WO2002088091A3 - Inhibitors of human rhinovirus 2a cysteine protease - Google Patents
Inhibitors of human rhinovirus 2a cysteine protease Download PDFInfo
- Publication number
- WO2002088091A3 WO2002088091A3 PCT/US2002/013270 US0213270W WO02088091A3 WO 2002088091 A3 WO2002088091 A3 WO 2002088091A3 US 0213270 W US0213270 W US 0213270W WO 02088091 A3 WO02088091 A3 WO 02088091A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- human rhinovirus
- inhibitors
- halo
- amino
- cysteine protease
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
- C07D231/20—One oxygen atom attached in position 3 or 5
- C07D231/22—One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms
- C07D231/26—1-Phenyl-3-methyl-5- pyrazolones, unsubstituted or substituted on the phenyl ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
- C07D231/20—One oxygen atom attached in position 3 or 5
- C07D231/22—One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US28708301P | 2001-04-26 | 2001-04-26 | |
US60/287,083 | 2001-04-26 |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2002088091A2 WO2002088091A2 (en) | 2002-11-07 |
WO2002088091A3 true WO2002088091A3 (en) | 2002-12-19 |
Family
ID=23101374
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/US2002/013270 WO2002088091A2 (en) | 2001-04-26 | 2002-04-26 | Inhibitors of human rhinovirus 2a cysteine protease |
Country Status (1)
Country | Link |
---|---|
WO (1) | WO2002088091A2 (en) |
-
2002
- 2002-04-26 WO PCT/US2002/013270 patent/WO2002088091A2/en not_active Application Discontinuation
Non-Patent Citations (4)
Title |
---|
DATABASE CAPLUS [online] TANAKA E. ET AL.: "Comparison of trimethadione and antipyrine as indicators of oxidative drug metabolizing capacity in man", XP002958361, accession no. STN Database accession no. 1989:508460 * |
DATABASE CAPLUS [online] USUI Y. ET AL.: "Fungicides. XII. Synthesis and antifungal activity of halogen-substituted phenylpyrazolone derivatives", XP002958362, accession no. STN Database accession no. 1967:411452 * |
EUR. J. OF CLIN. PHARM., vol. 36, no. 6, 1989, pages 29 - 32 * |
YAKAGAKU ZASSHI, vol. 87, no. 1, 1967, pages 38 - 42 * |
Also Published As
Publication number | Publication date |
---|---|
WO2002088091A2 (en) | 2002-11-07 |
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