) CH2S (O) Pen-c H
CH (Me) CH2S (O) Hex-c H
CH (Me) CH2S (O) CH2CH = CH2                   H
CH (Me) CH2S (O) CH2C Three CH H
CH (Me) CH2S (O) CF2H H
CH (Me) CH2S (O) CFThree                        H
CH (Me) CH2S (O) CF2Cl H
CH (Me) CH2S (O) CH2CFThree                     H
CH (Me) CH2S (O) {D1-108c} H
CH (Me) CH2S (O)2Me H
CH (Me) CH2S (O)2Et H
CH (Me) CH2S (O)2Pr-n H
CH (Me) CH2S (O)2Pr-i H
CH (Me) CH2S (O)2Bu-n H
CH (Me) CH2S (O)2Bu-i H
CH (Me) CH2S (O)2Bu-t H
CH (Me) CH2S (O)2Pen-n H
CH (Me) CH2S (O)2Hex-n H
CH (Me) CH2S (O)2Pr-c H
CH (Me) CH2S (O)2Bu-c H
CH (Me) CH2S (O)2Pen-c H
CH (Me) CH2S (O)2Hex-c H
CH (Me) CH2S (O)2CH2CH = CH2                  H
CH (Me) CH2S (O)2CH2C Three CH H
CH (Me) CH2S (O)2CF2H H
CH (Me) CH2S (O)2CFThree                        H
CH (Me) CH2S (O)2CF2Cl H
CH (Me) CH2S (O)2CH2CFThree                     H
CH (Me) CH2S (O)2{D1-108c} H
CH (Me) CH (Me) SH H
CH (Me) CH (Me) SMe H
CH (Me) CH (Me) SEt H
CH (Me) CH (Me) SPr-n H
CH (Me) CH (Me) SPr-i H
CH (Me) CH (Me) SBu-n H
CH (Me) CH (Me) SBu-i H
CH (Me) CH (Me) SBu-t H
CH (Me) CH (Me) SPen-n H
CH (Me) CH (Me) SHex-n H
CH (Me) CH (Me) SPr-c H
CH (Me) CH (Me) SBu-c H
CH (Me) CH (Me) SPen-c H
CH (Me) CH (Me) SHex-c H
CH (Me) CH (Me) SCH2CH = CH2                    H
CH (Me) CH (Me) SCH2C Three CH H
CH (Me) CH (Me) SCF2H H
CH (Me) CH (Me) SCFThree                         H
CH (Me) CH (Me) SCF2Cl H
CH (Me) CH (Me) SCH2CFThree                       H
CH (Me) CH (Me) S {D1-108c} H
CH (Me) CH (Me) S (O) Me H
CH (Me) CH (Me) S (O) Et H
CH (Me) CH (Me) S (O) Pr-n H
CH (Me) CH (Me) S (O) Pr-i H
CH (Me) CH (Me) S (O) Bu-n H
CH (Me) CH (Me) S (O) Bu-i H
CH (Me) CH (Me) S (O) Bu-t H
CH (Me) CH (Me) S (O) Pen-n H
CH (Me) CH (Me) S (O) Hex-n H
CH (Me) CH (Me) S (O) Pr-c H
CH (Me) CH (Me) S (O) Bu-c H
CH (Me) CH (Me) S (O) Pen-c H
CH (Me) CH (Me) S (O) Hex-c H
CH (Me) CH (Me) S (O) CH2CH = CH2                 H
CH (Me) CH (Me) S (O) CH2C Three CH H
CH (Me) CH (Me) S (O) CF2H H
CH (Me) CH (Me) S (O) CFThree                      H
CH (Me) CH (Me) S (O) CF2Cl H
CH (Me) CH (Me) S (O) CH2CFThree                   H
CH (Me) CH (Me) S (O) {D1-108c} H
CH (Me) CH (Me) S (O)2Me H
CH (Me) CH (Me) S (O)2Et H
CH (Me) CH (Me) S (O)2Pr-n H
CH (Me) CH (Me) S (O)2Pr-i H
CH (Me) CH (Me) S (O)2Bu-n H
CH (Me) CH (Me) S (O)2Bu-i H
CH (Me) CH (Me) S (O)2Bu-t H
CH (Me) CH (Me) S (O)2Pen-n H
CH (Me) CH (Me) S (O)2Hex-n H
CH (Me) CH (Me) S (O)2Pr-c H
CH (Me) CH (Me) S (O)2Bu-c H
CH (Me) CH (Me) S (O)2Pen-c H
CH (Me) CH (Me) S (O)2Hex-c H
CH (Me) CH (Me) S (O)2CH2CH = CH2                H
CH (Me) CH (Me) S (O)2CH2C Three CH H
CH (Me) CH (Me) S (O)2CF2H H
CH (Me) CH (Me) S (O)2CFThree                      H
CH (Me) CH (Me) S (O)2CF2Cl H
CH (Me) CH (Me) S (O)2CH2CFThree                   H
CH (Me) CH (Me) S (O)2{D1-108c} H
CH2CH (Me) SH H
CH2CH (Me) SMe H
CH2CH (Me) SEt H
CH2CH (Me) SPr-n H
CH2CH (Me) SPr-i H
CH2CH (Me) SBu-n H
CH2CH (Me) SBu-i H
CH2CH (Me) SBu-t H
CH2CH (Me) SPen-n H
CH2CH (Me) SHex-n H
CH2CH (Me) SPr-c H
CH2CH (Me) SBu-c H
CH2CH (Me) SPen-c H
CH2CH (Me) SHex-c H
CH2CH (Me) SCH2CH = CH2                       H
CH2CH (Me) SCH2C Three CH H
CH2CH (Me) SCF2H H
CH2CH (Me) SCFThree                            H
CH2CH (Me) SCF2Cl H
CH2CH (Me) SCH2CFThree                          H
CH2CH (Me) S {D1-108c} H
CH2CH (Me) S (O) Me H
CH2CH (Me) S (O) Et H
CH2CH (Me) S (O) Pr-n H
CH2CH (Me) S (O) Pr-i H
CH2CH (Me) S (O) Bu-n H
CH2CH (Me) S (O) Bu-i H
CH2CH (Me) S (O) Bu-t H
CH2CH (Me) S (O) Pen-n H
CH2CH (Me) S (O) Hex-n H
CH2CH (Me) S (O) Pr-c H
CH2CH (Me) S (O) Bu-c H
CH2CH (Me) S (O) Pen-c H
CH2CH (Me) S (O) Hex-c H
CH2CH (Me) S (O) CH2CH = CH2                    H
CH2CH (Me) S (O) CH2C Three CH H
CH2CH (Me) S (O) CF2H H
CH2CH (Me) S (O) CFThree                         H
CH2CH (Me) S (O) CF2Cl H
CH2CH (Me) S (O) CH2CFThree                      H
CH2CH (Me) S (O) {D1-108c} H
CH2CH (Me) S (O)2Me H
CH2CH (Me) S (O)2Et H
CH2CH (Me) S (O)2Pr-n H
CH2CH (Me) S (O)2Pr-i H
CH2CH (Me) S (O)2Bu-n H
CH2CH (Me) S (O)2Bu-i H
CH2CH (Me) S (O)2Bu-t H
CH2CH (Me) S (O)2Pen-n H
CH2CH (Me) S (O)2Hex-n H
CH2CH (Me) S (O)2Pr-c H
CH2CH (Me) S (O)2Bu-c H
CH2CH (Me) S (O)2Pen-c H
CH2CH (Me) S (O)2Hex-c H
CH2CH (Me) S (O)2CH2CH = CH2                   H
CH2CH (Me) S (O)2CH2C Three CH H
CH2CH (Me) S (O)2CF2H H
CH2CH (Me) S (O)2CFThree                         H
CH2CH (Me) S (O)2CF2Cl H
CH2CH (Me) S (O)2CH2CFThree                      H
CH2CH (Me) S (O)2{D1-108c} H
C (O) OH H
C (O) OMe H
C (O) OEt H
C (O) OPr-n H
C (O) OPr-i H
C (O) OBu-n H
C (O) OBu-i H
C (O) OBu-s H
C (O) OBu-t H
C (O) OPen-n H
C (O) OHex-n H
CHO H
C (O) Me H
C (O) Et H
C (O) Pr-n H
C (O) Pr-i H
C (O) Bu-n H
C (O) Bu-i H
C (O) Bu-s H
C (O) Bu-t H
C (O) Pen-n H
C (O) Hex-n H
C (O) NHC (O) Me H
C (O) NHMe H
C (O) NHEt H
C (O) NHPr-n H
C (O) NHPr-i H
C (O) NHBu-n H
C (O) NHBu-i H
C (O) NHBu-s H
C (O) NHBu-t H
C (O) NHPen-n H
C (O) NHHex-n H
CN H
Ph H
CH2Cl H
CH2Br H
CH2I H
CH (Me) Cl H
CH (Me) Br H
CH (Me) I H
CH (Et) Cl H
CH (Et) Br H
CH (Et) I H
CH (n-Pr) Cl H
CH (n-Pr) Br H
CH (n-Pr) I H
CH (i-Pr) Cl H
CH (i-Pr) Br H
CH (i-Pr) I H
CH (n-Bu) Cl H
CH (n-Bu) Br H
CH (n-Bu) I H
CH (CH2OMe) Cl H
CH (CH2OMe) Br H
CH (CH2OMe) I H
CH (CH2CH = CH2) Cl H
CH (CH2CH = CH2) Br H
CH (CH2CH = CH2) I H
CH (CH2C3CH) Cl H
CH (CH2C3CH) Br H
CH (CH2C3CH) I H
CH (Me) CH2Cl H
CH (Me) CH2Br H
CH (Me) CH2I H
C (Me)2CH2Cl H
C (Me)2CH2Br H
C (Me)2CH2I H
CH2SCH2Pr-c Me
CH2SCH2Pr-c Et
CH2SCH2Pr-c Pr-n
CH2SCH2Pr-c Pr-i
CH2SCH2Pr-c Pr-c
CH2SCH2Pr-c Bu-n
CH2SCH2Pr-c Bu-i
CH2SCH2Pr-c Bu-c
CH2SCH2Pr-c Bu-s
CH2SCH2Pr-c Bu-t
CH2SCH2Pr-c Pen-n
CH2SCH2Pr-c Pen-c
CH2SCH2Pr-c Hex-n
CH2SCH2Pr-c Hex-c
CH2SCH2Pr-c CH2Pr-c
CH2SCH2Pr-c CH2Bu-c
CH2SCH2Pr-c CH2Pen-c
CH2SCH2Pr-c CH2Hex-c
CH2SCH2Pr-c CH2CH = CH2
CH2SCH2Pr-c CH2CH = C (Cl)2
CH2SCH2Pr-c CH2Pr-c
CH2SCH2Pr-c CH2CN
CH2SCH2Pr-c CH2CFThree
CH2SCH2Pr-c CH2OMe
CH2SCH2Pr-c CH2OCFThree
CH2SCH2Pr-c CH2SMe
CH2SCH2Pr-c CH2S (O) Me
CH2SCH2Pr-c CH2S (O)2Me
CH2SCH2Pr-c CH2SCFThree
CH2SCH2Pr-c CH2S (O) CFThree
CH2SCH2Pr-c CH2S (O)2CFThree
CH2SCH2Pr-c CH2CH (OMe)2
CH2SCH2Pr-c CH2CH (SMe)2
CH2SCH2Pr-c CH2C (O) Me
CH2SCH2Pr-c CH2C (O) CFThree
CH2SCH2Pr-c CH2C (O) OMe
CH2SCH2Pr-c CH2(D1-32a)
CH2SCH2Pr-c CH2(D1-33a)
CH2SCH2Pr-c CH2(D1-34a)
CH2SCH2Pr-c CH2(D1-37a)
CH2SCH2Pr-c CH2(D1-81a)
CH2SCH2Pr-c CH2(D1-82a)
CH2SCH2Pr-c CH2(D1-84a)
CH2SCH2Pr-c CH2(D1-85a)
CH2SCH2Pr-c CH2(D1-87a)
CH2SCH2Pr-c CH2(D1-92a)
CH2SCH2Pr-c CH2(D1-93a)
CH2SCH2Pr-c CH2(D1-95a)
CH2SCH2Pr-c CH2(D1-96a)
CH2SCH2Pr-c CH2(D1-98a)
CH2SCH2Pr-c CH2(D1-108a)
CH2SCH2Pr-c CH2(D1-108b, Z = 2-Cl)
CH2SCH2Pr-c CH2(D1-108b, Z = 3-Me)
CH2SCH2Pr-c CH2(D1-108b, Z = 4-OMe)
CH2SCH2Pr-c CH2(D1-108b, Z = 2-SMe)
CH2SCH2Pr-c CH2(D1-108b, Z = 3-CFThree)
CH2SCH2Pr-c CH2(D1-108b, Z = 4-OCFThree)
CH2SCH2Pr-c CH2(D1-108b, Z = 2-SCFThree)
CH2SCH2Pr-c CH2CH2CN
CH2SCH2Pr-c CH2CH2CFThree
CH2SCH2Pr-c CH2CH2OMe
CH2SCH2Pr-c CH2CH2SMe
CH2SCH2Pr-c CH2CH2S (O) Me
CH2SCH2Pr-c CH2CH2S (O)2Me
CH2SCH2Pr-c D1-32a
CH2SCH2Pr-c D1-33a
CH2SCH2Pr-c D1-34a
CH2SCH2Pr-c D1-37a
CH2SCH2Pr-c D1-81a
CH2SCH2Pr-c D1-82a
CH2SCH2Pr-c D1-84a
CH2SCH2Pr-c D1-85a
CH2SCH2Pr-c D1-87a
CH2SCH2Pr-c D1-92a
CH2SCH2Pr-c D1-93a
CH2SCH2Pr-c D1-95a
CH2SCH2Pr-c D1-96a
CH2SCH2Pr-c D1-98a
CH2SCH2Pr-c D1-108a
CH2SCH2Pr-c D1-108b (Z = 2-Cl)
CH2SCH2Pr-c D1-108b (Z = 3-Me)
CH2SCH2Pr-c D1-108b (Z = 4-OMe)
CH2SCH2Pr-c D1-108b (Z = 2-SMe)
CH2SCH2Pr-c D1-108b (Z = 3-CFThree)
CH2SCH2Pr-c D1-108b (Z = 4-OCFThree)
CH2SCH2Pr-c D1-108b (Z = 2-SCFThree)
CH2SCH2Pr-c C (O) Me
CH2SCH2Pr-c C (O) CFThree
CH2SCH2Pr-c C (O) OMe
CH2S (O) CH2Pr-c Me
CH2S (O) CH2Pr-c Et
CH2S (O) CH2Pr-c Pr-n
CH2S (O) CH2Pr-c Pr-i
CH2S (O) CH2Pr-c Pr-c
CH2S (O) CH2Pr-c Bu-n
CH2S (O) CH2Pr-c Bu-i
CH2S (O) CH2Pr-c Bu-c
CH2S (O) CH2Pr-c Bu-s
CH2S (O) CH2Pr-c Bu-t
CH2S (O) CH2Pr-c Pen-n
CH2S (O) CH2Pr-c Pen-c
CH2S (O) CH2Pr-c Hex-n
CH2S (O) CH2Pr-c Hex-c
CH2S (O) CH2Pr-c CH2Pr-c
CH2S (O) CH2Pr-c CH2Bu-c
CH2S (O) CH2Pr-c CH2Pen-c
CH2S (O) CH2Pr-c CH2Hex-c
CH2S (O) CH2Pr-c CH2CH = CH2
CH2S (O) CH2Pr-c CH2CH = C (Cl)2
CH2S (O) CH2Pr-c CH2C≡CH
CH2S (O) CH2Pr-c CH2CN
CH2S (O) CH2Pr-c CH2CFThree
CH2S (O) CH2Pr-c CH2OMe
CH2S (O) CH2Pr-c CH2OCFThree
CH2S (O) CH2Pr-c CH2SMe
CH2S (O) CH2Pr-c CH2S (O) Me
CH2S (O) CH2Pr-c CH2S (O)2Me
CH2S (O) CH2Pr-c CH2SCFThree
CH2S (O) CH2Pr-c CH2S (O) CFThree
CH2S (O) CH2Pr-c CH2S (O)2CFThree
CH2S (O) CH2Pr-c CH2CH (OMe)2
CH2S (O) CH2Pr-c CH2CH (SMe)2
CH2S (O) CH2Pr-c CH2C (O) Me
CH2S (O) CH2Pr-c CH2C (O) CFThree
CH2S (O) CH2Pr-c CH2C (O) OMe
CH2S (O) CH2Pr-c CH2(D1-32a)
CH2S (O) CH2Pr-c CH2(D1-33a)
CH2S (O) CH2Pr-c CH2(D1-34a)
CH2S (O) CH2Pr-c CH2(D1-37a)
CH2S (O) CH2Pr-c CH2(D1-81a)
CH2S (O) CH2Pr-c CH2(D1-82a)
CH2S (O) CH2Pr-c CH2(D1-84a)
CH2S (O) CH2Pr-c CH2(D1-85a)
CH2S (O) CH2Pr-c CH2(D1-87a)
CH2S (O) CH2Pr-c CH2(D1-92a)
CH2S (O) CH2Pr-c CH2(D1-93a)
CH2S (O) CH2Pr-c CH2(D1-95a)
CH2S (O) CH2Pr-c CH2(D1-96a)
CH2S (O) CH2Pr-c CH2(D1-98a)
CH2S (O) CH2Pr-c CH2(D1-108a)
CH2S (O) CH2Pr-c CH2(D1-108b, Z = 2-Cl)
CH2S (O) CH2Pr-c CH2(D1-108b, Z = 3-Me)
CH2S (O) CH2Pr-c CH2(D1-108b, Z = 4-OMe)
CH2S (O) CH2Pr-c CH2(D1-108b, Z = 2-SMe)
CH2S (O) CH2Pr-c CH2(D1-108b, Z = 3-CFThree)
CH2S (O) CH2Pr-c CH2(D1-108b, Z = 4-OCFThree)
CH2S (O) CH2Pr-c CH2(D1-108b, Z = 2-SCFThree)
CH2S (O) CH2Pr-c CH2CH2CN
CH2S (O) CH2Pr-c CH2CH2CFThree
CH2S (O) CH2Pr-c CH2CH2OMe
CH2S (O) CH2Pr-c CH2CH2SMe
CH2S (O) CH2Pr-c CH2CH2S (O) Me
CH2S (O) CH2Pr-c CH2CH2S (O)2Me
CH2S (O) CH2Pr-c D1-32a
CH2S (O) CH2Pr-c D1-33a
CH2S (O) CH2Pr-c D1-34a
CH2S (O) CH2Pr-c D1-37a
CH2S (O) CH2Pr-c D1-81a
CH2S (O) CH2Pr-c D1-82a
CH2S (O) CH2Pr-c D1-84a
CH2S (O) CH2Pr-c D1-85a
CH2S (O) CH2Pr-c D1-87a
CH2S (O) CH2Pr-c D1-92a
CH2S (O) CH2Pr-c D1-93a
CH2S (O) CH2Pr-c D1-95a
CH2S (O) CH2Pr-c D1-96a
CH2S (O) CH2Pr-c D1-98a
CH2S (O) CH2Pr-c D1-108a
CH2S (O) CH2Pr-c D1-108b (Z = 2-Cl)
CH2S (O) CH2Pr-c D1-108b (Z = 3-Me)
CH2S (O) CH2Pr-c D1-108b (Z = 4-OMe)
CH2S (O) CH2Pr-c D1-108b (Z = 2-SMe)
CH2S (O) CH2Pr-c D1-108b (Z = 3-CFThree)
CH2S (O) CH2Pr-c D1-108b (Z = 4-OCFThree)
CH2S (O) CH2Pr-c D1-108b (Z = 2-SCFThree)
CH2S (O) CH2Pr-c C (O) Me
CH2S (O) CH2Pr-c C (O) CFThree
CH2S (O) CH2Pr-c C (O) OMe
CH2S (O)2CH2Pr-c Me
CH2S (O)2CH2Pr-c Et
CH2S (O)2CH2Pr-c Pr-n
CH2S (O)2CH2Pr-c Pr-i
CH2S (O)2CH2Pr-c Pr-c
CH2S (O)2CH2Pr-c Bu-n
CH2S (O)2CH2Pr-c Bu-i
CH2S (O)2CH2Pr-c Bu-c
CH2S (O)2CH2Pr-c Bu-s
CH2S (O)2CH2Pr-c Bu-t
CH2S (O)2CH2Pr-c Pen-n
CH2S (O)2CH2Pr-c Pen-c
CH2S (O)2CH2Pr-c Hex-n
CH2S (O)2CH2Pr-c Hex-c
CH2S (O)2CH2Pr-c CH2Pr-c
CH2S (O)2CH2Pr-c CH2Bu-c
CH2S (O)2CH2Pr-c CH2Pen-c
CH2S (O)2CH2Pr-c CH2Hex-c
CH2S (O)2CH2Pr-c CH2CH = CH2
CH2S (O)2CH2Pr-c CH2CH = C (Cl)2
CH2S (O)2CH2Pr-c CH2C≡CH
CH2S (O)2CH2Pr-c CH2CN
CH2S (O)2CH2Pr-c CH2CFThree
CH2S (O)2CH2Pr-c CH2OMe
CH2S (O)2CH2Pr-c CH2OCFThree
CH2S (O)2CH2Pr-c CH2SMe
CH2S (O)2CH2Pr-c CH2S (O) Me
CH2S (O)2CH2Pr-c CH2S (O)2Me
CH2S (O)2CH2Pr-c CH2SCFThree
CH2S (O)2CH2Pr-c CH2S (O) CFThree
CH2S (O)2CH2Pr-c CH2S (O)2CFThree
CH2S (O)2CH2Pr-c CH2CH (OMe)2
CH2S (O)2CH2Pr-c CH2CH (SMe)2
CH2S (O)2CH2Pr-c CH2C (O) Me
CH2S (O)2CH2Pr-c CH2C (O) CFThree
CH2S (O)2CH2Pr-c CH2C (O) OMe
CH2S (O)2CH2Pr-c CH2(D1-32a)
CH2S (O)2CH2Pr-c CH2(D1-33a)
CH2S (O)2CH2Pr-c CH2(D1-34a)
CH2S (O)2CH2Pr-c CH2(D1-37a)
CH2S (O)2CH2Pr-c CH2(D1-81a)
CH2S (O)2CH2Pr-c CH2(D1-82a)
CH2S (O)2CH2Pr-c CH2(D1-84a)
CH2S (O)2CH2Pr-c CH2(D1-85a)
CH2S (O)2CH2Pr-c CH2(D1-87a)
CH2S (O)2CH2Pr-c CH2(D1-92a)
CH2S (O)2CH2Pr-c CH2(D1-93a)
CH2S (O)2CH2Pr-c CH2(D1-95a)
CH2S (O)2CH2Pr-c CH2(D1-96a)
CH2S (O)2CH2Pr-c CH2(D1-98a)
CH2S (O)2CH2Pr-c CH2(D1-108a)
CH2S (O)2CH2Pr-c CH2(D1-108b, Z = 2-Cl)
CH2S (O)2CH2Pr-c CH2(D1-108b, Z = 3-Me)
CH2S (O)2CH2Pr-c CH2(D1-108b, Z = 4-OMe)
CH2S (O)2CH2Pr-c CH2(D1-108b, Z = 2-SMe)
CH2S (O)2CH2Pr-c CH2(D1-108b, Z = 3-CFThree)
CH2S (O)2CH2Pr-c CH2(D1-108b, Z = 4-OCFThree)
CH2S (O)2CH2Pr-c CH2(D1-108b, Z = 2-SCFThree)
CH2S (O)2CH2Pr-c CH2CH2CN
CH2S (O)2CH2Pr-c CH2CH2CFThree
CH2S (O)2CH2Pr-c CH2CH2OMe
CH2S (O)2CH2Pr-c CH2CH2SMe
CH2S (O)2CH2Pr-c CH2CH2S (O) Me
CH2S (O)2CH2Pr-c CH2CH2S (O)2Me
CH2S (O)2CH2Pr-c D1-32a
CH2S (O)2CH2Pr-c D1-33a
CH2S (O)2CH2Pr-c D1-34a
CH2S (O)2CH2Pr-c D1-37a
CH2S (O)2CH2Pr-c D1-81a
CH2S (O)2CH2Pr-c D1-82a
CH2S (O)2CH2Pr-c D1-84a
CH2S (O)2CH2Pr-c D1-85a
CH2S (O)2CH2Pr-c D1-87a
CH2S (O)2CH2Pr-c D1-92a
CH2S (O)2CH2Pr-c D1-93a
CH2S (O)2CH2Pr-c D1-95a
CH2S (O)2CH2Pr-c D1-96a
CH2S (O)2CH2Pr-c D1-98a
CH2S (O)2CH2Pr-c D1-108a
CH2S (O)2CH2Pr-c D1-108b (Z = 2-Cl)
CH2S (O)2CH2Pr-c D1-108b (Z = 3-Me)
CH2S (O)2CH2Pr-c D1-108b (Z = 4-OMe)
CH2S (O)2CH2Pr-c D1-108b (Z = 2-SMe)
CH2S (O)2CH2Pr-c D1-108b (Z = 3-CFThree)
CH2S (O)2CH2Pr-c D1-108b (Z = 4-OCFThree)
CH2S (O)2CH2Pr-c D1-108b (Z = 2-SCFThree)
CH2S (O)2CH2Pr-c C (O) Me
CH2S (O)2CH2Pr-c C (O) CFThree
CH2S (O)2CH2Pr-c C (O) OMe
CH (Me) SCH2Pr-c Me
CH (Me) SCH2Pr-c Et
CH (Me) SCH2Pr-c Pr-n
CH (Me) SCH2Pr-c Pr-i
CH (Me) SCH2Pr-c Pr-c
CH (Me) SCH2Pr-c Bu-n
CH (Me) SCH2Pr-c Bu-i
CH (Me) SCH2Pr-c Bu-c
CH (Me) SCH2Pr-c Bu-s
CH (Me) SCH2Pr-c Bu-t
CH (Me) SCH2Pr-c Pen-n
CH (Me) SCH2Pr-c Pen-c
CH (Me) SCH2Pr-c Hex-n
CH (Me) SCH2Pr-c Hex-c
CH (Me) SCH2Pr-c CH2Pr-c
CH (Me) SCH2Pr-c CH2Bu-c
CH (Me) SCH2Pr-c CH2Pen-c
CH (Me) SCH2Pr-c CH2Hex-c
CH (Me) SCH2Pr-c CH2CH = CH2
CH (Me) SCH2Pr-c CH2CH = C (Cl)2
CH (Me) SCH2Pr-c CH2C≡CH
CH (Me) SCH2Pr-c CH2CN
CH (Me) SCH2Pr-c CH2CFThree
CH (Me) SCH2Pr-c CH2OMe
CH (Me) SCH2Pr-c CH2OCFThree
CH (Me) SCH2Pr-c CH2SMe
CH (Me) SCH2Pr-c CH2S (O) Me
CH (Me) SCH2Pr-c CH2S (O)2Me
CH (Me) SCH2Pr-c CH2SCFThree
CH (Me) SCH2Pr-c CH2S (O) CFThree
CH (Me) SCH2Pr-c CH2S (O)2CFThree
CH (Me) SCH2Pr-c CH2CH (OMe)2
CH (Me) SCH2Pr-c CH2CH (SMe)2
CH (Me) SCH2Pr-c CH2C (O) Me
CH (Me) SCH2Pr-c CH2C (O) CFThree
CH (Me) SCH2Pr-c CH2C (O) OMe
CH (Me) SCH2Pr-c CH2(D1-32a)
CH (Me) SCH2Pr-c CH2(D1-33a)
CH (Me) SCH2Pr-c CH2(D1-34a)
CH (Me) SCH2Pr-c CH2(D1-37a)
CH (Me) SCH2Pr-c CH2(D1-81a)
CH (Me) SCH2Pr-c CH2(D1-82a)
CH (Me) SCH2Pr-c CH2(D1-84a)
CH (Me) SCH2Pr-c CH2(D1-85a)
CH (Me) SCH2Pr-c CH2(D1-87a)
CH (Me) SCH2Pr-c CH2(D1-92a)
CH (Me) SCH2Pr-c CH2(D1-93a)
CH (Me) SCH2Pr-c CH2(D1-95a)
CH (Me) SCH2Pr-c CH2(D1-96a)
CH (Me) SCH2Pr-c CH2(D1-98a)
CH (Me) SCH2Pr-c CH2(D1-108a)
CH (Me) SCH2Pr-c CH2(D1-108b, Z = 2-Cl)
CH (Me) SCH2Pr-c CH2(D1-108b, Z = 3-Me)
CH (Me) SCH2Pr-c CH2(D1-108b, Z = 4-OMe)
CH (Me) SCH2Pr-c CH2(D1-108b, Z = 2-SMe)
CH (Me) SCH2Pr-c CH2(D1-108b, Z = 3-CFThree)
CH (Me) SCH2Pr-c CH2(D1-108b, Z = 4-OCFThree)
CH (Me) SCH2Pr-c CH2(D1-108b, Z = 2-SCFThree)
CH (Me) SCH2Pr-c CH2CH2CN
CH (Me) SCH2Pr-c CH2CH2CFThree
CH (Me) SCH2Pr-c CH2CH2OMe
CH (Me) SCH2Pr-c CH2CH2SMe
CH (Me) SCH2Pr-c CH2CH2S (O) Me
CH (Me) SCH2Pr-c CH2CH2S (O)2Me
CH (Me) SCH2Pr-c D1-32a
CH (Me) SCH2Pr-c D1-33a
CH (Me) SCH2Pr-c D1-34a
CH (Me) SCH2Pr-c D1-37a
CH (Me) SCH2Pr-c D1-81a
CH (Me) SCH2Pr-c D1-82a
CH (Me) SCH2Pr-c D1-84a
CH (Me) SCH2Pr-c D1-85a
CH (Me) SCH2Pr-c D1-87a
CH (Me) SCH2Pr-c D1-92a
CH (Me) SCH2Pr-c D1-93a
CH (Me) SCH2Pr-c D1-95a
CH (Me) SCH2Pr-c D1-96a
CH (Me) SCH2Pr-c D1-98a
CH (Me) SCH2Pr-c D1-108a
CH (Me) SCH2Pr-c D1-108b (Z = 2-Cl)
CH (Me) SCH2Pr-c D1-108b (Z = 3-Me)
CH (Me) SCH2Pr-c D1-108b (Z = 4-OMe)
CH (Me) SCH2Pr-c D1-108b (Z = 2-SMe)
CH (Me) SCH2Pr-c D1-108b (Z = 3-CFThree)
CH (Me) SCH2Pr-c D1-108b (Z = 4-OCFThree)
CH (Me) SCH2Pr-c D1-108b (Z = 2-SCFThree)
CH (Me) SCH2Pr-c C (O) Me
CH (Me) SCH2Pr-c C (O) CFThree
CH (Me) SCH2Pr-c C (O) OMe
CH (Me) S (O) CH2Pr-c Me
CH (Me) S (O) CH2Pr-c Et
CH (Me) S (O) CH2Pr-c Pr-n
CH (Me) S (O) CH2Pr-c Pr-i
CH (Me) S (O) CH2Pr-c Pr-c
CH (Me) S (O) CH2Pr-c Bu-n
CH (Me) S (O) CH2Pr-c Bu-i
CH (Me) S (O) CH2Pr-c Bu-c
CH (Me) S (O) CH2Pr-c Bu-s
CH (Me) S (O) CH2Pr-c Bu-t
CH (Me) S (O) CH2Pr-c Pen-n
CH (Me) S (O) CH2Pr-c Pen-c
CH (Me) S (O) CH2Pr-c Hex-n
CH (Me) S (O) CH2Pr-c Hex-c
CH (Me) S (O) CH2Pr-c CH2Pr-c
CH (Me) S (O) CH2Pr-c CH2Bu-c
CH (Me) S (O) CH2Pr-c CH2Pen-c
CH (Me) S (O) CH2Pr-c CH2Hex-c
CH (Me) S (O) CH2Pr-c CH2CH = CH2
CH (Me) S (O) CH2Pr-c CH2CH = C (Cl)2
CH (Me) S (O) CH2Pr-c CH2C≡CH
CH (Me) S (O) CH2Pr-c CH2CN
CH (Me) S (O) CH2Pr-c CH2CFThree
CH (Me) S (O) CH2Pr-c CH2OMe
CH (Me) S (O) CH2Pr-c CH2OCFThree
CH (Me) S (O) CH2Pr-c CH2SMe
CH (Me) S (O) CH2Pr-c CH2S (O) Me
CH (Me) S (O) CH2Pr-c CH2S (O)2Me
CH (Me) S (O) CH2Pr-c CH2SCFThree
CH (Me) S (O) CH2Pr-c CH2S (O) CFThree
CH (Me) S (O) CH2Pr-c CH2S (O)2CFThree
CH (Me) S (O) CH2Pr-c CH2CH (OMe)2
CH (Me) S (O) CH2Pr-c CH2CH (SMe)2
CH (Me) S (O) CH2Pr-c CH2C (O) Me
CH (Me) S (O) CH2Pr-c CH2C (O) CFThree
CH (Me) S (O) CH2Pr-c CH2C (O) OMe
CH (Me) S (O) CH2Pr-c CH2(D1-32a)
CH (Me) S (O) CH2Pr-c CH2(D1-33a)
CH (Me) S (O) CH2Pr-c CH2(D1-34a)
CH (Me) S (O) CH2Pr-c CH2(D1-37a)
CH (Me) S (O) CH2Pr-c CH2(D1-81a)
CH (Me) S (O) CH2Pr-c CH2(D1-82a)
CH (Me) S (O) CH2Pr-c CH2(D1-84a)
CH (Me) S (O) CH2Pr-c CH2(D1-85a)
CH (Me) S (O) CH2Pr-c CH2(D1-87a)
CH (Me) S (O) CH2Pr-c CH2(D1-92a)
CH (Me) S (O) CH2Pr-c CH2(D1-93a)
CH (Me) S (O) CH2Pr-c CH2(D1-95a)
CH (Me) S (O) CH2Pr-c CH2(D1-96a)
CH (Me) S (O) CH2Pr-c CH2(D1-98a)
CH (Me) S (O) CH2Pr-c CH2(D1-108a)
CH (Me) S (O) CH2Pr-c CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O) CH2Pr-c CH2(D1-108b, Z = 3-Me)
CH (Me) S (O) CH2Pr-c CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O) CH2Pr-c CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O) CH2Pr-c CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O) CH2Pr-c CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O) CH2Pr-c CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O) CH2Pr-c CH2CH2CN
CH (Me) S (O) CH2Pr-c CH2CH2CFThree
CH (Me) S (O) CH2Pr-c CH2CH2OMe
CH (Me) S (O) CH2Pr-c CH2CH2SMe
CH (Me) S (O) CH2Pr-c CH2CH2S (O) Me
CH (Me) S (O) CH2Pr-c CH2CH2S (O)2Me
CH (Me) S (O) CH2Pr-c D1-32a
CH (Me) S (O) CH2Pr-c D1-33a
CH (Me) S (O) CH2Pr-c D1-34a
CH (Me) S (O) CH2Pr-c D1-37a
CH (Me) S (O) CH2Pr-c D1-81a
CH (Me) S (O) CH2Pr-c D1-82a
CH (Me) S (O) CH2Pr-c D1-84a
CH (Me) S (O) CH2Pr-c D1-85a
CH (Me) S (O) CH2Pr-c D1-87a
CH (Me) S (O) CH2Pr-c D1-92a
CH (Me) S (O) CH2Pr-c D1-93a
CH (Me) S (O) CH2Pr-c D1-95a
CH (Me) S (O) CH2Pr-c D1-96a
CH (Me) S (O) CH2Pr-c D1-98a
CH (Me) S (O) CH2Pr-c D1-108a
CH (Me) S (O) CH2Pr-c D1-108b (Z = 2-Cl)
CH (Me) S (O) CH2Pr-c D1-108b (Z = 3-Me)
CH (Me) S (O) CH2Pr-c D1-108b (Z = 4-OMe)
CH (Me) S (O) CH2Pr-c D1-108b (Z = 2-SMe)
CH (Me) S (O) CH2Pr-c D1-108b (Z = 3-CFThree)
CH (Me) S (O) CH2Pr-c D1-108b (Z = 4-OCFThree)
CH (Me) S (O) CH2Pr-c D1-108b (Z = 2-SCFThree)
CH (Me) S (O) CH2Pr-c C (O) Me
CH (Me) S (O) CH2Pr-c C (O) CFThree
CH (Me) S (O) CH2Pr-c C (O) OMe
CH (Me) S (O)2CH2Pr-c Me
CH (Me) S (O)2CH2Pr-c Et
CH (Me) S (O)2CH2Pr-c Pr-n
CH (Me) S (O)2CH2Pr-c Pr-i
CH (Me) S (O)2CH2Pr-c Pr-c
CH (Me) S (O)2CH2Pr-c Bu-n
CH (Me) S (O)2CH2Pr-c Bu-i
CH (Me) S (O)2CH2Pr-c Bu-c
CH (Me) S (O)2CH2Pr-c Bu-s
CH (Me) S (O)2CH2Pr-c Bu-t
CH (Me) S (O)2CH2Pr-c Pen-n
CH (Me) S (O)2CH2Pr-c Pen-c
CH (Me) S (O)2CH2Pr-c Hex-n
CH (Me) S (O)2CH2Pr-c Hex-c
CH (Me) S (O)2CH2Pr-c CH2Pr-c
CH (Me) S (O)2CH2Pr-c CH2Bu-c
CH (Me) S (O)2CH2Pr-c CH2Pen-c
CH (Me) S (O)2CH2Pr-c CH2Hex-c
CH (Me) S (O)2CH2Pr-c CH2CH = CH2
CH (Me) S (O)2CH2Pr-c CH2CH = C (Cl)2
CH (Me) S (O)2CH2Pr-c CH2C≡CH
CH (Me) S (O)2CH2Pr-c CH2CN
CH (Me) S (O)2CH2Pr-c CH2CFThree
CH (Me) S (O)2CH2Pr-c CH2OMe
CH (Me) S (O)2CH2Pr-c CH2OCFThree
CH (Me) S (O)2CH2Pr-c CH2SMe
CH (Me) S (O)2CH2Pr-c CH2S (O) Me
CH (Me) S (O)2CH2Pr-c CH2S (O)2Me
CH (Me) S (O)2CH2Pr-c CH2SCFThree
CH (Me) S (O)2CH2Pr-c CH2S (O) CFThree
CH (Me) S (O)2CH2Pr-c CH2S (O)2CFThree
CH (Me) S (O)2CH2Pr-c CH2CH (OMe)2
CH (Me) S (O)2CH2Pr-c CH2CH (SMe)2
CH (Me) S (O)2CH2Pr-c CH2C (O) Me
CH (Me) S (O)2CH2Pr-c CH2C (O) CFThree
CH (Me) S (O)2CH2Pr-c CH2C (O) OMe
CH (Me) S (O)2CH2Pr-c CH2(D1-32a)
CH (Me) S (O)2CH2Pr-c CH2(D1-33a)
CH (Me) S (O)2CH2Pr-c CH2(D1-34a)
CH (Me) S (O)2CH2Pr-c CH2(D1-37a)
CH (Me) S (O)2CH2Pr-c CH2(D1-81a)
CH (Me) S (O)2CH2Pr-c CH2(D1-82a)
CH (Me) S (O)2CH2Pr-c CH2(D1-84a)
CH (Me) S (O)2CH2Pr-c CH2(D1-85a)
CH (Me) S (O)2CH2Pr-c CH2(D1-87a)
CH (Me) S (O)2CH2Pr-c CH2(D1-92a)
CH (Me) S (O)2CH2Pr-c CH2(D1-93a)
CH (Me) S (O)2CH2Pr-c CH2(D1-95a)
CH (Me) S (O)2CH2Pr-c CH2(D1-96a)
CH (Me) S (O)2CH2Pr-c CH2(D1-98a)
CH (Me) S (O)2CH2Pr-c CH2(D1-108a)
CH (Me) S (O)2CH2Pr-c CH2(D1-108b, Z = 2-Cl)
CH (Me) S (O)2CH2Pr-c CH2(D1-108b, Z = 3-Me)
CH (Me) S (O)2CH2Pr-c CH2(D1-108b, Z = 4-OMe)
CH (Me) S (O)2CH2Pr-c CH2(D1-108b, Z = 2-SMe)
CH (Me) S (O)2CH2Pr-c CH2(D1-108b, Z = 3-CFThree)
CH (Me) S (O)2CH2Pr-c CH2(D1-108b, Z = 4-OCFThree)
CH (Me) S (O)2CH2Pr-c CH2(D1-108b, Z = 2-SCFThree)
CH (Me) S (O)2CH2Pr-c CH2CH2CN
CH (Me) S (O)2CH2Pr-c CH2CH2CFThree
CH (Me) S (O)2CH2Pr-c CH2CH2OMe
CH (Me) S (O)2CH2Pr-c CH2CH2SMe
CH (Me) S (O)2CH2Pr-c CH2CH2S (O) Me
CH (Me) S (O)2CH2Pr-c CH2CH2S (O)2Me
CH (Me) S (O)2CH2Pr-c D1-32a
CH (Me) S (O)2CH2Pr-c D1-33a
CH (Me) S (O)2CH2Pr-c D1-34a
CH (Me) S (O)2CH2Pr-c D1-37a
CH (Me) S (O)2CH2Pr-c D1-81a
CH (Me) S (O)2CH2Pr-c D1-82a
CH (Me) S (O)2CH2Pr-c D1-84a
CH (Me) S (O)2CH2Pr-c D1-85a
CH (Me) S (O)2CH2Pr-c D1-87a
CH (Me) S (O)2CH2Pr-c D1-92a
CH (Me) S (O)2CH2Pr-c D1-93a
CH (Me) S (O)2CH2Pr-c D1-95a
CH (Me) S (O)2CH2Pr-c D1-96a
CH (Me) S (O)2CH2Pr-c D1-98a
CH (Me) S (O)2CH2Pr-c D1-108a
CH (Me) S (O)2CH2Pr-c D1-108b (Z = 2-Cl)
CH (Me) S (O)2CH2Pr-c D1-108b (Z = 3-Me)
CH (Me) S (O)2CH2Pr-c D1-108b (Z = 4-OMe)
CH (Me) S (O)2CH2Pr-c D1-108b (Z = 2-SMe)
CH (Me) S (O)2CH2Pr-c D1-108b (Z = 3-CFThree)
CH (Me) S (O)2CH2Pr-c D1-108b (Z = 4-OCFThree)
CH (Me) S (O)2CH2Pr-c D1-108b (Z = 2-SCFThree)
CH (Me) S (O)2CH2Pr-c C (O) Me
CH (Me) S (O)2CH2Pr-c C (O) CFThree
CH (Me) S (O)2CH2Pr-c C (O) OMe
CH (Et) SCH2Pr-c Me
CH (Et) SCH2Pr-c Et
CH (Et) SCH2Pr-c Pr-n
CH (Et) SCH2Pr-c Pr-i
CH (Et) SCH2Pr-c Pr-c
CH (Et) SCH2Pr-c Bu-n
CH (Et) SCH2Pr-c Bu-i
CH (Et) SCH2Pr-c Bu-c
CH (Et) SCH2Pr-c Bu-s
CH (Et) SCH2Pr-c Bu-t
CH (Et) SCH2Pr-c Pen-n
CH (Et) SCH2Pr-c Pen-c
CH (Et) SCH2Pr-c Hex-n
CH (Et) SCH2Pr-c Hex-c
CH (Et) SCH2Pr-c CH2Pr-c
CH (Et) SCH2Pr-c CH2Bu-c
CH (Et) SCH2Pr-c CH2Pen-c
CH (Et) SCH2Pr-c CH2Hex-c
CH (Et) SCH2Pr-c CH2CH = CH2
CH (Et) SCH2Pr-c CH2CH = C (Cl)2
CH (Et) SCH2Pr-c CH2C≡CH
CH (Et) SCH2Pr-c CH2CN
CH (Et) SCH2Pr-c CH2CFThree
CH (Et) SCH2Pr-c CH2OMe
CH (Et) SCH2Pr-c CH2OCFThree
CH (Et) SCH2Pr-c CH2SMe
CH (Et) SCH2Pr-c CH2S (O) Me
CH (Et) SCH2Pr-c CH2S (O)2Me
CH (Et) SCH2Pr-c CH2SCFThree
CH (Et) SCH2Pr-c CH2S (O) CFThree
CH (Et) SCH2Pr-c CH2S (O)2CFThree
CH (Et) SCH2Pr-c CH2CH (OMe)2
CH (Et) SCH2Pr-c CH2CH (SMe)2
CH (Et) SCH2Pr-c CH2C (O) Me
CH (Et) SCH2Pr-c CH2C (O) CFThree
CH (Et) SCH2Pr-c CH2C (O) OMe
CH (Et) SCH2Pr-c CH2(D1-32a)
CH (Et) SCH2Pr-c CH2(D1-33a)
CH (Et) SCH2Pr-c CH2(D1-34a)
CH (Et) SCH2Pr-c CH2(D1-37a)
CH (Et) SCH2Pr-c CH2(D1-81a)
CH (Et) SCH2Pr-c CH2(D1-82a)
CH (Et) SCH2Pr-c CH2(D1-84a)
CH (Et) SCH2Pr-c CH2(D1-85a)
CH (Et) SCH2Pr-c CH2(D1-87a)
CH (Et) SCH2Pr-c CH2(D1-92a)
CH (Et) SCH2Pr-c CH2(D1-93a)
CH (Et) SCH2Pr-c CH2(D1-95a)
CH (Et) SCH2Pr-c CH2(D1-96a)
CH (Et) SCH2Pr-c CH2(D1-98a)
CH (Et) SCH2Pr-c CH2(D1-108a)
CH (Et) SCH2Pr-c CH2(D1-108b, Z = 2-Cl)
CH (Et) SCH2Pr-c CH2(D1-108b, Z = 3-Me)
CH (Et) SCH2Pr-c CH2(D1-108b, Z = 4-OMe)
CH (Et) SCH2Pr-c CH2(D1-108b, Z = 2-SMe)
CH (Et) SCH2Pr-c CH2(D1-108b, Z = 3-CFThree)
CH (Et) SCH2Pr-c CH2(D1-108b, Z = 4-OCFThree)
CH (Et) SCH2Pr-c CH2(D1-108b, Z = 2-SCFThree)
CH (Et) SCH2Pr-c CH2CH2CN
CH (Et) SCH2Pr-c CH2CH2CFThree
CH (Et) SCH2Pr-c CH2CH2OMe
CH (Et) SCH2Pr-c CH2CH2SMe
CH (Et) SCH2Pr-c CH2CH2S (O) Me
CH (Et) SCH2Pr-c CH2CH2S (O)2Me
CH (Et) SCH2Pr-c D1-32a
CH (Et) SCH2Pr-c D1-33a
CH (Et) SCH2Pr-c D1-34a
CH (Et) SCH2Pr-c D1-37a
CH (Et) SCH2Pr-c D1-81a
CH (Et) SCH2Pr-c D1-82a
CH (Et) SCH2Pr-c D1-84a
CH (Et) SCH2Pr-c D1-85a
CH (Et) SCH2Pr-c D1-87a
CH (Et) SCH2Pr-c D1-92a
CH (Et) SCH2Pr-c D1-93a
CH (Et) SCH2Pr-c D1-95a
CH (Et) SCH2Pr-c D1-96a
CH (Et) SCH2Pr-c D1-98a
CH (Et) SCH2Pr-c D1-108a
CH (Et) SCH2Pr-c D1-108b (Z = 2-Cl)
CH (Et) SCH2Pr-c D1-108b (Z = 3-Me)
CH (Et) SCH2Pr-c D1-108b (Z = 4-OMe)
CH (Et) SCH2Pr-c D1-108b (Z = 2-SMe)
CH (Et) SCH2Pr-c D1-108b (Z = 3-CFThree)
CH (Et) SCH2Pr-c D1-108b (Z = 4-OCFThree)
CH (Et) SCH2Pr-c D1-108b (Z = 2-SCFThree)
CH (Et) SCH2Pr-c C (O) Me
CH (Et) SCH2Pr-c C (O) CFThree
CH (Et) SCH2Pr-c C (O) OMe
CH (Et) S (O) CH2Pr-c Me
CH (Et) S (O) CH2Pr-c Et
CH (Et) S (O) CH2Pr-c Pr-n
CH (Et) S (O) CH2Pr-c Pr-i
CH (Et) S (O) CH2Pr-c Pr-c
CH (Et) S (O) CH2Pr-c Bu-n
CH (Et) S (O) CH2Pr-c Bu-i
CH (Et) S (O) CH2Pr-c Bu-c
CH (Et) S (O) CH2Pr-c Bu-s
CH (Et) S (O) CH2Pr-c Bu-t
CH (Et) S (O) CH2Pr-c Pen-n
CH (Et) S (O) CH2Pr-c Pen-c
CH (Et) S (O) CH2Pr-c Hex-n
CH (Et) S (O) CH2Pr-c Hex-c
CH (Et) S (O) CH2Pr-c CH2Pr-c
CH (Et) S (O) CH2Pr-c CH2Bu-c
CH (Et) S (O) CH2Pr-c CH2Pen-c
CH (Et) S (O) CH2Pr-c CH2Hex-c
CH (Et) S (O) CH2Pr-c CH2CH = CH2
CH (Et) S (O) CH2Pr-c CH2CH = C (Cl)2
CH (Et) S (O) CH2Pr-c CH2C≡CH
CH (Et) S (O) CH2Pr-c CH2CN
CH (Et) S (O) CH2Pr-c CH2CFThree
CH (Et) S (O) CH2Pr-c CH2OMe
CH (Et) S (O) CH2Pr-c CH2OCFThree
CH (Et) S (O) CH2Pr-c CH2SMe
CH (Et) S (O) CH2Pr-c CH2S (O) Me
CH (Et) S (O) CH2Pr-c CH2S (O)2Me
CH (Et) S (O) CH2Pr-c CH2SCFThree
CH (Et) S (O) CH2Pr-c CH2S (O) CFThree
CH (Et) S (O) CH2Pr-c CH2S (O)2CFThree
CH (Et) S (O) CH2Pr-c CH2CH (OMe)2
CH (Et) S (O) CH2Pr-c CH2CH (SMe)2
CH (Et) S (O) CH2Pr-c CH2C (O) Me
CH (Et) S (O) CH2Pr-c CH2C (O) CFThree
CH (Et) S (O) CH2Pr-c CH2C (O) OMe
CH (Et) S (O) CH2Pr-c CH2(D1-32a)
CH (Et) S (O) CH2Pr-c CH2(D1-33a)
CH (Et) S (O) CH2Pr-c CH2(D1-34a)
CH (Et) S (O) CH2Pr-c CH2(D1-37a)
CH (Et) S (O) CH2Pr-c CH2(D1-81a)
CH (Et) S (O) CH2Pr-c CH2(D1-82a)
CH (Et) S (O) CH2Pr-c CH2(D1-84a)
CH (Et) S (O) CH2Pr-c CH2(D1-85a)
CH (Et) S (O) CH2Pr-c CH2(D1-87a)
CH (Et) S (O) CH2Pr-c CH2(D1-92a)
CH (Et) S (O) CH2Pr-c CH2(D1-93a)
CH (Et) S (O) CH2Pr-c CH2(D1-95a)
CH (Et) S (O) CH2Pr-c CH2(D1-96a)
CH (Et) S (O) CH2Pr-c CH2(D1-98a)
CH (Et) S (O) CH2Pr-c CH2(D1-108a)
CH (Et) S (O) CH2Pr-c CH2(D1-108b, Z = 2-Cl)
CH (Et) S (O) CH2Pr-c CH2(D1-108b, Z = 3-Me)
CH (Et) S (O) CH2Pr-c CH2(D1-108b, Z = 4-OMe)
CH (Et) S (O) CH2Pr-c CH2(D1-108b, Z = 2-SMe)
CH (Et) S (O) CH2Pr-c CH2(D1-108b, Z = 3-CFThree)
CH (Et) S (O) CH2Pr-c CH2(D1-108b, Z = 4-OCFThree)
CH (Et) S (O) CH2Pr-c CH2(D1-108b, Z = 2-SCFThree)
CH (Et) S (O) CH2Pr-c CH2CH2CN
CH (Et) S (O) CH2Pr-c CH2CH2CFThree
CH (Et) S (O) CH2Pr-c CH2CH2OMe
CH (Et) S (O) CH2Pr-c CH2CH2SMe
CH (Et) S (O) CH2Pr-c CH2CH2S (O) Me
CH (Et) S (O) CH2Pr-c CH2CH2S (O)2Me
CH (Et) S (O) CH2Pr-c D1-32a
CH (Et) S (O) CH2Pr-c D1-33a
CH (Et) S (O) CH2Pr-c D1-34a
CH (Et) S (O) CH2Pr-c D1-37a
CH (Et) S (O) CH2Pr-c D1-81a
CH (Et) S (O) CH2Pr-c D1-82a
CH (Et) S (O) CH2Pr-c D1-84a
CH (Et) S (O) CH2Pr-c D1-85a
CH (Et) S (O) CH2Pr-c D1-87a
CH (Et) S (O) CH2Pr-c D1-92a
CH (Et) S (O) CH2Pr-c D1-93a
CH (Et) S (O) CH2Pr-c D1-95a
CH (Et) S (O) CH2Pr-c D1-96a
CH (Et) S (O) CH2Pr-c D1-98a
CH (Et) S (O) CH2Pr-c D1-108a
CH (Et) S (O) CH2Pr-c D1-108b (Z = 2-Cl)
CH (Et) S (O) CH2Pr-c D1-108b (Z = 3-Me)
CH (Et) S (O) CH2Pr-c D1-108b (Z = 4-OMe)
CH (Et) S (O) CH2Pr-c D1-108b (Z = 2-SMe)
CH (Et) S (O) CH2Pr-c D1-108b (Z = 3-CFThree)
CH (Et) S (O) CH2Pr-c D1-108b (Z = 4-OCFThree)
CH (Et) S (O) CH2Pr-c D1-108b (Z = 2-SCFThree)
CH (Et) S (O) CH2Pr-c C (O) Me
CH (Et) S (O) CH2Pr-c C (O) CFThree
CH (Et) S (O) CH2Pr-c C (O) OMe
CH (Et) S (O)2CH2Pr-c Me
CH (Et) S (O)2CH2Pr-c Et
CH (Et) S (O)2CH2Pr-c Pr-n
CH (Et) S (O)2CH2Pr-c Pr-i
CH (Et) S (O)2CH2Pr-c Pr-c
CH (Et) S (O)2CH2Pr-c Bu-n
CH (Et) S (O)2CH2Pr-c Bu-i
CH (Et) S (O)2CH2Pr-c Bu-c
CH (Et) S (O)2CH2Pr-c Bu-s
CH (Et) S (O)2CH2Pr-c Bu-t
CH (Et) S (O)2CH2Pr-c Pen-n
CH (Et) S (O)2CH2Pr-c Pen-c
CH (Et) S (O)2CH2Pr-c Hex-n
CH (Et) S (O)2CH2Pr-c Hex-c
CH (Et) S (O)2CH2Pr-c CH2Pr-c
CH (Et) S (O)2CH2Pr-c CH2Bu-c
CH (Et) S (O)2CH2Pr-c CH2Pen-c
CH (Et) S (O)2CH2Pr-c CH2Hex-c
CH (Et) S (O)2CH2Pr-c CH2CH = CH2
CH (Et) S (O)2CH2Pr-c CH2CH = C (Cl)2
CH (Et) S (O)2CH2Pr-c CH2C≡CH
CH (Et) S (O)2CH2Pr-c CH2CN
CH (Et) S (O)2CH2Pr-c CH2CFThree
CH (Et) S (O)2CH2Pr-c CH2OMe
CH (Et) S (O)2CH2Pr-c CH2OCFThree
CH (Et) S (O)2CH2Pr-c CH2SMe
CH (Et) S (O)2CH2Pr-c CH2S (O) Me
CH (Et) S (O)2CH2Pr-c CH2S (O)2Me
CH (Et) S (O)2CH2Pr-c CH2SCFThree
CH (Et) S (O)2CH2Pr-c CH2S (O) CFThree
CH (Et) S (O)2CH2Pr-c CH2S (O)2CFThree
CH (Et) S (O)2CH2Pr-c CH2CH (OMe)2
CH (Et) S (O)2CH2Pr-c CH2CH (SMe)2
CH (Et) S (O)2CH2Pr-c CH2C (O) Me
CH (Et) S (O)2CH2Pr-c CH2C (O) CFThree
CH (Et) S (O)2CH2Pr-c CH2C (O) OMe
CH (Et) S (O)2CH2Pr-c CH2(D1-32a)
CH (Et) S (O)2CH2Pr-c CH2(D1-33a)
CH (Et) S (O)2CH2Pr-c CH2(D1-34a)
CH (Et) S (O)2CH2Pr-c CH2(D1-37a)
CH (Et) S (O)2CH2Pr-c CH2(D1-81a)
CH (Et) S (O)2CH2Pr-c CH2(D1-82a)
CH (Et) S (O)2CH2Pr-c CH2(D1-84a)
CH (Et) S (O)2CH2Pr-c CH2(D1-85a)
CH (Et) S (O)2CH2Pr-c CH2(D1-87a)
CH (Et) S (O)2CH2Pr-c CH2(D1-92a)
CH (Et) S (O)2CH2Pr-c CH2(D1-93a)
CH (Et) S (O)2CH2Pr-c CH2(D1-95a)
CH (Et) S (O)2CH2Pr-c CH2(D1-96a)
CH (Et) S (O)2CH2Pr-c CH2(D1-98a)
CH (Et) S (O)2CH2Pr-c CH2(D1-108a)
CH (Et) S (O)2CH2Pr-c CH2(D1-108b, Z = 2-Cl)
CH (Et) S (O)2CH2Pr-c CH2(D1-108b, Z = 3-Me)
CH (Et) S (O)2CH2Pr-c CH2(D1-108b, Z = 4-OMe)
CH (Et) S (O)2CH2Pr-c CH2(D1-108b, Z = 2-SMe)
CH (Et) S (O)2CH2Pr-c CH2(D1-108b, Z = 3-CFThree)
CH (Et) S (O)2CH2Pr-c CH2(D1-108b, Z = 4-OCFThree)
CH (Et) S (O)2CH2Pr-c CH2(D1-108b, Z = 2-SCFThree)
CH (Et) S (O)2CH2Pr-c CH2CH2CN
CH (Et) S (O)2CH2Pr-c CH2CH2CFThree
CH (Et) S (O)2CH2Pr-c CH2CH2OMe
CH (Et) S (O)2CH2Pr-c CH2CH2SMe
CH (Et) S (O)2CH2Pr-c CH2CH2S (O) Me
CH (Et) S (O)2CH2Pr-c CH2CH2S (O)2Me
CH (Et) S (O)2CH2Pr-c D1-32a
CH (Et) S (O)2CH2Pr-c D1-33a
CH (Et) S (O)2CH2Pr-c D1-34a
CH (Et) S (O)2CH2Pr-c D1-37a
CH (Et) S (O)2CH2Pr-c D1-81a
CH (Et) S (O)2CH2Pr-c D1-82a
CH (Et) S (O)2CH2Pr-c D1-84a
CH (Et) S (O)2CH2Pr-c D1-85a
CH (Et) S (O)2CH2Pr-c D1-87a
CH (Et) S (O)2CH2Pr-c D1-92a
CH (Et) S (O)2CH2Pr-c D1-93a
CH (Et) S (O)2CH2Pr-c D1-95a
CH (Et) S (O)2CH2Pr-c D1-96a
CH (Et) S (O)2CH2Pr-c D1-98a
CH (Et) S (O)2CH2Pr-c D1-108a
CH (Et) S (O)2CH2Pr-c D1-108b (Z = 2-Cl)
CH (Et) S (O)2CH2Pr-c D1-108b (Z = 3-Me)
CH (Et) S (O)2CH2Pr-c D1-108b (Z = 4-OMe)
CH (Et) S (O)2CH2Pr-c D1-108b (Z = 2-SMe)
CH (Et) S (O)2CH2Pr-c D1-108b (Z = 3-CFThree)
CH (Et) S (O)2CH2Pr-c D1-108b (Z = 4-OCFThree)
CH (Et) S (O)2CH2Pr-c D1-108b (Z = 2-SCFThree)
CH (Et) S (O)2CH2Pr-c C (O) Me
CH (Et) S (O)2CH2Pr-c C (O) CFThree
CH (Et) S (O)2CH2Pr-c C (O) OMe
CH2SCH2C (O) OMe Me
CH2SCH2C (O) OEt Me
CH2SCH2C (O) OPr-n Me
CH2SCH2C (O) OPr-i Me
CH2SCH2C (O) OBu-n Me
CH2SCH2C (O) OBu-i Me
CH2SCH2C (O) OBu-t Me
CH2SCH2C (O) OPen-n Me
CH2SCH2C (O) OHex-n Me
CH2SCH2C (O) OMe Et
CH2SCH2C (O) OMe Pr-n
CH2SCH2C (O) OMe Pr-i
CH2SCH2C (O) OMe Pr-c
CH2SCH2C (O) OMe Bu-n
CH2SCH2C (O) OMe Bu-i
CH2SCH2C (O) OMe Bu-c
CH2SCH2C (O) OMe Bu-s
CH2SCH2C (O) OMe Bu-t
CH2SCH2C (O) OMe Pen-n
CH2SCH2C (O) OMe Pen-c
CH2SCH2C (O) OMe Hex-n
CH2SCH2C (O) OMe Hex-c
CH2SCH2C (O) OMe CH2Pr-c
CH2SCH2C (O) OMe CH2Bu-c
CH2SCH2C (O) OMe CH2Pen-c
CH2SCH2C (O) OMe CH2Hex-c
CH2SCH2C (O) OMe CH2CH = CH2
CH2SCH2C (O) OMe CH2CH = C (Cl)2
CH2SCH2C (O) OMe CH2C≡CH
CH2SCH2C (O) OMe CH2CN
CH2SCH2C (O) OMe CH2CFThree
CH2SCH2C (O) OMe CH2OMe
CH2SCH2C (O) OMe CH2OCFThree
CH2SCH2C (O) OMe CH2SMe
CH2SCH2C (O) OMe CH2S (O) Me
CH2SCH2C (O) OMe CH2S (O)2Me
CH2SCH2C (O) OMe CH2SCFThree
CH2SCH2C (O) OMe CH2S (O) CFThree
CH2SCH2C (O) OMe CH2S (O)2CFThree
CH2SCH2C (O) OMe CH2CH (OMe)2
CH2SCH2C (O) OMe CH2CH (SMe)2
CH2SCH2C (O) OMe CH2C (O) Me
CH2SCH2C (O) OMe CH2C (O) CFThree
CH2SCH2C (O) OMe CH2C (O) OMe
CH2S (O) CH2C (O) OMe Me
CH2S (O) CH2C (O) OEt Me
CH2S (O) CH2C (O) OPr-n Me
CH2S (O) CH2C (O) OPr-i Me
CH2S (O) CH2C (O) OBu-n Me
CH2S (O) CH2C (O) OBu-i Me
CH2S (O) CH2C (O) OBu-t Me
CH2S (O) CH2C (O) OPen-n Me
CH2S (O) CH2C (O) OHex-n Me
CH2S (O) CH2C (O) OMe Et
CH2S (O) CH2C (O) OMe Pr-n
CH2S (O) CH2C (O) OMe Pr-i
CH2S (O) CH2C (O) OMe Pr-c
CH2S (O) CH2C (O) OMe Bu-n
CH2S (O) CH2C (O) OMe Bu-i
CH2S (O) CH2C (O) OMe Bu-c
CH2S (O) CH2C (O) OMe Bu-s
CH2S (O) CH2C (O) OMe Bu-t
CH2S (O) CH2C (O) OMe Pen-n
CH2S (O) CH2C (O) OMe Pen-c
CH2S (O) CH2C (O) OMe Hex-n
CH2S (O) CH2C (O) OMe Hex-c
CH2S (O) CH2C (O) OMe CH2Pr-c
CH2S (O) CH2C (O) OMe CH2Bu-c
CH2S (O) CH2C (O) OMe CH2Pen-c
CH2S (O) CH2C (O) OMe CH2Hex-c
CH2S (O) CH2C (O) OMe CH2CH = CH2
CH2S (O) CH2C (O) OMe CH2CH = C (Cl)2
CH2S (O) CH2C (O) OMe CH2C≡CH
CH2S (O) CH2C (O) OMe CH2CN
CH2S (O) CH2C (O) OMe CH2CFThree
CH2S (O) CH2C (O) OMe CH2OMe
CH2S (O) CH2C (O) OMe CH2OCFThree
CH2S (O) CH2C (O) OMe CH2SMe
CH2S (O) CH2C (O) OMe CH2S (O) Me
CH2S (O) CH2C (O) OMe CH2S (O)2Me
CH2S (O) CH2C (O) OMe CH2SCFThree
CH2S (O) CH2C (O) OMe CH2S (O) CFThree
CH2S (O) CH2C (O) OMe CH2S (O)2CFThree
CH2S (O) CH2C (O) OMe CH2CH (OMe)2
CH2S (O) CH2C (O) OMe CH2CH (SMe)2
CH2S (O) CH2C (O) OMe CH2C (O) Me
CH2S (O) CH2C (O) OMe CH2C (O) CFThree
CH2S (O) CH2C (O) OMe CH2C (O) OMe
CH2S (O)2CH2C (O) OMe Me
CH2S (O)2CH2C (O) OEt Me
CH2S (O)2CH2C (O) OPr-n Me
CH2S (O)2CH2C (O) OPr-i Me
CH2S (O)2CH2C (O) OBu-n Me
CH2S (O)2CH2C (O) OBu-i Me
CH2S (O)2CH2C (O) OBu-t Me
CH2S (O)2CH2C (O) OPen-n Me
CH2S (O)2CH2C (O) OHex-n Me
CH2S (O)2CH2C (O) OMe Et
CH2S (O)2CH2C (O) OMe Pr-n
CH2S (O)2CH2C (O) OMe Pr-i
CH2S (O)2CH2C (O) OMe Pr-c
CH2S (O)2CH2C (O) OMe Bu-n
CH2S (O)2CH2C (O) OMe Bu-i
CH2S (O)2CH2C (O) OMe Bu-c
CH2S (O)2CH2C (O) OMe Bu-s
CH2S (O)2CH2C (O) OMe Bu-t
CH2S (O)2CH2C (O) OMe Pen-n
CH2S (O)2CH2C (O) OMe Pen-c
CH2S (O)2CH2C (O) OMe Hex-n
CH2S (O)2CH2C (O) OMe Hex-c
CH2S (O)2CH2C (O) OMe CH2Pr-c
CH2S (O)2CH2C (O) OMe CH2Bu-c
CH2S (O)2CH2C (O) OMe CH2Pen-c
CH2S (O)2CH2C (O) OMe CH2Hex-c
CH2S (O)2CH2C (O) OMe CH2CH = CH2
CH2S (O)2CH2C (O) OMe CH2CH = C (Cl)2
CH2S (O)2CH2C (O) OMe CH2C≡CH
CH2S (O)2CH2C (O) OMe CH2CN
CH2S (O)2CH2C (O) OMe CH2CFThree
CH2S (O)2CH2C (O) OMe CH2OMe
CH2S (O)2CH2C (O) OMe CH2OCFThree
CH2S (O)2CH2C (O) OMe CH2SMe
CH2S (O)2CH2C (O) OMe CH2S (O) Me
CH2S (O)2CH2C (O) OMe CH2S (O)2Me
CH2S (O)2CH2C (O) OMe CH2SCFThree
CH2S (O)2CH2C (O) OMe CH2S (O) CFThree
CH2S (O)2CH2C (O) OMe CH2S (O)2CFThree
CH2S (O)2CH2C (O) OMe CH2CH (OMe)2
CH2S (O)2CH2C (O) OMe CH2CH (SMe)2
CH2S (O)2CH2C (O) OMe CH2C (O) Me
CH2S (O)2CH2C (O) OMe CH2C (O) CFThree
CH2S (O)2CH2C (O) OMe CH2C (O) OMe
CH (Me) SCH2C (O) OMe Me
CH (Me) SCH2C (O) OEt Me
CH (Me) SCH2C (O) OPr-n Me
CH (Me) SCH2C (O) OPr-i Me
CH (Me) SCH2C (O) OBu-n Me
CH (Me) SCH2C (O) OBu-i Me
CH (Me) SCH2C (O) OBu-t Me
CH (Me) SCH2C (O) OPen-n Me
CH (Me) SCH2C (O) OHex-n Me
CH (Me) SCH2C (O) OMe Et
CH (Me) SCH2C (O) OMe Pr-n
CH (Me) SCH2C (O) OMe Pr-i
CH (Me) SCH2C (O) OMe Pr-c
CH (Me) SCH2C (O) OMe Bu-n
CH (Me) SCH2C (O) OMe Bu-i
CH (Me) SCH2C (O) OMe Bu-c
CH (Me) SCH2C (O) OMe Bu-s
CH (Me) SCH2C (O) OMe Bu-t
CH (Me) SCH2C (O) OMe Pen-n
CH (Me) SCH2C (O) OMe Pen-c
CH (Me) SCH2C (O) OMe Hex-n
CH (Me) SCH2C (O) OMe Hex-c
CH (Me) SCH2C (O) OMe CH2Pr-c
CH (Me) SCH2C (O) OMe CH2Bu-c
CH (Me) SCH2C (O) OMe CH2Pen-c
CH (Me) SCH2C (O) OMe CH2Hex-c
CH (Me) SCH2C (O) OMe CH2CH = CH2
CH (Me) SCH2C (O) OMe CH2CH = C (Cl)2
CH (Me) SCH2C (O) OMe CH2C≡CH
CH (Me) SCH2C (O) OMe CH2CN
CH (Me) SCH2C (O) OMe CH2CFThree
CH (Me) SCH2C (O) OMe CH2OMe
CH (Me) SCH2C (O) OMe CH2OCFThree
CH (Me) SCH2C (O) OMe CH2SMe
CH (Me) SCH2C (O) OMe CH2S (O) Me
CH (Me) SCH2C (O) OMe CH2S (O)2Me
CH (Me) SCH2C (O) OMe CH2SCFThree
CH (Me) SCH2C (O) OMe CH2S (O) CFThree
CH (Me) SCH2C (O) OMe CH2S (O)2CFThree
CH (Me) SCH2C (O) OMe CH2CH (OMe)2
CH (Me) SCH2C (O) OMe CH2CH (SMe)2
CH (Me) SCH2C (O) OMe CH2C (O) Me
CH (Me) SCH2C (O) OMe CH2C (O) CFThree
CH (Me) SCH2C (O) OMe CH2C (O) OMe
CH (Me) S (O) CH2C (O) OMe Me
CH (Me) S (O) CH2C (O) OEt Me
CH (Me) S (O) CH2C (O) OPr-n Me
CH (Me) S (O) CH2C (O) OPr-i Me
CH (Me) S (O) CH2C (O) OBu-n Me
CH (Me) S (O) CH2C (O) OBu-i Me
CH (Me) S (O) CH2C (O) OBu-t Me
CH (Me) S (O) CH2C (O) OPen-n Me
CH (Me) S (O) CH2C (O) OHex-n Me
CH (Me) S (O) CH2C (O) OMe Et
CH (Me) S (O) CH2C (O) OMe Pr-n
CH (Me) S (O) CH2C (O) OMe Pr-i
CH (Me) S (O) CH2C (O) OMe Pr-c
CH (Me) S (O) CH2C (O) OMe Bu-n
CH (Me) S (O) CH2C (O) OMe Bu-i
CH (Me) S (O) CH2C (O) OMe Bu-c
CH (Me) S (O) CH2C (O) OMe Bu-s
CH (Me) S (O) CH2C (O) OMe Bu-t
CH (Me) S (O) CH2C (O) OMe Pen-n
CH (Me) S (O) CH2C (O) OMe Pen-c
CH (Me) S (O) CH2C (O) OMe Hex-n
CH (Me) S (O) CH2C (O) OMe Hex-c
CH (Me) S (O) CH2C (O) OMe CH2Pr-c
CH (Me) S (O) CH2C (O) OMe CH2Bu-c
CH (Me) S (O) CH2C (O) OMe CH2Pen-c
CH (Me) S (O) CH2C (O) OMe CH2Hex-c
CH (Me) S (O) CH2C (O) OMe CH2CH = CH2
CH (Me) S (O) CH2C (O) OMe CH2CH = C (Cl)2
CH (Me) S (O) CH2C (O) OMe CH2C≡CH
CH (Me) S (O) CH2C (O) OMe CH2CN
CH (Me) S (O) CH2C (O) OMe CH2CFThree
CH (Me) S (O) CH2C (O) OMe CH2OMe
CH (Me) S (O) CH2C (O) OMe CH2OCFThree
CH (Me) S (O) CH2C (O) OMe CH2SMe
CH (Me) S (O) CH2C (O) OMe CH2S (O) Me
CH (Me) S (O) CH2C (O) OMe CH2S (O)2Me
CH (Me) S (O) CH2C (O) OMe CH2SCFThree
CH (Me) S (O) CH2C (O) OMe CH2S (O) CFThree
CH (Me) S (O) CH2C (O) OMe CH2S (O)2CFThree
CH (Me) S (O) CH2C (O) OMe CH2CH (OMe)2
CH (Me) S (O) CH2C (O) OMe CH2CH (SMe)2
CH (Me) S (O) CH2C (O) OMe CH2C (O) Me
CH (Me) S (O) CH2C (O) OMe CH2C (O) CFThree
CH (Me) S (O) CH2C (O) OMe CH2C (O) OMe
CH (Me) S (O)2CH2C (O) OMe Me
CH (Me) S (O)2CH2C (O) OEt Me
CH (Me) S (O)2CH2C (O) OPr-n Me
CH (Me) S (O)2CH2C (O) OPr-i Me
CH (Me) S (O)2CH2C (O) OBu-n Me
CH (Me) S (O)2CH2C (O) OBu-i Me
CH (Me) S (O)2CH2C (O) OBu-t Me
CH (Me) S (O)2CH2C (O) OPen-n Me
CH (Me) S (O)2CH2C (O) OHex-n Me
CH (Me) S (O)2CH2C (O) OMe Et
CH (Me) S (O)2CH2C (O) OMe Pr-n
CH (Me) S (O)2CH2C (O) OMe Pr-i
CH (Me) S (O)2CH2C (O) OMe Pr-c
CH (Me) S (O)2CH2C (O) OMe Bu-n
CH (Me) S (O)2CH2C (O) OMe Bu-i
CH (Me) S (O)2CH2C (O) OMe Bu-c
CH (Me) S (O)2CH2C (O) OMe Bu-s
CH (Me) S (O)2CH2C (O) OMe Bu-t
CH (Me) S (O)2CH2C (O) OMe Pen-n
CH (Me) S (O)2CH2C (O) OMe Pen-c
CH (Me) S (O)2CH2C (O) OMe Hex-n
CH (Me) S (O)2CH2C (O) OMe Hex-c
CH (Me) S (O)2CH2C (O) OMe CH2Pr-c
CH (Me) S (O)2CH2C (O) OMe CH2Bu-c
CH (Me) S (O)2CH2C (O) OMe CH2Pen-c
CH (Me) S (O)2CH2C (O) OMe CH2Hex-c
CH (Me) S (O)2CH2C (O) OMe CH2CH = CH2
CH (Me) S (O)2CH2C (O) OMe CH2CH = C (Cl)2
CH (Me) S (O)2CH2C (O) OMe CH2C≡CH
CH (Me) S (O)2CH2C (O) OMe CH2CN
CH (Me) S (O)2CH2C (O) OMe CH2CFThree
CH (Me) S (O)2CH2C (O) OMe CH2OMe
CH (Me) S (O)2CH2C (O) OMe CH2OCFThree
CH (Me) S (O)2CH2C (O) OMe CH2SMe
CH (Me) S (O)2CH2C (O) OMe CH2S (O) Me
CH (Me) S (O)2CH2C (O) OMe CH2S (O)2Me
CH (Me) S (O)2CH2C (O) OMe CH2SCFThree
CH (Me) S (O)2CH2C (O) OMe CH2S (O) CFThree
CH (Me) S (O)2CH2C (O) OMe CH2S (O)2CFThree
CH (Me) S (O)2CH2C (O) OMe CH2CH (OMe)2
CH (Me) S (O)2CH2C (O) OMe CH2CH (SMe)2
CH (Me) S (O)2CH2C (O) OMe CH2C (O) Me
CH (Me) S (O)2CH2C (O) OMe CH2C (O) CFThree
CH (Me) S (O)2CH2C (O) OMe CH2C (O) OMe
CH (Et) SCH2C (O) OMe Me
CH (Et) SCH2C (O) OEt Me
CH (Et) SCH2C (O) OPr-n Me
CH (Et) SCH2C (O) OPr-i Me
CH (Et) SCH2C (O) OBu-n Me
CH (Et) SCH2C (O) OBu-i Me
CH (Et) SCH2C (O) OBu-t Me
CH (Et) SCH2C (O) OPen-n Me
CH (Et) SCH2C (O) OHex-n Me
CH (Et) SCH2C (O) OMe Et
CH (Et) SCH2C (O) OMe Pr-n
CH (Et) SCH2C (O) OMe Pr-i
CH (Et) SCH2C (O) OMe Pr-c
CH (Et) SCH2C (O) OMe Bu-n
CH (Et) SCH2C (O) OMe Bu-i
CH (Et) SCH2C (O) OMe Bu-c
CH (Et) SCH2C (O) OMe Bu-s
CH (Et) SCH2C (O) OMe Bu-t
CH (Et) SCH2C (O) OMe Pen-n
CH (Et) SCH2C (O) OMe Pen-c
CH (Et) SCH2C (O) OMe Hex-n
CH (Et) SCH2C (O) OMe Hex-c
CH (Et) SCH2C (O) OMe CH2Pr-c
CH (Et) SCH2C (O) OMe CH2Bu-c
CH (Et) SCH2C (O) OMe CH2Pen-c
CH (Et) SCH2C (O) OMe CH2Hex-c
CH (Et) SCH2C (O) OMe CH2CH = CH2
CH (Et) SCH2C (O) OMe CH2CH = C (Cl)2
CH (Et) SCH2C (O) OMe CH2C≡CH
CH (Et) SCH2C (O) OMe CH2CN
CH (Et) SCH2C (O) OMe CH2CFThree
CH (Et) SCH2C (O) OMe CH2OMe
CH (Et) SCH2C (O) OMe CH2OCFThree
CH (Et) SCH2C (O) OMe CH2SMe
CH (Et) SCH2C (O) OMe CH2S (O) Me
CH (Et) SCH2C (O) OMe CH2S (O)2Me
CH (Et) SCH2C (O) OMe CH2SCFThree
CH (Et) SCH2C (O) OMe CH2S (O) CFThree
CH (Et) SCH2C (O) OMe CH2S (O)2CFThree
CH (Et) SCH2C (O) OMe CH2CH (OMe)2
CH (Et) SCH2C (O) OMe CH2CH (SMe)2
CH (Et) SCH2C (O) OMe CH2C (O) Me
CH (Et) SCH2C (O) OMe CH2C (O) CFThree
CH (Et) SCH2C (O) OMe CH2C (O) OMe
CH (Et) S (O) CH2C (O) OMe Me
CH (Et) S (O) CH2C (O) OEt Me
CH (Et) S (O) CH2C (O) OPr-n Me
CH (Et) S (O) CH2C (O) OPr-i Me
CH (Et) S (O) CH2C (O) OBu-n Me
CH (Et) S (O) CH2C (O) OBu-i Me
CH (Et) S (O) CH2C (O) OBu-t Me
CH (Et) S (O) CH2C (O) OPen-n Me
CH (Et) S (O) CH2C (O) OHex-n Me
CH (Et) S (O) CH2C (O) OMe Et
CH (Et) S (O) CH2C (O) OMe Pr-n
CH (Et) S (O) CH2C (O) OMe Pr-i
CH (Et) S (O) CH2C (O) OMe Pr-c
CH (Et) S (O) CH2C (O) OMe Bu-n
CH (Et) S (O) CH2C (O) OMe Bu-i
CH (Et) S (O) CH2C (O) OMe Bu-c
CH (Et) S (O) CH2C (O) OMe Bu-s
CH (Et) S (O) CH2C (O) OMe Bu-t
CH (Et) S (O) CH2C (O) OMe Pen-n
CH (Et) S (O) CH2C (O) OMe Pen-c
CH (Et) S (O) CH2C (O) OMe Hex-n
CH (Et) S (O) CH2C (O) OMe Hex-c
CH (Et) S (O) CH2C (O) OMe CH2Pr-c
CH (Et) S (O) CH2C (O) OMe CH2Bu-c
CH (Et) S (O) CH2C (O) OMe CH2Pen-c
CH (Et) S (O) CH2C (O) OMe CH2Hex-c
CH (Et) S (O) CH2C (O) OMe CH2CH = CH2
CH (Et) S (O) CH2C (O) OMe CH2CH = C (Cl)2
CH (Et) S (O) CH2C (O) OMe CH2C≡CH
CH (Et) S (O) CH2C (O) OMe CH2CN
CH (Et) S (O) CH2C (O) OMe CH2CFThree
CH (Et) S (O) CH2C (O) OMe CH2OMe
CH (Et) S (O) CH2C (O) OMe CH2OCFThree
CH (Et) S (O) CH2C (O) OMe CH2SMe
CH (Et) S (O) CH2C (O) OMe CH2S (O) Me
CH (Et) S (O) CH2C (O) OMe CH2S (O)2Me
CH (Et) S (O) CH2C (O) OMe CH2SCFThree
CH (Et) S (O) CH2C (O) OMe CH2S (O) CFThree
CH (Et) S (O) CH2C (O) OMe CH2S (O)2CFThree
CH (Et) S (O) CH2C (O) OMe CH2CH (OMe)2
CH (Et) S (O) CH2C (O) OMe CH2CH (SMe)2
CH (Et) S (O) CH2C (O) OMe CH2C (O) Me
CH (Et) S (O) CH2C (O) OMe CH2C (O) CFThree
CH (Et) S (O) CH2C (O) OMe CH2C (O) OMe
CH (Et) S (O)2CH2C (O) OMe Me
CH (Et) S (O)2CH2C (O) OEt Me
CH (Et) S (O)2CH2C (O) OPr-n Me
CH (Et) S (O)2CH2C (O) OPr-i Me
CH (Et) S (O)2CH2C (O) OBu-n Me
CH (Et) S (O)2CH2C (O) OBu-i Me
CH (Et) S (O)2CH2C (O) OBu-t Me
CH (Et) S (O)2CH2C (O) OPen-n Me
CH (Et) S (O)2CH2C (O) OHex-n Me
CH (Et) S (O)2CH2C (O) OMe Et
CH (Et) S (O)2CH2C (O) OMe Pr-n
CH (Et) S (O)2CH2C (O) OMe Pr-i
CH (Et) S (O)2CH2C (O) OMe Pr-c
CH (Et) S (O)2CH2C (O) OMe Bu-n
CH (Et) S (O)2CH2C (O) OMe Bu-i
CH (Et) S (O)2CH2C (O) OMe Bu-c
CH (Et) S (O)2CH2C (O) OMe Bu-s
CH (Et) S (O)2CH2C (O) OMe Bu-t
CH (Et) S (O)2CH2C (O) OMe Pen-n
CH (Et) S (O)2CH2C (O) OMe Pen-c
CH (Et) S (O)2CH2C (O) OMe Hex-n
CH (Et) S (O)2CH2C (O) OMe Hex-c
CH (Et) S (O)2CH2C (O) OMe CH2Pr-c
CH (Et) S (O)2CH2C (O) OMe CH2Bu-c
CH (Et) S (O)2CH2C (O) OMe CH2Pen-c
CH (Et) S (O)2CH2C (O) OMe CH2Hex-c
CH (Et) S (O)2CH2C (O) OMe CH2CH = CH2
CH (Et) S (O)2CH2C (O) OMe CH2CH = C (Cl)2
CH (Et) S (O)2CH2C (O) OMe CH2C≡CH
CH (Et) S (O)2CH2C (O) OMe CH2CN
CH (Et) S (O)2CH2C (O) OMe CH2CFThree
CH (Et) S (O)2CH2C (O) OMe CH2OMe
CH (Et) S (O)2CH2C (O) OMe CH2OCFThree
CH (Et) S (O)2CH2C (O) OMe CH2SMe
CH (Et) S (O)2CH2C (O) OMe CH2S (O) Me
CH (Et) S (O)2CH2C (O) OMe CH2S (O)2Me
CH (Et) S (O)2CH2C (O) OMe CH2SCFThree
CH (Et) S (O)2CH2C (O) OMe CH2S (O) CFThree
CH (Et) S (O)2CH2C (O) OMe CH2S (O)2CFThree
CH (Et) S (O)2CH2C (O) OMe CH2CH (OMe)2
CH (Et) S (O)2CH2C (O) OMe CH2CH (SMe)2
CH (Et) S (O)2CH2C (O) OMe CH2C (O) Me
CH (Et) S (O)2CH2C (O) OMe CH2C (O) CFThree
CH (Et) S (O)2CH2C (O) OMe CH2C (O) OMe
CH2SCH2C (O) Me Me
CH2SCH2C (O) Et Me
CH2SCH2C (O) Pr-n Me
CH2SCH2C (O) Pr-i Me
CH2SCH2C (O) Pr-c Me
CH2SCH2C (O) Bu-n Me
CH2SCH2C (O) Bu-i Me
CH2SCH2C (O) Bu-c Me
CH2SCH2C (O) Bu-t Me
CH2SCH2C (O) Pen-n Me
CH2SCH2C (O) Pen-c Me
CH2SCH2C (O) Hex-n Me
CH2SCH2C (O) Hex-c Me
CH2SCH2C (O) Me Et
CH2SCH2C (O) Me Pr-n
CH2SCH2C (O) Me Pr-i
CH2SCH2C (O) Me Pr-c
CH2SCH2C (O) Me Bu-n
CH2SCH2C (O) Me Bu-i
