WO2007093530A1

WO2007093530A1 - Thioamide compounds for combating animal pest

Info

Publication number: WO2007093530A1
Application number: PCT/EP2007/051145
Authority: WO
Inventors: Florian Kaiser; Wolfgang Von Deyn; Matthias Pohlman; Douglas D. Anspaugh; Deborah L. Culbertson; Henry Van Tuyl Cotter
Original assignee: Basf Se
Priority date: 2006-02-16
Filing date: 2007-02-07
Publication date: 2007-08-23
Also published as: PE20071233A1; UY30162A1; TW200738606A; AR059553A1

Abstract

The present invention relates to thioamide compounds of the general formula (I) and to the agriculturally useful salts thereof and to compositions comprising such compounds. The invention also relates to the use of the thioamide compounds, of their salts or of compositions comprising them for combating animal pests. wherein R1,R2, R3,R4,R6 and X are defined as in the description.

Description

Thioamide compounds for combating animal pest

The present invention relates to thioamide compounds, to the enantiomers, diasteromers and the agriculturally useful salts thereof and to compositions comprising such compounds. The invention also relates to the use of the thioamide compounds, of their salts or of compositions comprising them for combating animal pests.

Animal pests destroy growing and harvested crops and attack wooden dwelling and commercial structures, causing large economic loss to the food supply and to property. While a large number of pesticidal agents are known, due to the ability of target pests to develop resistance to said agents, there is an ongoing need for new agents for combating animal pests. In particular, animal pests such as insects and acaridae are difficult to be effectively controlled.

EP 33984 discloses 2-cyanobenzene sulfonamides having aphicidal activity. Their activity, however, is not satisfactory. Similar compounds are described in WO 2005/035486.

EP 0203825 describes thiocarbonyl-sulfonylureas having herbicidal and plant growth regulant activity.

It is therefore an object of the present invention to provide compounds having a good pesticidal activity, especially against difficult to control insects and acaridae.

It has been found that these objects are solved by thioamide derivatives of the general formula I:

wherein

X is N, NO or C-R⁵

R¹ and R² are, independently of one another, selected from the group consisting of hydrogen, C(=O)-R⁷, Ci-Cio-alkyl, C₂-Cio-alkenyl, C₂-Cio-alkinyl, Ci-Cio-alkoxy or C3-Cio-cycloalkyl, wherein the five last-mentioned radicals may be unsubstituted, partially or fully halogenated and/or may carry 1 , 2 or 3 radicals, independently of one another each selected from the group consisting of cyano, nitro, amino, Ci-Cio-alkoxy, Ci-Cio-alkylthio, Ci-Cio-alkylsulfinyl, C1-C10- alkylsulfonyl, Ci-Cio-haloalkoxy, Ci-Cio-haloalkylthio, Ci-Cio-alkoxycarbonyl, (Ci- Cio-alkyl)amino, di-(Ci-Cio-alkyl)amino, C3-Cio-cycloalkyl and phenyl, it being possible for phenyl to be unsubstituted, partially or fully halogenated and/or to carry 1 , 2 or 3 substituents, independently of one another selected from the group consisting of Ci-C4-alkyl, Ci-C4-haloalkyl, Ci-C4-alkoxy and C1-C4- haloalkoxy; or wherein

R¹ and R² together with the adjacent nitrogen form a 3 to 10-membered ring, optionally substituted by 1 , 2 or 3 Ci-Cs-alkyl radicals, wherein the ring may contain, in addition to the nitrogen and carbon ring members, 1 , 2 or 3 heteroatoms as ring members selected from the group consisting of nitrogen, oxygen, sulfur, a group SO, SO2 or N-R⁸;

R³ is hydrogen, nitro, cyano, azido, amino, halogen, sulfonylamino, sulfenylamino, sulfinylamino, C(=O)R⁷ , Ci-Cβ-alkyl, C2-C6-alkenyl, C2-C6-alkinyl, C3-C8-cycloalkyl, Ci-Cβ-alkoxy, Ci-Cβ-alkylthio, (Ci-C6-alkyl)amino, di(Ci-C6- alkyl)amino, C 1 -Ce-a I ky I s u If i nyl , d-Cδ-alkylsulfenyl or Ci-Cδ-alkylsulfonyl, wherein the eleven last-mentioned radicals may be unsubstituted, partially or fully halogenated and/or may carry 1 , 2 or 3 radicals, selected from the group consisting of cyano, nitro, amino, Ci-C4-alkoxy, Ci-C4-alkylthio, C1-C4- alkylsulfinyl, Ci-C4-alkylsulfonyl, Ci-C4-haloalkoxy, Ci-C4-haloalkylthio, (C1-C4- alkoxy)carbonyl, (Ci-C4-alkyl)amino, di(Ci-C4-alkyl)amino, Ca-Cs-cycloalkyl and phenyl, it being possible for phenyl to be unsubstituted, partially or fully halogenated and/or to carry 1 , 2 or 3 substituents, independently of one another selected from the group consisting of Ci-C4-alkyl, Ci-C4-haloalkyl, Ci-C4-alkoxy and Ci-C4-haloalkoxy;

R⁴, R⁵ and R⁶ are independently of one another selected from the group consisting of hydrogen, halogen, cyano, azido, nitro, Ci-Cδ-alkyl, C3-C8- cycloalkyl, Ci-C4-haloalkyl, Ci-C4-alkoxy, Ci-C4-alkylthio, Ci-C4-alkylsulfinyl, Ci- C4-alkylsulfonyl, Ci-C4-haloalkoxy, Ci-C4-haloalkylthio, C2-C6-alkenyl, C2-C6- alkinyl, (Ci-C4-alkoxy)carbonyl, amino, (Ci-C4-alkyl)amino, di(Ci-C4-alkyl)amino, aminocarbonyl, (Ci-C4-alkyl)aminocarbonyl, di(Ci-C4-alkyl)aminocarbonyl, sulfonyl, sulfonylamino, sulfenylamino, sulfanylamino and C(=O)-R⁷;

R⁷ is hydrogen, hydroxy, Ci-Cβ-alkoxy, amino, Ci-C4-alkyl, aryl, aryl-Ci-C4-alkyl, a 3- to 7-membered heteroaryl or heteroaryl-Ci-C4-alkyl, wherein the heteroaryl ring contains as ring members 1 ,2 or 3 heteroatoms, selected from the group consisting of nitrogen, oxygen, sulfur, a group SO, SO2 or N-R⁸; or a 3- to 7-membered heterocyclyl or heterocyclyl-Ci-C4-alkyl, wherein the heterocyclic ring contains as ring members 1 , 2 or 3 heteroatoms, selected from the group consisting of nitrogen, oxygen, sulfur, a group SO, SO2 or N-R⁸ and wherein the carbon atoms of the heterocyclic rings may by unsubstituted or substituted by 1 or 2 Ci-C4-alkyl groups; R⁸ is hydrogen or Ci-C4-alkyl

and/or the enantiomers, diastereomers or salts thereof.

The compounds of the formula I, and their agriculturally acceptable salts are highly active against animal pest, i.e. harmful arthropodes and nematodes, especially against difficult to control insects and acaridae.

Accordingly, the present invention relates to thioamide compounds of the general formula I and to their agriculturally useful salts.

The present invention relates also to polymorphic forms of thioamide compounds of the general formula I.

The expression "compound of formula I" in this specification includes whenever used compounds of formula I, their enantiomers, distereomers, salts and polymorphic forms.

Moreover, the present invention relates to: agricultural compositions comprising such an amount of at least one thioamide derivative of the formula I and/or at least one agriculturally useful salt of I and at least one inert liquid and/or solid agronomically acceptable carrier that it has a pesticidal action and, if desired, at least one surfactant; the use of compounds of formula I and/or their salts for combating animal pests; and - a method of combating animal pests which comprises contacting the animal pests, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal attack or infestation with a pesticidally effective amount of at least one compound of the formula I and/or at least one agriculturally acceptable salt thereof, as defined herein, and to a method for protecting crops from attack or infestation by animal pests, which comprises contacting a crop with a pesticidally effective amount of at least one compound of the formula I and/or at least one salt thereof.

Salts of the compounds of the formula I are preferably agriculturally and veterinarily acceptable salts. They can be formed in a customary method, e.g. by reacting the compound with an acid of the anion in question if the compound of formula I has a basic functionality or by reacting an acidic compound of formula I with a suitable base.

Suitable agriculturally useful salts are especially the salts of those cations or the acid addition salts of those acids whose cations and anions, respectively, do not have any adverse effect on the action of the compounds according to the present invention. Suitable cations are in particular the ions of the alkali metals, preferably lithium, sodium and potassium, of the alkaline earth metals, preferably calcium, magnesium and barium, and of the transition metals, preferably manganese, copper, zinc and iron, and also ammonium (NH₄ ⁺) and substituted ammonium in which one to four of the hydrogen atoms are replaced by Ci-C4-alkyl, Ci-C4-hydroxyalkyl, Ci-C4-alkoxy, Ci-C4-alkoxy-Ci- C4-alkyl, hydroxy-Ci-C4-alkoxy-Ci-C4-alkyl, phenyl or benzyl. Examples of substituted ammonium ions comprise methylammonium, isopropylammonium, dimethylammonium, diisopropylammonium, trimethylammonium, tetramethylammonium, tetraethylammonium, tetrabutylammonium, 2-hydroxyethylammonium, 2-(2- hydroxyethoxy)ethylammonium, bis(2-hydroxyethyl)ammonium, benzyltrimethylammonium and benzyltriethylammonium, furthermore phosphonium ions, sulfonium ions, preferably tri(Ci-C4-alkyl)sulfonium, and sulfoxonium ions, preferably tri(Ci-C4-alkyl)sulfoxonium.

Anions of useful acid addition salts are primarily chloride, bromide, fluoride, hydrogen sulfate, sulfate, dihydrogen phosphate, hydrogen phosphate, phosphate, nitrate, hydrogen carbonate, carbonate, hexafluorosilicate, hexafluorophosphate, benzoate, and the anions of Ci-C4-alkanoic acids, preferably formate, acetate, propionate and butyrate. They can be formed by reacting the compounds of the formulae I with an acid of the corresponding anion, preferably of hydrochloric acid, hydrobromic acid, sulfuric acid, phosphoric acid or nitric acid.

By the term "veterinarily acceptable salts" is meant salts the anions of which are known and accepted in the art for the formation of salts for veterinary use. Suitable acid addition salts, e.g. formed by compounds of formula I containing a basic nitrogen atom, e.g. an amino group, include salts with inorganic acids, for example hydrochlorids, sulphates, phosphates, and nitrates and salts of organic acids for example acetic acid, maleic acid, dimaleic acid, fumaric acid, difumaric acid, methane sulfenic acid, methane sulfonic acid, and succinic acid.

The organic moieties mentioned in the above definitions of the variables are - like the term halogen - collective terms for individual listings of the individual group members. The prefix C_n-Cm indicates in each case the possible number of carbon atoms in the group.

"Halogen" will be taken to mean fluoro, chloro, bromo and iodo.

The term "partially or fully halogenated" will be taken to mean that 1 or more, e.g. 1 , 2, 3, 4 or 5 or all of the hydrogen atoms of a given radical have been replaced by a halogen atom, in particular by fluorine or chlorine.

The term "Cn-C_m-alkyl" as used herein (and also in Cn-C_m-alkylamino, di-C_n-C_m- alkylamino, Cn-Cm-alkylaminocarbonyl, di-(Cn-C_m-alkylamino)carbonyl, Cn-C_m-alkylthio, Cn-Cm-alkylsulfinyl and C_n-C_m-alkylsulfonyl) refers to a branched or unbranched saturated hydrocarbon group having n to m, e.g. 1 to 10 carbon atoms, preferably 1 to 6 carbon atoms, for example methyl, ethyl, propyl, 1-methylethyl, butyl, 1-methylpropyl, 2-methylpropyl, 1 ,1-dimethylethyl, pentyl, 1-methylbutyl, 2-methylbutyl, 3-methylbutyl, 2,2-dimethylpropyl, 1-ethylpropyl, hexyl, 1 ,1-dimethylpropyl, 1 ,2-dimethylpropyl, 1- methylpentyl, 2-methylpentyl, 3-methylpentyl, 4-methylpentyl, 1 ,1-dimethylbutyl, 1 ,2- dimethylbutyl, 1 ,3-dimethylbutyl, 2,2-dimethylbutyl, 2,3-dimethylbutyl, 3,3-dimethylbutyl, 1-ethylbutyl, 2-ethylbutyl, 1 ,1 ,2-trimethylpropyl, 1 ,2,2-trimethylpropyl, 1 -ethyl-1 - methylpropyl, 1-ethyl-2-methylpropyl, heptyl, octyl, 2-ethylhexyl, nonyl and decyl and their isomers. Ci-C4-alkyl means for example methyl, ethyl, propyl, 1-methylethyl, butyl, 1-methylpropyl, 2-methylpropyl or 1 ,1-dimethylethyl.

The term "Cn-C_m-haloalkyl" as used herein (and also in C_n-C_m-haloalkylsulfinyl and C_n- Cm-haloalkylsulfonyl) refers to a straight-chain or branched alkyl group having n to m carbon atoms, e.g. 1 to 10 in particular 1 to 6 carbon atoms (as mentioned above), where some or all of the hydrogen atoms in these groups may be replaced by halogen atoms as mentioned above, for example Ci-C4-haloalkyl, such as chloromethyl, bromomethyl, dichloromethyl, trichloromethyl, fluoromethyl, difluoromethyl, trifluoromethyl, chlorofluoromethyl, dichlorofluoromethyl, chlorodifluoromethyl, 1- chloroethyl, 1-bromoethyl, 1-fluoroethyl, 2-fluoroethyl, 2,2-difluoroethyl, 2,2,2- trifluoroethyl, 2-chloro-2-fluoroethyl, 2-chloro-2,2-difluoroethyl, 2,2-dichloro-2- fluoroethyl, 2,2,2-trichloroethyl, pentafluoroethyl and the like. The term Ci-Cio-haloalkyl in particular comprises Ci-C2-fluoroalkyl, which is synonym with methyl or ethyl, wherein 1 , 2, 3, 4 or 5 hydrogen atoms are substituted by fluorine atoms, such as fluoromethyl, difluoromethyl, trifluoromethyl, 1-fluoroethyl, 2-fluoroethyl, 2,2- difluoroethyl, 2,2,2-trifluoroethyl and pentafluoromethyl.

Similarly, "C_n-C_m-alkoxy" and "C_n-C_m-alkylthio" (or C_n-C_m-alkylsulfenyl, respectively) refer to straight-chain or branched alkyl groups having n to m carbon atoms, e.g. 1 to 10, in particular 1 to 6 or 1 to 4 carbon atoms (as mentioned above) bonded through oxygen or sulfur linkages, respectively, at any bond in the alkyl group. Examples include Ci-C4-alkoxy such as methoxy, ethoxy, propoxy, isopropoxy, butoxy, sec- butoxy, isobutoxy and tert-butoxy, futher Ci-C4-alkylthio such as methylthio, ethylthio, propylthio, isopropylthio, and n-butylthio.

Accordingly, the terms "C_n-C_m-haloalkoxy" and "C_n-C_m-haloalkylthio" (or C_n-Cm- haloalkylsulfenyl, respectively) refer to straight-chain or branched alkyl groups having n to m carbon atoms, e.g. 1 to 10, in particular 1 to 6 or 1 to 4 carbon atoms (as mentioned above) bonded through oxygen or sulfur linkages, respectively, at any bond in the alkyl group, where some or all of the hydrogen atoms in these groups may be replaced by halogen atoms as mentioned above, for example Ci-C2-haloalkoxy, such as chloromethoxy, bromomethoxy, dichloromethoxy, trichloromethoxy, fluoromethoxy, difluoromethoxy, trifluoromethoxy, chlorofluoromethoxy, dichlorofluoromethoxy, chlorodifluoromethoxy, 1-chloroethoxy, 1-bromoethoxy, 1-fluoroethoxy, 2-fluoroethoxy, 2,2-difluoroethoxy, 2,2,2-trifluoroethoxy, 2-chloro-2-fluoroethoxy, 2-chloro-2,2- difluoroethoxy, 2,2-dichloro-2-fluoroethoxy, 2,2,2-trichloroethoxy and pentafluoroethoxy, further Ci-C2-haloalkylthio, such as chloromethylthio, bromomethylthio, dichloromethylthio, trichloromethylthio, fluoromethylthio, difluoromethylthio, trifluoromethylthio, chlorofluoromethylthio, dichlorofluoromethylthio, chlorodifluoromethylthio, 1-chloroethylthio, 1-bromoethylthio, 1-fluoroethylthio, 2- fluoroethylthio, 2,2-difluoroethylthio, 2,2,2-trifluoroethylthio, 2-chloro-2-fluoroethylthio, 2-chloro-2,2-difluoroethylthio, 2,2-dichloro-2-fluoroethylthio, 2,2,2-trichloroethylthio and pentafluoroethylthio and the like. Similarly the terms Ci-C2-fluoroalkoxy and C1-C2- fluoroalkylthio refer to Ci-C2-fluoroalkyl which is bound to the remainder of the molecule via an oxygen atom or a sulfur atom, respectively.

The term "C2-C_m-alkenyl" as used herein referrs to a branched or unbranched unsaturated hydrocarbon group having 2 to m, e.g. 2 to 10 or 2 to 6 carbon atoms and a double bond in any position, such as ethenyl, 1-propenyl, 2-propenyl, 1-methyl- ethenyl, 1-butenyl, 2-butenyl, 3-butenyl, 1-methyl-1-propenyl, 2-methyl-1-propenyl, 1- methyl-2-propenyl, 2-methyl-2-propenyl, 1-pentenyl, 2-pentenyl, 3-pentenyl, 4-pentenyl, 1-methyl-1-butenyl, 2-methyl-1-butenyl, 3-methyl-1-butenyl, 1-methyl-2-butenyl, 2- methyl-2-butenyl , 3-methyl-2-butenyl , 1 -methyl-3-butenyl , 2-methyl-3-butenyl , 3-methyl- 3-butenyl, 1 ,1-dimethyl-2-propenyl, 1 ,2-dimethyl-1-propenyl, 1 ,2-dimethyl-2-propenyl, 1-ethyl-1-propenyl, 1-ethyl-2-propenyl, 1-hexenyl, 2-hexenyl, 3-hexenyl, 4-hexenyl, 5- hexenyl, 1-methyl-1-pentenyl, 2-methyl-1-pentenyl, 3-methyl-1-pentenyl, 4-methyl-1- pentenyl, 1-methyl-2-pentenyl, 2-methyl-2-pentenyl, 3-methyl-2-pentenyl, 4-methyl-2- pentenyl, 1-methyl-3-pentenyl, 2-methyl-3-pentenyl, 3-methyl-3-pentenyl, 4-methyl-3- pentenyl, 1-methyl-4-pentenyl, 2-methyl-4-pentenyl, 3-methyl-4-pentenyl, 4-methyl-4- pentenyl, 1 ,1-dimethyl-2-butenyl, 1 ,1-dimethyl-3-butenyl, 1 ,2-dimethyl-1-butenyl, 1 ,2- dimethyl-2-butenyl, 1 ,2-dimethyl-3-butenyl, 1 ,3-dimethyl-1-butenyl, 1 ,3-dimethyl-2- butenyl, 1 ,3-dimethyl-3-butenyl, 2,2-dimethyl-3-butenyl, 2,3-dimethyl-1-butenyl, 2,3- dimethyl-2-butenyl, 2,3-dimethyl-3-butenyl, 3,3-dimethyl-1-butenyl, 3,3-dimethyl-2- butenyl, 1-ethyl-1-butenyl, 1-ethyl-2-butenyl, 1-ethyl-3-butenyl, 2-ethyl-1-butenyl, 2- ethyl-2-butenyl, 2-ethyl-3-butenyl, 1 ,1 ,2-trimethyl-2-propenyl, 1-ethyl-1-methyl-2- propenyl, 1-ethyl-2-methyl-1-propenyl and 1-ethyl-2-methyl-2-propenyl.

The term "C2-C_m-alkynyl" as used herein refers to a branched or unbranched unsaturated hydrocarbon group having 2 to m, e.g. 2 to 10 or 2 to 6 carbon atoms and containing at least one triple bond, such as ethynyl, propynyl, 1-butynyl, 2-butynyl, and the like.

The term Ci-C4-alkoxy-Ci-C4-alkyl as used herein refers to alkyl having 1 to 4 carbon atoms, wherein one hydrogen atom of the alkyl radical is replaced by an Ci-C4-alkoxy group. The term Ci-C4-alkylthio-Ci-C4-alkyl as used herein refers to alkyl having 1 to 4 carbon atoms, wherein one hydrogen atom of the alkyl radical is replaced by a Ci-C4-alkylthio group.

The term "C3-C_m-cycloalkyl" as used herein refers to a monocyclic 3- to m-membered saturated cycloaliphatic radicals, e.g. cyclopropyl, cyclobutyl, cyclopentyl, cyclohexyl, cycloheptyl, cyclooctyl and cyclodecyl.

The term aryl as used herein refers to an aromatic hydrocarbon radical such as naphthyl or in particular phenyl.

The term aryl-Ci-C4-alkyl as used herein refers to an aromatic hydrocarbon radical, which is bound to the remainder of the molecule via a Ci-C4-alkylene group, examples comprise benzyl, 1-phenylethyl or 2-phenylethyl.

The term "3- to 7-membered heterocyclyl" as used herein (and also in "heterocyclyl-Ci- C4-alkyl") refers to a saturated or partially unsaturated non-aromatic heterocyclic radical havin 3 to 7 ring members, wherein 1 , 2 or 3 ring members are heteroatoms selected from O, N and S or heteroatom groups, selected from S=O, S(O)2 or N-R with R being H or alkyl. Examples for non-aromatic rings include azetidiyl, pyrrolidinyl, pyrazolinyl, imidazolinyl, pyrrolinyl, pyrazolinyl, imidazolinyl, tetrahydrofuranyl, dihydrofuranyl, 1 ,3-dioxolanyl, dioxolenyl, thiolanyl, dihydrothienyl, oxazolidinyl, isoxazolidinyl, oxazolinyl, isoxazolinyl, thiazolinyl, isothiazolinyl, thiazolidinyl, isothiazolidinyl, oxathiolanyl, piperidinyl, piperazinyl, pyranyl, dihydropyranyl, tetrahydropyranyl, dioxanyl, thiopyranyl, dihydrothiopyranyl, tetrahydrothiopyranyl, morpholinyl, thiazinyl and the like.

The term "3- to 7-membered heteroaryl" as used herein (and also in "heteroaryl-Ci-C4- alkyl") refers to an aromatic heterocyclic radical havin 3 to 7 ring members, wherein 1 , 2 or 3 ring members are heteroatoms selected from O, N and S or heteroatom groups, selected from S=O, S(O)2 or N-R with R being H or alkyl. Examples for monocyclic 3- to 7-membered heteroaromatic rings include triazinyl, pyrazinyl, pyrimidyl, pyridazinyl, pyridyl, thienyl, furyl, pyrrolyl, pyrazolyl, imidazolyl, triazolyl, tetrazolyl, thiazolyl, oxazolyl, thiadiazolyl, oxadiazolyl, isothiazolyl and isoxazolyl.

The terms heterocyclyl-Ci-C4-alkyl and heteroaryl-Ci-C4-alkyl as used herein refer to an aromatic or non-aromatic heterocyclic radical, which is bound to the remainder of the molecule via a Ci-C4-alkylene group.

With respect to the use according to the invention of the thioamide compounds of formula I, particular preference is given to the following meanings of the substituents and variables, in each case on their own or in combination: Thioamide compounds of the formula I, wherein R¹ and R² are, independently of one another, selected from the group consisting of hydrogen, Ci-Cδ-alkyl, Ci-Cβ-haloalkyl, C2-C6-alkenyl, C2-C6-haloalkenyl, C2-C6-alkinyl, C2-C6-haloalkinyl, C3-C6-cycloalkyl, Ci- C4-alkoxy-Ci-C4-alkyl and Ci-C4-alkylthio-Ci-C4-alkyl. However R¹ may also form a radical C(=O)-R⁷, wherein R⁷ is selected from Ci-C4-alkyl, Ci-C3-alkoxy-Ci-C3-alkyl, Ci- C3-alkylthio-Ci-C3-alkyl or Ci-C4-haloalkyl, in particular R⁷ being Ci-C4-alkyl or Cr haloalkyl, such as methyl, ethyl, trifluoromethyl or trichloromethyl. Preferably thioamide compounds of the formula I, wherein R¹ and R² are, independently of one another, selected from the group consisting of hydrogen, C1-C4- alkyl, in particular methyl, ethyl or 1-methylethyl, cyclopropyl, C2-C4-alkinyl, in particular prop-3-yn-1-yl, and C(=O)-R⁷, wherein R⁷ is selected from Ci-C4-alkyl, in particular methyl, ethyl, 1-methylethyl or 2-methylpropan-2-yl, Ci-C3-alkoxy-Ci-C3-alkyl, in particular 2-methoxyethyl, Ci-C3-alkylthio-Ci-C3-alkyl, in particular 2-methylthioethyl, and Ci-C4-haloalkyl, in particular trifluoromethyl or trichloromethyl. More preferably thioamide compounds of the formula I, wherein R¹ and R² are, independently of one another, selected from the group consisting of hydrogen, methyl, ethyl, 1-methylethyl, cyclopropyl or prop-3-yn-1-yl.

Especially preferred are also thioamide compounds of the formula I, wherein R¹ or R² is C(=O)-R⁷, and wherein R⁷ is selected from Ci-C₄-alkyl, Ci-C₃-alkoxy-Ci-C₃-alkyl, C1-C3- alkylthio-Ci-C3-alkyl or Ci-C4-haloalkyl.

In particular thioamide compounds of the formula I, wherein R¹ or R² is C(=O)-R⁷, and wherein R⁷ is selected from methyl, ethyl, 1-methylethyl, 2-methylpropan-2-yl, 2- methoxyethyl, 2-methylthioethyl, trifluoromethyl or trichlormethyl.

Thioamide compounds of the formula I, wherein R³ is halogen, Ci-C4-alkyl, C1-C4- haloalkyl, Ci-C4-alkoxy or Ci-C4-haloalkoxy.

Preferably thioamide compounds of the formula I, wherein R³ is halogen, Ci-C2-alkyl,

Ci-haloalkyl, Ci-C2-alkoxy or Ci-haloalkoxy. More preferred are thioamide compounds of the formula I, wherein R³ is methyl, trifluoromethyl, trichloromethyl, methoxy, trifluoromethoxy, difluoromethoxy, fluoromethoxy or chlorodifluoromethoxy, chlorine or fluorine.

Thioamide compounds of the formula I, wherein X is N and R⁴ and R⁶ are selected, independently from each other, from hydrogen, halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, Ci-C4-alkoxy or d- C4-haloalkoxy.

Preferably thioamide compounds of the formula I, wherein X is N and R⁴ and R⁶ are selected, independently from each other, from hydrogen, halogen, Ci-C2-alkyl, or Ci- haloalkyl. More preferred are thioamide compounds of the formula I , wherein X is N and R⁴ and R⁶ are selected, independently from each other, from H, Cl, Br, I, CH3 or CF3. Especially preferred are thioamide compounds of the formula I , wherein X is N and one of the radicals R⁴ or R⁶ being present, is different from hydrogen, while the other one being present is hydrogen.

In another embodiment of the invention, thioamide compounds of the formula I are also preferred, wherein X is N and both of the radicals R⁴ and R⁶ being present are hydrogen.

Thioamide compounds of the formula I, wherein X is C-R⁵ and R⁴, R⁵, and R⁶ are selected, independently from each other, from hydrogen, halogen, Ci-C4-alkyl, C1-C4- haloalkyl, Ci-C4-alkoxy or Ci-C4-haloalkoxy.

Preferably thioamide compounds of the formula I , wherein X is C-R⁵ and R⁴, R⁵, and

R⁶ are selected, independently from each other, from hydrogen, halogen, Ci-C2-alkyl or d-haloalkyl, More preferred are thioamide compound of the formula I , wherein X is C-R⁵ and R⁴,

R⁵, and R⁶ are selected, independently from each other, from H, Cl, Br, I, CH3 or CF3.

Especially preferred are thioamide compounds of the formula I, wherein X is C-R⁵ and one of the radicals R⁴, R⁵ or R⁶ being present, is different from hydrogen, while the other two being present are hydrogen,

In another embodiment of the invention, thioamide compound of the formula I are preferred, wherein X is C-R⁵ and all three of the radicals R⁴, R⁵ or R⁶ being present are hydrogen.

