WO2016063289A3 - Compositions de comprimé pharmaceutique comprenant de la rifaximine - Google Patents

Compositions de comprimé pharmaceutique comprenant de la rifaximine Download PDF

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Publication number
WO2016063289A3
WO2016063289A3 PCT/IN2015/000312 IN2015000312W WO2016063289A3 WO 2016063289 A3 WO2016063289 A3 WO 2016063289A3 IN 2015000312 W IN2015000312 W IN 2015000312W WO 2016063289 A3 WO2016063289 A3 WO 2016063289A3
Authority
WO
WIPO (PCT)
Prior art keywords
rifaximin
pharmaceutical tablet
tablet compositions
compositions
pharmaceutical
Prior art date
Application number
PCT/IN2015/000312
Other languages
English (en)
Other versions
WO2016063289A2 (fr
Inventor
Kumar Mohan
Kumar Anil
Dash Bidhubhusan
Original Assignee
Strides Arcolab Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Strides Arcolab Limited filed Critical Strides Arcolab Limited
Publication of WO2016063289A2 publication Critical patent/WO2016063289A2/fr
Publication of WO2016063289A3 publication Critical patent/WO2016063289A3/fr

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La présente invention concerne une composition de comprimé pharmaceutique comprenant de la rifaximine et un procédé de préparation de celle-ci.
PCT/IN2015/000312 2014-10-22 2015-08-04 Compositions de comprimé pharmaceutique comprenant de la rifaximine WO2016063289A2 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN3379/MUM/2014 2014-10-22
IN3379MU2014 2014-10-22

Publications (2)

Publication Number Publication Date
WO2016063289A2 WO2016063289A2 (fr) 2016-04-28
WO2016063289A3 true WO2016063289A3 (fr) 2016-07-14

Family

ID=55761708

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/IN2015/000312 WO2016063289A2 (fr) 2014-10-22 2015-08-04 Compositions de comprimé pharmaceutique comprenant de la rifaximine

Country Status (1)

Country Link
WO (1) WO2016063289A2 (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2522895T3 (es) 2005-03-03 2014-11-19 Alfa Wassermann S.P.A. Nuevas formas polimorfas de rifaximina, procedimientos para su producción y uso de las mismas en preparados medicinales
ES2810010T3 (es) 2014-05-12 2021-03-08 Alfasigma Spa Preparación y uso de la forma cristalina tau de rifaximina solvatada con DEGME
EP4137132A1 (fr) * 2016-09-30 2023-02-22 Salix Pharmaceuticals, Inc. Formes de dispersion solides de rifaximine
WO2020128583A1 (fr) * 2018-12-19 2020-06-25 Friulchem S.P.A. Procédé de fabrication d'un comprimé de rifaximine et comprimé de rifaximine

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20090312357A1 (en) * 2006-09-22 2009-12-17 Cipla Limited Rifaximin
US20120245192A1 (en) * 2010-09-22 2012-09-27 Alfa Wassermann, S.P.A. Pharmaceutical formulations containing rifaximin, processes for their obtainment and method of treating intestinal disease
US20130004576A1 (en) * 2010-03-05 2013-01-03 Alfa Wassermann S.P.A. Rifaximin powder, process for preparing the same and controlled release compositions containing said rifaximin useful for obtaining a long-lasting effect
US20140012001A1 (en) * 2010-09-13 2014-01-09 Sequent Scientific Ltd. Novel polymorphic form of rifaximin and process for its preparation

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20090312357A1 (en) * 2006-09-22 2009-12-17 Cipla Limited Rifaximin
US20130004576A1 (en) * 2010-03-05 2013-01-03 Alfa Wassermann S.P.A. Rifaximin powder, process for preparing the same and controlled release compositions containing said rifaximin useful for obtaining a long-lasting effect
US20140012001A1 (en) * 2010-09-13 2014-01-09 Sequent Scientific Ltd. Novel polymorphic form of rifaximin and process for its preparation
US20120245192A1 (en) * 2010-09-22 2012-09-27 Alfa Wassermann, S.P.A. Pharmaceutical formulations containing rifaximin, processes for their obtainment and method of treating intestinal disease

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
VISCOUNT ET AL.: "Crystal founds of rifaximin and their effect on pharmaceutical properties", CRYST. ENG. COMM., vol. 10, July 2008 (2008-07-01), pages 1077 - 1078, XP009152378 *

Also Published As

Publication number Publication date
WO2016063289A2 (fr) 2016-04-28

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