CH2SCH2C (O) Me Bu-c
CH2SCH2C (O) Me Bu-s
CH2SCH2C (O) Me Bu-t
CH2SCH2C (O) Me Pen-n
CH2SCH2C (O) Me Pen-c
CH2SCH2C (O) Me Hex-n
CH2SCH2C (O) Me Hex-c
CH2SCH2C (O) Me CH2Pr-c
CH2SCH2C (O) Me CH2Bu-c
CH2SCH2C (O) Me CH2Pen-c
CH2SCH2C (O) Me CH2Hex-c
CH2SCH2C (O) Me CH2CH = CH2
CH2SCH2C (O) Me CH2CH = C (Cl)2
CH2SCH2C (O) Me CH2C≡CH
CH2SCH2C (O) Me CH2CN
CH2SCH2C (O) Me CH2CFThree
CH2SCH2C (O) Me CH2OMe
CH2SCH2C (O) Me CH2OCFThree
CH2SCH2C (O) Me CH2SMe
CH2SCH2C (O) Me CH2S (O) Me
CH2SCH2C (O) Me CH2S (O)2Me
CH2SCH2C (O) Me CH2SCFThree
CH2SCH2C (O) Me CH2S (O) CFThree
CH2SCH2C (O) Me CH2S (O)2CFThree
CH2SCH2C (O) Me CH2CH (OMe)2
CH2SCH2C (O) Me CH2CH (SMe)2
CH2SCH2C (O) Me CH2C (O) Me
CH2SCH2C (O) Me CH2C (O) CFThree
CH2SCH2C (O) Me CH2C (O) OMe
CH2S (O) CH2C (O) Me Me
CH2S (O) CH2C (O) Et Me
CH2S (O) CH2C (O) Pr-n Me
CH2S (O) CH2C (O) Pr-i Me
CH2S (O) CH2C (O) Pr-c Me
CH2S (O) CH2C (O) Bu-n Me
CH2S (O) CH2C (O) Bu-i Me
CH2S (O) CH2C (O) Bu-c Me
CH2S (O) CH2C (O) Bu-t Me
CH2S (O) CH2C (O) Pen-n Me
CH2S (O) CH2C (O) Pen-c Me
CH2S (O) CH2C (O) Hex-n Me
CH2S (O) CH2C (O) Hex-c Me
CH2S (O) CH2C (O) Me Et
CH2S (O) CH2C (O) Me Pr-n
CH2S (O) CH2C (O) Me Pr-i
CH2S (O) CH2C (O) Me Pr-c
CH2S (O) CH2C (O) Me Bu-n
CH2S (O) CH2C (O) Me Bu-i
CH2S (O) CH2C (O) Me Bu-c
CH2S (O) CH2C (O) Me Bu-s
CH2S (O) CH2C (O) Me Bu-t
CH2S (O) CH2C (O) Me Pen-n
CH2S (O) CH2C (O) Me Pen-c
CH2S (O) CH2C (O) Me Hex-n
CH2S (O) CH2C (O) Me Hex-c
CH2S (O) CH2C (O) Me CH2Pr-c
CH2S (O) CH2C (O) Me CH2Bu-c
CH2S (O) CH2C (O) Me CH2Pen-c
CH2S (O) CH2C (O) Me CH2Hex-c
CH2S (O) CH2C (O) Me CH2CH = CH2
CH2S (O) CH2C (O) Me CH2CH = C (Cl)2
CH2S (O) CH2C (O) Me CH2C≡CH
CH2S (O) CH2C (O) Me CH2CN
CH2S (O) CH2C (O) Me CH2CFThree
CH2S (O) CH2C (O) Me CH2OMe
CH2S (O) CH2C (O) Me CH2OCFThree
CH2S (O) CH2C (O) Me CH2SMe
CH2S (O) CH2C (O) Me CH2S (O) Me
CH2S (O) CH2C (O) Me CH2S (O)2Me
CH2S (O) CH2C (O) Me CH2SCFThree
CH2S (O) CH2C (O) Me CH2S (O) CFThree
CH2S (O) CH2C (O) Me CH2S (O)2CFThree
CH2S (O) CH2C (O) Me CH2CH (OMe)2
CH2S (O) CH2C (O) Me CH2CH (SMe)2
CH2S (O) CH2C (O) Me CH2C (O) Me
CH2S (O) CH2C (O) Me CH2C (O) CFThree
CH2S (O) CH2C (O) Me CH2C (O) OMe
CH2S (O)2CH2C (O) Me Me
CH2S (O)2CH2C (O) Et Me
CH2S (O)2CH2C (O) Pr-n Me
CH2S (O)2CH2C (O) Pr-i Me
CH2S (O)2CH2C (O) Pr-c Me
CH2S (O)2CH2C (O) Bu-n Me
CH2S (O)2CH2C (O) Bu-i Me
CH2S (O)2CH2C (O) Bu-c Me
CH2S (O)2CH2C (O) Bu-t Me
CH2S (O)2CH2C (O) Pen-n Me
CH2S (O)2CH2C (O) Pen-c Me
CH2S (O)2CH2C (O) Hex-n Me
CH2S (O)2CH2C (O) Hex-c Me
CH2S (O)2CH2C (O) Me Et
CH2S (O)2CH2C (O) Me Pr-n
CH2S (O)2CH2C (O) Me Pr-i
CH2S (O)2CH2C (O) Me Pr-c
CH2S (O)2CH2C (O) Me Bu-n
CH2S (O)2CH2C (O) Me Bu-i
CH2S (O)2CH2C (O) Me Bu-c
CH2S (O)2CH2C (O) Me Bu-s
CH2S (O)2CH2C (O) Me Bu-t
CH2S (O)2CH2C (O) Me Pen-n
CH2S (O)2CH2C (O) Me Pen-c
CH2S (O)2CH2C (O) Me Hex-n
CH2S (O)2CH2C (O) Me Hex-c
CH2S (O)2CH2C (O) Me CH2Pr-c
CH2S (O)2CH2C (O) Me CH2Bu-c
CH2S (O)2CH2C (O) Me CH2Pen-c
CH2S (O)2CH2C (O) Me CH2Hex-c
CH2S (O)2CH2C (O) Me CH2CH = CH2
CH2S (O)2CH2C (O) Me CH2CH = C (Cl)2
CH2S (O)2CH2C (O) Me CH2C≡CH
CH2S (O)2CH2C (O) Me CH2CN
CH2S (O)2CH2C (O) Me CH2CFThree
CH2S (O)2CH2C (O) Me CH2OMe
CH2S (O)2CH2C (O) Me CH2OCFThree
CH2S (O)2CH2C (O) Me CH2SMe
CH2S (O)2CH2C (O) Me CH2S (O) Me
CH2S (O)2CH2C (O) Me CH2S (O)2Me
CH2S (O)2CH2C (O) Me CH2SCFThree
CH2S (O)2CH2C (O) Me CH2S (O) CFThree
CH2S (O)2CH2C (O) Me CH2S (O)2CFThree
CH2S (O)2CH2C (O) Me CH2CH (OMe)2
CH2S (O)2CH2C (O) Me CH2CH (SMe)2
CH2S (O)2CH2C (O) Me CH2C (O) Me
CH2S (O)2CH2C (O) Me CH2C (O) CFThree
CH2S (O)2CH2C (O) Me CH2C (O) OMe
CH (Me) SCH2C (O) Me Me
CH (Me) SCH2C (O) Et Me
CH (Me) SCH2C (O) Pr-n Me
CH (Me) SCH2C (O) Pr-i Me
CH (Me) SCH2C (O) Pr-c Me
CH (Me) SCH2C (O) Bu-n Me
CH (Me) SCH2C (O) Bu-i Me
CH (Me) SCH2C (O) Bu-c Me
CH (Me) SCH2C (O) Bu-t Me
CH (Me) SCH2C (O) Pen-n Me
CH (Me) SCH2C (O) Pen-c Me
CH (Me) SCH2C (O) Hex-n Me
CH (Me) SCH2C (O) Hex-c Me
CH (Me) SCH2C (O) Me Et
CH (Me) SCH2C (O) Me Pr-n
CH (Me) SCH2C (O) Me Pr-i
CH (Me) SCH2C (O) Me Pr-c
CH (Me) SCH2C (O) Me Bu-n
CH (Me) SCH2C (O) Me Bu-i
CH (Me) SCH2C (O) Me Bu-c
CH (Me) SCH2C (O) Me Bu-s
CH (Me) SCH2C (O) Me Bu-t
CH (Me) SCH2C (O) Me Pen-n
CH (Me) SCH2C (O) Me Pen-c
CH (Me) SCH2C (O) Me Hex-n
CH (Me) SCH2C (O) Me Hex-c
CH (Me) SCH2C (O) Me CH2Pr-c
CH (Me) SCH2C (O) Me CH2Bu-c
CH (Me) SCH2C (O) Me CH2Pen-c
CH (Me) SCH2C (O) Me CH2Hex-c
CH (Me) SCH2C (O) Me CH2CH = CH2
CH (Me) SCH2C (O) Me CH2CH = C (Cl)2
CH (Me) SCH2C (O) Me CH2C≡CH
CH (Me) SCH2C (O) Me CH2CN
CH (Me) SCH2C (O) Me CH2CFThree
CH (Me) SCH2C (O) Me CH2OMe
CH (Me) SCH2C (O) Me CH2OCFThree
CH (Me) SCH2C (O) Me CH2SMe
CH (Me) SCH2C (O) Me CH2S (O) Me
CH (Me) SCH2C (O) Me CH2S (O)2Me
CH (Me) SCH2C (O) Me CH2SCFThree
CH (Me) SCH2C (O) Me CH2S (O) CFThree
CH (Me) SCH2C (O) Me CH2S (O)2CFThree
CH (Me) SCH2C (O) Me CH2CH (OMe)2
CH (Me) SCH2C (O) Me CH2CH (SMe)2
CH (Me) SCH2C (O) Me CH2C (O) Me
CH (Me) SCH2C (O) Me CH2C (O) CFThree
CH (Me) SCH2C (O) Me CH2C (O) OMe
CH (Me) S (O) CH2C (O) Me Me
CH (Me) S (O) CH2C (O) Et Me
CH (Me) S (O) CH2C (O) Pr-n Me
CH (Me) S (O) CH2C (O) Pr-i Me
CH (Me) S (O) CH2C (O) Pr-c Me
CH (Me) S (O) CH2C (O) Bu-n Me
CH (Me) S (O) CH2C (O) Bu-i Me
CH (Me) S (O) CH2C (O) Bu-t Me
CH (Me) S (O) CH2C (O) Pen-n Me
CH (Me) S (O) CH2C (O) Pen-c Me
CH (Me) S (O) CH2C (O) Hex-n Me
CH (Me) S (O) CH2C (O) Hex-c Me
CH (Me) S (O) CH2C (O) Me Et
CH (Me) S (O) CH2C (O) Me Pr-n
CH (Me) S (O) CH2C (O) Me Pr-i
CH (Me) S (O) CH2C (O) Me Pr-c
CH (Me) S (O) CH2C (O) Me Bu-n
CH (Me) S (O) CH2C (O) Me Bu-i
CH (Me) S (O) CH2C (O) Me Bu-c
CH (Me) S (O) CH2C (O) Me Bu-s
CH (Me) S (O) CH2C (O) Me Bu-t
CH (Me) S (O) CH2C (O) Me Pen-n
CH (Me) S (O) CH2C (O) Me Pen-c
CH (Me) S (O) CH2C (O) Me Hex-n
CH (Me) S (O) CH2C (O) Me Hex-c
CH (Me) S (O) CH2C (O) Me CH2Pr-c
CH (Me) S (O) CH2C (O) Me CH2Bu-c
CH (Me) S (O) CH2C (O) Me CH2Pen-c
CH (Me) S (O) CH2C (O) Me CH2Hex-c
CH (Me) S (O) CH2C (O) Me CH2CH = CH2
CH (Me) S (O) CH2C (O) Me CH2CH = C (Cl)2
CH (Me) S (O) CH2C (O) Me CH2C≡CH
CH (Me) S (O) CH2C (O) Me CH2CN
CH (Me) S (O) CH2C (O) Me CH2CFThree
CH (Me) S (O) CH2C (O) Me CH2OMe
CH (Me) S (O) CH2C (O) Me CH2OCFThree
CH (Me) S (O) CH2C (O) Me CH2SMe
CH (Me) S (O) CH2C (O) Me CH2S (O) Me
CH (Me) S (O) CH2C (O) Me CH2S (O)2Me
CH (Me) S (O) CH2C (O) Me CH2SCFThree
CH (Me) S (O) CH2C (O) Me CH2S (O) CFThree
CH (Me) S (O) CH2C (O) Me CH2S (O)2CFThree
CH (Me) S (O) CH2C (O) Me CH2CH (OMe)2
CH (Me) S (O) CH2C (O) Me CH2CH (SMe)2
CH (Me) S (O) CH2C (O) Me CH2C (O) Me
CH (Me) S (O) CH2C (O) Me CH2C (O) CFThree
CH (Me) S (O) CH2C (O) Me CH2C (O) OMe
CH (Me) S (O)2CH2C (O) Me Me
CH (Me) S (O)2CH2C (O) Et Me
CH (Me) S (O)2CH2C (O) Pr-n Me
CH (Me) S (O)2CH2C (O) Pr-i Me
CH (Me) S (O)2CH2C (O) Pr-c Me
CH (Me) S (O)2CH2C (O) Bu-n Me
CH (Me) S (O)2CH2C (O) Bu-i Me
CH (Me) S (O)2CH2C (O) Bu-t Me
CH (Me) S (O)2CH2C (O) Pen-n Me
CH (Me) S (O)2CH2C (O) Pen-c Me
CH (Me) S (O)2CH2C (O) Hex-n Me
CH (Me) S (O)2CH2C (O) Hex-c Me
CH (Me) S (O)2CH2C (O) Me Et
CH (Me) S (O)2CH2C (O) Me Pr-n
CH (Me) S (O)2CH2C (O) Me Pr-i
CH (Me) S (O)2CH2C (O) Me Pr-c
CH (Me) S (O)2CH2C (O) Me Bu-n
CH (Me) S (O)2CH2C (O) Me Bu-i
CH (Me) S (O)2CH2C (O) Me Bu-c
CH (Me) S (O)2CH2C (O) Me Bu-s
CH (Me) S (O)2CH2C (O) Me Bu-t
CH (Me) S (O)2CH2C (O) Me Pen-n
CH (Me) S (O)2CH2C (O) Me Pen-c
CH (Me) S (O)2CH2C (O) Me Hex-n
CH (Me) S (O)2CH2C (O) Me Hex-c
CH (Me) S (O)2CH2C (O) Me CH2Pr-c
CH (Me) S (O)2CH2C (O) Me CH2Bu-c
CH (Me) S (O)2CH2C (O) Me CH2Pen-c
CH (Me) S (O)2CH2C (O) Me CH2Hex-c
CH (Me) S (O)2CH2C (O) Me CH2CH = CH2
CH (Me) S (O)2CH2C (O) Me CH2CH = C (Cl)2
CH (Me) S (O)2CH2C (O) Me CH2C≡CH
CH (Me) S (O)2CH2C (O) Me CH2CN
CH (Me) S (O)2CH2C (O) Me CH2CFThree
CH (Me) S (O)2CH2C (O) Me CH2OMe
CH (Me) S (O)2CH2C (O) Me CH2OCFThree
CH (Me) S (O)2CH2C (O) Me CH2SMe
CH (Me) S (O)2CH2C (O) Me CH2S (O) Me
CH (Me) S (O)2CH2C (O) Me CH2S (O)2Me
CH (Me) S (O)2CH2C (O) Me CH2SCFThree
CH (Me) S (O)2CH2C (O) Me CH2S (O) CFThree
CH (Me) S (O)2CH2C (O) Me CH2S (O)2CFThree
CH (Me) S (O)2CH2C (O) Me CH2CH (OMe)2
CH (Me) S (O)2CH2C (O) Me CH2CH (SMe)2
CH (Me) S (O)2CH2C (O) Me CH2C (O) Me
CH (Me) S (O)2CH2C (O) Me CH2C (O) CFThree
CH (Me) S (O)2CH2C (O) Me CH2C (O) OMe
CH (Et) SCH2C (O) Me Me
CH (Et) SCH2C (O) Et Me
CH (Et) SCH2C (O) Pr-n Me
CH (Et) SCH2C (O) Pr-i Me
CH (Et) SCH2C (O) Pr-c Me
CH (Et) SCH2C (O) Bu-n Me
CH (Et) SCH2C (O) Bu-i Me
CH (Et) SCH2C (O) Bu-c Me
CH (Et) SCH2C (O) Bu-t Me
CH (Et) SCH2C (O) Pen-n Me
CH (Et) SCH2C (O) Pen-c Me
CH (Et) SCH2C (O) Hex-n Me
CH (Et) SCH2C (O) Hex-c Me
CH (Et) SCH2C (O) Me Et
CH (Et) SCH2C (O) Me Pr-n
CH (Et) SCH2C (O) Me Pr-i
CH (Et) SCH2C (O) Me Pr-c
CH (Et) SCH2C (O) Me Bu-n
CH (Et) SCH2C (O) Me Bu-i
CH (Et) SCH2C (O) Me Bu-c
CH (Et) SCH2C (O) Me Bu-s
CH (Et) SCH2C (O) Me Bu-t
CH (Et) SCH2C (O) Me Pen-n
CH (Et) SCH2C (O) Me Pen-c
CH (Et) SCH2C (O) Me Hex-n
CH (Et) SCH2C (O) Me Hex-c
CH (Et) SCH2C (O) Me CH2Pr-c
CH (Et) SCH2C (O) Me CH2Bu-c
CH (Et) SCH2C (O) Me CH2Pen-c
CH (Et) SCH2C (O) Me CH2Hex-c
CH (Et) SCH2C (O) Me CH2CH = CH2
CH (Et) SCH2C (O) Me CH2CH = C (Cl)2
CH (Et) SCH2C (O) Me CH2C≡CH
CH (Et) SCH2C (O) Me CH2CN
CH (Et) SCH2C (O) Me CH2CFThree
CH (Et) SCH2C (O) Me CH2OMe
CH (Et) SCH2C (O) Me CH2OCFThree
CH (Et) SCH2C (O) Me CH2SMe
CH (Et) SCH2C (O) Me CH2S (O) Me
CH (Et) SCH2C (O) Me CH2S (O)2Me
CH (Et) SCH2C (O) Me CH2SCFThree
CH (Et) SCH2C (O) Me CH2S (O) CFThree
CH (Et) SCH2C (O) Me CH2S (O)2CFThree
CH (Et) SCH2C (O) Me CH2CH (OMe)2
CH (Et) SCH2C (O) Me CH2CH (SMe)2
CH (Et) SCH2C (O) Me CH2C (O) Me
CH (Et) SCH2C (O) Me CH2C (O) CFThree
CH (Et) SCH2C (O) Me CH2C (O) OMe
CH (Et) S (O) CH2C (O) Me Me
CH (Et) S (O) CH2C (O) Et Me
CH (Et) S (O) CH2C (O) Pr-n Me
CH (Et) S (O) CH2C (O) Pr-i Me
CH (Et) S (O) CH2C (O) Pr-c Me
CH (Et) S (O) CH2C (O) Bu-n Me
CH (Et) S (O) CH2C (O) Bu-i Me
CH (Et) S (O) CH2C (O) Bu-t Me
CH (Et) S (O) CH2C (O) Pen-n Me
CH (Et) S (O) CH2C (O) Pen-c Me
CH (Et) S (O) CH2C (O) Hex-n Me
CH (Et) S (O) CH2C (O) Hex-c Me
CH (Et) S (O) CH2C (O) Me Et
CH (Et) S (O) CH2C (O) Me Pr-n
CH (Et) S (O) CH2C (O) Me Pr-i
CH (Et) S (O) CH2C (O) Me Pr-c
CH (Et) S (O) CH2C (O) Me Bu-n
CH (Et) S (O) CH2C (O) Me Bu-i
CH (Et) S (O) CH2C (O) Me Bu-c
CH (Et) S (O) CH2C (O) Me Bu-s
CH (Et) S (O) CH2C (O) Me Bu-t
CH (Et) S (O) CH2C (O) Me Pen-n
CH (Et) S (O) CH2C (O) Me Pen-c
CH (Et) S (O) CH2C (O) Me Hex-n
CH (Et) S (O) CH2C (O) Me Hex-c
CH (Et) S (O) CH2C (O) Me CH2Pr-c
CH (Et) S (O) CH2C (O) Me CH2Bu-c
CH (Et) S (O) CH2C (O) Me CH2Pen-c
CH (Et) S (O) CH2C (O) Me CH2Hex-c
CH (Et) S (O) CH2C (O) Me CH2CH = CH2
CH (Et) S (O) CH2C (O) Me CH2CH = C (Cl)2
CH (Et) S (O) CH2C (O) Me CH2C≡CH
CH (Et) S (O) CH2C (O) Me CH2CN
CH (Et) S (O) CH2C (O) Me CH2CFThree
CH (Et) S (O) CH2C (O) Me CH2OMe
CH (Et) S (O) CH2C (O) Me CH2OCFThree
CH (Et) S (O) CH2C (O) Me CH2SMe
CH (Et) S (O) CH2C (O) Me CH2S (O) Me
CH (Et) S (O) CH2C (O) Me CH2S (O)2Me
CH (Et) S (O) CH2C (O) Me CH2SCFThree
CH (Et) S (O) CH2C (O) Me CH2S (O) CFThree
CH (Et) S (O) CH2C (O) Me CH2S (O)2CFThree
CH (Et) S (O) CH2C (O) Me CH2CH (OMe)2
CH (Et) S (O) CH2C (O) Me CH2CH (SMe)2
CH (Et) S (O) CH2C (O) Me CH2C (O) Me
CH (Et) S (O) CH2C (O) Me CH2C (O) CFThree
CH (Et) S (O) CH2C (O) Me CH2C (O) OMe
CH (Et) S (O)2CH2C (O) Me Me
CH (Et) S (O)2CH2C (O) Et Me
CH (Et) S (O)2CH2C (O) Pr-n Me
CH (Et) S (O)2CH2C (O) Pr-i Me
CH (Et) S (O)2CH2C (O) Pr-c Me
CH (Et) S (O)2CH2C (O) Bu-n Me
CH (Et) S (O)2CH2C (O) Bu-i Me
CH (Et) S (O)2CH2C (O) Bu-t Me
CH (Et) S (O)2CH2C (O) Pen-n Me
CH (Et) S (O)2CH2C (O) Pen-c Me
CH (Et) S (O)2CH2C (O) Hex-n Me
CH (Et) S (O)2CH2C (O) Hex-c Me
CH (Et) S (O)2CH2C (O) Me Et
CH (Et) S (O)2CH2C (O) Me Pr-n
CH (Et) S (O)2CH2C (O) Me Pr-i
CH (Et) S (O)2CH2C (O) Me Pr-c
CH (Et) S (O)2CH2C (O) Me Bu-n
CH (Et) S (O)2CH2C (O) Me Bu-i
CH (Et) S (O)2CH2C (O) Me Bu-c
CH (Et) S (O)2CH2C (O) Me Bu-s
CH (Et) S (O)2CH2C (O) Me Bu-t
CH (Et) S (O)2CH2C (O) Me Pen-n
CH (Et) S (O)2CH2C (O) Me Pen-c
CH (Et) S (O)2CH2C (O) Me Hex-n
CH (Et) S (O)2CH2C (O) Me Hex-c
CH (Et) S (O)2CH2C (O) Me CH2Pr-c
CH (Et) S (O)2CH2C (O) Me CH2Bu-c
CH (Et) S (O)2CH2C (O) Me CH2Pen-c
CH (Et) S (O)2CH2C (O) Me CH2Hex-c
CH (Et) S (O)2CH2C (O) Me CH2CH = CH2
CH (Et) S (O)2CH2C (O) Me CH2CH = C (Cl)2
CH (Et) S (O)2CH2C (O) Me CH2C≡CH
CH (Et) S (O)2CH2C (O) Me CH2CN
CH (Et) S (O)2CH2C (O) Me CH2CFThree
CH (Et) S (O)2CH2C (O) Me CH2OMe
CH (Et) S (O)2CH2C (O) Me CH2OCFThree
CH (Et) S (O)2CH2C (O) Me CH2SMe
CH (Et) S (O)2CH2C (O) Me CH2S (O) Me
CH (Et) S (O)2CH2C (O) Me CH2S (O)2Me
CH (Et) S (O)2CH2C (O) Me CH2SCFThree
CH (Et) S (O)2CH2C (O) Me CH2S (O) CFThree
CH (Et) S (O)2CH2C (O) Me CH2S (O)2CFThree
CH (Et) S (O)2CH2C (O) Me CH2CH (OMe)2
CH (Et) S (O)2CH2C (O) Me CH2CH (SMe)2
CH (Et) S (O)2CH2C (O) Me CH2C (O) Me
CH (Et) S (O)2CH2C (O) Me CH2C (O) CFThree
CH (Et) S (O)2CH2C (O) Me CH2C (O) OMe
CH2SCH2C (O) NHMe Me
CH2SCH2C (O) NHEt Me
CH2SCH2C (O) NHPr-n Me
CH2SCH2C (O) NHPr-i Me
CH2SCH2C (O) NHPr-c Me
CH2SCH2C (O) NHBu-n Me
CH2SCH2C (O) NHBu-i Me
CH2SCH2C (O) NHBu-c Me
CH2SCH2C (O) NHBu-t Me
CH2SCH2C (O) NHPen-n Me
CH2SCH2C (O) NHPen-c Me
CH2SCH2C (O) NHHex-n Me
CH2SCH2C (O) NHHex-c Me
CH2SCH2C (O) N (Me)2                      Me
CH2SCH2C (O) N (Et)2                     Me
CH2SCH2C (O) NHMe Et
CH2SCH2C (O) NHMe Pr-n
CH2SCH2C (O) NHMe Pr-i
CH2SCH2C (O) NHMe Pr-c
CH2SCH2C (O) NHMe Bu-n
CH2SCH2C (O) NHMe Bu-i
CH2SCH2C (O) NHMe Bu-c
CH2SCH2C (O) NHMe Bu-s
CH2SCH2C (O) NHMe Bu-t
CH2SCH2C (O) NHMe Pen-n
CH2SCH2C (O) NHMe Pen-c
CH2SCH2C (O) NHMe Hex-n
CH2SCH2C (O) NHMe Hex-c
CH2SCH2C (O) NHMe CH2Pr-c
CH2SCH2C (O) NHMe CH2Bu-c
CH2SCH2C (O) NHMe CH2Pen-c
CH2SCH2C (O) NHMe CH2Hex-c
CH2SCH2C (O) NHMe CH2CH = CH2
CH2SCH2C (O) NHMe CH2CH = C (Cl)2
CH2SCH2C (O) NHMe CH2C≡CH
CH2SCH2C (O) NHMe CH2CN
CH2SCH2C (O) NHMe CH2CFThree
CH2SCH2C (O) NHMe CH2OMe
CH2SCH2C (O) NHMe CH2OCFThree
CH2SCH2C (O) NHMe CH2SMe
CH2SCH2C (O) NHMe CH2S (O) Me
CH2SCH2C (O) NHMe CH2S (O)2Me
CH2SCH2C (O) NHMe CH2SCFThree
CH2SCH2C (O) NHMe CH2S (O) CFThree
CH2SCH2C (O) NHMe CH2S (O)2CFThree
CH2SCH2C (O) NHMe CH2CH (OMe)2
CH2SCH2C (O) NHMe CH2CH (SMe)2
CH2SCH2C (O) NHMe CH2C (O) Me
CH2SCH2C (O) NHMe CH2C (O) CFThree
CH2SCH2C (O) NHMe CH2C (O) OMe
CH2S (O) CH2C (O) NHMe Me
CH2S (O) CH2C (O) NHEt Me
CH2S (O) CH2C (O) NHPr-n Me
CH2S (O) CH2C (O) NHPr-i Me
CH2S (O) CH2C (O) NHPr-c Me
CH2S (O) CH2C (O) NHBu-n Me
CH2S (O) CH2C (O) NHBu-i Me
CH2S (O) CH2C (O) NHBu-c Me
CH2S (O) CH2C (O) NHBu-t Me
CH2S (O) CH2C (O) NHPen-n Me
CH2S (O) CH2C (O) NHPen-c Me
CH2S (O) CH2C (O) NHHex-n Me
CH2S (O) CH2C (O) NHHex-c Me
CH2S (O) CH2C (O) N (Me)2                   Me
CH2S (O) CH2C (O) N (Et)2                  Me
CH2S (O) CH2C (O) NHMe Et
CH2S (O) CH2C (O) NHMe Pr-n
CH2S (O) CH2C (O) NHMe Pr-i
CH2S (O) CH2C (O) NHMe Pr-c
CH2S (O) CH2C (O) NHMe Bu-n
CH2S (O) CH2C (O) NHMe Bu-i
CH2S (O) CH2C (O) NHMe Bu-c
CH2S (O) CH2C (O) NHMe Bu-s
CH2S (O) CH2C (O) NHMe Bu-t
CH2S (O) CH2C (O) NHMe Pen-n
CH2S (O) CH2C (O) NHMe Pen-c
CH2S (O) CH2C (O) NHMe Hex-n
CH2S (O) CH2C (O) NHMe Hex-c
CH2S (O) CH2C (O) NHMe CH2Pr-c
CH2S (O) CH2C (O) NHMe CH2Bu-c
CH2S (O) CH2C (O) NHMe CH2Pen-c
CH2S (O) CH2C (O) NHMe CH2Hex-c
CH2S (O) CH2C (O) NHMe CH2CH = CH2
CH2S (O) CH2C (O) NHMe CH2CH = C (Cl)2
CH2S (O) CH2C (O) NHMe CH2C≡CH
CH2S (O) CH2C (O) NHMe CH2CN
CH2S (O) CH2C (O) NHMe CH2CFThree
CH2S (O) CH2C (O) NHMe CH2OMe
CH2S (O) CH2C (O) NHMe CH2OCFThree
CH2S (O) CH2C (O) NHMe CH2SMe
CH2S (O) CH2C (O) NHMe CH2S (O) Me
CH2S (O) CH2C (O) NHMe CH2S (O)2Me
CH2S (O) CH2C (O) NHMe CH2SCFThree
CH2S (O) CH2C (O) NHMe CH2S (O) CFThree
CH2S (O) CH2C (O) NHMe CH2S (O)2CFThree
CH2S (O) CH2C (O) NHMe CH2CH (OMe)2
CH2S (O) CH2C (O) NHMe CH2CH (SMe)2
CH2S (O) CH2C (O) NHMe CH2C (O) Me
CH2S (O) CH2C (O) NHMe CH2C (O) CFThree
CH2S (O) CH2C (O) NHMe CH2C (O) OMe
CH2S (O)2CH2C (O) NHMe Me
CH2S (O)2CH2C (O) NHMe Me
CH2S (O)2CH2C (O) NHEt Me
CH2S (O)2CH2C (O) NHPr-n Me
CH2S (O)2CH2C (O) NHPr-i Me
CH2S (O)2CH2C (O) NHPr-c Me
CH2S (O)2CH2C (O) NHBu-n Me
CH2S (O)2CH2C (O) NHBu-i Me
CH2S (O)2CH2C (O) NHBu-c Me
CH2S (O)2CH2C (O) NHBu-t Me
CH2S (O)2CH2C (O) NHPen-n Me
CH2S (O)2CH2C (O) NHPen-c Me
CH2S (O)2CH2C (O) NHHex-n Me
CH2S (O)2CH2C (O) NHHex-c Me
CH2S (O)2CH2C (O) N (Me)2                   Me
CH2S (O)2CH2C (O) N (Et)2                  Me
CH2S (O)2CH2C (O) NHMe Et
CH2S (O)2CH2C (O) NHMe Pr-n
CH2S (O)2CH2C (O) NHMe Pr-i
CH2S (O)2CH2C (O) NHMe Pr-c
CH2S (O)2CH2C (O) NHMe Bu-n
CH2S (O)2CH2C (O) NHMe Bu-i
CH2S (O)2CH2C (O) NHMe Bu-c
CH2S (O)2CH2C (O) NHMe Bu-s
CH2S (O)2CH2C (O) NHMe Bu-t
CH2S (O)2CH2C (O) NHMe Pen-n
CH2S (O)2CH2C (O) NHMe Pen-c
CH2S (O)2CH2C (O) NHMe Hex-n
CH2S (O)2CH2C (O) NHMe Hex-c
CH2S (O)2CH2C (O) NHMe CH2Pr-c
CH2S (O)2CH2C (O) NHMe CH2Bu-c
CH2S (O)2CH2C (O) NHMe CH2Pen-c
CH2S (O)2CH2C (O) NHMe CH2Hex-c
CH2S (O)2CH2C (O) NHMe CH2CH = CH2
CH2S (O)2CH2C (O) NHMe CH2CH = C (Cl)2
CH2S (O)2CH2C (O) NHMe CH2C≡CH
CH2S (O)2CH2C (O) NHMe CH2CN
CH2S (O)2CH2C (O) NHMe CH2CFThree
CH2S (O)2CH2C (O) NHMe CH2OMe
CH2S (O)2CH2C (O) NHMe CH2OCFThree
CH2S (O)2CH2C (O) NHMe CH2SMe
CH2S (O)2CH2C (O) NHMe CH2S (O) Me
CH2S (O)2CH2C (O) NHMe CH2S (O)2Me
CH2S (O)2CH2C (O) NHMe CH2SCFThree
CH2S (O)2CH2C (O) NHMe CH2S (O) CFThree
CH2S (O)2CH2C (O) NHMe CH2S (O)2CFThree
CH2S (O)2CH2C (O) NHMe CH2CH (OMe)2
CH2S (O)2CH2C (O) NHMe CH2CH (SMe)2
CH2S (O)2CH2C (O) NHMe CH2C (O) Me
CH2S (O)2CH2C (O) NHMe CH2C (O) CFThree
CH2S (O)2CH2C (O) NHMe CH2C (O) OMe
CH (Me) SCH2C (O) NHMe Me
CH (Me) SCH2C (O) NHEt Me
CH (Me) SCH2C (O) NHPr-n Me
CH (Me) SCH2C (O) NHPr-i Me
CH (Me) SCH2C (O) NHPr-c Me
CH (Me) SCH2C (O) NHBu-n Me
CH (Me) SCH2C (O) NHBu-i Me
CH (Me) SCH2C (O) NHBu-c Me
CH (Me) SCH2C (O) NHBu-t Me
CH (Me) SCH2C (O) NHPen-n Me
CH (Me) SCH2C (O) NHPen-c Me
CH (Me) SCH2C (O) NHHex-n Me
CH (Me) SCH2C (O) NHHex-c Me
CH (Me) SCH2C (O) N (Me)2                   Me
CH (Me) SCH2C (O) N (Et)2                   Me
CH (Me) SCH2C (O) NHMe Et
CH (Me) SCH2C (O) NHMe Pr-n
CH (Me) SCH2C (O) NHMe Pr-i
CH (Me) SCH2C (O) NHMe Pr-c
CH (Me) SCH2C (O) NHMe Bu-n
CH (Me) SCH2C (O) NHMe Bu-i
CH (Me) SCH2C (O) NHMe Bu-c
CH (Me) SCH2C (O) NHMe Bu-s
CH (Me) SCH2C (O) NHMe Bu-t
CH (Me) SCH2C (O) NHMe Pen-n
CH (Me) SCH2C (O) NHMe Pen-c
CH (Me) SCH2C (O) NHMe Hex-n
CH (Me) SCH2C (O) NHMe Hex-c
CH (Me) SCH2C (O) NHMe CH2Pr-c
CH (Me) SCH2C (O) NHMe CH2Bu-c
CH (Me) SCH2C (O) NHMe CH2Pen-c
CH (Me) SCH2C (O) NHMe CH2Hex-c
CH (Me) SCH2C (O) NHMe CH2CH = CH2
CH (Me) SCH2C (O) NHMe CH2CH = C (Cl)2
CH (Me) SCH2C (O) NHMe CH2C≡CH
CH (Me) SCH2C (O) NHMe CH2CN
CH (Me) SCH2C (O) NHMe CH2CFThree
CH (Me) SCH2C (O) NHMe CH2OMe
CH (Me) SCH2C (O) NHMe CH2OCFThree
CH (Me) SCH2C (O) NHMe CH2SMe
CH (Me) SCH2C (O) NHMe CH2S (O) Me
CH (Me) SCH2C (O) NHMe CH2S (O)2Me
CH (Me) SCH2C (O) NHMe CH2SCFThree
CH (Me) SCH2C (O) NHMe CH2S (O) CFThree
CH (Me) SCH2C (O) NHMe CH2S (O)2CFThree
CH (Me) SCH2C (O) NHMe CH2CH (OMe)2
CH (Me) SCH2C (O) NHMe CH2CH (SMe)2
CH (Me) SCH2C (O) NHMe CH2C (O) Me
CH (Me) SCH2C (O) NHMe CH2C (O) CFThree
CH (Me) SCH2C (O) NHMe CH2C (O) OMe
CH (Me) S (O) CH2C (O) NHMe Me
CH (Me) S (O) CH2C (O) NHEt Me
CH (Me) S (O) CH2C (O) NHPr-n Me
CH (Me) S (O) CH2C (O) NHPr-i Me
CH (Me) S (O) CH2C (O) NHPr-c Me
CH (Me) S (O) CH2C (O) NHBu-n Me
CH (Me) S (O) CH2C (O) NHBu-i Me
CH (Me) S (O) CH2C (O) NHBu-c Me
CH (Me) S (O) CH2C (O) NHBu-t Me
CH (Me) S (O) CH2C (O) NHPen-n Me
CH (Me) S (O) CH2C (O) NHPen-c Me
CH (Me) S (O) CH2C (O) NHHex-n Me
CH (Me) S (O) CH2C (O) NHHex-c Me
CH (Et) S (O) CH2C (O) N (Me)2                Me
CH (Et) S (O) CH2C (O) N (Et)2                Me
CH (Me) S (O) CH2C (O) NHMe Et
CH (Me) S (O) CH2C (O) NHMe Pr-n
CH (Me) S (O) CH2C (O) NHMe Pr-i
CH (Me) S (O) CH2C (O) NHMe Pr-c
CH (Me) S (O) CH2C (O) NHMe Bu-n
CH (Me) S (O) CH2C (O) NHMe Bu-i
CH (Me) S (O) CH2C (O) NHMe Bu-c
CH (Me) S (O) CH2C (O) NHMe Bu-s
CH (Me) S (O) CH2C (O) NHMe Bu-t
CH (Me) S (O) CH2C (O) NHMe Pen-n
CH (Me) S (O) CH2C (O) NHMe Pen-c
CH (Me) S (O) CH2C (O) NHMe Hex-n
CH (Me) S (O) CH2C (O) NHMe Hex-c
CH (Me) S (O) CH2C (O) NHMe CH2Pr-c
CH (Me) S (O) CH2C (O) NHMe CH2Bu-c
CH (Me) S (O) CH2C (O) NHMe CH2Pen-c
CH (Me) S (O) CH2C (O) NHMe CH2Hex-c
CH (Me) S (O) CH2C (O) NHMe CH2CH = CH2
CH (Me) S (O) CH2C (O) NHMe CH2CH = C (Cl)2
CH (Me) S (O) CH2C (O) NHMe CH2C≡CH
CH (Me) S (O) CH2C (O) NHMe CH2CN
CH (Me) S (O) CH2C (O) NHMe CH2CFThree
CH (Me) S (O) CH2C (O) NHMe CH2OMe
CH (Me) S (O) CH2C (O) NHMe CH2OCFThree
CH (Me) S (O) CH2C (O) NHMe CH2SMe
CH (Me) S (O) CH2C (O) NHMe CH2S (O) Me
CH (Me) S (O) CH2C (O) NHMe CH2S (O)2Me
CH (Me) S (O) CH2C (O) NHMe CH2SCFThree
CH (Me) S (O) CH2C (O) NHMe CH2S (O) CFThree
CH (Me) S (O) CH2C (O) NHMe CH2S (O)2CFThree
CH (Me) S (O) CH2C (O) NHMe CH2CH (OMe)2
CH (Me) S (O) CH2C (O) NHMe CH2CH (SMe)2
CH (Me) S (O) CH2C (O) NHMe CH2C (O) Me
CH (Me) S (O) CH2C (O) NHMe CH2C (O) CFThree
CH (Me) S (O) CH2C (O) NHMe CH2C (O) OMe
CH (Me) S (O)2CH2C (O) NHMe Me
CH (Me) S (O)2CH2C (O) NHEt Me
CH (Me) S (O)2CH2C (O) NHPr-n Me
CH (Me) S (O)2CH2C (O) NHPr-i Me
CH (Me) S (O)2CH2C (O) NHPr-c Me
CH (Me) S (O)2CH2C (O) NHBu-n Me
CH (Me) S (O)2CH2C (O) NHBu-i Me
CH (Me) S (O)2CH2C (O) NHBu-c Me
CH (Me) S (O)2CH2C (O) NHBu-t Me
CH (Me) S (O)2CH2C (O) NHPen-n Me
CH (Me) S (O)2CH2C (O) NHPen-c Me
CH (Me) S (O)2CH2C (O) NHHex-n Me
CH (Me) S (O)2CH2C (O) NHHex-c Me
CH (Me) S (O)2CH2C (O) N (Me)2                Me
CH (Me) S (O)2CH2C (O) N (Et)2               Me
CH (Me) S (O)2CH2C (O) NHMe Et
CH (Me) S (O)2CH2C (O) NHMe Pr-n
CH (Me) S (O)2CH2C (O) NHMe Pr-i
CH (Me) S (O)2CH2C (O) NHMe Pr-c
CH (Me) S (O)2CH2C (O) NHMe Bu-n
CH (Me) S (O)2CH2C (O) NHMe Bu-i
CH (Me) S (O)2CH2C (O) NHMe Bu-c
CH (Me) S (O)2CH2C (O) NHMe Bu-s
CH (Me) S (O)2CH2C (O) NHMe Bu-t
CH (Me) S (O)2CH2C (O) NHMe Pen-n
CH (Me) S (O)2CH2C (O) NHMe Pen-c
CH (Me) S (O)2CH2C (O) NHMe Hex-n
CH (Me) S (O)2CH2C (O) NHMe Hex-c
CH (Me) S (O)2CH2C (O) NHMe CH2Pr-c
CH (Me) S (O)2CH2C (O) NHMe CH2Bu-c
CH (Me) S (O)2CH2C (O) NHMe CH2Pen-c
CH (Me) S (O)2CH2C (O) NHMe CH2Hex-c
CH (Me) S (O)2CH2C (O) NHMe CH2CH = CH2
CH (Me) S (O)2CH2C (O) NHMe CH2CH = C (Cl)2
CH (Me) S (O)2CH2C (O) NHMe CH2C≡CH
CH (Me) S (O)2CH2C (O) NHMe CH2CN
CH (Me) S (O)2CH2C (O) NHMe CH2CFThree
CH (Me) S (O)2CH2C (O) NHMe CH2OMe
CH (Me) S (O)2CH2C (O) NHMe CH2OCFThree
CH (Me) S (O)2CH2C (O) NHMe CH2SMe
CH (Me) S (O)2CH2C (O) NHMe CH2S (O) Me
CH (Me) S (O)2CH2C (O) NHMe CH2S (O)2Me
CH (Me) S (O)2CH2C (O) NHMe CH2SCFThree
CH (Me) S (O)2CH2C (O) NHMe CH2S (O) CFThree
CH (Me) S (O)2CH2C (O) NHMe CH2S (O)2CFThree
CH (Me) S (O)2CH2C (O) NHMe CH2CH (OMe)2
CH (Me) S (O)2CH2C (O) NHMe CH2CH (SMe)2
CH (Me) S (O)2CH2C (O) NHMe CH2C (O) Me
CH (Me) S (O)2CH2C (O) NHMe CH2C (O) CFThree
CH (Me) S (O)2CH2C (O) NHMe CH2C (O) OMe
CH (Et) SCH2C (O) NHMe Me
CH (Et) SCH2C (O) NHEt Me
CH (Et) SCH2C (O) NHPr-n Me
CH (Et) SCH2C (O) NHPr-i Me
CH (Et) SCH2C (O) NHPr-c Me
CH (Et) SCH2C (O) NHBu-n Me
CH (Et) SCH2C (O) NHBu-i Me
CH (Et) SCH2C (O) NHBu-c Me
CH (Et) SCH2C (O) NHBu-t Me
CH (Et) SCH2C (O) NHPen-n Me
CH (Et) SCH2C (O) NHPen-c Me
CH (Et) SCH2C (O) NHHex-n Me
CH (Et) SCH2C (O) NHHex-c Me
CH (Et) SCH2C (O) N (Me)2                   Me
CH (Et) SCH2C (O) N (Et)2                   Me
CH (Et) SCH2C (O) NHMe Et
CH (Et) SCH2C (O) NHMe Pr-n
CH (Et) SCH2C (O) NHMe Pr-i
CH (Et) SCH2C (O) NHMe Pr-c
CH (Et) SCH2C (O) NHMe Bu-n
CH (Et) SCH2C (O) NHMe Bu-i
CH (Et) SCH2C (O) NHMe Bu-c
CH (Et) SCH2C (O) NHMe Bu-s
CH (Et) SCH2C (O) NHMe Bu-t
CH (Et) SCH2C (O) NHMe Pen-n
CH (Et) SCH2C (O) NHMe Pen-c
CH (Et) SCH2C (O) NHMe Hex-n
CH (Et) SCH2C (O) NHMe Hex-c
CH (Et) SCH2C (O) NHMe CH2Pr-c
CH (Et) SCH2C (O) NHMe CH2Bu-c
CH (Et) SCH2C (O) NHMe CH2Pen-c
CH (Et) SCH2C (O) NHMe CH2Hex-c
CH (Et) SCH2C (O) NHMe CH2CH = CH2
CH (Et) SCH2C (O) NHMe CH2CH = C (Cl)2
CH (Et) SCH2C (O) NHMe CH2C≡CH
CH (Et) SCH2C (O) NHMe CH2CN
CH (Et) SCH2C (O) NHMe CH2CFThree
CH (Et) SCH2C (O) NHMe CH2OMe
CH (Et) SCH2C (O) NHMe CH2OCFThree
CH (Et) SCH2C (O) NHMe CH2SMe
CH (Et) SCH2C (O) NHMe CH2S (O) Me
CH (Et) SCH2C (O) NHMe CH2S (O)2Me
CH (Et) SCH2C (O) NHMe CH2SCFThree
CH (Et) SCH2C (O) NHMe CH2S (O) CFThree
CH (Et) SCH2C (O) NHMe CH2S (O)2CFThree
CH (Et) SCH2C (O) NHMe CH2CH (OMe)2
CH (Et) SCH2C (O) NHMe CH2CH (SMe)2
CH (Et) SCH2C (O) NHMe CH2C (O) Me
CH (Et) SCH2C (O) NHMe CH2C (O) CFThree
CH (Et) SCH2C (O) NHMe CH2C (O) OMe
CH (Et) S (O) CH2C (O) NHMe Me
CH (Et) S (O) CH2C (O) NHEt Me
CH (Et) S (O) CH2C (O) NHPr-n Me
CH (Et) S (O) CH2C (O) NHPr-i Me
CH (Et) S (O) CH2C (O) NHPr-c Me
CH (Et) S (O) CH2C (O) NHBu-n Me
CH (Et) S (O) CH2C (O) NHBu-i Me
CH (Et) S (O) CH2C (O) NHBu-c Me
CH (Et) S (O) CH2C (O) NHBu-t Me
CH (Et) S (O) CH2C (O) NHPen-n Me
CH (Et) S (O) CH2C (O) NHPen-c Me
CH (Et) S (O) CH2C (O) NHHex-n Me
CH (Et) S (O) CH2C (O) NHHex-c Me
CH (Et) S (O) CH2C (O) N (Me)2                Me
CH (Et) S (O) CH2C (O) N (Et)2                Me
CH (Et) S (O) CH2C (O) NHMe Et
CH (Et) S (O) CH2C (O) NHMe Pr-n
CH (Et) S (O) CH2C (O) NHMe Pr-i
CH (Et) S (O) CH2C (O) NHMe Pr-c
CH (Et) S (O) CH2C (O) NHMe Bu-n
CH (Et) S (O) CH2C (O) NHMe Bu-i
CH (Et) S (O) CH2C (O) NHMe Bu-c
CH (Et) S (O) CH2C (O) NHMe Bu-s
CH (Et) S (O) CH2C (O) NHMe Bu-t
CH (Et) S (O) CH2C (O) NHMe Pen-n
CH (Et) S (O) CH2C (O) NHMe Pen-c
CH (Et) S (O) CH2C (O) NHMe Hex-n
CH (Et) S (O) CH2C (O) NHMe Hex-c
CH (Et) S (O) CH2C (O) NHMe CH2Pr-c
CH (Et) S (O) CH2C (O) NHMe CH2Bu-c
CH (Et) S (O) CH2C (O) NHMe CH2Pen-c
CH (Et) S (O) CH2C (O) NHMe CH2Hex-c
CH (Et) S (O) CH2C (O) NHMe CH2CH = CH2
CH (Et) S (O) CH2C (O) NHMe CH2CH = C (Cl)2
CH (Et) S (O) CH2C (O) NHMe CH2C≡CH
CH (Et) S (O) CH2C (O) NHMe CH2CN
CH (Et) S (O) CH2C (O) NHMe CH2CFThree
CH (Et) S (O) CH2C (O) NHMe CH2OMe
CH (Et) S (O) CH2C (O) NHMe CH2OCFThree
CH (Et) S (O) CH2C (O) NHMe CH2SMe
CH (Et) S (O) CH2C (O) NHMe CH2S (O) Me
CH (Et) S (O) CH2C (O) NHMe CH2S (O)2Me
CH (Et) S (O) CH2C (O) NHMe CH2SCFThree
CH (Et) S (O) CH2C (O) NHMe CH2S (O) CFThree
CH (Et) S (O) CH2C (O) NHMe CH2S (O)2CFThree
CH (Et) S (O) CH2C (O) NHMe CH2CH (OMe)2
CH (Et) S (O) CH2C (O) NHMe CH2CH (SMe)2
CH (Et) S (O) CH2C (O) NHMe CH2C (O) Me
CH (Et) S (O) CH2C (O) NHMe CH2C (O) CFThree
CH (Et) S (O) CH2C (O) NHMe CH2C (O) OMe
CH (Et) S (O)2CH2C (O) NHMe Me
CH (Et) S (O)2CH2C (O) NHEt Me
CH (Et) S (O)2CH2C (O) NHPr-n Me
CH (Et) S (O)2CH2C (O) NHPr-i Me
CH (Et) S (O)2CH2C (O) NHPr-c Me
CH (Et) S (O)2CH2C (O) NHBu-n Me
CH (Et) S (O)2CH2C (O) NHBu-i Me
CH (Et) S (O)2CH2C (O) NHBu-c Me
CH (Et) S (O)2CH2C (O) NHBu-t Me
CH (Et) S (O)2CH2C (O) NHPen-n Me
CH (Et) S (O)2CH2C (O) NHPen-c Me
CH (Et) S (O)2CH2C (O) NHHex-n Me
CH (Et) S (O)2CH2C (O) NHHex-c Me
CH (Et) S (O)2CH2C (O) N (Me)2                Me
CH (Et) S (O)2CH2C (O) N (Et)2               Me
CH (Et) S (O)2CH2C (O) NHMe Et
CH (Et) S (O)2CH2C (O) NHMe Pr-n
CH (Et) S (O)2CH2C (O) NHMe Pr-i
CH (Et) S (O)2CH2C (O) NHMe Pr-c
CH (Et) S (O)2CH2C (O) NHMe Bu-n
CH (Et) S (O)2CH2C (O) NHMe Bu-i
CH (Et) S (O)2CH2C (O) NHMe Bu-c
CH (Et) S (O)2CH2C (O) NHMe Bu-s
CH (Et) S (O)2CH2C (O) NHMe Bu-t
CH (Et) S (O)2CH2C (O) NHMe Pen-n
CH (Et) S (O)2CH2C (O) NHMe Pen-c
CH (Et) S (O)2CH2C (O) NHMe Hex-n
CH (Et) S (O)2CH2C (O) NHMe Hex-c
CH (Et) S (O)2CH2C (O) NHMe CH2Pr-c
CH (Et) S (O)2CH2C (O) NHMe CH2Bu-c
CH (Et) S (O)2CH2C (O) NHMe CH2Pen-c
CH (Et) S (O)2CH2C (O) NHMe CH2Hex-c
CH (Et) S (O)2CH2C (O) NHMe CH2CH = CH2
CH (Et) S (O)2CH2C (O) NHMe CH2CH = C (Cl)2
CH (Et) S (O)2CH2C (O) NHMe CH2C≡CH
CH (Et) S (O)2CH2C (O) NHMe CH2CN
CH (Et) S (O)2CH2C (O) NHMe CH2CFThree
CH (Et) S (O)2CH2C (O) NHMe CH2OMe
CH (Et) S (O)2CH2C (O) NHMe CH2OCFThree
CH (Et) S (O)2CH2C (O) NHMe CH2SMe
CH (Et) S (O)2CH2C (O) NHMe CH2S (O) Me
CH (Et) S (O)2CH2C (O) NHMe CH2S (O)2Me
CH (Et) S (O)2CH2C (O) NHMe CH2SCFThree
CH (Et) S (O)2CH2C (O) NHMe CH2S (O) CFThree
CH (Et) S (O)2CH2C (O) NHMe CH2S (O)2CFThree
CH (Et) S (O)2CH2C (O) NHMe CH2CH (OMe)2
CH (Et) S (O)2CH2C (O) NHMe CH2CH (SMe)2
CH (Et) S (O)2CH2C (O) NHMe CH2C (O) Me
CH (Et) S (O)2CH2C (O) NHMe CH2C (O) CFThree
CH (Et) S (O)2CH2C (O) NHMe CH2C (O) OMe
CH2SCH (Me) C (O) OMe Me
CH2SCH (Me) C (O) OEt Me
CH2SCH (Me) C (O) OPr-n Me
CH2SCH (Me) C (O) OPr-i Me
CH2SCH (Me) C (O) OBu-n Me
CH2SCH (Me) C (O) OBu-i Me
CH2SCH (Me) C (O) OBu-t Me
CH2SCH (Me) C (O) OPen-n Me
CH2SCH (Me) C (O) OHex-n Me
CH2SCH (Me) C (O) OMe Et
CH2SCH (Me) C (O) OMe Pr-n
CH2SCH (Me) C (O) OMe Pr-i
CH2SCH (Me) C (O) OMe Pr-c
CH2SCH (Me) C (O) OMe Bu-n
CH2SCH (Me) C (O) OMe Bu-i
CH2SCH (Me) C (O) OMe Bu-c
CH2SCH (Me) C (O) OMe Bu-s
CH2SCH (Me) C (O) OMe Bu-t
CH2SCH (Me) C (O) OMe Pen-n
CH2SCH (Me) C (O) OMe Pen-c
CH2SCH (Me) C (O) OMe Hex-n
CH2SCH (Me) C (O) OMe Hex-c
CH2SCH (Me) C (O) OMe CH2Pr-c
CH2SCH (Me) C (O) OMe CH2Bu-c
CH2SCH (Me) C (O) OMe CH2Pen-c
CH2SCH (Me) C (O) OMe CH2Hex-c
CH2SCH (Me) C (O) OMe CH2CH = CH2
CH2SCH (Me) C (O) OMe CH2CH = C (Cl)2
CH2SCH (Me) C (O) OMe CH2C≡CH
CH2SCH (Me) C (O) OMe CH2CN
CH2SCH (Me) C (O) OMe CH2CFThree
CH2SCH (Me) C (O) OMe CH2OMe
CH2SCH (Me) C (O) OMe CH2OCFThree
CH2SCH (Me) C (O) OMe CH2SMe
CH2SCH (Me) C (O) OMe CH2S (O) Me
CH2SCH (Me) C (O) OMe CH2S (O)2Me
CH2SCH (Me) C (O) OMe CH2SCFThree
CH2SCH (Me) C (O) OMe CH2S (O) CFThree
CH2SCH (Me) C (O) OMe CH2S (O)2CFThree
CH2SCH (Me) C (O) OMe CH2CH (OMe)2
CH2SCH (Me) C (O) OMe CH2CH (SMe)2
CH2SCH (Me) C (O) OMe CH2C (O) Me
CH2SCH (Me) C (O) OMe CH2C (O) CFThree
CH2SCH (Me) C (O) OMe CH2C (O) OMe
CH2S (O) CH (Me) C (O) OMe Me
CH2S (O) CH (Me) C (O) OEt Me
CH2S (O) CH (Me) C (O) OPr-n Me
CH2S (O) CH (Me) C (O) OPr-i Me
CH2S (O) CH (Me) C (O) OBu-n Me
CH2S (O) CH (Me) C (O) OBu-i Me
CH2S (O) CH (Me) C (O) OBu-t Me
CH2S (O) CH (Me) C (O) OPen-n Me
CH2S (O) CH (Me) C (O) OHex-n Me
CH2S (O) CH (Me) C (O) OMe Et
CH2S (O) CH (Me) C (O) OMe Pr-n
CH2S (O) CH (Me) C (O) OMe Pr-i
CH2S (O) CH (Me) C (O) OMe Pr-c
CH2S (O) CH (Me) C (O) OMe Bu-n
CH2S (O) CH (Me) C (O) OMe Bu-i
CH2S (O) CH (Me) C (O) OMe Bu-c
CH2S (O) CH (Me) C (O) OMe Bu-s
CH2S (O) CH (Me) C (O) OMe Bu-t
CH2S (O) CH (Me) C (O) OMe Pen-n
CH2S (O) CH (Me) C (O) OMe Pen-c
CH2S (O) CH (Me) C (O) OMe Hex-n
CH2S (O) CH (Me) C (O) OMe Hex-c
CH2S (O) CH (Me) C (O) OMe CH2Pr-c
CH2S (O) CH (Me) C (O) OMe CH2Bu-c
CH2S (O) CH (Me) C (O) OMe CH2Pen-c
CH2S (O) CH (Me) C (O) OMe CH2Hex-c
CH2S (O) CH (Me) C (O) OMe CH2CH = CH2
CH2S (O) CH (Me) C (O) OMe CH2CH = C (Cl)2
CH2S (O) CH (Me) C (O) OMe CH2C≡CH
CH2S (O) CH (Me) C (O) OMe CH2CN
CH2S (O) CH (Me) C (O) OMe CH2CFThree
CH2S (O) CH (Me) C (O) OMe CH2OMe
CH2S (O) CH (Me) C (O) OMe CH2OCFThree
CH2S (O) CH (Me) C (O) OMe CH2SMe
CH2S (O) CH (Me) C (O) OMe CH2S (O) Me
CH2S (O) CH (Me) C (O) OMe CH2S (O)2Me
CH2S (O) CH (Me) C (O) OMe CH2SCFThree
CH2S (O) CH (Me) C (O) OMe CH2S (O) CFThree
CH2S (O) CH (Me) C (O) OMe CH2S (O)2CFThree
CH2S (O) CH (Me) C (O) OMe CH2CH (OMe)2
CH2S (O) CH (Me) C (O) OMe CH2CH (SMe)2
CH2S (O) CH (Me) C (O) OMe CH2C (O) Me
CH2S (O) CH (Me) C (O) OMe CH2C (O) CFThree
CH2S (O) CH (Me) C (O) OMe CH2C (O) OMe
CH2S (O)2CH (Me) C (O) OMe Me
CH2S (O)2CH (Me) C (O) OEt Me
CH2S (O)2CH (Me) C (O) OPr-n Me
CH2S (O)2CH (Me) C (O) OPr-i Me
CH2S (O)2CH (Me) C (O) OBu-n Me
CH2S (O)2CH (Me) C (O) OBu-i Me
CH2S (O)2CH (Me) C (O) OBu-t Me
CH2S (O)2CH (Me) C (O) OPen-n Me
CH2S (O)2CH (Me) C (O) OHex-n Me
CH2S (O)2CH (Me) C (O) OMe Et
CH2S (O)2CH (Me) C (O) OMe Pr-n
CH2S (O)2CH (Me) C (O) OMe Pr-i
CH2S (O)2CH (Me) C (O) OMe Pr-c
CH2S (O)2CH (Me) C (O) OMe Bu-n
CH2S (O)2CH (Me) C (O) OMe Bu-i
CH2S (O)2CH (Me) C (O) OMe Bu-c
CH2S (O)2CH (Me) C (O) OMe Bu-s
CH2S (O)2CH (Me) C (O) OMe Bu-t
CH2S (O)2CH (Me) C (O) OMe Pen-n
CH2S (O)2CH (Me) C (O) OMe Pen-c
CH2S (O)2CH (Me) C (O) OMe Hex-n
CH2S (O)2CH (Me) C (O) OMe Hex-c
CH2S (O)2CH (Me) C (O) OMe CH2Pr-c
CH2S (O)2CH (Me) C (O) OMe CH2Bu-c
CH2S (O)2CH (Me) C (O) OMe CH2Pen-c
CH2S (O)2CH (Me) C (O) OMe CH2Hex-c
CH2S (O)2CH (Me) C (O) OMe CH2CH = CH2
CH2S (O)2CH (Me) C (O) OMe CH2CH = C (Cl)2
CH2S (O)2CH (Me) C (O) OMe CH2C≡CH
CH2S (O)2CH (Me) C (O) OMe CH2CN
CH2S (O)2CH (Me) C (O) OMe CH2CFThree
CH2S (O)2CH (Me) C (O) OMe CH2OMe
CH2S (O)2CH (Me) C (O) OMe CH2OCFThree
CH2S (O)2CH (Me) C (O) OMe CH2SMe
CH2S (O)2CH (Me) C (O) OMe CH2S (O) Me
CH2S (O)2CH (Me) C (O) OMe CH2S (O)2Me
CH2S (O)2CH (Me) C (O) OMe CH2SCFThree
CH2S (O)2CH (Me) C (O) OMe CH2S (O) CFThree
CH2S (O)2CH (Me) C (O) OMe CH2S (O)2CFThree
CH2S (O)2CH (Me) C (O) OMe CH2CH (OMe)2
CH2S (O)2CH (Me) C (O) OMe CH2CH (SMe)2
CH2S (O)2CH (Me) C (O) OMe CH2C (O) Me
CH2S (O)2CH (Me) C (O) OMe CH2C (O) CFThree
CH2S (O)2CH (Me) C (O) OMe CH2C (O) OMe
CH (Me) SCH (Me) C (O) OMe Me
CH (Me) SCH (Me) C (O) OEt Me
CH (Me) SCH (Me) C (O) OPr-n Me
CH (Me) SCH (Me) C (O) OPr-i Me
CH (Me) SCH (Me) C (O) OBu-n Me
CH (Me) SCH (Me) C (O) OBu-i Me
CH (Me) SCH (Me) C (O) OBu-t Me
CH (Me) SCH (Me) C (O) OPen-n Me
CH (Me) SCH (Me) C (O) OHex-n Me
CH (Me) SCH (Me) C (O) OMe Et
CH (Me) SCH (Me) C (O) OMe Pr-n
CH (Me) SCH (Me) C (O) OMe Pr-i
CH (Me) SCH (Me) C (O) OMe Pr-c
CH (Me) SCH (Me) C (O) OMe Bu-n
CH (Me) SCH (Me) C (O) OMe Bu-i
CH (Me) SCH (Me) C (O) OMe Bu-c
CH (Me) SCH (Me) C (O) OMe Bu-s
CH (Me) SCH (Me) C (O) OMe Bu-t
CH (Me) SCH (Me) C (O) OMe Pen-n
CH (Me) SCH (Me) C (O) OMe Pen-c
CH (Me) SCH (Me) C (O) OMe Hex-n
CH (Me) SCH (Me) C (O) OMe Hex-c
CH (Me) SCH (Me) C (O) OMe CH2Pr-c
CH (Me) SCH (Me) C (O) OMe CH2Bu-c
CH (Me) SCH (Me) C (O) OMe CH2Pen-c
CH (Me) SCH (Me) C (O) OMe CH2Hex-c
CH (Me) SCH (Me) C (O) OMe CH2CH = CH2
CH (Me) SCH (Me) C (O) OMe CH2CH = C (Cl)2
CH (Me) SCH (Me) C (O) OMe CH2C≡CH
CH (Me) SCH (Me) C (O) OMe CH2CN
CH (Me) SCH (Me) C (O) OMe CH2CFThree
CH (Me) SCH (Me) C (O) OMe CH2OMe
CH (Me) SCH (Me) C (O) OMe CH2OCFThree
CH (Me) SCH (Me) C (O) OMe CH2SMe
CH (Me) SCH (Me) C (O) OMe CH2S (O) Me
CH (Me) SCH (Me) C (O) OMe CH2S (O)2Me
CH (Me) SCH (Me) C (O) OMe CH2SCFThree
CH (Me) SCH (Me) C (O) OMe CH2S (O) CFThree
CH (Me) SCH (Me) C (O) OMe CH2S (O)2CFThree
CH (Me) SCH (Me) C (O) OMe CH2CH (OMe)2
CH (Me) SCH (Me) C (O) OMe CH2CH (SMe)2
CH (Me) SCH (Me) C (O) OMe CH2C (O) Me
CH (Me) SCH (Me) C (O) OMe CH2C (O) CFThree
CH (Me) SCH (Me) C (O) OMe CH2C (O) OMe
CH (Me) S (O) CH (Me) C (O) OMe Me
CH (Me) S (O) CH (Me) C (O) OEt Me
CH (Me) S (O) CH (Me) C (O) OPr-n Me
CH (Me) S (O) CH (Me) C (O) OPr-i Me
CH (Me) S (O) CH (Me) C (O) OBu-n Me
CH (Me) S (O) CH (Me) C (O) OBu-i Me
CH (Me) S (O) CH (Me) C (O) OBu-t Me
CH (Me) S (O) CH (Me) C (O) OPen-n Me
CH (Me) S (O) CH (Me) C (O) OHex-n Me
CH (Me) S (O) CH (Me) C (O) OMe Et
CH (Me) S (O) CH (Me) C (O) OMe Pr-n
CH (Me) S (O) CH (Me) C (O) OMe Pr-i
CH (Me) S (O) CH (Me) C (O) OMe Pr-c
CH (Me) S (O) CH (Me) C (O) OMe Bu-n
CH (Me) S (O) CH (Me) C (O) OMe Bu-i
CH (Me) S (O) CH (Me) C (O) OMe Bu-c
CH (Me) S (O) CH (Me) C (O) OMe Bu-s
CH (Me) S (O) CH (Me) C (O) OMe Bu-t
CH (Me) S (O) CH (Me) C (O) OMe Pen-n
CH (Me) S (O) CH (Me) C (O) OMe Pen-c
CH (Me) S (O) CH (Me) C (O) OMe Hex-n
CH (Me) S (O) CH (Me) C (O) OMe Hex-c
CH (Me) S (O) CH (Me) C (O) OMe CH2Pr-c
CH (Me) S (O) CH (Me) C (O) OMe CH2Bu-c
CH (Me) S (O) CH (Me) C (O) OMe CH2Pen-c
CH (Me) S (O) CH (Me) C (O) OMe CH2Hex-c
CH (Me) S (O) CH (Me) C (O) OMe CH2CH = CH2
CH (Me) S (O) CH (Me) C (O) OMe CH2CH = C (Cl)2
CH (Me) S (O) CH (Me) C (O) OMe CH2C≡CH
CH (Me) S (O) CH (Me) C (O) OMe CH2CN
CH (Me) S (O) CH (Me) C (O) OMe CH2CFThree
CH (Me) S (O) CH (Me) C (O) OMe CH2OMe
CH (Me) S (O) CH (Me) C (O) OMe CH2OCFThree
CH (Me) S (O) CH (Me) C (O) OMe CH2SMe
CH (Me) S (O) CH (Me) C (O) OMe CH2S (O) Me
CH (Me) S (O) CH (Me) C (O) OMe CH2S (O)2Me
CH (Me) S (O) CH (Me) C (O) OMe CH2SCFThree
CH (Me) S (O) CH (Me) C (O) OMe CH2S (O) CFThree
CH (Me) S (O) CH (Me) C (O) OMe CH2S (O)2CFThree
CH (Me) S (O) CH (Me) C (O) OMe CH2CH (OMe)2
CH (Me) S (O) CH (Me) C (O) OMe CH2CH (SMe)2
CH (Me) S (O) CH (Me) C (O) OMe CH2C (O) Me
CH (Me) S (O) CH (Me) C (O) OMe CH2C (O) CFThree
CH (Me) S (O) CH (Me) C (O) OMe CH2C (O) OMe
CH (Me) S (O)2CH (Me) C (O) OMe Me
CH (Me) S (O)2CH (Me) C (O) OEt Me
CH (Me) S (O)2CH (Me) C (O) OPr-n Me
CH (Me) S (O)2CH (Me) C (O) OPr-i Me
CH (Me) S (O)2CH (Me) C (O) OBu-n Me
CH (Me) S (O)2CH (Me) C (O) OBu-i Me
CH (Me) S (O)2CH (Me) C (O) OBu-t Me
CH (Me) S (O)2CH (Me) C (O) OPen-n Me
CH (Me) S (O)2CH (Me) C (O) OMe Et
CH (Me) S (O)2CH (Me) C (O) OMe Pr-n
CH (Me) S (O)2CH (Me) C (O) OMe Pr-i
CH (Me) S (O)2CH (Me) C (O) OMe Pr-c
CH (Me) S (O)2CH (Me) C (O) OMe Bu-n
CH (Me) S (O)2CH (Me) C (O) OMe Bu-i
CH (Me) S (O)2CH (Me) C (O) OMe Bu-c
CH (Me) S (O)2CH (Me) C (O) OMe Bu-s
CH (Me) S (O)2CH (Me) C (O) OMe Bu-t
CH (Me) S (O)2CH (Me) C (O) OMe Pen-n
CH (Me) S (O)2CH (Me) C (O) OMe Pen-c
CH (Me) S (O)2CH (Me) C (O) OMe Hex-n
CH (Me) S (O)2CH (Me) C (O) OMe Hex-c
CH (Me) S (O)2CH (Me) C (O) OMe CH2Pr-c
CH (Me) S (O)2CH (Me) C (O) OMe CH2Bu-c
CH (Me) S (O)2CH (Me) C (O) OMe CH2Pen-c
CH (Me) S (O)2CH (Me) C (O) OMe CH2Hex-c
CH (Me) S (O)2CH (Me) C (O) OMe CH2CH = CH2
CH (Me) S (O)2CH (Me) C (O) OMe CH2CH = C (Cl)2
CH (Me) S (O)2CH (Me) C (O) OMe CH2C≡CH
CH (Me) S (O)2CH (Me) C (O) OMe CH2CN
CH (Me) S (O)2CH (Me) C (O) OMe CH2CFThree
CH (Me) S (O)2CH (Me) C (O) OMe CH2OMe
CH (Me) S (O)2CH (Me) C (O) OMe CH2OCFThree
CH (Me) S (O)2CH (Me) C (O) OMe CH2SMe
CH (Me) S (O)2CH (Me) C (O) OMe CH2S (O) Me
CH (Me) S (O)2CH (Me) C (O) OMe CH2S (O)2Me
CH (Me) S (O)2CH (Me) C (O) OMe CH2SCFThree
CH (Me) S (O)2CH (Me) C (O) OMe CH2S (O) CFThree
CH (Me) S (O)2CH (Me) C (O) OMe CH2S (O)2CFThree
CH (Me) S (O)2CH (Me) C (O) OMe CH2CH (OMe)2
CH (Me) S (O)2CH (Me) C (O) OMe CH2CH (SMe)2
CH (Me) S (O)2CH (Me) C (O) OMe CH2C (O) Me
CH (Me) S (O)2CH (Me) C (O) OMe CH2C (O) CFThree
CH (Me) S (O)2CH (Me) C (O) OMe CH2C (O) OMe
CH (Et) SCH (Me) C (O) OMe Me
CH (Et) SCH (Me) C (O) OEt Me
CH (Et) SCH (Me) C (O) OPr-n Me
CH (Et) SCH (Me) C (O) OPr-i Me
CH (Et) SCH (Me) C (O) OBu-n Me
CH (Et) SCH (Me) C (O) OBu-i Me
CH (Et) SCH (Me) C (O) OBu-t Me
CH (Et) SCH (Me) C (O) OPen-n Me
CH (Et) SCH (Me) C (O) OHex-n Me
CH (Et) SCH (Me) C (O) OMe Et
CH (Et) SCH (Me) C (O) OMe Pr-n
CH (Et) SCH (Me) C (O) OMe Pr-i
CH (Et) SCH (Me) C (O) OMe Pr-c
CH (Et) SCH (Me) C (O) OMe Bu-n
CH (Et) SCH (Me) C (O) OMe Bu-i
CH (Et) SCH (Me) C (O) OMe Bu-c
CH (Et) SCH (Me) C (O) OMe Bu-s
CH (Et) SCH (Me) C (O) OMe Bu-t
CH (Et) SCH (Me) C (O) OMe Pen-n
CH (Et) SCH (Me) C (O) OMe Pen-c
CH (Et) SCH (Me) C (O) OMe Hex-n
CH (Et) SCH (Me) C (O) OMe Hex-c
CH (Et) SCH (Me) C (O) OMe CH2Pr-c
CH (Et) SCH (Me) C (O) OMe CH2Bu-c
CH (Et) SCH (Me) C (O) OMe CH2Pen-c
CH (Et) SCH (Me) C (O) OMe CH2Hex-c
CH (Et) SCH (Me) C (O) OMe CH2CH = CH2
CH (Et) SCH (Me) C (O) OMe CH2CH = C (Cl)2
CH (Et) SCH (Me) C (O) OMe CH2C≡CH
CH (Et) SCH (Me) C (O) OMe CH2CN
CH (Et) SCH (Me) C (O) OMe CH2CFThree
CH (Et) SCH (Me) C (O) OMe CH2OMe
CH (Et) SCH (Me) C (O) OMe CH2OCFThree
CH (Et) SCH (Me) C (O) OMe CH2SMe
CH (Et) SCH (Me) C (O) OMe CH2S (O) Me
CH (Et) SCH (Me) C (O) OMe CH2S (O)2Me
CH (Et) SCH (Me) C (O) OMe CH2SCFThree
CH (Et) SCH (Me) C (O) OMe CH2S (O) CFThree
CH (Et) SCH (Me) C (O) OMe CH2S (O)2CFThree
CH (Et) SCH (Me) C (O) OMe CH2CH (OMe)2
CH (Et) SCH (Me) C (O) OMe CH2CH (SMe)2
CH (Et) SCH (Me) C (O) OMe CH2C (O) Me
CH (Et) SCH (Me) C (O) OMe CH2C (O) CFThree
CH (Et) SCH (Me) C (O) OMe CH2C (O) OMe
CH (Et) S (O) CH (Me) C (O) OMe Me
CH (Et) S (O) CH (Me) C (O) OEt Me
CH (Et) S (O) CH (Me) C (O) OPr-n Me
CH (Et) S (O) CH (Me) C (O) OPr-i Me
CH (Et) S (O) CH (Me) C (O) OBu-n Me
CH (Et) S (O) CH (Me) C (O) OBu-i Me
CH (Et) S (O) CH (Me) C (O) OBu-t Me
CH (Et) S (O) CH (Me) C (O) OPen-n Me
CH (Et) S (O) CH (Me) C (O) OHex-n Me
CH (Et) S (O) CH (Me) C (O) OMe Et
CH (Et) S (O) CH (Me) C (O) OMe Pr-n
CH (Et) S (O) CH (Me) C (O) OMe Pr-i
CH (Et) S (O) CH (Me) C (O) OMe Pr-c
CH (Et) S (O) CH (Me) C (O) OMe Bu-n
CH (Et) S (O) CH (Me) C (O) OMe Bu-i
CH (Et) S (O) CH (Me) C (O) OMe Bu-c
CH (Et) S (O) CH (Me) C (O) OMe Bu-s
CH (Et) S (O) CH (Me) C (O) OMe Bu-t
CH (Et) S (O) CH (Me) C (O) OMe Pen-n
CH (Et) S (O) CH (Me) C (O) OMe Pen-c
CH (Et) S (O) CH (Me) C (O) OMe Hex-n
CH (Et) S (O) CH (Me) C (O) OMe Hex-c
CH (Et) S (O) CH (Me) C (O) OMe CH2Pr-c
CH (Et) S (O) CH (Me) C (O) OMe CH2Bu-c
CH (Et) S (O) CH (Me) C (O) OMe CH2Pen-c
CH (Et) S (O) CH (Me) C (O) OMe CH2Hex-c
CH (Et) S (O) CH (Me) C (O) OMe CH2CH = CH2
CH (Et) S (O) CH (Me) C (O) OMe CH2CH = C (Cl)2
CH (Et) S (O) CH (Me) C (O) OMe CH2C≡CH
CH (Et) S (O) CH (Me) C (O) OMe CH2CN
CH (Et) S (O) CH (Me) C (O) OMe CH2CFThree
CH (Et) S (O) CH (Me) C (O) OMe CH2OMe
CH (Et) S (O) CH (Me) C (O) OMe CH2OCFThree
CH (Et) S (O) CH (Me) C (O) OMe CH2SMe
CH (Et) S (O) CH (Me) C (O) OMe CH2S (O) Me
CH (Et) S (O) CH (Me) C (O) OMe CH2S (O)2Me
CH (Et) S (O) CH (Me) C (O) OMe CH2SCFThree
CH (Et) S (O) CH (Me) C (O) OMe CH2S (O) CFThree
CH (Et) S (O) CH (Me) C (O) OMe CH2S (O)2CFThree
CH (Et) S (O) CH (Me) C (O) OMe CH2CH (OMe)2
CH (Et) S (O) CH (Me) C (O) OMe CH2CH (SMe)2
CH (Et) S (O) CH (Me) C (O) OMe CH2C (O) Me
CH (Et) S (O) CH (Me) C (O) OMe CH2C (O) CFThree
CH (Et) S (O) CH (Me) C (O) OMe CH2C (O) OMe
CH (Et) S (O)2CH (Me) C (O) OMe Me
CH (Et) S (O)2CH (Me) C (O) OEt Me
CH (Et) S (O)2CH (Me) C (O) OPr-n Me
CH (Et) S (O)2CH (Me) C (O) OPr-i Me
CH (Et) S (O)2CH (Me) C (O) OBu-n Me
CH (Et) S (O)2CH (Me) C (O) OBu-i Me
CH (Et) S (O)2CH (Me) C (O) OBu-t Me
CH (Et) S (O)2CH (Me) C (O) OPen-n Me
CH (Et) S (O)2CH (Me) C (O) OHex-n Me
CH (Et) S (O)2CH (Me) C (O) OMe Et
CH (Et) S (O)2CH (Me) C (O) OMe Pr-n
CH (Et) S (O)2CH (Me) C (O) OMe Pr-i
CH (Et) S (O)2CH (Me) C (O) OMe Pr-c
CH (Et) S (O)2CH (Me) C (O) OMe Bu-n
CH (Et) S (O)2CH (Me) C (O) OMe Bu-i
CH (Et) S (O)2CH (Me) C (O) OMe Bu-c
CH (Et) S (O)2CH (Me) C (O) OMe Bu-s
CH (Et) S (O)2CH (Me) C (O) OMe Bu-t
CH (Et) S (O)2CH (Me) C (O) OMe Pen-n
CH (Et) S (O)2CH (Me) C (O) OMe Pen-c
CH (Et) S (O)2CH (Me) C (O) OMe Hex-n
CH (Et) S (O)2CH (Me) C (O) OMe Hex-c
CH (Et) S (O)2CH (Me) C (O) OMe CH2Pr-c
CH (Et) S (O)2CH (Me) C (O) OMe CH2Bu-c
CH (Et) S (O)2CH (Me) C (O) OMe CH2Pen-c
CH (Et) S (O)2CH (Me) C (O) OMe CH2Hex-c
CH (Et) S (O)2CH (Me) C (O) OMe CH2CH = CH2
CH (Et) S (O)2CH (Me) C (O) OMe CH2CH = C (Cl)2
CH (Et) S (O)2CH (Me) C (O) OMe CH2C≡CH
CH (Et) S (O)2CH (Me) C (O) OMe CH2CN
CH (Et) S (O)2CH (Me) C (O) OMe CH2CFThree
CH (Et) S (O)2CH (Me) C (O) OMe CH2OMe
CH (Et) S (O)2CH (Me) C (O) OMe CH2OCFThree
CH (Et) S (O)2CH (Me) C (O) OMe CH2SMe
CH (Et) S (O)2CH (Me) C (O) OMe CH2S (O) Me
CH (Et) S (O)2CH (Me) C (O) OMe CH2S (O)2Me
CH (Et) S (O)2CH (Me) C (O) OMe CH2SCFThree
CH (Et) S (O)2CH (Me) C (O) OMe CH2S (O) CFThree
CH (Et) S (O)2CH (Me) C (O) OMe CH2S (O)2CFThree
CH (Et) S (O)2CH (Me) C (O) OMe CH2CH (OMe)2
CH (Et) S (O)2CH (Me) C (O) OMe CH2CH (SMe)2
CH (Et) S (O)2CH (Me) C (O) OMe CH2C (O) Me
CH (Et) S (O)2CH (Me) C (O) OMe CH2C (O) CFThree
CH (Et) S (O)2CH (Me) C (O) OMe CH2C (O) OMe
-------------------------------------------------- -
  The compounds of the present invention are stored in warehouses, so-called agricultural pests that harm agricultural and horticultural crops and trees, so-called livestock pests that parasitize livestock and poultry, so-called sanitary pests that cause various adverse effects in the human living environment such as houses. It is possible to effectively control insects such as so-called stored grain pests that harm cereals and the like, and pests such as mites, crustaceans, molluscs, and nematodes that occur and harm in similar situations at low concentrations.

