WO2012026907A3 - Cefpodoxime proxetil formulations - Google Patents

Cefpodoxime proxetil formulations Download PDF

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Publication number
WO2012026907A3
WO2012026907A3 PCT/TR2011/000200 TR2011000200W WO2012026907A3 WO 2012026907 A3 WO2012026907 A3 WO 2012026907A3 TR 2011000200 W TR2011000200 W TR 2011000200W WO 2012026907 A3 WO2012026907 A3 WO 2012026907A3
Authority
WO
WIPO (PCT)
Prior art keywords
formulations
cefpodoxime proxetil
proxetil
cefpodoxime
relates
Prior art date
Application number
PCT/TR2011/000200
Other languages
French (fr)
Other versions
WO2012026907A2 (en
Inventor
Mahmut Bilgic
Original Assignee
Mahmut Bilgic
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mahmut Bilgic filed Critical Mahmut Bilgic
Priority to EP11782258.5A priority Critical patent/EP2608776A2/en
Publication of WO2012026907A2 publication Critical patent/WO2012026907A2/en
Publication of WO2012026907A3 publication Critical patent/WO2012026907A3/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0087Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/424Oxazoles condensed with heterocyclic ring systems, e.g. clavulanic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • A61K31/546Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine containing further heterocyclic rings, e.g. cephalothin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/143Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Abstract

The present invention relates to pharmaceutical formulations comprising cefpodoxime proxetil.
PCT/TR2011/000200 2010-08-25 2011-08-24 Cefpodoxime proxetil formulations WO2012026907A2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
EP11782258.5A EP2608776A2 (en) 2010-08-25 2011-08-24 Cefpodoxime proxetil formulations

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
TR2010/07106 2010-08-25
TR2010/07106A TR201007106A1 (en) 2010-08-25 2010-08-25 Cefpodoxime proxetil formulations.

Publications (2)

Publication Number Publication Date
WO2012026907A2 WO2012026907A2 (en) 2012-03-01
WO2012026907A3 true WO2012026907A3 (en) 2012-09-13

Family

ID=44947169

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/TR2011/000200 WO2012026907A2 (en) 2010-08-25 2011-08-24 Cefpodoxime proxetil formulations

Country Status (3)

Country Link
EP (1) EP2608776A2 (en)
TR (1) TR201007106A1 (en)
WO (1) WO2012026907A2 (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103142506B (en) * 2013-04-03 2015-02-25 天津医药集团津康制药有限公司 Cefpodoxime proxetil granules and preparation method thereof
CN103230367B (en) * 2013-05-07 2014-11-12 山东罗欣药业集团股份有限公司 Cefpodoxime proxetil composition dry suspension and preparation method thereof
CN107693491B (en) * 2017-04-20 2020-06-30 广东金城金素制药有限公司 Pharmaceutical composition and preparation for children
CN108815130A (en) * 2018-08-27 2018-11-16 邓倩 A kind of Cefpodoxime Proxetil tablet and its production technology

Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002067943A1 (en) * 2001-02-27 2002-09-06 Ranbaxy Laboratories Limited Oral pharmaceutical composition of cefpodoxime proxetil
WO2004004737A1 (en) * 2002-07-08 2004-01-15 Sankyo Company, Limited Cephalosporin preparation for oral use
WO2004006917A1 (en) * 2002-07-16 2004-01-22 Ranbaxy Laboratories Limited Dispersible tablets for oral administration
WO2007017895A2 (en) * 2005-05-05 2007-02-15 Lupin Limited Stabilized oral pharmaceutical compositions of cephalosporins
WO2011129792A1 (en) * 2010-04-13 2011-10-20 Mahmut Bilgic Water dispersible formulations comprising cefpodoxime proxetil

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4486425A (en) 1980-09-30 1984-12-04 Sankyo Company Limited 7-[2-(2-Aminothiazol-4-yl)-2-(syn)-methoxyiminoacetamido]-3-methoxymethyl-3-cephem-4-carboxylates

Patent Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002067943A1 (en) * 2001-02-27 2002-09-06 Ranbaxy Laboratories Limited Oral pharmaceutical composition of cefpodoxime proxetil
WO2004004737A1 (en) * 2002-07-08 2004-01-15 Sankyo Company, Limited Cephalosporin preparation for oral use
WO2004006917A1 (en) * 2002-07-16 2004-01-22 Ranbaxy Laboratories Limited Dispersible tablets for oral administration
WO2007017895A2 (en) * 2005-05-05 2007-02-15 Lupin Limited Stabilized oral pharmaceutical compositions of cephalosporins
WO2011129792A1 (en) * 2010-04-13 2011-10-20 Mahmut Bilgic Water dispersible formulations comprising cefpodoxime proxetil

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
DATABASE WPI Week 200416, Derwent World Patents Index; AN 2004-169094, XP002676813 *

Also Published As

Publication number Publication date
EP2608776A2 (en) 2013-07-03
WO2012026907A2 (en) 2012-03-01
TR201007106A1 (en) 2012-03-21

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