Preferred substituents X, R⁴, R⁵ and R⁶ are defined in the following formulas W1 to W243:

W1 W2 W3 W4

W9 W10 W1 1 W12

W13 W14 W15 W16

W17 W18 W19 W20

W21 W22 W23

W24 W25 W26 W27

W28 W29 W30 W31

W32 W33 W34 W35

W40 W41 W42

W43 W44 W45

W47 W48 W49

W50 W51 W52

W53 W54 W55

W61

W62 W63 W64

W81 W82 W83 W84

W89 W90 W91 W92

W95

W105 W106 W107

W111 W112 W113

W114 W115 W116

W117 W118 W119

W120 W121 W122

W123 W124 W125 W126 R³

W127 W128 W129 W130

W131 W132 W133

W134 W135 W136

W137 W138 W139

W140 W141 W142 W143

R³

W144 W145 W146 W147

W148 W149 W150

W151 W152 W153

W 154 W155 W156

W160 W161 W162 W163

W170 W171 W172

W173 W174 W175

W180 W181 W182 W183

W191 W192 W193 W194

W195 W196 W197

W202 W203 W204 W205

W209 W210 W21 1

W212 W213 W214

W219 W220 W221

W222 W223 W224

W225 W226 W227

W228 W229 W230

W234 W235 W236

Preparation methods

Thioamide compounds of the formula I can be prepared, for example, by reacting a α- cyano sulfonamide (II) with a thionating agent (III), for example gaseous hydrogen sulfide (see Scheme 1), as described in Journal of the Chemical Society, 1952, 742-4. In Scheme 1 the variables X and R¹ to R⁶ are as defined above. Scheme 1 :

In general, the thionating reagent, for example hydrogen sulphide, is employed in at least equimolar amount. Other thionating reagents that are also suitable include, for example, sodium hydrogen sulphate / magnesium chloride as described in Synthetic Communications 2005, 35, 761-764; or ammonium sulphide, as described in Synlett 2004, 14, 2615-2617; or sulfide salts in aqueous solution as described in WO 2003072547, or sodium trimethylsilyl sulfide as described in Synthesis 1992, 12, 1219- 1220, or phosphorus decasulfide/ sodium sulfide as described in Synthetic Communications 1992, 22, 1397-1401 ; or Diphenylphosphinodithioic acid as described in Tetrahedron Letters 1981 , 22, 1851-1854.

If gaseous hydrogen sulfide is used as a reagent, then the reaction should be performed in the presence of an amide base, for example trimethylamine, triethylamine or diisopropylamine, N-methylpiperidine, pyridine, substituted pyridines such as 2,3,5- collidine, 2,4,6-collidine, 2,4-lutidine, 3,5-lutidine or 2,6-lutidine.

The reaction of (II) and (III) is usually carried out in the presence of a solvent. Suitable solvents are solvents which are inert under the reaction conditions, for example (hetero)aromatic hydrocarbons like pyridine, benzene, toluene; dialkyl ethers such as diethyl ether, diisopropyl ether or methyl tert-butyl ether, cyclic ethers such as dioxane or tetrahydrofuran, acetonitrile, carboxamides such as N,N-dimethyl formamide, N₁N- dimethyl acetamide or N-methylpyrrolidinone, water, (provided the α-cyano sulfonamide (II) is sufficiently resistant to hydrolysis under the reaction conditions used) or a mixture thereof.

The reaction of (II) and (III) is usually carried out at a reaction temperature ranging from 0°C to the boiling point of the solvent, preferably from 0 to 30°C.

The α-cyano sulfonamides with X = C-R⁵ (VIII) can be prepared, for example, according to the reaction sequence shown in scheme 2 where the variables R¹, R², R³, R⁴, R⁵, and R⁶ are as defined above:

Scheme 2:

a) Conversion of the 2,6-difluoro-benzonitriles (IV) to the alkyl- or alkoxy analogues (V) by reacting (IV) with an appropriate alkoxide such as sodium methoxide and sodium ethoxide or, if R3 is an alkyl group, be reacting with an alkylate such as methyl magnesium chloride, in an inert organic solvent, for example an ether such as diethyl ether, diisopropyl ether, tetrahydrofuran, dioxane, or in the respective alcohol, or in a carboxamide such as N,N-dimethyl formamide, N,N-dimethyl acetamide or N- methylpyrrolidinone, or in dimethylsulfoxide or in a mixture of the above mentioned solvents providing the solvent is inert under the reaction conditions.

b) Transformation of fluorobenzene (V) into thioether (Vl) wherein y is an alkyl or phenyl group by reacting with alkyl- or benzylthiol in the presence of a base. Suitable bases are alkali metal alkoxides such as sodium methoxide, potassium methoxide or potassium tert-butoxide, alkali metal hydroxides such as sodium hydroxide or potassium hydroxide. The reaction is usually carried out in a solvent, for example an ether such as diethyl ether, diisopropyl ether, tetrahydrofuran, ethylen glycol dimethylether, dioxane, or in a carboxamide such as N,N-dimethyl formamide, N₁N- dimethyl acetamide or N-methylpyrrolidinone or in dimethylsulfoxide or in water. It may also be possible to use an excess of the alkyl- or benzylthiol, which then serves as solvent.

c) Transformation of thioether (Vl) into sulfonylchloride (VII) in analogy to a process described in WO 96/33167 by reacting (Vl) with chlorine in a suitable solvent, for example chlorobenzene or dichloromethane in the presence of water.

d) Reaction of the sulfonylchloride (VII), with an amine can be carried out similarly to standard methods of reacting sulfonylhalides with primary or secondary amines as described in J. March, 4^th edition 1992, p. 499 and in the literature cited therein. In general, the amine is employed in an at least equimolar amount, preferably at least 2- fold molar excess, based on the sulfonylchloride (VII), to bind the hydrogen halide formed. It may be advantageous to employ the amine in an up to 6-fold molar excess, based on the sulfonylchloride (VII). It may be advantageous to carry out the reaction in the presence of an auxiliary base. Suitable auxiliary bases include organic bases, for example tertiary amines, such as aliphatic tertiary amines, such as trimethylamine, triethylamine or diisopropylamine, cycloaliphatic tertiary amines such as N- methylpiperidine or aromatic amines such pyridine, substituted pyridines such as 2,3,5- collidine, 2,4,6-collidine, 2,4-lutidine, 3,5-lutidine or 2,6-lutidine and inorganic bases for example alkali metal hydrides such as sodium hydride and potassium hydride, alkali metal carbonates and alkaline earth metal carbonates such as lithium carbonate, potassium carbonate and sodium carbonate, calcium carbonate and alkaline metal hydrogencarbonates such as sodium hydrogen carbonate. The molar ratio of auxiliary base to sulfonylchloride (VII) is preferably in the range of from 1 :1 to 4:1 , preferably 1 :1 to 2:1. If the reaction is carried out in the presence of an auxiliary base, the molar ratio of the amine to sulfonylchloride (VII) usually is 1 :1 to 1.5:1.

The reaction of VII with an amine is usually carried out in the presence of a solvent. Suitable solvents are polar solvents which are inert under the reaction conditions, for example Ci-C4-alkanols such as methanol, ethanol, n-propanol or isopropanol, dialkyl ethers such as diethyl ether, diisopropyl ether or methyl tert-butyl ether, cyclic ethers such as dioxane or tetrahydrofuran, acetonitrile, carboxamides such as N,N-dimethyl formamide, N,N-dimethyl acetamide or N-methylpyrrolidinone, water, (provided the sulfonylchloride (VII) is sufficiently resistent to hydrolysis under the reaction conditions used) or a mixture thereof. The reaction of (VII) with the amine is usually carried out at a reaction temperature ranging from 0°C to the boiling point of the solvent, preferably from 0 to 30⁰C.

The α-Cyano sulfonamides with X = C-R⁵ and R⁶ = F (XII) can be prepared, for example, according to the reaction sequence shown in scheme 3 where the variables R¹, R², R³, R⁴ and R⁵ are as defined above:

Scheme 3:

a) if the nitrile (X) is not commercial available, it can be prepared by conversion of a 2,5-difluoro benzonitrile (IX) into 2-alkyl- or 2-alkoxy-5-fluorobenzonitrile (X), if R³ is an alkyl or alkoxy group via introduction of an alkyl or alkoxide substituent, which can be carried out, for example, in analogy to a process described in Tetrahedron Letters 1996, 37, 6439-6442, by reacting (IX) with an alkali metal alkylate or alkali metal alkoxide like, for example, sodium methylate in an inert organic solvent, for example dialkyl ethers such as diethyl ether, diisopropyl ether or methyl tert-butyl ether, cyclic ethers such as dioxane or tetrahydrofuran, acetonitrile, carboxamides such as N₁N- dimethyl formamide, N,N-dimethyl acetamide or N-methylpyrrolidinone. The reaction is usually carried out at a reaction temperature ranging from 0 °C to the boiling point of the solvent. The molar ratio of the alkali metal alkylate or alkali metal alkoxide to 2,5- difluoro benzonitrile (IX) is preferably in the range from 1 :1 to 10:1 ; and subsequent

b) directed ortho-metalation of (X), which can be carried out using, for example, a strong amide base like lithium diisopropylamide or lithium tetramethylpiperidide in an inert organic solvent, for example dialkyl ethers such as diethyl ether, diisopropyl ether or methyl tert-butyl ether or cyclic ethers such as dioxane or tetrahydrofuran, as described in Tetrahedron Letters 1992, 3349, 7495-7498 or Journal of Organic Chemistry 2004, 69, 556-569, followed by transformation of the intermediate aryllithium species into the sulfonyl chloride (Xl) by subsequent reaction of the corresponding lithiated intermediate with sulphur dioxide followed by a chlorinating agent like sulfuryl chloride or N-chlorosuccinimide, as described in Journal of Organic Chemistry 2003, 68, 8274-8276 or Tetrahedron 1999, 55, 237-254; and subsequent

c) reaction of the sulfonylchloride (Xl) with an amine, which can be carried out similarly to standard methods of reacting sulfonylhalides with primary or secondary amines as described in J. March, 4^th edition 1992, p. 499 and in the literature cited therein. In general, the amine is employed in an at least equimolar amount, preferably at least 2-fold molar excess, based on the sulfonylchloride (Xl), to bind the hydrogen halide formed. It may be advantageous to employ the amine in an up to 6-fold molar excess, based on the sulfonylchloride (Xl). It may be advantageous to carry out the reaction in the presence of an auxiliary base. Suitable auxiliary bases include organic bases, for example tertiary amines, such as aliphatic tertiary amines, such as trimethylamine, triethylamine or diisopropylamine, cycloaliphatic tertiary amines such as N-methylpiperidine or aromatic amines such pyridine, substituted pyridines such as 2,3,5-collidine, 2,4,6-collidine, 2,4-lutidine, 3,5-lutidine or 2,6-lutidine and inorganic bases for example alkali metal hydrides such as sodium hydride and potassium hydride, alkali metal carbonates and alkaline earth metal carbonates such as lithium carbonate, potassium carbonate and sodium carbonate, calcium carbonate and alkaline metal hydrogencarbonates such as sodium hydrogen carbonate. The molar ratio of auxiliary base to sulfonylchloride (Xl) is preferably in the range of from 1 :1 to 4:1 , preferably 1 :1 to 2:1. If the reaction is carried out in the presence of an auxiliary base, the molar ratio of the amine to sulfonylchloride (Xl) usually is 1 :1 to 1.5:1. The reaction of (Xl) with an amine is usually carried out in the presence of a solvent. Suitable solvents are polar solvents which are inert under the reaction conditions, for example Ci-C4-alkanols such as methanol, ethanol, n-propanol or isopropanol, dialkyl ethers such as diethyl ether, diisopropyl ether or methyl tert-butyl ether, cyclic ethers such as dioxane or tetrahydrofuran, acetonitrile, carboxamides such as N,N-dimethyl formamide, N,N-dimethyl acetamide or N-methylpyrrolidinone, water, (provided the sulfonylchloride (Xl) is sufficiently resistant to hydrolysis under the reaction conditions used) or a mixture thereof. The reaction of (Xl) with the amine is usually carried out at a reaction temperature ranging from 0°C to the boiling point of the solvent, preferably from 0 to 30°C.

The α-Cyano sulfonamides with X = N (XVII) can be prepared, for example, according to the reaction sequence shown in scheme 4 where the variables R¹, R², R³, R⁴ and R⁶ are as defined above:

Scheme 4:

(XIII) (XIV) (XV)

a) conversion of a dichloroisonicotinonitrile (XIII) into a thioalkylether or thiophenylether (XIV) wherein z is an alkyl or phenyl group, preferably a thiopropyl- or thiobenzylether, for example, in analogy to a process described in Heterocycles Vol. 43, No. 9, (1996), pp. 1893-1899, by reacting (XIII) with an alkaline thiopropylate or alkaline thiobenzylate reagent formed from propanethiol respective benzylthiol and a base such as for example alkali metal hydrides such as sodium hydride and potassium hydride, alkali metal carbonates and alkaline earth metal carbonates such as lithium carbonate, potassium carbonate and sodium carbonate, calcium carbonate, alkaline metal hydrogencarbonates such as sodium hydrogen carbonate, or an organo alkyl metal reagent like butyllithium. The reaction can be performed in an inert organic solvent, for example dialkyl ethers such as diethyl ether, diisopropyl ether or methyl tert-butyl ether, cyclic ethers such as dioxane or tetrahydrofuran, acetonitrile, carboxamides such as N,N-dimethyl formamide, N,N-dimethyl acetamide or N- methylpyrrolidinone. The reaction is usually carried out at a reaction temperature ranging from 0 °C to the boiling point of the solvent. The molar ratio of the alkaline thiopropylate or thiobenzylate to dichloroisonicotinonitrile (XIII) is preferably in the range from 1 :1 to 1.5:1.

The dichloroisonicotinonitrile (XIII) can be prepared in analogy to a process described in Heterocycles Vol. 43, No. 9, (1996), pp. 1893-1899; or a process described in Journal of Medicinal Chemistry, Vol. 44, No.6, (2001 ), pp. 988-100; and subsequent

b) Introduction of an alkyl or alkoxide substituent, if R³ is an alkyl or alkoxide group, for example, in analogy to a process described in Heterocycles Vol. 43, No. 9, (1996), pp. 1893-1899, by reacting (XIV) with an alkali metal alkylate or alkali metal alkoxide like, for example, sodium methylate in an inert organic solvent, for example dialkyl ethers such as diethyl ether, diisopropyl ether or methyl tert-butyl ether, cyclic ethers such as dioxane or tetrahydrofuran, acetonitrile, carboxamides such as N₁N- dimethyl formamide, N,N-dimethyl acetamide or N-methylpyrrolidinone. The reaction is usually carried out at a reaction temperature ranging from 0 °C to the boiling point of the solvent. The molar ratio of the alkali metal alkylate or alkali metal alkoxide to chloronicotononitrile (XIV) is preferably in the range from 1 :1 to 10:1 ; and subsequent

c) oxidative cleavage of the thioether (XV) to obtain the sulfonylchloride (XVI) for example, by reacting the thioether (XV) with chlorine in water or a water-solvent mixture, e. g. a mixture of water and acetic acid or water and dichloromethane, in analogy to a process described in Canadian Journal of Chemistry, Vol. 74, No. 9, (1996), pp. 1638-1648; and subsequent

d) reaction of the sulfonylchloride (XVI), with an amine, which can be carried out similarly to standard methods of reacting sulfonylhalides with primary or secondary amines as described in J. March, 4^th edition 1992, p. 499 and in the literature cited therein. In general, the amine is employed in an at least equimolar amount, preferably at least 2-fold molar excess, based on the sulfonylchloride (XVI), to bind the hydrogen halide formed. It may be advantageous to employ the amine in an up to 6-fold molar excess, based on the sulfonylchloride (XVI). It may be advantageous to carry out the reaction in the presence of an auxiliary base. Suitable auxiliary bases include organic bases, for example tertiary amines, such as aliphatic tertiary amines, such as trimethylamine, triethylamine or diisopropylamine, cycloaliphatic tertiary amines such as N-methylpiperidine or aromatic amines such pyridine, substituted pyridines such as 2,3,5-collidine, 2,4,6-collidine, 2,4-lutidine, 3,5-lutidine or 2,6-lutidine and inorganic bases for example alkali metal hydrides such as sodium hydride and potassium hydride, alkali metal carbonates and alkaline earth metal carbonates such as lithium carbonate, potassium carbonate and sodium carbonate, calcium carbonate and alkaline metal hydrogencarbonates such as sodium hydrogen carbonate. The molar ratio of auxiliary base to sulfonylchloride (XVI) is preferably in the range of from 1 :1 to 4:1 , preferably 1 :1 to 2:1. If the reaction is carried out in the presence of an auxiliary base, the molar ratio of the amine to sulfonylchloride (XVI) usually is 1 :1 to 1.5:1. The reaction of (XVI) with an amine is usually carried out in the presence of a solvent. Suitable solvents are polar solvents which are inert under the reaction conditions, for example Ci-C4-alkanols such as methanol, ethanol, n-propanol or isopropanol, dialkyl ethers such as diethyl ether, diisopropyl ether or methyl tert-butyl ether, cyclic ethers such as dioxane or tetrahydrofuran, acetonitrile, carboxamides such as N,N-dimethyl formamide, N,N-dimethyl acetamide or N-methylpyrrolidinone, water, (provided the sulfonylchloride (XVI) is sufficiently resistant to hydrolysis under the reaction conditions used) or a mixture thereof. The reaction of (XVI) with the amine is usually carried out at a reaction temperature ranging from 0°C to the boiling point of the solvent, preferably from O to 30⁰C.

α-Cyano sulfonamides with X = NO (XIX) can be prepared, for example, by reacting the corresponding pyridine compound (XVIII), and an oxidation reagent (XX), for example a peroxide reagent like 3-chloroperbenzoic acid (see Scheme 9), similarly to a process described in Synthetic Communications 1977, Vol. 7, No. 8, pp. 509-14.

Scheme 5:

(XVIII)

If individual compounds cannot be prepared via the above-described routes, they can be prepared by derivatization of other compounds I or by customary modifications of the synthesis routes described.

The reaction mixtures are worked up in the customary manner, for example by mixing with water, separating the phases, and, if appropriate, purifying the crude products by chromatography, for example on alumina or silica gel may be employed. Some of the intermediates and end products may be obtained in the form of colorless or pale brown viscous oils, which are freed or purified from volatile components under reduced pressure and at moderately elevated temperature. If the intermediates and end products are obtained as solids, they may be purified by recrystallization or digestion.

Agriculturally acceptable salts of the compounds I can be formed in a customary manner, e.g. by reaction with an acid of the anion in question.

Examples of preferred compounds of the formula I are given in the following tables A1 to A2700, wherein X, R⁴,R⁵ and R⁶ are defined as in formulas W1-W243 above and R¹ and R² are defined as in table A below: Table A1 : Compounds of the formula W1 , wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A2: Compounds of the formula W1 , wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A3: Compounds of the formula W1 , wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A4: Compounds of the formula W1 , wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A5: Compounds of the formula W1 , wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A6: Compounds of the formula W1 , wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A7: Compounds of the formula W1 , wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A8: Compounds of the formula W1 , wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A9: Compounds of the formula W1 , wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A10: Compounds of the formula W1 , wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A11 : Compounds of the formula W1 , wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A12: Compounds of the formula W1 , wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A13: Compounds of the formula W1 , wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A14: Compounds of the formula W1 , wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A15: Compounds of the formula W1 , wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A16: Compounds of the formula W1 , wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A17: Compounds of the formula W1 , wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A18: Compounds of the formula W1 , wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A19: Compounds of the formula W2, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A20: Compounds of the formula W2, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A21 : Compounds of the formula W2, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A22: Compounds of the formula W2, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A23: Compounds of the formula W2, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A24: Compounds of the formula W2, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A25: Compounds of the formula W2, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A26: Compounds of the formula W2, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A27: Compounds of the formula W2, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A28: Compounds of the formula W2, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A29: Compounds of the formula W2, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A30: Compounds of the formula W2, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A31 : Compounds of the formula W2, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A32: Compounds of the formula W2, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A33: Compounds of the formula W2, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A34: Compounds of the formula W2, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A35: Compounds of the formula W2, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A36: Compounds of the formula W2, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A37: Compounds of the formula W3, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A38: Compounds of the formula W3, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A39: Compounds of the formula W3, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A40: Compounds of the formula W3, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A41 : Compounds of the formula W3, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A42: Compounds of the formula W3, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A43: Compounds of the formula W3, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A44: Compounds of the formula W3, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A45: Compounds of the formula W3, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A46: Compounds of the formula W3, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A47: Compounds of the formula W3, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A48: Compounds of the formula W3, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A49: Compounds of the formula W3, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A50: Compounds of the formula W3, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A51 : Compounds of the formula W3, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A52: Compounds of the formula W3, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A53: Compounds of the formula W3, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A54: Compounds of the formula W4, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A55: Compounds of the formula W4, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A56: Compounds of the formula W4, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A57: Compounds of the formula W4, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A58: Compounds of the formula W4, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A59: Compounds of the formula W4, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A60: Compounds of the formula W4, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A61 : Compounds of the formula W4, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A62: Compounds of the formula W4, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A63: Compounds of the formula W4, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A64: Compounds of the formula W4, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A65: Compounds of the formula W4, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A66: Compounds of the formula W4, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A67: Compounds of the formula W4, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A68: Compounds of the formula W4, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A69: Compounds of the formula W4, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A70: Compounds of the formula W4, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A71 : Compounds of the formula W4, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A72: Compounds of the formula W6, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A73: Compounds of the formula W6, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A74: Compounds of the formula W6, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A75: Compounds of the formula W6, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A76: Compounds of the formula W6, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A77: Compounds of the formula W6, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A78: Compounds of the formula W6, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A79: Compounds of the formula W6, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A80: Compounds of the formula W6, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A81 : Compounds of the formula W6, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A82: Compounds of the formula W6, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A83: Compounds of the formula W6, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A84: Compounds of the formula W6, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A85: Compounds of the formula W6, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A86: Compounds of the formula W6, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A87: Compounds of the formula W6, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A88: Compounds of the formula W6, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A89: Compounds of the formula W6, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A90: Compounds of the formula W9, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A91 : Compounds of the formula W9, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A92: Compounds of the formula W9, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A93: Compounds of the formula W9, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A94: Compounds of the formula W9, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A95: Compounds of the formula W9, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A96: Compounds of the formula W9, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A97: Compounds of the formula W9, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A98: Compounds of the formula W9, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A99: Compounds of the formula W3, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A100: Compounds of the formula W9, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A101 : Compounds of the formula W9, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A102: Compounds of the formula W9, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A103: Compounds of the formula W9, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A104: Compounds of the formula W9, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A105: Compounds of the formula W9, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A106: Compounds of the formula W9, wherein R³ is OCH2CI and R¹ and R² are as defined in one row of table A;

Table A107: Compounds of the formula W9, wherein R³ is OCH2-OCH3 and R¹ and

R² are as defined in one row of table A;

Table A108: Compounds of the formula W9, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A109: Compounds of the formula W12, wherein R³ is CH3 and R¹ and R² are as defined in one row of table A;

Table A110: Compounds of the formula W12, wherein R³ is C2H5 and R¹ and R² are as defined in one row of table A;

Table A111: Compounds of the formula W12, wherein R³ is CF3 and R¹ and R² are as defined in one row of table A;

Table A112: Compounds of the formula W12, wherein R³ is CCb and R¹ and R² are as defined in one row of table A;

Table A113: Compounds of the formula W12, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A114: Compounds of the formula W12, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A115: Compounds of the formula W12, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A116: Compounds of the formula W12, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A117: Compounds of the formula W12, wherein R³ is OCH3 and R¹ and R² are as defined in one row of table A;

Table A118: Compounds of the formula W12, wherein R³ is OCF3 and R¹ and R² are as defined in one row of table A;

Table A119: Compounds of the formula W12, wherein R³ is OCCI3 and R¹ and R² are as defined in one row of table A;

Table A120: Compounds of the formula W12, wherein R³ is OCHF2 and R¹ and R² are as defined in one row of table A;

Table A121: Compounds of the formula W12, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A122: Compounds of the formula W12, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A123: Compounds of the formula W12, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A124: Compounds of the formula W12, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A125: Compounds of the formula W12, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A;

