ZA982369B - Dihydropyrazino[1,2-a]indol-1-one derivatives their preparation and their use in therapy - Google Patents

Dihydropyrazino[1,2-a]indol-1-one derivatives their preparation and their use in therapy

Info

Publication number
ZA982369B
ZA982369B ZA982369A ZA982369A ZA982369B ZA 982369 B ZA982369 B ZA 982369B ZA 982369 A ZA982369 A ZA 982369A ZA 982369 A ZA982369 A ZA 982369A ZA 982369 B ZA982369 B ZA 982369B
Authority
ZA
South Africa
Prior art keywords
dihydropyrazino
indol
therapy
derivatives
preparation
Prior art date
Application number
ZA982369A
Other languages
English (en)
Inventor
Gary Mccort
Christian Hoornaert
Caroline Cadilhac
Olivier Duclos
Eric Guilpain
Genevieve Dellac
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of ZA982369B publication Critical patent/ZA982369B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ZA982369A 1997-03-20 1998-03-19 Dihydropyrazino[1,2-a]indol-1-one derivatives their preparation and their use in therapy ZA982369B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9703389A FR2761070B1 (fr) 1997-03-20 1997-03-20 Derives de dihydropyrazino[1,2-a]indole-1-one, leur preparation et leur application en therapeutique

Publications (1)

Publication Number Publication Date
ZA982369B true ZA982369B (en) 1998-09-23

Family

ID=9505000

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA982369A ZA982369B (en) 1997-03-20 1998-03-19 Dihydropyrazino[1,2-a]indol-1-one derivatives their preparation and their use in therapy

Country Status (6)

Country Link
EP (1) EP0971926A1 (es)
AR (1) AR012095A1 (es)
AU (1) AU6924098A (es)
FR (1) FR2761070B1 (es)
WO (1) WO1998042710A1 (es)
ZA (1) ZA982369B (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2001232319B2 (en) 2000-02-18 2005-01-13 Meiji Seika Kaisha, Ltd. Phenoxyalkylamine derivates useful as opioid delta receptor ligands
DK2825542T3 (en) 2012-03-16 2017-01-09 Vitae Pharmaceuticals Inc LIVER-X-receptor modulators
AU2013232066B2 (en) 2012-03-16 2017-07-06 Vitae Pharmaceuticals, Inc. Liver X receptor modulators
CA2943815C (en) 2014-03-27 2023-04-04 Vanderbilt University Substituted indole mcl-1 inhibitors
US9949965B2 (en) 2014-10-17 2018-04-24 Vanderbilt University Tricyclic indole Mcl-1 inhibitors and uses thereof
BR112018067775B1 (pt) 2016-03-04 2024-02-15 Vanderbilt University Compostos inibidores de mcl-1 indol substituídos, composição farmacêutica compreendendo ditos compostos e usos terapêuticos dos mesmos

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2027898A6 (es) * 1991-01-24 1992-06-16 Espanola Prod Quimicos Procedimiento de preparacion de nuevos derivados de la 2-metoxifenilpiperacina.
EP0572863A1 (de) * 1992-06-05 1993-12-08 F. Hoffmann-La Roche Ag ZNS Pyrazinoindole

Also Published As

Publication number Publication date
WO1998042710A1 (fr) 1998-10-01
AU6924098A (en) 1998-10-20
EP0971926A1 (fr) 2000-01-19
FR2761070A1 (fr) 1998-09-25
FR2761070B1 (fr) 1999-04-23
AR012095A1 (es) 2000-09-27

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