WO2002088125A3 - Triazolopyrimidine mit fungizider wirkung - Google Patents

Triazolopyrimidine mit fungizider wirkung Download PDF

Info

Publication number
WO2002088125A3
WO2002088125A3 PCT/EP2002/004187 EP0204187W WO02088125A3 WO 2002088125 A3 WO2002088125 A3 WO 2002088125A3 EP 0204187 W EP0204187 W EP 0204187W WO 02088125 A3 WO02088125 A3 WO 02088125A3
Authority
WO
WIPO (PCT)
Prior art keywords
triazolopyrimidines
novel
fungicidal effect
producing
methods
Prior art date
Application number
PCT/EP2002/004187
Other languages
English (en)
French (fr)
Other versions
WO2002088125A2 (de
Inventor
Olaf Gebauer
Joerg Nico Greul
Ulrich Heinemann
Hans-Ludwig Elbe
Bernd-Wieland Krueger
Ralf Dunkel
Arnd Voerste
Ronald Ebbert
Astrid Mauler-Machnik
Ulrike Wachendorff-Neumann
Karl-Heinz Kuck
Yoshinori Kitagawa
Original Assignee
Bayer Ag
Olaf Gebauer
Joerg Nico Greul
Ulrich Heinemann
Hans-Ludwig Elbe
Bernd-Wieland Krueger
Ralf Dunkel
Arnd Voerste
Ronald Ebbert
Astrid Mauler-Machnik
Ulrike Wachendorff-Neumann
Karl-Heinz Kuck
Yoshinori Kitagawa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag, Olaf Gebauer, Joerg Nico Greul, Ulrich Heinemann, Hans-Ludwig Elbe, Bernd-Wieland Krueger, Ralf Dunkel, Arnd Voerste, Ronald Ebbert, Astrid Mauler-Machnik, Ulrike Wachendorff-Neumann, Karl-Heinz Kuck, Yoshinori Kitagawa filed Critical Bayer Ag
Priority to EP02737963A priority Critical patent/EP1397362A2/de
Priority to JP2002585424A priority patent/JP2004533436A/ja
Priority to US10/475,317 priority patent/US7189680B2/en
Priority to AU2002312826A priority patent/AU2002312826A1/en
Publication of WO2002088125A2 publication Critical patent/WO2002088125A2/de
Publication of WO2002088125A3 publication Critical patent/WO2002088125A3/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/02—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having no bond to a nitrogen atom
    • A01N47/04—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having no bond to a nitrogen atom containing >N—S—C≡(Hal)3 groups
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/34—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the groups, e.g. biuret; Thio analogues thereof; Urea-aldehyde condensation products
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/01—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms
    • C07C211/02—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C211/15—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton the carbon skeleton being further substituted by halogen atoms or by nitro or nitroso groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/01—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms
    • C07C211/20—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an acyclic unsaturated carbon skeleton
    • C07C211/24—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an acyclic unsaturated carbon skeleton the carbon skeleton being further substituted by halogen atoms or by nitro or nitroso groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C239/00—Compounds containing nitrogen-to-halogen bonds; Hydroxylamino compounds or ethers or esters thereof
    • C07C239/08—Hydroxylamino compounds or their ethers or esters
    • C07C239/20—Hydroxylamino compounds or their ethers or esters having oxygen atoms of hydroxylamino groups etherified
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06—Esters of carbamic acids
    • C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C271/12—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06—Esters of carbamic acids
    • C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
    • C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C271/16—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by singly-bound oxygen atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Neue Triazolopyrimidine der Formel (I), in welcher R?1, R2, R3¿ und X die in der Beschreibung angegebenen Bedeutungen haben sowie Säureadditions-Salze davon, mehrere Verfahren zur Herstellung dieser neuen Stoffe und deren Verwendung zur Bekämpfung von unerwünschten Mikroorganismen. Neue Amine und Carbamate der in der Beschreibung angegebenen Formeln sowie Verfahren zur Herstellung dieser Zwischenprodukte.
PCT/EP2002/004187 2001-04-27 2002-04-16 Triazolopyrimidine mit fungizider wirkung WO2002088125A2 (de)