本発明化合物を用いて防除しうる昆虫類、ダニ類、甲殻類、軟体動物及び線虫類には具体的に、例えば、下記の生物が挙げられるが、本発明はこれらのみに限定されるものではない。   Specific examples of insects, mites, crustaceans, molluscs and nematodes that can be controlled using the compounds of the present invention include the following organisms, but the present invention is not limited to these. is not.

チャノコカクモンハマキ(Adoxophyes honmai)、リンゴコカクモンハマキ(Adoxophyes orana faciata)、リンゴモンハマキ(Archips breviplicanus)、ミダレカクモンハマキ(Archips fuscocupreanus)、ナシヒメシンクイ(Grapholita molesta)、チャハマキ(Homona magnanima)、マメシンクイガ(Leguminivora glycinivorella)、マメヒメサヤムシガ(Matsumuraeses phaseoli)、トビハマキ(Pandemis heparana)、ナシチビガ(Bucculatrix pyrivorella)、モモハモグリガ(Lyonetia clerkella)、ギンモンハモグリガ(Lyonetia prunifoliella malinella)、チャノホソガ(Caloptilia theivora)、キンモンホソガ(Phyllonorycter ringoniella)、ミカンハモグリガ(Phyllocnistis citrella)、ネギコガ(Acrolepiopsis sapporensis)、ヤマノイモコガ(Acrolepiopsis suzukiella)、コナガ(Plutella xylostella)、カキノヘタムシガ(Stathmopoda masinissa)、イモキバガ(Helcystogramma triannulella)、ワタアカミムシ(Pectinophora gossypiella)、モモシンクイガ(Carposina sasakii)、コドリンガ(Cydla pomonella)、ニカメイガ(Chilo suppressalis)、コブノメイガ(Cnaphalocrocis medinalis)、モモノゴマダラノメイガ(Conogethes punctiferalis)、ワタヘリクロノメイガ(Diaphania indica)、シロイチモジマダラメイガ(Etiella zinckenella)、クワノメイガ(Glyphodes pyloalis)、ハイマダラノメイガ(Hellula undalis)、アワノメイガ(Ostrinia furnacalis)、アズキノメイガ(Ostrinia scapulalis)、ヨーロピアンコーンボーラー(Ostrinia nubilalis)、シバツトガ(Parapediasia teterrella)、イチモンジセセリ(Parnara guttata)、オオモンシロチョウ(Pieris brassicae)、モンシロチョウ(Pieris rapae crucivora)、ヨモギエダシャク(Ascotis selenaria)、ソイビーンルーパー(Pseudoplusia includens)、チャドクガ(Euproctis pseudoconspersa)、マイマイガ(Lymantria dispar)、ヒメシロモンドクガ(Orgyia thyellina)、アメリカシロヒトリ(Hyphantria cunea)、クワゴマダラヒトリ(Lemyra imparilis)、アケビコノハ(Adris tyrannus)、ナカジロシタバ(Aedia leucomelas)、タマナヤガ(Agrotis ipsilon)、カブラヤガ(Agrotis segetum)、タマナギンウワバ(Autographa nigrisigna)、ミツモンキンウワバ(Ctenoplusia agnata)、オオタバコガ(Helicoverpa armigera)、タバコガ(Helicoverpa assulta)、コットンボールワーム(Helicoverpa zea)、タバコバッドワーム(Heliothis virescens)、ヨトウガ(Mamestra brassicae)、アワヨトウ(Mythimna separata)、フタオビコヤガ(Naranga aenescens)、サザンアーミーワーム(Spodoptera eridania)、シロイチモジヨトウ(Spodoptera exigua)、フォールアーミーワーム(Spodoptera frugiperda)、コットンリーフワーム(Spodoptera littoralis)、ハスモンヨトウ(Spodoptera litura)、スジキリヨトウ(Spodoptera depravata)、イラクサギンウワバ(Trichoplusia ni)、グレープベリーモス(Endopiza viteana)、トマトホーンワーム(Manduca quinquemaculata)、タバコホーンワーム(Manduca sexta)等の鱗翅目昆虫。   Adoxophyes honmai, Adoxophyes orana faciata, Archips breviplicanus, Archips fuscocupreanus, Grapholita molesta, Chama magnan Leguminivora glycinivorella), Matsumuraeses phaseoli, Pandemis heparana, Bucculatrix pyrivorella, Lyonetia clerkella, Lyonetia prunifal ringoniella), mandarin leaf moth (Phyllocnistis citrella), green moth (Acrolepiopsis sapporensis), wild moth (Acrolepiopsis suzukiella), black moth (Plutella xylostella), oyster leaf moth (Stathmopoda masinissa), cystogram tria ora gossypiella), peach sinker moth (Carposina sasakii), codling moth (Cydla pomonella), green moth (Chilo suppressalis), corn borer (Cnaphalocrocis medinalis), peach moth (Conogethes punctiferalis), cotton moth (Dia) (Etiella zinckenella), Glyphodes pyloalis, Hellula undalis, Ostrinia furnacalis, Ostrinia scapulalis, European corn borer (Ostrinia nubilaliseter, Pesta pal) ), White-tailed butterfly (Pieris brassicae), white-tailed butterfly (Pieris rapae crucivora), mugwort (Ascotis selenaria), soy bean looper (Pseudoplusia includens), chadokuga (Euproctis pseudoconspersa), maimaiga (Lymantria disparia), thymeina ), White-spotted starfish (Hyphantria cunea), white-spotted starfish (Lemyra imparilis), Akebiko-no-ha (Adris tyrannus), red-footed butterfly (Aedia leucomelas), red-footed squirrel (Agrotis ipsilon), red-tailed squirrel (Agrotis segetum) Uwaba (Ctenoplusia agnata), Helicoverpa armigera, Tobacco moth (Helicoverpa assulta), Cotton ball worm (Helicoverpa zea), Tobacco bad worm (Heliothis virescens), Mamestra brassicae, Mythimna naa ), Southern army worm (Spodoptera eridania), Spodoptera exigua, Fall army worm (Spodoptera frugiperda), Cotton leaf worm (Spodoptera littoralis), Spodoptera litura, Spodoptera litura, Spodoptera era ), Leeb Berry Moss (Endopiza viteana), tomato horn worm (Manduca quinquemaculata), tobacco horn worm (Manduca sexta) lepidopteran insects such as.