Table A126: Compounds of the formula W12, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A; Table A127: Compounds of the formula W13, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A128: Compounds of the formula W13, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A129: Compounds of the formula W13, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A130: Compounds of the formula W13, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A131: Compounds of the formula W13, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A132: Compounds of the formula W13, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A133: Compounds of the formula W13, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A134: Compounds of the formula W13, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A135: Compounds of the formula W13, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A136: Compounds of the formula W13, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A137: Compounds of the formula W13, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A138: Compounds of the formula W13, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A139: Compounds of the formula W13, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A140: Compounds of the formula W13, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A141: Compounds of the formula W13, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A142: Compounds of the formula W13, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A143: Compounds of the formula W13, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A144: Compounds of the formula W13, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A145: Compounds of the formula W14, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A146: Compounds of the formula W14, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A147: Compounds of the formula W14, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A148: Compounds of the formula W14, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A149: Compounds of the formula W14, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A150: Compounds of the formula W14, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A151: Compounds of the formula W14, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A152: Compounds of the formula W14, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A153: Compounds of the formula W14, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A154: Compounds of the formula W14, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A155: Compounds of the formula W14, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A156: Compounds of the formula W14, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A157: Compounds of the formula W14, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A158: Compounds of the formula W14, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A159: Compounds of the formula W14, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A160: Compounds of the formula W14, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A161: Compounds of the formula W14, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A162: Compounds of the formula W14, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A163: Compounds of the formula W16, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A164: Compounds of the formula W16, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A165: Compounds of the formula W16, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A166: Compounds of the formula W16, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A167: Compounds of the formula W16, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A168: Compounds of the formula W16, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A169: Compounds of the formula W16, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A170: Compounds of the formula W16, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A171: Compounds of the formula W16, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A172: Compounds of the formula W16, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A173: Compounds of the formula W16, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A174: Compounds of the formula W16, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A175: Compounds of the formula W16, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A176: Compounds of the formula W16, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A177: Compounds of the formula W16, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A178: Compounds of the formula W16, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A179: Compounds of the formula W16, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A180: Compounds of the formula W16, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A181: Compounds of the formula W19, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A182: Compounds of the formula W19, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A183: Compounds of the formula W19, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A184: Compounds of the formula W19, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A185: Compounds of the formula W19, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A186: Compounds of the formula W19, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A187: Compounds of the formula W19, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A188: Compounds of the formula W19, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A189: Compounds of the formula W19, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A190: Compounds of the formula W19, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A191: Compounds of the formula W19, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A192: Compounds of the formula W19, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A193: Compounds of the formula W19, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A194: Compounds of the formula W19, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A195: Compounds of the formula W19, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A196: Compounds of the formula W19, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A197: Compounds of the formula W19, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A198: Compounds of the formula W19, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A199: Compounds of the formula W22, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A200: Compounds of the formula W22, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A201: Compounds of the formula W22, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A202: Compounds of the formula W22, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A203: Compounds of the formula W22, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A204: Compounds of the formula W22, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A205: Compounds of the formula W22, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A206: Compounds of the formula W22, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A207: Compounds of the formula W22, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A208: Compounds of the formula W22, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A209: Compounds of the formula W22, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A210: Compounds of the formula W22, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A211: Compounds of the formula W22, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A212: Compounds of the formula W22, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A213: Compounds of the formula W22, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A214: Compounds of the formula W22, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A215: Compounds of the formula W22, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A216: Compounds of the formula W22, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A217: Compounds of the formula W23, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A218: Compounds of the formula W23, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A219: Compounds of the formula W23, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A220: Compounds of the formula W23, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A221: Compounds of the formula W23, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A222: Compounds of the formula W23, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A223: Compounds of the formula W23, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A224: Compounds of the formula W23, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A225: Compounds of the formula W23, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A226: Compounds of the formula W23, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A227: Compounds of the formula W23, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A228: Compounds of the formula W23, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A229: Compounds of the formula W23, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A230: Compounds of the formula W23, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A231 : Compounds of the formula W23, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A232: Compounds of the formula W23, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A233: Compounds of the formula W23, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A234: Compounds of the formula W23, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A235: Compounds of the formula W27, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A236: Compounds of the formula W27, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A237: Compounds of the formula W27, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A238: Compounds of the formula W27, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A239: Compounds of the formula W27, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A240: Compounds of the formula W27, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A241: Compounds of the formula W27, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A242: Compounds of the formula W27, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A243: Compounds of the formula W27, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A244: Compounds of the formula W27, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A245: Compounds of the formula W27, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A246: Compounds of the formula W27, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A247: Compounds of the formula W27, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A248: Compounds of the formula W27, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A249: Compounds of the formula W27, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A250: Compounds of the formula W27, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A251: Compounds of the formula W27, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A252: Compounds of the formula W27, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A; Table A253: Compounds of the formula W28, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A254: Compounds of the formula W28, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A255: Compounds of the formula W28, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A256: Compounds of the formula W28, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A257: Compounds of the formula W28, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A258: Compounds of the formula W28, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A259: Compounds of the formula W28, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A260: Compounds of the formula W28, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A261: Compounds of the formula W28, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A262: Compounds of the formula W28, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A263: Compounds of the formula W28, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A264: Compounds of the formula W28, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A265: Compounds of the formula W28, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A266: Compounds of the formula W28, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A267: Compounds of the formula W28, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A268: Compounds of the formula W28, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A269: Compounds of the formula W28, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A270: Compounds of the formula W28, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A271: Compounds of the formula W31 , wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A272: Compounds of the formula W31 , wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A273: Compounds of the formula W31 , wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A274: Compounds of the formula W31 , wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A275: Compounds of the formula W31 , wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A276: Compounds of the formula W31 , wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A277: Compounds of the formula W31 , wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A278: Compounds of the formula W31 , wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A279: Compounds of the formula W31 , wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A280: Compounds of the formula W31 , wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A281: Compounds of the formula W31 , wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A282: Compounds of the formula W31 , wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A283: Compounds of the formula W31 , wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A284: Compounds of the formula W31 , wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A285: Compounds of the formula W31 , wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A286: Compounds of the formula W31 , wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A287: Compounds of the formula W31 , wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A288: Compounds of the formula W31 , wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A289: Compounds of the formula W32, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A290: Compounds of the formula W32, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A291: Compounds of the formula W32, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A292: Compounds of the formula W32, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A293: Compounds of the formula W32, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A294: Compounds of the formula W32, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A295: Compounds of the formula W32, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A296: Compounds of the formula W32, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A297: Compounds of the formula W32, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A298: Compounds of the formula W32, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A299: Compounds of the formula W32, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A300: Compounds of the formula W32, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A301: Compounds of the formula W32, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A302: Compounds of the formula W32, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A303: Compounds of the formula W32, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A304: Compounds of the formula W32, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A305: Compounds of the formula W32, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A306: Compounds of the formula W32, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A307: Compounds of the formula W33, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A308: Compounds of the formula W33, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A309: Compounds of the formula W33, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A310: Compounds of the formula W33, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A311: Compounds of the formula W33, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A312: Compounds of the formula W33, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A313: Compounds of the formula W33, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A314: Compounds of the formula W33, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A315: Compounds of the formula W33, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A316: Compounds of the formula W33, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A317: Compounds of the formula W33, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A318: Compounds of the formula W33, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A319: Compounds of the formula W33, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A320: Compounds of the formula W33, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A321: Compounds of the formula W33, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A322: Compounds of the formula W33, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A323: Compounds of the formula W33, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A324: Compounds of the formula W33, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A325: Compounds of the formula W36, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A326: Compounds of the formula W36, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A327: Compounds of the formula W36, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A328: Compounds of the formula W36, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A329: Compounds of the formula W36, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A330: Compounds of the formula W36, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A331: Compounds of the formula W36, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A332: Compounds of the formula W36, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A333: Compounds of the formula W36, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A334: Compounds of the formula W36, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A335: Compounds of the formula W36, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A336: Compounds of the formula W36, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A337: Compounds of the formula W36, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A338: Compounds of the formula W36, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A339: Compounds of the formula W36, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A340: Compounds of the formula W36, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A341: Compounds of the formula W36, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A342: Compounds of the formula W36, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A343: Compounds of the formula W37, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A344: Compounds of the formula W37, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A345: Compounds of the formula W37, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A346: Compounds of the formula W37, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A347: Compounds of the formula W37, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A348: Compounds of the formula W37, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A349: Compounds of the formula W37, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A350: Compounds of the formula W37, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A351: Compounds of the formula W37, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A352: Compounds of the formula W37, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A353: Compounds of the formula W37, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A354: Compounds of the formula W37, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A355: Compounds of the formula W37, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A356: Compounds of the formula W37, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A357: Compounds of the formula W37, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A358: Compounds of the formula W37, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A359: Compounds of the formula W37, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A360: Compounds of the formula W37, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A361: Compounds of the formula W38, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A362: Compounds of the formula W38, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A363: Compounds of the formula W38, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A364: Compounds of the formula W38, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A365: Compounds of the formula W38, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A366: Compounds of the formula W38, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A367: Compounds of the formula W38, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A368: Compounds of the formula W38, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A369: Compounds of the formula W38, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A370: Compounds of the formula W38, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A371: Compounds of the formula W38, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A372: Compounds of the formula W38, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A373: Compounds of the formula W38, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A374: Compounds of the formula W38, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A375: Compounds of the formula W38, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A376: Compounds of the formula W38, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A377: Compounds of the formula W38, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A378: Compounds of the formula W38, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A; Table A379: Compounds of the formula W40, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A380: Compounds of the formula W40, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A381: Compounds of the formula W40, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A382: Compounds of the formula W40, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A383: Compounds of the formula W40, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A384: Compounds of the formula W40, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A385: Compounds of the formula W40, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A386: Compounds of the formula W40, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A387: Compounds of the formula W40, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A388: Compounds of the formula W40, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A389: Compounds of the formula W40, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A390: Compounds of the formula W40, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A391: Compounds of the formula W40, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A392: Compounds of the formula W40, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A393: Compounds of the formula W40, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A394: Compounds of the formula W40, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A395: Compounds of the formula W40, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A396: Compounds of the formula W40, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A397: Compounds of the formula W41 , wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A398: Compounds of the formula W41 , wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A399: Compounds of the formula W41 , wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A400: Compounds of the formula W41 , wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A401: Compounds of the formula W41 , wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A402: Compounds of the formula W41 , wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A403: Compounds of the formula W41 , wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A404: Compounds of the formula W41 , wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A405: Compounds of the formula W41 , wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A406: Compounds of the formula W41 , wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A407: Compounds of the formula W41 , wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A408: Compounds of the formula W41 , wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A409: Compounds of the formula W41 , wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A410: Compounds of the formula W41 , wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A411: Compounds of the formula W41 , wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A412: Compounds of the formula W41 , wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A413: Compounds of the formula W41 , wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A414: Compounds of the formula W41 , wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A415: Compounds of the formula W44, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A416: Compounds of the formula W44, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A417: Compounds of the formula W44, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A418: Compounds of the formula W44, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A419: Compounds of the formula W44, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A420: Compounds of the formula W44, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A421: Compounds of the formula W44, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A422: Compounds of the formula W44, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A423: Compounds of the formula W44, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A424: Compounds of the formula W44, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A425: Compounds of the formula W44, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A426: Compounds of the formula W44, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A427: Compounds of the formula W44, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A428: Compounds of the formula W44, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A429: Compounds of the formula W44, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A430: Compounds of the formula W44, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A431: Compounds of the formula W44, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A432: Compounds of the formula W44, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A433: Compounds of the formula W45, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A434: Compounds of the formula W45, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A435: Compounds of the formula W45, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A436: Compounds of the formula W45, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A437: Compounds of the formula W45, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A438: Compounds of the formula W45, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A439: Compounds of the formula W45, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A440: Compounds of the formula W45, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A441 : Compounds of the formula W45, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A442: Compounds of the formula W45, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A443: Compounds of the formula W45, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A444: Compounds of the formula W45, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A445: Compounds of the formula W45, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A446: Compounds of the formula W45, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A447: Compounds of the formula W45, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A448: Compounds of the formula W45, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A449: Compounds of the formula W45, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A450: Compounds of the formula W45, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A451: Compounds of the formula W46, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A452: Compounds of the formula W46, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A453: Compounds of the formula W46, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A454: Compounds of the formula W46, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A455: Compounds of the formula W46, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A456: Compounds of the formula W46, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A457: Compounds of the formula W46, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A458: Compounds of the formula W46, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A459: Compounds of the formula W46, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A460: Compounds of the formula W46, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A461: Compounds of the formula W46, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A462: Compounds of the formula W46, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A463: Compounds of the formula W46, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A464: Compounds of the formula W46, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A465: Compounds of the formula W46, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A466: Compounds of the formula W46, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A467: Compounds of the formula W46, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A;

Table A468: Compounds of the formula W46, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A469: Compounds of the formula W51 , wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A470: Compounds of the formula W51 , wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A471: Compounds of the formula W51 , wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A472: Compounds of the formula W51 , wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A473: Compounds of the formula W51 , wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A474: Compounds of the formula W51 , wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A475: Compounds of the formula W51 , wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A476: Compounds of the formula W51 , wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A477: Compounds of the formula W51 , wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A478: Compounds of the formula W51 , wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A479: Compounds of the formula W51 , wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A480: Compounds of the formula W51 , wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A481: Compounds of the formula W51 , wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A482: Compounds of the formula W51 , wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A483: Compounds of the formula W51 , wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A484: Compounds of the formula W51 , wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A485: Compounds of the formula W51 , wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A486: Compounds of the formula W51 , wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A487: Compounds of the formula W55, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A488: Compounds of the formula W55, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A489: Compounds of the formula W55, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A490: Compounds of the formula W55, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A491: Compounds of the formula W55, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A492: Compounds of the formula W55, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A493: Compounds of the formula W55, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A494: Compounds of the formula W55, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A495: Compounds of the formula W55, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A496: Compounds of the formula W55, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A497: Compounds of the formula W55, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A498: Compounds of the formula W55, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A499: Compounds of the formula W55, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A500: Compounds of the formula W55, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A501: Compounds of the formula W55, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A502: Compounds of the formula W55, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A503: Compounds of the formula W55, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A504: Compounds of the formula W55, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A; Table A505: Compounds of the formula W56, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A506: Compounds of the formula W56, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A507: Compounds of the formula W56, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A508: Compounds of the formula W56, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A509: Compounds of the formula W56, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A510: Compounds of the formula W56, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A511: Compounds of the formula W56, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A512: Compounds of the formula W56, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A513: Compounds of the formula W56, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A514: Compounds of the formula W56, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A515: Compounds of the formula W56, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A516: Compounds of the formula W56, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A517: Compounds of the formula W56, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A518: Compounds of the formula W56, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A519: Compounds of the formula W56, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A520: Compounds of the formula W56, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A521: Compounds of the formula W56, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A522: Compounds of the formula W56, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A523: Compounds of the formula W57, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A524: Compounds of the formula W57, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A525: Compounds of the formula W57, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A526: Compounds of the formula W57, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A527: Compounds of the formula W57, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A528: Compounds of the formula W57, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A529: Compounds of the formula W57, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A530: Compounds of the formula W57, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A531: Compounds of the formula W57, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A532: Compounds of the formula W57, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A533: Compounds of the formula W57, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A534: Compounds of the formula W57, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A535: Compounds of the formula W57, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A536: Compounds of the formula W57, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A537: Compounds of the formula W57, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A538: Compounds of the formula W57, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A539: Compounds of the formula W57, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A540: Compounds of the formula W57, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A541: Compounds of the formula W59, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A542: Compounds of the formula W59, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A543: Compounds of the formula W59, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A544: Compounds of the formula W59, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A545: Compounds of the formula W59, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A546: Compounds of the formula W59, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A547: Compounds of the formula W59, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A548: Compounds of the formula W59, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A549: Compounds of the formula W59, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A550: Compounds of the formula W59, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A551: Compounds of the formula W59, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A552: Compounds of the formula W59, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A553: Compounds of the formula W59, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A554: Compounds of the formula W59, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A555: Compounds of the formula W59, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A556: Compounds of the formula W59, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A557: Compounds of the formula W59, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A558: Compounds of the formula W59, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A559: Compounds of the formula W65, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A560: Compounds of the formula W65, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A561: Compounds of the formula W65, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A562: Compounds of the formula W65, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A563: Compounds of the formula W65, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A564: Compounds of the formula W65, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A565: Compounds of the formula W65, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A566: Compounds of the formula W65, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A567: Compounds of the formula W65, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A568: Compounds of the formula W65, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A569: Compounds of the formula W65, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A570: Compounds of the formula W65, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A571: Compounds of the formula W65, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A572: Compounds of the formula W65, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A573: Compounds of the formula W65, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A574: Compounds of the formula W65, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A575: Compounds of the formula W65, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A576: Compounds of the formula W65, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A577: Compounds of the formula W66, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A578: Compounds of the formula W66, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A579: Compounds of the formula W66, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A580: Compounds of the formula W66, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A581: Compounds of the formula W66, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A582: Compounds of the formula W66, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A583: Compounds of the formula W66, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A584: Compounds of the formula W66, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A585: Compounds of the formula W66, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A586: Compounds of the formula W66, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A587: Compounds of the formula W66, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A588: Compounds of the formula W66, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A589: Compounds of the formula W66, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A590: Compounds of the formula W66, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A591: Compounds of the formula W66, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A592: Compounds of the formula W66, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A593: Compounds of the formula W66, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A594: Compounds of the formula W66, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A595: Compounds of the formula W67, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A596: Compounds of the formula W67, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A597: Compounds of the formula W67, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A598: Compounds of the formula W67, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A599: Compounds of the formula W67, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A600: Compounds of the formula W67, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A601: Compounds of the formula W67, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A602: Compounds of the formula W67, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A603: Compounds of the formula W67, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A604: Compounds of the formula W67, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A605: Compounds of the formula W67, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A606: Compounds of the formula W67, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A607: Compounds of the formula W67, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A608: Compounds of the formula W67, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A609: Compounds of the formula W67, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A610: Compounds of the formula W67, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A611: Compounds of the formula W67, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A612: Compounds of the formula W67, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A613: Compounds of the formula W68, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A614: Compounds of the formula W68, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A615: Compounds of the formula W68, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A616: Compounds of the formula W68, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A617: Compounds of the formula W68, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A618: Compounds of the formula W68, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A619: Compounds of the formula W68, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A620: Compounds of the formula W68, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A621: Compounds of the formula W68, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A622: Compounds of the formula W68, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A623: Compounds of the formula W68, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A624: Compounds of the formula W68, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A625: Compounds of the formula W68, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A626: Compounds of the formula W68, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A627: Compounds of the formula W68, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A628: Compounds of the formula W68, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A629: Compounds of the formula W68, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A630: Compounds of the formula W68, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A; Table A631: Compounds of the formula W69, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A632: Compounds of the formula W69, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A633: Compounds of the formula W69, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A634: Compounds of the formula W69, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A635: Compounds of the formula W69, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A636: Compounds of the formula W69, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A637: Compounds of the formula W69, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A638: Compounds of the formula W69, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A639: Compounds of the formula W69, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A640: Compounds of the formula W69, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A641: Compounds of the formula W69, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A642: Compounds of the formula W69, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A643: Compounds of the formula W69, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A644: Compounds of the formula W69, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A645: Compounds of the formula W69, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A646: Compounds of the formula W69, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A647: Compounds of the formula W69, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A648: Compounds of the formula W69, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A649: Compounds of the formula W70, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A650: Compounds of the formula W70, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A651 : Compounds of the formula W70, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A652: Compounds of the formula W70, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A653: Compounds of the formula W70, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A654: Compounds of the formula W70, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A655: Compounds of the formula W70, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A656: Compounds of the formula W70, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A657: Compounds of the formula W70, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A658: Compounds of the formula W70, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A659: Compounds of the formula W70, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A660: Compounds of the formula W70, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A661: Compounds of the formula W70, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A662: Compounds of the formula W70, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A663: Compounds of the formula W70, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A664: Compounds of the formula W70, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A665: Compounds of the formula W70, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A666: Compounds of the formula W70, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A667: Compounds of the formula W71 , wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A668: Compounds of the formula W71 , wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A669: Compounds of the formula W71 , wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A670: Compounds of the formula W71 , wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A671: Compounds of the formula W71 , wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A672: Compounds of the formula W71 , wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A673: Compounds of the formula W71 , wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A674: Compounds of the formula W71 , wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A675: Compounds of the formula W71 , wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A676: Compounds of the formula W71 , wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A677: Compounds of the formula W71 , wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A678: Compounds of the formula W71 , wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A679: Compounds of the formula W71 , wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A680: Compounds of the formula W71 , wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A681: Compounds of the formula W71 , wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A682: Compounds of the formula W71 , wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A683: Compounds of the formula W71 , wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A684: Compounds of the formula W71 , wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A685: Compounds of the formula W72, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A686: Compounds of the formula W72, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A687: Compounds of the formula W72, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A688: Compounds of the formula W72, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A689: Compounds of the formula W72, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A690: Compounds of the formula W72, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A691: Compounds of the formula W72, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A692: Compounds of the formula W72, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A693: Compounds of the formula W72, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A694: Compounds of the formula W72, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A695: Compounds of the formula W72, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A696: Compounds of the formula W72, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A697: Compounds of the formula W72, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A698: Compounds of the formula W72, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A699: Compounds of the formula W72, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A700: Compounds of the formula W72, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A701: Compounds of the formula W72, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A702: Compounds of the formula W72, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A703: Compounds of the formula W73, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A704: Compounds of the formula W73, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A705: Compounds of the formula W73, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A706: Compounds of the formula W73, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A707: Compounds of the formula W73, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A708: Compounds of the formula W73, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A709: Compounds of the formula W73, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A710: Compounds of the formula W73, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A711: Compounds of the formula W73, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A712: Compounds of the formula W73, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A713: Compounds of the formula W73, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A714: Compounds of the formula W73, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A715: Compounds of the formula W73, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A716: Compounds of the formula W73, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A717: Compounds of the formula W73, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A718: Compounds of the formula W73, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A719: Compounds of the formula W73, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A720: Compounds of the formula W73, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A721: Compounds of the formula W74, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A722: Compounds of the formula W74, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A723: Compounds of the formula W74, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A724: Compounds of the formula W74, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A725: Compounds of the formula W74, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A726: Compounds of the formula W74, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A727: Compounds of the formula W74, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A728: Compounds of the formula W74, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A729: Compounds of the formula W74, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A730: Compounds of the formula W74, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A731: Compounds of the formula W74, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A732: Compounds of the formula W74, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A733: Compounds of the formula W74, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A734: Compounds of the formula W74, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A735: Compounds of the formula W74, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A736: Compounds of the formula W74, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A737: Compounds of the formula W74, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A738: Compounds of the formula W74, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A739: Compounds of the formula W75, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A740: Compounds of the formula W75, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A741: Compounds of the formula W75, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A742: Compounds of the formula W75, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A743: Compounds of the formula W75, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A744: Compounds of the formula W75, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A745: Compounds of the formula W75, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A746: Compounds of the formula W75, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A747: Compounds of the formula W75, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A748: Compounds of the formula W75, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A749: Compounds of the formula W75, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A750: Compounds of the formula W75, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A751: Compounds of the formula W75, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A752: Compounds of the formula W75, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A753: Compounds of the formula W75, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A754: Compounds of the formula W75, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A755: Compounds of the formula W75, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A756: Compounds of the formula W75, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A; Table A757: Compounds of the formula W76, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A758: Compounds of the formula W76, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A759: Compounds of the formula W76, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A760: Compounds of the formula W76, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A761: Compounds of the formula W76, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A762: Compounds of the formula W76, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A763: Compounds of the formula W76, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A764: Compounds of the formula W76, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A765: Compounds of the formula W76, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A766: Compounds of the formula W76, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A767: Compounds of the formula W76, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A768: Compounds of the formula W76, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A769: Compounds of the formula W76, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A770: Compounds of the formula W76, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A771: Compounds of the formula W76, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A772: Compounds of the formula W76, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A773: Compounds of the formula W76, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A774: Compounds of the formula W76, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A775: Compounds of the formula W77, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A776: Compounds of the formula W77, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A777: Compounds of the formula W77, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A778: Compounds of the formula W77, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A779: Compounds of the formula W77, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A780: Compounds of the formula W77, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A781: Compounds of the formula W77, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A782: Compounds of the formula W77, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A783: Compounds of the formula W77, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A784: Compounds of the formula W77, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A785: Compounds of the formula W77, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A786: Compounds of the formula W77, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A787: Compounds of the formula W77, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A788: Compounds of the formula W77, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A789: Compounds of the formula W77, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A790: Compounds of the formula W77, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A791: Compounds of the formula W77, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A792: Compounds of the formula W77, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A793: Compounds of the formula W80, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A794: Compounds of the formula W80, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A795: Compounds of the formula W80, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A796: Compounds of the formula W80, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A797: Compounds of the formula W80, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A798: Compounds of the formula W80, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A799: Compounds of the formula W80, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A800: Compounds of the formula W80, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A801: Compounds of the formula W80, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A802: Compounds of the formula W80, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A803: Compounds of the formula W80, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A804: Compounds of the formula W80, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A805: Compounds of the formula W80, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A806: Compounds of the formula W80, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A807: Compounds of the formula W80, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A808: Compounds of the formula W80, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A809: Compounds of the formula W80, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A810: Compounds of the formula W80, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A811: Compounds of the formula W81 , wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A812: Compounds of the formula W81 , wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A813: Compounds of the formula W81 , wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A814: Compounds of the formula W81 , wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A815: Compounds of the formula W81 , wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A816: Compounds of the formula W81 , wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A817: Compounds of the formula W81 , wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A818: Compounds of the formula W81 , wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A819: Compounds of the formula W81 , wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A820: Compounds of the formula W81 , wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A821: Compounds of the formula W81 , wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A822: Compounds of the formula W81 , wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A823: Compounds of the formula W81 , wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A824: Compounds of the formula W81 , wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A825: Compounds of the formula W81 , wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A826: Compounds of the formula W81 , wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A827: Compounds of the formula W81 , wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A828: Compounds of the formula W81 , wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A829: Compounds of the formula W82, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A830: Compounds of the formula W82, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A831: Compounds of the formula W82, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A832: Compounds of the formula W82, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A833: Compounds of the formula W82, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A834: Compounds of the formula W82, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A835: Compounds of the formula W82, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A836: Compounds of the formula W82, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A837: Compounds of the formula W82, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A838: Compounds of the formula W82, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A839: Compounds of the formula W82, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A840: Compounds of the formula W82, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A841: Compounds of the formula W82, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A842: Compounds of the formula W82, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A843: Compounds of the formula W82, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A844: Compounds of the formula W82, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A845: Compounds of the formula W82, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A846: Compounds of the formula W82, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A847: Compounds of the formula W85, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A848: Compounds of the formula W85, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A849: Compounds of the formula W85, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A850: Compounds of the formula W85, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A851: Compounds of the formula W85, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A852: Compounds of the formula W85, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A853: Compounds of the formula W85, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A854: Compounds of the formula W85, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A855: Compounds of the formula W85, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A856: Compounds of the formula W85, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A857: Compounds of the formula W85, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A858: Compounds of the formula W85, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A859: Compounds of the formula W85, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A860: Compounds of the formula W85, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A861 : Compounds of the formula W85, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A862: Compounds of the formula W85, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A863: Compounds of the formula W85, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A864: Compounds of the formula W85, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A865: Compounds of the formula W86, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A866: Compounds of the formula W86, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A867: Compounds of the formula W86, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A868: Compounds of the formula W86, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A869: Compounds of the formula W86, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A870: Compounds of the formula W86, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A871: Compounds of the formula W86, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A872: Compounds of the formula W86, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A873: Compounds of the formula W86, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A874: Compounds of the formula W86, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A875: Compounds of the formula W86, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A876: Compounds of the formula W86, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A877: Compounds of the formula W86, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A878: Compounds of the formula W86, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A879: Compounds of the formula W86, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A880: Compounds of the formula W86, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A881: Compounds of the formula W86, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A882: Compounds of the formula W86, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A; Table A883: Compounds of the formula W87, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A884: Compounds of the formula W87, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A885: Compounds of the formula W87, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A886: Compounds of the formula W87, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A887: Compounds of the formula W87, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A888: Compounds of the formula W87, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A889: Compounds of the formula W87, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A890: Compounds of the formula W87, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A891: Compounds of the formula W87, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A892: Compounds of the formula W87, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A893: Compounds of the formula W87, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A894: Compounds of the formula W87, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A895: Compounds of the formula W87, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A896: Compounds of the formula W87, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A897: Compounds of the formula W87, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A898: Compounds of the formula W87, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A899: Compounds of the formula W87, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A900: Compounds of the formula W87, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A901: Compounds of the formula W90, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A902: Compounds of the formula W90, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A903: Compounds of the formula W90, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A904: Compounds of the formula W90, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A905: Compounds of the formula W90, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A906: Compounds of the formula W90, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A907: Compounds of the formula W90, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A908: Compounds of the formula W90, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A909: Compounds of the formula W90, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A910: Compounds of the formula W90, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A911: Compounds of the formula W90, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A912: Compounds of the formula W90, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A913: Compounds of the formula W90, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A914: Compounds of the formula W90, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A915: Compounds of the formula W90, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A916: Compounds of the formula W90, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A917: Compounds of the formula W90, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A918: Compounds of the formula W90, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A919: Compounds of the formula W91 , wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A920: Compounds of the formula W91 , wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A921: Compounds of the formula W91 , wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A922: Compounds of the formula W91 , wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A923: Compounds of the formula W91 , wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A924: Compounds of the formula W91 , wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A925: Compounds of the formula W91 , wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A926: Compounds of the formula W91 , wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A927: Compounds of the formula W91 , wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A928: Compounds of the formula W91 , wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A929: Compounds of the formula W91 , wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A930: Compounds of the formula W91 , wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A931: Compounds of the formula W91 , wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A932: Compounds of the formula W91 , wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A933: Compounds of the formula W91 , wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A934: Compounds of the formula W91 , wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A935: Compounds of the formula W91 , wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A936: Compounds of the formula W91 , wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A937: Compounds of the formula W92, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A938: Compounds of the formula W92, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A939: Compounds of the formula W92, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A940: Compounds of the formula W92, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A941: Compounds of the formula W92, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A942: Compounds of the formula W92, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A943: Compounds of the formula W92, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A944: Compounds of the formula W92, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A945: Compounds of the formula W92, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A946: Compounds of the formula W92, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A947: Compounds of the formula W92, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A948: Compounds of the formula W92, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A949: Compounds of the formula W92, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A950: Compounds of the formula W92, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A951: Compounds of the formula W92, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A952: Compounds of the formula W92, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A953: Compounds of the formula W92, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A954: Compounds of the formula W92, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A955: Compounds of the formula W93, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A956: Compounds of the formula W93, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A957: Compounds of the formula W93, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A958: Compounds of the formula W93, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A959: Compounds of the formula W93, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A960: Compounds of the formula W93, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A961: Compounds of the formula W93, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A962: Compounds of the formula W93, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A963: Compounds of the formula W93, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A964: Compounds of the formula W93, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A965: Compounds of the formula W93, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A966: Compounds of the formula W93, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A967: Compounds of the formula W93, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A968: Compounds of the formula W93, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A969: Compounds of the formula W93, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A970: Compounds of the formula W93, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A971: Compounds of the formula W93, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A972: Compounds of the formula W93, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A973: Compounds of the formula W94, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A974: Compounds of the formula W94, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A975: Compounds of the formula W94, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A976: Compounds of the formula W94, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A977: Compounds of the formula W94, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A978: Compounds of the formula W94, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A979: Compounds of the formula W94, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A980: Compounds of the formula W94, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A981: Compounds of the formula W94, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A982: Compounds of the formula W94, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A983: Compounds of the formula W94, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A984: Compounds of the formula W94, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A985: Compounds of the formula W94, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A986: Compounds of the formula W94, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A987: Compounds of the formula W94, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A988: Compounds of the formula W94, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A989: Compounds of the formula W94, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A990: Compounds of the formula W94, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A991: Compounds of the formula W96, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A992: Compounds of the formula W96, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A993: Compounds of the formula W96, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A994: Compounds of the formula W96, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A995: Compounds of the formula W96, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A996: Compounds of the formula W96, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A997: Compounds of the formula W96, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A998: Compounds of the formula W96, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A999: Compounds of the formula W96, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1000: Compounds of the formula W96, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1001: Compounds of the formula W96, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1002: Compounds of the formula W96, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A1003: Compounds of the formula W96, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1004: Compounds of the formula W96, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1005: Compounds of the formula W96, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A1006: Compounds of the formula W96, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1007: Compounds of the formula W96, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1008: Compounds of the formula W96, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A; Table A1009: Compounds of the formula W97, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1010: Compounds of the formula W97, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1011 : Compounds of the formula W97, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1012: Compounds of the formula W97, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1013: Compounds of the formula W97, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1014: Compounds of the formula W97, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1015: Compounds of the formula W97, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1016: Compounds of the formula W97, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1017: Compounds of the formula W97, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1018: Compounds of the formula W97, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1019: Compounds of the formula W97, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1020: Compounds of the formula W97, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1021 : Compounds of the formula W97, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1022: Compounds of the formula W97, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1023: Compounds of the formula W97, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A1024: Compounds of the formula W97, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1025: Compounds of the formula W97, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1026: Compounds of the formula W97, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A; Table A1027: Compounds of the formula W98, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A1028: Compounds of the formula W98, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A1029: Compounds of the formula W98, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1030: Compounds of the formula W98, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1031 : Compounds of the formula W98, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1032: Compounds of the formula W98, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1033: Compounds of the formula W98, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A1034: Compounds of the formula W98, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1035: Compounds of the formula W98, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1036: Compounds of the formula W98, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1037: Compounds of the formula W98, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1038: Compounds of the formula W98, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A1039: Compounds of the formula W98, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1040: Compounds of the formula W98, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1041 : Compounds of the formula W98, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1042: Compounds of the formula W98, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1043: Compounds of the formula W98, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A;