Priority Applications (4)

Application Number Priority Date Filing Date Title
EP02737963A EP1397362A2 (de) 2001-04-27 2002-04-16 Triazolopyrimidine mit fungizider wirkung
JP2002585424A JP2004533436A (ja) 2001-04-27 2002-04-16 殺真菌作用を有するトリアゾロピリミジン
US10/475,317 US7189680B2 (en) 2001-04-27 2002-04-16 5-halo-6-aryl[1,2,4]triazolo[1,5-a]pyrimidin-7-amines
AU2002312826A AU2002312826A1 (en) 2001-04-27 2002-04-16 Triazolopyrimidines having a fungicidal effect

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10121101.5 2001-04-27
DE10121101A DE10121101A1 (de) 2001-04-27 2001-04-27 Triazolopyrimidine

Publications (2)

Publication Number Publication Date
WO2002088125A2 WO2002088125A2 (de) 2002-11-07
WO2002088125A3 true WO2002088125A3 (de) 2003-02-13

Family

ID=7683228

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/EP2002/004187 WO2002088125A2 (de) 2001-04-27 2002-04-16 Triazolopyrimidine mit fungizider wirkung

Country Status (6)

Country Link
US (1) US7189680B2 (de)
EP (1) EP1397362A2 (de)
JP (1) JP2004533436A (de)
AU (1) AU2002312826A1 (de)
DE (1) DE10121101A1 (de)
WO (1) WO2002088125A2 (de)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUP0300798A3 (en) * 2000-06-30 2006-02-28 Wyeth Corp Substituted-triazolopyrimidines and their use as anticancer agents and pharmaceutical compositions containing them
US7139344B2 (en) * 2001-05-16 2006-11-21 Lexmark International, Inc. Method and apparatus for effecting synchronous pulse generation for use in variable speed serial communications
GB0230020D0 (en) 2002-12-23 2003-01-29 Syngenta Ltd Fungicides
GB0230021D0 (en) * 2002-12-23 2003-01-29 Syngenta Ltd Fungicides
GB0230018D0 (en) 2002-12-23 2003-01-29 Syngenta Ltd Fungicides
DE10360370A1 (de) * 2003-12-22 2005-07-14 Bayer Cropscience Ag Triazolopyrimidine
US20070249634A1 (en) * 2004-06-09 2007-10-25 Carsten Blettner Triazolopyrimidine Compounds and Use Thereof for Controlling Harmful Fungi
EP1920654A1 (de) 2006-09-13 2008-05-14 Syngeta Participations AG Neue Pyridopyrazine N-Oxide
WO2008092836A2 (en) * 2007-01-30 2008-08-07 Basf Se Method for improving plant health
EP1952691A3 (de) * 2007-01-31 2008-09-17 Basf Se Verfahren zur Verbesserung der Gesundheit von Pflanzen unter Verwendung eines Triazolopyrimidin-Derivats

Citations (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3178467A (en) * 1961-03-07 1965-04-13 Du Pont N-alkylidene and arylidene-n-alkoxy and alkenoxy-n-methylammonium salts
US4408055A (en) * 1979-11-17 1983-10-04 Bayer Aktiengesellschaft Azolyloxy-carboxylic acid n-oxy-amide compounds
EP0550113A2 (de) * 1991-12-30 1993-07-07 Shell Internationale Researchmaatschappij B.V. Triazolopyrimidinderivate mit fungizider Aktivität
US5612345A (en) * 1993-03-04 1997-03-18 Shell Internationale Research Maatschappij B.V. Dihalotriazolopyrimidine derivatives as fungicides
WO1998046608A1 (en) * 1997-04-14 1998-10-22 American Cyanamid Company Fungicidal trifluoromethylalkylamino-triazolopyrimidines
WO1998046607A1 (en) * 1997-04-14 1998-10-22 American Cyanamid Company Fungicidal trifluorophenyl-triazolopyrimidines
US6020338A (en) * 1998-02-11 2000-02-01 American Cyanamid Company Fungicidal 7-alkyl-triazolopyrimidines