ヒラズハナアザミウマ(Frankliniella intonsa)、ミカンキイロアザミウマ(Frankliniella occidentalis)、クロトンアザミウマ(Heliothrips haemorrhoidalis)、チャノキイロアザミウマ(Scirtothrips dorsalis)、ミナミキイロアザミウマ(Thrips palmi)、ネギアザミウマ(Thrips tabaci)、カキクダアザミウマ(Ponticulothrips diospyrosi)等の総翅目昆虫。   Thrips thrips (Frankliniella intonsa), Citrus thrips (Frankliniella occidentalis), Croton thrips (Prithia thrips) Moths in total.

ブチヒゲカメムシ(Dolycoris baccarum)、ナガメ(Eurydema rugosum)、トゲシラホシカメムシ(Eysarcoris aeneus)、オオトゲシラホシカメムシ(Eysarcoris lewisi)、シラホシカメムシ(Eysarcoris ventralis)、ツヤアオカメムシ(Glaucias subpunctatus)、クサギカメムシ(Halyomorpha halys)、アオクサカメムシ(Nezara antennata)、ミナミアオカメムシ(Nezara viridula)、イチモンジカメムシ(Piezodorus hybneri)、チャバネアオカメムシ(Plautia crossota)、イネクロカメムシ(Scotinophora lurida)、ホソハリカメムシ(Cletus punctiger)、クモヘリカメムシ(Leptocorisa chinensis)、ホソヘリカメムシ(Riptortus clavatus)、アカヒメヘリカメムシ(Rhopalus msculatus)、カンシャコバネナガカメムシ(Cavelerius saccharivorus)、コバネヒョウタンナガカメムシ(Togo hemipterus)、アカホシカメムシ(Dysdercus cingulatus)、ツツジグンバイ(Stephanitis pyrioides)、クロトビカスミカメ(Halticus insularis)、ターニッシュドプラントバグ(Lygus lineolaris)、ナガムギカスミカメ(Stenodema sibiricum)、アカスジカスミカメ(Stenotus rubrovittatus)、イネホソミドリカスミカメ(Trigonotylus caelestialium)、フタテンヒメヨコバイ(Arboridia apicalis)、ミドリナガヨコバイ(Balclutha saltuella)、フタテンオオヨコバイ(Epiacanthus stramineus)、ポテトリーフホッパー(Empoasca fabae)、カキノヒメヨコバイ(Empoasca nipponica)、チャノミドリヒメヨコバイ(Empoasca onukii)、マメノミドリヒメヨコバイ(Empoasca sakaii)、ヒメフタテンヨコバイ(Macrosteles striifrons)、ツマグロヨコバイ(Nephotettix cinctinceps)、コットンフリーホッパー(Psuedatomoscelis seriatus)、ヒメトビウンカ(Laodelphax striatella)、トビイロウンカ(Nilaparvata lugens)、セジロウンカ(Sogatella furcifera)、ミカンキジラミ(Diaphorina citri)、ナシキジラミ(Psylla pyrisuga)、ミカントゲコナジラミ(Aleurocanthus spiniferus)、シルバーリーフコナジラミ(Bemisia argentifolii)、タバココナジラミ(Bemisia tabaci)、ミカンコナジラミ(Dialeurodes citri)、オンシツコナジラミ(Trialeurodes vaporariorum)、ブドウネアブラムシ(Viteus vitifolii)、ワタアブラムシ(Aphis gossypii)、ユキヤナギアブラムシ(Aphis spiraecola)、モモアカアブラムシ(Myzus persicae)、コミカンアブラムシ(Toxoptera aurantii)、オオワラジカイガラムシ(Drosicha corpulenta)、イセリアカイガラムシ(Icerya purchasi)、ナスコナカイガラムシ(Phenacoccus solani)、ミカンコナカイガラムシ(Planococcus citri)、フジコナカイガラムシ(Planococcus kuraunhiae)、クワコナカイガラムシ(Pseudococcus comstocki)、ツノロウムシ(Ceroplastes ceriferus)、ルビーロウムシ(Ceroplastes rubens)、アカマルカイガラムシ(Aonidiella aurantii)、ナシマルカイガラムシ(Comstockaspis perniciosa)、ティースケール(Fiorinia theae)、チャノマルカイガラムシ(Pseudaonidia paeoniae)、クワシロカイガラムシ(Pseudaulacaspis pentagona)、ウメシロカイガラムシ(Pseudaulacaspis prunicola)、マサキナガカイガラムシ(Unaspis euonymi)、ヤノネカイガラムシ(Unaspis yanonensis)、トコジラミ(Cimex lectularius)等の半翅目昆虫。   Spotted beetle (Dolycoris baccarum), sea turtle (Eurydema rugosum), bark beetle (Eysarcoris aeneus), horseshoe beetle (Eysarcoris lewisi), white-headed beetle (Eysarcoris ventralis), subtilus , Nezara antennata, Nezara viridula, Piezodorus hybneri, Plautia crossota, Scotinophora lurida, tiger C Stink bug (Leptocorisa chinensis), Hoso-heli beetle (Riptortus clavatus), Red-headed beetle (Rhopalus msculatus), Cavelerius saccharivorus, Toba hemipterus cus, Togo hemipterus (Stephanitis pyrioides), Kuroto Bikasumi turtle (Halticus insularis), Turned plant bug (Lygus lineolaris), Nagamu sika turtle (Stenodema sibiricum), Akasika sika turtle (Stenotus rubrovittatus), Rice moss turtle (Trigonotylus caelestialium), ical Arisbori dia Green leafhopper (Balclutha saltuella), butterfly leafhopper (Epiacanthus stramineus), potato leaf hopper (Empoasca fabae), oyster leafhopper (Empoasca nipponica), Chanomidorimempei (Empoasca onukii), omenosaka ), Leafhopper leafhopper (Macrosteles striifrons), leafhopper leafhopper (Nephotettix cinctinceps), cotton-free hopper (Psuedatomoscelis seriatus), leafhopper (Laodelphax striatella), leafhopper (Nilaparvata lugens) Psylla pyrisuga, Aleurocanthus spiniferus, Silver leaf whitefly (Bemisia argentifolii), Tobacco whitefly (Bemisia tabaci), Citrus whitefly (Dialeurodes citri), Onsitsuna whitefly (trialeurous grape rum, Trialeurodes vapor Cotton Aphid (Aphis gossypii), Snowy Aphid (Aphis spiraecola), Peach Aphid (Myzus persicae), Komikan Aphid (Toxoptera aurantii), Alaska Scale Aphid (Drosicha corpulenta), Iceria scale P solani), citrus scale insect (Planococcus citri), stag beetle scale (Planococcus kuraunhiae), stag beetle scale (Pseudococcus comstocki), horn beetle (Ceroplastes ceriferus), ruby rotum (Ceroplastes rubens), red scallop Nymphalidae (Comstockaspis perniciosa), tea scale (Fiorinia theae), chanomarine scale insect (Pseudaonidia paeoniae), stag beetle (Pseudaulacaspis pentagona), scallop scale (Pseudaulacaspis prunicola), euglena (Unaspis yanonensis), Hemiptera (Cimex lectularius) and other Hemiptera insects.

ドウガネブイブイ(Anomala cuprea)、ヒメコガネ(Anomala rufocuprea)、コアオハナムグリ(Gametis jucunda)、ナガチャコガネ(Heptophylla picea)、マメコガネ(Popillia japonica)、コロラドポテトビートル(Lepinotarsa decemlineata)、マルクビクシコメツキ(Melanotus fortnumi)、カンシャクシコメツキ(Melanotus tamsuyensis)、タバコシバンムシ(Lasioderma serricorne)、ヒメヒラタケシキスイ(Epuraea domina)、インゲンテントウ(Epilachna varivestis)、ニジュウヤホシテントウ(Epilachna vigintioctopunctata)、チャイロコメノゴミムシダマシ(Tenebrio molitor)、コクヌストモドキ(Tribolium castaneum)、ゴマダラカミキリ(Anoplophora malasiaca)、マツノマダラカミキリ(Monochamus alternatus)、キボシカミキリ(Psacothea hilaris)、ブドウトラカミキリ(Xylotrechus pyrrhoderus)、アズキゾウムシ(Callosobruchus chinensis)、ウリハムシ(Aulacophora femoralis)、テンサイトビハムシ(Chaetocnema concinna)、サザンコーンルートワーム(Diabrotica undecimpunctata)、ウエスタンコーンルートワーム(Diabrotica virgifera)、ノーザンコーンルートワーム(Diabrotica barberi)、イネドロオイムシ(Oulema oryzae)、キスジノミハムシ(Phyllotreta striolata)、ナスナガスネトビハムシ(Psylliodes angusticollis)、モモチョッキリゾウムシ(Rhynchites heros)、アリモドキゾウムシ(Cylas formicarius)、ワタミゾウムシ(Anthonomus grandis)、イネゾウムシ(Echinocnemus squameus)、イモゾウムシ(Euscepes postfasciatus)、アルファルファタコゾウムシ(Hypera postica)、イネミズゾウムシ(Lissohoptrus oryzophilus)、キンケクチブトゾウムシ(Otiorhynchus sulcatus)、グラナリーウィービル(Sitophilus granarius)、コクゾウムシ(Sitophilus zeamais)、シバオサゾウムシ(Sphenophorus venatus vestitus)、アオバアリガタハネカクシ(Paederus fuscipes)等の鞘翅目昆虫。   Douganebubui (Anomala cuprea), Japanese common squirrel (Anomala rufocuprea), Core ohanamuri (Gametis jucunda), Nagachakogane (Heptophylla picea), Japanese beetle (Popillia japonica), Colorado potato beetle (Lepinotarsa decemlineata) White-footed beetle (Melanotus tamsuyensis), Tobacco beetle (Lasioderma serricorne), Himetaketakekisui (Epuraea domina), Green beetle (Epilachna varivestis), Nijuya-hoshi-tento (Epilachna vigintioctopunctata), T. Tribolium castaneum, Anoplophora malasiaca, Monochamus alternatus, Psacothea hilaris, Xylotrechus pyrrhoderus, callosobruchus, Callosobruchus Western Root beetle (Chaetocnema concinna), Southern corn root worm (Diabrotica undecimpunctata), Western corn root worm (Diabrotica virgifera), Northern corn root worm (Diabrotica barberi), Inedro beetle (Oulema oryzae), Phyllotreta nastriatum, Phyllotreta striol Tobet beetle (Psylliodes angusticollis), peach weevil (Rhynchites heros), aphid weevil (Cylas formicarius), cotton weevil (Anthonomus grandis), weevil (Echinocnemus squameus), weevil (Euscepes postfasciatus) Rice weevil (Lissohoptrus oryzophilus), horned weevil (Otiorhynchus sulcatus), granary weevil (Sitophilus granarius), hornet weevil (Sitophilus zeamais), bark weevil (Sphenophorus venatus vestitus moth) erus fuscipes).

ダイズサヤタマバエ(Asphondylia yushimai)、ムギアカタマバエ(Sitodiplosis mosellana)、ウリミバエ(Bactrocera cucurbitae)、ミカンコミバエ(Bactrocera dorsalis)、チチュウカイミバエ(Ceratitis capitata)、イネヒメハモグリバエ(Hydrellia griseola)、オウトウショウジョウバエ(Drosophila suzukii)、イネハモグリバエ(Agromyza oryzae)、ナモグリバエ(Chromatomyia horticola)、ナスハモグリバエ(Liriomyza bryoniae)、ネギハモグリバエ(Liriomyza chinensis)、トマトハモグリバエ(Liriomyza sativae)、マメハモグリバエ(Liriomyza trifolii)、タネバエ(Delia platura)、テンサイモグリハナバエ(Pegomya cunicularia)、アップルマゴット(Rhagoletis pomonella)、ヘシアンフライ(Mayetiola destructor)、イエバエ(Musca domestica)、サシバエ(Stomoxys calcitrans)、ヒツジシラミバエ(Melophagus ovinus)、ウシバエ(Hypoderma bovis)、キスジウシバエ(Hypoderma lineatum)、ヒツジバエ(Oestrus ovis)、ツェツェバエ(Glossina palpalis, Glossina morsitans)、キアシオオブユ(Prosimulium yezoensis)、ウシアブ(Tabanus trigonus)、オオチョウバエ(Telmatoscopus albipunctatus)、トクナガヌカカ(Leptoconops nipponensis)、アカイエカ(Culex pipiens pallens)、ネッタイシマカ(Aedes aegypti)、ヒトスジシマカ(Aedes albopicutus)、シナハマダラカ(Anopheles hyracanus sinesis)等の双翅目昆虫。   Soybean flies (Asphondylia yushimai), mud wings (Sitodiplosis mosellana), fruit flies (Bactrocera cucurbitae), citrus fruit flies (Bactrocera dorsalis), citrus fruit flies (Ceratitis capitata), rice moth flies Leafhopper (Agromyza oryzae), Leafworm (Chromatomyia horticola), Eggplant leaffly (Liriomyza bryoniae), Leafhopper (Liriomyza chinensis), Tomato leaffly (Liriomyza sativae), Beanworm (Liriomyza trifoli), Liriomyza trifoli (Pegomya cunicularia), apple haggot (Rhagoletis pomonella), hessian fly (Mayetiola destructor), housefly (Musca domestica), barn fly (Stomoxys calcitrans), sheep flies (Melophagus ovinus), bullflies (Hypoderma bovisma), , Sheep flies (Oestrus ovis), tsetse flies (Glossina palpalis, Glossina morsitans), black-headed ayu (Prosimulium yezoensis), bullfly (Tabanus trigonus), giant fly (Telmatoscopus albipunctatus), nipponen sip (Leptocons) Diptera, such as Aedes aegypti, Aedes albopicutus, Anopheles hyracanus sinesis.

クリハバチ(Apethymus kuri)、カブラハバチ(Athalia rosae)、チュウレンジハバチ(Arge pagana)、マツノキハバチ(Neodiprion sertifer)、クリタマバチ(Dryocosmus kuriphilus)、グンタイアリ(Eciton burchelli, Eciton schmitti)、クロオオアリ(Camponotus japonicus)、オオスズメバチ(Vespa mandarina)、ブルドックアント(Myrmecia spp.)、ファイヤーアント類(Solenopsis spp.)、ファラオアント(Monomorium pharaonis)等の膜翅目昆虫。   Bumblebee (Apethymus kuri), Bumblebee (Athalia rosae), Bumblebee (Arge pagana), Bumblebee (Neodiprion sertifer), Bumblebee (Dryocosmus kuriphilus), Gantai (Eciton burchelli, Eciton schmitus), Eciton burchelli, Eciton schmitus Hymenoptera insects such as mandarina, bulldog ant (Myrmecia spp.), fire ant (Solenopsis spp.), pharaoh ant (Monomorium pharaonis).

エンマコオロギ(Teleogryllus emma)、ケラ(Gryllotalpa orientalis)、トノサマバッタ(Locusta migratoria)、コバネイナゴ(Oxya yezoensis)、サバクワタリバッタ(Schistocerca gregaria)等の直翅目昆虫。   Straight-legged insects such as Teleogryllus emma, Gryllotalpa orientalis, Locusta migratoria, Oxya yezoensis, Schistocerca gregaria and others.

トゲナシシロトビムシ(Onychiurus folsomi)、シベリアシロトビムシ(Onychiurus sibiricus)、キボシマルトビムシ(Bourletiella hortensis)等の粘管目昆虫。   Coleoptera insects such as Onychiurus folsomi, Onychiurus sibiricus and Bourletiella hortensis.

クロゴキブリ(Periplaneta fuliginosa)、ヤマトゴキブリ(Periplaneta japonica)、チャバネゴキブリ(Blattella germanica)等の網翅目昆虫。   Reticulate insects such as black cockroach (Periplaneta fuliginosa), cockroach (Periplaneta japonica), German cockroach (Blattella germanica).

イエシロアリ(Coptotermes formosanus)、ヤマトシロアリ(Reticulitermes speratus)、タイワンシロアリ(Odontotermes formosanus)等のシロアリ目昆虫。   Termite insects such as termites (Coptotermes formosanus), Yamato termites (Reticulitermes speratus), Taiwan termites (Odontotermes formosanus).

ネコノミ(Ctenocephalidae felis)、イヌノミ(Ctenocephalides canis)、ニワトリノミ(Echidnophaga gallinacea)、ヒトノミ(Pulex irritans)、ケオプスネズミノミ(Xenopsylla cheopis)等の等翅目昆虫。   Coleopterous insects such as cat fleas (Ctenocephalidae felis), dog fleas (Ctenocephalides canis), chicken fleas (Echidnophaga gallinacea), human fleas (Pulex irritans), keops rat fleas (Xenopsylla cheopis) and the like.

ニワトリオオハジラミ(Menacanthus stramineus)、ウシハジラミ(Bovicola bovis)等のハジラミ目昆虫。   White-headed insects such as chicken lice (Menacanthus stramineus) and bovine lice (Bovicola bovis).

ウシジラミ(Haematopinus eurysternus)、ブタジラミ(Haematopinus suis)、ウシホソジラミ(Linognathus vituli)、ケブカウシジラミ(Solenopotes capillatus)等のシラミ目昆虫。   Louse insects such as cattle lice (Haematopinus eurysternus), pig lice (Haematopinus suis), cattle white lice (Linognathus vituli), horned lice (Solenopotes capillatus) and the like.

シクラメンホコリダニ(Phytonemus pallidus)、チャノホコリダニ(Polyphagotarsonemus latus)、スジブトホコリダニ(Tarsonemus bilobatus)等のホコリダニ類。   Dust mites such as cyclamen dust mite (Phytonemus pallidus), chano dust mite (Polyphagotarsonemus latus), and Sudabuto dust mite (Tarsonemus bilobatus).

ハクサイダニ(Penthaleus erythrocephalus)、ムギダニ(Penthaleus major)等のハシリダニ類。   Spider mites such as cabbage mite (Penthaleus erythrocephalus) and wheat mite (Penthaleus major).

イネハダニ(Oligonychus shinkajii)、ミカンハダニ(Panonychus citri)、クワオオハダニ(Panonychus mori)、リンゴハダニ(Panonychus ulmi)、カンザワハダニ(Tetranychus kanzawai)、ナミハダニ(Tetranychus urticae)等のハダニ類。   Spider mites such as rice spider mite (Oligonychus shinkajii), citrus spider mite (Panonychus citri), blue spider mite (Panonychus mori), apple spider mite (Panonychus ulmi), Kanzawa spider mite (Tetranychus kanzawai), spider mite (Tetranychus urticae), etc.

チャノナガサビダニ(Acaphylla theavagrans)、チューリップサビダニ(Aceria tulipae)、トマトサビダニ(Aculops lycopersici)、ミカンサビダニ(Aculops pelekassi)、リンゴサビダニ(Aculus schlechtendali)、ニセナシサビダニ(Eriophyes chibaensis)、シトラスラストマイト(Phyllocoptruta oleivora)等のフシダニ類。   Chinese cabbage mite (Acaphylla theavagrans), tulip rust mite (Aceria tulipae), tomato rust mite (Aculops lycopersici), citrus red mite (Aculops pelekassi), apple rust mite (Aculus schlechtendali), black rust mite (Eriophyes chitrastrostrum) ) Etc.

ロビンネダニ(Rhizoglyphus robini)、ケナガコナダニ(Tyrophagus putrescentiae)、ホウレンソウケナガコナダニ(Tyrophagus similis)等のコナダニ類。   Acarids such as Robin tick (Rhizoglyphus robini), Tyrophagus putrescentiae, and Tyrophagus similis.

ミツバチヘギイタダニ(Varroa jacobsoni)等のハチダニ類。   Bee mites such as honeybee mite (Varroa jacobsoni).

オウシマダニ(Boophilus microplus)、クリイロコイタマダニ(Rhipicephalus sanguineus)、フタトゲチマダニ(Haemaphysalis longicornis)、キチマダニ(Haemophysalis flava)、ツリガネチマダニ(Haemophysalis campanulata)、ヤマトマダニ(Ixodes ovatus)、シュルツェマダニ(Ixodes persulcatus)、オオマダニ(Amblyomma spp.)、アミメマダニ(Dermacentor spp.)等のマダニ類。   Tick tick (Boophilus microplus), Rhipicephalus sanguineus, Tick tick (Haemaphysalis longicornis), Tick tick (Haemophysalis flava), Tick tick (Haemophysalis campanulata), Tick tick (Ixo tus tick) Tick such as Amblyomma spp.), Dermacentor spp.

イヌツメダニ(Cheyletiella yasguri)、ネコツメダニ(Cheyletiella blakei)等のツメダニ類。   Crawling ticks, such as the crayfish tick (Cheyletiella yasguri) and the cat crawfish tick (Cheyletiella blakei).

イヌニキビダニ(Demodex canis)、ネコニキビダニ(Demodex cati)などのニキビダニ類。   Acne mites, such as Inodex canis and Demodex cati.

ヒツジキュウセンダニ(Psoroptes ovis)等のキュウセンダニ類。   Cucumber mites such as sheep cucumber mites (Psoroptes ovis).

センコウヒゼンダニ(Sarcoptes scabiei)、ネコショウセンコウヒゼンダニ(Notoedres cati)、ニワトリヒゼンダニ(Knemidocoptes spp.)等のヒゼンダニ類。   Spider mites, such as Sarcoptes scabiei, Notoedres cati, and Knemidocoptes spp.

オカダンゴムシ(Armadillidium vulgare)等の甲殻類。   Crustacea such as Armadillidium vulgare.

スクミリンゴガイ(Pomacea canaliculata)、アフリカマイマイ(Achatina fulica)、ナメクジ(Meghimatium bilineatum)、チャコウラナメクジ(Limax Valentiana)、ウスカワマイマイ(Acusta despecta sieboldiana)、ミスジマイマイ(Euhadra peliomphala)等の腹足類。   Gastropods such as Pomacea canaliculata, African mussel (Achatina fulica), Slug (Meghimatium bilineatum), Chaukoura slug (Limax Valentiana), Uskawamai (Acusta despecta sieboldiana), Mishamai mai (Euhadra peliomphala).

ミナミネグサレセンチュウ(Prathylenchus coffeae)、キタネグサレセンチュウ(Prathylenchus penetrans)、クルミネグサレセンチュウ(Prathylenchus vulnus)、ジャガイモシストセンチュウ(Globodera rostochiensis)、ダイズシストセンチュウ(Heterodera glycines)、キタネコブセンチュウ(Meloidogyne hapla)、サツマイモネコブセンチュウ(Meloidogyne incognita)、イネシンガレセンチュウ(Aphelenchoides besseyi)、マツノザイセンチュウ(Bursaphelenchus xylophilus)等の線虫類。   Southern nematode nematode (Prathylenchus coffeae), Kitane-negususa nematode (Prathylenchus penetrans), Kurume rushes nematode (Prathylenchus vulnus), potato cyst nematode (Globodera rostochiensis), soybean cyst nematode (Heterodera lypter Nematodes such as root-knot nematodes (Meloidogyne incognita), rice-spotted nematodes (Aphelenchoides besseyi), and pine wood nematodes (Bursaphelenchus xylophilus).

また、本発明化合物を用いて防除しうる家畜、家禽、愛玩動物等の内部寄生虫としては具体的に、例えば、下記の生物が挙げられるが、本発明はこれらのみに限定されるものではない。   In addition, specific examples of endoparasites such as livestock, poultry, and pet animals that can be controlled using the compounds of the present invention include the following organisms, but the present invention is not limited to these. .

ヘモンクス属(Haemonchus)、トリコストロンギルス属(Trichostrongylus)、オステルターギヤ属(Ostertagia)、ネマトディルス属(Nematodirus)、クーペリア属(Cooperia)、アスカリス属(Ascaris)、ブノストムーム属(Bunostomum)、エスファゴストムーム属(Oesophagostomum)、チャベルチア属(Chabertia)、トリキュリス属(Trichuris)、ストロンギルス属(Storongylus)、トリコネマ属(Trichonema)、ディクチオカウルス属(Dictyocaulus)、キャピラリア属(Capillaria)、ヘテラキス属(Heterakis)、トキソカラ属(Toxocara)、アスカリディア属(Ascaridia)、オキシウリス属(Oxyuris)、アンキロストーマ属(Ancylostoma)、ウンシナリア属(Uncinaria)、トキサスカリス属(Toxascaris)、パラスカリス属(Parascaris)などの線虫類、
ブツヘレリア属(Wuchereria)、ブルージア属(Brugia)、オンコセルカ属(Onchoceca)、ディロフィラリア属(Dirofilaria)、ロア糸状虫属(Loa)などのフィラリア科(Filariidae)線虫類。
Haemonchus, Trichostrongylus, Ostertagia, Nematodirus, Cooperia, Ascaris, Bunostomum, Esphagostomum Genus (Oesophagostomum), Chabertia, Trichuris, Strongylus, Trichonema, Dictyocaulus, Capillaria, Heterakis ), Toxocara, Ascaridia, Oxyuris, Ancylostoma, Uncinaria, Toxacaris, Parascaris, and other nematodes ,
Filariidae nematodes such as Wuchereria, Blueia, Onchoceca, Dirofilaria and Loa.

ドラクンクルス属(Deacunculus)などの蛇状線虫科(Dracunculidae)線虫類。   Dracunculidae nematodes, such as the genus Deacunculus.

犬条虫(Dipylidium caninum)、猫条虫(Taenia taeniaeformis)、有鉤条虫(Taenia solium)、無鉤条虫(Taenia saginata)、縮小条虫(Hymenolepis diminuta)、ベネデン条虫(Moniezia benedeni)、広節裂頭条虫(Diphyllobothrium latum)、マンソン裂頭条虫(Diphyllobothrium erinacei)、単包条虫(Echinococcus granulosus)、多包条虫(Echinococcus multilocularis)などの条虫類。   Dogworms (Dipylidium caninum), caterpillars (Taenia taeniaeformis), rodents (Taenia solium), striped tapeworms (Taenia saginata), contracted tapeworms (Hymenolepis diminuta), Beneden tapeworms (Moniezia benedeni), Tapeworms such as Diphyllobothrium latum, Manson cleftworm (Diphyllobothrium erinacei), Echinococcus granulosus, Echinococcus multilocularis.

肝蛭(Fasciola hepatica,F.gigantica)、ウエステルマン肺吸虫(Paragonimus westermanii)、肥大吸虫(Fasciolopsic bruski)、膵吸虫(Eurytrema pancreaticum,E.coelomaticum)、肝吸虫(Clonorchis sinensis)、日本住血吸虫(Schistosoma japonicum)、ビルハルツ住血吸虫(Schistosoma haematobium)、マンソン住血吸虫(Schistosoma mansoni)などの吸虫類。   Fasciola hepatica (F. gigantica), Westermann lung fluke (Paragonimus westermanii), hypertrophic fluke (Fasciolopsic bruski), pancreatic fluke (Eurytrema pancreaticum, E. coelomaticum), liver fluke (Clonorchis sinensis), Schistosoma Schistosoma japonicum), Schistosoma haematobium, Schistosoma mansoni, etc.

エイメリア・テネラ(Eimeria tenella)、エイメリア・アセルブリナ(Eimeria acervulina)、エイメリア・ブルネッチ(Eimeria brunetti)、エイメリア・マクシマ(Eimeria maxima)、エイメリア・ネカトリクス(Eimeria necatrix)、エイメリア・ボビス(Eimeria bovis)、エイメリア・オビノイダリス(Eimeria ovinoidalis)のようなエイメリア類(Eimeria spp.)。   Eimeria tenella, Eimeria acervulina, Eimeria brunetti, Eimeria maxima, Eimeria necatrix, Eimeria bovis, Eimeria bovis Eimeria spp., Such as Eimeria ovinoidalis.

クルーズトリパノソーマ(Trypanosomsa cruzi)、リーシュマニア類(Leishmania spp.)、マラリア原虫(Plasmodium spp.)、バベシア類(Babesis spp.)、トリコモナス類(Trichomonadidae spp.)、ヒストモナス類(Histomanas spp.)、ジアルディア類(Giardia spp.)、トキソプラズマ類(Toxoplasma spp.)、赤痢アメーバ(Entamoeba histolytica)、タイレリア類(Theileria spp.)。   Trypanosomsa cruzi, Leishmania spp., Plasmodium spp., Babesis spp., Trichomonadidae spp., Histomanas spp., Giardia (Giardia spp.), Toxoplasma spp., Entamoeba histolytica, Theileria spp.

さらに、本発明化合物は、有機燐系化合物、カーバメート系化合物又はピレスロイド系化合物等の既存の殺虫剤に対して抵抗性の発達した有害生物に対しても有効である。   Furthermore, the compound of the present invention is also effective against pests that have developed resistance to existing insecticides such as organophosphorus compounds, carbamate compounds, and pyrethroid compounds.

すなわち、本発明化合物は、粘管目(トビムシ目)、網翅目(ゴキブリ目)、直翅目(バッタ目)、シロアリ目、総翅目(アザミウマ目)、半翅目(カメムシ目及びヨコバイ目)、鱗翅目(チョウ目)、鞘翅目(コウチュウ目)、膜翅目(ハチ目)、双翅目(ハエ目)、等翅目(ノミ目)及びシラミ目等の昆虫類、ダニ類、腹足類及び線虫類等に属する有害生物を低濃度で有効に防除することが出来る。一方、本発明化合物はホ乳類、魚類、甲殻類及び益虫(ミツバチ、マルハナバチ等の有用昆虫やツヤコバチ、アブラバチ、ヤドリバエ、ヒメハナカメムシ、カブリダニ等の天敵)に対してほとんど悪影響の無い極めて有用な特長を有している。   That is, the compound of the present invention is composed of the order of mucous eyes (Coleoptera), reticulates (Roaches), straight moths (Grasshoppers), termites, common moths (Thrips), hemimorphs (stink bugs and leafhoppers). Eyes), Lepidoptera (Lepidoptera), Coleoptera (Coleoptera), Hymenoptera (Hymenoptera), Diptera (Flyidae), Islamic (Flea), Liceid, and other insects, ticks In addition, pests belonging to gastropods and nematodes can be effectively controlled at low concentrations. On the other hand, the compounds of the present invention are extremely useful with little adverse effect on mammals, fish, crustaceans and beneficial insects (beneficial insects such as bees and bumblebees, natural enemies such as honeybees, wasps, mistletoe flies, mosquitoes, and mites). Has features.

本発明化合物を使用するにあたっては、通常適当な固体担体又は液体担体と混合し、更に所望により界面活性剤、浸透剤、展着剤、増粘剤、凍結防止剤、結合剤、固結防止剤、崩壊剤、消泡剤、防腐剤および分解防止剤等を添加して、液剤(soluble concentrate)、乳剤(emulsifiable concentrate)、水和剤(wettable powder)、水溶剤(water soluble powder)、顆粒水和剤(water dispersible granule)、顆粒水溶剤(water soluble granule)、懸濁剤(suspension concentrate)、乳濁剤(concentrated emulsion)、サスポエマルジョン(suspoemulsion)、マイクロエマルジョン(microemulsion)、粉剤(dustable powder)、粒剤(granule)錠剤(tablet)および乳化性ゲル剤(emulsifiable gel)等任意の剤型の製剤にて実用に供することができる。また、省力化および安全性向上の観点から、上記任意の剤型の製剤を、水溶性カプセルおよび水溶性フィルムの袋等の水溶性包装体に封入して供することもできる。   When using the compound of the present invention, it is usually mixed with a suitable solid carrier or liquid carrier, and if desired, a surfactant, penetrant, spreading agent, thickener, antifreezing agent, binder, anti-caking agent. , Disintegrating agents, antifoaming agents, preservatives and anti-degradation agents, etc., and soluble concentrate, emulsion (emulsifiable concentrate), wettable powder, water-soluble powder, granular water Water dispersible granule, water soluble granule, suspension concentrate, concentrated emulsion, suspoemulsion, microemulsion, dustable powder ), Granule tablets, and emulsifiable gels, and can be put to practical use. Further, from the viewpoint of labor saving and safety improvement, the preparations of any of the above dosage forms can be provided by being enclosed in a water-soluble package such as a water-soluble capsule and a bag of a water-soluble film.

固体担体としては、例えば石英、方解石、海泡石、ドロマイト、チョーク、カオリナイト、パイロフィライト、セリサイト、ハロサイト、メタハロサイト、木節粘土、蛙目粘土、陶石、ジークライト、アロフェン、シラス、きら、タルク、ベントナイト、活性白土、酸性白土、軽石、アタパルジャイト、ゼオライトおよび珪藻土等の天然鉱物質、例えば焼成クレー、パーライト、シラスバルーン、バーミキュライト、アタパルガスクレーおよび焼成珪藻土等の天然鉱物質の焼成品、例えば炭酸マグネシウム、炭酸カルシウム、炭酸ナトリウム、炭酸水素ナトリウム、硫酸アンモニウム、硫酸ナトリウム、硫酸マグネシウム、リン酸水素二アンモニウム、リン酸二水素アンモニウムおよび塩化カリウム等の無機塩類、例えばブドウ糖、果糖、しょ糖および乳糖などの糖類、例えば澱粉、粉末セルロースおよびデキストリン等の多糖類、例えば尿素、尿素誘導体、安息香酸および安息香酸の塩等の有機物、例えば木粉、コルク粉、トウモロコシ穂軸、クルミ殻およびタバコ茎等の植物類、フライアッシュ、ホワイトカーボン(例えば、含水合成シリカ、無水合成シリカおよび含水合成シリケート等)ならびに肥料等が挙げられる。   Examples of the solid carrier include quartz, calcite, gypsum, dolomite, chalk, kaolinite, pyrophyllite, sericite, halosite, metahalosite, kibushi clay, glazed clay, porcelain stone, siegrite, and allophane. Natural minerals such as shirasu, kira, talc, bentonite, activated clay, acid clay, pumice, attapulgite, zeolite and diatomaceous earth, for example, calcined clay, perlite, shirasu balloon, vermiculite, attapulgus clay and calcined diatomaceous earth Baked products such as magnesium carbonate, calcium carbonate, sodium carbonate, sodium bicarbonate, ammonium sulfate, sodium sulfate, magnesium sulfate, diammonium hydrogen phosphate, ammonium dihydrogen phosphate and potassium chloride, such as glucose, fructose , And Sugars such as sugar and lactose, polysaccharides such as starch, powdered cellulose and dextrin, organic materials such as urea, urea derivatives, benzoic acid and benzoic acid salts, such as wood flour, cork flour, corn cobs, walnut shells and Examples include plants such as tobacco stalks, fly ash, white carbon (for example, hydrous synthetic silica, anhydrous synthetic silica, hydrous synthetic silicate, etc.) and fertilizers.

液体担体としては、例えばキシレン、アルキル(C9又はC10等)ベンゼン、フェニルキシリルエタンおよびアルキル(C1又はC3等)ナフタレン等の芳香族炭化水素類、マシン油、ノルマルパラフィン、イソパラフィンおよびナフテン等の脂肪族炭化水素類、ケロシン等の芳香族炭化水素と脂肪族炭化水素の混合物、エタノール、イソプロパノール、シクロヘキサノール、フェノキシエタノールおよびベンジルアルコール等のアルコール、エチレングリコール、プロピレングリコール、ジエチレングリコール、ヘキシレングリコール、ポリエチレングリコールおよびポリプロピレングリコール等の多価アルコール、プロピルセロソルブ、ブチルセロソルブ、フェニルセロソルブ、プロピレングリコールモノメチルエーテル、プロピレングリコールモノエチルエーテル、プロピレングリコールモノプロピルエーテル、プロピレングリコールモノブチルエーテルおよびプロピレングリコールモノフェニルエーテル等のエーテル、アセトフェノン、シクロヘキサノンおよびγ−ブチロラクトン等のケトン、脂肪酸メチルエステル、コハク酸ジアルキルエステル、グルタミン酸ジアルキルエステル、アジピン酸ジアルキルエステルおよびフタル酸ジアルキルエステル等のエステル、N−アルキル(C1、C8又はC12等)ピロリドン等の酸アミド、大豆油、アマニ油、ナタネ油、ヤシ油、綿実油およびヒマシ油等の油脂、ジメチルスルホキシドならびに水が挙げられる。 Examples of the liquid carrier include xylene, alkyl (C 9 or C 10 etc.) benzene, phenyl xylyl ethane and alkyl (C 1 or C 3 etc.) naphthalene and other aromatic hydrocarbons, machine oil, normal paraffin, isoparaffin and Aliphatic hydrocarbons such as naphthene, mixtures of aromatic and aliphatic hydrocarbons such as kerosene, alcohols such as ethanol, isopropanol, cyclohexanol, phenoxyethanol and benzyl alcohol, ethylene glycol, propylene glycol, diethylene glycol, hexylene glycol , Polyhydric alcohols such as polyethylene glycol and polypropylene glycol, propyl cellosolve, butyl cellosolve, phenyl cellosolve, propylene glycol monomethyl ether, propylene glycol Ethers such as ethyl monoethyl ether, propylene glycol monopropyl ether, propylene glycol monobutyl ether and propylene glycol monophenyl ether, ketones such as acetophenone, cyclohexanone and γ-butyrolactone, fatty acid methyl esters, dialkyl esters of succinic acid, dialkyl esters of glutamic acid, adipine esters such as dialkyl ester and dialkyl phthalate esters, N- alkyl (C 1, C 8 or C 12, etc.) acid amide pyrrolidone, soybean oil, linseed oil, rapeseed oil, coconut oil, such as cottonseed oil and castor oil Examples include fats and oils, dimethyl sulfoxide and water.

これら固体および液体担体は、単独で用いても2種以上を併用してもよい。   These solid and liquid carriers may be used alone or in combination of two or more.

界面活性剤としては、例えばポリオキシエチレンアルキルエーテル、ポリオキシエチレンアルキル(モノ又はジ)フェニルエーテル、ポリオキシエチレン(モノ、ジ又はトリ)スチリルフェニルエーテル、ポリオキシエチレンポリオキシプロピレンブロックコポリマー、ポリオキシエチレン脂肪酸(モノ又はジ)エステル、ソルビタン脂肪酸エステル、ポリオキシエチレンソルビタン脂肪酸エステル、ヒマシ油エチレンオキサイド付加物、アセチレングリコール、アセチレンアルコール、アセチレングリコールのエチレンオキサイド付加物、アセチレンアルコールのエチレンオキサイド付加物およびアルキルグリコシド等のノニオン性界面活性剤、アルキル硫酸エステル塩、アルキルベンゼンスルホン酸塩、リグニンスルホン酸塩、アルキルスルホコハク酸塩、ナフタレンスルホン酸塩、アルキルナフタレンスルホン酸塩、ナフタレンスルホン酸のホルマリン縮合物の塩、アルキルナフタレンスルホン酸のホルマリン縮合物の塩、ポリオキシエチレンアルキルエーテル硫酸又は燐酸エステル塩、ポリオキシエチレン(モノ又はジ)アルキルフェニルエーテル硫酸又は燐酸エステル塩、ポリオキシエチレン(モノ、ジ又はトリ)スチリルフェニルエーテル硫酸又は燐酸エステル塩、ポリカルボン酸塩(例えば、ポリアクリル酸塩、ポリマレイン酸塩およびマレイン酸とオレフィンとの共重合物等)およびポリスチレンスルホン酸塩等のアニオン性界面活性剤、アルキルアミン塩およびアルキル4級アンモニウム塩等のカチオン性界面活性剤、アミノ酸型およびベタイン型等の両性界面活性剤、シリコーン系界面活性剤ならびにフッ素系界面活性剤が挙げられる。   Examples of the surfactant include polyoxyethylene alkyl ether, polyoxyethylene alkyl (mono or di) phenyl ether, polyoxyethylene (mono, di or tri) styryl phenyl ether, polyoxyethylene polyoxypropylene block copolymer, polyoxyethylene Ethylene fatty acid (mono or di) ester, sorbitan fatty acid ester, polyoxyethylene sorbitan fatty acid ester, castor oil ethylene oxide adduct, acetylene glycol, acetylene alcohol, ethylene oxide adduct of acetylene glycol, ethylene oxide adduct of acetylene alcohol and alkyl Nonionic surfactants such as glycosides, alkyl sulfate esters, alkylbenzene sulfonates, lignin sulfonates, alkyls Rufosuccinate, naphthalene sulfonate, alkyl naphthalene sulfonate, salt of formalin condensate of naphthalene sulfonic acid, salt of formalin condensate of alkyl naphthalene sulfonic acid, polyoxyethylene alkyl ether sulfate or phosphate ester salt, polyoxyethylene (Mono or di) alkyl phenyl ether sulfate or phosphate ester salt, polyoxyethylene (mono, di or tri) styryl phenyl ether sulfate or phosphate ester salt, polycarboxylate (eg polyacrylate, polymaleate and maleate) Copolymer of acid and olefin, etc.) and anionic surfactants such as polystyrene sulfonate, cationic surfactants such as alkylamine salts and alkyl quaternary ammonium salts, and amphoteric interfaces such as amino acid type and betaine type Sexual agents, silicone-based surfactants and fluorinated surfactants.

これら界面活性剤の含有量は、特に限定されるものではないが、本発明の製剤100重量部に対し、通常0.05〜20重量部の範囲が望ましい。また、これら界面活性剤は、単独で用いても2種以上を併用してもよい。   The content of these surfactants is not particularly limited, but is usually preferably in the range of 0.05 to 20 parts by weight with respect to 100 parts by weight of the preparation of the present invention. These surfactants may be used alone or in combination of two or more.

本発明化合物の施用薬量は適用場面、施用時期、施用方法、栽培作物等により差異は有るが、一般には有効成分量としてヘクタール(ha)当たり0.005〜50kg程度が適当である。   The application amount of the compound of the present invention varies depending on the application scene, application time, application method, cultivated crops, etc., but generally 0.005 to 50 kg per hectare (ha) is appropriate as the amount of active ingredient.

一方、家畜及び愛玩動物としての哺乳動物および鳥類の外部又は内部寄生虫の防除に本発明化合物を使用するにあたっては、有効量の本発明化合物を製剤用添加物とともに経口投与、注射(筋肉内、皮下、静脈内、腹腔内)などの非経口投与;浸漬、スプレー、入浴、洗浄、滴下(pouring-on)およびスポッティング(spotting-on)並びにダスティング(dusting)などの経皮投与;経鼻投与により投与することができる。本発明化合物はまた、細片、プレート、バンド、カラー、イヤー・マーク(ear mark)、リム(limb)・バンド、標識装置などを用いた成形製品により投与することができる。投与にあたっては本発明化合物を投与経路に適した任意の剤型とすることができる。   On the other hand, when using the compound of the present invention for the control of the ectoparasites of mammals and birds as domestic animals and pets, an effective amount of the compound of the present invention is administered orally together with injection additives (intramuscular, Parenteral administration such as subcutaneous, intravenous, intraperitoneal; transdermal administration such as immersion, spraying, bathing, washing, pouring-on and spotting-on and dusting; nasal administration Can be administered. The compounds of the present invention can also be administered by molded products using strips, plates, bands, collars, ear marks, limb bands, labeling devices and the like. In administration, the compound of the present invention can be in any dosage form suitable for the administration route.

調製される任意の剤型としては、粉剤、粒剤、水和剤、ペレット、錠剤、大丸薬、カプセル剤、活性化合物を含む成形製品などの固体調製物;注射用液剤、経口用液剤、皮膚上又は体腔中に用いる液剤;滴下(Pour-on)剤、点下(Spot-on)剤、フロアブル剤、乳剤などの溶液調製物;軟膏剤、ゲルなどの半固体調製物などが挙げられる。   Arbitrary forms to be prepared include solid preparations such as powders, granules, wettable powders, pellets, tablets, large pills, capsules, molded products containing active compounds; injection solutions, oral solutions, skin Liquid preparations used above or in body cavities; solution preparations such as Pour-on agents, spot-on agents, flowable agents and emulsions; semi-solid preparations such as ointments and gels.

固体調製物は、主に経口投与あるいは水などで希釈して経皮投与にあるいは環境処理にて用いることができる。固体調製物は、活性化合物を必要ならば補助剤を加えて適当な賦形剤と共に混合し、そして所望の形状に変えることにより調製できる。適当な賦形剤としては、例えば炭酸塩、炭酸水素塩、リン酸塩、酸化アルミニウム、シリカ、粘土などの無機物質、糖、セルロース、粉砕された穀物、澱粉などの有機物質がある。   The solid preparation can be used mainly for oral administration or diluted with water for transdermal administration or environmental treatment. Solid preparations can be prepared by adding the active compound, if necessary, with adjuncts, mixing with appropriate excipients, and converting to the desired shape. Suitable excipients include, for example, inorganic substances such as carbonates, bicarbonates, phosphates, aluminum oxides, silicas, clays, and organic substances such as sugars, cellulose, crushed grains, and starches.

注射用液剤は、静脈内、筋肉内および皮下に投与できる、注射用液剤は、活性化合物を適当な溶媒に溶解させ、そして必要ならば可溶化剤、酸、塩基、緩衝用塩、酸化防止剤および保護剤などの添加剤を加えることにより調製できる。適当な溶媒としては、水、エタノール、ブタノール、ベンジルアルコール、グリセリン、プロピレングリコール、ポリエチレングリコール、N−メチルピロリドン並びにこれらの混合物、生理学的に許容しうる植物油、注射に適する合成油などがあげられる。可溶化剤としては、ポリビニルピロリドン、ポリオキシエチル化されたヒマシ油およびポリオキシエチル化されたソルビタンエステルなどがあげられる。保護剤には、ベンジルアルコール、トリクロロブタノール、p−ヒドロキシ安息香酸エステルおよびn−ブタノールなどがある。   Injection solutions can be administered intravenously, intramuscularly and subcutaneously. Injection solutions dissolve the active compound in a suitable solvent and, if necessary, solubilizers, acids, bases, buffer salts, antioxidants. And can be prepared by adding additives such as protective agents. Suitable solvents include water, ethanol, butanol, benzyl alcohol, glycerin, propylene glycol, polyethylene glycol, N-methylpyrrolidone and mixtures thereof, physiologically acceptable vegetable oils, synthetic oils suitable for injection, and the like. Examples of solubilizers include polyvinylpyrrolidone, polyoxyethylated castor oil, and polyoxyethylated sorbitan ester. Protecting agents include benzyl alcohol, trichlorobutanol, p-hydroxybenzoic acid ester and n-butanol.

経口液剤は直接又は希釈して投与することができる。注射用液剤と同様に調製することができる。   Oral solutions can be administered directly or diluted. It can be prepared in the same manner as an injectable solution.

フロアブル剤、乳剤、などは直接又は希釈して経皮的に、又は環境処理にて投与できる。   Flowables, emulsions, etc. can be administered directly or diluted transdermally or by environmental treatment.

皮膚上で用いる液剤は、滴下し、広げ、すり込み、噴霧し、散布するか、又は浸漬(浸漬、入浴又は洗浄)により塗布することにより投与できる。これらの液剤は注射用液剤と同様に調製できる。   Solutions used on the skin can be administered by dripping, spreading, rubbing, spraying, spraying or applying by dipping (immersion, bathing or washing). These solutions can be prepared in the same manner as injection solutions.

滴下(Pour-on)剤および点下(Spot-on)剤は皮膚の限定された場所に滴下するか、又は噴霧し、これにより活性化合物を皮膚に浸漬させそして全身的に作用させることができる。滴下剤および点下剤は、有効成分を適当な皮膚適合性溶媒又は溶媒混合物に溶解するか、懸濁させるか又は乳化することにより調製できる。必要ならば、界面活性剤、着色剤、吸収促進物質、酸化防止剤、光安定剤および接着剤などの補助剤を加えてもよい。   Pour-on and spot-on agents can be dripped or sprayed onto a limited area of the skin, so that the active compound can be immersed in the skin and act systemically . Drops and drop preparations can be prepared by dissolving, suspending or emulsifying the active ingredient in suitable skin-compatible solvents or solvent mixtures. If necessary, auxiliary agents such as surfactants, colorants, absorption promoting substances, antioxidants, light stabilizers and adhesives may be added.

