WO2009012039A3 - Polymorphes cristallins - Google Patents
Polymorphes cristallins Download PDFInfo
- Publication number
- WO2009012039A3 WO2009012039A3 PCT/US2008/068558 US2008068558W WO2009012039A3 WO 2009012039 A3 WO2009012039 A3 WO 2009012039A3 US 2008068558 W US2008068558 W US 2008068558W WO 2009012039 A3 WO2009012039 A3 WO 2009012039A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- crystalline polymorphs
- present
- compositions
- provides
- ethoxycarbonylprop
- Prior art date
Links
- 125000002941 2-furyl group Chemical group O1C([*])=C([H])C([H])=C1[H] 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
- C07F9/65586—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system at least one of the hetero rings does not contain nitrogen as ring hetero atom
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La présente invention concerne des formes cristallines de 2-amino-5-(2,2~ diméthylpropionyl)-4-{[5-(N,N'-(2-éthoxycarbonylprop-2-yl)phosphonamido] furan-2-yl}thiazole et des compositions en contenant y compris des compositions pharmaceutiques. La présente invention concerne également des procédés d'utilisation et des procédés de fabrication de telles formes cristallines.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US94968107P | 2007-07-13 | 2007-07-13 | |
US60/949,681 | 2007-07-13 |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2009012039A2 WO2009012039A2 (fr) | 2009-01-22 |
WO2009012039A3 true WO2009012039A3 (fr) | 2009-03-19 |
Family
ID=40260294
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/US2008/068558 WO2009012039A2 (fr) | 2007-07-13 | 2008-06-27 | Polymorphes cristallins |
Country Status (1)
Country | Link |
---|---|
WO (1) | WO2009012039A2 (fr) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2011107494A1 (fr) | 2010-03-03 | 2011-09-09 | Sanofi | Nouveaux dérivés aromatiques de glycoside, médicaments contenants ces composés, et leur utilisation |
US8530413B2 (en) | 2010-06-21 | 2013-09-10 | Sanofi | Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments |
TW201215388A (en) | 2010-07-05 | 2012-04-16 | Sanofi Sa | (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments |
TW201221505A (en) | 2010-07-05 | 2012-06-01 | Sanofi Sa | Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament |
TW201215387A (en) | 2010-07-05 | 2012-04-16 | Sanofi Aventis | Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament |
WO2013037390A1 (fr) | 2011-09-12 | 2013-03-21 | Sanofi | Dérivés amides d'acide 6-(4-hydroxyphényl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylique en tant qu'inhibiteurs de kinase |
WO2013045413A1 (fr) | 2011-09-27 | 2013-04-04 | Sanofi | Dérivés d'amide d'acide 6-(4-hydroxyphényl)-3-alkyl-1h-pyrazolo[3,4-b] pyridine-4-carboxylique utilisés comme inhibiteurs de kinase |
Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6756360B1 (en) * | 1998-12-24 | 2004-06-29 | Metabasis Therapeutics, Inc. | Combination of FBPase inhibitors and insulin sensitizers for the treatment of diabetes |
WO2006023515A2 (fr) * | 2004-08-18 | 2006-03-02 | Metabasis Therapeutics, Inc. | Nouveaux inhibiteurs thiazole de la fructose 1,6-bisphosphatase |
-
2008
- 2008-06-27 WO PCT/US2008/068558 patent/WO2009012039A2/fr active Application Filing
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6756360B1 (en) * | 1998-12-24 | 2004-06-29 | Metabasis Therapeutics, Inc. | Combination of FBPase inhibitors and insulin sensitizers for the treatment of diabetes |
WO2006023515A2 (fr) * | 2004-08-18 | 2006-03-02 | Metabasis Therapeutics, Inc. | Nouveaux inhibiteurs thiazole de la fructose 1,6-bisphosphatase |
Also Published As
Publication number | Publication date |
---|---|
WO2009012039A2 (fr) | 2009-01-22 |
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