WO2019020981A1 - Dérivés de pyrazole, d'isothiazole et d'isoxazole utiles en tant que fongicides agricoles - Google Patents

Dérivés de pyrazole, d'isothiazole et d'isoxazole utiles en tant que fongicides agricoles Download PDF

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Publication number
WO2019020981A1
WO2019020981A1 PCT/GB2018/052071 GB2018052071W WO2019020981A1 WO 2019020981 A1 WO2019020981 A1 WO 2019020981A1 GB 2018052071 W GB2018052071 W GB 2018052071W WO 2019020981 A1 WO2019020981 A1 WO 2019020981A1
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WIPO (PCT)
Prior art keywords
alkyl
compound
haloalkyl
ring
independently
Prior art date
Application number
PCT/GB2018/052071
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English (en)
Inventor
Christopher John Urch
Victoria Elizabeth JACKSON
Linda Jordan
Effi BAETZNER
Oliver James Stephen MCGAW
Original Assignee
Redag Crop Protection Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB1711872.0A external-priority patent/GB201711872D0/en
Priority claimed from GBGB1719097.6A external-priority patent/GB201719097D0/en
Priority claimed from GBGB1807495.5A external-priority patent/GB201807495D0/en
Application filed by Redag Crop Protection Ltd. filed Critical Redag Crop Protection Ltd.
Publication of WO2019020981A1 publication Critical patent/WO2019020981A1/fr

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

La présente invention concerne des composés pyrazole, isoxazole et isothiazole qui sont utilisés dans le domaine de l'agriculture en tant que fongicides.
PCT/GB2018/052071 2017-07-24 2018-07-23 Dérivés de pyrazole, d'isothiazole et d'isoxazole utiles en tant que fongicides agricoles WO2019020981A1 (fr)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
GBGB1711872.0A GB201711872D0 (en) 2017-07-24 2017-07-24 Agricultural chemicals
GB1711872.0 2017-07-24
GBGB1719097.6A GB201719097D0 (en) 2017-11-17 2017-11-17 Agricultural chemicals
GB1719097.6 2017-11-17
GB1807495.5 2018-05-08
GBGB1807495.5A GB201807495D0 (en) 2018-05-08 2018-05-08 Agricultural chemicals

Publications (1)

Publication Number Publication Date
WO2019020981A1 true WO2019020981A1 (fr) 2019-01-31

Family

ID=63077899

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/GB2018/052071 WO2019020981A1 (fr) 2017-07-24 2018-07-23 Dérivés de pyrazole, d'isothiazole et d'isoxazole utiles en tant que fongicides agricoles

Country Status (1)

Country Link
WO (1) WO2019020981A1 (fr)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2020051402A1 (fr) 2018-09-06 2020-03-12 Fmc Corporation Pyrazoles fongicides substitués par nitroanilino
WO2021183721A1 (fr) 2020-03-11 2021-09-16 Fmc Corporation Mélanges fongicides contenant des dérivés de pyrazole
US20220306609A1 (en) * 2021-03-23 2022-09-29 Nido Biosciences, Inc. Bicyclic compounds as androgen receptor modulators

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20050137201A1 (en) * 2003-09-04 2005-06-23 Alex Aronov Compositions useful as inhibitors of protein kinases
WO2009127612A1 (fr) * 2008-04-14 2009-10-22 Syngenta Participations Ag Nouveaux dérivés de pyrazole
WO2012031061A2 (fr) 2010-09-01 2012-03-08 E. I. Du Pont De Nemours And Company Pyrazoles fongicides et mélanges associés
WO2016055801A2 (fr) 2014-10-10 2016-04-14 Redag Crop Protection Ltd Produits chimiques agricoles

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20050137201A1 (en) * 2003-09-04 2005-06-23 Alex Aronov Compositions useful as inhibitors of protein kinases
WO2009127612A1 (fr) * 2008-04-14 2009-10-22 Syngenta Participations Ag Nouveaux dérivés de pyrazole
WO2012031061A2 (fr) 2010-09-01 2012-03-08 E. I. Du Pont De Nemours And Company Pyrazoles fongicides et mélanges associés
WO2016055801A2 (fr) 2014-10-10 2016-04-14 Redag Crop Protection Ltd Produits chimiques agricoles

Non-Patent Citations (10)

* Cited by examiner, † Cited by third party
Title
E. L. ELIEL; S. H. WILEN: "Stereochemistry of Organic Compounds", 1994, WILEY
FA CAREY; RJ SUNDBERG: "Reactions and Synthesis", 2001, KLUWER ACADEMIC/PLENUM PUBLICATIONS, article "Advanced Organic Chemistry"
J. JOULE: "Heterocyclic Chemistry", 2010, WILEY
MB SMITH; J. MARCH: "Reactions, Mechanisms and Structure", WILEY, article "March's Advanced Organic Chemistry"
RAPHAEL DUMEUNIER ET AL: "Synthesis of Tetrasubstituted Pyrazoles through Different Cyclization Strategies; Isosteres of Imidazole Fungicides", SYNLETT, vol. 24, no. 09, 18 April 2013 (2013-04-18), DE, pages 1150 - 1154, XP055503319, ISSN: 0936-5214, DOI: 10.1055/s-0033-1338433 *
RC LAROCK: "A Guide to Functional Group Transformations", 1999, WILEY-VCH, article "Comprehensive Organic Transformations"
RK MACKIE; DM SMITH: "Guidebook To Organic Synthesis", 1982, LONGMAN
S WARREN: "Designing Organic Syntheses", 1983, WILEY
S WARREN: "Organic Synthesis - The Disconnection Approach", 1982, WILEY
TW GREENE; PGM WUTS: "Protective Groups in Organic Synthesis", 1999, JOHN WILEY & SONS INC.

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2020051402A1 (fr) 2018-09-06 2020-03-12 Fmc Corporation Pyrazoles fongicides substitués par nitroanilino
CN112969688A (zh) * 2018-09-06 2021-06-15 Fmc公司 杀真菌的硝基苯胺取代的吡唑类化合物
US20210317087A1 (en) * 2018-09-06 2021-10-14 Fmc Corporation Fungicidal nitroanilino substituted pyrazoles
WO2021183721A1 (fr) 2020-03-11 2021-09-16 Fmc Corporation Mélanges fongicides contenant des dérivés de pyrazole
US20220306609A1 (en) * 2021-03-23 2022-09-29 Nido Biosciences, Inc. Bicyclic compounds as androgen receptor modulators

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