WO2019209208A3 - Compositions pharmaceutiques d'ivabradine à libération contrôlée - Google Patents

Compositions pharmaceutiques d'ivabradine à libération contrôlée Download PDF

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Publication number
WO2019209208A3
WO2019209208A3 PCT/TR2018/050818 TR2018050818W WO2019209208A3 WO 2019209208 A3 WO2019209208 A3 WO 2019209208A3 TR 2018050818 W TR2018050818 W TR 2018050818W WO 2019209208 A3 WO2019209208 A3 WO 2019209208A3
Authority
WO
WIPO (PCT)
Prior art keywords
controlled
ivabradine
pharmaceutical compositions
release pharmaceutical
release
Prior art date
Application number
PCT/TR2018/050818
Other languages
English (en)
Other versions
WO2019209208A2 (fr
Inventor
Ali TÜRKYILMAZ
Arzu Palantöken
Dicle Güner
Original Assignee
Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi filed Critical Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi
Publication of WO2019209208A2 publication Critical patent/WO2019209208A2/fr
Publication of WO2019209208A3 publication Critical patent/WO2019209208A3/fr

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2009Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2031Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

Abstract

La présente invention concerne des compositions pharmaceutiques à libération contrôlée comprenant de l'ivabradine ou un sel, un solvate ou un polymorphe pharmaceutiquement acceptable de ce composé et au moins un agent à libération contrôlée.
PCT/TR2018/050818 2017-12-18 2018-12-17 Compositions pharmaceutiques d'ivabradine à libération contrôlée WO2019209208A2 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
TR2017/20672 2017-12-18
TR2017/20672A TR201720672A2 (tr) 2017-12-18 2017-12-18 İvabradi̇ni̇n kontrollü salimli farmasöti̇k kompozi̇syonlari

Publications (2)

Publication Number Publication Date
WO2019209208A2 WO2019209208A2 (fr) 2019-10-31
WO2019209208A3 true WO2019209208A3 (fr) 2020-01-16

Family

ID=67900851

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/TR2018/050818 WO2019209208A2 (fr) 2017-12-18 2018-12-17 Compositions pharmaceutiques d'ivabradine à libération contrôlée

Country Status (2)

Country Link
TR (1) TR201720672A2 (fr)
WO (1) WO2019209208A2 (fr)

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2010128525A2 (fr) * 2009-05-04 2010-11-11 Dinesh Shantilal Patel Préparation d'ivabradine dans le traitement des maladies cardiovasculaires
WO2011157720A2 (fr) * 2010-06-14 2011-12-22 Ratiopharm Gmbh Composition pharmaceutique contenant de l'ivabradine à libération modifiée
EP2740478A1 (fr) * 2011-08-05 2014-06-11 Jiangsu Hengrui Medicine Co., Ltd. Préparation à libération entretenue d'ivabradine ou de sels pharmaceutiquement acceptables de celle-ci

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2010128525A2 (fr) * 2009-05-04 2010-11-11 Dinesh Shantilal Patel Préparation d'ivabradine dans le traitement des maladies cardiovasculaires
WO2011157720A2 (fr) * 2010-06-14 2011-12-22 Ratiopharm Gmbh Composition pharmaceutique contenant de l'ivabradine à libération modifiée
EP2740478A1 (fr) * 2011-08-05 2014-06-11 Jiangsu Hengrui Medicine Co., Ltd. Préparation à libération entretenue d'ivabradine ou de sels pharmaceutiquement acceptables de celle-ci

Also Published As

Publication number Publication date
TR201720672A2 (tr) 2019-07-22
WO2019209208A2 (fr) 2019-10-31

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