Table A1044: Compounds of the formula W98, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A1045: Compounds of the formula W106, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1046: Compounds of the formula W106, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1047: Compounds of the formula W106, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1048: Compounds of the formula W106, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1049: Compounds of the formula W106, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1050: Compounds of the formula W106, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1051 : Compounds of the formula W106, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1052: Compounds of the formula W106, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1053: Compounds of the formula W106, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1054: Compounds of the formula W106, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1055: Compounds of the formula W106, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1056: Compounds of the formula W106, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1057: Compounds of the formula W106, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1058: Compounds of the formula W106, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1059: Compounds of the formula W106, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A1060: Compounds of the formula W106, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1061 : Compounds of the formula W106, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1062: Compounds of the formula W106, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1063: Compounds of the formula W107, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1064: Compounds of the formula W107, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A1065: Compounds of the formula W107, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A1066: Compounds of the formula W107, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1067: Compounds of the formula W107, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1068: Compounds of the formula W107, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1069: Compounds of the formula W107, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A1070: Compounds of the formula W107, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1071 : Compounds of the formula W107, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1072: Compounds of the formula W107, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1073: Compounds of the formula W107, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1074: Compounds of the formula W107, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1075: Compounds of the formula W107, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1076: Compounds of the formula W107, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1077: Compounds of the formula W107, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1078: Compounds of the formula W107, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1079: Compounds of the formula W107, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1080: Compounds of the formula W107, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A;

Table A1081 : Compounds of the formula W108, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A1082: Compounds of the formula W108, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1083: Compounds of the formula W108, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1084: Compounds of the formula W108, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1085: Compounds of the formula W108, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1086: Compounds of the formula W108, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A1087: Compounds of the formula W108, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1088: Compounds of the formula W108, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1089: Compounds of the formula W108, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1090: Compounds of the formula W108, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1091 : Compounds of the formula W108, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1092: Compounds of the formula W108, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1093: Compounds of the formula W108, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1094: Compounds of the formula W108, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1095: Compounds of the formula W108, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1096: Compounds of the formula W108, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1097: Compounds of the formula W108, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1098: Compounds of the formula W108, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1099: Compounds of the formula W1 12, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1100: Compounds of the formula W1 12, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1101 : Compounds of the formula W1 12, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A1102: Compounds of the formula W1 12, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1103: Compounds of the formula W1 12, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1104: Compounds of the formula W1 12, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1105: Compounds of the formula W1 12, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1106: Compounds of the formula W1 12, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1107: Compounds of the formula W1 12, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1108: Compounds of the formula W1 12, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1109: Compounds of the formula W1 12, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A11 10: Compounds of the formula W1 12, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A11 11 : Compounds of the formula W1 12, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A11 12: Compounds of the formula W1 12, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A11 13: Compounds of the formula W1 12, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A11 14: Compounds of the formula W1 12, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A11 15: Compounds of the formula W1 12, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A11 16: Compounds of the formula W1 12, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A11 17: Compounds of the formula W1 13, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A11 18: Compounds of the formula W1 13, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A1119: Compounds of the formula W113, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1120: Compounds of the formula W1 13, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1121 : Compounds of the formula W1 13, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1122: Compounds of the formula W1 13, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A1123: Compounds of the formula W1 13, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A1124: Compounds of the formula W1 13, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1125: Compounds of the formula W1 13, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1126: Compounds of the formula W1 13, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1127: Compounds of the formula W1 13, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1128: Compounds of the formula W1 13, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A1129: Compounds of the formula W1 13, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1130: Compounds of the formula W1 13, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1131 : Compounds of the formula W1 13, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1132: Compounds of the formula W1 13, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1133: Compounds of the formula W1 13, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1134: Compounds of the formula W1 13, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1135: Compounds of the formula W1 16, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1136: Compounds of the formula W1 16, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1137: Compounds of the formula W1 16, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1138: Compounds of the formula W1 16, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1139: Compounds of the formula W1 16, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1140: Compounds of the formula W116, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1141 : Compounds of the formula W1 16, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1142: Compounds of the formula W1 16, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1143: Compounds of the formula W1 16, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1144: Compounds of the formula W1 16, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1145: Compounds of the formula W1 16, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1146: Compounds of the formula W1 16, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1147: Compounds of the formula W1 16, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1148: Compounds of the formula W1 16, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1149: Compounds of the formula W1 16, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A1150: Compounds of the formula W1 16, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1151 : Compounds of the formula W1 16, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1152: Compounds of the formula W1 16, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1153: Compounds of the formula W1 17, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A1154: Compounds of the formula W1 17, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A1155: Compounds of the formula W1 17, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1156: Compounds of the formula W1 17, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1157: Compounds of the formula W1 17, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1158: Compounds of the formula W1 17, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1159: Compounds of the formula W1 17, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A1160: Compounds of the formula W1 17, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1161 : Compounds of the formula W117, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1162: Compounds of the formula W1 17, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1163: Compounds of the formula W1 17, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1164: Compounds of the formula W1 17, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A1165: Compounds of the formula W1 17, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1166: Compounds of the formula W1 17, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1167: Compounds of the formula W1 17, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1168: Compounds of the formula W1 17, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1169: Compounds of the formula W1 17, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A;

Table A1170: Compounds of the formula W1 17, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A1171 : Compounds of the formula W1 18, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1172: Compounds of the formula W1 18, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1173: Compounds of the formula W1 18, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1174: Compounds of the formula W1 18, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1175: Compounds of the formula W1 18, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1176: Compounds of the formula W1 18, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1177: Compounds of the formula W1 18, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1178: Compounds of the formula W1 18, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1179: Compounds of the formula W1 18, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1180: Compounds of the formula W1 18, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1181 : Compounds of the formula W1 18, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1182: Compounds of the formula W118, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1183: Compounds of the formula W1 18, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1184: Compounds of the formula W1 18, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1185: Compounds of the formula W1 18, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A1186: Compounds of the formula W1 18, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1187: Compounds of the formula W1 18, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1188: Compounds of the formula W1 18, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1189: Compounds of the formula W1 19, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1190: Compounds of the formula W1 19, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A1191 : Compounds of the formula W1 19, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A1192: Compounds of the formula W1 19, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1193: Compounds of the formula W1 19, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1194: Compounds of the formula W1 19, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1195: Compounds of the formula W1 19, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A1196: Compounds of the formula W1 19, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1197: Compounds of the formula W1 19, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1198: Compounds of the formula W1 19, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1199: Compounds of the formula W1 19, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1200: Compounds of the formula W119, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1201 : Compounds of the formula W1 19, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1202: Compounds of the formula W1 19, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1203: Compounds of the formula W119, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1204: Compounds of the formula W1 19, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1205: Compounds of the formula W1 19, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1206: Compounds of the formula W1 19, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A;

Table A1207: Compounds of the formula W120, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A1208: Compounds of the formula W120, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1209: Compounds of the formula W120, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1210: Compounds of the formula W120, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1211 : Compounds of the formula W120, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1212: Compounds of the formula W120, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A1213: Compounds of the formula W120, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1214: Compounds of the formula W120, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1215: Compounds of the formula W120, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1216: Compounds of the formula W120, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1217: Compounds of the formula W120, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1218: Compounds of the formula W120, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1219: Compounds of the formula W120, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1220: Compounds of the formula W120, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1221 : Compounds of the formula W120, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1222: Compounds of the formula W120, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1223: Compounds of the formula W120, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1224: Compounds of the formula W120, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1225: Compounds of the formula W122, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1226: Compounds of the formula W122, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1227: Compounds of the formula W122, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A1228: Compounds of the formula W122, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1229: Compounds of the formula W122, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1230: Compounds of the formula W122, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1231 : Compounds of the formula W122, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1232: Compounds of the formula W122, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1233: Compounds of the formula W122, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1234: Compounds of the formula W122, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1235: Compounds of the formula W122, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1236: Compounds of the formula W122, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1237: Compounds of the formula W122, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1238: Compounds of the formula W122, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1239: Compounds of the formula W122, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1240: Compounds of the formula W122, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1241 : Compounds of the formula W122, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1242: Compounds of the formula W122, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1243: Compounds of the formula W123, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A1244: Compounds of the formula W123, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A1245: Compounds of the formula W123, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1246: Compounds of the formula W123, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1247: Compounds of the formula W123, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1248: Compounds of the formula W123, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A1249: Compounds of the formula W123, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A1250: Compounds of the formula W123, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1251 : Compounds of the formula W123, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1252: Compounds of the formula W123, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1253: Compounds of the formula W123, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1254: Compounds of the formula W123, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A1255: Compounds of the formula W123, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1256: Compounds of the formula W123, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1257: Compounds of the formula W123, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1258: Compounds of the formula W123, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1259: Compounds of the formula W123, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1260: Compounds of the formula W123, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1261 : Compounds of the formula W124, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1262: Compounds of the formula W124, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1263: Compounds of the formula W124, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1264: Compounds of the formula W124, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1265: Compounds of the formula W124, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1266: Compounds of the formula W124, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1267: Compounds of the formula W124, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1268: Compounds of the formula W124, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1269: Compounds of the formula W124, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1270: Compounds of the formula W124, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1271 : Compounds of the formula W124, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1272: Compounds of the formula W124, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1273: Compounds of the formula W124, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1274: Compounds of the formula W124, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1275: Compounds of the formula W124, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A1276: Compounds of the formula W124, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1277: Compounds of the formula W124, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1278: Compounds of the formula W124, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1279: Compounds of the formula W125, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A1280: Compounds of the formula W125, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A1281 : Compounds of the formula W125, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1282: Compounds of the formula W125, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1283: Compounds of the formula W125, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1284: Compounds of the formula W125, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1285: Compounds of the formula W125, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A1286: Compounds of the formula W125, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1287: Compounds of the formula W125, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1288: Compounds of the formula W125, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1289: Compounds of the formula W125, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1290: Compounds of the formula W125, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A1291 : Compounds of the formula W125, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1292: Compounds of the formula W125, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1293: Compounds of the formula W125, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1294: Compounds of the formula W125, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1295: Compounds of the formula W125, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A;

Table A1296: Compounds of the formula W125, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A1297: Compounds of the formula W126, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1298: Compounds of the formula W126, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1299: Compounds of the formula W126, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1300: Compounds of the formula W126, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1301 : Compounds of the formula W126, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1302: Compounds of the formula W126, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1303: Compounds of the formula W126, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1304: Compounds of the formula W126, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1305: Compounds of the formula W126, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1306: Compounds of the formula W126, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1307: Compounds of the formula W126, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1308: Compounds of the formula W126, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1309: Compounds of the formula W126, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1310: Compounds of the formula W126, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1311 : Compounds of the formula W126, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A1312: Compounds of the formula W126, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1313: Compounds of the formula W126, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1314: Compounds of the formula W126, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1315: Compounds of the formula W128, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1316: Compounds of the formula W128, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A1317: Compounds of the formula W128, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A1318: Compounds of the formula W128, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1319: Compounds of the formula W128, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1320: Compounds of the formula W128, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1321 : Compounds of the formula W128, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A1322: Compounds of the formula W128, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1323: Compounds of the formula W128, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1324: Compounds of the formula W128, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1325: Compounds of the formula W128, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1326: Compounds of the formula W128, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1327: Compounds of the formula W128, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1328: Compounds of the formula W128, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1329: Compounds of the formula W128, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1330: Compounds of the formula W128, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1331 : Compounds of the formula W128, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1332: Compounds of the formula W128, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A;

Table A1333: Compounds of the formula W129, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A1334: Compounds of the formula W129, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1335: Compounds of the formula W129, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1336: Compounds of the formula W129, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1337: Compounds of the formula W129, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1338: Compounds of the formula W129, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A1339: Compounds of the formula W129, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1340: Compounds of the formula W129, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1341 : Compounds of the formula W129, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1342: Compounds of the formula W129, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1343: Compounds of the formula W129, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1344: Compounds of the formula W129, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1345: Compounds of the formula W129, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1346: Compounds of the formula W129, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1347: Compounds of the formula W129, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1348: Compounds of the formula W129, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1349: Compounds of the formula W129, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1350: Compounds of the formula W129, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1351 : Compounds of the formula W130, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1352: Compounds of the formula W130, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1353: Compounds of the formula W130, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A1354: Compounds of the formula W130, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1355: Compounds of the formula W130, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1356: Compounds of the formula W130, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1357: Compounds of the formula W130, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1358: Compounds of the formula W130, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1359: Compounds of the formula W130, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1360: Compounds of the formula W130, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1361 : Compounds of the formula W130, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1362: Compounds of the formula W130, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1363: Compounds of the formula W130, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1364: Compounds of the formula W130, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1365: Compounds of the formula W130, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1366: Compounds of the formula W130, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1367: Compounds of the formula W130, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1368: Compounds of the formula W130, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1369: Compounds of the formula W131 , wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A1370: Compounds of the formula W131 , wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A1371 : Compounds of the formula W131 , wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1372: Compounds of the formula W131 , wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1373: Compounds of the formula W131 , wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1374: Compounds of the formula W131 , wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A1375: Compounds of the formula W131 , wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A1376: Compounds of the formula W131 , wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1377: Compounds of the formula W131 , wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1378: Compounds of the formula W131 , wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1379: Compounds of the formula W131 , wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1380: Compounds of the formula W131 , wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A1381 : Compounds of the formula W131 , wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1382: Compounds of the formula W131 , wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1383: Compounds of the formula W131 , wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1384: Compounds of the formula W131 , wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1385: Compounds of the formula W131 , wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1386: Compounds of the formula W131 , wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1387: Compounds of the formula W134, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1388: Compounds of the formula W134, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1389: Compounds of the formula W134, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1390: Compounds of the formula W134, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1391 : Compounds of the formula W134, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1392: Compounds of the formula W134, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1393: Compounds of the formula W134, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1394: Compounds of the formula W134, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1395: Compounds of the formula W134, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1396: Compounds of the formula W134, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1397: Compounds of the formula W134, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1398: Compounds of the formula W134, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1399: Compounds of the formula W134, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1400: Compounds of the formula W134, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1401 : Compounds of the formula W134, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A1402: Compounds of the formula W134, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1403: Compounds of the formula W134, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1404: Compounds of the formula W134, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1405: Compounds of the formula W135, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A1406: Compounds of the formula W135, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A1407: Compounds of the formula W135, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1408: Compounds of the formula W135, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1409: Compounds of the formula W135, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1410: Compounds of the formula W135, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1411 : Compounds of the formula W135, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A1412: Compounds of the formula W135, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1413: Compounds of the formula W135, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1414: Compounds of the formula W135, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1415: Compounds of the formula W135, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1416: Compounds of the formula W135, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A1417: Compounds of the formula W135, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1418: Compounds of the formula W135, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1419: Compounds of the formula W135, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1420: Compounds of the formula W135, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1421 : Compounds of the formula W135, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A;

Table A1422: Compounds of the formula W135, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A1423: Compounds of the formula W136, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1424: Compounds of the formula W136, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1425: Compounds of the formula W136, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1426: Compounds of the formula W136, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1427: Compounds of the formula W136, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1428: Compounds of the formula W136, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1429: Compounds of the formula W136, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1430: Compounds of the formula W136, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1431 : Compounds of the formula W136, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1432: Compounds of the formula W136, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1433: Compounds of the formula W136, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1434: Compounds of the formula W136, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1435: Compounds of the formula W136, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1436: Compounds of the formula W136, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1437: Compounds of the formula W136, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A1438: Compounds of the formula W136, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1439: Compounds of the formula W136, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1440: Compounds of the formula W136, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1441 : Compounds of the formula W137, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1442: Compounds of the formula W137, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A1443: Compounds of the formula W137, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A1444: Compounds of the formula W137, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1445: Compounds of the formula W137, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1446: Compounds of the formula W137, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1447: Compounds of the formula W137, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A1448: Compounds of the formula W137, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1449: Compounds of the formula W137, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1450: Compounds of the formula W137, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1451 : Compounds of the formula W137, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1452: Compounds of the formula W137, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1453: Compounds of the formula W137, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1454: Compounds of the formula W137, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1455: Compounds of the formula W137, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1456: Compounds of the formula W137, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1457: Compounds of the formula W137, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1458: Compounds of the formula W137, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A;

Table A1459: Compounds of the formula W138, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A1460: Compounds of the formula W138, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1461 : Compounds of the formula W138, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1462: Compounds of the formula W138, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1463: Compounds of the formula W138, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1464: Compounds of the formula W138, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A1465: Compounds of the formula W138, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1466: Compounds of the formula W138, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1467: Compounds of the formula W138, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1468: Compounds of the formula W138, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1469: Compounds of the formula W138, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1470: Compounds of the formula W138, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1471 : Compounds of the formula W138, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1472: Compounds of the formula W138, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1473: Compounds of the formula W138, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1474: Compounds of the formula W138, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1475: Compounds of the formula W138, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1476: Compounds of the formula W138, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1477: Compounds of the formula W140, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1478: Compounds of the formula W140, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1479: Compounds of the formula W140, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A1480: Compounds of the formula W140, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1481 : Compounds of the formula W140, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1482: Compounds of the formula W140, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1483: Compounds of the formula W140, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1484: Compounds of the formula W140, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1485: Compounds of the formula W140, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1486: Compounds of the formula W140, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1487: Compounds of the formula W140, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1488: Compounds of the formula W140, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1489: Compounds of the formula W140, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1490: Compounds of the formula W140, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1491 : Compounds of the formula W140, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1492: Compounds of the formula W140, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1493: Compounds of the formula W140, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1494: Compounds of the formula W140, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1495: Compounds of the formula W141 , wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A1496: Compounds of the formula W141 , wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A1497: Compounds of the formula W141 , wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1498: Compounds of the formula W141 , wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1499: Compounds of the formula W141 , wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1500: Compounds of the formula W141 , wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A1501 : Compounds of the formula W141 , wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A1502: Compounds of the formula W141 , wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1503: Compounds of the formula W141 , wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1504: Compounds of the formula W141 , wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1505: Compounds of the formula W141 , wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1506: Compounds of the formula W141 , wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A1507: Compounds of the formula W141 , wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1508: Compounds of the formula W141 , wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1509: Compounds of the formula W141 , wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1510: Compounds of the formula W141 , wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1511 : Compounds of the formula W141 , wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1512: Compounds of the formula W141 , wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1513: Compounds of the formula W142, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1514: Compounds of the formula W142, wherein R³ is C2H5 and R¹ and R² are as defined in one row of table A; Table A1515: Compounds of the formula W142, wherein R³ is CF3 and R¹ and R² are as defined in one row of table A; Table A1516: Compounds of the formula W142, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1517: Compounds of the formula W142, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1518: Compounds of the formula W142, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1519: Compounds of the formula W142, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1520: Compounds of the formula W142, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1521 : Compounds of the formula W142, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1522: Compounds of the formula W142, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1523: Compounds of the formula W142, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1524: Compounds of the formula W142, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1525: Compounds of the formula W142, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1526: Compounds of the formula W142, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1527: Compounds of the formula W142, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A1528: Compounds of the formula W142, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1529: Compounds of the formula W142, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1530: Compounds of the formula W142, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1531 : Compounds of the formula W143, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A1532: Compounds of the formula W143, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A1533: Compounds of the formula W143, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1534: Compounds of the formula W143, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1535: Compounds of the formula W143, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1536: Compounds of the formula W143, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1537: Compounds of the formula W143, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A1538: Compounds of the formula W143, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1539: Compounds of the formula W143, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1540: Compounds of the formula W143, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1541 : Compounds of the formula W143, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1542: Compounds of the formula W143, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A1543: Compounds of the formula W143, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1544: Compounds of the formula W143, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1545: Compounds of the formula W143, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1546: Compounds of the formula W143, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1547: Compounds of the formula W143, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A;

Table A1548: Compounds of the formula W143, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A1549: Compounds of the formula W146, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1550: Compounds of the formula W146, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1551 : Compounds of the formula W146, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1552: Compounds of the formula W146, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1553: Compounds of the formula W146, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1554: Compounds of the formula W146, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1555: Compounds of the formula W146, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1556: Compounds of the formula W146, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1557: Compounds of the formula W146, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1558: Compounds of the formula W146, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1559: Compounds of the formula W146, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1560: Compounds of the formula W146, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1561 : Compounds of the formula W146, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1562: Compounds of the formula W146, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1563: Compounds of the formula W146, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A1564: Compounds of the formula W146, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1565: Compounds of the formula W146, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1566: Compounds of the formula W146, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1567: Compounds of the formula W147, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1568: Compounds of the formula W147, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A1569: Compounds of the formula W147, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A1570: Compounds of the formula W147, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1571 : Compounds of the formula W147, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1572: Compounds of the formula W147, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1573: Compounds of the formula W147, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A1574: Compounds of the formula W147, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1575: Compounds of the formula W147, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1576: Compounds of the formula W147, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1577: Compounds of the formula W147, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1578: Compounds of the formula W147, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1579: Compounds of the formula W147, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1580: Compounds of the formula W147, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1581 : Compounds of the formula W147, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1582: Compounds of the formula W147, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1583: Compounds of the formula W147, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1584: Compounds of the formula W147, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A;

Table A1585: Compounds of the formula W148, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A1586: Compounds of the formula W148, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1587: Compounds of the formula W148, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1588: Compounds of the formula W148, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1589: Compounds of the formula W148, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1590: Compounds of the formula W148, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A1591 : Compounds of the formula W148, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1592: Compounds of the formula W148, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1593: Compounds of the formula W148, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1594: Compounds of the formula W148, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1595: Compounds of the formula W148, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1596: Compounds of the formula W148, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1597: Compounds of the formula W148, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1598: Compounds of the formula W148, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1599: Compounds of the formula W148, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1600: Compounds of the formula W148, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1601 : Compounds of the formula W148, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1602: Compounds of the formula W148, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1603: Compounds of the formula W149, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1604: Compounds of the formula W149, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1605: Compounds of the formula W149, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A1606: Compounds of the formula W149, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1607: Compounds of the formula W149, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1608: Compounds of the formula W149, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1609: Compounds of the formula W149, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1610: Compounds of the formula W149, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1611 : Compounds of the formula W149, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1612: Compounds of the formula W149, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1613: Compounds of the formula W149, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1614: Compounds of the formula W149, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1615: Compounds of the formula W149, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1616: Compounds of the formula W149, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1617: Compounds of the formula W149, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1618: Compounds of the formula W149, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1619: Compounds of the formula W149, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1620: Compounds of the formula W149, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1621 : Compounds of the formula W152, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A1622: Compounds of the formula W152, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A1623: Compounds of the formula W152, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1624: Compounds of the formula W152, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1625: Compounds of the formula W152, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1626: Compounds of the formula W152, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A1627: Compounds of the formula W152, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A1628: Compounds of the formula W152, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1629: Compounds of the formula W152, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1630: Compounds of the formula W152, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1631 : Compounds of the formula W152, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1632: Compounds of the formula W152, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A1633: Compounds of the formula W152, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1634: Compounds of the formula W152, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1635: Compounds of the formula W152, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1636: Compounds of the formula W152, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1637: Compounds of the formula W152, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1638: Compounds of the formula W152, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1639: Compounds of the formula W153, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1640: Compounds of the formula W153, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1641 : Compounds of the formula W153, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1642: Compounds of the formula W153, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1643: Compounds of the formula W153, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1644: Compounds of the formula W153, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1645: Compounds of the formula W153, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1646: Compounds of the formula W153, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1647: Compounds of the formula W153, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1648: Compounds of the formula W153, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1649: Compounds of the formula W153, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1650: Compounds of the formula W153, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1651 : Compounds of the formula W153, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1652: Compounds of the formula W153, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1653: Compounds of the formula W153, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A1654: Compounds of the formula W153, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1655: Compounds of the formula W153, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1656: Compounds of the formula W153, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1657: Compounds of the formula W154, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A1658: Compounds of the formula W154, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A1659: Compounds of the formula W154, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1660: Compounds of the formula W154, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1661 : Compounds of the formula W154, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1662: Compounds of the formula W154, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1663: Compounds of the formula W154, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A1664: Compounds of the formula W154, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1665: Compounds of the formula W154, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1666: Compounds of the formula W154, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1667: Compounds of the formula W154, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1668: Compounds of the formula W154, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A1669: Compounds of the formula W154, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1670: Compounds of the formula W154, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1671 : Compounds of the formula W154, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1672: Compounds of the formula W154, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1673: Compounds of the formula W154, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A;

Table A1674: Compounds of the formula W154, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A1675: Compounds of the formula W155, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1676: Compounds of the formula W155, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1677: Compounds of the formula W155, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1678: Compounds of the formula W155, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1679: Compounds of the formula W155, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1680: Compounds of the formula W155, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1681 : Compounds of the formula W155, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1682: Compounds of the formula W155, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1683: Compounds of the formula W155, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1684: Compounds of the formula W155, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1685: Compounds of the formula W155, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1686: Compounds of the formula W155, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1687: Compounds of the formula W155, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1688: Compounds of the formula W155, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1689: Compounds of the formula W155, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A1690: Compounds of the formula W155, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1691 : Compounds of the formula W155, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1692: Compounds of the formula W155, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1693: Compounds of the formula W156, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1694: Compounds of the formula W156, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A1695: Compounds of the formula W156, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A1696: Compounds of the formula W156, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1697: Compounds of the formula W156, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1698: Compounds of the formula W156, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1699: Compounds of the formula W156, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A1700: Compounds of the formula W156, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1701 : Compounds of the formula W156, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1702: Compounds of the formula W156, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1703: Compounds of the formula W156, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1704: Compounds of the formula W156, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1705: Compounds of the formula W156, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1706: Compounds of the formula W156, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1707: Compounds of the formula W156, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1708: Compounds of the formula W156, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1709: Compounds of the formula W156, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1710: Compounds of the formula W156, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A;

Table A1711 : Compounds of the formula W158, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A1712: Compounds of the formula W158, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1713: Compounds of the formula W158, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1714: Compounds of the formula W158, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1715: Compounds of the formula W158, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1716: Compounds of the formula W158, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A1717: Compounds of the formula W158, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1718: Compounds of the formula W158, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1719: Compounds of the formula W158, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1720: Compounds of the formula W158, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1721 : Compounds of the formula W158, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1722: Compounds of the formula W158, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1723: Compounds of the formula W158, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1724: Compounds of the formula W158, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1725: Compounds of the formula W158, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1726: Compounds of the formula W158, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1727: Compounds of the formula W158, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1728: Compounds of the formula W158, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1729: Compounds of the formula W159, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1730: Compounds of the formula W159, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1731 : Compounds of the formula W159, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A1732: Compounds of the formula W159, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1733: Compounds of the formula W159, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1734: Compounds of the formula W159, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1735: Compounds of the formula W159, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1736: Compounds of the formula W159, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1737: Compounds of the formula W159, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1738: Compounds of the formula W159, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1739: Compounds of the formula W159, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1740: Compounds of the formula W159, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1741 : Compounds of the formula W159, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1742: Compounds of the formula W159, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1743: Compounds of the formula W159, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1744: Compounds of the formula W159, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1745: Compounds of the formula W159, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1746: Compounds of the formula W159, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1747: Compounds of the formula W160, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A1748: Compounds of the formula W160, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A1749: Compounds of the formula W160, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1750: Compounds of the formula W160, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1751 : Compounds of the formula W160, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1752: Compounds of the formula W160, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A1753: Compounds of the formula W160, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A1754: Compounds of the formula W160, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1755: Compounds of the formula W160, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1756: Compounds of the formula W160, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1757: Compounds of the formula W160, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1758: Compounds of the formula W160, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A1759: Compounds of the formula W160, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1760: Compounds of the formula W160, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1761 : Compounds of the formula W160, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1762: Compounds of the formula W160, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1763: Compounds of the formula W160, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1764: Compounds of the formula W160, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1765: Compounds of the formula W161 , wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1766: Compounds of the formula W161 , wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1767: Compounds of the formula W161 , wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1768: Compounds of the formula W161 , wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1769: Compounds of the formula W161 , wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1770: Compounds of the formula W161 , wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1771 : Compounds of the formula W161 , wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1772: Compounds of the formula W161 , wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1773: Compounds of the formula W161 , wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1774: Compounds of the formula W161 , wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1775: Compounds of the formula W161 , wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1776: Compounds of the formula W161 , wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1777: Compounds of the formula W161 , wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1778: Compounds of the formula W161 , wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1779: Compounds of the formula W161 , wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A1780: Compounds of the formula W161 , wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1781 : Compounds of the formula W161 , wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1782: Compounds of the formula W161 , wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1783: Compounds of the formula W164, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A1784: Compounds of the formula W164, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A1785: Compounds of the formula W164, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1786: Compounds of the formula W164, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1787: Compounds of the formula W164, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1788: Compounds of the formula W164, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1789: Compounds of the formula W164, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A1790: Compounds of the formula W164, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1791 : Compounds of the formula W164, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1792: Compounds of the formula W164, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1793: Compounds of the formula W164, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1794: Compounds of the formula W164, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A1795: Compounds of the formula W164, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1796: Compounds of the formula W164, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1797: Compounds of the formula W164, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1798: Compounds of the formula W164, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1799: Compounds of the formula W164, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A;