適当な溶媒としては、水、アルカノール、グリコール、ポリエチレングリコール、ポリプロピレングリコール、グリセリン、ベンジルアルコール、フェニルエタノール、フェノキシエタノール、酢酸エチル、酢酸ブチル、安息香酸ベンジル、ジプロピレングリコールモノメチルエーテル、ジエチレングリコールモノブチルエーテル、アセトン、メチルエチルケトン、芳香族および/又は脂肪族炭化水素、植物又は合成油、DMF、流動パラフィン、軽質流動パラフィン、シリコーン、ジメチルアセトアミド、N−メチルピロリドン又は2,2−ジメチル−4−オキシ−メチレン−1,3−ジオキソランが挙げられる。吸収促進物質には、DMSO、ミリスチン酸イソプロピル、ペラルゴン酸ジプロピレングリコール、シリコーン油、脂肪族エステル、トリグリセリドおよび脂肪アルコールが挙げられる。酸化防止剤には、亜硫酸塩、メタ重亜硫酸塩、アスコルビン酸、ブチルヒドロキシトルエン、ブチルヒドロキシアニソールおよびトコフェロールが挙げられる。   Suitable solvents include water, alkanol, glycol, polyethylene glycol, polypropylene glycol, glycerin, benzyl alcohol, phenylethanol, phenoxyethanol, ethyl acetate, butyl acetate, benzyl benzoate, dipropylene glycol monomethyl ether, diethylene glycol monobutyl ether, acetone, Methyl ethyl ketone, aromatic and / or aliphatic hydrocarbons, vegetable or synthetic oil, DMF, liquid paraffin, light liquid paraffin, silicone, dimethylacetamide, N-methylpyrrolidone or 2,2-dimethyl-4-oxy-methylene-1, 3-dioxolane is mentioned. Absorption enhancers include DMSO, isopropyl myristate, dipropylene glycol pelargonate, silicone oil, aliphatic esters, triglycerides and fatty alcohols. Antioxidants include sulfites, metabisulfites, ascorbic acid, butylhydroxytoluene, butylhydroxyanisole and tocopherol.

乳剤は、経口投与、経皮投与又は注射として投与できる。乳剤は、有効成分を疎水性相又は親水性相に溶解させ、このものを適当な乳化剤により、必要ならばさらに着色剤、吸収促進物質、保護剤、酸化防止剤、遮光剤および増粘物質などの補助剤と共に他の相の溶媒と均質化することにより調製できる。   The emulsion can be administered orally, transdermally or as an injection. In emulsions, active ingredients are dissolved in a hydrophobic phase or a hydrophilic phase, and this is further added with a suitable emulsifier, and if necessary, a colorant, an absorption promoting substance, a protective agent, an antioxidant, a light-shielding agent, a thickening substance, etc. Can be prepared by homogenizing with other phase solvents together with other auxiliary agents.

疎水性相(油)としては、パラフィン油、シリコーン油、ゴマ油、アーモンド油、ヒマシ油、合成トリグリセリド、ステアリン酸エチル、アジピン酸ジーn−ブチリル、ラウリル酸ヘキシル、ペラルゴン酸ジプロピレングリコール、分枝鎖状の短鎖長脂肪酸と鎖長C16〜C18の飽和脂肪酸とのエステル、ミリスチン酸イソプロピル、パルミチン酸イソプロピル、鎖長C12〜C18の飽和脂肪アルコールのカプリル/カプリン酸エステル、ステアリン酸イソプロピル、オレイン酸オレイル、オレイン酸デシル、オレイン酸エチル、乳酸エチル、ワックス状脂肪酸エステル、フタル酸ジブチル、アジピン酸ジイソプロピル、イソトリデシルアルコール、2−オクチルドデカノール、セチルステアリルアルコール、オレイルアルコールが挙げられる。   As hydrophobic phase (oil), paraffin oil, silicone oil, sesame oil, almond oil, castor oil, synthetic triglyceride, ethyl stearate, di-n-butyryl adipate, hexyl laurate, dipropylene glycol pelargonate, branched chain Of a short fatty acid having a chain length and a saturated fatty acid having a chain length of C16 to C18, isopropyl myristate, isopropyl palmitate, capryl / caprate of a saturated fatty alcohol having a chain length of C12 to C18, isopropyl stearate, oleyl oleate Decyl oleate, ethyl oleate, ethyl lactate, waxy fatty acid ester, dibutyl phthalate, diisopropyl adipate, isotridecyl alcohol, 2-octyldodecanol, cetyl stearyl alcohol, oleyl alcohol It is.

親水性相としては、水、プロピレングリコール、グリセリン、ソルビトールが挙げられる。   Examples of the hydrophilic phase include water, propylene glycol, glycerin, and sorbitol.

乳化剤としては、ポリオキシエチル化されたヒマシ油、ポリオキシエチル化されたモノオレフィン酸ソルビタン、モノステアリン酸ソルビタン、モノステアリン酸グリセリン、ステアリン酸ポリオキシエチル、アルキルフェノールポリグリコールエーテルなどの非イオン性界面活性剤;N−ラウリル−β−イミノジプロピオン酸二ナトリウム、レシチンなどの両性界面活性剤;ラウリル硫酸ナトリウム、脂肪アルコール硫酸エーテル、モノ/ジアルキルポリグリコールオルトリン酸エステルのモノエタノールアミン塩などの陰イオン性界面活性剤;塩化セチルトリメチルアンモニウムなどの陽イオン性界面活性剤などが挙げられる。   Emulsifiers include nonionic interfaces such as polyoxyethylated castor oil, polyoxyethylated sorbitan monoolefin acid, sorbitan monostearate, glyceryl monostearate, polyoxyethyl stearate, alkylphenol polyglycol ether, etc. Activators; amphoteric surfactants such as disodium N-lauryl-β-iminodipropionate and lecithin; anions such as sodium lauryl sulfate, fatty alcohol sulfate ether, monoethanolamine salt of mono / dialkyl polyglycol orthophosphate Surfactants; cationic surfactants such as cetyltrimethylammonium chloride.

他の補助剤として、カルボキシメチルセルロース、メチルセルロース、ポリアクリレート、アルギネート、ゼラチン、アラビアゴム、ポリビニルピロリドン、ポリビニルアルコール、メチルビニルエーテル、無水マレイン酸の共重合体、ポリエチレングリコール、ワックス、コロイド状シリカが挙げられる。   Other adjuvants include carboxymethyl cellulose, methyl cellulose, polyacrylate, alginate, gelatin, gum arabic, polyvinyl pyrrolidone, polyvinyl alcohol, methyl vinyl ether, a copolymer of maleic anhydride, polyethylene glycol, wax, colloidal silica.

半固体調製物は皮膚上に塗布するか、もしくは広げるか、又は体腔中に導入することにより投与できる。ゲルは注射用液剤について上記したように調製した溶液に、軟膏状の粘稠性を有する透明な物質を生じさせるに十分なシックナーを加えることにより調製できる。   Semi-solid preparations can be administered by application on the skin or spreading or introduction into body cavities. Gels can be prepared by adding sufficient thickener to a solution prepared as described above for an injectable solution to produce a clear material having an ointment-like consistency.

次に本発明化合物を用いる場合の製剤の配合例を示す。但し本発明の配合例は、これらのみに限定されるものではない。なお、以下の配合例において「部」は重量部を意味する。   Next, formulation examples of the preparation when the compound of the present invention is used are shown. However, the formulation examples of the present invention are not limited to these. In the following formulation examples, “parts” means parts by weight.

〔水和剤〕
本発明化合物 0.1〜80部
固体担体 5〜98.9部
界面活性剤 1〜10部
その他 0〜5部
その他として、例えば固結防止剤、分解防止剤等があげれらる。
[Wettable powder]
Compound of the present invention 0.1 to 80 parts Solid carrier 5 to 98.9 parts Surfactant 1 to 10 parts Others 0 to 5 parts Other examples include anti-caking agents and decomposition inhibitors.

〔乳剤〕
本発明化合物 0.1〜30部
液体担体 45〜95部
界面活性剤 4.9〜15部
その他 0〜10部
その他として、例えば展着剤、分解防止剤等が挙げられる。
〔emulsion〕
Compound of the present invention 0.1-30 parts Liquid carrier 45-95 parts Surfactant 4.9-15 parts Others 0-10 parts Others include, for example, spreading agents, decomposition inhibitors, and the like.

〔懸濁剤〕
本発明化合物 0.1〜70部
液体担体 15〜98.89部
界面活性剤 1〜12部
その他 0.01〜30部
その他として、例えば凍結防止剤、増粘剤等が挙げられる。
[Suspension]
Compound of the present invention 0.1 to 70 parts Liquid carrier 15 to 98.89 parts Surfactant 1 to 12 parts Others 0.01 to 30 parts Others include, for example, antifreezing agents and thickeners.

〔顆粒水和剤〕
本発明化合物 0.1〜90部
固体担体 0〜98.9部
界面活性剤 1〜20部
その他 0〜10部
その他として、例えば結合剤、分解防止剤等が挙げられる。
(Granule wettable powder)
Compound of the present invention 0.1 to 90 parts Solid carrier 0 to 98.9 parts Surfactant 1 to 20 parts Others 0 to 10 parts Others include, for example, binders and decomposition inhibitors.

〔液剤〕
本発明化合物 0.01〜70部
液体担体 20〜99.99部
その他 0〜10部
その他として、例えば凍結防止剤、展着剤等が挙げられる。
[Liquid]
Compound of the present invention 0.01 to 70 parts Liquid carrier 20 to 99.99 parts Others 0 to 10 parts Other examples include antifreezing agents and spreading agents.

〔粒剤〕
本発明化合物 0.01〜80部
固体担体 10〜99.99部
その他 0〜10部
その他として、例えば結合剤、分解防止剤等が挙げられる。
[Granule]
Compound of the present invention 0.01 to 80 parts Solid carrier 10 to 99.99 parts Others 0 to 10 parts Others include, for example, binders, decomposition inhibitors and the like.

〔粉剤〕
本発明化合物 0.01〜30部
固体担体 65〜99.99部
その他 0〜5部
その他として、例えばドリフト防止剤、分解防止剤等が挙げられる。
[Dust]
Compound of the present invention 0.01 to 30 parts Solid support 65 to 99.99 parts Others 0 to 5 parts Other examples include a drift inhibitor and a decomposition inhibitor.

次に、本発明化合物を有効成分とする製剤例をより具体的に示すが、本発明はこれらに限定されるものではない。   Next, although the formulation example which uses this invention compound as an active ingredient is shown more concretely, this invention is not limited to these.

尚、以下の配合例において、「部」は重量部を意味する。   In the following formulation examples, “parts” means parts by weight.

〔配合例1〕水和剤
本発明化合物No.1-001 20部
パイロフィライト 74部
ソルポール5039 4部
(非イオン性界面活性剤とアニオン性界面活性剤との混合物:東邦化学工業(株)商品名)
カープレックス#80D 2部
(合成含水珪酸:塩野義製薬(株)商品名)
以上を均一に混合粉砕して水和剤とする。
[Formulation Example 1] wettable powder Compound No.1-001 20 parts pyrophyllite 74 parts Solpol 5039 4 parts (mixture of nonionic surfactant and anionic surfactant: Toho Chemical Co., Ltd.) Product name)
Carplex # 80D 2 parts (Synthetic hydrous silicic acid: Shionogi & Co., Ltd. trade name)
The above is uniformly mixed and ground to obtain a wettable powder.

〔配合例2〕乳 剤
本発明化合物No.1-001 5部
キシレン 75部
N−メチルピロリドン 15部
ソルポール2680 5部
(非イオン性界面活性剤とアニオン性界面活性剤との混合物:東邦化学工業(株)商品名)
以上を均一に混合して乳剤とする。
[Formulation Example 2] Milk Compound of the present invention No.1-001 5 parts Xylene 75 parts N-methylpyrrolidone 15 parts Solpol 2680 5 parts (mixture of nonionic surfactant and anionic surfactant: Toho Chemical Industry (Product name)
The above is uniformly mixed to obtain an emulsion.

〔配合例3〕懸濁剤
本発明化合物No.1-001 25部
アグリゾールS−710 10部
(非イオン性界面活性剤:花王(株)商品名)
ルノックス1000C 0.5部
(アニオン性界面活性剤:東邦化学工業(株)商品名)
キサンタンガム 0.2部
水 64.3部
以上を均一に混合した後、湿式粉砕して懸濁剤とする。
[Formulation Example 3] Suspension Agent Compound No.1-001 25 parts Agrisol S-710 10 parts (Nonionic Surfactant: Kao Corporation trade name)
LUNOX 1000C 0.5 part (anionic surfactant: Toho Chemical Industries, Ltd. trade name)
Xanthan gum 0.2 parts water 64.3 parts After uniformly mixing the above, wet pulverize to make a suspension.

〔配合例4〕顆粒水和剤
本発明化合物No.1-001 75部
ハイテノールNE-15 5部
(アニオン性界面活性剤:第一工業製薬(株)商品名)
バニレックスN 10部
(アニオン性界面活性剤:日本製紙(株)商品名)
カープレックス#80D 10部
(合成含水珪酸:塩野義製薬(株)商品名)
以上を均一に混合粉砕した後、少量の水を加えて撹拌混合し、押出式造粒機で造粒し、乾燥して顆粒水和剤とする。
[Composition Example 4] Granule wettable powder Compound No.1-001 of the present invention 75 parts Hytenol NE-15 5 parts (anionic surfactant: trade name of Daiichi Kogyo Seiyaku Co., Ltd.)
Vanillex N 10 parts (anionic surfactant: Nippon Paper Industries Co., Ltd. trade name)
Carplex # 80D 10 parts (Synthetic hydrous silicic acid: Shionogi Pharmaceutical Co., Ltd. trade name)
After uniformly mixing and pulverizing the above, a small amount of water is added, stirred and mixed, granulated with an extrusion granulator, and dried to obtain a granulated wettable powder.

〔配合例5〕粒剤
本発明化合物No.1-001 5部
ベントナイト 50部
タルク 45部
以上を均一に混合粉砕した後、少量の水を加えて撹拌混合し、押出式造粒機で造粒し、乾燥して粒剤とする。
[Formulation Example 5] Granule Compound No. 1-001 of the present invention 5 parts Bentonite 50 parts Talc 45 parts After uniformly mixing and pulverizing the above, a small amount of water is added and mixed with stirring, and granulated with an extrusion granulator. And dried into granules.

〔配合例6〕粉剤
本発明化合物No.1-001 3部
カープレックス#80D 0.5部
(合成含水珪酸:塩野義製薬(株)商品名)
カオリナイト 95部
リン酸ジイソプロピル 1.5部
以上を均一に混合粉砕して粉剤とする。
[Formulation Example 6] Powder Compound of the present invention No.1-001 3 parts Carplex # 80D 0.5 part (Synthetic hydrous silicic acid: Shionogi Pharmaceutical Co., Ltd. trade name)
Kaolinite 95 parts Diisopropyl phosphate 1.5 parts The above is uniformly mixed and ground to obtain a powder.

使用に際しては、上記製剤を水で1〜10000倍に希釈して、又は希釈せずに直接散布する。   In use, the above preparation is diluted 1 to 10000 times with water or sprayed directly without dilution.

〔配合例7〕水和剤調製物
本発明化合物No.1-001 25部
ジイソブチルナフタレンスルホン酸ナトリウム 1部
n−ドデシルベンゼンスルホン酸カルシウム 10部
アルキルアリール ポリグリコールエーテル 12部
ナフタレンスルホン酸ホルマリン縮合物のナトリウム塩 3部
エマルジョン型シリコーン 1部
二酸化ケイ素 3部
カオリン 45部
〔配合例8〕水溶性濃厚剤調製物
本発明化合物No.1-001 20部
ポリオキシエチレンラウリルエーテル 3部
ジオクチルスルホコハク酸ナトリウム 3.5部
ジメチルスルホキシド 37部
2−プロパノール 36.5部
〔配合例9〕噴霧用液剤
本発明化合物No.1-001 2部
ジメチルスルホキシド 10部
2−プロパノール 35部
アセトン 53部
〔配合例10〕経皮投与用液剤
本発明化合物No.1-001 5部
ヘキシレングリコール 50部
イソプロパノール 45部
〔配合例11〕経皮投与用液剤
本発明化合物No.1-001 5部
プロピレングリコールモノメチルエーテル 50部
ジプロピレングリコール 45部
〔配合例12〕経皮投与(滴下)用液剤
本発明化合物No.1-001 2部
軽質流動パラフィン 98部
〔配合例13〕経皮投与(滴下)用液剤
本発明化合物No.1-001 2部
軽質流動パラフィン 58部
オリーブ油 30部
ODO−H 9部
信越シリコーン 1部
また、本発明化合物を農薬として使用する場合には、必要に応じて製剤時又は散布時に他種の除草剤、各種殺虫剤、殺ダニ剤、殺線虫剤、殺菌剤、植物生長調節剤、共力剤、肥料、土壌改良剤等と混合施用しても良い。
[Formulation Example 7] wettable powder preparation Compound No. 1-001 of the present invention 25 parts sodium diisobutylnaphthalenesulfonate 1 part calcium n-dodecylbenzenesulfonate 10 parts alkylaryl polyglycol ether 12 parts naphthalenesulfonic acid formalin condensate Sodium salt 3 parts Emulsion type silicone 1 part Silicon dioxide 3 parts Kaolin 45 parts [Formulation Example 8] Water-soluble thickener preparation Compound No.1-001 20 parts Polyoxyethylene lauryl ether 3 parts Sodium dioctyl sulfosuccinate 3. 5 parts dimethyl sulfoxide 37 parts 2-propanol 36.5 parts [Formulation Example 9] Solution for spraying the present compound No.1-001 2 parts dimethyl sulfoxide 10 parts 2-propanol 35 parts acetone 53 parts [Formulation Example 10] transdermal Solution for administration The present compound No.1-001 5 Parts hexylene glycol 50 parts isopropanol 45 parts [Formulation Example 11] Solution for transdermal administration Compound No. 1-001 5 parts propylene glycol monomethyl ether 50 parts Dipropylene glycol 45 parts [Formulation example 12] transdermal administration (instillation) ) Solution for the Invention Compound No.1-001 2 parts Light Liquid Paraffin 98 parts [Formulation Example 13] Solution for the transdermal administration (drip) Compound No.1-001 2 parts Light Liquid Paraffin 58 parts Olive Oil 30 parts ODO -H 9 parts Shin-Etsu Silicone 1 part In addition, when the compound of the present invention is used as an agrochemical, other types of herbicides, various insecticides, acaricides, nematicides, You may mix and apply with a disinfectant, a plant growth regulator, a synergist, a fertilizer, a soil conditioner, etc.

特に他の農薬あるいは植物ホルモンと混合施用することにより、施用薬量の低減による低コスト化、混合薬剤の相乗作用による殺虫スペクトラムの拡大やより高い有害生物防除効果が期待できる。この際、同時に複数の公知農薬との組み合わせも可能である。本発明化合物と混合使用する農薬の種類としては、例えばザ・ペスティサイド・マニュアル(The Pesticide Manual)15版、2009年に記載されている化合物等が挙げられる。具体的にその一般名を例示すれば次の通りであるが、必ずしもこれらのみに限定されるものではない。   In particular, when mixed with other pesticides or plant hormones, the cost can be reduced by reducing the amount of applied medicine, the insecticidal spectrum can be expanded by the synergistic action of the mixed drugs, and higher pest control effects can be expected. At this time, a combination with a plurality of known agricultural chemicals is also possible. Examples of the type of agricultural chemical used in combination with the compound of the present invention include compounds described in The Pesticide Manual 15th edition, 2009, and the like. Specific examples of common names are as follows, but the general names are not necessarily limited to these.

殺菌剤:アシベンゾラルーS−メチル(acibenzolar-S-methyl)、アシルアミノベンザミド(acylaminobenzamide)、アシペタックス(acypetacs)、アルジモルフ(aldimorph) 、アメトクトラジン(ametoctradin)、アミスルブロム(amisulbrom)、アンバム(amobam)、アムプロピルホス(ampropyfos)、アニラジン(anilazine)、アザコナゾール(azaconazole)、アジチラム(azithiram)、アゾキシストロビン(azoxystrobin)、バリウムポリサルファイド(barium polysulfide)、ベナラキシル(benalaxyl)、ベナラキシル−M(benalaxyl-M)、ベノダニル(benodanil)、ベノミル(benomyl)、ベンキノックス(benquinox)、ベンタルロン(bentaluron)、ベンチアバリカルブ(benthiavalicarb)、ベンチアゾール(benthiazole)、ベンザマクリル(benzamacril)、ベンズアモルフ(benzamorf)、ベトキサジン(bethoxazine)、ビナパクリル(binapacryl)、ビフェニル(biphenyl)、ビテルタノール(bitertanol)、ブラストサイジン−S(blasticidin-S)、ビキサフェン(bixafen)、ボルドー液(bordeaux mixture)、ボスカリド(boscalid)、ブロモコナゾール(bromoconazole)、ブピリメート(bupirimate)、ブチオベート(buthiobate)、石灰硫黄合剤(calcium polysulfide)、カルシウムポリスルフィド(calcium polysulfide)、キャプタフォール(captafol)、キャプタン(captan)、カルプロパミド(carpropamid)、カルバモルフ(carbamorph)、カルベンダジン(carbendazim)、カルボキシン(carboxin)、カルボン(carvone)、チェシュントミクスチャ(cheshunt mixture)、キノメチオネート(chinomethionat)、クロベンチアゾン(chlobenthiazone)、クロラニフォルメタン(chloraniformethane)、クロラニル(chloranil)、クロルフェナゾール(chlorfenazol)、クロロネブ(chloroneb)、クロロピクリン(chloropicrin)、クロロタロニル(chlorothalonil)、クロロキノックス(chlorquinox)、クロゾリネート(chlozolinate)、クリムバゾール(climbazole)、クロトリマゾール(clotrimazole)、カッパーアセテイト(copper acetate)、塩基性炭酸銅(copper carbonate, basic)、水酸化第二銅(copper hydroxide)、カッパーナフタレン(copper naphthenate)、カッパーオルアイト(copper oleate)、カッパーオキシクロリド(copper oxychloride)、硫酸銅(copper sulfate)、塩基性硫酸銅(copper sulfate, basic)、カッパージンククロメイト(copper zinc chromate)、クフラネブ(cufraneb)、クプロバム(cuprobam)、シアゾファミド(cyazofamid)、シクラフルアミド(cyclafuramid)、シクロヘキシミド(cycloheximide)、シフルフェナミド(cyflufenamid)、シモキサニル(cymoxanil)、サイペンダゾール(cypendazole)、シプロコナゾール(cyproconazol)、シプロジニル(cyprodinil)、シプロフラム(cyprofuram)、ダゾメット(dazomet)、デバカルブ(debacarb)、デカフェンチン(decafentin)、デハイドロアセテイト(dehydroacetic acid)、ジクロフルアニド(dichlofluanid)、ジクロン(dichlone)、ジクロロフェン(dichlorophen)、ジクロゾリン(dichlozoline)、ジクロブトラゾール(diclobutrazol)、ジクロシメット(diclocymet)、ジクロメジン(diclomedine)、ジクロラン(dicloran)など。   Bactericides: acibenzolar-S-methyl, acylaminobenzamide, acypetacs, aldimorph, ametoctradin, amisulbrom, amobam, ampropyl Phos (ampropyfos), anilazine, azaconazole, azithiram, azoxystrobin, barium polysulfide, benalaxyl, benalaxyl-M, benodaril (Benodanil), benomyl, benquinox, bentaluron, benthiavalicarb, benthiazole, benzamacril, benzamorf, bethoxazine, Binapacryl Biphenyl, bitertanol, blasticidin-S, bixafen, bordeaux mixture, boscalid, bromoconazole, bupirimate, buthiobate (Buthiobate), calcium polysulfide, calcium polysulfide, captafol, captan, carpropamid, carbamorph, carbendazim, carboxin (Carboxin), carvone, cheshunt mixture, chinomethionat, clobenthiazone, chloraniformethane, chloranil, chlorfenazol, Chloroneb (c hloroneb), chloropicrin, chlorothalonil, chlorquinox, chlozolinate, climbazole, clotrimazole, copper acetate, basic copper carbonate (copper carbonate, basic), cupric hydroxide, copper naphthenate, copper oleate, copper oxychloride, copper sulfate, basic sulfuric acid Copper sulfate, basic, copper zinc chromate, cufraneb, cuprobam, cyazofamid, cyclafuramid, cycloheximide, cyflufenamid, Simoxanil, cypendazole, cyproconazole (cyp) roconazol), cyprodinil, cyprofuram, dazomet, debacarb, decaentin, dehydroacetic acid, dichlorfluanid, dichlone, Dichlorophen, dichlozoline, diclobutrazol, diclocymet, diclomedine, dicloran, etc.

殺菌剤(続き):ジエトフェンカルブ(diethofencarb)、ジフェノコナゾール(difenoconazole)、ジフルメトリン(diflumetorim)、ジメチリモール(dimethirimol)、ジメトモルフ(dimethomorph)、ジモキシストロビン(dimoxystrobin)、ジニコナゾール(diniconazole)、ジニコナゾール−M(diniconazole-M)、ジノブトン(dinobuton)、ジノカップ(dinocap)、ジノカップ−4(dinocap-4)、ジノカップ−6(dinocap-6)、ジノクトン(dinocton)、ジノスルフォン(dinosulfon)、ジノテルボン(dinoterbon)、ジフェニルアミン(diphenylamine)、ジピリチオン(dipyrithione)、ジタリムホス(ditalimfos)、ジチアノン(dithianon)、ドデモルフ(dodemorph)、ドジン(dodine)、ドラゾクソロン(drazoxolon)、エデフェノホス(edifenphos)、エポキシコナゾール(epoxiconazole)、エタコナゾール(etaconazole)、エタボキサム(ethaboxam)、エテム(etem)、エチリモル(ethirimol)、エトキシキン(ethoxyquin)、エトリジアノール(etridiazole)、ファモキサゾン(famoxadone)、フェナリモル(fenarimol)、フェブコナゾール(febuconazole)、フェナミドン(fenamidone)、フェナミノスルフ(fenaminosulf)、フェナパニル(fenapanil)、フェンダゾスラム(fendazosulam)、フェンフラム(fenfuram)、フェンヘキサミド(fenhexamid)、フェニトロパン(fenitropan)、フェノキサニル(fenoxanil)、フェンピクロニル(fenpiclonil)、フェンプロピジン(fenpropidin)、フェンピラザミン(fenpyrazamine)、フェンプロピモルフ(fenpropimorph)、フェンチン(fentin)、フェルバン(ferbam)、フェリムゾン(ferimzone)、フルアジナム(fluazinam)、フルジオキソニル(fludioxonil)、フルメトベル(flumetover)、フルモルフ(flumorph)、フルオピコリド(fluopicolide)、フルオピラム(fluopyram)、フルオロイミド(fluoroimide)、フルオトリマゾール(fluotrimazole)、フルオキサストロビン(fluoxastrobin)、フルキンコナゾール(fluquinconazole)、フルシラゾール(flusilazole)、フルスルファミド(flusulfamide)、フルチアニル(flutianil)、フルトラニル(flutolanil)、フルトリアフォール(flutriafol)、フルキサピロキサド(fluxapyroxad)、フォルペット(folpet)、フォセチル−アルミニウム(fosetyl-aluminium)、フベリダゾール(fuberidazole)、フララキシル(furalaxyl)、フラメトピル(furametpyr)、フルカルバニル(furcarbanil)、フルコナゾール(furconazole)、フルコナゾール−シス(furconazole-cis)、フルメシクロックス(furmecyclox)、フルファネート(furphanate)、グリオジン(glyodin)、グリセオフルビン(griseofulvin)、グアザチン(guazatine)、ハラクリネイト(halacrinate)、ヘキサクロロベンゼン(hexachlorobenzene)、ヘキサコナゾール(hexaconazole)、ヘキシルチオフォス(hexylthiofos)、ハイドロキシキノリン サルフェイト(8-hydroxyquinoline sulfate)、ヒメキサゾール(hymexazol)、イマザリル(imazalil)、イミベンコナゾール(imibenconazole)、イミノクタジン(iminoctadine)、イプコナゾール(ipconazole)、イプロベンホス(iprobenfos)、イプロジオン(iprodione)、イプロバリカルブ(iprovalicarb)、イソプロチオラン(isoprothiolane)、イソバレジオン(isovaledione)など。   Bactericides (continued): diethofencarb, difenoconazole, diflumetorim, dimethirimol, dimethomorph, dimoxystrobin, diniconazole-M, diniconazole-M, diniconazole-M M), dinobuton, dinocap, dinocap-4, dinocap-6, dinoton, dinosulfon, dinoterbon, diphenylamine ), Dipyrithione, ditalimfos, dithianon, dodemorph, dodine, drazoxolon, edifenphos, epoxiconazole, etaconazole, etaconazole Xham (ethaboxam), etem, etirimol, ethoxyquin, etridianol, famoxadone, fenarimol, febuconazole, fenamidone, phenaminosulf ), Fenapanil, fendazosulam, fenfuram, fenhexamid, fenitropan, fenoxanil, fenpiclonil, fenpropidin, fenpyrazamine (fenpyrazamine), fenpropimorph, fentin, ferbam, ferimzone, fluazinam, fludioxonil, flumetover, flumorph, full Fluopicolide, fluopyram, fluoroimide, fluotrimazole, fluoxastrobin, fluquinconazole, flusilazole, flusulfamide, fluthianyl (fluoxanil) flutianil), flutolanil, flutriafol, fluxapyroxad, folpet, fosetyl-aluminium, fuberidazole, fluralaxyl, flametopyr ( furametpyr), furcarbanil, furconazole, fluconazole-cis, furmecyclox, furphanate, furyonate, glyodin, griseofulvin, guazachi (Guazatine), halacrinate, hexachlorobenzene, hexaconazole, hexylthiofos, hydroxyquinoline sulfate, hymexazol, imazalil, Imibenconazole, iminoctadine, ipconazole, iprobenfos, iprodione, iprovalicarb, isoprothiolane, isovaledione, etc.

殺菌剤(続き):カスガマイシン(kasugamycin)、クレソキシム−メチル(kresoxim-methyl)、マンカッパー(mancopper)、マンコゼブ(mancozeb)、マンジプロパミド(mandipropamid)、マンネブ(maneb)、メベニル(mebenil)、メカルビンジド(mecarbinzid)、メパニピリム(mepanipyrim)、メプロニル(mepronil)、メタラキシル(metalaxyl)、メタラキシル−M(metalaxyl-M)、メタム(metam)、メタゾキソロン(metazoxolon)、メトコナゾール(metconazole)、メタスルホカルブ(methasulfocarb)、メトフロキサム(methfuroxam)、メチルイソチオシアネイト(methyl isothiocyanate)、メチラム(metiram)、メトミノストロビン(metominostrobin)、メトラフェノン(metrafenone)、メトスルフォバックス(metsulfovax)、ミルネブ(milneb)、ミクロブタニル(myclobutanil)、ミクロゾリン(myclozolin)、ナバム(nabam)、ナタマイシン(natamycin)、ニッケルビス(ジメチルジチオカーバメート)(nickel bis(dimethyldithiocarbamate))、ニトロスチレン(nitrostyrene)、ニトロタール−イソプロピル(nitrothal-isopropyl)、ヌアリモル(nuarimol)、オーシーエイチ(OCH)、オクチリノン(octhilinone)、オフレース(ofurace)、オリサストロビン(orysastrobin)、オキサジキシル(oxadixyl)、有機銅(oxine copper)、オキシカルボキシン(oxycarboxin)、オキスポコナゾールフマール酸塩(oxpoconazole fumarate)、ペフラゾエート(pefurzoate)、ペンコナゾール(penconazole)、ペンフルフェン(penflufen)、ペンシクロン(pencycuron)、ペンチオピラド(penthiopyrad)、オルソフェニルフェノール(o-phenylphenol)、フォスジフェン(phosdiphen)、フタライド(phthalide)、ピコキシストロビン(picoxystrobin)、ピペラリン(piperalin)、ポリカーバメート(polycarbamate)、ポリオキシン(polyoxins)、ポリオクソリム(polyoxorim)、ポタシウムアザイド(potassium azide)、炭酸水素カリウム(potassium hydrogen carbonate)、プロキナジド(proquinazid)、プロベナゾール(probenazole)、プロクロラズ(prochloraz)、プロシミドン(procymidone)、プロパモカルブ塩酸塩(propamocarb hydrochloride)、プロピコナゾール(propiconazole)、プロピネブ(propineb)、プロチオカルブ(prothiocarb)、プロチオコナゾール(prothioconazole)、ピラカルボリド(pyracarbolid)、ピラクロストロビン(pyraclostrobin)、ピラゾホス(pyrazophos)、ピリジニトリル(pyridinitril)、ピリフェノックス(pyrifenox)、ピリメタニル(pyrimethanil)、ピリオフェノン(pyriofenone)、ピロキュロン(pyroquilon)、ピロキシクロル(pyroxychlor)、ピロキシフル(pyroxyfur)、キノメチオネート(quinomethionate)、キノキシフェン(quinoxyfen)、キントゼン(quintozene)、キナセトール・スルフェート(quinacetol-sulfate)、キナザミド(quinazamid)、キンコナゾール(quinconazole)、ラベンザゾール(rabenzazole)など。   Fungicide (continued): kasugamycin, kresoxim-methyl, mancopper, mancozeb, mandipropamid, maneb, mebenil, mecarbinzid , Mepanipyrim, mepronil, metalaxyl, metalaxyl-M, metam, metazoxolon, metconazole, metasulfocarb, metoxasulfocarb, metoxafloxam ), Methyl isothiocyanate, metiram, metinominostrobin, metrafenone, metsulfovax, milneb, microbutanil, microzoline (myclozo) lin), nabam, natamycin, nickel bis (dimethyldithiocarbamate), nitrostyrene, nitrothal-isopropyl, nuarimol, OH (OCH), octhilinone, offurace, orysastrobin, oxadixyl, oxine copper, oxycarboxin, oxpoconazole fumarate , Pefurzoate, penconazole, penflufen, penencycuron, penthiopyrad, o-phenylphenol, phosdiphen, phthalide, picoxis Robin (picoxystrobin), piperalin (piperalin), polycarbamate (polycarbamate), polyoxins (polyoxins), polyoxorim (polyoxorim), potassium azide (potassium hydrogen carbonate) (potassium hydrogen carbonate), proquinazid (proquinazid) probenazole), prochloraz, procymidone, propamocarb hydrochloride, propiconazole, propineb, prothiocarb, prothioconazole, pyracarbolid, Pyraclostrobin, pyrazophos, pyridinitril, pyrifenox, pyrimethanil, pyriofenone, pyroculone (pyroq) uilon, pyroxychlor, pyroxyfur, quinomethionate, quinoxyfen, quintozene, quinacetol-sulfate, quinazamid, quinazaazole, quinconazole rabenzazole).

殺菌剤(続き):アジ化ナトリウム(sodium azide)、炭酸水素ナトリウム(sodium hydrogen carbonate)、次亜塩素酸ナトリウム(sodium hypochlorite)、硫黄(sulfur)、スピロキサミン(spiroxamine)、サリチルアニリド(salycylanilide)、シルチオファム(silthiofam)、シメコナゾール(simeconazole)、テブコナゾール(tebuconazole)、テクナゼン(tecnazene)、テコラム(tecoram)、テトラコナゾール(tetraconazole)、チアベンダゾール(thiabendazole)、チアジフルオール(thiadifluor)、チシオフェン(thicyofen)、チフルザミド(thifluzamide)、チオクロルフェンフィム(thiochlorfenphim)、チオファネート(thiophanate)、チオファネート−メチル(thiophanate-methyl)、チオキノックス(thioquinox)、チラム(thiram)、チアジニル(tiadinil)、チオキシミド(tioxymid)、トルクロホス−メチル(tolclofos-methyl)、トリルフラニド(tolylfluanid)、トリアジメホン(triadimefon)、トリアジメノール(toriadimenol)、トリアミフォス(triamiphos)、トリアリモル(triarimol)、トリアゾキシド(triazoxide)、トリアズブチル(triazbutil)、トリブチルチンオキサイド(tributyltin oxide)、トリクラミド(trichlamide)、トリシクラゾール(tricyclazole)、トリデモルフ(tridemorph)、トリフロキシストロビン(trifloxystrobin)、トリフルミゾール(triflumizole)、トリホリン(triforine)、トリチコナゾール(triticonazole)、バリダマイシン(validamycin)、バリフェナレート(valifenalate)、ビンクロゾリン(vinclozolin)、ザリルアミド(zarilamide)、硫酸亜鉛(zinc sulfate)、ジネブ(zineb)、ジラム(ziram)、ゾキサミド(zoxamide)及びシイタケ菌糸体抽出物など。   Fungicide (continued): sodium azide, sodium hydrogen carbonate, sodium hypochlorite, sulfur, spiroxamine, salicylanilide, silthiofam (Silthiofam), simeconazole, tebuconazole, tecnazene, tecoram, tetraconazole, thiabendazole, thiadifluor, thicyofen, thifluzamide thifluzamide, thiochlorfenphim, thiophanate, thiophanate-methyl, thioquinox, thiram, thiadinyl, tioxymid, tolcrophos-me Tolclofos-methyl, tolylfluanid, triadimefon, triadimenol, triamiphos, triarimol, triazoxide, triazbutil, tributyltin oxide ), Trichlamide, tricyclazole, tridemorph, trifloxystrobin, triflumizole, triforine, triticonazole, validamycin, validamycin Examples include valifenalate, vinclozolin, zarilamide, zinc sulfate, zineb, ziram, zoxamide and shiitake mycelium extract.

殺バクテリア剤:ベンザルコニウムクロライド(benzalkonium chloride)、ビチオノール(bithionol)、ブロノポール(bronopol)、クレゾール(cresol)、ホルムアルデヒド(formaldehyde)、ニトラピリン(nitrapyrin)、オキソリニックアシド(oxolinic acid)、オキシテトラサイクリン(oxyterracycline)、ストレプトマイシン(streptomycin)及びテクロフタラム(tecloftalam)など。   Bactericides: benzalkonium chloride, bithionol, bronopol, cresol, formaldehyde, nitrapyrin, oxolinic acid, oxyterracycline , Streptomycin and tecloftalam.

殺線虫剤:アルドキシカルブ(aldoxycarb)、カズサホス(cadusafos)、デービーシーピー(DBCP)、ジクロフェンチオン(dichlofenthion)、デーエスピー(DSP)、エトプロホス(ethoprophos)、フェナミホス(fenamiphos)、フェンスルホチオン(fensulfothion)、フルエンスルホン(fluensulfone)、フォスチアゼート(fosthiazate)、フォスチエタン(fosthietan)、イミシアホス(imicyafos)、イサミドホス(isamidofos)、イサゾホス(isazofos)、オキサミル(oxamyl)及びチオナジン(thionazin)など。   Nematicides: aldoxycarb, cadusafos, DCP, DBCH, dichlofenthion, DSP (DSP), etoprophos, fenamiphos, fensulfothion, fluene Sulfone (fluensulfone), fosthiazate (fosthiazate), fosthietan (fosthietan), imisiafos (imicyafos), isamidofos (isamidofos), isazofos (isazofos), oxamyl (oxamyl) and thionazin (thionazin) and the like.

殺ダニ剤:アセキノシル(acequinocyl)、アクリナトリン(acrinathrin)、アミトラズ(amitraz)、BCI−033(試験名)、ビフェナゼート(bifenazate)、ブロモプロピレート(bromopropylate)、チノメチオネート(chinomethionat)、クロロベンジラート(chlorobezilate)、クロフェンテジン(clofentezine)、シエノピラフェン(cyenopyrafen)、シフルメトフェン(cyflumetofen)、サイヘキサチン(cyhexatine)、ジコフォール(dicofol)、ジエノクロール(dienochlor)、デーエヌオーシー(DNOC)、エトキサゾール(etoxazole)、フェナザキン(fenazaquin)、フェンブタチンオキシド(fenbutatin oxide)、フェノチオカルブ(fenothiocarb)、フェンプロパトリン(fenpropathrin)、フェンピロキシメート(fenpyroximate)、フルアクリピリム(fluacrypyrim)、ハルフェンプロックス(halfenprox)、ヘキシチアゾックス(hexythiazox)、ミルベメクチン(milbemectin)、プロパルギット(propargite)、ピリダベン(pyridaben)、ピリミジフェン(pyrimidifen)、S−1870(試験名)、スピロジクロフェン(spirodiclofen)、スピロメシフェン(spyromesifen)、NNI−0711(試験名)、CL900167(試験名)及びテブフェンピラド(tebufenpyrad)など。   Acaricide: acequinocyl, acrinathrin, amitraz, BCI-033 (test name), bifenazate, bromopropylate, chinomethionat, chlorobezilate , Clofentezine, cyenopyrafen, cyflumetofen, cyhexatine, dicofol, dienochlor, denochlor (DNOC), etoxazole, quinazaquin (fenaza) Fenbutatin oxide, fenothiocarb, fenpropathrin, fenpyroximate, fluacrypyrim, halfenprox (halfenpro) x), hexythiazox, milbemectin, propargite, pyridaben, pyrimidifen, S-1870 (test name), spirodiclofen, spiromesifen ( spyromesifen), NNI-0711 (test name), CL900187 (test name) and tebufenpyrad.

殺虫剤:アバメクチン(abamectin)、アセフェート(acephate)、アセタミピリド(acetamipirid)、アラニカルブ(alanycarb)、アルディカルブ(aldicarb)、アレスリン(allethrin)、アザメチホス(azamethiphos)、アジンホス−メチル(azinphos-methyl)、バチルスチューリンゲシス(bacillus thuringiensis)、ベンジオカルブ(bendiocarb)、ベンフルトリン(benfluthrin)、ベンフラカルブ(benfuracarb)、ベンスルタップ(bensultap)、ビフェントリン(bifenthrin)、ビオアレスリン(bioallethrin)、ビオレスメトリン(bioresmethrin)、ビストリフルロン(bistrifluron)、ブプロフェジン(buprofezin)、ブトカルボキシン(butocarboxim)、カルバリル(carbaryl)、カルボフラン(carbofuran)、カルボスルファン(carbosulfan)、カルタップ(cartap)、クロルアントラニリプロール(chlorantraniliprole)、クロルエトキシホス(chlorethxyfos)、クロルフェナピル(chlorfenapyr)、クロルフェンビンホス(chlorfenvinphos)、クロルフルアズロン(chlorfluazuron)、クロルメホス(chlormephos)、クロルピリホス(chlorpyrifos)、クロピリホス−メチル(chlorpyrifos-methyl)、クロマフェノジド(chromafenozide)、クロチアニジン(clothianidin)、シアントラニリプロール(cyantraniliprole)、シクロプロトリン(cycloprothrin)、シフルメトフェン(cyflumetofen)、シフルトリン(cyfluthrin)、ベータ−シフルトリン(beta-cyfluthrin)、シハロトリン(cyhalothrin)、ラムダ−シハロトリン(lambda-cyhalothrin)、シペルメトリン(cypermethrin)、アルファ−シペルメトリン(alpha-cypermethrin)、ベータ−シペルメトリン(beta-cypermethrin)、ゼタ−シペルメトリン(zeta-cypermethrin)、シロマジン(cyromazine)、デルタメトリン(deltamethrin)、ジアクロデン(diacloden)、ジアフェンチウロン(diafenthiuron)、ダイアジノン(diazinon)、ジクロルボス(dichlorvos)、ジフルベンズロン(diflubenzuron)、ジメチルビンホス(dimethylvinphos)、ジノテフラン(dinotefuran)、ジオフェノラン(diofenolan)、ジスルフォトン(disulfoton)、ジメトエート(dimethoate)、エマメクチンベンゾエート(emamectin-benzoate)、エンペントリン(empenthrin)、エンドスルファン(endosulfan)、アルファ−エンドスルファン(alpha-endosulfan)、イーピーエヌ(EPN)、エスフェンバレレート(esfenvalerate)、エチオフェンカルブ(ethiofencarb)、エチプロール(ethiprole)、エトフェンプロックス(etofenprox)、エトリムホス(etrimfos)、フェニトロチオン(fenitrothion)、フェノブカルブ(fenobucarb)、フェノキシカーブ(fenoxycarb)、フェンプロパトリン(fenpropathrin)、フェンチオン(fenthion)、フェンバレレート(fenvalerate)、フィプロニル(fipronil)、フロニカミド(flonicamid)、フルベンジアミド(flubendiamide)、フルシトリネート(flucythrinate)、フルフェネリム(flufenerim)、フルフェノクスウロン(flufenoxuron)、フルフェンプロックス(flufenprox)、フルメトリン(flumethrin)、フルバリネート(fluvalinate)、タウ−フルバリネート(tau-fluvalinate)、ホノホス(fonophos)、フォルメタネート(formetanate)、フォルモチオン(formothion)、フラチオカルブ(furathiocarb)、フルフィプロール(flufiprole)、フルピラジフロン(flupyradifurone)、フロメトキン(flometoquin)など。   Insecticides: abamectin, acephate, acetamipirid, alanamicarb, aldicarb, allethrin, azamethiphos, azinphos-methyl, bacillus tubulin Bacillus thuringiensis, bendiocarb, benfluthrin, benfuracarb, bensultap, bifenthrin, bioallethrin, bioresmethrin, bistrifluron, tris Buprofezin, butocarboxim, carbaryl, carbofuran, carbosulfan, cartap, chlorantraniliprole, Chlorethxyfos, chlorfenapyr, chlorfenvinphos, chlorfluazuron, chlormephos, chlorpyrifos, chlorpyrifos-methyl, chromafenozide, chromafenozide Clothianidin, cyantraniliprole, cycloprothrin, cyflumetofen, cyfluthrin, beta-cyfluthrin, cyhalothrin, lambda-cyhalothrin cyhalothrin), cypermethrin, alpha-cypermethrin, beta-cypermethrin, zeta-cypermethrin, cyromazine, Deltamethrin, diacloden, diafenthiuron, diazinon, dichlorvos, diflubenzuron, dimethylvinphos, dinotefuran, diofenolan, diofenolan Disulfoton, dimethoate, emamectin-benzoate, empenthrin, endosulfan, alpha-endosulfan, EP-N, EPN, esfenvalerate, etiophencarb (Ethiofencarb), ethiprole, etofenprox, etrimfos, fenitrothion, fenobucarb, fenobucarb Fenoxycarb, fenpropathrin, fenthion, fenvalerate, fipronil, flonicamid, flubendiamide, flucythrinate, flufenerim , Flufenoxuron, flufenprox, flumethrin, fluvalinate, tau-fluvalinate, fonophos, formetanate, formotaion ( formothion), furathiocarb, flufiprole, flupyradifurone, flometoquin and the like.

殺虫剤(続き):ハロフェノジド(halofenozide)、ヘキサフルムロン(hexaflumuron)、ヒドラメチルノン(hydramethylnon)、イミダクロプリド(imidacloprid)、イソフェンホス(isofenphos)、インドキサカルブ(indoxacarb)、イソプロカルブ(isoprocarb)、イソキサチオン(isoxathion)、レピメクチン(lepimectin)、ルフェヌウロン(lufenuron)、マラチオン(malathion)、メペルフルスリン(meperfluthrin)、メタフルミゾン(metaflumizone)、メタルデヒド(metaldehyde)、メタミドホス(methamidophos)、メチダチオン(methidathion)、メタクリホス(methacrifos)、メタフルミゾン(metaflumizone)、メタルカルブ(metalcarb)、メソミル(methomyl)、メソプレン(methoprene)、メトキシクロール(methoxychlor)、メトキシフェノジド(methoxyfenozide)、メチルブロマイド(methyl bromide)、モノクロトホス(monocrotophos)、ムスカルーレ(muscalure)、ニテンピラム(nitenpyram)、ノバルロン(novaluron)、ノビフルムロン(noviflumuron)、オメトエート(omethoate)、オキサミル(oxamyl)、オキシデメトン−メチル(oxydemeton-methyl)、オキシデプロホス(oxydeprofos)、パラチオン(parathion)、パラチオン−メチル(parathion-methyl)、ペンタクロロフェノール(pentachlorophenol(PCP))、ペルメトリン(permethrin)、フェノトリン(phenothrin)、フェントエート(phenthoate)、フォキシム(phoxim)、ホレート(phorate)、ホサロン(phosalone)、ホスメット(phosmet)、ホスファミドン(phosphamidon)、ピリミカルブ(pirimicarb)、ピリミホス−メチル(pirimiphos-methyl)、プロフェノホス(profenofos)、プロチオホス(prothiofos)、プロパホス(propaphos)、プロトリフェンブト(protrifenbute)、ピメトロジン(pymetrozine)、ピラクロホス(pyraclofos)、ピレトリン(pyrethrins)、ピリダリル(pyridalyl)、ピリフルキナゾン(pyrifluquinazon)、ピリプロール(pyriprole)、ピラフルプロール(pyrafluprole)、、ピリプロキシフェン(pyriproxyfen)、レスメトリン(resmethrin)、ロテノン(rotenone)、SI−0405(試験名)、スルプロホス(sulprofos)、シラフルオフェン(silafluofen)、スピネトラム(spinetoram)、スピノサド(spinosad)、スピロテトラマート(spirotetramat)、スルホキサフロール(sulfoxaflor)、スルホテップ(sulfotep)、SYJ−159(試験名)、テブフェノジド(tebfenozide)、テフルベンズロン(teflubenzuron)、テフルトリン(tefluthorin)、テルブホス(terbufos)、テトラクロロビンホス(tetrachlorvinphos)、テトラメトリン(tetramethrin)、d−T−80−フタルスリン(d-tetramethrin)、テトラメチルフルスリン(tetramethylfluthrin)、チアクロプリド(thiacloprid)、チオシクラム(thiocyclam)、チオジカルブ(thiodicarb)、チアメトキサム(thiamethoxam)、チオファノックス(thiofanox)、チオメトン(thiometon)、トルフェンピラド(tolfenpyrad)、トラロメスリン(tralomethrin)、トリクロルホン(trichlorfon)、トリアズロン(triazuron)、トリフルムロン(triflumuron)、バミドチオン(vamidothion)及びME−5343(試験名)など。   Insecticides (continued): halofenozide, hexaflumuron, hydramethylnon, imidacloprid, isofenphos, indoxacarb, isoprocarb, isoxathion ), Lepimectin, lufenuron, malathion, meperfluthrin, metaflumizone, metalaldehyde, methamidophos, methidathion, methidathion, methacrifos (methacrifos) ), Metalcarb, methomyl, metoprene, methoxychlor, methoxyfenozide, methyl bromide , Monocrotophos, muscalure, nitenpyram, novaluron, noviflumuron, omethoate, oxamyl, oxydemeton-methyl, oxydemeton-methyl (oxydemeton-methyl) oxydeprofos, parathion, parathion-methyl, pentachlorophenol (PCP), permethrin, phenothrin, phenthoate, phoxim, phorate ), Phosalone, phosmet, phosphamidon, pirimicarb, pirimiphos-methyl, profenofos, prothiofos, propaphos, prototri Protrifenbute, pyrometrozine, pyraclofos, pyrethrins, pyridalalyl, pyrifluquinazon, pyriprole, pyrafluprole, proxy, pyrifiprofen, py Resmethrin, rotenone, SI-0405 (study name), sulprofos, silafluofen, spinetram, spinosad, spirotetramat, sulfoxaflor ), Sulfotep, SYJ-159 (test name), tebfenozide, teflubenzuron, tefluthorin, terbufos, tetrachlorvinphos, tetrame Trimethrin, dT-80-phthalthrin, d-tetramethrin, tetramethylfluthrin, thiacloprid, thiocyclam, thiodicarb, thiamethoxam, thiophanox ( thiofanox, thiometon, tolfenpyrad, tralomethrin, trichlorfon, triazuron, triflumuron, vamidomion and ME-5343 (test name).

以下に本発明化合物の合成例、試験例を実施例として具体的に述べることで、本発明をさらに詳しく説明するが、本発明はこれらによって限定されるものではない。   Hereinafter, the present invention will be described in more detail by specifically describing synthesis examples and test examples of the compounds of the present invention as examples, but the present invention is not limited thereto.

合成例に記載した中圧分取液体クロマトグラフィーは、山善株式会社中圧分取装置;YFLC−Wprep(流速18ml/min、シリカゲル40μmのカラム)を使用した。   The medium pressure preparative liquid chromatography described in the synthesis example used an intermediate pressure preparative apparatus (Yamazen Co., Ltd.); YFLC-Wprep (flow rate 18 ml / min, silica gel 40 μm column).

