WO2009111623A3 - Tartrate de varénicline amorphe - Google Patents
Tartrate de varénicline amorphe Download PDFInfo
- Publication number
- WO2009111623A3 WO2009111623A3 PCT/US2009/036157 US2009036157W WO2009111623A3 WO 2009111623 A3 WO2009111623 A3 WO 2009111623A3 US 2009036157 W US2009036157 W US 2009036157W WO 2009111623 A3 WO2009111623 A3 WO 2009111623A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- varenicline tartrate
- amorphous
- amorphous varenicline
- tartrate
- processes
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/08—Bridged systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Abstract
L’invention concerne le tartrate de varénicline amorphe, des dispersions solides amorphes de tartrate de varénicline et un excipient pharmaceutique, et leurs procédés de préparation.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP09716470A EP2262780A4 (fr) | 2008-03-06 | 2009-03-05 | Tartrate de varénicline amorphe |
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN571CH2008 | 2008-03-06 | ||
IN571/CHE/2008 | 2008-03-06 | ||
US7384408P | 2008-06-19 | 2008-06-19 | |
US61/073,844 | 2008-06-19 |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2009111623A2 WO2009111623A2 (fr) | 2009-09-11 |
WO2009111623A3 true WO2009111623A3 (fr) | 2009-12-10 |
Family
ID=41056650
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/US2009/036157 WO2009111623A2 (fr) | 2008-03-06 | 2009-03-05 | Tartrate de varénicline amorphe |
Country Status (2)
Country | Link |
---|---|
EP (1) | EP2262780A4 (fr) |
WO (1) | WO2009111623A2 (fr) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2801842A1 (fr) | 2009-06-10 | 2010-12-16 | Actavis Group Ptc Ehf | Co-precipites amorphes de tartrate de varenicline |
US20120004239A1 (en) | 2010-06-11 | 2012-01-05 | Medichem, S.A. | Process for Preparing Quinoxaline Derivatives |
WO2013160916A1 (fr) * | 2012-04-25 | 2013-10-31 | Hetero Research Foundation | Dispersion solide de malate de sunitinib |
CN104478803A (zh) * | 2014-12-19 | 2015-04-01 | 连云港恒运医药科技有限公司 | 伐尼克兰中间体及其硝基还原杂质的制备方法 |
US11266658B2 (en) * | 2017-03-03 | 2022-03-08 | Ctc Bio, Inc. | Preparation, comprising inclusion complex of varenicline or pharmaceutically acceptable salt thereof, for oral administration |
US11602537B2 (en) | 2022-03-11 | 2023-03-14 | Par Pharmaceutical, Inc. | Varenicline compound and process of manufacture thereof |
Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2002092089A1 (fr) * | 2001-05-14 | 2002-11-21 | Pfizer Products Inc. | Sels de tartrate de 5,8,14-triazatetracyclo[10.3.1.02,11.04,9]-hexadeca-2(11),3,5,7,9-pentaene |
US6558435B2 (en) * | 2000-05-26 | 2003-05-06 | Pfizer, Inc. | Reactive crystallization method to improve particle size |
WO2007012963A1 (fr) * | 2005-07-26 | 2007-02-01 | Pfizer Products Inc. | Système transdermique pour la varenicline |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5683720A (en) * | 1994-10-28 | 1997-11-04 | Fuisz Technologies Ltd. | Liquiflash particles and method of making same |
JP2008516942A (ja) * | 2004-10-15 | 2008-05-22 | ファイザー・プロダクツ・インク | バレニクリンの鼻腔内、バッカル、舌下および肺送達のための組成物および方法 |
EP1843769A1 (fr) * | 2005-01-07 | 2007-10-17 | Pfizer Products Incorporated | Formes posologiques a desintegration rapide de 5,8,14-triazatetracyclo[10.3.1.02,11.04,9]-hexadeca-2(11),3,5,7,9-pentaene |
-
2009
- 2009-03-05 WO PCT/US2009/036157 patent/WO2009111623A2/fr active Application Filing
- 2009-03-05 EP EP09716470A patent/EP2262780A4/fr not_active Withdrawn
Patent Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6558435B2 (en) * | 2000-05-26 | 2003-05-06 | Pfizer, Inc. | Reactive crystallization method to improve particle size |
WO2002092089A1 (fr) * | 2001-05-14 | 2002-11-21 | Pfizer Products Inc. | Sels de tartrate de 5,8,14-triazatetracyclo[10.3.1.02,11.04,9]-hexadeca-2(11),3,5,7,9-pentaene |
WO2007012963A1 (fr) * | 2005-07-26 | 2007-02-01 | Pfizer Products Inc. | Système transdermique pour la varenicline |
Non-Patent Citations (2)
Title |
---|
NIAURA, RAYMOND ET AL.: "Varenicline", NATURE REVIEWS DRUG DISCOVERY, vol. 5, no. 7, 2006, pages 537 - 538, XP008138247 * |
See also references of EP2262780A4 * |
Also Published As
Publication number | Publication date |
---|---|
EP2262780A2 (fr) | 2010-12-22 |
EP2262780A4 (fr) | 2012-01-25 |
WO2009111623A2 (fr) | 2009-09-11 |
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