Table A1800: Compounds of the formula W164, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A1801 : Compounds of the formula W165, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1802: Compounds of the formula W165, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1803: Compounds of the formula W165, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1804: Compounds of the formula W165, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1805: Compounds of the formula W165, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1806: Compounds of the formula W165, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1807: Compounds of the formula W165, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1808: Compounds of the formula W165, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1809: Compounds of the formula W165, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1810: Compounds of the formula W165, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1811 : Compounds of the formula W165, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1812: Compounds of the formula W165, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1813: Compounds of the formula W165, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1814: Compounds of the formula W165, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1815: Compounds of the formula W165, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A1816: Compounds of the formula W165, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1817: Compounds of the formula W165, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1818: Compounds of the formula W165, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1819: Compounds of the formula W166, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1820: Compounds of the formula W166, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A1821 : Compounds of the formula W166, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A1822: Compounds of the formula W166, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1823: Compounds of the formula W166, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1824: Compounds of the formula W166, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1825: Compounds of the formula W166, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A1826: Compounds of the formula W166, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1827: Compounds of the formula W166, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1828: Compounds of the formula W166, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1829: Compounds of the formula W166, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1830: Compounds of the formula W166, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1831 : Compounds of the formula W166, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1832: Compounds of the formula W166, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1833: Compounds of the formula W166, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1834: Compounds of the formula W166, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1835: Compounds of the formula W166, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1836: Compounds of the formula W166, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A;

Table A1837: Compounds of the formula W167, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A1838: Compounds of the formula W167, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1839: Compounds of the formula W167, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1840: Compounds of the formula W167, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1841 : Compounds of the formula W167, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1842: Compounds of the formula W167, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A1843: Compounds of the formula W167, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1844: Compounds of the formula W167, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1845: Compounds of the formula W167, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1846: Compounds of the formula W167, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1847: Compounds of the formula W167, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1848: Compounds of the formula W167, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1849: Compounds of the formula W167, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1850: Compounds of the formula W167, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1851 : Compounds of the formula W167, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1852: Compounds of the formula W167, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1853: Compounds of the formula W167, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1854: Compounds of the formula W167, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1855: Compounds of the formula W170, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1856: Compounds of the formula W170, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1857: Compounds of the formula W170, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A1858: Compounds of the formula W170, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1859: Compounds of the formula W170, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1860: Compounds of the formula W170, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1861 : Compounds of the formula W170, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1862: Compounds of the formula W170, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1863: Compounds of the formula W170, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1864: Compounds of the formula W170, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1865: Compounds of the formula W170, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1866: Compounds of the formula W170, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1867: Compounds of the formula W170, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1868: Compounds of the formula W170, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1869: Compounds of the formula W170, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1870: Compounds of the formula W170, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1871 : Compounds of the formula W170, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1872: Compounds of the formula W170, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1873: Compounds of the formula W171 , wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A1874: Compounds of the formula W171 , wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A1875: Compounds of the formula W171 , wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1876: Compounds of the formula W171 , wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1877: Compounds of the formula W171 , wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1878: Compounds of the formula W171 , wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A1879: Compounds of the formula W171 , wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A1880: Compounds of the formula W171 , wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1881 : Compounds of the formula W171 , wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1882: Compounds of the formula W171 , wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1883: Compounds of the formula W171 , wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1884: Compounds of the formula W171 , wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A1885: Compounds of the formula W171 , wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1886: Compounds of the formula W171 , wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1887: Compounds of the formula W171 , wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1888: Compounds of the formula W171 , wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1889: Compounds of the formula W171 , wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1890: Compounds of the formula W171 , wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1891 : Compounds of the formula W172, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1892: Compounds of the formula W172, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1893: Compounds of the formula W172, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1894: Compounds of the formula W172, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1895: Compounds of the formula W172, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1896: Compounds of the formula W172, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1897: Compounds of the formula W172, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1898: Compounds of the formula W172, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1899: Compounds of the formula W172, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1900: Compounds of the formula W172, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1901 : Compounds of the formula W172, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1902: Compounds of the formula W172, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1903: Compounds of the formula W172, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1904: Compounds of the formula W172, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1905: Compounds of the formula W172, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A1906: Compounds of the formula W172, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1907: Compounds of the formula W172, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1908: Compounds of the formula W172, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1909: Compounds of the formula W173, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A1910: Compounds of the formula W173, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A1911 : Compounds of the formula W173, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1912: Compounds of the formula W173, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1913: Compounds of the formula W173, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1914: Compounds of the formula W173, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1915: Compounds of the formula W173, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A1916: Compounds of the formula W173, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1917: Compounds of the formula W173, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1918: Compounds of the formula W173, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1919: Compounds of the formula W173, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1920: Compounds of the formula W173, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A1921 : Compounds of the formula W173, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1922: Compounds of the formula W173, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1923: Compounds of the formula W173, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1924: Compounds of the formula W173, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1925: Compounds of the formula W173, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A;

Table A1926: Compounds of the formula W173, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A1927: Compounds of the formula W176, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1928: Compounds of the formula W176, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1929: Compounds of the formula W176, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1930: Compounds of the formula W176, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1931 : Compounds of the formula W176, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1932: Compounds of the formula W176, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1933: Compounds of the formula W176, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1934: Compounds of the formula W176, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1935: Compounds of the formula W176, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1936: Compounds of the formula W176, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1937: Compounds of the formula W176, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1938: Compounds of the formula W176, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1939: Compounds of the formula W176, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1940: Compounds of the formula W176, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1941 : Compounds of the formula W176, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A1942: Compounds of the formula W176, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1943: Compounds of the formula W176, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1944: Compounds of the formula W176, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1945: Compounds of the formula W177, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1946: Compounds of the formula W177, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A1947: Compounds of the formula W177, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A1948: Compounds of the formula W177, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1949: Compounds of the formula W177, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1950: Compounds of the formula W177, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1951 : Compounds of the formula W177, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A1952: Compounds of the formula W177, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1953: Compounds of the formula W177, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1954: Compounds of the formula W177, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1955: Compounds of the formula W177, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1956: Compounds of the formula W177, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1957: Compounds of the formula W177, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1958: Compounds of the formula W177, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1959: Compounds of the formula W177, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1960: Compounds of the formula W177, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1961 : Compounds of the formula W177, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1962: Compounds of the formula W177, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A;

Table A1963: Compounds of the formula W178, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A1964: Compounds of the formula W178, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1965: Compounds of the formula W178, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A1966: Compounds of the formula W178, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A1967: Compounds of the formula W178, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A1968: Compounds of the formula W178, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A1969: Compounds of the formula W178, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1970: Compounds of the formula W178, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A1971 : Compounds of the formula W178, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A1972: Compounds of the formula W178, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A1973: Compounds of the formula W178, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A1974: Compounds of the formula W178, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1975: Compounds of the formula W178, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A1976: Compounds of the formula W178, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A1977: Compounds of the formula W178, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1978: Compounds of the formula W178, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A1979: Compounds of the formula W178, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1980: Compounds of the formula W178, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1981 : Compounds of the formula W179, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A1982: Compounds of the formula W179, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A1983: Compounds of the formula W179, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A1984: Compounds of the formula W179, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A1985: Compounds of the formula W179, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A1986: Compounds of the formula W179, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A1987: Compounds of the formula W179, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A1988: Compounds of the formula W179, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A1989: Compounds of the formula W179, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A1990: Compounds of the formula W179, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A1991 : Compounds of the formula W179, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A1992: Compounds of the formula W179, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A1993: Compounds of the formula W179, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A1994: Compounds of the formula W179, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A1995: Compounds of the formula W179, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A1996: Compounds of the formula W179, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A1997: Compounds of the formula W179, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A1998: Compounds of the formula W179, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A1999: Compounds of the formula W182, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A2000: Compounds of the formula W182, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A2001 : Compounds of the formula W182, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2002: Compounds of the formula W182, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A2003: Compounds of the formula W182, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A2004: Compounds of the formula W182, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A2005: Compounds of the formula W182, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A2006: Compounds of the formula W182, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A2007: Compounds of the formula W182, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2008: Compounds of the formula W182, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A2009: Compounds of the formula W182, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A2010: Compounds of the formula W182, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A2011 : Compounds of the formula W182, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A2012: Compounds of the formula W182, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A2013: Compounds of the formula W182, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2014: Compounds of the formula W182, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A2015: Compounds of the formula W182, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A2016: Compounds of the formula W182, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2017: Compounds of the formula W183, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A2018: Compounds of the formula W183, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A2019: Compounds of the formula W183, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2020: Compounds of the formula W183, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A2021 : Compounds of the formula W183, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A2022: Compounds of the formula W183, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2023: Compounds of the formula W183, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A2024: Compounds of the formula W183, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A2025: Compounds of the formula W183, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A2026: Compounds of the formula W183, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A2027: Compounds of the formula W183, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A2028: Compounds of the formula W183, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2029: Compounds of the formula W183, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A2030: Compounds of the formula W183, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A2031 : Compounds of the formula W183, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A2032: Compounds of the formula W183, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A2033: Compounds of the formula W183, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A2034: Compounds of the formula W183, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2035: Compounds of the formula W184, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A2036: Compounds of the formula W184, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A2037: Compounds of the formula W184, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2038: Compounds of the formula W184, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A2039: Compounds of the formula W184, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A2040: Compounds of the formula W184, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2041 : Compounds of the formula W184, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A2042: Compounds of the formula W184, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A2043: Compounds of the formula W184, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2044: Compounds of the formula W184, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A2045: Compounds of the formula W184, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A2046: Compounds of the formula W184, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A2047: Compounds of the formula W184, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A2048: Compounds of the formula W184, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A2049: Compounds of the formula W184, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2050: Compounds of the formula W184, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A2051 : Compounds of the formula W184, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A;

Table A2052: Compounds of the formula W184, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A2053: Compounds of the formula W186, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A2054: Compounds of the formula W186, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A2055: Compounds of the formula W186, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2056: Compounds of the formula W186, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A2057: Compounds of the formula W186, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A2058: Compounds of the formula W186, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2059: Compounds of the formula W186, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A2060: Compounds of the formula W186, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A2061 : Compounds of the formula W186, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2062: Compounds of the formula W186, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A2063: Compounds of the formula W186, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A2064: Compounds of the formula W186, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2065: Compounds of the formula W186, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A2066: Compounds of the formula W186, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A2067: Compounds of the formula W186, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A2068: Compounds of the formula W186, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A2069: Compounds of the formula W186, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A2070: Compounds of the formula W186, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2071 : Compounds of the formula W187, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A2072: Compounds of the formula W187, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A2073: Compounds of the formula W187, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A2074: Compounds of the formula W187, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A2075: Compounds of the formula W187, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A2076: Compounds of the formula W187, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2077: Compounds of the formula W187, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A2078: Compounds of the formula W187, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A2079: Compounds of the formula W187, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2080: Compounds of the formula W187, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A2081 : Compounds of the formula W187, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A2082: Compounds of the formula W187, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2083: Compounds of the formula W187, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A2084: Compounds of the formula W187, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A2085: Compounds of the formula W187, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2086: Compounds of the formula W187, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A2087: Compounds of the formula W187, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A2088: Compounds of the formula W187, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A;

Table A2089: Compounds of the formula W190, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A2090: Compounds of the formula W190, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A2091 : Compounds of the formula W190, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2092: Compounds of the formula W190, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A2093: Compounds of the formula W190, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A2094: Compounds of the formula W190, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A2095: Compounds of the formula W190, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A2096: Compounds of the formula W190, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A2097: Compounds of the formula W190, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2098: Compounds of the formula W190, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A2099: Compounds of the formula W190, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A2100: Compounds of the formula W190, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2101 : Compounds of the formula W190, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A2102: Compounds of the formula W190, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A2103: Compounds of the formula W190, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2104: Compounds of the formula W190, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A2105: Compounds of the formula W190, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A2106: Compounds of the formula W190, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2107: Compounds of the formula W191 , wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A2108: Compounds of the formula W191 , wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A2109: Compounds of the formula W191 , wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A21 10: Compounds of the formula W191 , wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A21 11 : Compounds of the formula W191 , wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A21 12: Compounds of the formula W191 , wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A21 13: Compounds of the formula W191 , wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A21 14: Compounds of the formula W191 , wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A21 15: Compounds of the formula W191 , wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A21 16: Compounds of the formula W191 , wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A21 17: Compounds of the formula W191 , wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A21 18: Compounds of the formula W191 , wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A21 19: Compounds of the formula W191 , wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A2120: Compounds of the formula W191 , wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A2121 : Compounds of the formula W191 , wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2122: Compounds of the formula W191 , wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A2123: Compounds of the formula W191 , wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A2124: Compounds of the formula W191 , wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2125: Compounds of the formula W192, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A2126: Compounds of the formula W192, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A2127: Compounds of the formula W192, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2128: Compounds of the formula W192, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A2129: Compounds of the formula W192, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A2130: Compounds of the formula W192, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A2131 : Compounds of the formula W192, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A2132: Compounds of the formula W192, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A2133: Compounds of the formula W192, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2134: Compounds of the formula W192, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A2135: Compounds of the formula W192, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A2136: Compounds of the formula W192, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A2137: Compounds of the formula W192, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A2138: Compounds of the formula W192, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A2139: Compounds of the formula W192, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2140: Compounds of the formula W192, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A2141 : Compounds of the formula W192, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A2142: Compounds of the formula W192, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2143: Compounds of the formula W193, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A2144: Compounds of the formula W193, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A2145: Compounds of the formula W193, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2146: Compounds of the formula W193, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A2147: Compounds of the formula W193, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A2148: Compounds of the formula W193, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2149: Compounds of the formula W193, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A2150: Compounds of the formula W193, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A2151 : Compounds of the formula W193, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A2152: Compounds of the formula W193, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A2153: Compounds of the formula W193, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A2154: Compounds of the formula W193, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2155: Compounds of the formula W193, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A2156: Compounds of the formula W193, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A2157: Compounds of the formula W193, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A2158: Compounds of the formula W193, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A2159: Compounds of the formula W193, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A2160: Compounds of the formula W193, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2161 : Compounds of the formula W194, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A2162: Compounds of the formula W194, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A2163: Compounds of the formula W194, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2164: Compounds of the formula W194, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A2165: Compounds of the formula W194, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A2166: Compounds of the formula W194, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2167: Compounds of the formula W194, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A2168: Compounds of the formula W194, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A2169: Compounds of the formula W194, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2170: Compounds of the formula W194, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A2171 : Compounds of the formula W194, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A2172: Compounds of the formula W194, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A2173: Compounds of the formula W194, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A2174: Compounds of the formula W194, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A2175: Compounds of the formula W194, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2176: Compounds of the formula W194, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A2177: Compounds of the formula W194, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A;

Table A2178: Compounds of the formula W194, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A2179: Compounds of the formula W195, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A2180: Compounds of the formula W195, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A2181 : Compounds of the formula W195, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2182: Compounds of the formula W195, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A2183: Compounds of the formula W195, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A2184: Compounds of the formula W195, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2185: Compounds of the formula W195, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A2186: Compounds of the formula W195, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A2187: Compounds of the formula W195, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2188: Compounds of the formula W195, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A2189: Compounds of the formula W195, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A2190: Compounds of the formula W195, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2191 : Compounds of the formula W195, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A2192: Compounds of the formula W195, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A2193: Compounds of the formula W195, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A2194: Compounds of the formula W195, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A2195: Compounds of the formula W195, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A2196: Compounds of the formula W195, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2197: Compounds of the formula W197, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A2198: Compounds of the formula W197, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A2199: Compounds of the formula W197, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A2200: Compounds of the formula W197, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A2201 : Compounds of the formula W197, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A2202: Compounds of the formula W197, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2203: Compounds of the formula W197, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A2204: Compounds of the formula W197, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A2205: Compounds of the formula W197, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2206: Compounds of the formula W197, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A2207: Compounds of the formula W197, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A2208: Compounds of the formula W197, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2209: Compounds of the formula W197, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A2210: Compounds of the formula W197, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A2211 : Compounds of the formula W197, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2212: Compounds of the formula W197, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A2213: Compounds of the formula W197, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A2214: Compounds of the formula W197, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A;

Table A2215: Compounds of the formula W198, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A2216: Compounds of the formula W198, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A2217: Compounds of the formula W198, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2218: Compounds of the formula W198, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A2219: Compounds of the formula W198, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A2220: Compounds of the formula W198, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A2221 : Compounds of the formula W198, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A2222: Compounds of the formula W198, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A2223: Compounds of the formula W198, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2224: Compounds of the formula W198, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A2225: Compounds of the formula W198, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A2226: Compounds of the formula W198, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2227: Compounds of the formula W198, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A2228: Compounds of the formula W198, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A2229: Compounds of the formula W198, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2230: Compounds of the formula W198, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A2231 : Compounds of the formula W198, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A2232: Compounds of the formula W198, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2233: Compounds of the formula W199, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A2234: Compounds of the formula W199, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A2235: Compounds of the formula W199, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A2236: Compounds of the formula W199, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A2237: Compounds of the formula W199, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A2238: Compounds of the formula W199, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2239: Compounds of the formula W199, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A2240: Compounds of the formula W199, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A2241 : Compounds of the formula W199, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A2242: Compounds of the formula W199, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A2243: Compounds of the formula W199, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A2244: Compounds of the formula W199, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2245: Compounds of the formula W199, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A2246: Compounds of the formula W199, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A2247: Compounds of the formula W199, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2248: Compounds of the formula W199, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A2249: Compounds of the formula W199, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A2250: Compounds of the formula W199, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2251 : Compounds of the formula W200, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A2252: Compounds of the formula W200, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A2253: Compounds of the formula W200, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2254: Compounds of the formula W200, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A2255: Compounds of the formula W200, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A2256: Compounds of the formula W200, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A2257: Compounds of the formula W200, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A2258: Compounds of the formula W200, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A2259: Compounds of the formula W200, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2260: Compounds of the formula W200, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A2261 : Compounds of the formula W200, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A2262: Compounds of the formula W200, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A2263: Compounds of the formula W200, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A2264: Compounds of the formula W200, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A2265: Compounds of the formula W200, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2266: Compounds of the formula W200, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A2267: Compounds of the formula W200, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A2268: Compounds of the formula W200, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2269: Compounds of the formula W203, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A2270: Compounds of the formula W203, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A2271 : Compounds of the formula W203, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2272: Compounds of the formula W203, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A2273: Compounds of the formula W203, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A2274: Compounds of the formula W203, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2275: Compounds of the formula W203, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A2276: Compounds of the formula W203, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A2277: Compounds of the formula W203, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A2278: Compounds of the formula W203, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A2279: Compounds of the formula W203, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A2280: Compounds of the formula W203, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2281 : Compounds of the formula W203, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A2282: Compounds of the formula W203, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A2283: Compounds of the formula W203, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A2284: Compounds of the formula W203, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A2285: Compounds of the formula W203, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A2286: Compounds of the formula W203, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2287: Compounds of the formula W204, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A2288: Compounds of the formula W204, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A2289: Compounds of the formula W204, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2290: Compounds of the formula W204, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A2291 : Compounds of the formula W204, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A2292: Compounds of the formula W204, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2293: Compounds of the formula W204, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A2294: Compounds of the formula W204, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A2295: Compounds of the formula W204, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2296: Compounds of the formula W204, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A2297: Compounds of the formula W204, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A2298: Compounds of the formula W204, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A2299: Compounds of the formula W204, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A2300: Compounds of the formula W204, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A2301 : Compounds of the formula W204, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2302: Compounds of the formula W204, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A2303: Compounds of the formula W204, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A;

Table A2304: Compounds of the formula W204, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A2305: Compounds of the formula W205, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A2306: Compounds of the formula W205, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A2307: Compounds of the formula W205, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2308: Compounds of the formula W205, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A2309: Compounds of the formula W205, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A2310: Compounds of the formula W205, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2311 : Compounds of the formula W205, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A2312: Compounds of the formula W205, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A2313: Compounds of the formula W205, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2314: Compounds of the formula W205, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A2315: Compounds of the formula W205, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A2316: Compounds of the formula W205, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2317: Compounds of the formula W205, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A2318: Compounds of the formula W205, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A2319: Compounds of the formula W205, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A2320: Compounds of the formula W205, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A2321 : Compounds of the formula W205, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A2322: Compounds of the formula W205, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2323: Compounds of the formula W207, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A2324: Compounds of the formula W207, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A2325: Compounds of the formula W207, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A2326: Compounds of the formula W207, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A2327: Compounds of the formula W207, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A2328: Compounds of the formula W207, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2329: Compounds of the formula W207, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A2330: Compounds of the formula W207, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A2331 : Compounds of the formula W207, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2332: Compounds of the formula W207, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A2333: Compounds of the formula W207, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A2334: Compounds of the formula W207, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2335: Compounds of the formula W207, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A2336: Compounds of the formula W207, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A2337: Compounds of the formula W207, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2338: Compounds of the formula W207, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A2339: Compounds of the formula W207, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A2340: Compounds of the formula W207, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A;

Table A2341 : Compounds of the formula W209, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A2342: Compounds of the formula W209, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A2343: Compounds of the formula W209, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2344: Compounds of the formula W209, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A2345: Compounds of the formula W209, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A2346: Compounds of the formula W209, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A2347: Compounds of the formula W209, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A2348: Compounds of the formula W209, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A2349: Compounds of the formula W209, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2350: Compounds of the formula W209, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A2351 : Compounds of the formula W209, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A2352: Compounds of the formula W209, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2353: Compounds of the formula W209, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A2354: Compounds of the formula W209, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A2355: Compounds of the formula W209, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2356: Compounds of the formula W209, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A2357: Compounds of the formula W209, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A2358: Compounds of the formula W209, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2359: Compounds of the formula W210, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A2360: Compounds of the formula W210, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A2361 : Compounds of the formula W210, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A2362: Compounds of the formula W210, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A2363: Compounds of the formula W210, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A2364: Compounds of the formula W210, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2365: Compounds of the formula W210, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A2366: Compounds of the formula W210, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A2367: Compounds of the formula W210, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A2368: Compounds of the formula W210, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A2369: Compounds of the formula W210, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A2370: Compounds of the formula W210, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2371 : Compounds of the formula W210, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A2372: Compounds of the formula W210, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A2373: Compounds of the formula W210, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2374: Compounds of the formula W210, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A2375: Compounds of the formula W210, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A2376: Compounds of the formula W210, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2377: Compounds of the formula W21 1 , wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A2378: Compounds of the formula W21 1 , wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A2379: Compounds of the formula W211 , wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2380: Compounds of the formula W21 1 , wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A2381 : Compounds of the formula W21 1 , wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A2382: Compounds of the formula W211 , wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A2383: Compounds of the formula W211 , wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A2384: Compounds of the formula W21 1 , wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A2385: Compounds of the formula W21 1 , wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2386: Compounds of the formula W21 1 , wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A2387: Compounds of the formula W21 1 , wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A2388: Compounds of the formula W21 1 , wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A2389: Compounds of the formula W21 1 , wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A2390: Compounds of the formula W21 1 , wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A2391 : Compounds of the formula W21 1 , wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2392: Compounds of the formula W21 1 , wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A2393: Compounds of the formula W21 1 , wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A2394: Compounds of the formula W21 1 , wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2395: Compounds of the formula W212, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A2396: Compounds of the formula W212, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A2397: Compounds of the formula W212, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2398: Compounds of the formula W212, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A2399: Compounds of the formula W212, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A2400: Compounds of the formula W212, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2401 : Compounds of the formula W212, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A2402: Compounds of the formula W212, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A2403: Compounds of the formula W212, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A2404: Compounds of the formula W212, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A2405: Compounds of the formula W212, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A2406: Compounds of the formula W212, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2407: Compounds of the formula W212, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A2408: Compounds of the formula W212, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A2409: Compounds of the formula W212, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A2410: Compounds of the formula W212, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A2411 : Compounds of the formula W212, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A2412: Compounds of the formula W212, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2413: Compounds of the formula W215, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A2414: Compounds of the formula W215, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A2415: Compounds of the formula W215, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2416: Compounds of the formula W215, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A2417: Compounds of the formula W215, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A2418: Compounds of the formula W215, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2419: Compounds of the formula W215, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A2420: Compounds of the formula W215, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A2421 : Compounds of the formula W215, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2422: Compounds of the formula W215, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A2423: Compounds of the formula W215, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A2424: Compounds of the formula W215, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A2425: Compounds of the formula W215, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A2426: Compounds of the formula W215, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A2427: Compounds of the formula W215, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2428: Compounds of the formula W215, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A2429: Compounds of the formula W215, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A;

Table A2430: Compounds of the formula W215, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A2431 : Compounds of the formula W216, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A2432: Compounds of the formula W216, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A2433: Compounds of the formula W216, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2434: Compounds of the formula W216, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A2435: Compounds of the formula W216, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A2436: Compounds of the formula W216, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2437: Compounds of the formula W216, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A2438: Compounds of the formula W216, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A2439: Compounds of the formula W216, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2440: Compounds of the formula W216, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A2441 : Compounds of the formula W216, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A2442: Compounds of the formula W216, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2443: Compounds of the formula W216, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A2444: Compounds of the formula W216, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A2445: Compounds of the formula W216, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A2446: Compounds of the formula W216, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A2447: Compounds of the formula W216, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A2448: Compounds of the formula W216, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2449: Compounds of the formula W217, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A2450: Compounds of the formula W217, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A2451 : Compounds of the formula W217, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A2452: Compounds of the formula W217, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A2453: Compounds of the formula W217, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A2454: Compounds of the formula W217, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2455: Compounds of the formula W217, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A2456: Compounds of the formula W217, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A2457: Compounds of the formula W217, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2458: Compounds of the formula W217, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A2459: Compounds of the formula W217, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A2460: Compounds of the formula W217, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2461 : Compounds of the formula W217, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A2462: Compounds of the formula W217, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A2463: Compounds of the formula W217, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2464: Compounds of the formula W217, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A2465: Compounds of the formula W217, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A2466: Compounds of the formula W217, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A;

Table A2467: Compounds of the formula W221 , wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A2468: Compounds of the formula W221 , wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A2469: Compounds of the formula W221 , wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2470: Compounds of the formula W221 , wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A2471 : Compounds of the formula W221 , wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A2472: Compounds of the formula W221 , wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A2473: Compounds of the formula W221 , wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A2474: Compounds of the formula W221 , wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A2475: Compounds of the formula W221 , wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2476: Compounds of the formula W221 , wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A2477: Compounds of the formula W221 , wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A2478: Compounds of the formula W221 , wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2479: Compounds of the formula W221 , wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A2480: Compounds of the formula W221 , wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A2481 : Compounds of the formula W221 , wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2482: Compounds of the formula W221 , wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A2483: Compounds of the formula W221 , wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A2484: Compounds of the formula W221 , wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2485: Compounds of the formula W222, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A2486: Compounds of the formula W222, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A2487: Compounds of the formula W222, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A2488: Compounds of the formula W222, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A2489: Compounds of the formula W222, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A2490: Compounds of the formula W222, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2491 : Compounds of the formula W222, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A2492: Compounds of the formula W222, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A2493: Compounds of the formula W222, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A2494: Compounds of the formula W222, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A2495: Compounds of the formula W222, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A2496: Compounds of the formula W222, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2497: Compounds of the formula W222, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A2498: Compounds of the formula W222, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A2499: Compounds of the formula W222, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2500: Compounds of the formula W222, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A2501 : Compounds of the formula W222, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A2502: Compounds of the formula W222, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2503: Compounds of the formula W223, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A2504: Compounds of the formula W223, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A2505: Compounds of the formula W223, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2506: Compounds of the formula W223, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A2507: Compounds of the formula W223, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A2508: Compounds of the formula W223, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A2509: Compounds of the formula W223, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A2510: Compounds of the formula W223, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A2511 : Compounds of the formula W223, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2512: Compounds of the formula W223, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A2513: Compounds of the formula W223, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A2514: Compounds of the formula W223, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A2515: Compounds of the formula W223, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A2516: Compounds of the formula W223, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A2517: Compounds of the formula W223, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2518: Compounds of the formula W223, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A2519: Compounds of the formula W223, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A2520: Compounds of the formula W223, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2521 : Compounds of the formula W227, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A2522: Compounds of the formula W227, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A2523: Compounds of the formula W227, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2524: Compounds of the formula W227, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A2525: Compounds of the formula W227, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A2526: Compounds of the formula W227, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2527: Compounds of the formula W227, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A2528: Compounds of the formula W227, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A2529: Compounds of the formula W227, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A2530: Compounds of the formula W227, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A2531 : Compounds of the formula W227, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A2532: Compounds of the formula W227, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2533: Compounds of the formula W227, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A2534: Compounds of the formula W227, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A2535: Compounds of the formula W227, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A2536: Compounds of the formula W227, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A2537: Compounds of the formula W227, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A2538: Compounds of the formula W227, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2539: Compounds of the formula W228, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A2540: Compounds of the formula W228, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A2541 : Compounds of the formula W228, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2542: Compounds of the formula W228, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A2543: Compounds of the formula W228, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A2544: Compounds of the formula W228, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2545: Compounds of the formula W228, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A2546: Compounds of the formula W228, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A2547: Compounds of the formula W228, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2548: Compounds of the formula W228, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A2549: Compounds of the formula W228, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A2550: Compounds of the formula W228, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A2551 : Compounds of the formula W228, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A2552: Compounds of the formula W228, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A2553: Compounds of the formula W228, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2554: Compounds of the formula W228, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A2555: Compounds of the formula W228, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A;

