WO2011083112A3 - Solid oral dosage form containing olmesartan medoxomil - Google Patents

Solid oral dosage form containing olmesartan medoxomil Download PDF

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Publication number
WO2011083112A3
WO2011083112A3 PCT/EP2011/050061 EP2011050061W WO2011083112A3 WO 2011083112 A3 WO2011083112 A3 WO 2011083112A3 EP 2011050061 W EP2011050061 W EP 2011050061W WO 2011083112 A3 WO2011083112 A3 WO 2011083112A3
Authority
WO
WIPO (PCT)
Prior art keywords
dosage form
oral dosage
solid oral
olmesartan medoxomil
form containing
Prior art date
Application number
PCT/EP2011/050061
Other languages
French (fr)
Other versions
WO2011083112A2 (en
Inventor
Ganesh V. Gat
Jawed Hussain
Parshwakumar V. Kalyankar
Original Assignee
Ratiopharm Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ratiopharm Gmbh filed Critical Ratiopharm Gmbh
Priority to CA2785920A priority Critical patent/CA2785920A1/en
Priority to EP11701630.3A priority patent/EP2521540A2/en
Publication of WO2011083112A2 publication Critical patent/WO2011083112A2/en
Publication of WO2011083112A3 publication Critical patent/WO2011083112A3/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2031Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41781,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/44221,4-Dihydropyridines, e.g. nifedipine, nicardipine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/549Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame having two or more nitrogen atoms in the same ring, e.g. hydrochlorothiazide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

The present invention provides a solid oral dosage form comprising olmesartan medoxomil and polyethylene glycol having a molecular weight of about 1,000 - 10,000.
PCT/EP2011/050061 2010-01-05 2011-01-04 Solid oral dosage form containing olmesartan medoxomil WO2011083112A2 (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
CA2785920A CA2785920A1 (en) 2010-01-05 2011-01-04 Solid oral dosage form containing olmesartan medoxomil
EP11701630.3A EP2521540A2 (en) 2010-01-05 2011-01-04 Solid oral dosage form containing olmesartan medoxomil

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN26DE2010 2010-01-05
IN26/DEL/2010 2010-01-05

Publications (2)

Publication Number Publication Date
WO2011083112A2 WO2011083112A2 (en) 2011-07-14
WO2011083112A3 true WO2011083112A3 (en) 2011-12-29

Family

ID=43795169

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/EP2011/050061 WO2011083112A2 (en) 2010-01-05 2011-01-04 Solid oral dosage form containing olmesartan medoxomil

Country Status (3)

Country Link
EP (1) EP2521540A2 (en)
CA (1) CA2785920A1 (en)
WO (1) WO2011083112A2 (en)

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20040198789A1 (en) * 2003-02-28 2004-10-07 Recordati Ireland Limited Lercanidipine/ARB/diuretic therapeutic combinations
CN101066264A (en) * 2007-06-12 2007-11-07 杨喜鸿 Solid olmesartan medoxmil dispersion and its prepn and medicinal application
CN101313907A (en) * 2008-07-07 2008-12-03 北京润德康医药技术有限公司 Medicament composition for treating hyperpiesis
WO2008149338A2 (en) * 2007-06-06 2008-12-11 Dexcel Ltd. Process for forming solid oral dosage forms of angiotensin ii receptor antagonists

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2229000C (en) 1991-02-21 2002-04-09 Sankyo Company, Limited 1-biphenylimidazole derivatives, their preparation and their therapeutic use
US20060281800A1 (en) 2005-04-12 2006-12-14 Glenmark Pharmaceuticals Limited Polymorphic form of olmesartan and process for its preparation
EP1910343B1 (en) 2005-07-29 2014-10-29 Krka Process for the preparation of olmesartan medoxomil
EP1801111B1 (en) 2005-12-20 2014-07-16 LEK Pharmaceuticals d.d. Novel polymorph forms of olmesartan medoxomil
EP1891952B1 (en) 2006-05-04 2011-10-05 LEK Pharmaceuticals d.d. Pharmaceutical composition of olmesartan medoxomil
GB0710905D0 (en) 2007-06-07 2007-07-18 Generics Uk Ltd Amorphous olmesartan medoxomil

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20040198789A1 (en) * 2003-02-28 2004-10-07 Recordati Ireland Limited Lercanidipine/ARB/diuretic therapeutic combinations
WO2008149338A2 (en) * 2007-06-06 2008-12-11 Dexcel Ltd. Process for forming solid oral dosage forms of angiotensin ii receptor antagonists
CN101066264A (en) * 2007-06-12 2007-11-07 杨喜鸿 Solid olmesartan medoxmil dispersion and its prepn and medicinal application
CN101313907A (en) * 2008-07-07 2008-12-03 北京润德康医药技术有限公司 Medicament composition for treating hyperpiesis

Also Published As

Publication number Publication date
CA2785920A1 (en) 2011-07-14
WO2011083112A2 (en) 2011-07-14
EP2521540A2 (en) 2012-11-14

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