FI903297A0 - 4h-indolo/1,2-d//1,2,4/triazolo/4,3-a// 1,4/benzodiazepiner, foerfarande foer deras framstaellning och deras anvaendning som laekemedel. - Google Patents

4h-indolo/1,2-d//1,2,4/triazolo/4,3-a// 1,4/benzodiazepiner, foerfarande foer deras framstaellning och deras anvaendning som laekemedel.

Info

Publication number
FI903297A0
FI903297A0 FI903297A FI903297A FI903297A0 FI 903297 A0 FI903297 A0 FI 903297A0 FI 903297 A FI903297 A FI 903297A FI 903297 A FI903297 A FI 903297A FI 903297 A0 FI903297 A0 FI 903297A0
Authority
FI
Finland
Prior art keywords
deras
benzodiazepiner
indolo
triazolo
foerfarande foer
Prior art date
Application number
FI903297A
Other languages
English (en)
Inventor
John Joseph Tegeler
Eileen Mary Gardenhire
Grover Cleveland Helsley
Original Assignee
Hoechst Roussel Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Roussel Pharma filed Critical Hoechst Roussel Pharma
Publication of FI903297A0 publication Critical patent/FI903297A0/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
FI903297A 1989-07-03 1990-06-29 4h-indolo/1,2-d//1,2,4/triazolo/4,3-a// 1,4/benzodiazepiner, foerfarande foer deras framstaellning och deras anvaendning som laekemedel. FI903297A0 (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/375,444 US4897392A (en) 1989-07-03 1989-07-03 4H-indolo(1,2-d)(1,2,4)triazolo(4,3-A)(1,4)benzodiazepines

Publications (1)

Publication Number Publication Date
FI903297A0 true FI903297A0 (fi) 1990-06-29

Family

ID=23480913

Family Applications (1)

Application Number Title Priority Date Filing Date
FI903297A FI903297A0 (fi) 1989-07-03 1990-06-29 4h-indolo/1,2-d//1,2,4/triazolo/4,3-a// 1,4/benzodiazepiner, foerfarande foer deras framstaellning och deras anvaendning som laekemedel.

Country Status (13)

Country Link
US (1) US4897392A (fi)
EP (1) EP0406719A1 (fi)
JP (1) JPH0344392A (fi)
KR (1) KR910002858A (fi)
AU (1) AU5801490A (fi)
CA (1) CA2020297A1 (fi)
FI (1) FI903297A0 (fi)
IE (1) IE902393A1 (fi)
IL (1) IL94950A0 (fi)
NO (1) NO902934L (fi)
NZ (1) NZ234316A (fi)
PT (1) PT94567A (fi)
ZA (1) ZA905149B (fi)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW201311B (fi) * 1991-06-17 1993-03-01 Hoffmann La Roche
US6515122B1 (en) * 1999-09-24 2003-02-04 Lion Bioscience Ag Tetracyclic benzimidazole derivatives and combinatorial libraries thereof
EP1809297B1 (en) * 2004-10-12 2008-07-30 F. Hoffmann-Roche AG Imidazo[1,5a]triazolo[1,5d]benzodiazepine derivatives for the treatment of cognitive disorders
WO2006045429A1 (en) * 2004-10-20 2006-05-04 F. Hoffmann-La Roche Ag Halogen substituted benzodiazepine derivatives
WO2006045430A1 (en) * 2004-10-20 2006-05-04 F. Hoffmann-La Roche Ag Imidazo-benzodiazepine derivatives
BRPI0515800A (pt) * 2004-12-14 2008-08-05 Hoffmann La Roche imidazo-benzodiazepinas tetracìclicas como moduladores de receptores de gaba
ES2374870T3 (es) * 2008-03-27 2012-02-22 Bristol-Myers Squibb Company Inhibidores de ns5b de vhc de indolobenzadiazepina fusionada con heterocíclicos aromáticos.

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3375246A (en) * 1965-06-11 1968-03-26 Sandoz Ag Isoindolines
US3642779A (en) * 1969-10-22 1972-02-15 Robins Co Inc A H Indolo(1 2-d)(1 4)benzodiazepin-6-ones
US3642778A (en) * 1969-10-22 1972-02-15 Robins Co Inc A H Benzimidazo(1 2-d)(1 4)benzodiazepin-6(5h)-ones
US4013763A (en) * 1974-07-12 1977-03-22 Takeda Chemical Industries, Ltd. Heterocyclic compounds
JPS5572177A (en) * 1978-11-27 1980-05-30 Shionogi & Co Ltd 4,1-benzoxazepine or 4,1-benzothiazepine
US4587244A (en) * 1984-04-11 1986-05-06 Mcneilab, Inc. Amidine benzodiazepines, methods for their use and intermediates
US4596799A (en) * 1985-01-29 1986-06-24 Ciba-Geigy Corporation 9H-pyrrolo[2,1-c]-1,2,4-triazolo[4,3-a][1,4]benzodiazepines
US4737496A (en) * 1986-10-01 1988-04-12 Ciba-Geigy Corporation 1,3,4,16b-tetrahydro-2H,10H-indolo[2,1-c]pyrazino-[1,2-a][1,4]benzodiazepines useful as serotonin-2 receptor antagonists

Also Published As

Publication number Publication date
EP0406719A1 (en) 1991-01-09
AU5801490A (en) 1991-01-03
NO902934L (no) 1991-01-04
KR910002858A (ko) 1991-02-26
JPH0344392A (ja) 1991-02-26
ZA905149B (en) 1991-04-24
NZ234316A (en) 1992-03-26
IL94950A0 (en) 1991-06-10
PT94567A (pt) 1991-03-20
US4897392A (en) 1990-01-30
CA2020297A1 (en) 1991-01-04
IE902393A1 (en) 1991-06-19
NO902934D0 (no) 1990-07-02

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Legal Events

Date Code Title Description
FA Application withdrawn

Owner name: HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED