WO2020055359A3 - Forme posologique orale de tosylate de sorafénib - Google Patents

Forme posologique orale de tosylate de sorafénib Download PDF

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Publication number
WO2020055359A3
WO2020055359A3 PCT/TR2019/050578 TR2019050578W WO2020055359A3 WO 2020055359 A3 WO2020055359 A3 WO 2020055359A3 TR 2019050578 W TR2019050578 W TR 2019050578W WO 2020055359 A3 WO2020055359 A3 WO 2020055359A3
Authority
WO
WIPO (PCT)
Prior art keywords
dosage form
oral dosage
sorafenib tosylate
present
sorafenib
Prior art date
Application number
PCT/TR2019/050578
Other languages
English (en)
Other versions
WO2020055359A2 (fr
Inventor
Ali Turkyilmaz
Ali Ihsan SECKIN
Irem Yenice
Yuksel TOPALOGLU
Original Assignee
Arven Ilac Sanayi Ve Ticaret Anonim Sirketi
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Arven Ilac Sanayi Ve Ticaret Anonim Sirketi filed Critical Arven Ilac Sanayi Ve Ticaret Anonim Sirketi
Publication of WO2020055359A2 publication Critical patent/WO2020055359A2/fr
Publication of WO2020055359A3 publication Critical patent/WO2020055359A3/fr

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2009Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Inorganic Chemistry (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)

Abstract

L'invention concerne une forme posologique orale comprenant du tosylate de sorafénib en tant que principe actif qui présente des propriétés améliorées. La présente invention concerne également un procédé de préparation de ladite composition.
PCT/TR2019/050578 2018-08-10 2019-07-16 Forme posologique orale de tosylate de sorafénib WO2020055359A2 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
TR2018/11686 2018-08-10
TR201811686 2018-08-10

Publications (2)

Publication Number Publication Date
WO2020055359A2 WO2020055359A2 (fr) 2020-03-19
WO2020055359A3 true WO2020055359A3 (fr) 2020-06-04

Family

ID=69776588

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/TR2019/050578 WO2020055359A2 (fr) 2018-08-10 2019-07-16 Forme posologique orale de tosylate de sorafénib

Country Status (1)

Country Link
WO (1) WO2020055359A2 (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2023155182A1 (fr) * 2022-02-21 2023-08-24 北京睿创康泰医药研究院有限公司 Formulation orale de sorafénib ou de donafénib à faible dose et à exposition de forte intensité, et son utilisation

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20030125359A1 (en) * 2001-12-04 2003-07-03 Lyons John F. RAF-MEK-ERK pathway inhibitors to treat cancer
WO2007059154A2 (fr) * 2005-11-14 2007-05-24 Bayer Healthcare Llc Traitement de cancers a resistance acquise a des inhibiteurs de kit

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20030125359A1 (en) * 2001-12-04 2003-07-03 Lyons John F. RAF-MEK-ERK pathway inhibitors to treat cancer
WO2007059154A2 (fr) * 2005-11-14 2007-05-24 Bayer Healthcare Llc Traitement de cancers a resistance acquise a des inhibiteurs de kit

Also Published As

Publication number Publication date
WO2020055359A2 (fr) 2020-03-19

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