[合成例]
合成例1
N−エチル−2−(メトキシイミノ)−3−(メチルチオ)−N−{1−(ピリジン−3−イル)−1H−1,2,3−トリアゾール−4−イル}プロパンアミドの製造(本発明化合物1−001)
工程1
1−(ピリジン−3−イル)−1H−1,2,3−トリアゾ−ル−4−アミドの製造
バイオオーガニック アンド メディシナル ケミストリー レターズ 2008年,18巻,1195頁記載の方法により合成した1−(ピリジン−3−イル)−1H−1,2,3−トリアゾ−ル−4−カルボン酸1.9gのジクロロメタン20ml溶液に、室温下で塩化オキサリル3.8g、N,N−ジメチルホルムアミド20mgを順次添加した。該反応混合物を室温で30分間撹拌した後、減圧下にて溶媒を留去した。溶媒を留去した後に得られた残渣をジクロロメタン5mlに溶解させ、28%アンモニア水溶液30mlに投入した。該反応混合物を室温で2時間撹拌した後、析出した固体をろ過にて取り出た。得られた固体を水洗後、乾燥して目的物1.4gを茶色固体として得た。
H NMR(測定溶媒DMSO−d6)δ9.34(s,1H),9.18(d,J=2.4Hz,1H),8.72(d,J=4.8Hz,1H),8.38(d,J=8.1Hz,1H),8.05(brs,1H),7.70−7.60(m,2H)
融点;260−263℃
工程2
メチル {1−(ピリジン−3−イル)−1H−1,2,3−トリアゾ−ル−4−イル}カーバメートの製造
1−(ピリジン−3−イル)−1H−1,2,3−トリアゾ−ル−4−アミド900mgのメタノール60ml溶液に、室温下にて8重量%次亜塩素酸ナトリウム水溶液4.9gを添加した。添加終了後、加熱還流下で20時間撹拌した。反応終了後、反応混合物を室温まで放冷した後、溶媒を減圧下にて留去した。溶媒を留去した後に得られた残渣に、水50mlを加え、酢酸エチル200mlにて抽出した。得られた有機層を、無水硫酸ナトリウムで脱水・乾燥後、減圧下にて溶媒を留去した。溶媒を留去した後に得られた残渣を酢酸エチル−メタノール〔10:1(体積比、以下同じである)〕にて溶出する中圧分取液体クロマトグラフィーにて精製し、目的物700mgを白色固体として得た。
H NMR(測定溶媒CDCl)δ9.06(d,J=2.4Hz,1H),8.72(dd,J=1.5,4.8Hz,1H),8.29(s,1H),8.13(ddd,J=1.5,2.4,8.4Hz,1H),7.72(brs,1H),7.51(dd,J=4.8,8.4Hz,1H),3.86(s,3H)
融点;168−169℃
工程3
メチル エチル{1−(ピリジン−3−イル)−1H−1,2,3−トリアゾ−ル−4−イル}カーバメートの製造
60重量%水素化ナトリウム(鉱油中に分散)165mgのN,N−ジメチルホルムアミド5ml溶液に、氷冷下でメチル {1−(ピリジン−3−イル)−1H−1,2,3−トリアゾ−ル−4−イル}カーバメート600mgを添加した。添加終了後、室温まで昇温し、30分間撹拌した。反応混合物にヨウ化エチル468mgを添加し、更に室温で1時間撹拌を継続した。反応終了後、反応混合物を氷水に注ぎ、酢酸エチル100mlにて抽出した。得られた有機層を無水硫酸ナトリウムで脱水・乾燥後、減圧下にて溶媒を留去した。残留物をn−ヘキサン−酢酸エチル(15:85)にて溶出する中圧分取液体クロマトグラフィーにて精製し、目的物500mgを白色固体として得た。
H NMR(測定溶媒CDCl)δ9.05(d,J=2.4Hz,1H),8.70(d,J=4.5Hz,1H),8.43(s,1H),8.14(m,1H),7.50(dd,J=4.5,8.4Hz,1H),4.18(q,J=7.2Hz,2H),3.88(s,3H),1.33(t,J=7.2Hz,3H)
融点;161−163℃
工程4
N−エチル−1−(ピリジン−3−イル)−1H−1,2,3−トリアゾ−ル−4−アミンの製造
メチル エチル{1−(ピリジン−3−イル)−1H−1,2,3−トリアゾ−ル−4−イル}カーバメート500mgの1,4−ジオキサン12ml溶液に、1N水酸化ナトリウム水溶液12mlを加え100℃にて2時間撹拌した。反応完結後、反応混合物を室温まで放冷した後、水200mlを添加し、酢酸エチル100mで3回抽出した。得られた有機層を混合し、無水硫酸ナトリウムで脱水・乾燥した。減圧下にて溶媒を留去し、目的物400mgを淡黄色固体として得た。
H NMR(測定溶媒CDCl)δ8.96(d,J=2.4Hz,1H),8.63(dd,J=1.5,4.8Hz,1H),8.10(ddd,J=1.5,2.4,8.4Hz,1H),7.45(dd,J=4.8,8.4Hz,1H),7.25(s,1H),3.97(brs,1H),3.19(q,J=7.2Hz,2H),1.29(t,J=7.2Hz,3H)
工程5
N−エチル−2−(メトキシイミノ)−3−(メチルチオ)−N−{1−(ピリジン−3−イル)−1H−1,2,3−トリアゾール−4−イル}プロパンアミドの製造
2−(メトキシイミノ)−3−(メチルチオ)プロパン酸259mgのジクロロメタン3ml溶液に、オキサリルクロリド2ml、次いでN,N−ジメチルホルムアミド10mgの順に添加し、室温にて1時間撹拌した。撹拌終了後、該反応溶液を、別途調整したN−エチル−1−(ピリジン−3−イル)−1H−1,2,3−トリアゾ−ル−4−アミン200mg及びトリエチルアミン215mgのジクロロメタン3ml溶液に滴下し、室温にて30分撹拌した。反応終了後、該反応混合物を水10ml、次いで飽和炭酸水素ナトリウム水溶液10mlで洗浄した。得られた有機層を、飽和食塩水次いで無水硫酸ナトリウムの順で洗浄・乾燥し、減圧下にて溶媒を留去した。得られた残留物を、n−ヘキサン−酢酸エチル(7:3〜3:7のグラジエント)にて溶出する中圧分取液体クロマトグラフィーにて精製し、目的物100mgを白色結晶として得た。
融点;101−105℃
合成例2
2−(メトキシイミノ)−N−{3−メチル−5−(ピリジン−3−イル)−1,3,4−チアジアゾール−2(3H)−イリデン}−3−(メチルチオ)プロパンアミドの製造(本発明化合物2−001)
工程1
3−メチル−5−(ピリジン−3−イル)−1,3,4−チアジアゾール−2(3H)−イミンの製造
ジャーナル オブ オーガニック ケミストリー 1959年,24巻,1925頁記載の方法により合成した3−{(2−メチルヒドラゾノ)メチル}ピリジン1gのジクロロメタン50ml溶液に、臭素1.2gを添加した。室温にて2時間撹拌した後、該反応溶液を減圧下で濃縮した。得られた残留物にエタノール50ml及びチオシアン酸カリウム1gを順次添加し、室温にて一晩撹拌した。反応終了後、該反応溶液を減圧下にて溶媒を留去し、得られた残留物に飽和炭酸水素ナトリウム水溶液50mlを添加した後、酢酸エチル50mlにて抽出した。得られた有機層を無水硫酸ナトリウムで乾燥し、減圧下にて溶媒を留去して、目的物700mgを黒色粘性物質として得た。この化合物は精製せずにそのまま次の工程に用いた。
[Synthesis example]
Synthesis example 1
Preparation of N-ethyl-2- (methoxyimino) -3- (methylthio) -N- {1- (pyridin-3-yl) -1H-1,2,3-triazol-4-yl} propanamide (present Invention Compound 1-001)
Process 1
Production of 1- (pyridin-3-yl) -1H-1,2,3-triazol-4-amide Bioorganic and Medicinal Chemistry Letters 2008, Vol. 18, p. 1195 To a solution of 1.9 g of pyridine-3-yl) -1H-1,2,3-triazol-4-carboxylic acid in 20 ml of dichloromethane, 3.8 g of oxalyl chloride and 20 mg of N, N-dimethylformamide were successively added at room temperature. Added. The reaction mixture was stirred at room temperature for 30 minutes, and then the solvent was distilled off under reduced pressure. The residue obtained after distilling off the solvent was dissolved in 5 ml of dichloromethane and poured into 30 ml of 28% aqueous ammonia solution. The reaction mixture was stirred at room temperature for 2 hours, and the precipitated solid was removed by filtration. The obtained solid was washed with water and dried to obtain 1.4 g of the desired product as a brown solid.
1 H NMR (measurement solvent DMSO-d6) δ 9.34 (s, 1H), 9.18 (d, J = 2.4 Hz, 1H), 8.72 (d, J = 4.8 Hz, 1H), 8 .38 (d, J = 8.1 Hz, 1H), 8.05 (brs, 1H), 7.70-7.60 (m, 2H)
Melting point: 260-263 ° C
Process 2
Preparation of methyl {1- (pyridin-3-yl) -1H-1,2,3-triazol-4-yl} carbamate 1- (pyridin-3-yl) -1H-1,2,3-triazo -To a solution of 900 mg of 4-l-amide in 60 ml of methanol, 4.9 g of an 8 wt% aqueous sodium hypochlorite solution was added at room temperature. After completion of the addition, the mixture was stirred for 20 hours under reflux with heating. After completion of the reaction, the reaction mixture was allowed to cool to room temperature, and then the solvent was distilled off under reduced pressure. To the residue obtained after distilling off the solvent, 50 ml of water was added and extracted with 200 ml of ethyl acetate. The obtained organic layer was dehydrated and dried over anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure. The residue obtained after distilling off the solvent was purified by medium pressure preparative liquid chromatography eluting with ethyl acetate-methanol [10: 1 (volume ratio, the same shall apply hereinafter)] to obtain 700 mg of the objective product as white. Obtained as a solid.
1 H NMR (measurement solvent CDCl 3 ) δ 9.06 (d, J = 2.4 Hz, 1H), 8.72 (dd, J = 1.5, 4.8 Hz, 1H), 8.29 (s, 1H ), 8.13 (ddd, J = 1.5, 2.4, 8.4 Hz, 1H), 7.72 (brs, 1H), 7.51 (dd, J = 4.8, 8.4 Hz, 1H), 3.86 (s, 3H)
Melting point: 168-169 ° C
Process 3
Preparation of methyl ethyl {1- (pyridin-3-yl) -1H-1,2,3-triazol-4-yl} carbamate 60% by weight sodium hydride (dispersed in mineral oil) 165 mg N, N- To 5 ml of dimethylformamide solution, 600 mg of methyl {1- (pyridin-3-yl) -1H-1,2,3-triazol-4-yl} carbamate was added under ice cooling. After the addition, the temperature was raised to room temperature and stirred for 30 minutes. 468 mg of ethyl iodide was added to the reaction mixture, and stirring was further continued at room temperature for 1 hour. After completion of the reaction, the reaction mixture was poured into ice water and extracted with 100 ml of ethyl acetate. The obtained organic layer was dehydrated and dried over anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure. The residue was purified by medium pressure preparative liquid chromatography eluting with n-hexane-ethyl acetate (15:85) to obtain 500 mg of the desired product as a white solid.
1 H NMR (measurement solvent CDCl 3 ) δ 9.05 (d, J = 2.4 Hz, 1H), 8.70 (d, J = 4.5 Hz, 1H), 8.43 (s, 1H), 8. 14 (m, 1H), 7.50 (dd, J = 4.5, 8.4 Hz, 1H), 4.18 (q, J = 7.2 Hz, 2H), 3.88 (s, 3H), 1.33 (t, J = 7.2 Hz, 3H)
Melting point: 161-163 ° C
Process 4
Preparation of N-ethyl-1- (pyridin-3-yl) -1H-1,2,3-triazol-4-amine Methyl ethyl {1- (pyridin-3-yl) -1H-1,2, To a solution of 500 mg of 3-triazol-4-yl} carbamate in 12 ml of 1,4-dioxane, 12 ml of 1N aqueous sodium hydroxide solution was added and stirred at 100 ° C. for 2 hours. After completion of the reaction, the reaction mixture was allowed to cool to room temperature, 200 ml of water was added, and the mixture was extracted 3 times with 100 m of ethyl acetate. The obtained organic layers were mixed, dehydrated and dried over anhydrous sodium sulfate. The solvent was distilled off under reduced pressure to obtain 400 mg of the desired product as a pale yellow solid.
1 H NMR (measurement solvent CDCl 3 ) δ 8.96 (d, J = 2.4 Hz, 1H), 8.63 (dd, J = 1.5, 4.8 Hz, 1H), 8.10 (ddd, J = 1.5, 2.4, 8.4 Hz, 1H), 7.45 (dd, J = 4.8, 8.4 Hz, 1H), 7.25 (s, 1H), 3.97 (brs, 1H), 3.19 (q, J = 7.2 Hz, 2H), 1.29 (t, J = 7.2 Hz, 3H)
Process 5
Preparation of N-ethyl-2- (methoxyimino) -3- (methylthio) -N- {1- (pyridin-3-yl) -1H-1,2,3-triazol-4-yl} propanamide 2- To a solution of (methoxyimino) -3- (methylthio) propanoic acid (259 mg) in dichloromethane (3 ml) was added oxalyl chloride (2 ml) and then N, N-dimethylformamide (10 mg) in that order, and the mixture was stirred at room temperature for 1 hour. After completion of the stirring, the reaction solution was added to a separately prepared solution of N-ethyl-1- (pyridin-3-yl) -1H-1,2,3-triazol-4-amine (200 mg) and triethylamine (215 mg) in dichloromethane (3 ml). The solution was added dropwise and stirred at room temperature for 30 minutes. After completion of the reaction, the reaction mixture was washed with 10 ml of water and then with 10 ml of saturated aqueous sodium hydrogen carbonate solution. The obtained organic layer was washed and dried in the order of saturated brine and then anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure. The obtained residue was purified by medium pressure preparative liquid chromatography eluting with n-hexane-ethyl acetate (gradient of 7: 3 to 3: 7) to obtain 100 mg of the desired product as white crystals.
Melting point: 101-105 ° C
Synthesis example 2
Preparation of 2- (methoxyimino) -N- {3-methyl-5- (pyridin-3-yl) -1,3,4-thiadiazole-2 (3H) -ylidene} -3- (methylthio) propanamide ( The present compound 2-001)
Process 1
Production of 3-methyl-5- (pyridin-3-yl) -1,3,4-thiadiazole-2 (3H) -imine 3- of synthesized by the method described in Journal of Organic Chemistry 1959, 24, 1925 1.2 g of bromine was added to a solution of 1 g of {(2-methylhydrazono) methyl} pyridine in 50 ml of dichloromethane. After stirring at room temperature for 2 hours, the reaction solution was concentrated under reduced pressure. To the obtained residue, 50 ml of ethanol and 1 g of potassium thiocyanate were sequentially added and stirred overnight at room temperature. After completion of the reaction, the solvent was distilled off from the reaction solution under reduced pressure, and 50 ml of a saturated aqueous sodium hydrogen carbonate solution was added to the resulting residue, followed by extraction with 50 ml of ethyl acetate. The obtained organic layer was dried over anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure to obtain 700 mg of the desired product as a black viscous substance. This compound was directly used in the next step without purification.

工程2
2−(メトキシイミノ)−N−{3−メチル−5−(ピリジン−3−イル)−1,3,4−チアジアゾール−2(3H)−イリデン}−3−(メチルチオ)プロパンアミドの製造
2−(メトキシイミノ)−3−(メチルチオ)プロパン酸200mgのジクロロメタン10ml溶液に、室温にてオキサリルクロリド200mg、次いでN,N−ジメチルホルムアミド10mgの順に添加した。添加終了後、同温度にて1時間撹拌した。反応終了後、減圧下にて溶媒を留去した。得られた残留物を、別途調整した3−メチル−5−(ピリジン−3−イル)−1,3,4−チアジアゾール−2(3H)−イミン115mg及びトリエチルアミン1gのジクロロメタン5ml、アセトン3ml及び酢酸エチル3mlの溶液に添加した。添加終了後、室温にて3時間間撹拌した。反応終了後、該反応溶液から減圧下にて溶媒を留去した後、得られた残留物をn−ヘキサン−酢酸エチル(3:2)にて溶出するシリカゲルクロマトグラフィーにて精製し、目的物50mgを薄黄色樹脂状物として得た。
H NMR(CDCl,MeSi,300MHz)δ9.09(d,J=1.5Hz,1H),8.73(d,J=4.8Hz,1H),8.15−8.05(m,1H)、7.50−7.40(m,1H),4.12(s,3H),4.11(s,3H),3.78(s,2H),2.16(s,3H)
合成例3
2−(メトキシイミノ)−N−{1−メチル−3−(ピリジン−3−イル)−1H−ピラゾール−5−イル}−3−(メチルチオ)ブタンアミドの製造(本発明化合物4−001)
2−(メトキシイミノ)−3−(メチルチオ)ブタン酸0.56gのジクロロメタン5ml溶液に、室温にてオキサリルクロリド0.47g、次いでN,N−ジメチルホルムアミド10mgの順に添加した。添加終了後、同温度にて2時間撹拌した。反応終了後、減圧下にて溶媒を留去した。得られた残留物を、別途調整した1−メチル−3−(ピリジン−3−イル)−1H−ピラゾール−5−アミン0.5g及びピリジン0.57gのジクロロメタン5ml溶液に添加し、室温にて30分間撹拌した。反応終了後、該反応溶液に飽和炭酸水素ナトリウム水溶液を添加し、有機層を分液にて取り出した。得られた有機層を、水洗した後、飽和食塩水次いで無水硫酸ナトリウムの順で洗浄・乾燥し、減圧下にて溶媒を留去した。得られた残留物をn−ヘキサン−酢酸エチル(1:1〜0:1のグラジエント)にて溶出する中圧分取液体クロマトグラフィーにて精製し、目的物265mgを薄黄色結晶として得た。
融点;81−91℃
合成例4
2−(メトキシイミノ)−N−{2−メチル−4−(ピリジン−3−イル)−1H−イミダゾール−1−イル}−3−(メチルチオ)ペンタンアミドの製造
工程1
2−メチル−4−(ピリジン−3−イル)−1H−イミダゾール−1−アミン 塩酸塩の製造
国際公開第2012/061288号明細書に記載の方法に準じて合成したtert−ブチル {2−メチル−4−(ピリジン−3−イル)−1H−イミダゾール−1−イル}カーバメート350mgの1,4−ジオキサン5ml溶液に、約4M塩化水素の1,4−ジオキサン溶液10mlを添加した。添加終了後、該反応溶液を室温にて一晩撹拌した。反応終了後、該反応溶液中に析出した固体をろ過によりろ別し、目的物0.25gを薄茶色固体として得た。融点;195−200℃
工程2
2−(メトキシイミノ)−N−{2−メチル−4−(ピリジン−3−イル)−1H−イミダゾール−1−イル}−3−(メチルチオ)ペンタンアミドの製造
2−(メトキシイミノ)−3−(メチルチオ)ペンタン酸100mgのジクロロメタン5ml溶液に、オキサリルクロリド0.1g、次いでN,N−ジメチルホルムアミド5mgの順に添加した。添加終了後、該反応溶液を室温にて1時間撹拌した。撹拌終了後、該反応溶液を、別途調整した2−メチル−4−(ピリジン−3−イル)−1H−イミダゾール−1−アミン 塩酸塩120mg及びピリジン210mgのジクロロメタン5ml溶液に滴下した。滴下終了後、該反応溶液を室温にて2時間撹拌した。反応終了後、該反応溶液を水10ml、次いで飽和炭酸水素ナトリウム水溶液10mlで洗浄した。得られた有機層を、飽和食塩水次いで無水硫酸ナトリウムの順で洗浄・乾燥し、減圧下にて溶媒を留去した。得られた残留物を、n−ヘキサン−アセトン(2:1)にて溶出するシリカゲルクロマトグラフィーにて精製し、目的物81mgを橙色結晶として得た。
融点;148−150℃
参考例1
2−(メトキシイミノ)−3−(メチルチオ)プロパン酸の製造
工程1
エチル 2−(メトキシイミノ)−3−(メチルチオ)プロパノエートの製造
エチル 3−ブロモ−2−(メトキシイミノ)プロパノエート2.0gのN,N−ジメチルホルムアミド30mlの溶液に、メチルメルカプタンナトリウム750mgを添加し、室温にて2時間攪拌した。攪拌終了後、80℃に昇温した後、同温度で1時間撹拌を継続した。反応終了後、該反応混合物に水30mlを添加し、酢酸エチル50mlで抽出した。得られた有機層を、飽和炭酸水素ナトリウム水溶液で洗浄した後、飽和食塩水次いで無水硫酸ナトリウムの順で洗浄・乾燥した。減圧下にて溶媒を留去し、目的物2gを薄黄色油状物として得た。
H NMR(CDCl,MeSi,300MHz)δ4.34(q,J=7.2Hz,2H),4.04(s,3H),3.55(s,2H),2.10(s,3H),1.35(t,J=7.2Hz,3H)
工程2
2−(メトキシイミノ)−3−(メチルチオ)プロパン酸の製造
エチル 2−(メトキシイミノ)−3−(メチルチオ)プロパノエート1.84gの水10ml及びエタノール10mlの混合溶液に、水酸化ナトリウム430mgを添加し、室温にて2日間撹拌した。反応終了後、該反応溶液に1N塩酸水溶液を添加し、該反応溶液のpHを2とした後、酢酸エチル20mlで2回抽出した。得られた有機層を、飽和食塩水次いで無水硫酸ナトリウムの順で洗浄・乾燥し、減圧下にて溶媒を留去した。得られた固体を、ヘキサン:イソプロピルエーテル(5:1)の混合溶液6mlで洗浄し、目的物0.4gを黄白色固体として得た。
H NMR(CDCl,MeSi,300MHz)δ4.08(s,3H),3.53(s,2H),2.14(s,3H)
参考例2
2−(メトキシイミノ)−3−(メチルチオ)ブタン酸の製造
工程1
エチル 2−(メトキシイミノ)−3−(トシルオキシ)ブタノエートの製造(化合物D−001)
独国特許出願公開第3220524号明細書に記載の方法に従って合成したエチル 3−ヒドロキシ−2−(メトキシイミノ)ブタノエート1.63gのジクロロメタン10ml溶液に、トリエチルアミン2.36g、p−トルエンスルホニルクロリド2.14g及び4−ジメチルアミノピリジン0.34gを順次添加した。添加終了後、該反応混合物を室温にて一晩撹拌した。反応終了後、該反応溶液に飽和炭酸水素ナトリウム水溶液20mlを添加し、酢酸エチル30mlにて抽出した。得られた有機層を水洗した後、飽和食塩水次いで無水硫酸ナトリウムの順で洗浄・乾燥し、減圧下にて溶媒を留去した。得られた残渣をn−ヘキサン−酢酸エチル(5:1)にて溶出する中圧分取液体クロマトグラフィーにて精製し、目的物0.8gを黄色油状物として得た。
H NMR(CDCl,MeSi,300MHz)δ7.78(d,J=8.1Hz,2H),7.32(d,J=8.1Hz,2H),5.31(q,J=6.9Hz,1H),4.28−4.16(m,2H),3.82(s,3H),2.44(s,3H),1.53(d,J=6.9Hz,3H), 1.27(t,J=7.2Hz,3H)
工程2
エチル 2−(メトキシイミノ)−3−(メチルチオ)ブタノエートの製造(化合物E−001)
エチル 2−(メトキシイミノ)−3−(トシルオキシ)ブタノエート0.8gのN,N−ジメチルホルムアミド5ml溶液に、0℃にてメチルメルカプタンナトリウム0.2gを添加した。添加終了後、同温度にて30分撹拌した。反応終了後、該反応溶液に水10mlを添加し、酢酸エチル10mlにて抽出した。得られた有機層を、飽和食塩水次いで無水硫酸ナトリウムの順で洗浄・乾燥した後、減圧下にて溶媒を留去し、目的物0.45gを黄色油状物として得た。
H NMR(CDCl,MeSi,300MHz)δ4.32(q,J=7.2Hz,2H),3.87(s,3H),3.60(q,J=7.2Hz,1H),2.05(s,3H),1.46(d,J=7.2Hz,3H), 1.33(t,J=7.2Hz,3H) 工程3
2−(メトキシイミノ)−3−(メチルチオ)ブタン酸の製造(化合物F−001)
エチル 2−(メトキシイミノ)−3−(メチルチオ)ブタノエート0.45gのエタノール5ml溶液に、1N水酸化ナトリウム水溶液3.3mlを添加した。添加終了後、室温にて2時間撹拌した。反応終了後、該反応溶液から減圧下にてエタノールを留去した。得られた残留物を酢酸エチルで洗浄した。洗浄終了後、1N塩酸水溶液でpH3とした後、酢酸エチル(5mlx2)にて抽出した。得られた有機層を、飽和食塩水次いで無水硫酸ナトリウムの順で洗浄・乾燥した後、減圧下にて溶媒を留去し、目的物0.4gを黄色油状物として得た。
H NMR(CDCl,MeSi,300MHz)δ4.06(s,3H),3.88−3.77(m,1H),2.06(s,3H),1.49(d,J=6.9Hz,3H)(COHのプロトンピークは観測されなかった。)
また、参考例2と同様の合成法にて、以下の中間体を合成した。
Process 2
Preparation of 2- (methoxyimino) -N- {3-methyl-5- (pyridin-3-yl) -1,3,4-thiadiazole-2 (3H) -ylidene} -3- (methylthio) propanamide 2 200 mg of oxalyl chloride and then 10 mg of N, N-dimethylformamide were added to a solution of 200 mg of-(methoxyimino) -3- (methylthio) propanoic acid in 10 ml of dichloromethane at room temperature. After completion of the addition, the mixture was stirred at the same temperature for 1 hour. After completion of the reaction, the solvent was distilled off under reduced pressure. The residue thus obtained was prepared by separately preparing 3-methyl-5- (pyridin-3-yl) -1,3,4-thiadiazole-2 (3H) -imine (115 mg) and triethylamine (1 g) in dichloromethane (5 ml), acetone (3 ml) and acetic acid. Added to a solution of 3 ml of ethyl. After completion of the addition, the mixture was stirred at room temperature for 3 hours. After completion of the reaction, the solvent was distilled off from the reaction solution under reduced pressure, and the obtained residue was purified by silica gel chromatography eluting with n-hexane-ethyl acetate (3: 2). 50 mg was obtained as a pale yellow resin.
1 H NMR (CDCl 3 , Me 4 Si, 300 MHz) δ 9.09 (d, J = 1.5 Hz, 1H), 8.73 (d, J = 4.8 Hz, 1H), 8.15-8.05 (M, 1H), 7.50-7.40 (m, 1H), 4.12 (s, 3H), 4.11 (s, 3H), 3.78 (s, 2H), 2.16 ( s, 3H)
Synthesis example 3
Preparation of 2- (methoxyimino) -N- {1-methyl-3- (pyridin-3-yl) -1H-pyrazol-5-yl} -3- (methylthio) butanamide (present compound 4-001)
To a solution of 0.56 g of 2- (methoxyimino) -3- (methylthio) butanoic acid in 5 ml of dichloromethane was added 0.47 g of oxalyl chloride and then 10 mg of N, N-dimethylformamide at room temperature. After completion of the addition, the mixture was stirred at the same temperature for 2 hours. After completion of the reaction, the solvent was distilled off under reduced pressure. The obtained residue was added to a separately prepared solution of 0.5 g of 1-methyl-3- (pyridin-3-yl) -1H-pyrazol-5-amine and 0.57 g of pyridine in 5 ml of dichloromethane at room temperature. Stir for 30 minutes. After completion of the reaction, a saturated aqueous sodium hydrogen carbonate solution was added to the reaction solution, and the organic layer was taken out by liquid separation. The obtained organic layer was washed with water, then washed and dried in the order of saturated brine and then anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure. The obtained residue was purified by medium pressure preparative liquid chromatography eluting with n-hexane-ethyl acetate (1: 1 to 0: 1 gradient) to obtain 265 mg of the desired product as pale yellow crystals.
Melting point: 81-91 ° C
Synthesis example 4
Production of 2- (methoxyimino) -N- {2-methyl-4- (pyridin-3-yl) -1H-imidazol-1-yl} -3- (methylthio) pentanamide Step 1
Preparation of 2-methyl-4- (pyridin-3-yl) -1H-imidazol-1-amine hydrochloride Tert-butyl synthesized according to the method described in WO 2012/061288 {2-methyl To a solution of 350 mg of -4- (pyridin-3-yl) -1H-imidazol-1-yl} carbamate in 5 ml of 1,4-dioxane, 10 ml of a 1,4-dioxane solution of about 4M hydrogen chloride was added. After completion of the addition, the reaction solution was stirred overnight at room temperature. After completion of the reaction, the solid precipitated in the reaction solution was filtered off to obtain 0.25 g of the desired product as a light brown solid. Melting point: 195-200 ° C
Process 2
Preparation of 2- (methoxyimino) -N- {2-methyl-4- (pyridin-3-yl) -1H-imidazol-1-yl} -3- (methylthio) pentanamide 2- (methoxyimino) -3 -To a solution of 100 mg of (methylthio) pentanoic acid in 5 ml of dichloromethane, 0.1 g of oxalyl chloride and then 5 mg of N, N-dimethylformamide were added in this order. After completion of the addition, the reaction solution was stirred at room temperature for 1 hour. After completion of the stirring, the reaction solution was added dropwise to a solution of 2-methyl-4- (pyridin-3-yl) -1H-imidazol-1-amine hydrochloride (120 mg) and pyridine (210 mg) in dichloromethane (5 ml). After completion of the dropwise addition, the reaction solution was stirred at room temperature for 2 hours. After completion of the reaction, the reaction solution was washed with 10 ml of water and then with 10 ml of a saturated aqueous sodium hydrogen carbonate solution. The obtained organic layer was washed and dried in the order of saturated brine and then anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure. The obtained residue was purified by silica gel chromatography eluting with n-hexane-acetone (2: 1) to obtain 81 mg of the objective product as orange crystals.
Melting point: 148-150 ° C
Reference example 1
Production of 2- (methoxyimino) -3- (methylthio) propanoic acid Step 1
Preparation of ethyl 2- (methoxyimino) -3- (methylthio) propanoate To a solution of 2.0 g of ethyl 3-bromo-2- (methoxyimino) propanoate in 30 ml of N, N-dimethylformamide was added 750 mg of sodium methyl mercaptan. The mixture was stirred at room temperature for 2 hours. After completion of stirring, the temperature was raised to 80 ° C., and stirring was continued for 1 hour at the same temperature. After completion of the reaction, 30 ml of water was added to the reaction mixture and extracted with 50 ml of ethyl acetate. The obtained organic layer was washed with a saturated aqueous solution of sodium hydrogen carbonate, washed with saturated brine and then dried over anhydrous sodium sulfate in that order. The solvent was distilled off under reduced pressure to obtain 2 g of the desired product as a pale yellow oil.
1 H NMR (CDCl 3 , Me 4 Si, 300 MHz) δ 4.34 (q, J = 7.2 Hz, 2H), 4.04 (s, 3H), 3.55 (s, 2H), 2.10 ( s, 3H), 1.35 (t, J = 7.2 Hz, 3H)
Process 2
Preparation of 2- (methoxyimino) -3- (methylthio) propanoic acid Ethyl 2- (methoxyimino) -3- (methylthio) propanoate 430 mg of sodium hydroxide was added to a mixed solution of 1.84 g of water and 10 ml of ethanol. And stirred at room temperature for 2 days. After completion of the reaction, 1N aqueous hydrochloric acid solution was added to the reaction solution to adjust the pH of the reaction solution to 2, and then extracted twice with 20 ml of ethyl acetate. The obtained organic layer was washed and dried in the order of saturated brine and then anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure. The obtained solid was washed with 6 ml of a mixed solution of hexane: isopropyl ether (5: 1) to obtain 0.4 g of the objective product as a yellowish white solid.
1 H NMR (CDCl 3 , Me 4 Si, 300 MHz) δ 4.08 (s, 3H), 3.53 (s, 2H), 2.14 (s, 3H)
Reference example 2
Production of 2- (methoxyimino) -3- (methylthio) butanoic acid Step 1
Preparation of ethyl 2- (methoxyimino) -3- (tosyloxy) butanoate (Compound D-001)
To a solution of 1.63 g of ethyl 3-hydroxy-2- (methoxyimino) butanoate synthesized in accordance with the method described in German Patent Application No. 3220524 in 10 ml of dichloromethane, 2.36 g of triethylamine and p-toluenesulfonyl chloride. 14 g and 4-dimethylaminopyridine 0.34 g were added sequentially. After the addition was complete, the reaction mixture was stirred overnight at room temperature. After completion of the reaction, 20 ml of saturated aqueous sodium hydrogen carbonate solution was added to the reaction solution, and extracted with 30 ml of ethyl acetate. The obtained organic layer was washed with water, then washed and dried with saturated brine and then anhydrous sodium sulfate in this order, and the solvent was distilled off under reduced pressure. The obtained residue was purified by medium pressure preparative liquid chromatography eluting with n-hexane-ethyl acetate (5: 1) to obtain 0.8 g of the objective product as a yellow oil.
1 H NMR (CDCl 3 , Me 4 Si, 300 MHz) δ 7.78 (d, J = 8.1 Hz, 2H), 7.32 (d, J = 8.1 Hz, 2H), 5.31 (q, J = 6.9 Hz, 1H), 4.28-4.16 (m, 2H), 3.82 (s, 3H), 2.44 (s, 3H), 1.53 (d, J = 6.9 Hz) , 3H), 1.27 (t, J = 7.2 Hz, 3H)
Process 2
Preparation of ethyl 2- (methoxyimino) -3- (methylthio) butanoate (Compound E-001)
To a solution of 0.8 g of ethyl 2- (methoxyimino) -3- (tosyloxy) butanoate in 5 ml of N, N-dimethylformamide was added 0.2 g of sodium methyl mercaptan at 0 ° C. After completion of the addition, the mixture was stirred at the same temperature for 30 minutes. After completion of the reaction, 10 ml of water was added to the reaction solution and extracted with 10 ml of ethyl acetate. The obtained organic layer was washed and dried in the order of saturated brine and then anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure to obtain 0.45 g of the desired product as a yellow oil.
1 H NMR (CDCl 3 , Me 4 Si, 300 MHz) δ 4.32 (q, J = 7.2 Hz, 2H), 3.87 (s, 3H), 3.60 (q, J = 7.2 Hz, 1H) ), 2.05 (s, 3H), 1.46 (d, J = 7.2 Hz, 3H), 1.33 (t, J = 7.2 Hz, 3H) Step 3
Production of 2- (methoxyimino) -3- (methylthio) butanoic acid (Compound F-001)
To a solution of ethyl 2- (methoxyimino) -3- (methylthio) butanoate 0.45 g in ethanol 5 ml was added 1N sodium hydroxide aqueous solution 3.3 ml. After completion of the addition, the mixture was stirred at room temperature for 2 hours. After completion of the reaction, ethanol was distilled off from the reaction solution under reduced pressure. The resulting residue was washed with ethyl acetate. After the completion of washing, the pH was adjusted to 3 with 1N aqueous hydrochloric acid solution, followed by extraction with ethyl acetate (5 ml × 2). The obtained organic layer was washed and dried in the order of saturated brine and then anhydrous sodium sulfate, and the solvent was evaporated under reduced pressure to obtain 0.4 g of the objective product as a yellow oil.
1 H NMR (CDCl 3 , Me 4 Si, 300 MHz) δ 4.06 (s, 3H), 3.88-3.77 (m, 1H), 2.06 (s, 3H), 1.49 (d, J = 6.9 Hz, 3H) (The proton peak of CO 2 H was not observed.)
In addition, the following intermediate was synthesized by the same synthesis method as in Reference Example 2.

メチル 2−(メトキシイミノ)−3−(メチルチオ)ペンタノエート;
H NMR(CDCl,MeSi,300MHz)δ3.89(s,3H),3.84(s,3H),3.33(t,J=7.5Hz,1H),2.04(s,3H),1.93−1.60(m,2H),1.05(t,J=7.5Hz,3H)
メチル 3−(アリルチオ)−2−(メトキシイミノ)ペンタノエート(2種の異性体混合物 異性体比7:3);
異性体比7
H NMR(CDCl,MeSi,300MHz)δ5.85−5.66(m,1H),5.18−5.02(m,2H),3.87(s,3H),3.83(s,3H),3.43−3.02(m,2H),2.65−2.45(m,1H),2.05−1.60(m,2H),1.30−0.87(m,3H)
異性体比3
H NMR(CDCl,MeSi,300MHz)δ5.85−5.66(m,1H),5.18−5.02(m,2H),4.00(s,3H),3.83(s,3H),3.43−3.02(m,2H),2.65−2.45(m,1H),2.05−1.60(m,2H),1.30−0.87(m,3H)
2−(メトキシイミノ)−3−(メチルチオ)ペンタン酸;
H NMR(CDCl,MeSi,300MHz)δ4.03(s,3H),3.53(t,J=7.8Hz,1H),2.04(s,3H),1.96−1.70(m,2H),1.04(t,J=7.2Hz,3H)(COHのプロトンピークは観測されなかった。)
3−(アリルチオ)−2−(メトキシイミノ)ペンタン酸(2種の異性体混合物 異性体比7:3);
異性体比7
H NMR(CDCl,MeSi,300MHz)δ5.90−5.70(m,1H),5.22−5.06(m,2H),4.02(s,3H),3.60−3.04(m,2H),2.70−2.48(m,1H),2.10−1.72(m,2H),1.08−0.85(m,3H)
異性体比3
H NMR(CDCl,MeSi,300MHz)δ5.90−5.70(m,1H),5.22−5.06(m,2H),4.05(s,3H),3.60−3.04(m,2H),2.70−2.48(m,1H),2.10−1.72(m,2H),1.08−0.85(m,3H)
参考例3
1−メチル−3−(ピリジン−3−イル)−1H−ピラゾール−5−アミンの製造
60重量%水素化ナトリウム(鉱油中に分散)2.9gのテトラヒドロフラン溶液に、0℃にてアセトニトリル1.5g、ニコチン酸エチル5.0gを順次添加し、テトラヒドロフランの還流温度で4時間撹拌した。反応終了後、該反応溶液を氷水50mlに添加し、濃塩酸にてpH2とした後、エタノール150ml、メチルヒドラジン2.3gを添加し、エタノールの還流温度にて4時間撹拌した。反応終了後、該反応溶液を減圧下にて溶媒を留去し、得られた残留物に1N塩酸水溶液を添加してpH1とした後、酢酸エチルで洗浄した。この水層を1N水酸化ナトリウム水溶液で中和し、酢酸エチル50mlにて3回抽出した。得られた有機層を飽和食塩水次いで無水硫酸ナトリウムの順で洗浄・乾燥した後、減圧下にて溶媒を留去し、目的物3.1gを橙色結晶として得た。
融点;120−128℃
参考例4
5−クロロ−N−エチル−2−(ピリジン−3−イル)−2H−1,2,3−トリアゾ−ル−4−アミンの製造
工程1
N−{5−クロロ−2−(ピリジン−3−イル)−2H−1,2,3−トリアゾ−ル−4−イル}アセトアミドの製造
テトラへドロン 1993年,49巻,5339頁記載の方法に準して合成した4−アセトアミド−2−(ピリジン−3−イル)−2H−1,2,3−トリアゾ−ル 1−オキシド1.0gのオキシ塩化リン3ml溶液を、110℃で3時間撹拌した。反応完結後、反応溶液を水20mlに滴下した。滴下終了後、該反応溶液に1N水酸化ナトリウム水溶液を添加してpH6〜7とし、該反応溶液中に析出した固体を、減圧ろ過にてろ別した。得られた個体を水、酢酸エチルの順番で洗浄した。洗浄後に得られた固体を減圧乾燥した後、目的物0.64gを黄土色結晶として得た。
融点;215−225℃
工程2
N−{5−クロロ−2−(ピリジン−3−イル)−2H−1,2,3−トリアゾ−ル−4−イル}−N−エチルアセトアミドの製造
60重量%水素化ナトリウム(鉱油中に分散)96mgのN,N−ジメチルホルムアミド5ml溶液に、氷冷下にてN−{5−クロロ−2−(ピリジン−3−イル)−2H−1,2,3−トリアゾ−ル−4−イル}アセトアミド500mgを添加した。添加終了後、該反応溶液を室温まで昇温し、30分間撹拌した。撹拌終了後、該反応溶液にヨウ化エチル360mgを添加し、更に室温にて2時間撹拌を継続した。反応終了後、該反応溶液を氷水に注ぎ、酢酸エチル10mlにて抽出した。得られた有機層を無水硫酸ナトリウムにて脱水・乾燥後、減圧下にて溶媒を留去した。残留物をn−ヘキサン−酢酸エチル(3:1)にて溶出する中圧分取液体クロマトグラフィーにて精製し、目的物377mgを黄色油状物として得た。
H NMR(測定溶媒CDCl)δ9.30(d,J=2.4Hz,1H),8.66(d,J=4.8Hz,1H),8.32−8.24(m,1H),7.46(dd,J=8.4,4.8Hz,1H),3.78(q,J=7.2Hz,2H),1.96(brs,3H),1.18(t,J=7.2Hz,3H)
工程3
5−クロロ−N−エチル−2−(ピリジン−3−イル)−2H−1,2,3−トリアゾ−ル−4−アミンの製造
N−{5−クロロ−2−(ピリジン−3−イル)−2H−1,2,3−トリアゾ−ル−4−イル}−N−エチルアセトアミド300mgのエタノール10ml溶液に、水0.5ml及び濃硫酸150mgを添加し、加熱還流下にて12時間攪拌した。撹拌終了後、該反応溶液に、水0.5ml及び濃硫酸300mgを添加し、加熱還流下にて12時間攪拌を継続した。反応終了後、該反応溶液を室温まで冷却し、1N水酸化ナトリウム水溶液を添加してpH7〜8とし、該反応溶液中に析出した固体を、減圧濾過にてろ別。得られた固体を水洗し、減圧乾燥後、目的物213mgを黄白色固体として得た。
融点;103−108℃
本発明化合物は、前記製造法及び実施例に準じて製造することができる。合成例1〜3と同様に製造した本発明化合物の例を第2表乃至第9表に示し、それらの物性値を第10表に示すが、本発明はこれらのみに限定されるものではない。
Methyl 2- (methoxyimino) -3- (methylthio) pentanoate;
1 H NMR (CDCl 3 , Me 4 Si, 300 MHz) δ 3.89 (s, 3H), 3.84 (s, 3H), 3.33 (t, J = 7.5 Hz, 1H), 2.04 ( s, 3H), 1.93-1.60 (m, 2H), 1.05 (t, J = 7.5 Hz, 3H)
Methyl 3- (allylthio) -2- (methoxyimino) pentanoate (mixture of two isomers, isomer ratio 7: 3);
Isomeric ratio 7
1 H NMR (CDCl 3 , Me 4 Si, 300 MHz) δ 5.85-5.66 (m, 1H), 5.18-5.02 (m, 2H), 3.87 (s, 3H), 3. 83 (s, 3H), 3.43-3.02 (m, 2H), 2.65-2.45 (m, 1H), 2.05-1.60 (m, 2H), 1.30- 0.87 (m, 3H)
Isomer ratio 3
1 H NMR (CDCl 3 , Me 4 Si, 300 MHz) δ 5.85-5.66 (m, 1H), 5.18-5.02 (m, 2H), 4.00 (s, 3H), 3. 83 (s, 3H), 3.43-3.02 (m, 2H), 2.65-2.45 (m, 1H), 2.05-1.60 (m, 2H), 1.30- 0.87 (m, 3H)
2- (methoxyimino) -3- (methylthio) pentanoic acid;
1 H NMR (CDCl 3 , Me 4 Si, 300 MHz) δ 4.03 (s, 3H), 3.53 (t, J = 7.8 Hz, 1H), 2.04 (s, 3H), 1.96- 1.70 (m, 2H), 1.04 (t, J = 7.2 Hz, 3H) (The proton peak of CO 2 H was not observed.)
3- (allylthio) -2- (methoxyimino) pentanoic acid (mixture of two isomers, isomer ratio 7: 3);
Isomeric ratio 7
1 H NMR (CDCl 3 , Me 4 Si, 300 MHz) δ 5.90-5.70 (m, 1H), 5.22-5.06 (m, 2H), 4.02 (s, 3H), 3. 60-3.04 (m, 2H), 2.70-2.48 (m, 1H), 2.10-1.72 (m, 2H), 1.08-0.85 (m, 3H)
Isomer ratio 3
1 H NMR (CDCl 3 , Me 4 Si, 300 MHz) δ 5.90-5.70 (m, 1H), 5.22-5.06 (m, 2H), 4.05 (s, 3H), 3. 60-3.04 (m, 2H), 2.70-2.48 (m, 1H), 2.10-1.72 (m, 2H), 1.08-0.85 (m, 3H)
Reference example 3
Preparation of 1-methyl-3- (pyridin-3-yl) -1H-pyrazol-5-amine 60 wt% sodium hydride (dispersed in mineral oil) in 2.9 g tetrahydrofuran solution at 0 ° C. with acetonitrile 1. 5 g and 5.0 g of ethyl nicotinate were sequentially added, and the mixture was stirred at the reflux temperature of tetrahydrofuran for 4 hours. After completion of the reaction, the reaction solution was added to 50 ml of ice water, adjusted to pH 2 with concentrated hydrochloric acid, 150 ml of ethanol and 2.3 g of methyl hydrazine were added, and the mixture was stirred at the reflux temperature of ethanol for 4 hours. After completion of the reaction, the solvent was distilled off from the reaction solution under reduced pressure, and 1N hydrochloric acid aqueous solution was added to the resulting residue to adjust to pH 1, followed by washing with ethyl acetate. The aqueous layer was neutralized with 1N aqueous sodium hydroxide solution and extracted three times with 50 ml of ethyl acetate. The obtained organic layer was washed and dried in the order of saturated brine and then anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure to obtain 3.1 g of the objective product as orange crystals.
Melting point: 120-128 ° C
Reference example 4
Production of 5-chloro-N-ethyl-2- (pyridin-3-yl) -2H-1,2,3-triazol-4-amine Step 1
Preparation of N- {5-chloro-2- (pyridin-3-yl) -2H-1,2,3-triazol-4-yl} acetamide Tetrahedron 1993, 49, 5339 4-acetamido-2- (pyridin-3-yl) -2H-1,2,3-triazol 1-oxide 1.0 g synthesized in a similar manner to 3 ml of phosphorus oxychloride was added at 110 ° C. for 3 hours. Stir. After completion of the reaction, the reaction solution was added dropwise to 20 ml of water. After completion of the dropwise addition, 1N aqueous sodium hydroxide solution was added to the reaction solution to adjust the pH to 6-7, and the solid precipitated in the reaction solution was filtered off under reduced pressure. The obtained solid was washed in the order of water and ethyl acetate. The solid obtained after washing was dried under reduced pressure, and 0.64 g of the desired product was obtained as ocher crystals.
Melting point: 215-225 ° C
Process 2
Preparation of N- {5-chloro-2- (pyridin-3-yl) -2H-1,2,3-triazol-4-yl} -N-ethylacetamide 60% by weight sodium hydride (in mineral oil) Dispersion) N- {5-Chloro-2- (pyridin-3-yl) -2H-1,2,3-triazol-4-l in 96 mg N, N-dimethylformamide 5 ml solution under ice-cooling 500 mg of yl} acetamide was added. After completion of the addition, the reaction solution was warmed to room temperature and stirred for 30 minutes. After the completion of stirring, 360 mg of ethyl iodide was added to the reaction solution, and stirring was further continued at room temperature for 2 hours. After completion of the reaction, the reaction solution was poured into ice water and extracted with 10 ml of ethyl acetate. The obtained organic layer was dehydrated and dried over anhydrous sodium sulfate, and then the solvent was distilled off under reduced pressure. The residue was purified by medium pressure preparative liquid chromatography eluting with n-hexane-ethyl acetate (3: 1) to obtain 377 mg of the desired product as a yellow oil.
1 H NMR (measurement solvent CDCl 3 ) δ 9.30 (d, J = 2.4 Hz, 1H), 8.66 (d, J = 4.8 Hz, 1H), 8.32-8.24 (m, 1H ), 7.46 (dd, J = 8.4, 4.8 Hz, 1H), 3.78 (q, J = 7.2 Hz, 2H), 1.96 (brs, 3H), 1.18 (t , J = 7.2Hz, 3H)
Process 3
Preparation of 5-chloro-N-ethyl-2- (pyridin-3-yl) -2H-1,2,3-triazol-4-amine N- {5-chloro-2- (pyridin-3-yl) ) -2H-1,2,3-triazol-4-yl} -N-ethylacetamide 300 mg of ethanol in 10 ml solution was added 0.5 ml of water and 150 mg of concentrated sulfuric acid and stirred for 12 hours under heating and reflux. did. After completion of the stirring, 0.5 ml of water and 300 mg of concentrated sulfuric acid were added to the reaction solution, and stirring was continued for 12 hours under heating and reflux. After completion of the reaction, the reaction solution is cooled to room temperature, 1N aqueous sodium hydroxide solution is added to adjust the pH to 7-8, and the solid precipitated in the reaction solution is separated by filtration under reduced pressure. The obtained solid was washed with water and dried under reduced pressure to obtain 213 mg of the desired product as a yellowish white solid.
Melting point: 103-108 ° C
This invention compound can be manufactured according to the said manufacturing method and an Example. Examples of the compounds of the present invention produced in the same manner as in Synthesis Examples 1 to 3 are shown in Tables 2 to 9 and their physical properties are shown in Table 10. However, the present invention is not limited to these. .

また、「*1」は樹脂状を表し、「m.p.」は融点を表す。「*2」は樹脂状で、同一構造であるが2種類の異性体混合物の場合を表す。異性体比が判明した場合は、第10表にその比を記載する。   “* 1” represents a resinous shape, and “m.p.” represents a melting point. “* 2” represents a resinous structure having the same structure but a mixture of two isomers. If the isomer ratio is known, the ratio is listed in Table 10.

第10表の記号は下記の意味を表す。
s:シングレット、d:ダブレット、t:トリプレット、q:カルテット、m:マルチプレット、brs:ブロードピーク。
〔第2表〕
The symbols in Table 10 represent the following meanings.
s: singlet, d: doublet, t: triplet, q: quartet, m: multiplet, brs: broad peak.
[Table 2]

Figure 2015147757
Figure 2015147757

―――――――――――――――――――――――――――――――――――――
No. Y Ra Rb-1 m.p.(℃)
―――――――――――――――――――――――――――――――――――――
1-001 O CH2CH3 C(=NOCH3)CH2SCH3 101-105
―――――――――――――――――――――――――――――――――――――
〔第3表〕
―――――――――――――――――――――――――――――――――――――
No. YR a R b-1 mp (℃)
―――――――――――――――――――――――――――――――――――――
1-001 O CH 2 CH 3 C (= NOCH 3 ) CH 2 SCH 3 101-105
―――――――――――――――――――――――――――――――――――――
[Table 3]

Figure 2015147757
Figure 2015147757

―――――――――――――――――――――――――――――――――――――
No. Y R3a Rb-1 m.p.(℃)
―――――――――――――――――――――――――――――――――――――
2-001 O CH3 C(=NOCH3)CH2SCH3 *1
―――――――――――――――――――――――――――――――――――――
〔第4表〕
―――――――――――――――――――――――――――――――――――――
No. YR 3a R b-1 mp (℃)
―――――――――――――――――――――――――――――――――――――
2-001 O CH 3 C (= NOCH 3 ) CH 2 SCH 3 * 1
―――――――――――――――――――――――――――――――――――――
[Table 4]

Figure 2015147757
Figure 2015147757

―――――――――――――――――――――――――――――――――――――
No. Y Ra Rb-1 m.p.(℃)
―――――――――――――――――――――――――――――――――――――
3-001 O H C(=NOCH3)CH3 219-220
3-002 O H C(=NOCH2CH3)CH3 169-171
3-003 O H C(=NOCH3)CH2SCH3 200-202
―――――――――――――――――――――――――――――――――――――
〔第5表〕
―――――――――――――――――――――――――――――――――――――
No. YR a R b-1 mp (℃)
―――――――――――――――――――――――――――――――――――――
3-001 OHC (= NOCH 3 ) CH 3 219-220
3-002 OHC (= NOCH 2 CH 3 ) CH 3 169-171
3-003 OHC (= NOCH 3 ) CH 2 SCH 3 200-202
―――――――――――――――――――――――――――――――――――――
[Table 5]

Figure 2015147757
Figure 2015147757

―――――――――――――――――――――――――――――――――――――
No. Y R3a Ra Rb-1 m.p.(℃)
―――――――――――――――――――――――――――――――――――――
4-001 O CH3 H C(=NOCH3)CH(CH3)SCH3 81-91
4-002 O CH3 H C(=NOCH3)CH(CH3)S(O)CH3 *2(52:48)
4-003 O CH3 H C(=NOCH3)CH(CH3)S(O)2CH3 *2(53:47)
4-004 O CH3 H C(=NOCH3)CH2SCH3 150-155
4-005 O CH3 H C(=NOCH3)CH2S(O)2CH3 157-162
4-006 O CH3 H C(=NOCH3)CH(CH2CH3)SCH2CH=CH2 *1
4-007 O CH3 H C(=NOCH3)CH(CH2CH3)S(O)2CH2CH=CH2 *1
―――――――――――――――――――――――――――――――――――――
〔第6表〕
―――――――――――――――――――――――――――――――――――――
No. YR 3a R a R b-1 mp (℃)
―――――――――――――――――――――――――――――――――――――
4-001 O CH 3 HC (= NOCH 3 ) CH (CH 3 ) SCH 3 81-91
4-002 O CH 3 HC (= NOCH 3 ) CH (CH 3 ) S (O) CH 3 * 2 (52:48)
4-003 O CH 3 HC (= NOCH 3 ) CH (CH 3 ) S (O) 2 CH 3 * 2 (53:47)
4-004 O CH 3 HC (= NOCH 3 ) CH 2 SCH 3 150-155
4-005 O CH 3 HC (= NOCH 3 ) CH 2 S (O) 2 CH 3 157-162
4-006 O CH 3 HC (= NOCH 3 ) CH (CH 2 CH 3 ) SCH 2 CH = CH 2 * 1
4-007 O CH 3 HC (= NOCH 3 ) CH (CH 2 CH 3 ) S (O) 2 CH 2 CH = CH 2 * 1
―――――――――――――――――――――――――――――――――――――
[Table 6]

Figure 2015147757
Figure 2015147757

―――――――――――――――――――――――――――――――――――――
No. Y Ra Rb-1 m.p.(℃)
―――――――――――――――――――――――――――――――――――――
5-001 O H C(=NOCH3)CH(CH3)SCH3 165-175
―――――――――――――――――――――――――――――――――――――
〔第7表〕
―――――――――――――――――――――――――――――――――――――
No. YR a R b-1 mp (℃)
―――――――――――――――――――――――――――――――――――――
5-001 OHC (= NOCH 3 ) CH (CH 3 ) SCH 3 165-175
―――――――――――――――――――――――――――――――――――――
[Table 7]

Figure 2015147757
Figure 2015147757

―――――――――――――――――――――――――――――――――――――
No. Y R3 Ra Rb-1 m.p.(℃)
―――――――――――――――――――――――――――――――――――――
6-001 O CH3 H C(=NOCH3)CH(CH2CH3)SCH3 *1
―――――――――――――――――――――――――――――――――――――
〔第8表〕
―――――――――――――――――――――――――――――――――――――
No. YR 3 R a R b-1 mp (℃)
―――――――――――――――――――――――――――――――――――――
6-001 O CH 3 HC (= NOCH 3 ) CH (CH 2 CH 3 ) SCH 3 * 1
―――――――――――――――――――――――――――――――――――――
[Table 8]

Figure 2015147757
Figure 2015147757

――――――――――――――――――――――――――――――――――――――――
No. Y R3 Ra Rb-1 m.p.(℃)
――――――――――――――――――――――――――――――――――――――――
7-001 O Cl H C(=NOCH3)CH2SCH3 84-87
――――――――――――――――――――――――――――――――――――――――
〔第9表〕
――――――――――――――――――――――――――――――――――――――――
No. YR 3 R a R b-1 mp (℃)
――――――――――――――――――――――――――――――――――――――――
7-001 O Cl HC (= NOCH 3 ) CH 2 SCH 3 84-87
――――――――――――――――――――――――――――――――――――――――
[Table 9]