Table A2556: Compounds of the formula W228, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A2557: Compounds of the formula W230, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A2558: Compounds of the formula W230, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A2559: Compounds of the formula W230, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2560: Compounds of the formula W230, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A2561 : Compounds of the formula W230, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A2562: Compounds of the formula W230, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2563: Compounds of the formula W230, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A2564: Compounds of the formula W230, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A2565: Compounds of the formula W230, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2566: Compounds of the formula W230, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A2567: Compounds of the formula W230, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A2568: Compounds of the formula W230, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2569: Compounds of the formula W230, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A2570: Compounds of the formula W230, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A2571 : Compounds of the formula W230, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A2572: Compounds of the formula W230, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A2573: Compounds of the formula W230, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A2574: Compounds of the formula W230, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2575: Compounds of the formula W234, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A2576: Compounds of the formula W234, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A2577: Compounds of the formula W234, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A2578: Compounds of the formula W234, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A2579: Compounds of the formula W234, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A2580: Compounds of the formula W234, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2581 : Compounds of the formula W234, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A2582: Compounds of the formula W234, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A2583: Compounds of the formula W234, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2584: Compounds of the formula W234, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A2585: Compounds of the formula W234, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A2586: Compounds of the formula W234, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2587: Compounds of the formula W234, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A2588: Compounds of the formula W234, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A2589: Compounds of the formula W234, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2590: Compounds of the formula W234, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A2591 : Compounds of the formula W234, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A2592: Compounds of the formula W234, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A;

Table A2593: Compounds of the formula W235, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A2594: Compounds of the formula W235, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A2595: Compounds of the formula W235, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2596: Compounds of the formula W235, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A2597: Compounds of the formula W235, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A2598: Compounds of the formula W235, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A2599: Compounds of the formula W235, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A2600: Compounds of the formula W235, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A2601 : Compounds of the formula W235, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2602: Compounds of the formula W235, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A2603: Compounds of the formula W235, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A2604: Compounds of the formula W235, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2605: Compounds of the formula W235, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A2606: Compounds of the formula W235, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A2607: Compounds of the formula W235, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2608: Compounds of the formula W235, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A2609: Compounds of the formula W235, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A2610: Compounds of the formula W235, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2611 : Compounds of the formula W236, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A2612: Compounds of the formula W236, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A2613: Compounds of the formula W236, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A;

Table A2614: Compounds of the formula W236, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A2615: Compounds of the formula W236, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A2616: Compounds of the formula W236, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2617: Compounds of the formula W236, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A2618: Compounds of the formula W236, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A2619: Compounds of the formula W236, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A2620: Compounds of the formula W236, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A2621 : Compounds of the formula W236, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A2622: Compounds of the formula W236, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2623: Compounds of the formula W236, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A2624: Compounds of the formula W236, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A2625: Compounds of the formula W236, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2626: Compounds of the formula W236, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A2627: Compounds of the formula W236, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A2628: Compounds of the formula W236, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2629: Compounds of the formula W238, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A2630: Compounds of the formula W238, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A2631 : Compounds of the formula W238, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2632: Compounds of the formula W238, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A2633: Compounds of the formula W238, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A2634: Compounds of the formula W238, wherein R³ is Cl and R¹ and R² are as defined in one row of table A;

Table A2635: Compounds of the formula W238, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A2636: Compounds of the formula W238, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A2637: Compounds of the formula W238, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2638: Compounds of the formula W238, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A2639: Compounds of the formula W238, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A2640: Compounds of the formula W238, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A2641 : Compounds of the formula W238, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A2642: Compounds of the formula W238, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A2643: Compounds of the formula W238, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2644: Compounds of the formula W238, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A2645: Compounds of the formula W238, wherein R³ is OCH₂-OCH₃ and R¹ and R² are as defined in one row of table A;

Table A2646: Compounds of the formula W238, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2647: Compounds of the formula W239, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A2648: Compounds of the formula W239, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A2649: Compounds of the formula W239, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2650: Compounds of the formula W239, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A2651 : Compounds of the formula W239, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A2652: Compounds of the formula W239, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2653: Compounds of the formula W239, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A2654: Compounds of the formula W239, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A2655: Compounds of the formula W239, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A;

Table A2656: Compounds of the formula W239, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A2657: Compounds of the formula W239, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A2658: Compounds of the formula W239, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2659: Compounds of the formula W239, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A2660: Compounds of the formula W239, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A;

Table A2661 : Compounds of the formula W239, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A2662: Compounds of the formula W239, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A2663: Compounds of the formula W239, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A2664: Compounds of the formula W239, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A; Table A2665: Compounds of the formula W240, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A;

Table A2666: Compounds of the formula W240, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A;

Table A2667: Compounds of the formula W240, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2668: Compounds of the formula W240, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A; Table A2669: Compounds of the formula W240, wherein R³ is F and R¹ and R² are as defined in one row of table A; Table A2670: Compounds of the formula W240, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2671 : Compounds of the formula W240, wherein R³ is Br and R¹ and R² are as defined in one row of table A;

Table A2672: Compounds of the formula W240, wherein R³ is I and R¹ and R² are as defined in one row of table A;

Table A2673: Compounds of the formula W240, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2674: Compounds of the formula W240, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A; Table A2675: Compounds of the formula W240, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A; Table A2676: Compounds of the formula W240, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A;

Table A2677: Compounds of the formula W240, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A;

Table A2678: Compounds of the formula W240, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A2679: Compounds of the formula W240, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A; Table A2680: Compounds of the formula W240, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A; Table A2681 : Compounds of the formula W240, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A;

Table A2682: Compounds of the formula W240, wherein R³ is OCH₂CH₃ and R¹ and R² are as defined in one row of table A;

Table A2683: Compounds of the formula W243, wherein R³ is CH₃ and R¹ and R² are as defined in one row of table A; Table A2684: Compounds of the formula W243, wherein R³ is C₂H₅ and R¹ and R² are as defined in one row of table A; Table A2685: Compounds of the formula W243, wherein R³ is CF₃ and R¹ and R² are as defined in one row of table A; Table A2686: Compounds of the formula W243, wherein R³ is CCI₃ and R¹ and R² are as defined in one row of table A;

Table A2687: Compounds of the formula W243, wherein R³ is F and R¹ and R² are as defined in one row of table A;

Table A2688: Compounds of the formula W243, wherein R³ is Cl and R¹ and R² are as defined in one row of table A; Table A2689: Compounds of the formula W243, wherein R³ is Br and R¹ and R² are as defined in one row of table A; Table A2690: Compounds of the formula W243, wherein R³ is I and R¹ and R² are as defined in one row of table A; Table A2691 : Compounds of the formula W243, wherein R³ is OCH₃ and R¹ and R² are as defined in one row of table A; Table A2692: Compounds of the formula W243, wherein R³ is OCF₃ and R¹ and R² are as defined in one row of table A;

Table A2693: Compounds of the formula W243, wherein R³ is OCCI₃ and R¹ and R² are as defined in one row of table A;

Table A2694: Compounds of the formula W243, wherein R³ is OCHF₂ and R¹ and R² are as defined in one row of table A; Table A2695: Compounds of the formula W243, wherein R³ is OCCIF₂ and R¹ and R² are as defined in one row of table A; Table A2696: Compounds of the formula W243, wherein R³ is OCH₂F and R¹ and R² are as defined in one row of table A; Table A2697: Compounds of the formula W243, wherein R³ is OCHCI₂ and R¹ and R² are as defined in one row of table A;

Table A2698: Compounds of the formula W243, wherein R³ is OCH₂CI and R¹ and R² are as defined in one row of table A;

Table A2699: Compounds of the formula W243, wherein R³ is OCH₂-OCH₃ and R¹ and

R² are as defined in one row of table A; Table A2700: Compounds of the formula W243, wherein R³ is OCH₂CH₃ and R¹ and

R² are as defined in one row of table A;

Table A:

Pests

The compounds of the formula I, and their salts are in particular suitable for efficiently controlling arthropodal pests such as arachnids, myriapedes and insects as well as nematodes.

In particular, they are suitable for controlling insect pests, such as insects from the order of

Lepidoptera: for example Agrotis ypsilon, Agrotis segetum, Alabama argillacea, Anticarsia gemmatalis, Argyresthia conjugella, Autographa gamma, Bupalus piniarius, Cacoecia murinana, Capua reticulana, Cheimatobia brumata, Choristoneura fumiferana, Choristoneura occidentalis, Cirphis unipuncta, Cydia pomonella, Dendrolimus pini, Diaphania nitidalis, Diatraea grandiosella, Earias insulana, Elasmopalpus lignosellus, Eupoecilia ambiguella, Evetria bouliana, Feltia subterranea, Galleria mellonella, Grapholitha funebrana, Grapholitha molesta, Heliothis armigera, Heliothis virescens, Heliothis zea, HeIIuIa undalis, Hibernia defoliaria, Hyphantria cunea, Hyponomeuta malinellus, Keiferia lycopersicella, Lambdina fiscellaria,

Laphygma exigua, Leucoptera coffeella, Leucoptera scitella, Lithocolletis blancardella, Lobesia botrana, Loxostege sticticalis, Lymantria dispar, Lymantria monacha, Lyonetia clerkella, Malacosoma neustria, Mamestra brassicae, Orgyia pseudotsugata, Ostrinia nubilalis, Panolis flammea, Pectinophora gossypiella, Peridroma saucia, Phalera bucephala, Phthorimaea operculella, Phyllocnistis citrella, Pieris brassicae, Plathypena scabra, Plutella xylostella, Pseudoplusia includens, Rhyacionia frustrana, Scrobipalpula absoluta, Sitotroga cerealella, Sparganothis pilleriana, Spodoptera eridania, Spodoptera frugiperda, Spodoptera littoralis, Spodoptera litura, Thaumatopoea pityocampa, Tortrix viridana, Trichoplusia ni and Zeiraphera canadensis,

Coleoptera (beetles), for example Agrilus sinuatus, Agriotes lineatus, Agriotes obscurus, Amphimallus solstitialis, Anisandrus dispar, Anthonomus grandis, Anthonomus pomorum, Atomaria linearis, Blastophagus piniperda, Blitophaga undata, Bruchus rufimanus, Bruchus pisorum, Bruchus lentis, Byctiscus betulae, Cassida nebulosa, Cerotoma trifurcata, Ceuthorrhynchus assimilis, Ceuthorrhynchus napi, Chaetocnema tibialis, Conoderus vespertinus, Crioceris asparagi, Diabrotica Iongicornis, Diabrotica 12-punctata, Diabrotica virgifera, Epilachna varivestis, Epitrix hirtipennis, Eutinobothrus brasiliensis, Hylobius abietis, Hypera brunneipennis, Hypera postica, lps typographus, Lema bilineata, Lema melanopus, Leptinotarsa decemlineata, Limonius californicus, Lissorhoptrus oryzophilus, Melanotus communis, Meligethes aeneus, Melolontha hippocastani, Melolontha melolontha, Oulema oryzae, Ortiorrhynchus sulcatus, Otiorrhynchus ovatus, Phaedon cochleariae, Phyllotreta chrysocephala, Phyllophaga sp., Phyllopertha horticola, Phyllotreta nemorum, Phyllotreta striolata, Popillia japonica, Sitona lineatus and Sitophilus granaria,

Diptera, for example Aedes aegypti, Aedes vexans, Anastrepha ludens, Anopheles maculipennis, Ceratitis capitata, Chrysomya bezziana, Chrysomya hominivorax, Chrysomya macellaria, Contarinia sorghicola, Cordylobia anthropophaga, Culex pipiens, Dacus cucurbitae, Dacus oleae, Dasineura brassicae, Fannia canicularis, Gasterophilus intestinalis, Glossina morsitans, Haematobia irritans, Haplodiplosis equestris, Hylemyia platura, Hypoderma lineata, Liriomyza sativae, Liriomyza trifolii, Lucilia caprina, Lucilia cuprina, Lucilia sericata, Lycoria pectoralis, Mayetiola destructor, Musca domestica, Muscina stabulans, Oestrus ovis, Oscinella frit, Pegomya hysocyami, Phorbia antiqua, Phorbia brassicae, Phorbia coarctata, Rhagoletis cerasi, Rhagoletis pomonella, Tabanus bovinus, Tipula oleracea and Tipula paludosa,

Thysanoptera (thrips), e.g. Dichromothrips spp., Frankliniella fusca, Frankliniella occidentalis, Frankliniella tritici, Scirtothrips citri, Thrips oryzae, Thrips palmi and Thrips tabaci,

Hymenoptera e.g. Athalia rosae, Atta cephalotes, Atta sexdens, Atta texana, Hoplocampa minuta, Hoplocampa testudinea, Monomorium pharaonis, Solenopsis geminata and Solenopsis invicta,

Heteroptera, e.g. Acrosternum hilare, Blissus leucopterus, Cyrtopeltis notatus, Dysdercus cingulatus, Dysdercus intermedius, Eurygaster integriceps, Euschistus impictiventris, Leptoglossus phyllopus, Lygus lineolaris, Lygus pratensis, Nezara viridula, Piesma quadrata, Solubea insularis and Thyanta perditor,

Homoptera (in particular aphids), e.g. Acyrthosiphon onobrychis, Adelges laricis, Aphidula nasturtii, Aphis craccivora, Aphis fabae, Aphis forbesi, Aphis pomi, Aphis gossypii, Aphis grossulariae, Aphis schneideri, Aphis spiraecola, Aphis sambuci, Acyrthosiphon pisum, Aulacorthum solani, Bemisa tabaci, Bemisa argentifolii, Brachycaudus cardui, Brachycaudus helichrysi, Brachycaudus persicae, Brachycaudus prunicola, Brevicoryne brassicae, Capitophorus horni, Cerosipha gossypii, Chaetosiphon fragaefolii, Cryptomyzus ribis, Dreyfusia nordmannianae, Dreyfusia piceae, Dysaphis radicola, Dysaulacorthum pseudosolani, Dysaphis plantaginea, Dysaphis pyri, Empoasca fabae, Hyalopterus pruni, Hyperomyzus lactucae, Macrosiphum avenae, Macrosiphum euphorbiae, Macrosiphon rosae, Megoura viciae, Melanaphis pyrarius, Metopolophium dirhodum, Myzodes persicae, Myzus ascalonicus, Myzus cerasi, Myzus varians, Nasonovia ribis-nigri, Nilaparvata lugens, Pemphigus bursarius, Perkinsiella saccharicida, Phorodon humuli, Psylla mali, Psylla piri, Rhopalomyzus ascalonicus, Rhopalosiphum maidis, Rhopalosiphum padi, Rhopalosiphum insertum, Sappaphis mala, Sappaphis mali, Schizaphis graminum, Schizoneura lanuginosa, Sitobion avenae, Trialeurodes vaporariorum, Toxoptera aurantiiand, and Viteus vitifolii,

lsoptera (termites), e.g. Calotermes flavicollis, Leucotermes flavipes, Reticulitermes lucifugus und Termes natalensis,

Orthoptera, e.g. Acheta domestica, Blatta orientalis, Blattella germanica, Forficula auricularia, Gryllotalpa gryllotalpa, Locusta migratoria, Melanoplus bivittatus, Melanoplus femur-rubrum, Melanoplus mexicanus, Melanoplus sanguinipes, Melanoplus spretus, Nomadacris septemfasciata, Periplaneta americana, Schistocerca americana, Schistocerca peregrina, Stauronotus maroccanus and Tachycines asynamorus, and

Collembola (springtails), e.g. Onychiurus ssp..

They are also suitable for controlling Nematodes : plant parasitic nematodes such as root knot nematodes, Meloidogyne hapla, Meloidogyne incognita, Meloidogyne javanica, and other Meloidogyne species; cyst-forming nematodes, Globodera rostochiensis and other Globodera species; Heterodera avenae, Heterodera glycines, Heterodera schachtii, Heterodera trifolii, and other Heterodera species; Seed gall nematodes, Anguina species; Stem and foliar nematodes, Aphelenchoides species; Sting nematodes, Belonolaimus longicaudatus and other Belonolaimus species; Pine nematodes, Bursaphelenchus xylophilus and other Bursaphelenchus species; Ring nematodes, Criconema species, Criconemella species, Criconemoides species, Mesocriconema species; Stem and bulb nematodes, Ditylenchus destructor, Ditylenchus dipsaci and other Ditylenchus species; AwI nematodes, Dolichodorus species; Spiral nematodes, Heliocotylenchus multicinctus and other Helicotylenchus species; Sheath and sheathoid nematodes, Hemicycliophora species and Hemicriconemoides species; Hirshmanniella species; Lance nematodes, Hoploaimus species; false rootknot nematodes, Nacobbus species; Needle nematodes, Longidorus elongatus and other Longidorus species; Lesion nematodes, Pratylenchus neglectus, Pratylenchus penetrans, Pratylenchus curvitatus, Pratylenchus goodeyi and other Pratylenchus species; Burrowing nematodes, Radopholus similis and other Radopholus species; Reniform nematodes, Rotylenchus robustus and other Rotylenchus species; Scutellonema species; Stubby root nematodes, Trichodorus primitivus and other Trichodorus species, Paratrichodorus species; Stunt nematodes, Tylenchorhynchus claytoni, Tylenchorhynchus dubius and other Tylenchorhynchus species; Citrus nematodes, Tylenchulus species; Dagger nematodes, Xiphinema species; and other plant parasitic nematode species.

The compounds of the formula I and their salts are also useful for controlling arachnids (Arachnoidea), such as acarians (Acarina), e.g. of the families Argasidae, Ixodidae and Sarcoptidae, such as Amblyomma americanum, Amblyomma variegatum, Argas persicus, Boophilus annulatus, Boophilus decoloratus, Boophilus microplus, Dermacentor silvarum, Hyalomma truncatum, Ixodes ricinus, Ixodes rubicundus, Ornithodorus moubata, Otobius megnini, Dermanyssus gallinae, Psoroptes ovis, Rhipicephalus appendiculatus, Rhipicephalus evertsi, Sarcoptes scabiei, and Eriophyidae spp. such as Aculus schlechtendali, Phyllocoptrata oleivora and Eriophyes sheldoni; Tarsonemidae spp. such as Phytonemus pallidus and Polyphagotarsonemus latus; Tenuipalpidae spp. such as Brevipalpus phoenicis; Tetranychidae spp. such as Tetranychus cinnabarinus, Tetranychus kanzawai, Tetranychus pacificus, Tetranychus telarius and Tetranychus urticae, Panonychus ulmi, Panonychus citri, and oligonychus pratensis.

Compounds of the formula I are particularly useful for controlling insects, preferably sucking or piercing insects such as insects from the genera Thysanoptera, Hymenoptera, Orthoptera and Homptera, in particular the following species:

Thysanoptera (thrips): Frankliniella fusca, Frankliniella occidentalis, Frankliniella tritici, Scirtothrips citri, Thrips oryzae, Thrips palmi and Thrips tabaci,

Hymenoptera: Athalia rosae, Atta cephalotes, Atta sexdens, Atta texana, Hoplocampa minuta, Hoplocampa testudinea, Monomorium pharaonis, Solenopsis geminata and Solenopsis invicta,

Orthoptera: Acheta domestica, Blatta orientalis, Blattella germanica, Forficula auricularia, Gryllotalpa gryllotalpa, Locusta migratoria, Melanoplus bivittatus, Melanoplus femur-rubrum, Melanoplus mexicanus, Melanoplus sanguinipes, Melanoplus spretus, Nomadacris septemfasciata, Periplaneta americana, Schistocerca americana, Schistocerca peregrina, Stauronotus maroccanus and Tachycines asynamorus ;

Homoptera, in particular aphids: Acyrthosiphon onobrychis, Adelges laricis, Aphidula nasturtii, Aphis fabae, Aphis forbesi, Aphis pomi, Aphis gossypii, Aphis grossulariae, Aphis schneideri, Aphis spiraecola, Aphis sambuci, Acyrthosiphon pisum, Aulacorthum solani, Brachycaudus cardui, Brachycaudus helichrysi, Brachycaudus persicae, Brachycaudus prunicola, Brevicoryne brassicae, Capitophorus horni, Cerosipha gossypii, Chaetosiphon fragaefolii, Cryptomyzus ribis, Dreyfusia nordmannianae, Dreyfusia piceae, Dysaphis radicola, Dysaulacorthum pseudosolani, Dysaphis plantaginea, Dysaphis pyri, Empoasca fabae, Hyalopterus pruni, Hyperomyzus lactucae, Macrosiphum avenae, Macrosiphum euphorbiae, Macrosiphon rosae, Megoura viciae, Melanaphis pyrarius, Metopolophium dirhodum, Myzodes persicae, Myzus ascalonicus, Myzus cerasi, Myzus varians, Nasonovia ribis-nigri, Nilaparvata lugens, Pemphigus bursarius, Perkinsiella saccharicida, Phorodon humuli, Psylla mali, Psylla piri, Rhopalomyzus ascalonicus, Rhopalosiphum maidis, Rhopalosiphum padi, Rhopalosiphum insertum, Sappaphis mala, Sappaphis mali, Schizaphis graminum, Schizoneura lanuginosa, Sitobion avenae, Trialeurodes vaporariorum, Toxoptera aurantiiand, and Viteus vitifolii;

Compounds of the formula I are particularly useful for controlling insects of the orders Homoptera and Thysanoptera and more preferably for controlling aphids.

Formulations

For use in a method according to the present invention, the compounds I can be converted into the customary formulations, e.g. solutions, emulsions, suspensions, dusts, powders, pastes, granules and directly sprayable solutions. The use form depends on the particular purpose and application method. Formulations and application methods are chosen to ensure in each case a fine and uniform distribution of the compound of the formula I according to the present invention.

The formulations are prepared in a known manner (see e.g. for review US 3,060,084, EP-A 707 445 (for liquid concentrates), Browning, "Agglomeration", Chemical

Engineering, Dec. 4, 1967, 147-48, Perry's Chemical Engineer's Handbook, 4th Ed., McGraw-Hill, New York, 1963, pages 8-57 and et seq. WO 91/13546, US 4,172,714, US 4,144,050, US 3,920,442, US 5,180,587, US 5,232,701 , US 5,208,030, GB 2,095,558, US 3,299,566, Klingman, Weed Control as a Science, John Wiley and Sons, Inc., New York, 1961 , Hance et al., Weed Control Handbook, 8th Ed., Blackwell Scientific Publications, Oxford, 1989 and Mollet, H., Grubemann, A., Formulation technology, Wiley VCH Verlag GmbH, Weinheim (Germany), 2001 , 2. D. A. Knowles, Chemistry and Technology of Agrochemical Formulations, Kluwer Academic Publishers, Dordrecht, 1998 (ISBN 0-7514-0443-8), for example by extending the active compound with auxiliaries suitable for the formulation of agrochemicals, such as solvents and/or carriers, if desired emulsifiers, surfactants and dispersants, preservatives, antifoaming agents, anti-freezing agents, for seed treatment formulation also optionally colorants and/or binders and/or gelling agents.

Solvents/carriers, which are suitable, are e.g.:

solvents such as water, aromatic solvents (for example Solvesso products, xylene and the like), paraffins (for example mineral fractions), alcohols (for example methanol, butanol, pentanol, benzyl alcohol), ketones (for example cyclohexanone, gamma-butyrolactone), pyrrolidones (N-metyhl-pyrrolidone (NMP),N-octylpyrrolidone NOP), acetates (glycol diacetate), alkyl lactates, lactones such as g-butyrolactone, glycols, fatty acid dimethylamides, fatty acids and fatty acid esters, triglycerides, oils of vegetable or animal origin and modified oils such as alkylated plant oils. In principle, solvent mixtures may also be used, carriers such as ground natural minerals and ground synthetic minerals, such as silica gels, finely divided silicic acid, silicates, talc, kaolin, attaclay, limestone, lime, chalk, bole, loess, clay, dolomite, diatomaceous earth, calcium sulfate and magnesium sulfate, magnesium oxide, ground synthetic materials, fertilizers, such as, for example, ammonium sulfate, ammonium phosphate, ammonium nitrate, ureas and products of vegetable origin, such as cereal meal, tree bark meal, wood meal and nutshell meal, cellulose powders and other solid carriers. Suitable emulsifiers are nonionic and anionic emulsifiers (for example polyoxyethylene fatty alcohol ethers, alkylsulfonates and arylsulfonates).

Examples of dispersants are lignin-sulfite waste liquors and methylcellulose.

Suitable surfactants are alkali metal, alkaline earth metal and ammonium salts of lignosulfonic acid, naphthalenesulfonic acid, phenolsulfonic acid, dibutylnaphthalenesulfonic acid, alkylarylsulfonates, alkyl sulfates, alkylsulfonates, fatty alcohol sulfates, fatty acids and sulfated fatty alcohol glycol ethers, furthermore condensates of sulfonated naphthalene and naphthalene derivatives with formaldehyde, condensates of naphthalene or of naphthalenesulfonic acid with phenol and formaldehyde, polyoxyethylene octylphenyl ether, ethoxylated isooctylphenol, octylphenol, nonylphenol, alkylphenyl polyglycol ethers, tributylphenyl polyglycol ether, tristearylphenyl polyglycol ether, alkylaryl polyether alcohols, alcohol and fatty alcohol/ethylene oxide condensates, ethoxylated castor oil, polyoxyethylene alkyl ethers, ethoxylated polyoxypropylene, lauryl alcohol polyglycol ether acetal, sorbitol esters,

Also anti-freezing agents such as glycerin, ethylene glycol, propylene glycol and bactericides such as can be added to the formulation. Suitable antifoaming agents are for example antifoaming agents based on silicon or magnesium stearate.

Suitable preservatives are for example dichlorophen und benzyl alcohol hemiformal

Suitable thickeners are compounds which confer a pseudoplastic flow behavior to the formulation, i.e. high viscosity at rest and low viscosity in the agitated stage. Mention may be made, in this context, for example, of commercial thickeners based on polysaccharides, such as Xanthan Gum^® (Kelzan^® from Kelco), Rhodopol^® 23 (Rhone Poulenc) or Veegum^® (from R. T. Vanderbilt), or organic phyllosilicates, such as Attaclay^® (from Engelhardt). Antifoam agents suitable for the dispersions according to the invention are, for example, silicone emulsions (such as, for example, Silikon^® SRE, Wacker or Rhodorsil^® from Rhodia), long-chain alcohols, fatty acids, organofluorine compounds and mixtures thereof. Biocides can be added to stabilize the compositions according to the invention against attack by microorganisms. Suitable biocides are, for example, based on isothiazolones such as the compounds marketed under the trademarks Proxel^® from Avecia (or Arch) or Acticide^® RS from Thor Chemie and Kathon^® MK from Rohm & Haas. Suitable antifreeze agents are organic polyols, for example ethylene glycol, propylene glycol or glycerol. These are usually employed in amounts of not more than 10% by weight, based on the total weight of the active compound composition. If appropriate, the active compound compositions according to the invention may comprise 1 to 5% by weight of buffer, based on the total amount of the formulation prepared, to regulate the pH, the amount and type of the buffer used depending on the chemical properties of the active compound or the active compounds. Examples of buffers are alkali metal salts of weak inorganic or organic acids, such as, for example, phosphoric acid, boronic acid, acetic acid, propionic acid, citric acid, fumaric acid, tartaric acid, oxalic acid and succinic acid.

Substances which are suitable for the preparation of directly sprayable solutions, emulsions, pastes or oil dispersions are mineral oil fractions of medium to high boiling point, such as kerosene or diesel oil, furthermore coal tar oils and oils of vegetable or animal origin, aliphatic, cyclic and aromatic hydrocarbons, for example toluene, xylene, paraffin, tetrahydronaphthalene, alkylated naphthalenes or their derivatives, methanol, ethanol, propanol, butanol, cyclohexanol, cyclohexanone, isophorone, strongly polar solvents, for example dimethyl sulfoxide, N-methylpyrrolidone and water.

Powders, materials for spreading and dusts can be prepared by mixing or concomitantly grinding the active substances with a solid carrier.

