WO2007103711A3 - Polymorphic forms of rimonabant - Google Patents

Polymorphic forms of rimonabant Download PDF

Info

Publication number
WO2007103711A3
WO2007103711A3 PCT/US2007/063042 US2007063042W WO2007103711A3 WO 2007103711 A3 WO2007103711 A3 WO 2007103711A3 US 2007063042 W US2007063042 W US 2007063042W WO 2007103711 A3 WO2007103711 A3 WO 2007103711A3
Authority
WO
WIPO (PCT)
Prior art keywords
rimonabant
polymorphic forms
amorphous
vi
iv
Prior art date
Application number
PCT/US2007/063042
Other languages
French (fr)
Other versions
WO2007103711A2 (en
Inventor
Ramulu Akula
Anuradha Bhimireddy
Vijayabhaskar Bolugoddu
Purandhar Kolkonda
Vijaya Kumar Kotagiri
Sashikanth Suthrapu
Original Assignee
Ramulu Akula
Anuradha Bhimireddy
Vijayabhaskar Bolugoddu
Purandhar Kolkonda
Vijaya Kumar Kotagiri
Reddys Lab Inc Dr
Reddys Lab Ltd Dr
Sashikanth Suthrapu
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to IN358CH2006 priority Critical
Priority to IN358/CHE/2006 priority
Priority to IN611CH2006 priority
Priority to IN611/CHE/2006 priority
Priority to US60/805,679 priority
Priority to US80567906P priority
Priority to US80778506P priority
Priority to US60/807,785 priority
Application filed by Ramulu Akula, Anuradha Bhimireddy, Vijayabhaskar Bolugoddu, Purandhar Kolkonda, Vijaya Kumar Kotagiri, Reddys Lab Inc Dr, Reddys Lab Ltd Dr, Sashikanth Suthrapu filed Critical Ramulu Akula
Publication of WO2007103711A2 publication Critical patent/WO2007103711A2/en
Publication of WO2007103711A3 publication Critical patent/WO2007103711A3/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Abstract

Polymorphic crystalline Forms III, IV, V, and VI of rimonabant, amorphous rimonabant, and amorphous rimonabant in an intimate dispersion with a pharmaceutically acceptable carrier.
PCT/US2007/063042 2006-03-01 2007-03-01 Polymorphic forms of rimonabant WO2007103711A2 (en)

Priority Applications (8)

Application Number Priority Date Filing Date Title
IN358CH2006 2006-03-01
IN358/CHE/2006 2006-03-01
IN611CH2006 2006-04-04
IN611/CHE/2006 2006-04-04
US80567906P true 2006-06-23 2006-06-23
US60/805,679 2006-06-23
US80778506P true 2006-07-19 2006-07-19
US60/807,785 2006-07-19

Publications (2)

Publication Number Publication Date
WO2007103711A2 WO2007103711A2 (en) 2007-09-13
WO2007103711A3 true WO2007103711A3 (en) 2009-04-02

Family

ID=38475673

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/US2007/063042 WO2007103711A2 (en) 2006-03-01 2007-03-01 Polymorphic forms of rimonabant

Country Status (1)

Country Link
WO (1) WO2007103711A2 (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20100076022A1 (en) * 2006-09-01 2010-03-25 Hetero Drugs Limited Novel polymorphs of rimonabant
WO2008056377A2 (en) * 2006-11-06 2008-05-15 Cadila Healthcare Limited Polymorphic forms of rimonabant
CZ300115B6 (en) * 2006-12-01 2009-02-11 Zentiva, A. S. Process for preparing N-piperidino-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxamide (rimonabant)
WO2008064615A2 (en) * 2006-12-01 2008-06-05 Zentiva, A.S. Crystalline and amorphous forms of rimonabant and processes for obtaining them
US20080182877A1 (en) * 2007-01-05 2008-07-31 Westheim Raymond J H Rimonabant forms and methods of making the same
WO2008088900A2 (en) * 2007-01-18 2008-07-24 Teva Pharmaceutical Industries Ltd. Polymorphic forms of rimonabant base and processes for preparation thereof
FR2913018A1 (en) * 2007-02-23 2008-08-29 Sanofi Aventis Sa New pyrazol-3-carboxamide derivative in amorphous form comprising surinabant and rimonabant form, useful for preparing amorphous solid solution

