WO2006089215A3 - Compositions pharmaceutiques et procedes associes - Google Patents

Compositions pharmaceutiques et procedes associes Download PDF

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Publication number
WO2006089215A3
WO2006089215A3 PCT/US2006/005821 US2006005821W WO2006089215A3 WO 2006089215 A3 WO2006089215 A3 WO 2006089215A3 US 2006005821 W US2006005821 W US 2006005821W WO 2006089215 A3 WO2006089215 A3 WO 2006089215A3
Authority
WO
WIPO (PCT)
Prior art keywords
methods
pharmaceutical compositions
disclosed
effective amount
composition
Prior art date
Application number
PCT/US2006/005821
Other languages
English (en)
Other versions
WO2006089215A2 (fr
Inventor
Vinod V Tuliani
Michael A Brandley
Original Assignee
Glaxo Group Ltd
Vinod V Tuliani
Michael A Brandley
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd, Vinod V Tuliani, Michael A Brandley filed Critical Glaxo Group Ltd
Publication of WO2006089215A2 publication Critical patent/WO2006089215A2/fr
Publication of WO2006089215A3 publication Critical patent/WO2006089215A3/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/38Heterocyclic compounds having sulfur as a ring hetero atom
    • A61K31/381Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2009Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Inorganic Chemistry (AREA)
  • Organic Chemistry (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

L'invention porte, entre autres, sur une composition pharmaceutique qui se présente sous la forme d'un comprimé contenant une quantité efficace d'un composé A, un polymère gonflant, un polymère de matrice, un agent flottant, et facultativement un diluant, un liant, un glissant, et/ou un lubrifiant. L'invention porte aussi sur un procédé de traitement ou de prévention de troubles thromboemboliques consistant à administrer une quantité efficace de la composition à un patient qui en a besoin.
PCT/US2006/005821 2005-02-18 2006-02-17 Compositions pharmaceutiques et procedes associes WO2006089215A2 (fr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US65427905P 2005-02-18 2005-02-18
US60/654,279 2005-02-18
US69612105P 2005-07-01 2005-07-01
US60/696,121 2005-07-01

Publications (2)

Publication Number Publication Date
WO2006089215A2 WO2006089215A2 (fr) 2006-08-24
WO2006089215A3 true WO2006089215A3 (fr) 2006-11-23

Family

ID=36917125

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/US2006/005821 WO2006089215A2 (fr) 2005-02-18 2006-02-17 Compositions pharmaceutiques et procedes associes

Country Status (4)

Country Link
AR (1) AR054226A1 (fr)
PE (1) PE20061010A1 (fr)
TW (1) TW200640449A (fr)
WO (1) WO2006089215A2 (fr)

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5169838A (en) * 1989-09-22 1992-12-08 Fournier Industrie Et Sante Benzopyranone-β-D-thioxylosides and their use in therapy
US6602899B1 (en) * 1999-11-17 2003-08-05 Fournier Industrie & Sante β-D-5 thioxylose derivatives, preparation method and therapeutic use

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5169838A (en) * 1989-09-22 1992-12-08 Fournier Industrie Et Sante Benzopyranone-β-D-thioxylosides and their use in therapy
US6602899B1 (en) * 1999-11-17 2003-08-05 Fournier Industrie & Sante β-D-5 thioxylose derivatives, preparation method and therapeutic use

Also Published As

Publication number Publication date
WO2006089215A2 (fr) 2006-08-24
AR054226A1 (es) 2007-06-13
TW200640449A (en) 2006-12-01
PE20061010A1 (es) 2006-11-11

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