Granules, for example coated granules, impregnated granules and homogeneous granules, can be prepared by binding the active ingredients to solid carriers. Examples of solid carriers are mineral earths such as silica gels, silicates, talc, kaolin, attaclay, limestone, lime, chalk, bole, loess, clay, dolomite, diatomaceous earth, calcium sulfate, magnesium sulfate, magnesium oxide, ground synthetic materials, fertilizers, such as, for example, ammonium sulfate, ammonium phosphate, ammonium nitrate, ureas, and products of vegetable origin, such as cereal meal, tree bark meal, wood meal and nutshell meal, cellulose powders and other solid carriers.

In general, the formulations comprise from 0.01 to 95% by weight, preferably from 0.1 to 90% by weight, of the active ingredient. The active ingredients are employed in a purity of from 90% to 100%, preferably 95% to 100% (according to NMR spectrum).

For seed treatment purposes, respective formulations can be diluted 2-10 fold leading to concentrations in the ready to use preparations of 0,01 to 60% by weight active compound, preferably 0,1 to 40% by weight.

The compounds of formula I can be used as such, in the form of their formulations or the use forms prepared therefrom, for example in the form of directly sprayable solutions, powders, suspensions or dispersions, emulsions, oil dispersions, pastes, dustable products, materials for spreading, or granules, by means of spraying, atomizing, dusting, spreading or pouring. The use forms depend entirely on the intended purposes; they are intended to ensure in each case the finest possible distribution of the active compounds according to the invention.

The following are examples of formulations:

1. Products for dilution with water. For seed treatment purposes, such products may be applied to the seed diluted or undiluted.

A) Water-soluble concentrates (SL, LS)

10 parts by weight of the active compound is dissolved in 90 parts by weight of water or a water-soluble solvent. As an alternative, wetters or other auxiliaries are added. The active compound dissolves upon dilution with water, whereby a formulation with 10 % (w/w) of active compound is obtained.

B) Dispersible concentrates (DC) 20 parts by weight of the active compound is dissolved in 70 parts by weight of cyclohexanone with addition of 10 parts by weight of a dispersant, for example polyvinylpyrrolidone. Dilution with water gives a dispersion, whereby a formulation with 20% (w/w) of active compounds is obtained.

C) Emulsifiable concentrates (EC)

15 parts by weight of the active compounds is dissolved in 7 parts by weight of xylene with addition of calcium dodecylbenzenesulfonate and castor oil ethoxylate (in each case 5 parts by weight). Dilution with water gives an emulsion, whereby a formulation with 15% (w/w) of active compounds is obtained.

D) Emulsions (EW, EO, ES)

25 parts by weight of the active compound is dissolved in 35 parts by weight of xylene with addition of calcium dodecylbenzenesulfonate and castor oil ethoxylate (in each case 5 parts by weight). This mixture is introduced into 30 parts by weight of water by means of an emulsifier machine (e.g. Ultraturrax) and made into a homogeneous emulsion. Dilution with water gives an emulsion, whereby a formulation with 25% (w/w) of active compound is obtained.

E) Suspensions (SC, OD, FS)

In an agitated ball mill, 20 parts by weight of the active compound is comminuted with addition of 10 parts by weight of dispersants, wetters and 70 parts by weight of water or of an organic solvent to give a fine active compound suspension. Dilution with water gives a stable suspension of the active compound, whereby a formulation with 20% (w/w) of active compound is obtained.

F) Water-dispersible granules and water-soluble granules (WG, SG)

50 parts by weight of the active compound is ground finely with addition of 50 parts by weight of dispersants and wetters and made as water-dispersible or water-soluble granules by means of technical appliances (for example extrusion, spray tower, fluidized bed). Dilution with water gives a stable dispersion or solution of the active compound, whereby a formulation with 50% (w/w) of active compound is obtained.

G) Water-dispersible powders and water-soluble powders (WP, SP, SS, WS) 75 parts by weight of the active compound are ground in a rotor-stator mill with addition of 25 parts by weight of dispersants, wetters and silica gel. Dilution with water gives a stable dispersion or solution of the active compound, whereby a formulation with 75% (w/w) of active compound is obtained.

H) Gel-Formulation (GF) (for seed treatment purposes only)

In an agitated ball mill, 20 parts by weight of the active compound is comminuted with addition of 10 parts by weight of dispersants, 1 part by weight of a gelling agent wetters and 70 parts by weight of water or of an organic solvent to give a fine active compound suspension. Dilution with water gives a stable suspension of the active compound, whereby a formulation with 20% (w/w) of active compound is obtained.

2. Products to be applied undiluted for foliar applications. For seed treatment purposes, such products may be applied to the seed diluted or undiluted. I) Dustable powders (DP, DS)

5 parts by weight of the active compound are ground finely and mixed intimately with 95 parts by weight of finely divided kaolin. This gives a dustable product having 5% (w/w) of active compound.

J) Granules (GR, FG, GG, MG)

0.5 part by weight of the active compound is ground finely and associated with 95.5 parts by weight of carriers, whereby a formulation with 0.5% (w/w) of active compound is obtained. Current methods are extrusion, spray-drying or the fluidized bed. This gives granules to be applied undiluted for foliar use.

K) ULV solutions (UL)

10 parts by weight of the active compound is dissolved in 90 parts by weight of an organic solvent, for example xylene. This gives a product having 10% (w/w) of active compound, which is applied undiluted for foliar use.

Aqueous use forms can be prepared from emulsion concentrates, pastes or wettable powders (sprayable powders, oil dispersions) by adding water. To prepare emulsions, pastes or oil dispersions, the substances, as such or dissolved in an oil or solvent, can be homogenized in water by means of a wetter, tackifier, dispersant or emulsifier. Alternatively, it is possible to prepare concentrates composed of active substance, wetter, tackifier, dispersant or emulsifier and, if appropriate, solvent or oil, and such concentrates are suitable for dilution with water.

The active ingredient concentrations in the ready-to-use products can be varied within relatively wide ranges. In general, they are from 0.0001 to 10%, preferably from 0.01 to 1 %.

The active ingredients may also be used successfully in the ultra-low-volume process (ULV), it being possible to apply formulations comprising over 95% by weight of active ingredient, or even to apply the active ingredient without additives.

In the method of this invention compounds I may be applied with other active ingredients, for example with other pesticides, insecticides, herbicides, fertilizers such as ammonium nitrate, urea, potash, and superphosphate, phytotoxicants and plant growth regulators, safeners and nematicides. These additional ingredients may be used sequentially or in combination with the above-described compositions, if appropriate also added only immediately prior to use (tank mix). For example, the plant(s) may be sprayed with a composition of this invention either before or after being treated with other active ingredients. These additional agents can be admixed with the agents used according to the invention in a weight ratio of 1 :10 to 10:1. Mixing the compounds I or the compositions comprising them in the use form as pesticides with other pesticides frequently results in a broader pesticidal spectrum of action.

The following list M of pesticides together with which the compounds according to the invention can be used and with which potential synergistic effects might be produced, is intended to illustrate the possible combinations, but not to impose any limitation:

M.1. Organo(thio)phosphates: acephate, azamethiphos, azinphos-methyl, chlorpyrifos, chlorpyrifos-methyl, chlorfenvinphos, diazinon, dichlorvos, dicrotophos, dimethoate, disulfoton, ethion, fenitrothion, fenthion, isoxathion, malathion, methamidophos, methidathion, methyl-parathion, mevinphos, monocrotophos, oxydemeton-methyl, paraoxon, parathion, phenthoate, phosalone, phosmet, phosphamidon, phorate, phoxim, pirimiphos-methyl, profenofos, prothiofos, sulprophos, tetrachlorvinphos, terbufos, triazophos, trichlorfon;

M.2. Carbamates: alanycarb, aldicarb, bendiocarb, benfuracarb, carbaryl, carbofuran, carbosulfan, fenoxycarb, furathiocarb, methiocarb, methomyl, oxamyl, pirimicarb, propoxur, thiodicarb, triazamate;

M.3. Pyrethroids: allethrin, bifenthrin, cyfluthrin, cyhalothrin, cyphenothrin, cypermethrin, alpha-cypermethrin, beta-cypermethrin, zeta-cypermethrin, deltamethrin, empenthrin, esfenvalerate, etofenprox, fenpropathrin, fenvalerate, imiprothrin, lambda- cyhalothrin, permethrin, prallethrin, pyrethrin I and II, resmethrin, silafluofen, tau- fluvalinate, tefluthrin, tetramethrin, tralomethrin, transfluthrin, profluthrin, dimefluthrin;

M.4. Growth regulators: a) chitin synthesis inhibitors: benzoylureas: chlorfluazuron, diflubenzuron, flucycloxuron, flufenoxuron, hexaflumuron, lufenuron, novaluron, teflubenzuron, triflumuron; buprofezin, diofenolan, hexythiazox, etoxazole, clofentazine; b) ecdysone antagonists: halofenozide, methoxyfenozide, tebufenozide, azadirachtin; c) juvenoids: pyriproxyfen, methoprene, fenoxycarb; d) lipid biosynthesis inhibitors: spirodiclofen, spiromesifen, spirotetramat;

M.5. Nicotinic receptor agonists/antagonists compounds: clothianidin, dinotefuran, imidacloprid, thiamethoxam, nitenpyram, acetamiprid, thiacloprid and AKD-1022;

M.6. GABA antagonist compounds: acetoprole, endosulfan, ethiprole, fipronil, vaniliprole, pyrafluprole, pyriprole, the phenylpyrazole compound of formula M^{6 1}

M.7. Macrocyclic lactone insecticides: abamectin, emamectin, milbemectin, lepimectin, spinosad

M.8. METI I compounds: fenazaquin, pyridaben, tebufenpyrad, tolfenpyrad, flufenerim;

M.9. METI Il and III compounds: acequinocyl, fluacyprim, hydramethylnon;

M.10. Uncoupler compounds: chlorfenapyr;

M.1 1. Oxidative phosphorylation inhibitor compounds: cyhexatin, diafenthiuron, fenbutatin oxide, propargite;

M.12. Moulting disruptor compounds: cyromazine;

M.13. Mixed Function Oxidase inhibitor compounds: piperonyl butoxide;

M.14. Sodium channel blocker compounds: indoxacarb, metaflumizone,

M.15. Various: amitraz, benclothiaz, bifenazate, cartap, flonicamid, pyridalyl, pymetrozine, sulfur, thiocyclam, flubendiamide, cyenopyrafen, flupyrazofos, cyflumetofen, amidoflumet, pyrifluquinazon, N-R'-2,2-dihalo-1-R"cyclo- propanecarboxamide-2-(2,6-dichloro- α ,α ,α -tri-fluoro-p-tolyl)hydrazone or N-R'2,2- di(R"')propionamide-2-(2,6-dichloro- α ,α ,α -trifluoro-p-tolyl)-hydrazone, wherein R' s methyl or ethyl, halo is chloro or bromo, R" is hydrogen or methyl and R'" is methyl or ethyl, anthranilamide compounds as chlorantraniliprole or the compound of formula M^{15 1}.

and malononitrile compounds as described in JP 2002 284608, WO 02/89579, WO 02/90320, WO 02/90321 , WO 04/06677, WO 04/20399, JP 2004 99597, WO 05/68423, WO 05/68432, or WO 05/63694, especially the malononitrile compounds CF3(CH2)2C(CN)2CH2(CF2)3CF₂H, CF3(CH2)2C(CN)2CH2(CF2)5CF₂H, CF₃(CH2)2C(CN)2(CH2)2C(CF₃)2F, CF₃(CH2)2C(CN)2(CH2)2(CF2)3CF₃, CF₂H(CF₂)SCH₂C(CN)₂CH₂(CF₂)SCF₂H, CF₃(CH₂)2C(CN)2CH2(CF₂)₃CF₃, CF₃(CF₂)₂CH₂C(CN)₂CH₂(CF₂)sCF₂H, and CF₃CF₂CH₂C(CN)₂CH₂(CF₂)₃CF₂H.

The commercially available compounds of the group M may be found in The Pesticide Manual, 13^th Edition, British Crop Protection Council (2003) among other publications. The phenylpyrazole of formula M^{6 1} and the preparation thereof has been described in WO 98/28279. Lepimectin is known from Agro Project, PJB Publications Ltd, November 2004.

Benclothiaz and its preparation have been described in EP-A1 454621. Methidathion and Paraoxon and their preparation have been described in Farm Chemicals Handbook, Volume 88, Meister Publishing Company, 2001. Acetoprole and its preparation have been described in WO 98/28277. Metaflumizone and its preparation have been described in EP-A1 462 456. Flupyrazofos has been described in Pesticide Science 54, 1988, p.237-243 and in US 4822779. Pyrafluprole and its preparation have been described in JP 2002193709 and in WO 01/00614. Pyriprole and its preparation have been described in WO 98/45274 and in US 6335357. Amidoflumet and its preparation have been described in US 6221890 and in JP 21010907. Flufenerim and its preparation have been described in WO 03/007717 and in WO 03/007718. Cyflumetofen and its preparation have been described in WO 04/080180. The aminoquinazolinone pyrifluquinazone has been described in EP A 109 7932.

Anthranilamides as the one of formula M^{15 1} or as chloranthraniliprole and their preparations have been described in WO 01/70671 ; WO 02/48137; WO 03/24222, WO 03/15518, WO 04/67528; WO 04/33468; and WO 05/1 18552. The malononitrile compounds CF₃(CH₂)₂C(CN)₂CH₂(CF₂)₃CF₂H, CF₃(CH₂)₂C(CN)₂CH₂(CF₂)₅CF₂H, CF₃(CH₂)₂C(CN)₂(CH₂)₂C(CF₃)₂F, CF₃(CH₂)₂C(CN)₂(CH₂)₂(CF₂)₃CF₃, CF₂H(CF₂)₃CH₂C(CN)₂CH₂(CF₂)₃CF₂H, CF₃(CH₂)₂C(CN)₂CH₂(CF₂)₃CF₃, CF₃(CF₂)₂CH₂C(CN)₂CH₂(CF₂)₃CF₂H, and CF₃CF₂CH₂C(CN)₂CH₂(CF₂)₃CF₂H have been described in WO 05/63694.

Fungicidal mixing partners are those selected from the group F consisting of

F.1 acylalanines such as benalaxyl, metalaxyl, ofurace, oxadixyl;

F.2 amine derivatives such as aldimorph, dodine, dodemorph, fenpropimorph, fenpropidin, guazatine, iminoctadine, spiroxamin, tridemorph;

F.3 anilinopyrimidines such as pyrimethanil, mepanipyrim or cyrodinyl;

F.4 antibiotics such as cycloheximid, griseofulvin, kasugamycin, natamycin, polyoxin or streptomycin;

F.5 azoles such as bitertanol, bromoconazole, cyproconazole, difenoconazole, dinitroconazole, epoxiconazole, fenbuconazole, fluquiconazole, flusilazole, hexaconazole, imazalil, metconazole, myclobutanil, penconazole, propiconazole, prochloraz, prothioconazole, tebuconazole, triadimefon, triadimenol, triflumizol, triticonazole, flutriafol;

F.6 dicarboximides such as iprodion, myclozolin, procymidon, vinclozolin; F.7 dithiocarbamates such as ferbam, nabam, maneb, mancozeb, metam, metiram, propineb, polycarbamate, thiram, ziram, zineb;

F.8 heterocyclic compounds such as anilazine, benomyl, boscalid, carbendazim, carboxin, oxycarboxin, cyazofamid, dazomet, dithianon, famoxadon, fenamidon, fenarimol, fuberidazole, flutolanil, furametpyr, isoprothiolane, mepronil, nuarimol, probenazole, proquinazid, pyrifenox, pyroquilon, quinoxyfen, silthiofam, thiabendazole, thifluzamid, thiophanate-methyl, tiadinil, tricyclazole, triforine;

F.9 copper fungicides such as Bordeaux mixture, copper acetate, copper oxychloride, basic copper sulfate;

F.10 nitrophenyl derivatives such as binapacryl, dinocap, dinobuton, nitrophthalisopropyl;

F.1 1 phenylpyrroles such as fenpiclonil or fludioxonil;

F.12 strobilurins such as azoxystrobin, dimoxystrobin, fluoxastrobin, kresoxim-methyl, metominostrobin, orysastrobin, picoxystrobin or trifloxystrobin;

F.13 sulfenic acid derivatives such as captafol, captan, dichlofluanid, folpet, tolylfluanid; F.14 cinnemamides and analogs such as dimethomorph, flumetover or flumorph; F.15 sulfur, and other fungicides such as acibenzolar-S-methyl, benthiavalicarb, carpropamid, chlorothalonil, cyflufenamid, cymoxanil, dazomet, diclomezin, diclocymet, diethofencarb, edifenphos, ethaboxam, fenhexamid, fentin-acetate, fenoxanil, ferimzone, fluazinam, fosetyl, fosetyl-aluminum, iprovalicarb, hexachlorobenzene, metrafenon, pencycuron, propamocarb, phthalide, toloclofos-methyl, quintozene, zoxamid.

Applications

In the methods according to the invention the pests are controlled by contacting the target parasite/pest, its food supply, habitat, breeding ground or its locus with a pesticidally effective amount of compounds of formula I or with a salt thereof or with a composition, containing a pesticidally effective amount of a compound of formula I or a salt thereof.

"Locus" means a habitat, breeding ground, plant, seed, soil, area, material or environment in which a pest or parasite is growing or may grow.

In general, "pesticidally effective amount" means the amount of active ingredient needed to achieve an observable effect on growth, including the effects of necrosis, death, retardation, prevention, and removal, destruction, or otherwise diminishing the occurrence and activity of the target organism. The pesticidally effective amount can vary for the various compounds/compositions used in the invention. A pesticidally effective amount of the compositions will also vary according to the prevailing conditions such as desired pesticidal effect and duration, weather, target species, locus, mode of application, and the like.

The compounds of the invention can also be applied preventively to places at which occurrence of the pests is expected.

The compounds of formula I may be also used to protect growing plants from attack or infestation by pests by contacting the plant with a pesticidally effective amount of compounds of formula I. As such, "contacting" includes both direct contact (applying the compounds/compositions directly on the pest and/or plant - typically to the foliage, stem or roots of the plant) and indirect contact (applying the compounds/compositions to the locus of the pest and/or plant).

The aforementioned compositions are particularly useful for protecting crop plants against infestation of said pests or for combating these pests in infested plants.

For use in treating crop plants, the rate of application of the active ingredients of this invention may be in the range of 0.1 g to 4000 g per hectare, desirably from 25 g to 600 g per hectare, more desirably from 50 g to 500 g per hectare.

In the case of soil treatment or of application to the pests dwelling place or nest, the quantity of active ingredient ranges from 0.0001 to 500 g per 100 m², preferably from 0.001 to 2O g per 100 m².

The compounds of the invention may also be applied against non-crop insect pests, such as ants, termites, wasps, flies, mosquitos, crickets, or cockroaches. For use against said non-crop pests, compounds of formula I are preferably used in a bait composition.

The bait can be a liquid, a solid or a semisolid preparation (e.g. a gel). Solid baits can be formed into various shapes and forms suitable to the respective application e.g. granules, blocks, sticks, disks. Liquid baits can be filled into various devices to ensure proper application, e.g. open containers, spray devices, droplet sources, or evaporation sources. Gels can be based on aqueous or oily matrices and can be formulated to particular necessities in terms of stickyness, moisture retention or aging characteristics.

The bait employed in the composition is a product which is sufficiently attractive to incite insects such as ants, termites, wasps, flies, mosquitos, crickets etc. or cockroaches to eat it. The attractiveness can be manipulated by using feeding stimulants or sex pheromones. Food stimulants are chosen, for example, but not exclusively, from animal and/or plant proteins (meat-, fish- or blood meal, insect parts, egg yolk), from fats and oils of animal and/or plant origin, or mono-, oligo- or polyorganosaccharides, especially from sucrose, lactose, fructose, dextrose, glucose, starch, pectin or even molasses or honey. Fresh or decaying parts of fruits, crops, plants, animals, insects or specific parts thereof can also serve as a feeding stimulant. Sex pheromones are known to be more insect specific. Specific pheromones are described in the literature and are known to those skilled in the art.

For use in bait compositions, the typical content of active ingredient is from 0.001 weight % to 15 weight %, desirably from 0.001 weight % to 5% weight % of active compound.

Formulations of compounds of formula I as aerosols (e.g in spray cans), oil sprays or pump sprays are highly suitable for the non-professional user for controlling pests such as flies, fleas, ticks, mosquitos or cockroaches. Aerosol recipes are preferably composed of the active compound, solvents such as lower alcohols (e.g. methanol, ethanol, propanol, butanol), ketones (e.g. acetone, methyl ethyl ketone), paraffin hydrocarbons (e.g. kerosenes) having boiling ranges of approximately 50 to 250 °C, dimethylformamide, N-methylpyrrolidone, dimethyl sulfoxide, aromatic hydrocarbons such as toluene, xylene, water, furthermore auxiliaries such as emulsifiers such as sorbitol monooleate, oleyl ethoxylate having 3-7 mol of ethylene oxide, fatty alcohol ethoxylate, perfume oils such as ethereal oils, esters of medium fatty acids with lower alcohols, aromatic carbonyl compounds, if appropriate stabilizers such as sodium benzoate, amphoteric surfactants, lower epoxides, triethyl orthoformate and, if required, propellants such as propane, butane, nitrogen, compressed air, dimethyl ether, carbon dioxide, nitrous oxide, or mixtures of these gases.

The oil spray formulations differ from the aerosol recipes in that no propellants are used.

For use in spray compositions, the content of active ingredient is from 0.001 to 80 weights %, preferably from 0.01 to 50 weight % and most preferably from 0.01 to 15 weight %.

The compounds of formula I and its respective compositions can also be used in mosquito and fumigating coils, smoke cartridges, vaporizer plates or long-term vaporizers and also in moth papers, moth pads or other heat-independent vaporizer systems.

Seed treatment The compounds of formula I are also suitable for the treatment of seeds in order to protect the seed from insect pest, in particular from soil-living insect pests and the resulting plant's roots and shoots against soil pests and foliar insects.

The compounds of formula I are particularly useful for the protection of the seed from soil pests and the resulting plant's roots and shoots against soil pests and foliar insects. The protection of the resulting plant's roots and shoots is preferred. More preferred is the protection of resulting plant's shoots from piercing and sucking insects, wherein the protection from aphids is most preferred.

The present invention therefore comprises a method for the protection of seeds from insects, in particular from soil insects and of the seedlings' roots and shoots from insects, in particular from soil and foliar insects, said method comprising contacting the seeds before sowing and/or after pregermination with a compound of the general formula I or a salt thereof. Particularly preferred is a method, wherein the plant's roots and shoots are protected, more preferably a method, wherein the plants shoots are protected form piercing and sucking insects, most preferably aa method, wherein the plants shoots are protected from aphids.

The term seed embraces seeds and plant propagules of all kinds including but not limited to true seeds, seed pieces, suckers, corms, bulbs, fruit, tubers, grains, cuttings, cut shoots and the like and means in a preferred embodiment true seeds.

The term seed treatment comprises all suitable seed treatment techniques known in the art, such as seed dressing, seed coating, seed dusting, seed soaking and seed pelleting.

The present invention also comprises seeds coated with or containing the active compound.

The term "coated with and/or containing" generally signifies that the active ingredient is for the most part on the surface of the propagation product at the time of application, although a greater or lesser part of the ingredient may penetrate into the propagation product, depending on the method of application. When the said propagation product is (re)planted, it may absorb the active ingredient.

Suitable seed is seed of cereals, root crops, oil crops, vegetables, spices, ornamentals, for example seed of durum and other wheat, barley, oats, rye, maize (fodder maize and sugar maize / sweet and field corn), soybeans, oil crops, crucifers, cotton, sunflowers, bananas, rice, oilseed rape, turnip rape, sugarbeet, fodder beet, eggplants, potatoes, grass, lawn, turf, fodder grass, tomatoes, leeks, pumpkin/squash, cabbage, iceberg lettuce, pepper, cucumbers, melons, Brassica species, melons, beans, peas, garlic, onions, carrots, tuberous plants such as potatoes, sugar cane, tobacco, grapes, petunias, geranium/pelargoniums, pansies and impatiens. In addition, the active compound may also be used for the treatment seeds from plants, which tolerate the action of herbicides or fungicides or insecticides owing to breeding, including genetic engineering methods.

For example, the active compound can be employed in treatment of seeds from plants, which are resistant to herbicides from the group consisting of the sulfonylureas, imidazolinones, glufosinate-ammonium or glyphosate-isopropylammonium and analogous active substances (see for example, EP-A-0242236, EP-A-242246) (WO 92/00377) (EP-A-0257993, U.S. Pat. No. 5,013,659) or in transgenic crop plants, for example cotton, with the capability of producing Bacillus thuringiensis toxins (Bt toxins) which make the plants resistant to certain pests (E P-A-0142924, E P-A-0193259),

Furthermore, the active compound can be used also for the treatment of seeds from plants, which have modified characteristics in comparison with existing plants consist, which can be generated for example by traditional breeding methods and/or the generation of mutants, or by recombinant procedures). For example, a number of cases have been described of recombinant modifications of crop plants for the purpose of modifying the starch synthesized in the plants (e.g. WO 92/1 1376, WO 92/14827, WO 91/19806) or of transgenic crop plants having a modified fatty acid composition (WO 91/13972).

The seed treatment application of the active compound is carried out by spraying or dusting the seeds before sowing of the plants and before emergence of the plants.

In the treatment of seeds the corresponding formulations are applied by treating the seeds with an effective amount of the active compound. Herein, the application rates of the active compound are generally from 0,1 g to 10 kg per 100 kg of seed, preferably from 1 g to 5 kg per 100 kg of seed, in particular from 1 g to 2,5 kg per 100 kg of seed. For specific crops such as lettuce the rate can be higher.

Compositions which are useful for seed treatment are e.g.:

A Soluble concentrates (SL, LS)

D Emulsions (EW, EO, ES) E Suspensions (SC, OD, FS)

F Water-dispersible granules and water-soluble granules (WG, SG)

G Water-dispersible powders and water-soluble powders (WP, SP, WS)

H Dustable powders (DP, DS)

Conventional seed treatment formulations include for example flowable concentrates FS, solutions LS, powders for dry treatment DS, water dispersible powders for slurry treatment WS, water-soluble powders SS and emulsion ES and EC and gel formulation GF. These formulation can be applied to the seed diluted or undiluted. Application to the seeds is carried out before sowing, either directly on the seeds or after having pregerminated the latter

In a preferred embodiment a FS formulation is used for seed treatment. Typcially, a FS formulation may comprise 1-800 g/l of active ingredient, 1-200 g/l Surfactant, 0 to 200 g/l antifreezing agent, 0 to 400 g/l of binder, 0 to 200 g/l of a pigment and up to 1 liter of a solvent, preferably water.

Preferred FS formulations of compounds of formula I for seed treatment usually comprise from 0.1 to 80% by weight (1 to 800 g/L) of the active ingredient, from 0.1 to 20 % by weight (1 to 200 g/L) of at least one surfactant, e.g. 0.05 to 5 % by weight of a wetter and from 0.5 to 15 % by weight of a dispersing agent, up to 20 % by weight, e.g. from 5 to 20 % of an anti-freeze agent, from 0 to 15 % by weight, e.g. 1 to 15 % by weight of a pigment and/or a dye, from 0 to 40 % by weight, e.g. 1 to 40 % by weight of a binder (sticker /adhesion agent), optionally up to 5 % by weight, e.g. from 0.1 to 5 % by weight of a thickener, optionally from 0.1 to 2 % of an anti-foam agent, and optionally a preservative such as a biocide, antioxidant or the like, e.g. in an amount from 0.01 to 1 % by weight and a filler/vehicle up to 100 % by weight.

Seed Treatment formulations may additionally also comprise binders and optionally colorants.

Binders can be added to improve the adhesion of the active materials on the seeds after treatment. Suitable binders are homo- and copolymers from alkylene oxides like ethylene oxide or propylene oxide, polyvinylacetate, polyvinylalcohols, polyvinylpyrrolidones, and copolymers thereof, ethylene-vinyl acetate copolymers, acrylic homo- and copolymers, polyethyleneamines, polyethyleneamides and polyethyleneimines, polysaccharides like celluloses, tylose and starch, polyolefin homo- and copolymers like olefin/maleic anhydride copolymers, polyurethanes, polyesters, polystyrene homo and copolymers.

Optionally, also colorants can be included in the formulation. Suitable colorants or dyes for seed treatment formulations are Rhodamin B, C.I. Pigment Red 1 12, C.I. Solvent Red 1 , pigment blue 15:4, pigment blue 15:3, pigment blue 15:2, pigment blue 15:1 , pigment blue 80, pigment yellow 1 , pigment yellow 13, pigment red 1 12, pigment red 48:2, pigment red 48:1 , pigment red 57:1 , pigment red 53:1 , pigment orange 43, pigment orange 34, pigment orange 5, pigment green 36, pigment green 7, pigment white 6, pigment brown 25, basic violet 10, basic violet 49, acid red 51 , acid red 52, acid red 14, acid blue 9, acid yellow 23, basic red 10, basic red 108.