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6284277B1 (en) * 1995-11-03 2001-09-04 Sanofi-Synthelabo Stable freeze-dried pharmaceutical formulation
US20050202092A1 (en) * 2002-07-18 2005-09-15 Skantze Tommy U. Process for the preparation of crystalline nano-particle dispersions
WO2006087732A1 (en) * 2005-01-06 2006-08-24 Cadila Healthcare Limited An amorphous and three crystalline forms of rimonabant hydrochloride
US20080070949A1 (en) * 2006-09-19 2008-03-20 Cipla Limited Polymorphs of rimonabant

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6284277B1 (en) * 1995-11-03 2001-09-04 Sanofi-Synthelabo Stable freeze-dried pharmaceutical formulation
US20050202092A1 (en) * 2002-07-18 2005-09-15 Skantze Tommy U. Process for the preparation of crystalline nano-particle dispersions
WO2006087732A1 (en) * 2005-01-06 2006-08-24 Cadila Healthcare Limited An amorphous and three crystalline forms of rimonabant hydrochloride
US20080070949A1 (en) * 2006-09-19 2008-03-20 Cipla Limited Polymorphs of rimonabant

Also Published As

Publication number Publication date
WO2007103711A2 (en) 2007-09-13

Similar Documents

Publication Publication Date Title
EP1890746B8 (en) Injection device
EP2461418B8 (en) Battery module, and method for cooling a battery module
EP1720485B8 (en) Highly crystalline cross-linked oxidation-resistant polyethylene
EP2409707B8 (en) Polymer-based sustained release device
EP2046246B8 (en) Multi-planar taper lock screw
EP1970084B8 (en) Insertion device for an insertion head, in particular for an infusion set
EP1956806B8 (en) Method and device for communication channel selection
EP1773933A4 (en) Fuel supplies for fuel cells
WO2007121252A3 (en) Tandem photovoltaic cells
PL2364988T3 (en) Stable NAD/NADH derivatives
EP2163171A4 (en) Vehicle seat device
WO2007007140A3 (en) Communication mehtod
EP2058865A4 (en) Method for forming semiconductor substrate and electrode, and method for manufacturing solar battery
AU2009292594A8 (en) Solar cell module, installation structure for solar cell module, and installation method for solar cell module
EP1755712B8 (en) Injection device
EP1928488A4 (en) Oligodendrocyte precursor cell proliferation regulated by prolactin
EP1714381B8 (en) Power amplifier with stabilising network
EP1947704A4 (en) Cis-type thin-film solar battery module and process for producing the same
EP2234172A4 (en) Solar cell module and method for manufacturing the same
EP1866178B8 (en) Seat mount with integrated adjustment
EP2264779A4 (en) Solar cell, solar cell string and solar cell module
AU2009286380A8 (en) Dioxa-bicyclo[3.2.1.]octane-2,3,4-triol derivatives
EP1725536B8 (en) Imidazoline derivatives having cb1-antagonistic activity
EP1973719A4 (en) Patterning substrates employing multiple chucks
EP2175675B8 (en) Radio cell size management

Legal Events

Date Code Title Description
121 Ep: the epo has been informed by wipo that ep was designated in this application

Ref document number: 07757692

Country of ref document: EP

Kind code of ref document: A2

NENP Non-entry into the national phase in:

Ref country code: DE

122 Ep: pct application non-entry in european phase

Ref document number: 07757692

Country of ref document: EP

Kind code of ref document: A2