ZA200608778B - Pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists - Google Patents

Pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists

Info

Publication number
ZA200608778B
ZA200608778B ZA200608778A ZA200608778A ZA200608778B ZA 200608778 B ZA200608778 B ZA 200608778B ZA 200608778 A ZA200608778 A ZA 200608778A ZA 200608778 A ZA200608778 A ZA 200608778A ZA 200608778 B ZA200608778 B ZA 200608778B
Authority
ZA
South Africa
Prior art keywords
triazolo
pyrazolo
receptor antagonists
pyrimidine adenosine
adenosine
Prior art date
Application number
ZA200608778A
Inventor
Bernard R Neustadt
Hao Jinsong
Liu Hong
Craig D Boyle
Chackalamannil Samuel
Unmesh G Shah
Stamford Andrew
Joel M Harris
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Publication of ZA200608778B publication Critical patent/ZA200608778B/en

Links

ZA200608778A 2004-04-21 2006-10-20 Pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists ZA200608778B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US56391304P 2004-04-21 2004-04-21

Publications (1)

Publication Number Publication Date
ZA200608778B true ZA200608778B (en) 2008-09-25

Family

ID=38126306

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200608778A ZA200608778B (en) 2004-04-21 2006-10-20 Pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists

Country Status (2)

Country Link
CN (1) CN1976935A (en)
ZA (1) ZA200608778B (en)

Also Published As

Publication number Publication date
CN1976935A (en) 2007-06-06

Similar Documents

Publication Publication Date Title
IL178674A0 (en) PYRAZOLO-[4,3-e]-1,2,4-TRIAZOLO-[1,5-c]-PYRIMIDINE ADENOSINE A2A RECEPTOR ANTAGONISTS
HK1085466A1 (en) 2-alkynyl-and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c] - pyrimidine adenosine a2a receptor antagonists
IL160878A0 (en) Imidazo (4,3-e)-1,2,4-triazolo (1,5-c) pyrimidines as adenosine a2a receptor antagonists
IL220174A0 (en) 5-AMINO - {PYRAZOLO-[4,3-e]-1,2,4-TRIAZOLO[1,5-c]PYRIMIDINE}-2-AND 7-SUBSTITUTED DERIVATIVES AS ADENOSINE A2A RECEPTOR INHIBITORS
DK2217578T5 (en) [1,2,4] triazolo [1,5-A] pyridine and [1,2,4] triazolo [1,5-C] pyrimidine compounds and their use
IL175759A0 (en) A2b adenosine receptor antagonists
IL178365A (en) Selective antagonists of a2a adenosine receptors
IL190336A0 (en) Imidazopyridine derivatives as a2b adenosine receptor antagonists
SG160438A1 (en) Process for preparing pyrido[2,3-d]pyrimidin-7-one and 3,4-dihydropyrimido[4,5- d]pyrimidin-2(1h)-one derivatives
IL158214A0 (en) 8-heteroaryl xanthine adenosine a2b receptor antagonists
HK1137753A1 (en) Pyrido[4,3-d]pyrimidin-4(3h)-one derivatives as calcium receptor antagonists
EP1599482A4 (en) Pyrazolo 1,5-a pyrimidine derivatives
HUP0402324A3 (en) [1,2,4]triazolo[1,5-a]pyridine and [1,2,4]triazolo[1,5-c]pyrimidine derivatives as adenosine a2a receptor antagonists and pharmaceutical compositions containing them
IL182528A0 (en) Purine derivatives for use as adenosin a-2a receptor antagonists
HK1063780A1 (en) Adenosine a2a receptor antagonists
IL161572A0 (en) Adenosine a2a receptor antagonists
HK1138581A1 (en) Triazolo [1, 5-a] quinolines as adenosine a3 receptor ligands
PL370565A1 (en) 5-methoxy-8-aryl-[1,2,4] triazolo [1,5-a] pyridine derivatives as adenosine receptor antagonists
PL1678182T3 (en) Process for preparing substituted 5-amino-pyrazolo- [4,3-e]-1,2,4-triazolo [1,5-c]pyrimidines
ZA200608778B (en) Pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists
GB2454549B (en) Uses of 2-[piperidinyl]methyl-2,3-dihydroimidazo[1,2-c]quinazolin-5(6H)-one for providing an anti-allergic effect and histamine H1 receptor antagonism effect
EP1636230A4 (en) A1 adenosine receptor antagonists
TH0401001406A (en) 2-alkynyl-and 2-alkenyl-pyrasolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidines which is an antagonist of the adenosine A2a receptor.
PL366807A1 (en) New derivatives of 1h-pyrazolo[4,3-e]-1,2,4-triazolo[3,4-b][1,2,4]- triazine system