Examples of a gelling agent is carrageen (Satiagel^®) In the treatment of seed, the application rates of the compounds I are generally from 0.1 g to 10 kg per 100 kg of seed, preferably from 1 g to 5 kg per 100 kg of seed, in particular from 1 g to 1000 g per 100 kg of seed.

The invention therefore also relates to seed comprising a compound of the formula I, or an agriculturally useful salt of I, as defined herein. The amount of the compound I or the agriculturally useful salt thereof will in general vary from 0.1 g to 10 kg per 100 kg of seed, preferably from 1 g to 5 kg per 100 kg of seed, in particular from 1 g to 1000 g per 100 kg of seed.

The present invention is now illustrated in further details by the following examples.

I. Synthesis Examples

Example 1.1 : 2-Difluoromethoxy-6-prop-2-ynylsulfamoyl-thiobenzamide (4)

1.1. 2-Fluoro-6-methoxybenzonitrile:

640.5 g (4.6 mol) of difluorobenzonitrile have been dissolved in 3.5 I of methanol and then cooled to 0-5 °C. 828.8 g of 30% strength sodium methoxide solution have been added dropwise in this temperature range, and the reaction mixture has been stirred at room temperature overnight. Then the reaction mixture has been added to 20 I of water and the precipitate has been filtered off with suction and washed twice with water and twice with heptane. The solid has been dried in vacuo at 50 °C to yield 740 g (455 mmol) of the title compound as a white solid.

1.2. 2-Fluoro-6-hydroxybenzonitrile: 151 g (1 mol) of 2-fluoro-6-methoxybenzonitrile and 346.5 g (3 mol) of pyridinium hydrochloride have been introduced into a 2 I flask and then slowly heated to 190°C under a protective gas atmosphere and then stirred at this temperature for 5 h. The mixture has been cooled with slow stirring to room temperature overnight. Then 1000 ml of water have been added, and the mixture has been heated to 80°C. After adding 1000 ml of methyl tert-butyl ether, the phases have been are separated and the aqueous phase has been back-extracted twice with 500 ml of methyl tert-butyl ether. The combined methyl tert-butyl ether phases have been washed once with 800 ml of 10% strength NaOH and once with 400 ml of water. The two aqueous phases have been combined, adjusted to pH 2 with concentrated hydrochloric acid and washed three times with 500 ml of methylene chloride. Then, the combined organic phases have been washed once with 10% strength hydrochloric acid. The organic phase has been dried over sodium sulfate. Finally, the solvent has been distilled off in vacuo to give 120 g (870 mmol) of the desired product.

1.3. 2-Difluoromethoxy-6-fluorobenzonitrile:

150 g (1.1 mol) of 2-fluoro-6-hydroxybenzonitrile have been introduced into 2000 ml of ethylene glycol dimethyl ether. Then, 262.8 g (3.3 mol) of concentrated NaOH have been added dropwise. The reaction mixture has been heated to 65°C and 95 g (1.1 mol) of chlorodifluoromethane have been passed in. The mixture has been stirred at 65°C for one hour and at room temperature overnight. Then, the reaction mixture has been stirred into 3 I of water, followed by three times extraction with 800 ml of methyl tert-butyl ether. The combined organic phases have been washed twice with 500 ml of water, once with 250 ml of sodium chloride solution and dried over sodium sulfate. Finally, the solvent has been distilled off in vacuo to yield 21 1 g (1.1 mmol) of the desired product.

1.4. 2-Difluoromethoxy-6-propylsulfanylbenzonitrile:

180 g (0.96 mol) 2-difluoromethoxy-6-fluorobenzonitrile have been introduced into 1.5 I of dimethylformamide at room temperature. 73.2 g (0.96 mol) of propanethiol have been added dropwise and, after cooling to 0 °C, 70 g (1.25 mol) of potassium hydroxide pellets, dissolved in 600 ml of water, have been added dropwise at 0 °C. The mixture has been stirred for one hour and then warmed to room temperature. The reaction mixture has been stirred into 3.5 I of ice-water and extracted three times with 500 ml of methyl tert-butyl ether. The combined organic phases have been washed twice with 500 ml of 1 N hydrochloric acid and dried over sodium sulfate. Then, the solvent has been distilled off in vacuo. The oil obtained has been distilled in vacuo (b.p.: 180-185°C/0.5 mbar) to give 730 mmol of the title compound.

1.5. 2-Cyano-3-difluoromethoxyphenylsulfonyl chloride: A mixture of 100 ml of chlorobenzene and 20 ml of water has been cooled to 10°C and presaturated with gaseous chlorine. A solution of 20 g (0.08 mol) of 2-difluoro-methoxy- 6-propylsulfanylbenzonitrile in 200 ml of chlorobenzene has been added dropwise while passing chlorine through the solution. After 2 hours of stirring the conversion has been complete. The mixture has been cooled to 0-5 °C, dried over sodium sulfate and evaporated. The oily residue (27.8 g) contained byproducts formed from chlorobenzene but has been used without further purification for the next step. If necessary, the sulfonyl chloride could have been purified by column chromatography using cyclohexane and toluene as eluents.

1.6. N-Propargyl-2-cyano-3-difluoromethoxyphenylsulfonamide:

To a solution of 0.65 g (2.4 mmol) of purified 2-cyano-3-difluoromethoxyphenylsulfonyl chloride in 20 ml of tetrahydrofuran a solution of 274 mg (2.4 mmol) of dimethylamine and 510 mg of sodium carbonate in 15 ml of water has been added at room temperature. The reaction mixture has been stirred at room temperature for 5 minutes before water has been added. The aqueous phase has been acidified to pH = 1 using hydrochloric acid (10% strength by weight, aqueous solution). The aqueous phase has then been extracted three times with dichloromethane. The combined organic extracts have been dried over sodium sulfate and filtered. The filtrate has been concentrated in vacuo and the resulting residue has been triturated with methyl tert-butyl ether to yield 0.53 g (1.9 mmol) of the title compound having a melting point of 100-102°C.

1.7. 2-Difluoromethoxy-6-prop-2-ynylsulfamoyl-thiobenzamide (4): 0.46 g (1.52 mmol) of 2-(Ethyl-methyl-sulfamoyl)-3-fluoro-6-methoxy-benzonitrile was dissolved in 20 ml of pyridine. 1.9 ml (17.3 mmol) of triethylamine was added. Hydrogen sulphide was passed through the reaction mixture for 3 h. Then the reaction mixture was stirred at room temperature for 2 days. 60 ml of water was added to the solution. The aqueous mixture was extracted with ethyl acetate. The combined organic layers were washed with diluted aqueous HCI, water and brine. Then they were dried over Na2SU4 and filtered. The filtrate was concentrated in vacuo. The residue was purified by flash chromatography to give 0.20 g (0.61 mmol) of the title compound as colorless solid.

Example 1.2: 2-(Ethyl-methyl-sulfamoyl)-3-fluoro-6-methoxy-thiobenzamide (6)

2.1. 5-Fluoro-2-methoxy-1-cyano-phenyl sulfonyl chloride: 3.085 g (20 mmol) of (commercial available) 5-Fluoro-2-methoxybenzonitrile was dissolved in 20 ml of dry tetrahydrofurane under an argon atmosphere and cooled to - 78 °C. A solution of freshly prepared lithium diisopropyl amide (40 mmol in 20 ml of dry tetrahydrofurane) was added over a period of 10 min. The resulting solution was stirred at - 40 °C for 2 h and then was cooled to - 78 °C again. In a separate flask 20 ml of dry tetrahydrofurane was cooled to - 78 °C. Approximately 10 g of gaseous sulphur dioxide was added. Then the solution of the lithiated starting material from the first flask was added at - 78 °C drop wise via syringe. The resulting reaction mixture was stirred at 0 °C for 1 h. Then 5.51 g (40 mmol) of sulfurylchloride was added drop wise at 0 °C. The resulting reaction mixture was further stirred at room temperature for 30 min before the reaction was quenched by addition of water. After phase separation, the aqueous phase was extracted with dichloromethane. The combined organic layers were washed with brine, dried over Na2SU4 and evaporated. The crude sulfonyl chloride (6.6 g, 20 mmol, purity approx. 75%) was directly used in the subsequent step without further purification. If necessary, the sulfonyl chloride could have been purified by column chromatography using cyclohexane and toluene as eluents. 2.2. 2-(Ethyl-methyl-sulfamoyl)-3-fluoro-6-methoxy-benzonitrile:

1.49 g (20 mmol) of N-methylisopropyl amine were dissolved in 20 ml of tetrahydrofurane and cooled to 0 °C. A solution of 1.5 g (contains 4 mmol) of 5-Fluoro- 2-methoxy-1-cyano-phenyl sulfonyl chloride in 10 ml of tetrahydrofurane was added dropwise. The reaction mixture was stirred at 0 °C for 3 h before the reaction was quenched by addition of water. The aqueous solution was extracted with dichloromethane. The combined organic layers were washed with brine, dried over Na2SU4 and evaporated. The resulting residue was crystallized from ethyl eacetate/hexane to afford 0.97 g (3.2 mmol) of the title compound.

2.3. 2-(Ethyl-methyl-sulfamoyl)-3-fluoro-6-methoxy-thiobenzamide (6):

0.50 g (1.84 mmol) of 2-(Ethyl-methyl-sulfamoyl)-3-fluoro-6-methoxy-benzonitrile was dissolved in 20 ml of pyridine. 2.1 ml (17.3 mmol) of triethylamine was added. Hydrogen sulphide was passed through the reaction mixture for 3 h. Then the reaction mixture was stirred at room temperature for 3 days. 60 ml of water was added to the solution. The aqueous mixture was extracted with ethyl acetate. The combined organic layers were washed with diluted aqueous HCI, water and brine. Then they were dried over Na2SU4 and filtered. The filtrate was concentrated in vacuo. The residue was purified by flash chromatography to give 0.12 g (0.38 mmol) of the title compound as colourless solid.

The compounds nos. 1 to 7 of the formula I with X = C-R⁵ listed in the following table 1 were prepared analogously.

Table 1 :

Example 1.3: 3-(lsopropyl-methyl-sulfamoyl)-5-methoxy-thioisonicotinamide (9)

3.1. S.δ-Dichloro-isonicotinonitrile:

30.0 g (170.5 mmol) 3,5-dichloro-4-pyridine carbaldehyde was dissolved in 200 ml of formic acid. 15.4 g (221.6 mmol) of hydroxylamine hydrochloride and 2 drops of concentrate sulfuric acid were added and the resulting mixture was refluxed for 3.5 hours. The reaction mixture was cooled to room temperature, the solvent was evaporated under reduced pressure and the residue was redissolved in methyl tert- butyl ether. The resulting solution was washed with water, aqueous saturated solution of NaHCO₃ and again with water. The organic phase was dried over Na₂SO₄ and the solvent was evaporated under reduced pressure to give 28.3 g (163.6 mmol) of the title compound, which was used in the following reaction without further purification.

3.2. 3-Chloro-5-propylsulfanylisonicotinonitrile:

At - 78 °C, a solution of 6.47 g (85 mmol) of propane-1 -thiol in 100 ml of dry tetrahydrofuran was treated with 53.1 ml (85 mmol) of a 1.6 molar solution of n-butyl lithium in hexane. The resulting milky white suspension was allowed to warm to room temperature and stirred for additional 15 minutes. In a separate flask, 14.0 g (80.9 mmol) of 3,5-dichloro-isonicotinonitrile were dissolved in 100 ml of dry tetrahydrofuran. At room temperature, the lithium thiopropylate solution was slowly added over a period of 30 minutes. After the addition was complete, the resulting solution was stirred for further 1 hour, after which the reaction was quenched by addition of 200 ml of saturated aqueous NH₄CI solution. After addition of ethyl acetate, the phases were separated, and the aqueous layer was extracted three times with ethyl acetate. The combined organic layers were washed with saturated brine, dried over Na₂SO₄ and evaporated. The residue slowly crystallized to give 16.95 g (79.7 mmol) of the title compound without further purification.

3.3. 3-Methoxy-5-propylsulfanyl-isonicotinonitrile:

15.2 g (84.3 mmol) of a 30 % by weight solution of sodium methylate in methanol were dissolved in 50 ml of dry tetrahydrofuran. 17.9 g (84.3 mmol) of 3-chloro-5- propylsulfanyl-isonicotinonitrile dissolved in 150 ml of dry tetrahydrofuran were added at room temperature. The resulting mixture was refluxed for 2.5 hours. Then the mixture was cooled to room temperature and water was added. The aqueous mixture was extracted three times with ethyl acetate. The combined organic layers were washed with saturated brine, dried over Na2SU4 and evaporated. The residue was purified by flash chromatography to give 7.0 g (33.6 mmol) of the title compound as a colourless solid.

3.4. 4-Cyano-5-methoxypyridine-3-sulfonylchloride:

1.8 g (7.4 mmol) of S-methoxy-δ-propylsulfanylisonicotinonitrile was dissolved in 30 ml of dichloromethane and 3 ml of water. At 0 °C chlorine gas was passed through the reaction mixture for 1 h, whereupon the reaction mixture was stirred at 5 °C for 30 minutes. The reaction was quenched by addition of water. After phase separation, the aqueous layer was extracted three times with dichloromethane. The combined organic layers were washed with water and dried over Na2SU4 to afford 2.0 g (-6.6 mmol) of the title compound, which was used in the following reaction without further purification.

3.5. 4-Cyano-5-methoxypyridine-3-sulfonic acid methylisopropylamide:

A solution of 2.6 g (7.8 mmol) of 4-cyano-5-dimethoxy-pyridin-3-sulfonylchloride in 20 ml of tetrahydrofuran was added to a solution of 1.45 g (19.5 mmol) of methylisopropylamine in 20 ml of tetrahydrofuran at 0 °C. The reaction mixture was stirred at 0 °C for 2 hours whereupon water was added. Tetrahydrofuran was removed from the reaction mixture by evaporation. The resulting aqueous mixture was extracted three times with dichloromethane. The combined organic extracts were dried over Na2SU4 and filtered. The filtrate was concentrated in vacuo. The residue was purified by flash chromatography to give 1.05 g (3.7 mmol) of the title compound.

3.6. 3-(lsopropyl-methyl-sulfamoyl)-5-methoxy-thioisonicotinamide (9):

0.93 g (3.45 mmol) of 4-Cyano-5-methoxypyridine-3-sulfonic acid methylisopropylamide was dissolved in 30 ml of pyridine. 2.1 ml (17.3 mmol) of triethylamine was added. Hydrogen sulphide was passed through the reaction mixture for 3 h. Then the reaction mixture was stirred at room temperature for 3 days. 60 ml of water was added to the solution. The aqueous mixture was extracted with ethyl acetate. The combined organic layers were washed with diluted aqueous HCI, water and brine. Then they were dried over Na2SU4 and filtered. The filtrate was concentrated in vacuo. The residue was purified by flash chromatography to give 0.59 g (1.85 mmol) of the title compound as colourless solid.

The compounds nos. 8 to 10 of the formula I with X= N, listed in the following table 2 were prepared analogously to example 1.3.

Table 2:

II. Biological examples of action against pests

The active compounds were formulated in a mixture of 50 vol.-% acetone:50 vol.-% water. A nonionic surfactant (Kinetic®) was included in the solution at a volume of 0.01 % v/v.

In the following tests, the formulated solutions of the active compounds were diluted to an active ingredient concentration of 300 ppm and the diluted solutions were applied in the below mentioned tests.

The action of the compounds of the formula I against pests was demonstrated by the following experiments:

11.1 Cotton aphid (aphis gossypii), mixed life stages

Cotton plants at the cotyledon stage were infested prior to treatment by placing a heavily infested leaf from the main aphid colony on top of each cotyledon. The aphids were allowed to transfer overnight and the host leaf was removed. The infested cotyledons were then dipped and agitated in the test solution for 3 seconds and allowed to dry in a fume hood, est plants were maintained under fluorescent lighting in a 24-hr photoperiod at 25°C and 20-40% relative humidity. Aphid mortality on the treated plants, relative to mortality on untreated check plants, was determined after 5 days.

In this test each compound of examples 1-10 of tables 1 and 2 provided at 300 ppm least 90 % mortality of cotton aphid (Aphis gossypii, mixed life stages) in comparison with untreated controls.

11.2 Green Peach Aphid (Myzus persicae), mixed life stages

Bell pepper plants at the first true-leaf stage were infested prior to treatment by placing heavily infested leaves from the main aphid colony on top of the treatment plants. The aphids were allowed to transfer overnight to accomplish an infestation of 30-40 aphids per plant and the host leaves were removed. The infested leaves of the test plants were then dipped and agitated in the test solution for 3 seconds and allowed to dry in a fume hood. Test plants were maintained under fluorescent lighting in a 24-hr photoperiod at 25°C and 20-40% relative humidity. Aphid mortality on the treated plants, relative to mortality on untreated check plants, was determined after 5 days.

In this test each compound of examples 1-10 of tables 1 and 2 provided at 300 ppm at least 90 % mortality of green peach aphid in comparison with untreated controls.

II.3 Bean Aphid (Aphis fabae)

Nasturtium plants grown in Metro mix in the 1^st leaf-pair stage (variety 'Mixed Jewel') were infested with approximately 2-30 laboratory-reared aphids by placing infested cut plants on top of the test plants. The cut plants were removed after 24 hr. Each plant was dipped into the test solution to provide complete coverage of the foliage, stem, protruding seed surface and surrounding cube surface and allowed to dry in the fume hood. The treated plants were kept at about 25°C with continuous fluorescent light. Aphid mortality is determined after 3 days.

In this test each compound of examples 1-10 in tables 1 and 2 provided at 300 ppm at least 90 % mortality of bean aphid in comparison with untreated controls.

Claims

We claim:

1. A thioamide compound of the formula I

wherein

X is N, NO or C-R⁵

R¹ and R² are, independently of one another, selected from the group consisting of hydrogen, C(=O)-R⁷, Ci-Cio-alkyl, C₂-Cio-alkenyl, C₂-Cio-alkinyl, Ci-Cio-alkoxy or C3-Cio-cycloalkyl, wherein the five last-mentioned radicals may be unsubstituted, partially or fully halogenated and/or may carry 1 , 2 or 3 radicals, independently of one another each selected from the group consisting of cyano, nitro, amino, C1-C10- alkoxy, Ci-Cio-alkylthio, Ci-Cio-alkylsulfinyl, Ci-Cio-alkylsulfonyl, Ci- Cio-haloalkoxy, Ci-Cio-haloalkylthio, Ci-Cio-alkoxycarbonyl, (C1-C10- alkyl)amino, di-(Ci-Cio-alkyl)amino, C3-Cio-cycloalkyl and phenyl, it being possible for phenyl to be unsubstituted, partially or fully halogenated and/or to carry 1 , 2 or 3 substituents, independently of one another selected from the group consisting of Ci-C4-alkyl, C1-C4- haloalkyl, Ci-C4-alkoxy and Ci-C4-haloalkoxy; or wherein R¹ and R² together with the adjacent nitrogen form a 3 to 10- membered ring, optionally substituted by 1 , 2 or 3 Ci-Cs-alkyl radicals, wherein the ring may contain, in addition to the nitrogen and carbon ring members, 1 , 2 or 3 heteroatoms as ring members selected from the group consisting of nitrogen, oxygen, sulfur, a group SO, SO₂ or N-R⁸;

R³ is hydrogen, nitro, cyano, azido, amino, halogen, sulfonylamino, sulfenylamino, sulfinylamino, C(=O)R⁷ , Ci-Cδ-alkyl, C₂-C6-alkenyl, C₂-Cδ- alkinyl, Ca-Cs-cycloalkyl, Ci-Cβ-alkoxy, Ci-Cβ-alkylthio, (Ci-C6-alkyl)amino, di(Ci-C6-alkyl)amino, C 1 -Ce-a I ky I s u If i nyl , Ci-Cβ-alkylsulfenyl or Ci-Cβ- alkylsulfonyl, wherein the eleven last-mentioned radicals may be unsubstituted, partially or fully halogenated and/or may carry 1 , 2 or 3 radicals, selected from the group consisting of cyano, nitro, amino, C1-C4- alkoxy, Ci-C4-alkylthio, Ci-C4-alkylsulfinyl, Ci-C4-alkylsulfonyl, CrC₄- haloalkoxy, Ci-C4-haloalkylthio, (Ci-C4-alkoxy)carbonyl, (Ci-C4-alkyl)amino, di(Ci-C4-alkyl)amino, Ca-Cs-cycloalkyl and phenyl, it being possible for phenyl to be unsubstituted, partially or fully halogenated and/or to carry 1 , 2 or 3 substituents, independently of one another selected from the group consisting of Ci-C4-alkyl, Ci-C4-haloalkyl, Ci-C4-alkoxy and CrC₄- haloalkoxy;

R⁴, R⁵ and R⁶ are independently of one another selected from the group consisting of hydrogen, halogen, cyano, azido, nitro, Ci-Cβ- alkyl, C₃-C₈-cycloalkyl, Ci-C₄-haloalkyl, Ci-C₄-alkoxy, CrC₄- alkylthio, Ci-C₄-alkylsulfinyl, Ci-C₄-alkylsulfonyl, CrC₄- haloalkoxy, CrC₄-haloalkylthio, C2-C6-alkenyl, C2-C6-alkinyl, (CrC₄-alkoxy)carbonyl, amino, (CrC₄-alkyl)amino, di(Ci-C₄- alkyl)amino, aminocarbonyl, (CrC₄-alkyl)aminocarbonyl, di(d-

C₄-alkyl)aminocarbonyl, sulfonyl, sulfonylamino, sulfenylamino, sulfanylamino and C(=O)-R⁷;

R⁷ is hydrogen, hydroxy, CrCs-alkoxy, amino, CrC₄-alkyl, aryl, aryl-Ci-C₄- alkyl, a 3- to 7-membered heteroaryl or heteroaryl-CrC₄ -alkyl, wherein the heteroaryl ring contains as ring members 1 ,2 or 3 heteroatoms, selected from the group consisting of nitrogen, oxygen, sulfur, a group SO, SO2 or N-R⁸; a 3- to 7-membered heterocyclyl or heterocyclyl-CrC₄-alkyl, wherein the heterocyclic ring contains as ring members 1 ,

2 or 3 heteroatoms, selected from the group consisting of nitrogen, oxygen, sulfur, a group SO, SO2 or N-R⁸ and wherein the carbon atoms of the heterocyclic rings may by unsubstituted or substituted by one or two CrC₄-alkyl groups;

R⁸ is hydrogen or CrC₄-alkyl

and/or the enantiomers, diastereomers or salts thereof.

A thioamide compound of the formula I according to claim 1 , wherein R¹ and R² are, independently of one another, selected from the group consisting of hydrogen, CrCralkyl, CrCrhaloalkyl, C2-C6-alkenyl, C2-C6-haloalkenyl, C2-C6- alkinyl, C₂-C₆-haloalkinyl, C₃-C₆-cycloalkyl, Ci-C₄-alkoxy-CrC₄-alkyl, CrC₄- alkylthio-CrC₄-alkyl and C(=O)-R⁷, wherein R⁷ is CrC₄-alkyl, CrCa-alkoxy-CrCa- alkyl, CrCa-alkylthio-CrCa-alkyl or CrC₄-haloalkyl.

3. A thioamide compound of the formula I according to claim 1 , wherein R¹ and R² are, independently of one another, selected from the group consisting of hydrogen, Ci-C4-alkyl, C2-C4-alkinyl and C(=O)-R⁷, wherein R⁷ is selected from Ci-C₄-alkyl, Ci-C₃-alkoxy-Ci-C₃-alkyl, Ci-C₃-alkylthio-Ci-C₃-alkyl and CrC₄- haloalkyl.

4. A thioamide compound of the formula I according to claim 1 , wherein R¹ and R² are, independently of one another, selected from the group consisting of hydrogen, methyl, ethyl, 1-methylethyl, cyclopropyl or prop-3-yn-1-yl.

5. A thioamide compound of the formula I according to claim 1 , wherein one or both of R¹ and R² are C(=O)-R⁷, and wherein R⁷ is selected from Ci-C₄-alkyl, CrC₃- alkoxy-CrC₃-alkyl, Ci-C₃-alkylthio-CrC₃-alkyl or CrC₄-haloalkyl.

6. A thioamide compound of the formula I according to claim 1 , wherein one or both of R¹ and R² are selected from C(=O)-R⁷, and wherein R⁷ is selected from methyl, ethyl, 1-methylethyl, 2-methylpropan-2-yl, 2-methoxyethyl, 2-methylthioethyl, trifluoromethyl or trichloromethyl.

7. A thioamide compound of the formula I according to claim 1 , wherein R³ is halogen, CrC₄-alkyl, CrC₄-haloalkyl, CrC₄-alkoxy or CrC₄-haloalkoxy.

8. A thioamide compound of the formula I according to claim 1 , wherein R³ is halogen, CrC2-alkyl, d-haloalkyl, CrC2-alkoxy or Crhaloalkoxy.

9. A thioamide compound of the formula I according to claim 1 , wherein R³ is methyl, trifluoromethyl, trichloromethyl, methoxy, trifluoromethoxy, difluoromethoxy, fluoromethoxy or chlorodifluoromethoxy, chlorine or fluorine.

10. A thioamide compound of the formula I according to claim 1 , wherein X is N and R⁴ and R⁶ are selected, independently from each other, from hydrogen, halogen, CrC₄-alkyl, CrC₄-haloalkyl, CrC₄-alkoxy or Cr C₄-haloalkoxy.

1 1. A thioamide compound of the formula I according to claim 1 , wherein X is N and R⁴ and R⁶ are selected, independently from each other, from hydrogen, halogen,

CrC2-alkyl, or d-haloalkyl.

12. A thioamide compound of the formula I according to claim 1 , wherein X is N and R⁴ and R⁶ are selected, independently from each other, from H, Cl, Br, I, CH₃ or CF₃.

13. A thioamide compound of the formula I according to claim 1 , wherein X is N and wherein one or both of the radicals R⁴ or R⁶ being present are hydrogen.

14. A thioamide compound of the formula I according to claim 1 , wherein X is C-R⁵ and wherein R⁴, R⁵, and R⁶ are selected, independently from each other, from hydrogen, halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, Ci-C4-alkoxy or C1-C4- haloalkoxy.

15. A thioamide compound of the formula I according to claim 1 , wherein X is C-R⁵ and wherein R⁴, R⁵, and R⁶ are selected, independently from each other, from hydrogen, halogen, Ci-C2-alkyl or Ci-haloalkyl.

16. A thioamide compound of the formula I according to claim 1 , wherein X is C-R⁵ and wherein R⁴, R⁵, and R⁶ are selected, independently from each other, from H, CI₁ Br₁ I₁ CH₃ Or CF₃.

17. A thioamide compound of the formula I according to claim 1 , wherein X is C-R⁵ and at least two or all three of the radicals R⁴, R⁵ or R⁶ being present are hydrogen.

18. A composition comprising at least one thioamide compound of the formula I as defined in any one of claims 1 to 17 or an enantiomer, diastereomer and/or salt thereof and at least one inert liquid and/or solid carrier.

19. An agricultural composition comprising such a pesticidal effective amount of at least one compound of the formula I and/or its enantiomer, diastereomer or agriculturally useful salt of I, as defined in any of claims 1 to 17, and at least one inert liquid and/or solid agriculturally acceptable carrier and, if desired, at least one surfactant.

20. A method of combating animal pests which comprises contacting the animal pests, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal attack or infestation with a pesticidally effective amount of at least one thioamide compound of the formula I, as defined in any of claims 1 to 17, or its enantiomer, diastereomer or at least one agriculturally acceptable salt thereof.

21. A method as defined in claim 21 , where the animal pest is from the order Homoptera or Thysanoptera.

22. A method for protecting crops from attack or infestation by animal pests, which comprises contacting a crop with a pesticidal effective amount of at least one thioamide compound of the formula I as defined in claims 1-17 and/or its enantiomer, diastereomer or at least one agricultural acceptable salt thereof.

23. A method for the protection of seeds from soil insects and of the seedlings' roots and shoots from insects comprising contacting the seeds before sowing and/or after pregermination with a thioamide compound of the formula I as defined in any of claims 1 to 17, or its enantiomers, diastereomers or at least one agriculturally acceptable salt thereof in a pesticidal effective amount.

24. The method according toclaim 24, wherein the compound of formula I is applied in an amount of from 100 mg to 10 kg per 100 kg of seeds.

25. A method according to claims 24 or 25, wherein of the resulting plant' s roots and shoots are protected.

26. A method according to claims 24 to 26, wherein the resulting plant' s shoots are protected from aphids.

27. Seed comprising a compound of the formula I as defined in any of claims 1 to 17 or its enantiomer, diastereomer or agriculturally useful salt thereof in an amount of from 0.1 g to 10 kg per 100 kg of seed.