ZA9510960B - Heterocyclic keto arginine peptided as thrombin inhibitors - Google Patents

Heterocyclic keto arginine peptided as thrombin inhibitors

Info

Publication number
ZA9510960B
ZA9510960B ZA9510960A ZA9510960A ZA9510960B ZA 9510960 B ZA9510960 B ZA 9510960B ZA 9510960 A ZA9510960 A ZA 9510960A ZA 9510960 A ZA9510960 A ZA 9510960A ZA 9510960 B ZA9510960 B ZA 9510960B
Authority
ZA
South Africa
Prior art keywords
peptided
thrombin inhibitors
arginine
heterocyclic keto
heterocyclic
Prior art date
Application number
ZA9510960A
Inventor
John W Gillard
John Dimaio
Arshad M Siddiqui
Patrice Preville
Doninique Lafleur
Annette Marian Doherty
Jeremy John Edmonds
Original Assignee
Iaf Biochem Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Iaf Biochem Int filed Critical Iaf Biochem Int
Publication of ZA9510960B publication Critical patent/ZA9510960B/en

Links

ZA9510960A 1994-12-22 1995-12-22 Heterocyclic keto arginine peptided as thrombin inhibitors ZA9510960B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9426038.7A GB9426038D0 (en) 1994-12-22 1994-12-22 Low molecular weight bicyclic thrombin inhibitors

Publications (1)

Publication Number Publication Date
ZA9510960B true ZA9510960B (en) 1996-07-09

Family

ID=10766468

Family Applications (2)

Application Number Title Priority Date Filing Date
ZA9510960A ZA9510960B (en) 1994-12-22 1995-12-22 Heterocyclic keto arginine peptided as thrombin inhibitors
ZA9510961A ZA9510961B (en) 1994-12-22 1995-12-22 Low molecular weight bicyclic thrombin inhibitors

Family Applications After (1)

Application Number Title Priority Date Filing Date
ZA9510961A ZA9510961B (en) 1994-12-22 1995-12-22 Low molecular weight bicyclic thrombin inhibitors

Country Status (3)

Country Link
GB (2) GB9426038D0 (en)
LT (1) LT4368B (en)
ZA (2) ZA9510960B (en)

Family Cites Families (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4097472A (en) 1974-11-08 1978-06-27 Mitsubishi Chemical Industries Limited N2 -arylsulfonyl-l-argininamides and the pharmaceutically acceptable salts thereof
US4097591A (en) 1974-11-08 1978-06-27 Mitsubishi Chemical Industries Limited N2 -arylsulfonyl-L-argininamides and the pharmaceutically acceptable salts thereof
US4096255A (en) 1974-11-08 1978-06-20 Mitsubishi Chemical Industries Limited N2 -naphthalenesulfonyl-L-argininamides, and pharmaceutical salts, compositions and methods
US4173630A (en) 1974-11-08 1979-11-06 Mitsubishi Chemical Industries Limited N2 Arylsulfonyl-L-argininamides and the pharmaceutically acceptable salts thereof
CA1131621A (en) 1977-01-19 1982-09-14 Shosuke Okamoto N.sup.2-arylsulfonyl-l-argininamides and the pharmaceutically acceptable salts thereof
US4046876A (en) 1974-11-08 1977-09-06 Mitsubishi Chemical Industries Limited N2 -alkoxynaphthalenesulfonyl-L-argininamides and the pharmaceutically acceptable salts thereof
US4318904A (en) 1980-04-25 1982-03-09 Research Corporation Peptide affinity labels for thrombin and other trypsin-like proteases
US4781866A (en) 1985-03-15 1988-11-01 Mcneilab, Inc. Process for producing amidine sulfonic acid intermediates for guanidines
CA1341032C (en) 1987-01-23 2000-06-20 John L. Krstenansky Anticoagulant peptides
US4753077A (en) 1987-06-01 1988-06-28 Synthetic Sink Multi-staged turbine system with bypassable bottom stage
AU3098289A (en) 1988-03-04 1989-09-07 Biogen, Inc. Hirudin peptides
NZ228995A (en) 1988-05-10 1992-03-26 Merrell Dow Pharma Hirudin peptide derivatives and pharmaceutical compositions
US5196404B1 (en) 1989-08-18 1996-09-10 Biogen Inc Inhibitors of thrombin
US5138650A (en) 1990-09-27 1992-08-11 Motorola, Inc. Cordless telephone with internal debit and credit memory
JPH05503300A (en) 1990-11-15 1993-06-03 ペンタファルム　アクチェンゲゼルシャフト Meta-substituted phenylalanine derivatives
US5158091A (en) 1990-11-30 1992-10-27 Ivac Corporation Tonometry system for determining blood pressure
DE4127404A1 (en) 1991-08-19 1993-02-25 Thomae Gmbh Dr K CYCLIC IMINODERIVATES, MEDICAMENTS CONTAINING SUCH COMPOUNDS AND METHOD FOR THE PRODUCTION THEREOF
DE69321344D1 (en) 1992-02-14 1998-11-05 Corvas Int Inc INHIBITORS OF THROMBOSE
GB9209032D0 (en) 1992-04-25 1992-06-10 Ciba Geigy Ag New peptide derivatives
US5371072A (en) 1992-10-16 1994-12-06 Corvas International, Inc. Asp-Pro-Arg α-keto-amide enzyme inhibitors
JPH06219948A (en) 1993-01-25 1994-08-09 Mitsubishi Kasei Corp Antithrombin agent and its production
WO1994017817A1 (en) 1993-02-12 1994-08-18 Corvas International, Inc. Inhibitors of thrombosis

Also Published As

Publication number Publication date
LT4368B (en) 1998-08-25
GB9426038D0 (en) 1995-02-22
LT97132A (en) 1998-03-25
GB9503136D0 (en) 1995-04-05
ZA9510961B (en) 1996-07-09

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