Figure 2015147757
Figure 2015147757

――――――――――――――――――――――――――――――――――――――――
No. Y R3 Ra Rb-1 m.p.(℃)
――――――――――――――――――――――――――――――――――――――――
8-001 O Cl CH2CH3 C(=NOCH3)CH2SCH3 148-150
8-002 O CH3 H C(=NOCH3)CH(CH2CH3)SCH2CH=CH2 *1
8-003 O CH3 C(O)C(=NOCH3)CH(CH2CH3)SCH2CH=CH2
C(=NOCH3)CH(CH2CH3)SCH2CH=CH2 *1
――――――――――――――――――――――――――――――――――――――――
〔第10表〕
―――――――――――――――――――――――――――――――――――――――
No. プロトン核磁気共鳴ケミカルシフト値(CDCl中):σ(ppm)
―――――――――――――――――――――――――――――――――――――――
2−001;
9.09(d,J=1.5Hz,1H),8.73(d,J=4.8Hz,1H),8.15−8.05(m,1H)、7.50−7.40(m,1H),4.12(s,3H),4.11(s,3H),3.78(s,2H),2.16(s,3H)
4−002;
(異性体比52)9.63(brs,1H),9.02−8.97(m,1H),8.56−8.50(m,1H),8.10−8.02(m,1H),7.35−7.26(m,1H),6.82(s,1H),4.56(q,J=7.2Hz,1H),4.14(s,3H),3.86(s,3H),2.69(s,3H),1.64(d,J=7.2Hz,3H)
(異性体比48) 9.02−8.97(m,1H),8.57(brs,1H),8.56−8.50(m,1H),8.10−8.02(m,1H),7.35−7.26(m,1H),6.75(s,1H),4.38(q,J=7.2Hz,1H),4.14(s,3H),3.85(s,3H),2.55(s,3H),1.71(d,J=7.2Hz,3H)
4−003;
(異性体比53)9.15(brs,1H),9.02−8.97(m,1H),8.60−8.50(m,1H),8.10−8.04(m,1H),7.35−7.28(m,1H),6.76(s,1H),4.71(q,J=7.5Hz,1H),4.18(s,3H),3.84(s,3H),3.01(s,3H),1.70(d,J=7.5Hz,3H)
(異性体比47) 9.02−8.97(m,1H),8.60−8.50(m,1H),8.47(brs,1H),8.10−8.04(m,1H),7.35−7.28(m,1H),6.69(s,1H),4.99(q,J=7.5Hz,1H),4.18(s,3H),3.85(s,3H),3.09(s,3H),1.82(d,J=7.5Hz,3H)
4−006;
9.00(d,J=2.4Hz,1H),8.86−8.80(m,2H),8.10−8.03(m,1H),7.34−7.26(m,1H),6.75(s,1H),5.92−5.74(m,1H),5.22−5.08(m,2H),3.93−3.80(m,1H),4.08(s,3H),3.84(s,3H),3.17(d,J=7,2Hz,2H),2.15−1.90(m,2H),0.97(d,J=7.5Hz,3H)
4−007;
9.01−8.98(m,1H),8.57−8.49(m,2H),8.10−8.00(m,1H),7.35−7.28(m,1H),6.71(s,1H),6.03−5.86(m,1H),5.56−5.47(m,2H),4.96(dd,J=10.8,5.4Hz,1H),4.17(m,3H),3.91(d,J=7.2Hz,2H),3.85(s,3H),2.58−2.40(m,1H),2.28−2.10(m,1H),1.00(t,J=7.5Hz,3H)
8−002;
9.21(s,1H),8.91(d,J=1.8Hz,1H),8.46(dd,J=4.8,1.8Hz,1H),8.06(m,1H),7.31−7.25(m,2H),5.80(m,1H),5.14(m,2H),4.08−4.03(m,4H),3.17(d,J=7.2Hz,2H),2.38(s,3H),1.95(m,2H),0.97(t,J=7.3Hz,3H)
8−003
8.92(s,1H),8.48(d,J=4.5Hz,1H),8.06(m,1H),8.04−7.25(m,2H),5.73(m,2H),5.05(m,4H),4.98−3.89(m,8H),3.05(m,4H),2.43(m,3H),1.95(m,4H)1.01(m,6H)
―――――――――――――――――――――――――――――――――――――――
第10表のプロトン核磁気共鳴ケミカルシフト値は、基準物質としてMeSi(テトラメチルシラン)を用い、300MHzにて測定した。
[試験例]
次に、本発明化合物の有害生物防除剤としての有用性について、以下の試験例において具体的に説明するが、本発明はこれらのみに限定されるものではない。
試験例1 トビイロウンカに対する殺虫試験
本発明化合物の10%乳剤(化合物によっては10%水和剤を供試)を展着剤の入った水で希釈して、500ppm濃度の薬液を調製した。この薬液中にイネの葉鞘を約10秒間浸漬し、風乾後試験管に入れ、この中にトビイロウンカ(Nilaparvata lugens)の2齢幼虫を試験管当たり5頭放虫し、スポンジで蓋をして25℃恒温室に収容した。6日後の死虫数を調査し、死虫率(%)(死虫数÷供試虫数×100)を算出した。尚、試験は2連制で行なった。
――――――――――――――――――――――――――――――――――――――――
No. YR 3 R a R b-1 mp (℃)
――――――――――――――――――――――――――――――――――――――――
8-001 O Cl CH 2 CH 3 C (= NOCH 3 ) CH 2 SCH 3 148-150
8-002 O CH 3 HC (= NOCH 3 ) CH (CH 2 CH 3 ) SCH 2 CH = CH 2 * 1
8-003 O CH 3 C (O) C (= NOCH 3 ) CH (CH 2 CH 3 ) SCH 2 CH = CH 2
C (= NOCH 3 ) CH (CH 2 CH 3 ) SCH 2 CH = CH 2 * 1
――――――――――――――――――――――――――――――――――――――――
[Table 10]
―――――――――――――――――――――――――――――――――――――――
No. Proton nuclear magnetic resonance chemical shift value (in CDCl 3 ): σ (ppm)
―――――――――――――――――――――――――――――――――――――――
2-001;
9.09 (d, J = 1.5 Hz, 1H), 8.73 (d, J = 4.8 Hz, 1H), 8.15-8.05 (m, 1H), 7.50-7.40 (M, 1H), 4.12 (s, 3H), 4.11 (s, 3H), 3.78 (s, 2H), 2.16 (s, 3H)
4-002;
(Isomer ratio 52) 9.63 (brs, 1H), 9.02-8.97 (m, 1H), 8.56-8.50 (m, 1H), 8.10-8.02 (m , 1H), 7.35-7.26 (m, 1H), 6.82 (s, 1H), 4.56 (q, J = 7.2 Hz, 1H), 4.14 (s, 3H), 3.86 (s, 3H), 2.69 (s, 3H), 1.64 (d, J = 7.2 Hz, 3H)
(Isomer ratio 48) 9.02-8.97 (m, 1H), 8.57 (brs, 1H), 8.56-8.50 (m, 1H), 8.10-8.02 (m , 1H), 7.35-7.26 (m, 1H), 6.75 (s, 1H), 4.38 (q, J = 7.2 Hz, 1H), 4.14 (s, 3H), 3.85 (s, 3H), 2.55 (s, 3H), 1.71 (d, J = 7.2 Hz, 3H)
4-003;
(Isomer ratio 53) 9.15 (brs, 1H), 9.02-8.97 (m, 1H), 8.60-8.50 (m, 1H), 8.10-8.04 (m , 1H), 7.35-7.28 (m, 1H), 6.76 (s, 1H), 4.71 (q, J = 7.5 Hz, 1H), 4.18 (s, 3H), 3.84 (s, 3H), 3.01 (s, 3H), 1.70 (d, J = 7.5 Hz, 3H)
(Isomer ratio 47) 9.02-8.97 (m, 1H), 8.60-8.50 (m, 1H), 8.47 (brs, 1H), 8.10-8.04 (m , 1H), 7.35-7.28 (m, 1H), 6.69 (s, 1H), 4.99 (q, J = 7.5 Hz, 1H), 4.18 (s, 3H), 3.85 (s, 3H), 3.09 (s, 3H), 1.82 (d, J = 7.5 Hz, 3H)
4-006;
9.00 (d, J = 2.4 Hz, 1H), 8.86-8.80 (m, 2H), 8.10-8.03 (m, 1H), 7.34-7.26 (m , 1H), 6.75 (s, 1H), 5.92-5.74 (m, 1H), 5.22-5.08 (m, 2H), 3.93-3.80 (m, 1H) ), 4.08 (s, 3H), 3.84 (s, 3H), 3.17 (d, J = 7, 2 Hz, 2H), 2.15-1.90 (m, 2H),. 97 (d, J = 7.5Hz, 3H)
4-007;
9.01-8.98 (m, 1H), 8.57-8.49 (m, 2H), 8.10-8.00 (m, 1H), 7.35-7.28 (m, 1H) ), 6.71 (s, 1H), 6.03-5.86 (m, 1H), 5.56-5.47 (m, 2H), 4.96 (dd, J = 10.8, 5 .4 Hz, 1H), 4.17 (m, 3H), 3.91 (d, J = 7.2 Hz, 2H), 3.85 (s, 3H), 2.58-2.40 (m, 1H) ), 2.28-2.10 (m, 1H), 1.00 (t, J = 7.5 Hz, 3H)
8-002;
9.21 (s, 1H), 8.91 (d, J = 1.8 Hz, 1H), 8.46 (dd, J = 4.8, 1.8 Hz, 1H), 8.06 (m, 1H) ), 7.31-7.25 (m, 2H), 5.80 (m, 1H), 5.14 (m, 2H), 4.08-4.03 (m, 4H), 3.17 ( d, J = 7.2 Hz, 2H), 2.38 (s, 3H), 1.95 (m, 2H), 0.97 (t, J = 7.3 Hz, 3H)
8-003
8.92 (s, 1H), 8.48 (d, J = 4.5 Hz, 1H), 8.06 (m, 1H), 8.04-7.25 (m, 2H), 5.73 ( m, 2H), 5.05 (m, 4H), 4.98-3.89 (m, 8H), 3.05 (m, 4H), 2.43 (m, 3H), 1.95 (m , 4H) 1.01 (m, 6H)
―――――――――――――――――――――――――――――――――――――――
The proton nuclear magnetic resonance chemical shift values in Table 10 were measured at 300 MHz using Me 4 Si (tetramethylsilane) as a reference material.
[Test example]
Next, the usefulness of the compound of the present invention as a pest control agent will be specifically described in the following test examples, but the present invention is not limited to these.
Test Example 1 Insecticidal test against brown planthopper A 10% emulsion of the compound of the present invention (depending on the compound, 10% wettable powder) was diluted with water containing a spreading agent to prepare a chemical solution having a concentration of 500 ppm. Rice leaf sheaths are immersed in this chemical solution for about 10 seconds, air-dried and placed in a test tube, and 5 second-instar larvae of the green planthopper (Nilaparvata lugens) are released per test tube and covered with a sponge. Housed in a constant temperature room. The number of dead insects after 6 days was investigated, and the death rate (%) (number of dead insects ÷ number of test insects × 100) was calculated. In addition, the test was performed by 2 continuous systems.

その結果、供試した化合物の内、下記の化合物が90%以上の死虫率を示した。
本発明化合物:1−001、2−001、3−001、3−002、3−003、4−001〜4−007、5−001、6−001、7−001、8−001、8−002
試験例2 シルバーリーフコナジラミに対する殺虫試験
内径7cmのスチロールカップに湿った濾紙を敷き、その上に3cmに切り取ったインゲンの葉を置いた。本発明化合物の10%乳剤(化合物によっては10%水和剤を供試)を展着剤の入った水で希釈して、500ppm濃度の薬液を調製し、回転式散布塔を用いて薬液をスチロールカップ当たり2.5mlずつ散布した(2.5mg/cm)。葉を風乾後、シルバーリーフコナジラミ(Bemisia argentifolii)の成虫を放虫し、蓋をして25℃恒温室に収容した。5日後の死虫数を調査し、試験例1と同様の計算式から死虫率を算出した。尚、試験は2連制で行なった。
As a result, among the compounds tested, the following compounds showed a death rate of 90% or more.
Compounds of the present invention: 1-001, 2-001, 3-001, 3-002, 3-003, 4-001 to 4-007, 5-001, 6-001, 7-001, 8-001, 8- 002
Test Example 2 Insecticidal test against silver leaf whitefly A moist filter paper was laid on a 7 cm inner diameter styrol cup, and a green leaf cut into 3 cm was placed thereon. A 10% emulsion of a compound of the present invention (depending on the compound, 10% wettable powder) is diluted with water containing a spreading agent to prepare a chemical solution with a concentration of 500 ppm, and the chemical solution is prepared using a rotary spray tower. 2.5 ml was sprayed per styrene cup (2.5 mg / cm 2 ). After the leaves were air-dried, adults of silver leaf whiteflies (Bemisia argentifolii) were released, covered, and housed in a thermostatic chamber at 25 ° C. The number of dead insects after 5 days was investigated, and the dead insect rate was calculated from the same calculation formula as in Test Example 1. In addition, the test was performed by 2 continuous systems.

その結果、供試した化合物の内、下記の化合物が90%以上の死虫率を示した。
本発明化合物:1−001、4−001〜4−007、5−001、7−001、8−001、8−002
試験例3 モモアカアブラムシに対する殺虫試験
内径3cmのガラスシャーレに湿った脱脂綿を敷き、その上に同径に切り取ったカンランの葉を置き、モモアカアブラムシ(Myzus persicae)無翅成虫を4頭放虫した。1日後、本発明化合物の10%乳剤(化合物によっては10%水和剤を供試)を展着剤の入った水で希釈して、500ppm濃度の薬液を調製し、回転式散布塔にて薬液を散布(2.5mg/cm)、蓋をして25℃恒温室に収容した。6日後の死虫数を調査し、試験例1と同様の計算式から死虫率を算出した。尚、試験は2連制で行なった。
As a result, among the compounds tested, the following compounds showed a death rate of 90% or more.
Compounds of the present invention: 1-001, 4-001 to 4-007, 5-001, 7-001, 8-001, 8-002
Test Example 3 Insecticidal test against peach aphid A moist absorbent cotton was laid on a glass petri dish with an inner diameter of 3 cm, and kanran leaves cut out to the same diameter were placed on it. did. One day later, a 10% emulsion of the compound of the present invention (depending on the compound, 10% wettable powder was tested) was diluted with water containing a spreading agent to prepare a chemical solution with a concentration of 500 ppm. The chemical solution was sprayed (2.5 mg / cm 2 ), covered, and stored in a constant temperature room at 25 ° C. The number of dead insects after 6 days was investigated, and the death rate was calculated from the same calculation formula as in Test Example 1. In addition, the test was performed by 2 continuous systems.

その結果、供試した化合物の内、下記の化合物が90%以上の死虫率を示した。
本発明化合物:1−001、2−001、3−001、3−002、4−001〜4−007、5−001、6−001、7−001、8−001、8−002
試験例4 ワタアブラムシに対する殺虫試験
内径3cmのガラスシャーレに湿った脱脂綿を敷き、その上に同径に切り取ったキュウリの葉を置き、ワタアブラムシ(Aphis gossypii)無翅成虫を4頭放虫した。1日後、本発明化合物の10%乳剤(化合物によっては10%水和剤を供試)を展着剤の入った水で希釈して、500ppm濃度の薬液を調製し、回転式散布塔にて薬液を散布(2.5mg/cm)、蓋をして25℃恒温室に収容した。6日後の死虫数を調査し、試験例1と同様の計算式から死虫率を算出した。尚、試験は2連制で行なった。
As a result, among the compounds tested, the following compounds showed a death rate of 90% or more.
Compounds of the present invention: 1-001, 2-001, 3-001, 3-002, 4-001 to 4-007, 5-001, 6-001, 7-001, 8-001, 8-002
Test Example 4 Insecticidal test for cotton aphids Wet cotton wool with a 3 cm inner diameter petri dish and a cucumber leaf cut out to the same diameter were placed on it, and four cotton aphids (Aphis gossypii) adults were released. One day later, a 10% emulsion of the compound of the present invention (depending on the compound, 10% wettable powder was tested) was diluted with water containing a spreading agent to prepare a chemical solution with a concentration of 500 ppm. The chemical solution was sprayed (2.5 mg / cm 2 ), covered, and stored in a constant temperature room at 25 ° C. The number of dead insects after 6 days was investigated, and the death rate was calculated from the same calculation formula as in Test Example 1. In addition, the test was performed by 2 continuous systems.

その結果、供試した化合物の内、下記の化合物が90%以上の死虫率を示した。
本発明化合物:1−001、2−001、3−001、3−002、4−001〜4−007、5−001、7−001,8−001、8−002
試験例5 モモアカアブラムシに対する土壌潅注処理試験
本発明化合物の10%乳剤を水道水で希釈して、濃度が100ppmの薬液を調製した。
As a result, among the compounds tested, the following compounds showed a death rate of 90% or more.
Compounds of the present invention: 1-001, 2-001, 3-001, 3-002, 4-001 to 4-007, 5-001, 7-001, 8-001, 8-002
Test Example 5 Soil irrigation treatment test for peach aphid A 10% emulsion of the compound of the present invention was diluted with tap water to prepare a chemical solution having a concentration of 100 ppm.

プラスチックカップ植えキャベツ苗(2.5本葉期)の株元土壌部分に10mlの薬液を潅注処理し、温室内に放置した。潅注処理1日後にモモアカアブラムシ(Myzus persicae)の成虫を20頭/株で放虫し、その後温室内に放置した。放虫6日後の生存虫数を調査し、下記の計算式から対照値を算出した。
対照値(%)={1−(Cb×Tai)/(Cai×Tb)}×100
式中の文字は下記を表している。
Cb:無処理区における処理前の虫の数
Cai:無処理区における最終調査時の生存虫数
Tb:処理区における処理前の虫の数
Cai:処理区における最終調査時の生存虫数
その結果、供試した化合物の内、下記の化合物が90%以上の対照値を示した。
本発明化合物:1−001、4−001
10 ml of the chemical solution was irrigated to the stock soil portion of the plastic cup planted cabbage seedling (2.5 true leaf stage) and left in the greenhouse. One day after the irrigation treatment, 20 mosquitoes / strain of adult peach aphid (Myzus persicae) were released and then left in the greenhouse. The number of surviving insects 6 days after the release was examined, and a control value was calculated from the following formula.
Control value (%) = {1- (Cb × Tai) / (Cai × Tb)} × 100
The characters in the formula represent the following:
Cb: number of insects before treatment in the untreated group Cai: number of live insects at the time of final survey in the untreated group Tb: number of insects before treatment in the treated group Cai: number of live insects at the time of final survey in the treated group Among the compounds tested, the following compounds showed a control value of 90% or more.
Compounds of the present invention: 1-001, 4-001

本発明における新規な複素環誘導体は、優れた有害生物防除活性、特に殺虫・殺ダニ活性を示し、且つ、ホ乳動物、魚類及び益虫等の非標的生物に対してほとんど悪影響の無い、極めて有用な化合物である。   The novel heterocyclic derivative in the present invention exhibits excellent pest control activity, particularly insecticidal / miticidal activity, and has very little adverse effect on non-target organisms such as mammals, fish and beneficial insects. Compound.

Claims (9)

式(1):
Figure 2015147757

[式中、Aは、−N(−O)m2又は−CRを表し、
、R、R、R4a及びR4bは、各々独立して水素原子、ハロゲン原子、シアノ、ニトロ、−OH、−SH、−NH、C〜Cアルキル、R28aによって任意に置換された(C〜C)アルキル、C〜Cシクロアルキル、R28aによって任意に置換された(C〜C)シクロアルキル、C〜Cアルケニル、R28aによって任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R28aによって任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R28aによって任意に置換された(C〜C)アルキニル、C〜Cアルコキシ、C〜Cハロアルコキシ、C〜Cアルケニルオキシ、C〜Cアルキルチオ、C〜Cアルキルスルフィニル、C〜Cアルキルスルホニル、C〜Cハロアルキルチオ、C〜Cハロアルキルスルフィニル、C〜Cハロアルキルスルホニル、C〜Cアルキルカルボニル、C〜Cシクロアルキルカルボニル、C〜Cハロアルキルカルボニル、C〜Cハロシクロアルキルカルボニル、C〜Cアルコキシカルボニル、C〜Cハロアルコキシカルボニル、C〜Cアルキルチオカルボニル、C〜Cアルコキシチオカルボニル、C〜Cアルキルジチオカルボニル、C〜Cアルキルアミノカルボニル、C〜Cハロアルキルアミノカルボニル、ジ(C〜Cアルキル)アミノカルボニル、トリ(C〜Cアルキル)シリル、C〜Cアルキルアミノスルホニル、ジ(C〜Cアルキル)アミノスルホニル、C〜Cアルキルカルボニルオキシ、C〜Cアルキルスルホニルオキシ、C〜Cハロアルキルスルホニルオキシ、C〜Cアルキルアミノ、ジ(C〜Cアルキル)アミノ、フェニル、ナフチル、(Z)で置換されたフェニル、(Z)で置換されたナフチル又はD1−1〜D1−99を表し、
は、ハロゲン原子、シアノ、ニトロ、−OH、−SH、−NH、C〜Cアルキル、R28aによって任意に置換された(C〜C)アルキル、C〜Cシクロアルキル、R28aによって任意に置換された(C〜C)シクロアルキル、C〜Cアルケニル、R28aによって任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R28aによって任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R28aによって任意に置換された(C〜C)アルキニル、C〜Cアルコキシ、C〜Cハロアルコキシ、C〜Cアルケニルオキシ、C〜Cアルキルチオ、C〜Cアルキルスルフィニル、C〜Cアルキルスルホニル、C〜Cハロアルキルチオ、C〜Cハロアルキルスルフィニル、C〜Cハロアルキルスルホニル、C〜Cアルキルカルボニル、C〜Cシクロアルキルカルボニル、C〜Cハロアルキルカルボニル、C〜Cハロシクロアルキルカルボニル、C〜Cアルコキシカルボニル、C〜Cハロアルコキシカルボニル、C〜Cアルキルチオカルボニル、C〜Cアルコキシチオカルボニル、C〜Cアルキルジチオカルボニル、C〜Cアルキルアミノカルボニル、C〜Cハロアルキルアミノカルボニル、ジ(C〜Cアルキル)アミノカルボニル、トリ(C〜Cアルキル)シリル、C〜Cアルキルアミノスルホニル、ジ(C〜Cアルキル)アミノスルホニル、C〜Cアルキルカルボニルオキシ、C〜Cアルキルスルホニルオキシ、C〜Cハロアルキルスルホニルオキシ、C〜Cアルキルアミノ、ジ(C〜Cアルキル)アミノ、フェニル、ナフチル、(Z)で置換されたフェニル、(Z)で置換されたナフチル又はD1−1〜D1−99を表し、nが2以上の整数を表すとき、各々のRは互いに同一であっても又は互いに相異なってもよく、
3aは、水素原子、シアノ、ニトロ、−OH、−SH、−NH、C〜Cアルキル、R28aによって任意に置換された(C〜C)アルキル、C〜Cシクロアルキル、R28aによって任意に置換された(C〜C)シクロアルキル、C〜Cアルケニル、R28aによって任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R28aによって任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R28aによって任意に置換された(C〜C)アルキニル、C〜Cアルコキシ、C〜Cハロアルコキシ、C〜Cアルケニルオキシ、C〜Cアルキルチオ、C〜Cアルキルスルフィニル、C〜Cアルキルスルホニル、C〜Cハロアルキルチオ、C〜Cハロアルキルスルフィニル、C〜Cハロアルキルスルホニル、C〜Cアルキルカルボニル、C〜Cシクロアルキルカルボニル、C〜Cハロアルキルカルボニル、C〜Cハロシクロアルキルカルボニル、C〜Cアルコキシカルボニル、C〜Cハロアルコキシカルボニル、C〜Cアルキルチオカルボニル、C〜Cアルコキシチオカルボニル、C〜Cアルキルジチオカルボニル、C〜Cアルキルアミノカルボニル、C〜Cハロアルキルアミノカルボニル、ジ(C〜Cアルキル)アミノカルボニル、トリ(C〜Cアルキル)シリル、C〜Cアルキルアミノスルホニル、ジ(C〜Cアルキル)アミノスルホニル、C〜Cアルキルカルボニルオキシ、C〜Cアルキルスルホニルオキシ、C〜Cハロアルキルスルホニルオキシ、C〜Cアルキルアミノ、ジ(C〜Cアルキル)アミノ、フェニル、ナフチル、(Z)で置換されたフェニル、(Z)で置換されたナフチル又はD1−1〜D1−99を表し、
Bは、B−1〜B−34を表し、
B−1〜B−34は、以下の構造を表し、
Figure 2015147757

Figure 2015147757

明細書中
環Bの記載において、「*」は置換基「−N(R)R」との結合位置を表し、「**」は置換基「=NR」との結合位置を表し、「***」は下記に示した置換基との結合位置を表す。
Figure 2015147757

は、酸素原子又は硫黄原子を表し、
は、水素原子、シアノ、C〜C12アルキル、R5aによって任意に置換された(C〜C12)アルキル、C〜C12シクロアルキル、R5aによって任意に置換された(C〜C12)シクロアルキル、C〜C12アルケニル、R5aによって任意に置換された(C〜C12)アルケニル、C〜C12シクロアルケニル、R5aによって任意に置換された(C〜C12)シクロアルケニル、C〜C12アルキニル、R5aによって任意に置換された(C〜C12)アルキニル、、−OH、−OR6a、−SH、−S(O)r26a、−C(O)OR6a、−C(O)SR6a、−C(S)OR6a、−C(S)SR6a、−C(O)R7a、−C(S)R7a、−N(R8a)R9a、−C(O)N(R8a)R9a、−C(S)N(R8a)R9a、−S(O)r2N(R8a)R9a、−Si(R40a)(R40b)R40、−P(O)(OR41、−P(S)(OR41、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル又はD1−1〜D1−99のいずれかの基を表すか、或いは、RはRと一緒になってC〜Cのアルキレン鎖又はC〜Cアルケニレン鎖を形成することにより、Rが結合する炭素原子及びRが結合する炭素原子と共に5〜8員環を形成してもよく、このときこのアルキレン鎖又はアルケニレン鎖は酸素原子、硫黄原子又は窒素原子を1又は2個含んでもよく、且つハロゲン原子、シアノ、ニトロ、C〜Cアルキル、−OH、−OR11a、−SH、−S(O)11a、オキソ基又はチオキソ基によって任意に置換されてもよく、
は、−C(O)R7b又は−C(S)R7bを表すか、或いは、RはRと一緒になって=C(Rb2)Rb3を形成してもよく、
b2は、−OR6a又は−S(O)6aを表し、
b3は、−C(=NOH)R12b、−C(=NOR11b)R12b又は−C{=NN(R13b)R14b}R12bを表し、
5aは、ハロゲン原子、シアノ、ニトロ、C〜Cシクロアルキル、R10aによって任意に置換された(C〜C)シクロアルキル、−OH、−OR11a、−SH、−S(O)r211a、−N(R13a)R14a、−C(O)OH、−C(O)OR11a、−C(O)SR11a、−C(S)OR11a、−C(S)SR11a、−C(O)R12a、−C(S)R12a、−C(O)N(R13a)R14a、−C(S)N(R13a)R14a、−S(O)r2N(R13a)R14a、−Si(R40a)(R40b)R40、−P(O)(OR41、−P(S)(OR41、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル又はD1−1〜D1−99のいずれかの基を表すか、或いは、2つのR5aが同一の炭素上に置換している場合、2つのR5aは一緒になってオキソ、チオキソ、イミノ、C〜Cアルキルイミノ、C〜Cアルコキシイミノ又はC〜Cアルキリデンを形成してもよい。
6a、R8a及びR9aは、各々独立して水素原子、C〜Cアルキル、R10aによって任意に置換された(C〜C)アルキル、C〜Cアルケニル、R10aによって任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R10aによって任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R10aによって任意に置換された(C〜C)アルキニル、C〜Cシクロアルキル、R10aによって任意に置換された(C〜C)シクロアルキル、−S(O)r211a、−C(O)OR11a、−C(O)SR11a、−C(S)OR11a、−C(S)SR11a、−C(O)R12a、−C(S)R12a、−C(O)N(R13a)R14a、−C(S)N(R13a)R14a、−S(O)r2N(R13a)R14a、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル又はD1−1〜D1−99のいずれかの基を表すか、或いは、R8aはR9aと一緒になってC〜Cのアルキレン鎖又はC〜Cのアルケニレン鎖を形成することにより、R8a及びR9aが結合する窒素原子と共に3〜8員環を形成してもよく、このときこのアルキレン鎖又はアルケニレン鎖は酸素原子、硫黄原子又は窒素原子を1個含んでもよく、且つ、R42、R10aで任意に置換された(C〜C)アルキル、オキソ基又はチオキソ基によって任意に置換されてもよい。
7aは、R6a、−C(=NR13a)R12a、−C(=NOH)R12a、−C(=NOR11a)R12a又は−C{=NN(R13a)R14a}R12aを表し、
7bは、−C(=NOH)R12b、−C(=NOR11b)R12b又は−C{=NN(R13b)R14b}R12bを表し、
10aは、ハロゲン原子、シアノ、ニトロ、C〜Cシクロアルキル、C〜Cハロシクロアルキル、−OH、−OR11a、−SH、−S(O)11a、−P(O)(OR41、−P(S)(OR41又は−Si(R40a)(R40b)R40を表すか、或いは、2つのR10aが同一の炭素上に置換している場合、2つのR10aは一緒になってオキソ、チオキソ、イミノ、C〜Cアルキルイミノ、C〜Cアルコキシイミノ又はC〜Cアルキリデンを形成してもよい。
11aは、C〜Cアルキル、R15aによって任意に置換された(C〜C)アルキル、C〜Cアルケニル、R15aによって任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R15aによって任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R15aによって任意に置換された(C〜C)アルキニル、C〜Cシクロアルキル、R15aによって任意に置換された(C〜C)シクロアルキル、−S(O)r216a、−C(O)OR16a、−C(O)SR16a、−C(S)OR16a、−C(S)SR16a、−C(O)R17a、−C(S)R17a、−N(R18a)R19a、−C(O)N(R18a)R19a、−C(S)N(R18a)R19a、−S(O)r2N(R18a)R19a、−Si(R40a)(R40b)R40、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル又はD1−1〜D1−99を表し、
11bは、C〜Cアルキル、R15bによって任意に置換された(C〜C)アルキル、C〜Cアルケニル、R15bによって任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R15bによって任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R15bによって任意に置換された(C〜C)アルキニル、C〜Cシクロアルキル、R15bによって任意に置換された(C〜C)シクロアルキル、−S(O)r316b、−C(O)OR16b、−C(O)SR16b、−C(S)OR16b、−C(S)SR16b、−C(O)R17b、−C(S)R17b、−C(O)N(R18b)R19b、−C(S)N(R18b)R19b、−S(O)r3N(R18b)R19b、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル又はD1−1〜D1−99を表し、
12aは、水素原子、ハロゲン原子、シアノ、C〜Cアルキル、R15aによって任意に置換された(C〜C)アルキル、C〜Cアルケニル、R15aによって任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R15aによって任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R15aによって任意に置換された(C〜C)アルキニル、C〜Cシクロアルキル、R15aによって任意に置換された(C〜C)シクロアルキル、−OR16a、−S(O)r216a、−C(O)OR16a、−C(O)SR16a、−C(S)OR16a、−C(S)SR16a、−C(O)R17a、−C(S)R17a、−N(R18a)R19a、−C(O)N(R18a)R19a、−C(S)N(R18a)R19a、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル又はD1−1〜D1−99を表し、
12bは、水素原子、ハロゲン原子、シアノ、C〜Cアルキル、R15cによって任意に置換された(C〜C)アルキル、C〜Cアルケニル、R15cによって任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R15cによって任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R15cによって任意に置換された(C〜C)アルキニル、C〜Cシクロアルキル、R15cによって任意に置換された(C〜C)シクロアルキル、−OR16c、−S(O)16c、−C(O)OR16c、−C(O)SR16c、−C(S)OR16c、−C(S)SR16c、−C(O)R17c、−C(S)R17c、−N(R18c)R19c、−C(O)N(R18c)R19c、−C(S)N(R18c)R19c、−S(O)N(R18c)R19c、−C(=NOH)R17c、−C(=NOR16c)R17c、−C{=NN(R18c)R19c}R17c、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル又はD1−1〜D1−99を表し、
13a及びR14aは、各々独立して水素原子又はC〜Cアルキルを表すか、或いは、R13aはR14aと一緒になってC〜Cのアルキレン鎖又はC〜Cのアルケニレン鎖を形成することにより、R13a及びR14aが結合する窒素原子と共に3〜8員環を形成してもよく、このときこのアルキレン鎖又はアルケニレン鎖は酸素原子、硫黄原子又は窒素原子を1個含んでもよく、且つハロゲン原子、シアノ、C〜Cアルキル、R15aによって任意に置換された(C〜C)アルキル、C〜Cアルコキシ、C〜Cハロアルコキシ、C〜Cアルキルチオ、C〜Cハロアルキルチオ、C〜Cアルキルスルフィニル、C〜Cハロアルキルスルフィニル、C〜Cアルキルスルホニル、C〜Cハロアルキルスルホニル、フェニル、(Z)によって置換されたフェニル、オキソ基又はチオキソ基によって任意に置換されてもよく、
13bは、水素原子、シアノ、ニトロ、C〜Cアルキル、R15bによって任意に置換された(C〜C)アルキル、C〜Cアルケニル、R15bによって任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R15bによって任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R15bによって任意に置換された(C〜C)アルキニル、C〜Cシクロアルキル、R15bによって任意に置換された(C〜C)シクロアルキル、−OR16b、−S(O)r316b、−C(O)OR16b、−C(O)SR16b、−C(S)OR16b、−C(S)SR16b、−C(O)R17b、−C(S)R17b、−C(O)N(R18b)R19b、−C(S)N(R18b)R19b、−S(O)r3N(R18b)R19b、−P(O)(OR41、−P(S)(OR41、−Si(R40a)(R40b)R40、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル又はD1−1〜D1−99を表すか、或いは、R13bはR14bと一緒になってC〜Cのアルキレン鎖又はC〜Cのアルケニレン鎖を形成することにより、R13b及びR14bが結合する窒素原子と共に3〜8員環を形成してもよく、このときこのアルキレン鎖又はアルケニレン鎖は酸素原子、硫黄原子又は窒素原子を1個含んでもよく、且つハロゲン原子、シアノ、C〜Cアルキル、R15bによって任意に置換された(C〜C)アルキル、C〜Cアルコキシ、C〜Cハロアルコキシ、C〜Cアルキルチオ、C〜Cハロアルキルチオ、C〜Cアルキルスルフィニル、C〜Cハロアルキルスルフィニル、C〜Cアルキルスルホニル、C〜Cハロアルキルスルホニル、フェニル、(Z)によって置換されたフェニル、オキソ基又はチオキソ基によって任意に置換されてもよく、
14bは、水素原子、シアノ、ニトロ、C〜Cアルキル、R15dで任意に置換された(C〜C)アルキル、C〜Cアルケニル、R15dで任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R15dで任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R15dで任意に置換された(C〜C)アルキニル、C〜Cシクロアルキル、R15dで任意に置換された(C〜C)シクロアルキル、−OR16d、−S(O)r316d、−C(O)OR16d、−C(O)SR16d、−C(S)OR16d、−C(S)SR16d、−C(O)R17d、−C(S)R17d、−C(O)N(R18d)R19d、−C(S)N(R18d)R19d、−S(O)r3N(R18d)R19d、−Si(R40a)(R40b)R40、−P(O)(OR41、−P(S)(OR41、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル又はD1−1〜D1−99のいずれかの基を表すか、或いは、R14bはR13bと一緒になって=C(R14e)R14fを形成してもよい。
14e及びR14fは、各々独立して水素原子、シアノ、ニトロ、C〜Cアルキル、R15bで任意に置換された(C〜C)アルキル、C〜Cアルケニル、R15bで任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R15bで任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R15bで任意に置換された(C〜C)アルキニル、C〜Cシクロアルキル、R15bで任意に置換された(C〜C)シクロアルキル、−OR16b、−S(O)r316b、−C(O)OR16b、−C(O)SR16b、−C(S)OR16b、−C(S)SR16b、−C(O)R17b、−C(S)R17b、−C(O)N(R18b)R19b、−C(S)N(R18b)R19b、−S(O)r3N(R18b)R19b、−Si(R40a)(R40b)R40、−P(O)(OR41、−P(S)(OR41、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル又はD1−1〜D1−99のいずれかの基を表すか、或いは、R14eはR14fと一緒になってC〜Cのアルキレン鎖又はC〜Cのアルケニレン鎖を形成することにより、R14e及びR14fが結合する炭素原子と共に3〜8員環を形成してもよく、このときこのアルキレン鎖又はアルケニレン鎖は酸素原子、硫黄原子又は窒素原子を1、2又は3個含んでもよく、且つR42、R15bで任意に置換された(C〜C)アルキル、オキソ基又はチオキソ基によって任意に置換されてもよい。
15aは、ハロゲン原子、シアノ、ニトロ、C〜Cシクロアルキル、C〜Cハロシクロアルキル、−OH、−OR16a、−SH、−S(O)r216a、−S(=NR18a)R16a、−S(O)(=NR18a)R16a、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル、D1−1〜D1−99又は−Si(R40a)(R40b)R40を表すか、、或いは、2つのR15aが同一の炭素上に置換している場合、2つのR15aは一緒になってオキソ、チオキソ、イミノ、C〜Cアルキルイミノ、C〜Cアルコキシイミノ又はC〜Cアルキリデンを形成してもよい。
15bは、ハロゲン原子、シアノ、ニトロ、C〜Cシクロアルキル、C〜Cハロシクロアルキル、−OH、−OR16b、−SH、−S(O)r316b、−S(=NR18b)R16b、−S(O)(=NR18b)R16b、−C(O)OH、−C(O)OR16b、−C(O)R17b、−C(O)N(R18b)R19b、−C(=NOR16b)R17b、−P(O)(OR41、−P(S)(OR41、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル、D1−1〜D1−99又は−Si(R40a)(R40b)R40を表すか、、或いは、2つのR15bが同一の炭素上に置換している場合、2つのR15bは一緒になってオキソ、チオキソ、イミノ、C〜Cアルキルイミノ、C〜Cアルコキシイミノ又はC〜Cアルキリデンを形成してもよい。
15cは、ハロゲン原子、シアノ、ニトロ、C〜Cシクロアルキル、C〜Cハロシクロアルキル、−OH、−OR16c、−SH、−S(O)16c、−S(=NR18c)R16c、−S(O)(=NR18c)R16c、−P(O)(OR41、−P(S)(OR41、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル、D1−1〜D1−99又は−Si(R40a)(R40b)R40を表すか、或いは、2つのR15cが同一の炭素上に置換している場合、2つのR15cは一緒になってオキソ、チオキソ、イミノ、C〜Cアルキルイミノ、C〜Cアルコキシイミノ又はC〜Cアルキリデンを形成してもよい。
15dは、ハロゲン原子、シアノ、ニトロ、C〜Cシクロアルキル、C〜Cハロシクロアルキル、−OH、−OR16d、−SH、−S(O)r316d、−S(=NR18d)R16d、−S(O)(=NR18d)R16d、−P(O)(OR41、−P(S)(OR41、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル、D1−1〜D1−99のいずれかの基又は−Si(R40a)(R40b)R40を表すか、或いは、2つのR15dが同一の炭素上に置換している場合、2つのR5aは一緒になってオキソ、チオキソ、イミノ、C〜Cアルキルイミノ、C〜Cアルコキシイミノ又はC〜Cアルキリデンを形成してもよく、
16a、R16b、R16c及びR16dは、各々独立してシアノ、C〜Cアルキル、C〜Cアルケニル、C〜Cアルキニル、C〜Cシクロアルキル、C〜Cシクロアルケニル、R20によって任意に置換された(C〜C)アルキル、R20によって任意に置換された(C〜C)アルケニル、R20によって任意に置換された(C〜C)アルキニル、R20によって任意に置換された(C〜C)シクロアルキル、R20によって任意に置換された(C〜C)シクロアルケニル、−S(O)21、−C(O)R22、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル又はD1−1〜D1−99のいずれかの基を表し、
17a、R17b、R17c及びR17dは、各々独立して水素原子、C〜Cアルキル、C〜Cアルケニル、C〜Cアルキニル、C〜Cシクロアルキル、C〜Cシクロアルケニル、R20によって任意に置換された(C〜C)アルキル、R20で任意に置換された(C〜C)アルケニル、R20で任意に置換された(C〜C)アルキニル、R20で任意に置換された(C〜C)シクロアルキル、R20で任意に置換された(C〜C)シクロアルケニル、−C(O)R22、−C(=NOR21)R22、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル又はD1−1〜D1−99のいずれかの基を表し、
18a及びR19aは、各々独立して水素原子,シアノ又はC〜Cアルキルを表し、
18b、R19b、R18d及びR19dは、各々独立して水素原子,シアノ、C〜Cアルキル、C〜Cアルケニル、C〜Cアルキニル、C〜Cシクロアルキル、C〜Cシクロアルケニル、R20で任意に置換された(C〜C)アルキル、R20で任意に置換された(C〜C)アルケニル、R20で任意に置換された(C〜C)アルキニル、R20で任意に置換された(C〜C)シクロアルキル、R20で任意に置換された(C〜C)シクロアルケニル、フェニル、(Z)によって置換されたフェニル、ナフチル、(Z)によって置換されたナフチル又はD1−1〜D1−99のいずれかの基を表すか、或いは、R18bはR19bと一緒になってC〜Cのアルキレン鎖又はC〜Cのアルケニレン鎖を形成することにより、R18b及びR19bが結合する窒素原子と共に3〜8員環を形成してもよく、このときこのアルキレン鎖又はアルケニレン鎖は酸素原子、硫黄原子又は窒素原子を1又は2個含んでもよく、且つR42、R20で任意に置換された(C〜C)アルキル、オキソ基又はチオキソ基によって任意に置換されてもよい。
18c及びR19cは、各々独立して水素原子,シアノ、C〜Cアルキル、R20で任意に置換された(C〜C)アルキル、−OR21、−S(O)21、−C(O)OR21、−C(O)R22、−C(S)R22、フェニル又は(Z)によって置換されたフェニルを表し、
20は、ハロゲン原子、シアノ、ニトロ、−OH、−SH、−NH、C〜Cシクロアルキル、C〜Cハロシクロアルキル、C〜Cシクロアルケニル、C〜Cハロシクロアルケニル、C〜Cアルコキシ、C〜Cハロアルコキシ、C〜Cアルケニルオキシ、C〜Cアルキルチオ、C〜Cアルキルスルフィニル、C〜Cアルキルスルホニル、C〜Cハロアルキルチオ、C〜Cハロアルキルスルフィニル、C〜Cハロアルキルスルホニル、C〜Cアルキルカルボニル、C〜Cシクロアルキルカルボニル、C〜Cハロアルキルカルボニル、C〜Cハロシクロアルキルカルボニル、C〜Cアルコキシカルボニル、C〜Cハロアルコキシカルボニル、C〜Cアルキルチオカルボニル、C〜Cアルコキシチオカルボニル、C〜Cアルキルジチオカルボニル、C〜Cアルキルアミノカルボニル、C〜Cハロアルキルアミノカルボニル、ジ(C〜Cアルキル)アミノカルボニル、トリ(C〜Cアルキル)シリル、C〜Cアルキルアミノスルホニル、ジ(C〜Cアルキル)アミノスルホニル、C〜Cアルキルカルボニルオキシ、C〜Cアルキルスルホニルオキシ、C〜Cハロアルキルスルホニルオキシ、C〜Cアルキルアミノ、ジ(C〜Cアルキル)アミノ、C〜Cアルキルイミノ、C〜Cアルコキシイミノ、フェニル、ナフチル、(Z)で置換されたフェニル、(Z)で置換されたナフチル又はD1−1〜D1−99を表すか、、或いは、2つのR20が同一の炭素上に置換している場合、2つのR20は一緒になってオキソ、チオキソ、イミノ、C〜Cアルキルイミノ、C〜Cアルコキシイミノ又はC〜Cアルキリデンを形成してもよく、
D1−1〜D1−99は、それぞれ下記の構造で表される環を表し、
Figure 2015147757

Figure 2015147757

Figure 2015147757

は、ハロゲン原子、シアノ、ニトロ、−OH、−SH又はR24を表し、g1、g2又はg4が2以上の整数を表すとき、各々のXは互いに同一であっても又は互いに相異なってもよく、更に2つのXが隣接する場合には、隣接する2つのXは、−CHCHCH−、−CHCHO−、−CHOCH−、−OCHO−、−CHCHS−、−CHSCH−、−CHCHCHCH−、−CHCHCHO−、−CHCHOCH−、−CHOCHO−、−OCHCHO−、−CHCHCHS−、−OCHCHS−、−CHCH=CH−、−OCH=CH−、−SCH=CH−、−N(X1a)CH=CH−、−OCH=N−、−SCH=N−、−N(X1a)CH=N−、−N(X1a)N=CH−、−OCHCH=CH−、−CH=CHCH=CH−、−N=CHCH=CH−、−CH=NCH=CH−、−N=NCH=CH−、−CH=NN=CH−、−N=CHCH=N−又は−N=CHN=CH−を形成することにより、それぞれのXが結合する炭素原子と共に5員環又は6員環を形成してもよく、このとき環を形成する各々の炭素原子に結合した水素原子は、ハロゲン原子、シアノ、ニトロ、C〜Cアルキル基、C〜Cハロアルキル基、C〜Cアルコキシ基、C〜Cハロアルコキシ基、C〜Cアルキルチオ基、C〜Cアルキルスルフィニル基、C〜Cアルキルスルホニル基、C〜Cハロアルキルチオ基、C〜Cハロアルキルスルフィニル基、C〜Cハロアルキルスルホニル基、C〜Cアルキルカルボニル基、C〜Cシクロアルキルカルボニル基、C〜Cハロアルキルカルボニル基、C〜Cハロシクロアルキルカルボニル基、C〜Cアルコキシカルボニル基又はC〜Cハロアルコキシカルボニル基によって任意に置換されてもよく、
1aは、水素原子、シアノ、−OH又はR24を表し、
1aの隣接位にXが存在する場合には、隣接するX1aとXは、−CHCHCHCH−、−CH=CHCH=CH−、−N=CHCH=CH−、−CH=N−CH=CH−、−CH=CH−N=CH−又は−CH=CH−CH=N−を形成することにより、X1a及びXのそれぞれが結合する原子と共に6員環を形成してもよく、このとき、環を形成する各々の炭素原子に結合する水素原子は、ハロゲン原子、シアノ、ニトロ、C〜Cアルキル基、C〜Cハロアルキル基、C〜Cアルコキシ基、C〜Cアルキルチオ基、C〜Cアルキルスルフィニル基又はC〜Cアルキルスルホニル基によって任意に置換されてもよい。
1bは、ハロゲン原子、シアノ、ニトロ、−OH、−SH又はR24を表し、f1、f2、f4、f5、f6、f7、f8又はf9が2以上の整数を表すとき、各々のX1bは互いに同一であっても又は互いに相異なってもよく、さらに、2つのX1bが同一の炭素上に置換している場合、2つのX1bは一緒になってオキソ、チオキソ、イミノ、C〜Cアルキルイミノ、C〜Cアルコキシイミノ又はC〜Cアルキリデンを形成してもよく、
Zは、ハロゲン原子、シアノ、ニトロ、−OH、−SH又はR24を表し、qが2以上の整数を表すとき、各々のZは互いに同一であっても又は互いに相異なってもよく、更に2つのZが隣接する場合には、隣接する2つのZは、−CHCHCH−、−CHCHO−、−CHOCH−、−OCHO−、−CHCHS−、−CHSCH−、−CHCHCHCH−、−CHCHCHO−、−CHCHOCH−、−CHOCHO−、−OCHCHO−、−CHCHCHS−、−OCHCHS−、−CHCH=CH−、−OCH=CH−、−SCH=CH−、−N(X1a)CH=CH−、−OCH=N−、−SCH=N−、−N(X1a)CH=N−、−N(X1a)N=CH−、−OCHCH=CH−、−N=CHCH=CH−、−CH=NCH=CH−、−N=NCH=CH−、−CH=NN=CH−、−N=CHCH=N−又は−N=CHN=CH−を形成することにより、それぞれのZが結合する炭素原子と共に5員環又は6員環を形成してもよく、このとき環を形成する各々の炭素原子に結合した水素原子は、ハロゲン原子、シアノ、ニトロ、C〜Cアルキル基、C〜Cハロアルキル基、C〜Cアルコキシ基、C〜Cハロアルコキシ基、C〜Cアルキルチオ基、C〜Cアルキルスルフィニル基、C〜Cアルキルスルホニル基、C〜Cハロアルキルチオ基、C〜Cハロアルキルスルフィニル基、C〜Cハロアルキルスルホニル基、C〜Cアルキルカルボニル基、C〜Cシクロアルキルカルボニル基、C〜Cハロアルキルカルボニル基、C〜Cハロシクロアルキルカルボニル基、C〜Cアルコキシカルボニル基又はC〜Cハロアルコキシカルボニル基によって任意に置換されてもよく、
24は、C〜Cアルキル、R28によって任意に置換された(C〜C)アルキル、C〜Cシクロアルキル、R28によって任意に置換された(C〜C)シクロアルキル、C〜Cアルケニル、R28によって任意に置換された(C〜C)アルケニル、C〜Cシクロアルケニル、R28によって任意に置換された(C〜C)シクロアルケニル、C〜Cアルキニル、R28によって任意に置換された(C〜C)アルキニル、C〜Cアルコキシ、C〜Cハロアルコキシ、C〜Cアルケニルオキシ、C〜Cアルキルチオ、C〜Cアルキルスルフィニル、C〜Cアルキルスルホニル、C〜Cハロアルキルチオ、C〜Cハロアルキルスルフィニル、C〜Cハロアルキルスルホニル、C〜Cアルキルカルボニル、C〜Cシクロアルキルカルボニル、C〜Cハロアルキルカルボニル、C〜Cハロシクロアルキルカルボニル、C〜Cアルコキシカルボニル、C〜Cハロアルコキシカルボニル、C〜Cアルキルチオカルボニル、C〜Cアルコキシチオカルボニル、C〜Cアルキルジチオカルボニル、C〜Cアルキルアミノカルボニル、C〜Cハロアルキルアミノカルボニル、ジ(C〜Cアルキル)アミノカルボニル、トリ(C〜Cアルキル)シリル、C〜Cアルキルアミノスルホニル、ジ(C〜Cアルキル)アミノスルホニル、C〜Cアルキルカルボニルオキシ、C〜Cアルキルスルホニルオキシ、C〜Cハロアルキルスルホニルオキシ、C〜Cアルキルアミノ、ジ(C〜Cアルキル)アミノ、−C(=NOR29)R30、フェニル、ナフチル、C〜Cアルキルで任意に置換されたフェニル又はハロゲン原子で任意に置換されたフェニルを表し、
28、R28a、R31及びR32は、各々独立してハロゲン原子、シアノ、−OH、−SH、−NH、−CHO、−C(O)OH、−C(O)NH、−C(S)NH、−S(O)NH、−Si(R40a)(R40b)R40、C〜Cアルコキシ、C〜Cハロアルコキシ、C〜Cアルケニルオキシ、C〜Cアルキルチオ、C〜Cアルキルスルフィニル、C〜Cアルキルスルホニル、C〜Cハロアルキルチオ、C〜Cハロアルキルスルフィニル、C〜Cハロアルキルスルホニル、C〜Cアルキルカルボニル、C〜Cシクロアルキルカルボニル、C〜Cハロアルキルカルボニル、C〜Cハロシクロアルキルカルボニル、C〜Cアルコキシカルボニル、C〜Cハロアルコキシカルボニル、C〜C6アルキルアミノスルホニル、ジ(C〜Cアルキル)アミノスルホニル、C〜C6アルキルアミノカルボニル、ジ(C〜Cアルキル)アミノカルボニル、C〜Cアルキルアミノ、ジ(C〜Cアルキル)アミノ、フェニル、C〜Cアルキルで任意に置換されたフェニル又はハロゲン原子で任意に置換されたフェニルを表し、
29及びR29aは、各々独立してC〜Cアルキル、C〜Cアルケニル、C〜Cアルキニル、C〜Cシクロアルキル、C〜Cシクロアルケニル、R31で任意に置換された(C〜C)アルキル、R31で任意に置換された(C〜C)アルケニル、R31で任意に置換された(C〜C)アルキニル、R31で任意に置換された(C〜C)シクロアルキル又はR31で任意に置換された(C〜C)シクロアルケニルを表す。
30及びR30aは、各々独立してC〜Cアルキル、C〜Cアルケニル、C〜Cアルキニル、C〜Cシクロアルキル、C〜Cシクロアルケニル、R32で任意に置換された(C〜C)アルキル、R32で任意に置換された(C〜C)アルケニル、R32で任意に置換された(C〜C)アルキニル、R32で任意に置換された(C〜C)シクロアルキル、R32で任意に置換された(C〜C)シクロアルケニル、フェニル、C〜Cアルキルで任意に置換されたフェニル又はハロゲン原子で任意に置換されたフェニルを表す。
40、R40a及びR40bは、各々独立してC〜Cアルキル、C〜Cアルコキシ又はフェニルを表し、
41は、C〜Cアルキルを表し、
42は、ハロゲン原子、シアノ、C〜Cアルキル、C〜Cアルコキシ、C〜Cハロアルコキシ、C〜Cアルキルチオ、C〜Cハロアルキルチオ、C〜Cアルキルスルフィニル、C〜Cハロアルキルスルフィニル、C〜Cアルキルスルホニル、C〜Cハロアルキルスルホニル、フェニル又は(Z)によって置換されたフェニルを表す。
n、g1及びf1は、各々独立して0、1、2又は3の整数を表し、
g2及びf2は、各々独立して0、1又は2の整数を表し、
g3は、0又は1の整数を表し、
g4及びf4は、各々独立して0、1、2、3又は4の整数を表し、
f5は、0、1、2、3、4又は5の整数を表し、
f6は、0、1、2、3、4、5又は6の整数を表し、
f7は、0、1、2、3、4、5、6又は7の整数を表し、
f8は、0、1、2、3、4、5、6、7又は8の整数を表し、
f9は、0、1、2、3、4、5、6、7、8又は9の整数を表し、
qは、1、2、3、4又は5の整数を表し、
m1、m2及びm3は、各々独立して0又は1の整数を表し、
r及びr2は、各々独立して0、1又は2の整数を表す。〕で表される複素環誘導体又はその塩。
Formula (1):
Figure 2015147757

