WO2015092687A3 - Process for the purification of darapladib - Google Patents

Process for the purification of darapladib Download PDF

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Publication number
WO2015092687A3
WO2015092687A3 PCT/IB2014/066980 IB2014066980W WO2015092687A3 WO 2015092687 A3 WO2015092687 A3 WO 2015092687A3 IB 2014066980 W IB2014066980 W IB 2014066980W WO 2015092687 A3 WO2015092687 A3 WO 2015092687A3
Authority
WO
WIPO (PCT)
Prior art keywords
darapladib
purification
provides
present
Prior art date
Application number
PCT/IB2014/066980
Other languages
French (fr)
Other versions
WO2015092687A2 (en
Inventor
Md Abul Kalam AZAD
Amit K. Jain
Gyanendra Pandey
Kaptan Singh
Mohan Prasad
Original Assignee
Ranbaxy Laboratories Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ranbaxy Laboratories Limited filed Critical Ranbaxy Laboratories Limited
Publication of WO2015092687A2 publication Critical patent/WO2015092687A2/en
Publication of WO2015092687A3 publication Critical patent/WO2015092687A3/en

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Ladders (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

The present invention provides a process for the purification of darapladib.
PCT/IB2014/066980 2013-12-17 2014-12-16 Process for the purification of darapladib WO2015092687A2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN3675DE2013 2013-12-17
IN3675/DEL/2013 2013-12-17

Publications (2)

Publication Number Publication Date
WO2015092687A2 WO2015092687A2 (en) 2015-06-25
WO2015092687A3 true WO2015092687A3 (en) 2015-08-13

Family

ID=53264685

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/IB2014/066980 WO2015092687A2 (en) 2013-12-17 2014-12-16 Process for the purification of darapladib

Country Status (1)

Country Link
WO (1) WO2015092687A2 (en)

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003016287A2 (en) * 2001-08-14 2003-02-27 Smithkline Beecham P.L.C. Process for preparing 1-(carboxymethyl)- and 1-(aminocarbonyl)- pyrimidin-4-one derivatives
WO2011146494A1 (en) * 2010-05-17 2011-11-24 Glaxo Group Limited Novel processes

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2400554C (en) 2000-02-16 2009-04-07 Smithkline Beecham P.L.C. Pyrimidine-4-one derivatives as ldl-pla2 inhibitors

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003016287A2 (en) * 2001-08-14 2003-02-27 Smithkline Beecham P.L.C. Process for preparing 1-(carboxymethyl)- and 1-(aminocarbonyl)- pyrimidin-4-one derivatives
WO2011146494A1 (en) * 2010-05-17 2011-11-24 Glaxo Group Limited Novel processes

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
VOGEL A I: "VOGEL'S TEXTBOOK OF PRACTICAL ORGANIC CHEMISTRY", VOGEL'S TEXTBOOK OF PRACTICAL ORGANIC CHEMISTRY, XX, XX, 1 January 1989 (1989-01-01), pages 135 - 139, XP003004371 *

Also Published As

Publication number Publication date
WO2015092687A2 (en) 2015-06-25

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