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL254901A (de) * 1959-08-24
FR1592328A (de) * 1968-11-19 1970-05-11
US5593996A (en) * 1991-12-30 1997-01-14 American Cyanamid Company Triazolopyrimidine derivatives
IL108731A (en) * 1993-03-04 1997-03-18 Shell Int Research 6, N-DISUBSTITUTED-£1, 2, 4| TRIAZOLO-£1, 5-a| PYRIMIDINE- 7-AMINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS FUNGICIDES
RU2147584C1 (ru) * 1995-10-27 2000-04-20 Американ Цианамид Компани Способ получения дигалоидазолопиримидинов и способ получения дигидроксиазолопиримидинов
US5817663A (en) * 1996-10-07 1998-10-06 American Cyanamid Company Pentafluorophenylazolopyrimidines
HUP0300798A3 (en) * 2000-06-30 2006-02-28 Wyeth Corp Substituted-triazolopyrimidines and their use as anticancer agents and pharmaceutical compositions containing them

Patent Citations (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3178467A (en) * 1961-03-07 1965-04-13 Du Pont N-alkylidene and arylidene-n-alkoxy and alkenoxy-n-methylammonium salts
US4408055A (en) * 1979-11-17 1983-10-04 Bayer Aktiengesellschaft Azolyloxy-carboxylic acid n-oxy-amide compounds
EP0550113A2 (de) * 1991-12-30 1993-07-07 Shell Internationale Researchmaatschappij B.V. Triazolopyrimidinderivate mit fungizider Aktivität
US5612345A (en) * 1993-03-04 1997-03-18 Shell Internationale Research Maatschappij B.V. Dihalotriazolopyrimidine derivatives as fungicides
WO1998046608A1 (en) * 1997-04-14 1998-10-22 American Cyanamid Company Fungicidal trifluoromethylalkylamino-triazolopyrimidines
WO1998046607A1 (en) * 1997-04-14 1998-10-22 American Cyanamid Company Fungicidal trifluorophenyl-triazolopyrimidines
US6020338A (en) * 1998-02-11 2000-02-01 American Cyanamid Company Fungicidal 7-alkyl-triazolopyrimidines

Also Published As

Publication number Publication date
US7189680B2 (en) 2007-03-13
US20040176398A1 (en) 2004-09-09
EP1397362A2 (de) 2004-03-17
AU2002312826A1 (en) 2002-11-11
JP2004533436A (ja) 2004-11-04
DE10121101A1 (de) 2002-10-31
WO2002088125A2 (de) 2002-11-07

