WO2007123855A3 - Pyrazolines for controlling invertebrate pests - Google Patents

Pyrazolines for controlling invertebrate pests Download PDF

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Publication number
WO2007123855A3
WO2007123855A3 PCT/US2007/009184 US2007009184W WO2007123855A3 WO 2007123855 A3 WO2007123855 A3 WO 2007123855A3 US 2007009184 W US2007009184 W US 2007009184W WO 2007123855 A3 WO2007123855 A3 WO 2007123855A3
Authority
WO
WIPO (PCT)
Prior art keywords
optionally substituted
pyrazolines
nr12r13
alkylcycloalkyl
cycloalkylalkyl
Prior art date
Application number
PCT/US2007/009184
Other languages
French (fr)
Other versions
WO2007123855B1 (en
WO2007123855A2 (en
Inventor
Stephen Frederick Mccann
Brenton Todd Smith
Original Assignee
Du Pont
Stephen Frederick Mccann
Brenton Todd Smith
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Du Pont, Stephen Frederick Mccann, Brenton Todd Smith filed Critical Du Pont
Priority to BRPI0710403-0A priority Critical patent/BRPI0710403A2/en
Priority to AU2007240954A priority patent/AU2007240954A1/en
Priority to MX2008013307A priority patent/MX2008013307A/en
Publication of WO2007123855A2 publication Critical patent/WO2007123855A2/en
Publication of WO2007123855A3 publication Critical patent/WO2007123855A3/en
Publication of WO2007123855B1 publication Critical patent/WO2007123855B1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/06—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings

Abstract

Disclosed are compounds of Formula 1, including all geometric and stereoisomers N-oxides, and salts thereof; wherein Z is N or CR2; R1 is cyano; or C1-C6 alkyl, C2-C6 alkenyl, C2-C6 alkynyl, C3-C6 cycloalkyl, C4-C7 alkylcycloalkyl or C4-C7 cycloalkylalkyl, each optionally substituted with one or more substituents independently selected from R17; R3 is H, cyano or -CHO; or C1-C6 alkyl, C2-C6 alkenyl, C2-C6 alkynyl, C3-C6 cycloalkyl, C4-C7 alkylcycloalkyl, C4-C7 cycloalkylalkyl, phenyl, C2-C6 alkylcarbonyl, C2-C6 alkoxycarbonyl, C2-C6 alkylaminocarbonyl or C3-C9 dialkylaminocarbonyl, each optionally substituted with one or more substituents independently selected from R18; Q is a 5- or 6-membered saturated or unsaturated heterocycle optionally substituted; or Q is C(O)NR12R13, C(S)NR12R13, S(O)2NR14R15 or R16. Also disclosed are compositions containing the compounds of Formula 1 and methods for controlling an invertebrate pest comprising contacting the invertebrate pest or its environment with a biologically effective amount of a compound or a composition of the invention.
PCT/US2007/009184 2006-04-20 2007-04-13 Pyrazolines for controlling invertebrate pests WO2007123855A2 (en)

Priority Applications (3)

Application Number Priority Date Filing Date Title
BRPI0710403-0A BRPI0710403A2 (en) 2006-04-20 2007-04-13 compound composition, control composition, spraying, bait, trap device, control methods, protection methods, treated seed, protective composition
AU2007240954A AU2007240954A1 (en) 2006-04-20 2007-04-13 Pyrazolines for controlling invertebrate pests
MX2008013307A MX2008013307A (en) 2006-04-20 2007-04-13 Pyrazolines for controlling invertebrate pests.

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US79357606P 2006-04-20 2006-04-20
US60/793,576 2006-04-20

Publications (3)

Publication Number Publication Date
WO2007123855A2 WO2007123855A2 (en) 2007-11-01
WO2007123855A3 true WO2007123855A3 (en) 2008-01-10
WO2007123855B1 WO2007123855B1 (en) 2008-02-21

Family

ID=38542963

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/US2007/009184 WO2007123855A2 (en) 2006-04-20 2007-04-13 Pyrazolines for controlling invertebrate pests

Country Status (5)

Country Link
KR (1) KR20090005201A (en)
AU (1) AU2007240954A1 (en)
BR (1) BRPI0710403A2 (en)
MX (1) MX2008013307A (en)
WO (1) WO2007123855A2 (en)

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CN102858161A (en) * 2010-04-27 2013-01-02 先正达参股股份有限公司 Methods of controlling neonicotinoid resistant aphids
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PL2811998T3 (en) 2012-02-06 2019-05-31 Merial Inc Parasiticidal oral veterinary compositions comprising systemically acting active agents, methods and uses thereof
JO3626B1 (en) 2012-02-23 2020-08-27 Merial Inc Topical compositions comprising fipronil and permethrin and methods of use
US20150057321A1 (en) 2012-04-04 2015-02-26 Intervet Inc. Soft chewable pharmaceutical products
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CN103355279B (en) * 2013-07-19 2014-11-26 江苏省农业科学院 Aphid extinguishing liquor and electrothermal aphid extinguishing method employing same for preventing and controlling aphid of facility crops
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Also Published As

Publication number Publication date
WO2007123855B1 (en) 2008-02-21
WO2007123855A2 (en) 2007-11-01
KR20090005201A (en) 2009-01-12
BRPI0710403A2 (en) 2011-08-09
MX2008013307A (en) 2008-10-27
AU2007240954A1 (en) 2007-11-01

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