DK1440075T3 - Hidtil ukendte heteroaromatiske 3beta-aminio-azabicyclooctan-amidderivater, fremgangsmåde til fremstilling deraf og terapeutisk anvendelse deraf - Google Patents

Hidtil ukendte heteroaromatiske 3beta-aminio-azabicyclooctan-amidderivater, fremgangsmåde til fremstilling deraf og terapeutisk anvendelse deraf

Info

Publication number
DK1440075T3
DK1440075T3 DK02785568T DK02785568T DK1440075T3 DK 1440075 T3 DK1440075 T3 DK 1440075T3 DK 02785568 T DK02785568 T DK 02785568T DK 02785568 T DK02785568 T DK 02785568T DK 1440075 T3 DK1440075 T3 DK 1440075T3
Authority
DK
Denmark
Prior art keywords
sub
pyridine
furo
thieno
group
Prior art date
Application number
DK02785568T
Other languages
English (en)
Inventor
Barbara Monse
Thierry Imbert
Wouter Koek
Original Assignee
Pf Medicament
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pf Medicament filed Critical Pf Medicament
Application granted granted Critical
Publication of DK1440075T3 publication Critical patent/DK1440075T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
DK02785568T 2001-11-02 2002-10-30 Hidtil ukendte heteroaromatiske 3beta-aminio-azabicyclooctan-amidderivater, fremgangsmåde til fremstilling deraf og terapeutisk anvendelse deraf DK1440075T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0114220A FR2831884B1 (fr) 2001-11-02 2001-11-02 Nouveaux derives amides heteroaromatiques de 3 beta-amino azabicyclooctane, leur procede de preparation et leurs applications en therapeutique
PCT/FR2002/003737 WO2003037904A1 (fr) 2001-11-02 2002-10-30 NOUVEAUX DERIVES AMIDES HETEROAROMATIQUES DE 3β-AMINO AZABICYCLOOCTANE, LEUR PROCEDE DE PREPARATION ET LEURS APPLICATIONS EN THERAPEUTIQUE

Publications (1)

Publication Number Publication Date
DK1440075T3 true DK1440075T3 (da) 2005-08-22

Family

ID=8869022

Family Applications (1)

Application Number Title Priority Date Filing Date
DK02785568T DK1440075T3 (da) 2001-11-02 2002-10-30 Hidtil ukendte heteroaromatiske 3beta-aminio-azabicyclooctan-amidderivater, fremgangsmåde til fremstilling deraf og terapeutisk anvendelse deraf

Country Status (9)

Country Link
US (1) US7456192B2 (da)
EP (1) EP1440075B1 (da)
AT (1) ATE297399T1 (da)
DE (1) DE60204582T2 (da)
DK (1) DK1440075T3 (da)
ES (1) ES2243779T3 (da)
FR (1) FR2831884B1 (da)
PT (1) PT1440075E (da)
WO (1) WO2003037904A1 (da)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU227684B1 (en) 2003-08-29 2011-11-28 Sanofi Aventis Adamantane and azabicyclo-octane and nonane derivatives and their use as dpp-iv inhibitors
ES2440746T3 (es) 2008-04-11 2014-01-30 Janssen Pharmaceutica, N.V. Triazolopiridina-2-iloxi-fenil y triazolopiridina-iloxi-fenil amino como moduladores del leucotrieno A4 hidrolasa
WO2010087762A1 (en) * 2009-01-28 2010-08-05 Astrazeneca Ab 2-aza-bicyclo[2.2.1]heptane compounds and uses thereof
JP5690286B2 (ja) * 2009-03-04 2015-03-25 イデニク プハルマセウティカルス，インコーポレイテッド ホスホチオフェン及びホスホチアゾールｈｃｖポリメラーゼ阻害剤
CN102459251B (zh) 2009-05-14 2015-05-20 詹森药业有限公司 作为白三烯a4水解酶的调节剂的具有两个稠合双环杂芳基部分的化合物
US9481679B2 (en) 2012-12-17 2016-11-01 Sun Pharmaceutical Industries Limited Process for the preparation of tofacitinib and intermediates thereof
CN109851551B (zh) * 2018-12-11 2022-05-20 大连金点生物科技有限公司 一种合成3-溴异烟酸中间体的方法
JP2022526901A (ja) 2019-03-19 2022-05-27 ベーリンガー インゲルハイム アニマル ヘルス ユーエスエイ インコーポレイテッド 駆虫性アザベンゾチオフェンおよびアザベンゾフラン化合物
PE20231205A1 (es) 2020-05-29 2023-08-17 Boehringer Ingelheim Animal Health Usa Inc Compuestos heterociclicos como anthelminticos

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL59004A0 (en) 1978-12-30 1980-03-31 Beecham Group Ltd Substituted benzamides their preparation and pharmaceutical compositions containing them
FR2476088A2 (fr) 1979-01-16 1981-08-21 Delalande Sa Nouveaux derives du nor-tropane, leur procede de preparation et leur application en therapeutique
US4910193A (en) 1985-12-16 1990-03-20 Sandoz Ltd. Treatment of gastrointestinal disorders
AU3364493A (en) 1992-01-28 1993-09-01 Smithkline Beecham Plc Compounds as calcium channel antagonists
FR2738569B1 (fr) * 1995-09-12 1997-11-28 Pf Medicament Nouveaux derives naphtamide de 3 beta-amino azabicyclo octane ou nonane, leur procede de preparation, leur utilisation a titre de medicament antipsychotique
SE9902987D0 (sv) 1999-08-24 1999-08-24 Astra Pharma Prod Novel compounds

Also Published As

Publication number Publication date
US7456192B2 (en) 2008-11-25
DE60204582T2 (de) 2006-03-16
ES2243779T3 (es) 2005-12-01
EP1440075B1 (fr) 2005-06-08
FR2831884A1 (fr) 2003-05-09
PT1440075E (pt) 2005-10-31
WO2003037904A1 (fr) 2003-05-08
US20050080085A1 (en) 2005-04-14
EP1440075A1 (fr) 2004-07-28
DE60204582D1 (de) 2005-07-14
ATE297399T1 (de) 2005-06-15
FR2831884B1 (fr) 2003-12-26

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