[Where A 1 Is -N (-O) m2 Or -CR 1 Represents
R 1 , R 3 , R 4 , R 4a And R 4b Each independently represents a hydrogen atom, a halogen atom, cyano, nitro, -OH, -SH, -NH 2 , C 1 ~ C 6 Alkyl, R 28a Optionally substituted by (C 1 ~ C 6 ) Alkyl, C 3 ~ C 8 Cycloalkyl, R 28a Optionally substituted by (C 3 ~ C 8 ) Cycloalkyl, C 2 ~ C 6 Alkenyl, R 28a Optionally substituted by (C 2 ~ C 6 ) Alkenyl, C 3 ~ C 8 Cycloalkenyl, R 28a Optionally substituted by (C 3 ~ C 8 ) Cycloalkenyl, C 2 ~ C 6 Alkynyl, R 28a Optionally substituted by (C 2 ~ C 6 ) Alkynyl, C 1 ~ C 6 Alkoxy, C 1 ~ C 6 Haloalkoxy, C 2 ~ C 6 Alkenyloxy, C 1 ~ C 6 Alkylthio, C 1 ~ C 6 Alkylsulfinyl, C 1 ~ C 6 Alkylsulfonyl, C 1 ~ C 6 Haloalkylthio, C 1 ~ C 6 Haloalkylsulfinyl, C 1 ~ C 6 Haloalkylsulfonyl, C 1 ~ C 6 Alkylcarbonyl, C 3 ~ C 8 Cycloalkylcarbonyl, C 1 ~ C 6 Haloalkylcarbonyl, C 3 ~ C 8 Halocycloalkylcarbonyl, C 1 ~ C 6 Alkoxycarbonyl, C 1 ~ C 6 Haloalkoxycarbonyl, C 1 ~ C 6 Alkylthiocarbonyl, C 1 ~ C 6 Alkoxythiocarbonyl, C 1 ~ C 6 Alkyldithiocarbonyl, C 1 ~ C 6 Alkylaminocarbonyl, C 1 ~ C 6 Haloalkylaminocarbonyl, di (C 1 ~ C 6 Alkyl) aminocarbonyl, tri (C 1 ~ C 6 Alkyl) silyl, C 1 ~ C 6 Alkylaminosulfonyl, di (C 1 ~ C 6 Alkyl) aminosulfonyl, C 1 ~ C 6 Alkylcarbonyloxy, C 1 ~ C 6 Alkylsulfonyloxy, C 1 ~ C 6 Haloalkylsulfonyloxy, C 1 ~ C 6 Alkylamino, di (C 1 ~ C 6 Alkyl) amino, phenyl, naphthyl, (Z) q Phenyl substituted with (Z) q Represents naphthyl or D1-1 to D1-99 substituted with
R 2 Is a halogen atom, cyano, nitro, -OH, -SH, -NH 2 , C 1 ~ C 6 Alkyl, R 28a Optionally substituted by (C 1 ~ C 6 ) Alkyl, C 3 ~ C 8 Cycloalkyl, R 28a Optionally substituted by (C 3 ~ C 8 ) Cycloalkyl, C 2 ~ C 6 Alkenyl, R 28a Optionally substituted by (C 2 ~ C 6 ) Alkenyl, C 3 ~ C 8 Cycloalkenyl, R 28a Optionally substituted by (C 3 ~ C 8 ) Cycloalkenyl, C 2 ~ C 6 Alkynyl, R 28a Optionally substituted by (C 2 ~ C 6 ) Alkynyl, C 1 ~ C 6 Alkoxy, C 1 ~ C 6 Haloalkoxy, C 2 ~ C 6 Alkenyloxy, C 1 ~ C 6 Alkylthio, C 1 ~ C 6 Alkylsulfinyl, C 1 ~ C 6 Alkylsulfonyl, C 1 ~ C 6 Haloalkylthio, C 1 ~ C 6 Haloalkylsulfinyl, C 1 ~ C 6 Haloalkylsulfonyl, C 1 ~ C 6 Alkylcarbonyl, C 3 ~ C 8 Cycloalkylcarbonyl, C 1 ~ C 6 Haloalkylcarbonyl, C 3 ~ C 8 Halocycloalkylcarbonyl, C 1 ~ C 6 Alkoxycarbonyl, C 1 ~ C 6 Haloalkoxycarbonyl, C 1 ~ C 6 Alkylthiocarbonyl, C 1 ~ C 6 Alkoxythiocarbonyl, C 1 ~ C 6 Alkyldithiocarbonyl, C 1 ~ C 6 Alkylaminocarbonyl, C 1 ~ C 6 Haloalkylaminocarbonyl, di (C 1 ~ C 6 Alkyl) aminocarbonyl, tri (C 1 ~ C 6 Alkyl) silyl, C 1 ~ C 6 Alkylaminosulfonyl, di (C 1 ~ C 6 Alkyl) aminosulfonyl, C 1 ~ C 6 Alkylcarbonyloxy, C 1 ~ C 6 Alkylsulfonyloxy, C 1 ~ C 6 Haloalkylsulfonyloxy, C 1 ~ C 6 Alkylamino, di (C 1 ~ C 6 Alkyl) amino, phenyl, naphthyl, (Z) q Phenyl substituted with (Z) q Represents naphthyl substituted with or D1-1 to D1-99, and when n represents an integer of 2 or more, each R 2 May be the same or different from each other,
R 3a Is a hydrogen atom, cyano, nitro, -OH, -SH, -NH 2 , C 1 ~ C 6 Alkyl, R 28a Optionally substituted by (C 1 ~ C 6 ) Alkyl, C 3 ~ C 8 Cycloalkyl, R 28a Optionally substituted by (C 3 ~ C 8 ) Cycloalkyl, C 2 ~ C 6 Alkenyl, R 28a Optionally substituted by (C 2 ~ C 6 ) Alkenyl, C 3 ~ C 8 Cycloalkenyl, R 28a Optionally substituted by (C 3 ~ C 8 ) Cycloalkenyl, C 2 ~ C 6 Alkynyl, R 28a Optionally substituted by (C 2 ~ C 6 ) Alkynyl, C 1 ~ C 6 Alkoxy, C 1 ~ C 6 Haloalkoxy, C 2 ~ C 6 Alkenyloxy, C 1 ~ C 6 Alkylthio, C 1 ~ C 6 Alkylsulfinyl, C 1 ~ C 6 Alkylsulfonyl, C 1 ~ C 6 Haloalkylthio, C 1 ~ C 6 Haloalkylsulfinyl, C 1 ~ C 6 Haloalkylsulfonyl, C 1 ~ C 6 Alkylcarbonyl, C 3 ~ C 8 Cycloalkylcarbonyl, C 1 ~ C 6 Haloalkylcarbonyl, C 3 ~ C 8 Halocycloalkylcarbonyl, C 1 ~ C 6 Alkoxycarbonyl, C 1 ~ C 6 Haloalkoxycarbonyl, C 1 ~ C 6 Alkylthiocarbonyl, C 1 ~ C 6 Alkoxythiocarbonyl, C 1 ~ C 6 Alkyldithiocarbonyl, C 1 ~ C 6 Alkylaminocarbonyl, C 1 ~ C 6 Haloalkylaminocarbonyl, di (C 1 ~ C 6 Alkyl) aminocarbonyl, tri (C 1 ~ C 6 Alkyl) silyl, C 1 ~ C 6 Alkylaminosulfonyl, di (C 1 ~ C 6 Alkyl) aminosulfonyl, C 1 ~ C 6 Alkylcarbonyloxy, C 1 ~ C 6 Alkylsulfonyloxy, C 1 ~ C 6 Haloalkylsulfonyloxy, C 1 ~ C 6 Alkylamino, di (C 1 ~ C 6 Alkyl) amino, phenyl, naphthyl, (Z) q Phenyl substituted with (Z) q Represents naphthyl or D1-1 to D1-99 substituted with
B represents B-1 to B-34;
B-1 to B-34 represent the following structures:
Figure 2015147757

Figure 2015147757

In the description
In the description of ring B, “*” represents the substituent “—N (R a ) R b "**" represents the substituent "= NR" b ”Represents a bonding position with the substituent shown below.
Figure 2015147757

Q 1 Represents an oxygen atom or a sulfur atom,
R a Is a hydrogen atom, cyano, C 1 ~ C 12 Alkyl, R 5a Optionally substituted by (C 1 ~ C 12 ) Alkyl, C 3 ~ C 12 Cycloalkyl, R 5a Optionally substituted by (C 3 ~ C 12 ) Cycloalkyl, C 2 ~ C 12 Alkenyl, R 5a Optionally substituted by (C 2 ~ C 12 ) Alkenyl, C 3 ~ C 12 Cycloalkenyl, R 5a Optionally substituted by (C 3 ~ C 12 ) Cycloalkenyl, C 2 ~ C 12 Alkynyl, R 5a Optionally substituted by (C 2 ~ C 12 ) Alkynyl, -OH, -OR 6a , -SH, -S (O) r2 R 6a , -C (O) OR 6a , -C (O) SR 6a , -C (S) OR 6a , -C (S) SR 6a , -C (O) R 7a , -C (S) R 7a , -N (R 8a ) R 9a , -C (O) N (R 8a ) R 9a , -C (S) N (R 8a ) R 9a , -S (O) r2 N (R 8a ) R 9a , -Si (R 40a ) (R 40b ) R 40 , -P (O) (OR 41 ) 2 , -P (S) (OR 41 ) 2 , Phenyl, (Z) q Phenyl, naphthyl, substituted by (Z) q Represents naphthyl or any group of D1-1 to D1-99 substituted by R, or R a Is R 3 Together with C 2 ~ C 5 An alkylene chain or C 2 ~ C 5 By forming an alkenylene chain, R a Carbon atom to which R is bonded and R 3 May form a 5- to 8-membered ring with the carbon atom to which is bonded, and in this case, the alkylene chain or alkenylene chain may contain one or two oxygen atoms, sulfur atoms or nitrogen atoms, and a halogen atom, cyano, Nitro, C 1 ~ C 6 Alkyl, -OH, -OR 11a , -SH, -S (O) r R 11a Optionally substituted by an oxo group or a thioxo group,
R b Is -C (O) R 7b Or -C (S) R 7b Or R b Is R a Together with = C (R b2 ) R b3 May form,
R b2 Is -OR 6a Or -S (O) r R 6a Represents
R b3 Is -C (= NOH) R 12b , -C (= NOR 11b ) R 12b Or -C {= NN (R 13b ) R 14b } R 12b Represents
R 5a Is a halogen atom, cyano, nitro, C 3 ~ C 8 Cycloalkyl, R 10a Optionally substituted by (C 3 ~ C 8 ) Cycloalkyl, -OH, -OR 11a , -SH, -S (O) r2 R 11a , -N (R 13a ) R 14a , -C (O) OH, -C (O) OR 11a , -C (O) SR 11a , -C (S) OR 11a , -C (S) SR 11a , -C (O) R 12a , -C (S) R 12a , -C (O) N (R 13a ) R 14a , -C (S) N (R 13a ) R 14a , -S (O) r2 N (R 13a ) R 14a , -Si (R 40a ) (R 40b ) R 40 , -P (O) (OR 41 ) 2 , -P (S) (OR 41 ) 2 , Phenyl, (Z) q Phenyl, naphthyl, substituted by (Z) q Represents naphthyl or any group of D1-1 to D1-99 substituted by 5a Are substituted on the same carbon, two R 5a Together oxo, thioxo, imino, C 1 ~ C 6 Alkylimino, C 1 ~ C 6 Alkoxyimino or C 1 ~ C 6 An alkylidene may be formed.
R 6a , R 8a And R 9a Are each independently a hydrogen atom, C 1 ~ C 6 Alkyl, R 10a Optionally substituted by (C 1 ~ C 6 ) Alkyl, C 2 ~ C 6 Alkenyl, R 10a Optionally substituted by (C 2 ~ C 6 ) Alkenyl, C 3 ~ C 8 Cycloalkenyl, R 10a Optionally substituted by (C 3 ~ C 8 ) Cycloalkenyl, C 2 ~ C 6 Alkynyl, R 10a Optionally substituted by (C 2 ~ C 6 ) Alkynyl, C 3 ~ C 8 Cycloalkyl, R 10a Optionally substituted by (C 3 ~ C 8 ) Cycloalkyl, -S (O) r2 R 11a , -C (O) OR 11a , -C (O) SR 11a , -C (S) OR 11a , -C (S) SR 11a , -C (O) R 12a , -C (S) R 12a , -C (O) N (R 13a ) R 14a , -C (S) N (R 13a ) R 14a , -S (O) r2 N (R 13a ) R 14a , Phenyl, (Z) q Phenyl, naphthyl, substituted by (Z) q Represents naphthyl or any group of D1-1 to D1-99 substituted by R, or R 8a Is R 9a Together with C 2 ~ C 7 An alkylene chain or C 2 ~ C 7 By forming an alkenylene chain of R 8a And R 9a May form a 3- to 8-membered ring together with the nitrogen atom to which is bonded, in which case the alkylene chain or alkenylene chain may contain one oxygen atom, sulfur atom or nitrogen atom, and R 42 , R 10a Optionally substituted with (C 1 ~ C 6 ) Optionally substituted by alkyl, oxo group or thioxo group.
R 7a Is R 6a , -C (= NR 13a ) R 12a , -C (= NOH) R 12a , -C (= NOR 11a ) R 12a Or -C {= NN (R 13a ) R 14a } R 12a Represents
R 7b Is -C (= NOH) R 12b, -C (= NOR 11b ) R 12b Or -C {= NN (R 13b ) R 14b } R 12b Represents
R 10a Is a halogen atom, cyano, nitro, C 3 ~ C 8 Cycloalkyl, C 3 ~ C 8 Halocycloalkyl, —OH, —OR 11a , -SH, -S (O) r R 11a , -P (O) (OR 41 ) 2 , -P (S) (OR 41 ) 2 Or -Si (R 40a ) (R 40b ) R 40 Or two R 10a Are substituted on the same carbon, two R 10a Together oxo, thioxo, imino, C 1 ~ C 6 Alkylimino, C 1 ~ C 6 Alkoxyimino or C 1 ~ C 6 An alkylidene may be formed.
R 11a Is C 1 ~ C 6 Alkyl, R 15a Optionally substituted by (C 1 ~ C 6 ) Alkyl, C 2 ~ C 6 Alkenyl, R 15a Optionally substituted by (C 2 ~ C 6 ) Alkenyl, C 3 ~ C 8 Cycloalkenyl, R 15a Optionally substituted by (C 3 ~ C 8 ) Cycloalkenyl, C 2 ~ C 6 Alkynyl, R 15a Optionally substituted by (C 2 ~ C 6 ) Alkynyl, C 3 ~ C 8 Cycloalkyl, R 15a Optionally substituted by (C 3 ~ C 8 ) Cycloalkyl, -S (O) r2 R 16a , -C (O) OR 16a , -C (O) SR 16a , -C (S) OR 16a , -C (S) SR 16a , -C (O) R 17a , -C (S) R 17a , -N (R 18a ) R 19a , -C (O) N (R 18a ) R 19a , -C (S) N (R 18a ) R 19a , -S (O) r2 N (R 18a ) R 19a , -Si (R 40a ) (R 40b ) R 40 , Phenyl, (Z) q Phenyl, naphthyl, substituted by (Z) q Represents naphthyl or D1-1 to D1-99 substituted by
R 11b Is C 1 ~ C 6 Alkyl, R 15b Optionally substituted by (C 1 ~ C 6 ) Alkyl, C 2 ~ C 6 Alkenyl, R 15b Optionally substituted by (C 2 ~ C 6 ) Alkenyl, C 3 ~ C 8 Cycloalkenyl, R 15b Optionally substituted by (C 3 ~ C 8 ) Cycloalkenyl, C 2 ~ C 6 Alkynyl, R 15b Optionally substituted by (C 2 ~ C 6 ) Alkynyl, C 3 ~ C 8 Cycloalkyl, R 15b Optionally substituted by (C 3 ~ C 8 ) Cycloalkyl, -S (O) r3 R 16b , -C (O) OR 16b , -C (O) SR 16b , -C (S) OR 16b , -C (S) SR 16b , -C (O) R 17b , -C (S) R 17b , -C (O) N (R 18b ) R 19b , -C (S) N (R 18b ) R 19b , -S (O) r3 N (R 18b ) R 19b , Phenyl, (Z) q Phenyl, naphthyl, substituted by (Z) q Represents naphthyl or D1-1 to D1-99 substituted by
R 12a Is a hydrogen atom, halogen atom, cyano, C 1 ~ C 6 Alkyl, R 15a Optionally substituted by (C 1 ~ C 6 ) Alkyl, C 2 ~ C 6 Alkenyl, R 15a Optionally substituted by (C 2 ~ C 6 ) Alkenyl, C 3 ~ C 8 Cycloalkenyl, R 15a Optionally substituted by (C 3 ~ C 8 ) Cycloalkenyl, C 2 ~ C 6 Alkynyl, R 15a Optionally substituted by (C 2 ~ C 6 ) Alkynyl, C 3 ~ C 8 Cycloalkyl, R 15a Optionally substituted by (C 3 ~ C 8 ) Cycloalkyl, -OR 16a , -S (O) r2 R 16a , -C (O) OR 16a , -C (O) SR 16a , -C (S) OR 16a , -C (S) SR 16a , -C (O) R 17a , -C (S) R 17a , -N (R 18a ) R 19a , -C (O) N (R 18a ) R 19a , -C (S) N (R 18a ) R 19a , Phenyl, (Z) q Phenyl, naphthyl, substituted by (Z) q Represents naphthyl or D1-1 to D1-99 substituted by
R 12b Is a hydrogen atom, halogen atom, cyano, C 1 ~ C 6 Alkyl, R 15c Optionally substituted by (C 1 ~ C 6 ) Alkyl, C 2 ~ C 6 Alkenyl, R 15c Optionally substituted by (C 2 ~ C 6 ) Alkenyl, C 3 ~ C 8 Cycloalkenyl, R 15c Optionally substituted by (C 3 ~ C 8 ) Cycloalkenyl, C 2 ~ C 6 Alkynyl, R 15c Optionally substituted by (C 2 ~ C 6 ) Alkynyl, C 3 ~ C 8 Cycloalkyl, R 15c Optionally substituted by (C 3 ~ C 8 ) Cycloalkyl, -OR 16c , -S (O) r R 16c , -C (O) OR 16c , -C (O) SR 16c , -C (S) OR 16c , -C (S) SR 16c , -C (O) R 17c , -C (S) R 17c , -N (R 18c ) R 19c , -C (O) N (R 18c ) R 19c , -C (S) N (R 18c ) R 19c , -S (O) r N (R 18c ) R 19c , -C (= NOH) R 17c , -C (= NOR 16c ) R 17c , -C {= NN (R 18c ) R 19c } R 17c , Phenyl, (Z) q Phenyl, naphthyl, substituted by (Z) q Represents naphthyl or D1-1 to D1-99 substituted by
R 13a And R 14a Each independently represents a hydrogen atom or C 1 ~ C 6 Represents alkyl or R 13a Is R 14a Together with C 2 ~ C 7 An alkylene chain or C 2 ~ C 7 By forming an alkenylene chain of R 13a And R 14a May form a 3- to 8-membered ring together with the nitrogen atom to which is bonded, and in this case, the alkylene chain or alkenylene chain may contain one oxygen atom, sulfur atom or nitrogen atom, and a halogen atom, cyano, C 1 ~ C 6 Alkyl, R 15a Optionally substituted by (C 1 ~ C 6 ) Alkyl, C 1 ~ C 6 Alkoxy, C 1 ~ C 6 Haloalkoxy, C 1 ~ C 6 Alkylthio, C 1 ~ C 6 Haloalkylthio, C 1 ~ C 6 Alkylsulfinyl, C 1 ~ C 6 Haloalkylsulfinyl, C 1 ~ C 6 Alkylsulfonyl, C 1 ~ C 6 Haloalkylsulfonyl, phenyl, (Z) q Optionally substituted by a phenyl, oxo group or thioxo group substituted by
R 13b Is a hydrogen atom, cyano, nitro, C 1 ~ C 6 Alkyl, R 15b Optionally substituted by (C 1 ~ C 6 ) Alkyl, C 2 ~ C 6 Alkenyl, R 15b Optionally substituted by (C 2 ~ C 6 ) Alkenyl, C 3 ~ C 8 Cycloalkenyl, R 15b Optionally substituted by (C 3 ~ C 8 ) Cycloalkenyl, C 2 ~ C 6 Alkynyl, R 15b Optionally substituted by (C 2 ~ C 6 ) Alkynyl, C 3 ~ C 8 Cycloalkyl, R 15b Optionally substituted by (C 3 ~ C 8 ) Cycloalkyl, -OR 16b , -S (O) r3 R 16b , -C (O) OR 16b , -C (O) SR 16b , -C (S) OR 16b , -C (S) SR 16b , -C (O) R 17b , -C (S) R 17b , -C (O) N (R 18b ) R 19b , -C (S) N (R 18b ) R 19b , -S (O) r3 N (R 18b ) R 19b , -P (O) (OR 41 ) 2 , -P (S) (OR 41 ) 2 , -Si (R 40a ) (R 40b ) R 40 , Phenyl, (Z) q Phenyl, naphthyl, substituted by (Z) q Represents naphthyl or D1-1 to D1-99 substituted by R, or R 13b Is R 14b Together with C 2 ~ C 7 An alkylene chain or C 2 ~ C 7 By forming an alkenylene chain of R 13b And R 14b May form a 3- to 8-membered ring together with the nitrogen atom to which is bonded, and in this case, the alkylene chain or alkenylene chain may contain one oxygen atom, sulfur atom or nitrogen atom, and a halogen atom, cyano, C 1 ~ C 6 Alkyl, R 15b Optionally substituted by (C 1 ~ C 6 ) Alkyl, C 1 ~ C 6 Alkoxy, C 1 ~ C 6 Haloalkoxy, C 1 ~ C 6 Alkylthio, C 1 ~ C 6 Haloalkylthio, C 1 ~ C 6 Alkylsulfinyl, C 1 ~ C 6 Haloalkylsulfinyl, C 1 ~ C 6 Alkylsulfonyl, C 1 ~ C 6 Haloalkylsulfonyl, phenyl, (Z) q Optionally substituted by a phenyl, oxo group or thioxo group substituted by
R 14b Is a hydrogen atom, cyano, nitro, C 1 ~ C 6 Alkyl, R 15d Optionally substituted with (C 1 ~ C 6 ) Alkyl, C 2 ~ C 6 Alkenyl, R 15d Optionally substituted with (C 2 ~ C 6 ) Alkenyl, C 3 ~ C 8 Cycloalkenyl, R 15d Optionally substituted with (C 3 ~ C 8 ) Cycloalkenyl, C 2 ~ C 6 Alkynyl, R 15d Optionally substituted with (C 2 ~ C 6 ) Alkynyl, C 3 ~ C 8 Cycloalkyl, R 15d Optionally substituted with (C 3 ~ C 8 ) Cycloalkyl, -OR 16d , -S (O) r3 R 16d , -C (O) OR 16d , -C (O) SR 16d , -C (S) OR 16d , -C (S) SR 16d , -C (O) R 17d , -C (S) R 17d , -C (O) N (R 18d ) R 19d , -C (S) N (R 18d ) R 19d , -S (O) r3 N (R 18d ) R 19d , -Si (R 40a ) (R 40b ) R 40 , -P (O) (OR 41 ) 2 , -P (S) (OR 41 ) 2 , Phenyl, (Z) q Phenyl, naphthyl, substituted by (Z) q Represents naphthyl or any group of D1-1 to D1-99 substituted by R, or R 14b Is R 13b Together with = C (R 14e ) R 14f May be formed.
R 14e And R 14f Each independently represents a hydrogen atom, cyano, nitro, C 1 ~ C 6 Alkyl, R 15b Optionally substituted with (C 1 ~ C 6 ) Alkyl, C 2 ~ C 6 Alkenyl, R 15b Optionally substituted with (C 2 ~ C 6 ) Alkenyl, C 3 ~ C 8 Cycloalkenyl, R 15b Optionally substituted with (C 3 ~ C 8 ) Cycloalkenyl, C 2 ~ C 6 Alkynyl, R 15b Optionally substituted with (C 2 ~ C 6 ) Alkynyl, C 3 ~ C 8 Cycloalkyl, R 15b Optionally substituted with (C 3 ~ C 8 ) Cycloalkyl, -OR 16b , -S (O) r3 R 16b , -C (O) OR 16b , -C (O) SR 16b , -C (S) OR 16b , -C (S) SR 16b , -C (O) R 17b , -C (S) R 17b , -C (O) N (R 18b ) R 19b , -C (S) N (R 18b ) R 19b , -S (O) r3 N (R 18b ) R 19b , -Si (R 40a ) (R 40b ) R 40 , -P (O) (OR 41 ) 2 , -P (S) (OR 41 ) 2 , Phenyl, (Z) q Phenyl, naphthyl, substituted by (Z) q Represents naphthyl or any group of D1-1 to D1-99 substituted by R, or R 14e Is R 14f Together with C 2 ~ C 7 An alkylene chain or C 2 ~ C 7 By forming an alkenylene chain of R 14e And R 14f May form a 3- to 8-membered ring together with the carbon atom to which is bonded, in which case the alkylene chain or alkenylene chain may contain 1, 2 or 3 oxygen atoms, sulfur atoms or nitrogen atoms, and R 42 , R 15b Optionally substituted with (C 1 ~ C 6 ) Optionally substituted by alkyl, oxo group or thioxo group.
R 15a Is a halogen atom, cyano, nitro, C 3 ~ C 8 Cycloalkyl, C 3 ~ C 8 Halocycloalkyl, —OH, —OR 16a , -SH, -S (O) r2 R 16a , -S (= NR 18a ) R 16a , -S (O) (= NR 18a ) R 16a , Phenyl, (Z) q Phenyl, naphthyl, substituted by (Z) q Naphthyl substituted by D1-1 to D1-99 or —Si (R 40a ) (R 40b ) R 40 Or two R 15a Are substituted on the same carbon, two R 15a Together oxo, thioxo, imino, C 1 ~ C 6 Alkylimino, C 1 ~ C 6 Alkoxyimino or C 1 ~ C 6 An alkylidene may be formed.
R 15b Is a halogen atom, cyano, nitro, C 3 ~ C 8 Cycloalkyl, C 3 ~ C 8 Halocycloalkyl, —OH, —OR 16b , -SH, -S (O) r3 R 16b , -S (= NR 18b ) R 16b , -S (O) (= NR 18b ) R 16b , -C (O) OH, -C (O) OR 16b , -C (O) R 17b , -C (O) N (R 18b ) R 19b , -C (= NOR 16b ) R 17b , -P (O) (OR 41 ) 2 , -P (S) (OR 41 ) 2 , Phenyl, (Z) q Phenyl, naphthyl, substituted by (Z) q Naphthyl substituted by D1-1 to D1-99 or —Si (R 40a ) (R 40b ) R 40 Or two R 15b Are substituted on the same carbon, two R 15b Together oxo, thioxo, imino, C 1 ~ C 6 Alkylimino, C 1 ~ C 6 Alkoxyimino or C 1 ~ C 6 An alkylidene may be formed.
R 15c Is a halogen atom, cyano, nitro, C 3 ~ C 8 Cycloalkyl, C 3 ~ C 8 Halocycloalkyl, —OH, —OR 16c , -SH, -S (O) r R 16c , -S (= NR 18c ) R 16c, -S (O) (= NR 18c ) R 16c , -P (O) (OR 41 ) 2 , -P (S) (OR 41 ) 2 , Phenyl, (Z) q Phenyl, naphthyl, substituted by (Z) q Naphthyl substituted by D1-1 to D1-99 or —Si (R 40a ) (R 40b ) R 40 Or two R 15c Are substituted on the same carbon, two R 15c Together oxo, thioxo, imino, C 1 ~ C 6 Alkylimino, C 1 ~ C 6 Alkoxyimino or C 1 ~ C 6 An alkylidene may be formed.
R 15d Is a halogen atom, cyano, nitro, C 3 ~ C 8 Cycloalkyl, C 3 ~ C 8 Halocycloalkyl, —OH, —OR 16d , -SH, -S (O) r3 R 16d , -S (= NR 18d ) R 16d , -S (O) (= NR 18d ) R 16d , -P (O) (OR 41 ) 2 , -P (S) (OR 41 ) 2 , Phenyl, (Z) q Phenyl, naphthyl, substituted by (Z) q A naphthyl substituted by any group of D1-1 to D1-99 or —Si (R 40a ) (R 40b ) R 40 Or two R 15d Are substituted on the same carbon, two R 5a Together oxo, thioxo, imino, C 1 ~ C 6 Alkylimino, C 1 ~ C 6 Alkoxyimino or C 1 ~ C 6 May form alkylidene,
R 16a , R 16b , R 16c And R 16d Are each independently cyano, C 1 ~ C 6 Alkyl, C 2 ~ C 6 Alkenyl, C 2 ~ C 6 Alkynyl, C 3 ~ C 8 Cycloalkyl, C 3 ~ C 8 Cycloalkenyl, R 20 Optionally substituted by (C 1 ~ C 6 ) Alkyl, R 20 Optionally substituted by (C 2 ~ C 6 ) Alkenyl, R 20 Optionally substituted by (C 2 ~ C 6 ) Alkynyl, R 20 Optionally substituted by (C 3 ~ C 8 ) Cycloalkyl, R 20 Optionally substituted by (C 3 ~ C 8 ) Cycloalkenyl, -S (O) r R 21 , -C (O) R 22 , Phenyl, (Z) q Phenyl, naphthyl, substituted by (Z) q Represents naphthyl or any group of D1-1 to D1-99 substituted by
R 17a , R 17b , R 17c And R 17d Are each independently a hydrogen atom, C 1 ~ C 6 Alkyl, C 2 ~ C 6 Alkenyl, C 2 ~ C 6 Alkynyl, C 3 ~ C 8 Cycloalkyl, C 3 ~ C 8 Cycloalkenyl, R 20 Optionally substituted by (C 1 ~ C 6 ) Alkyl, R 20 Optionally substituted with (C 2 ~ C 6 ) Alkenyl, R 20 Optionally substituted with (C 2 ~ C 6 ) Alkynyl, R 20 Optionally substituted with (C 3 ~ C 8 ) Cycloalkyl, R 20 Optionally substituted with (C 3 ~ C 8 ) Cycloalkenyl, -C (O) R 22 , -C (= NOR 21 ) R 22 , Phenyl, (Z) q Phenyl, naphthyl, substituted by (Z) q Represents naphthyl or any group of D1-1 to D1-99 substituted by
R 18a And R 19a Each independently represents a hydrogen atom, cyano or C 1 ~ C 6 Represents alkyl,
R 18b , R 19b , R 18d And R 19d Are each independently a hydrogen atom, cyano, C 1 ~ C 6 Alkyl, C 2 ~ C 6 Alkenyl, C 2 ~ C 6 Alkynyl, C 3 ~ C 8 Cycloalkyl, C 3 ~ C 8 Cycloalkenyl, R 20 Optionally substituted with (C 1 ~ C 6 ) Alkyl, R 20 Optionally substituted with (C 2 ~ C 6 ) Alkenyl, R 20 Optionally substituted with (C 2 ~ C 6 ) Alkynyl, R 20 Optionally substituted with (C 3 ~ C 8 ) Cycloalkyl, R 20 Optionally substituted with (C 3 ~ C 8 ) Cycloalkenyl, phenyl, (Z) q Phenyl, naphthyl, substituted by (Z) q Represents naphthyl or any group of D1-1 to D1-99 substituted by R, or R 18b Is R 19b Together with C 2 ~ C 7 An alkylene chain or C 2 ~ C 7 By forming an alkenylene chain of R 18b And R 19b May form a 3- to 8-membered ring together with the nitrogen atom to which is bonded, in which case the alkylene chain or alkenylene chain may contain one or two oxygen atoms, sulfur atoms or nitrogen atoms, and R 42 , R 20 Optionally substituted with (C 1 ~ C 6 ) Optionally substituted by alkyl, oxo group or thioxo group.
R 18c And R 19c Are each independently a hydrogen atom, cyano, C 1 ~ C 6 Alkyl, R 20 Optionally substituted with (C 1 ~ C 6 ) Alkyl, -OR 21 , -S (O) r R 21 , -C (O) OR 21 , -C (O) R 22 , -C (S) R 22 , Phenyl or (Z) q Represents phenyl substituted by
R 20 Is a halogen atom, cyano, nitro, -OH, -SH, -NH 2 , C 3 ~ C 8 Cycloalkyl, C 3 ~ C 8 Halocycloalkyl, C 3 ~ C 8 Cycloalkenyl, C 3 ~ C 8 Halocycloalkenyl, C 1 ~ C 6 Alkoxy, C 1 ~ C 6 Haloalkoxy, C 2 ~ C 6 Alkenyloxy, C 1 ~ C 6 Alkylthio, C 1 ~ C 6 Alkylsulfinyl, C 1 ~ C 6 Alkylsulfonyl, C 1 ~ C 6 Haloalkylthio, C 1 ~ C 6 Haloalkylsulfinyl, C 1 ~ C 6 Haloalkylsulfonyl, C 1 ~ C 6 Alkylcarbonyl, C 3 ~ C 8 Cycloalkylcarbonyl, C 1 ~ C 6 Haloalkylcarbonyl, C 3 ~ C 8 Halocycloalkylcarbonyl, C 1 ~ C 6 Alkoxycarbonyl, C 1 ~ C 6 Haloalkoxycarbonyl, C 1 ~ C 6 Alkylthiocarbonyl, C 1 ~ C 6 Alkoxythiocarbonyl, C 1 ~ C 6 Alkyldithiocarbonyl, C 1 ~ C 6 Alkylaminocarbonyl, C 1 ~ C 6 Haloalkylaminocarbonyl, di (C 1 ~ C 6 Alkyl) aminocarbonyl, tri (C 1 ~ C 6 Alkyl) silyl, C 1 ~ C 6 Alkylaminosulfonyl, di (C 1 ~ C 6 Alkyl) aminosulfonyl, C 1 ~ C 6 Alkylcarbonyloxy, C 1 ~ C 6 Alkylsulfonyloxy, C 1 ~ C 6 Haloalkylsulfonyloxy, C 1 ~ C 6 Alkylamino, di (C 1 ~ C 6 Alkyl) amino, C 1 ~ C 6 Alkylimino, C 1 ~ C 6 Alkoxyimino, phenyl, naphthyl, (Z) q Phenyl substituted with (Z) q Represents naphthyl or D1-1 to D1-99 substituted with or two R 20 Are substituted on the same carbon, two R 20 Together oxo, thioxo, imino, C 1 ~ C 6 Alkylimino, C 1 ~ C 6 Alkoxyimino or C 1 ~ C 6 May form alkylidene,
D1-1 to D1-99 each represent a ring represented by the following structure:
Figure 2015147757

Figure 2015147757

Figure 2015147757

X 1 Is a halogen atom, cyano, nitro, —OH, —SH or R 24 When g1, g2 or g4 represents an integer of 2 or more, each X 1 May be the same as or different from each other, and two X 1 Are adjacent, the two adjacent X 1 Is -CH 2 CH 2 CH 2 -, -CH 2 CH 2 O-, -CH 2 OCH 2 -, -OCH 2 O-, -CH 2 CH 2 S-, -CH 2 SCH 2 -, -CH 2 CH 2 CH 2 CH 2 -, -CH 2 CH 2 CH 2 O-, -CH 2 CH 2 OCH 2 -, -CH 2 OCH 2 O-, -OCH 2 CH 2 O-, -CH 2 CH 2 CH 2 S-, -OCH 2 CH 2 S-, -CH 2 CH = CH-, -OCH = CH-, -SCH = CH-, -N (X 1a ) CH = CH-, -OCH = N-, -SCH = N-, -N (X 1a ) CH = N-, -N (X 1a ) N = CH-, -OCH 2 CH = CH-, -CH = CHCH = CH-, -N = CHCH = CH-, -CH = NCH = CH-, -N = NCH = CH-, -CH = NN = CH-, -N = CHCH = By forming N- or -N = CHN = CH-, each X 1 May form a 5-membered ring or a 6-membered ring with the carbon atom to which is bonded, and at this time, the hydrogen atom bonded to each carbon atom forming the ring is a halogen atom, cyano, nitro, C 1 ~ C 6 Alkyl group, C 1 ~ C 6 Haloalkyl group, C 1 ~ C 6 Alkoxy group, C 1 ~ C 6 Haloalkoxy group, C 1 ~ C 6 Alkylthio group, C 1 ~ C 6 Alkylsulfinyl group, C 1 ~ C 6 Alkylsulfonyl group, C 1 ~ C 6 Haloalkylthio group, C 1 ~ C 6 Haloalkylsulfinyl group, C 1 ~ C 6 Haloalkylsulfonyl group, C 1 ~ C 6 Alkylcarbonyl group, C 3 ~ C 8 A cycloalkylcarbonyl group, C 1 ~ C 6 Haloalkylcarbonyl group, C 3 ~ C 8 Halocycloalkylcarbonyl group, C 1 ~ C 6 An alkoxycarbonyl group or C 1 ~ C 6 Optionally substituted by a haloalkoxycarbonyl group,
X 1a Is a hydrogen atom, cyano, -OH or R 24 Represents
X 1a X next to 1 Is adjacent X 1a And X 1 Is -CH 2 CH 2 CH 2 CH 2 -, -CH = CHCH = CH-, -N = CHCH = CH-, -CH = N-CH = CH-, -CH = CH-N = CH- or -CH = CH-CH = N-. X 1a And X 1 May form a 6-membered ring together with the atoms to which each of them is bonded, and in this case, a hydrogen atom bonded to each carbon atom forming the ring is a halogen atom, cyano, nitro, C 1 ~ C 6 Alkyl group, C 1 ~ C 6 Haloalkyl group, C 1 ~ C 6 Alkoxy group, C 1 ~ C 6 Alkylthio group, C 1 ~ C 6 An alkylsulfinyl group or C 1 ~ C 6 It may be optionally substituted with an alkylsulfonyl group.
X 1b Is a halogen atom, cyano, nitro, —OH, —SH or R 24 When f1, f2, f4, f5, f6, f7, f8 or f9 represents an integer of 2 or more, each X 1b May be the same as or different from each other, and two X 1b Are substituted on the same carbon, two X 1b Together oxo, thioxo, imino, C 1 ~ C 6 Alkylimino, C 1 ~ C 6 Alkoxyimino or C 1 ~ C 6 May form alkylidene,
Z is a halogen atom, cyano, nitro, —OH, —SH or R 24 When q represents an integer of 2 or more, each Z may be the same as or different from each other, and when two Zs are adjacent to each other, the two adjacent Zs are − CH 2 CH 2 CH 2 -, -CH 2 CH 2 O-, -CH 2 OCH 2 -, -OCH 2 O-, -CH 2 CH 2 S-, -CH 2 SCH 2 -, -CH 2 CH 2 CH 2 CH 2 -, -CH 2 CH 2 CH 2 O-, -CH 2 CH 2 OCH 2 -, -CH 2 OCH 2 O-, -OCH 2 CH 2 O-, -CH 2 CH 2 CH 2 S-, -OCH 2 CH 2 S-, -CH 2 CH = CH-, -OCH = CH-, -SCH = CH-, -N (X 1a ) CH = CH-, -OCH = N-, -SCH = N-, -N (X 1a ) CH = N-, -N (X 1a ) N = CH-, -OCH 2 CH = CH-, -N = CHCH = CH-, -CH = NCH = CH-, -N = NCH = CH-, -CH = NN = CH-, -N = CHCH = N- or -N = CHN = By forming CH—, a 5-membered ring or a 6-membered ring may be formed together with the carbon atom to which each Z is bonded. At this time, the hydrogen atom bonded to each carbon atom forming the ring is a halogen atom. , Cyano, nitro, C 1 ~ C 6 Alkyl group, C 1 ~ C 6 Haloalkyl group, C 1 ~ C 6 Alkoxy group, C 1 ~ C 6 Haloalkoxy group, C 1 ~ C 6 Alkylthio group, C 1 ~ C 6 Alkylsulfinyl group, C 1 ~ C 6 Alkylsulfonyl group, C 1 ~ C 6 Haloalkylthio group, C 1 ~ C 6 Haloalkylsulfinyl group, C 1 ~ C 6 Haloalkylsulfonyl group, C 1 ~ C 6 Alkylcarbonyl group, C 3 ~ C 8 A cycloalkylcarbonyl group, C 1 ~ C 6 Haloalkylcarbonyl group, C 3 ~ C 8 Halocycloalkylcarbonyl group, C 1 ~ C 6 An alkoxycarbonyl group or C 1 ~ C 6 Optionally substituted by a haloalkoxycarbonyl group,
R 24 Is C 1 ~ C 6 Alkyl, R 28 Optionally substituted by (C 1 ~ C 6 ) Alkyl, C 3 ~ C 8 Cycloalkyl, R 28 Optionally substituted by (C 3 ~ C 8 ) Cycloalkyl, C 2 ~ C 6 Alkenyl, R 28 Optionally substituted by (C 2 ~ C 6 ) Alkenyl, C 3 ~ C 8 Cycloalkenyl, R 28 Optionally substituted by (C 3 ~ C 8 ) Cycloalkenyl, C 2 ~ C 6 Alkynyl, R 28 Optionally substituted by (C 2 ~ C 6 ) Alkynyl, C 1 ~ C 6 Alkoxy, C 1 ~ C 6 Haloalkoxy, C 2 ~ C 6 Alkenyloxy, C 1 ~ C 6 Alkylthio, C 1 ~ C 6 Alkylsulfinyl, C 1 ~ C 6 Alkylsulfonyl, C 1 ~ C 6 Haloalkylthio, C 1 ~ C 6 Haloalkylsulfinyl, C 1 ~ C 6 Haloalkylsulfonyl, C 1 ~ C 6 Alkylcarbonyl, C 3 ~ C 8 Cycloalkylcarbonyl, C 1 ~ C 6 Haloalkylcarbonyl, C 3 ~ C 8 Halocycloalkylcarbonyl, C 1 ~ C 6 Alkoxycarbonyl, C 1 ~ C 6 Haloalkoxycarbonyl, C 1 ~ C 6 Alkylthiocarbonyl, C 1 ~ C 6 Alkoxythiocarbonyl, C 1 ~ C 6 Alkyldithiocarbonyl, C 1 ~ C 6 Alkylaminocarbonyl, C 1 ~ C 6 Haloalkylaminocarbonyl, di (C 1 ~ C 6 Alkyl) aminocarbonyl, tri (C 1 ~ C 6 Alkyl) silyl, C 1 ~ C 6 Alkylaminosulfonyl, di (C 1 ~ C 6 Alkyl) aminosulfonyl, C 1 ~ C 6 Alkylcarbonyloxy, C 1 ~ C 6 Alkylsulfonyloxy, C 1 ~ C 6 Haloalkylsulfonyloxy, C 1 ~ C 6 Alkylamino, di (C 1 ~ C 6 Alkyl) amino, -C (= NOR 29 ) R 30 , Phenyl, naphthyl, C 1 ~ C 6 Represents phenyl optionally substituted with alkyl or phenyl optionally substituted with halogen atoms;
R 28 , R 28a , R 31 And R 32 Are each independently a halogen atom, cyano, -OH, -SH, -NH 2 , -CHO, -C (O) OH, -C (O) NH 2 , -C (S) NH 2 , -S (O) 2 NH 2 , -Si (R 40a ) (R 40b ) R 40 , C 1 ~ C 6 Alkoxy, C 1 ~ C 6 Haloalkoxy, C 2 ~ C 6 Alkenyloxy, C 1 ~ C 6 Alkylthio, C 1 ~ C 6 Alkylsulfinyl, C 1 ~ C 6 Alkylsulfonyl, C 1 ~ C 6 Haloalkylthio, C 1 ~ C 6 Haloalkylsulfinyl, C 1 ~ C 6 Haloalkylsulfonyl, C 1 ~ C 6 Alkylcarbonyl, C 3 ~ C 8 Cycloalkylcarbonyl, C 1 ~ C 6 Haloalkylcarbonyl, C 3 ~ C 8 Halocycloalkylcarbonyl, C 1 ~ C 6 Alkoxycarbonyl, C 1 ~ C 6 Haloalkoxycarbonyl, C 1 ~ C 6 Alkylaminosulfonyl, di (C 1 ~ C 6 Alkyl) aminosulfonyl, C 1 ~ C 6 Alkylaminocarbonyl, di (C 1 ~ C 6 Alkyl) aminocarbonyl, C 1 ~ C 6 Alkylamino, di (C 1 ~ C 6 Alkyl) amino, phenyl, C 1 ~ C 6 Represents phenyl optionally substituted with alkyl or phenyl optionally substituted with halogen atoms;
R 29 And R 29a Are each independently C 1 ~ C 6 Alkyl, C 2 ~ C 6 Alkenyl, C 2 ~ C 6 Alkynyl, C 3 ~ C 8 Cycloalkyl, C 3 ~ C 8 Cycloalkenyl, R 31 Optionally substituted with (C 1 ~ C 6 ) Alkyl, R 31 Optionally substituted with (C 2 ~ C 6 ) Alkenyl, R 31 Optionally substituted with (C 2 ~ C 6 ) Alkynyl, R 31 Optionally substituted with (C 3 ~ C 8 ) Cycloalkyl or R 31 Optionally substituted with (C 3 ~ C 8 ) Represents cycloalkenyl.
R 30 And R 30a Are each independently C 1 ~ C 6 Alkyl, C 2 ~ C 6 Alkenyl, C 2 ~ C 6 Alkynyl, C 3 ~ C 8 Cycloalkyl, C 3 ~ C 8 Cycloalkenyl, R 32 Optionally substituted with (C 1 ~ C 6 ) Alkyl, R 32 Optionally substituted with (C 2 ~ C 6 ) Alkenyl, R 32 Optionally substituted with (C 2 ~ C 6 ) Alkynyl, R 32 Optionally substituted with (C 3 ~ C 8 ) Cycloalkyl, R 32 Optionally substituted with (C 3 ~ C 8 ) Cycloalkenyl, phenyl, C 1 ~ C 6 It represents phenyl optionally substituted with alkyl or phenyl optionally substituted with halogen atoms.
R 40 , R 40a And R 40b Are each independently C 1 ~ C 6 Alkyl, C 1 ~ C 6 Represents alkoxy or phenyl,
R 41 Is C 1 ~ C 6 Represents alkyl,
R 42 Is a halogen atom, cyano, C 1 ~ C 6 Alkyl, C 1 ~ C 6 Alkoxy, C 1 ~ C 6 Haloalkoxy, C 1 ~ C 6 Alkylthio, C 1 ~ C 6 Haloalkylthio, C 1 ~ C 6 Alkylsulfinyl, C 1 ~ C 6 Haloalkylsulfinyl, C 1 ~ C 6 Alkylsulfonyl, C 1 ~ C 6 Haloalkylsulfonyl, phenyl or (Z) q Represents phenyl substituted by
n, g1 and f1 each independently represent an integer of 0, 1, 2 or 3;
g2 and f2 each independently represent an integer of 0, 1 or 2;
g3 represents an integer of 0 or 1,
g4 and f4 each independently represent an integer of 0, 1, 2, 3 or 4;
f5 represents an integer of 0, 1, 2, 3, 4 or 5,
f6 represents an integer of 0, 1, 2, 3, 4, 5 or 6,
f7 represents an integer of 0, 1, 2, 3, 4, 5, 6 or 7,
f8 represents an integer of 0, 1, 2, 3, 4, 5, 6, 7 or 8;
f9 represents an integer of 0, 1, 2, 3, 4, 5, 6, 7, 8 or 9,
q represents an integer of 1, 2, 3, 4 or 5;
m1, m2 and m3 each independently represent an integer of 0 or 1,
r and r2 each independently represents an integer of 0, 1 or 2. Or a salt thereof.
は、−CRを表し、
は、水素原子、ハロゲン原子又はC〜Cアルキル表し、
は、ハロゲン原子又はC〜Cアルキルを表す請求項1記載の複素環誘導体又はその塩。
A 1 represents -CR 1
R 1 represents a hydrogen atom, a halogen atom or C 1 -C 6 alkyl,
The heterocyclic derivative or a salt thereof according to claim 1 , wherein R 2 represents a halogen atom or C 1 -C 6 alkyl.
は、水素原子を表し、
は、ハロゲン原子又はC〜Cアルキルを表し、
3aは、C〜Cアルキルを表し、
、R4a及びR4bは、水素原子を表し
Bは、B−1、B−2、B−3、B−5、B−7、B−9、B−17又はB−32を表し、
は、酸素原子を表し、
は、水素原子又はC〜Cアルキルを表し、
は、−C(O)R7bを表し、
7bは、−C(=NOR11b)R12bを表し、
11bは、C〜Cアルキルを表し、
12bは、C〜Cアルキル又はR15cによって任意に置換された(C〜C)アルキルを表し、
15cは、−S(O)16cを表し、
16cは、C〜Cアルキル又はC〜Cアルケニルを表し、
nは、0を表す請求項2記載の複素環誘導体又はその塩。
R 1 represents a hydrogen atom,
R 3 represents a halogen atom or C 1 -C 6 alkyl,
R 3a represents C 1 -C 6 alkyl;
R 4 , R 4a and R 4b represent a hydrogen atom. B represents B-1, B-2, B-3, B-5, B-7, B-9, B-17, or B-32. ,
Q 1 represents an oxygen atom,
R a represents a hydrogen atom or C 1 -C 6 alkyl;
R b represents -C (O) R 7b ;
R 7b represents -C (= NOR 11b ) R 12b ,
R 11b represents C 1 -C 6 alkyl,
R 12b represents C 1 -C 6 alkyl or (C 1 -C 6 ) alkyl optionally substituted with R 15c ,
R 15c represents -S (O) r R 16c ,
R 16c represents C 1 -C 6 alkyl or C 1 -C 6 alkenyl,
The heterocyclic derivative or a salt thereof according to claim 2, wherein n represents 0.
請求項1〜請求項3記載の複素環誘導体及びその塩から選ばれる1種又は2種以上を有効成分として含有する有害生物防除剤。   The pest control agent which contains 1 type, or 2 or more types chosen from the heterocyclic derivative and its salt of Claims 1-3 as an active ingredient. 請求項1〜請求項3記載の複素環誘導体及びその塩から選ばれる1種又は2種以上を有効成分として含有する農薬。   An agrochemical containing one or more selected from the heterocyclic derivatives according to claim 1 and a salt thereof as an active ingredient. 請求項1〜請求項3記載の複素環誘導体及びその塩から選ばれる1種又は2種以上を有効成分として含有する哺乳動物又は鳥類の内部もしくは外部寄生虫防除剤。   A mammalian or avian internal or ectoparasite control agent comprising one or more selected from the heterocyclic derivatives and salts thereof according to claim 1 as active ingredients. 請求項1〜請求項3記載の複素環誘導体及びその塩から選ばれる1種又は2種以上を有効成分として含有する殺虫剤又は殺ダニ剤。   The insecticide or acaricide which contains 1 type, or 2 or more types chosen from the heterocyclic derivative and its salt of Claims 1-3 as an active ingredient. 請求項1〜請求項3記載の複素環誘導体及びその塩から選ばれる1種又は2種以上を有効成分として含有する土壌処理剤。   The soil treatment agent which contains 1 type, or 2 or more types chosen from the heterocyclic derivative and its salt of Claims 1-3 as an active ingredient. 土壌処理方法が土壌潅注処理である請求項8記載の土壌処理剤。
The soil treatment agent according to claim 8, wherein the soil treatment method is soil irrigation treatment.
JP2014048820A 2013-03-12 2014-03-12 Heterocyclic derivative and pest control agent Pending JP2015147757A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2014048820A JP2015147757A (en) 2013-03-12 2014-03-12 Heterocyclic derivative and pest control agent

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
JP2013049500 2013-03-12
JP2013049500 2013-03-12
JP2014002935 2014-01-10
JP2014002935 2014-01-10
JP2014048820A JP2015147757A (en) 2013-03-12 2014-03-12 Heterocyclic derivative and pest control agent

Publications (1)

Publication Number Publication Date
JP2015147757A true JP2015147757A (en) 2015-08-20

Family

ID=53891465

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2014048820A Pending JP2015147757A (en) 2013-03-12 2014-03-12 Heterocyclic derivative and pest control agent

Country Status (1)

Country Link
JP (1) JP2015147757A (en)

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2019057724A1 (en) * 2017-09-22 2019-03-28 Syngenta Participations Ag Pyrazine-4carbamate or -urea derivatives as herbicides
WO2019057725A1 (en) * 2017-09-22 2019-03-28 Syngenta Participations Ag Pyrazine-4-carbamate or -urea derivatives as herbicides
WO2019057722A1 (en) * 2017-09-22 2019-03-28 Syngenta Participations Ag Pyrimidin-4-carbamate or urea derivatives as herbicides
JP2020534338A (en) * 2017-09-22 2020-11-26 シンジェンタ パーティシペーションズ アーゲー Pyrimidine- / pyrimidine-pyrimidine derivative with herbicidal activity
JP2020534339A (en) * 2017-09-22 2020-11-26 シンジェンタ パーティシペーションズ アーゲー Pyrimidine- / pyrimidine-pyrimidine derivative with herbicidal activity

Cited By (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2019057724A1 (en) * 2017-09-22 2019-03-28 Syngenta Participations Ag Pyrazine-4carbamate or -urea derivatives as herbicides
WO2019057725A1 (en) * 2017-09-22 2019-03-28 Syngenta Participations Ag Pyrazine-4-carbamate or -urea derivatives as herbicides
WO2019057722A1 (en) * 2017-09-22 2019-03-28 Syngenta Participations Ag Pyrimidin-4-carbamate or urea derivatives as herbicides
CN111315731A (en) * 2017-09-22 2020-06-19 先正达参股股份有限公司 Pyrazine-4-carbamate or-urea derivatives as herbicides
CN111315732A (en) * 2017-09-22 2020-06-19 先正达参股股份有限公司 Pyrazine-4-carbamate or-urea derivatives as herbicides
CN111356686A (en) * 2017-09-22 2020-06-30 先正达参股股份有限公司 Pyrimidine-4-carbamate or-urea derivatives as herbicides
JP2020534338A (en) * 2017-09-22 2020-11-26 シンジェンタ パーティシペーションズ アーゲー Pyrimidine- / pyrimidine-pyrimidine derivative with herbicidal activity
JP2020534340A (en) * 2017-09-22 2020-11-26 シンジェンタ パーティシペーションズ アーゲー Pyrazine-4-carbamate or urea derivative as a herbicide
JP2020534341A (en) * 2017-09-22 2020-11-26 シンジェンタ パーティシペーションズ アーゲー Pyrazine-4 carbamate or -urea derivative as a herbicide
JP2020534339A (en) * 2017-09-22 2020-11-26 シンジェンタ パーティシペーションズ アーゲー Pyrimidine- / pyrimidine-pyrimidine derivative with herbicidal activity
JP2020534342A (en) * 2017-09-22 2020-11-26 シンジェンタ パーティシペーションズ アーゲー Pyrimidine-4-carbamate or urea derivative as a herbicide
US11434221B2 (en) 2017-09-22 2022-09-06 Syngenta Participations Ag Pyrazine-4-carbamate or -urea derivatives as herbicides
JP7153068B2 (en) 2017-09-22 2022-10-13 シンジェンタ パーティシペーションズ アーゲー Pyrazine-4-carbamate or urea derivatives as herbicides
JP7206261B2 (en) 2017-09-22 2023-01-17 シンジェンタ パーティシペーションズ アーゲー Pyridyl-/pyrimidyl-pyrimidine derivatives with herbicidal activity
JP7237946B2 (en) 2017-09-22 2023-03-13 シンジェンタ パーティシペーションズ アーゲー Pyridyl-/pyrimidyl-pyrimidine derivatives with herbicidal activity
JP7252215B2 (en) 2017-09-22 2023-04-04 シンジェンタ パーティシペーションズ アーゲー Pyrimidine-4-carbamate or urea derivatives as herbicides
JP7271518B2 (en) 2017-09-22 2023-05-11 シンジェンタ パーティシペーションズ アーゲー Pyrazine-4 carbamate or -urea derivatives as herbicides
US11678665B2 (en) 2017-09-22 2023-06-20 Syngenta Participations Ag Pyrazine-4-carbamate or -urea derivatives as herbicides

Similar Documents

Publication Publication Date Title
JP5051340B2 (en) Substituted isoxazoline compounds and pest control agents
JP5007788B2 (en) Dihydroazole-substituted benzamide compounds and pest control agents
JP5316808B2 (en) Substituted isoxazoline or enone oxime compounds and pest control agents
JP5206993B2 (en) Isoxazoline-substituted benzamide compounds and pest control agents
KR101472517B1 (en) Substituted Isoxazoline Compound And Pest Control Agent
KR101416521B1 (en) Isoxazoline-substituted benzamide compound and harmful organism-controlling agent
US8268754B2 (en) Substituted dihydroazole compound and pest control agent
JP5365806B2 (en) Substituted isoxazoline compounds and pest control agents
JP2012188418A (en) Triazole derivative, and pest control agent
JP2013075871A (en) Thiazole derivative and pest controller
JP2013107867A (en) Pyrazole derivative and pest controlling agent
WO2012102387A1 (en) Pyrazole derivative and pest control agent
JP2007106756A (en) Substituted isoxazoline compound and pesticide
JP2013082699A (en) Pyrazole derivative and pest control agent
JP2013129651A (en) Thiazole derivative and pest control agent
JP2013082704A (en) Thiazole derivative and pest control agent
JP2013129653A (en) Triazole derivative and pest control agent
JP2008239611A (en) Isoxazoline-substituted benzamide compound and pesticide
JP2010083883A (en) Isoxazoline-substituted benzamide compound and harmful organism-controlling agent
JP2014208631A (en) Pyridine derivative and pest control agent
JP2018024672A (en) Condensed heterocyclic compound and pest control agent
JP2018024658A (en) Condensed heterocyclic compound and pest control agent
JP2010168367A (en) Substituted isoxazoline compound or substituted enone oxime compound, and pesticide
JP2015147757A (en) Heterocyclic derivative and pest control agent
JP2014015447A (en) Pyrazole derivative and pest control agent