Similar Documents

Publication Publication Date Title
WO2003051846A3 (de) Substituierte phenylderivate
WO2001090071A3 (de) Substituierte iminoazine als herbizide
WO2005061443A3 (de) Benzoylsubstituierte phenylalanin-amide
IL176062A0 (en) Dpp-iv inhibitors
WO2003016282A3 (en) Substituted 1h-dihydropyrazoles, their preparation and use
WO1999064409A3 (de) Benzothiepin-1,1-dioxidderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung
WO2003084922A8 (de) Acyl-4-carboxy-phenyl-harnstoffderivate, verfahren zu deren herstellung und deren verwendung
WO2002100860A3 (fr) Composes heterocycliques, leur preparation et leur utilisation comme medicaments, notamment comme anti-bacteriens
EP1382603A4 (de) Stickstoffhaltige verbindung mit kondensiertem ring und pyrazolylgruppe als substituent und medizinische zusammensetzung davon
HK1155146A1 (zh) 作為藥物活性劑的茚衍生物
WO2002088127A3 (de) Triazolopyrimidine
MX2007000240A (es) Derivados de [1.2]-oxazin-3,5-diona y dihidropirona sustituidos con fenilo.
WO2006119309A3 (en) 19,26,27-TRINOR-1α,25-DIHYDROXYVITAMIN D3 COMPOUNDS
WO2001077090A3 (en) Isothiazole derivatives and their use as microbicides
WO2002088125A3 (de) Triazolopyrimidine mit fungizider wirkung
WO2001090102A3 (de) 6-heterocyclyl-3-oxo-3,4-dihydro-chinoxaline
ATE353330T1 (de) Triazolopyrimidine fungizide
WO2002014313A3 (de) Neue beta-amyloid inhibitoren, verfahren zu deren herstellung und deren verwendung als arzneimittel
WO2008023003A8 (de) Arzneimittelkombinationen zur behandlung von atemwegserkrankungen
ZA200604654B (en) Pyrazolopyrimidines
WO1999037291A3 (de) Verwendung von substituierten sulfonamiden als antivirale mittel und neue stoffe
WO2002046152A3 (de) Coniosetin und derivate davon, verfahren zur herstellung und verwendung derselben
WO2003017766A3 (de) Herbizide auf basis von substituierten arylketonen
WO2002010160A3 (de) Substituierte heterocyclylalkylamino-1,3,5-triazine
WO2003014094A3 (de) Heterocyclylarylsulfonamide

Legal Events

Date Code Title Description
AK Designated states

Kind code of ref document: A2

Designated state(s): AE AG AL AM AT AU AZ BA BB BG BR BY BZ CA CH CN CO CR CU CZ DE DK DM DZ EC EE ES FI GB GD GE GH GM HR HU ID IL IN IS JP KE KG KP KR KZ LC LK LR LS LT LU LV MA MD MG MK MN MW MX MZ NO NZ OM PH PL PT RO RU SD SE SG SI SK SL TJ TM TN TR TT TZ UA UG US UZ VN YU ZA ZM ZW

AL Designated countries for regional patents

Kind code of ref document: A2

Designated state(s): GH GM KE LS MW MZ SD SL SZ TZ UG ZM ZW AM AZ BY KG KZ MD RU TJ TM AT BE CH CY DE DK ES FI FR GB GR IE IT LU MC NL PT SE TR BF BJ CF CG CI CM GA GN GQ GW ML MR NE SN TD TG

DFPE Request for preliminary examination filed prior to expiration of 19th month from priority date (pct application filed before 20040101)
121 Ep: the epo has been informed by wipo that ep was designated in this application
AK Designated states

Kind code of ref document: A3

Designated state(s): AE AG AL AM AT AU AZ BA BB BG BR BY BZ CA CH CN CO CR CU CZ DE DK DM DZ EC EE ES FI GB GD GE GH GM HR HU ID IL IN IS JP KE KG KP KR KZ LC LK LR LS LT LU LV MA MD MG MK MN MW MX MZ NO NZ OM PH PL PT RO RU SD SE SG SI SK SL TJ TM TN TR TT TZ UA UG US UZ VN YU ZA ZM ZW

AL Designated countries for regional patents

Kind code of ref document: A3

Designated state(s): GH GM KE LS MW MZ SD SL SZ TZ UG ZM ZW AM AZ BY KG KZ MD RU TJ TM AT BE CH CY DE DK ES FI FR GB GR IE IT LU MC NL PT SE TR BF BJ CF CG CI CM GA GN GQ GW ML MR NE SN TD TG

WWE Wipo information: entry into national phase

Ref document number: 2002737963

Country of ref document: EP

WWE Wipo information: entry into national phase

Ref document number: 2002585424

Country of ref document: JP

REG Reference to national code

Ref country code: DE

Ref legal event code: 8642

WWP Wipo information: published in national office

Ref document number: 2002737963

Country of ref document: EP

WWE Wipo information: entry into national phase

Ref document number: 10475317

Country of ref document: US