WO2020210320A8 - L,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-ones substituées - Google Patents
L,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-ones substituées Download PDFInfo
- Publication number
- WO2020210320A8 WO2020210320A8 PCT/US2020/027218 US2020027218W WO2020210320A8 WO 2020210320 A8 WO2020210320 A8 WO 2020210320A8 US 2020027218 W US2020027218 W US 2020027218W WO 2020210320 A8 WO2020210320 A8 WO 2020210320A8
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- pyrazolo
- pyrimidin
- dihydro
- ones
- substituted
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
L'invention concerne des composés de formule (I). De tels composés, ainsi que des sels pharmaceutiquement acceptables et des compositions de ceux-ci, sont utiles pour traiter des maladies ou des affections, y compris des affections caractérisées par une prolifération cellulaire excessive, telles que le cancer du sein.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201962832529P | 2019-04-11 | 2019-04-11 | |
US62/832,529 | 2019-04-11 |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2020210320A1 WO2020210320A1 (fr) | 2020-10-15 |
WO2020210320A8 true WO2020210320A8 (fr) | 2020-11-12 |
Family
ID=72750610
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/US2020/027218 WO2020210320A1 (fr) | 2019-04-11 | 2020-04-08 | L,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-ones substituées |
Country Status (1)
Country | Link |
---|---|
WO (1) | WO2020210320A1 (fr) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN111902413B (zh) | 2018-03-09 | 2023-10-17 | 里科瑞尔姆Ip控股有限责任公司 | 取代的1,2-二氢-3H-吡唑并[3,4-d]嘧啶-3-酮 |
JP2024517085A (ja) * | 2021-04-12 | 2024-04-19 | リキュリウム アイピー ホールディングス リミテッド ライアビリティー カンパニー | 子宮漿液性がんを治療するためのwee1化合物 |
CN117751122A (zh) * | 2021-08-11 | 2024-03-22 | 微境生物医药科技(上海)有限公司 | 作为Wee-1抑制剂的1,2-二氢-3H-吡唑[3,4-d]嘧啶-3-酮化合物 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AR060635A1 (es) * | 2006-04-27 | 2008-07-02 | Banyu Pharma Co Ltd | Derivados de 1,2-dihidro-3h-pirazolo[3,4-d]pirimidin-3-ona, composiciones farmaceuticas que los comprenden y su uso en el tratamiento del cancer |
US8329711B2 (en) * | 2007-10-23 | 2012-12-11 | Msd K.K. | Pyridone-substituted-dihydropyrazolopyrimidinone derivative |
WO2019028008A1 (fr) * | 2017-08-01 | 2019-02-07 | Zeno Royalties & Milestones, LLC | Analogues de 1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-one |
EP3694861A4 (fr) * | 2017-10-09 | 2021-05-19 | Nuvation Bio Inc. | Composés hétérocycliques et leurs utilisations |
CN111902413B (zh) * | 2018-03-09 | 2023-10-17 | 里科瑞尔姆Ip控股有限责任公司 | 取代的1,2-二氢-3H-吡唑并[3,4-d]嘧啶-3-酮 |
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2020
- 2020-04-08 WO PCT/US2020/027218 patent/WO2020210320A1/fr active Application Filing
Also Published As
Publication number | Publication date |
---|---|
WO2020210320A1 (fr) | 2020-10-15 |
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