WO2013109213A3 - Pharmaceutical formulations comprising tiotropium - Google Patents

Pharmaceutical formulations comprising tiotropium Download PDF

Info

Publication number
WO2013109213A3
WO2013109213A3 PCT/TR2013/000025 TR2013000025W WO2013109213A3 WO 2013109213 A3 WO2013109213 A3 WO 2013109213A3 TR 2013000025 W TR2013000025 W TR 2013000025W WO 2013109213 A3 WO2013109213 A3 WO 2013109213A3
Authority
WO
WIPO (PCT)
Prior art keywords
tiotropium
pharmaceutical formulations
order
dry powder
relates
Prior art date
Application number
PCT/TR2013/000025
Other languages
French (fr)
Other versions
WO2013109213A2 (en
Inventor
Mahmut Bilgic
Original Assignee
Mahmut Bilgic
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mahmut Bilgic filed Critical Mahmut Bilgic
Publication of WO2013109213A2 publication Critical patent/WO2013109213A2/en
Publication of WO2013109213A3 publication Critical patent/WO2013109213A3/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/007Pulmonary tract; Aromatherapy
    • A61K9/0073Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/0075Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/439Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Otolaryngology (AREA)
  • Pulmonology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

The present invention relates to pharmaceutical formulations in dry powder comprising tiotropium in order to be used in respiratory tract diseases.
PCT/TR2013/000025 2012-01-16 2013-01-16 Pharmaceutical formulations comprising tiotropium WO2013109213A2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
TR201200492 2012-01-16
TR2012/00492 2012-01-16

Publications (2)

Publication Number Publication Date
WO2013109213A2 WO2013109213A2 (en) 2013-07-25
WO2013109213A3 true WO2013109213A3 (en) 2013-09-06

Family

ID=48237229

Family Applications (2)

Application Number Title Priority Date Filing Date
PCT/TR2013/000025 WO2013109213A2 (en) 2012-01-16 2013-01-16 Pharmaceutical formulations comprising tiotropium
PCT/TR2013/000028 WO2013109216A2 (en) 2012-01-16 2013-01-16 Preparation of dry powder formulations comprising tiotropium

Family Applications After (1)

Application Number Title Priority Date Filing Date
PCT/TR2013/000028 WO2013109216A2 (en) 2012-01-16 2013-01-16 Preparation of dry powder formulations comprising tiotropium

Country Status (2)

Country Link
EP (1) EP2804591A2 (en)
WO (2) WO2013109213A2 (en)

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20040136919A1 (en) * 2002-11-28 2004-07-15 Boehringer Ingelheim Pharma Gmbh & Co. Kg Tiotropium containing powder formulation for inhalation
EP2172190A1 (en) * 2008-10-02 2010-04-07 Laboratorios Liconsa, S.A. Inhalable particles comprising tiotropium
WO2011093819A2 (en) * 2010-01-28 2011-08-04 Mahmut Bilgic New combination comprising tiotropium
WO2011093820A2 (en) * 2010-01-28 2011-08-04 Mahmut Bilgic A pharmaceutical combination comprising tiotropium

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3931041C2 (en) 1989-09-16 2000-04-06 Boehringer Ingelheim Kg Esters of thienyl carboxylic acids with amino alcohols, their quaternization products, processes for their preparation and medicaments containing them
WO2011152804A2 (en) * 2010-06-03 2011-12-08 Mahmut Bilgic Process for dry powder formulations

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20040136919A1 (en) * 2002-11-28 2004-07-15 Boehringer Ingelheim Pharma Gmbh & Co. Kg Tiotropium containing powder formulation for inhalation
EP2172190A1 (en) * 2008-10-02 2010-04-07 Laboratorios Liconsa, S.A. Inhalable particles comprising tiotropium
WO2011093819A2 (en) * 2010-01-28 2011-08-04 Mahmut Bilgic New combination comprising tiotropium
WO2011093820A2 (en) * 2010-01-28 2011-08-04 Mahmut Bilgic A pharmaceutical combination comprising tiotropium

Also Published As

Publication number Publication date
WO2013109213A2 (en) 2013-07-25
EP2804591A2 (en) 2014-11-26
WO2013109216A2 (en) 2013-07-25
WO2013109216A3 (en) 2014-04-17

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