WO2001017965A3 - Cyanopiperidines - Google Patents
Cyanopiperidines Download PDFInfo
- Publication number
- WO2001017965A3 WO2001017965A3 PCT/EP2000/008660 EP0008660W WO0117965A3 WO 2001017965 A3 WO2001017965 A3 WO 2001017965A3 EP 0008660 W EP0008660 W EP 0008660W WO 0117965 A3 WO0117965 A3 WO 0117965A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- cyanopiperidines
- pesticides
- compounds
- preparation
- pests
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
- A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
- A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
- A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
- A01N47/16—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof the nitrogen atom being part of a heterocyclic ring
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
- A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
- A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
- A01N47/38—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< where at least one nitrogen atom is part of a heterocyclic ring; Thio analogues thereof
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N53/00—Biocides, pest repellants or attractants, or plant growth regulators containing cyclopropane carboxylic acids or derivatives thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- Plant Pathology (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Agronomy & Crop Science (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
AU75147/00A AU7514700A (en) | 1999-09-07 | 2000-09-05 | Cyanopiperidines |
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH163999 | 1999-09-07 | ||
CH1639/99 | 1999-09-07 |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2001017965A2 WO2001017965A2 (fr) | 2001-03-15 |
WO2001017965A3 true WO2001017965A3 (fr) | 2003-04-17 |
Family
ID=4215173
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/EP2000/008660 WO2001017965A2 (fr) | 1999-09-07 | 2000-09-05 | Cyanopiperidines |
Country Status (2)
Country | Link |
---|---|
AU (1) | AU7514700A (fr) |
WO (1) | WO2001017965A2 (fr) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8889690B2 (en) | 2007-04-27 | 2014-11-18 | Purdue Pharma L.P. | TRPV1 antagonists including dihydroxy substituent and uses thereof |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7115632B1 (en) * | 1999-05-12 | 2006-10-03 | G. D. Searle & Co. | Sulfonyl aryl or heteroaryl hydroxamic acid compounds |
EP1184442A1 (fr) * | 2000-08-30 | 2002-03-06 | Clariant International Ltd. | Composition liquide cristalline |
US6953801B2 (en) | 2001-05-22 | 2005-10-11 | Neurogen Corporation | Melanin concentrating hormone receptor ligands: substituted 1-benzyl-4-aryl piperazine analogues |
GEP20094675B (en) | 2003-07-24 | 2009-05-10 | Euro Celtique Sa | Heteroaryl- tetra-hydropiperidyl compounds useful for treating or preventing pain |
GEP20094676B (en) * | 2003-07-24 | 2009-05-10 | Euro Celtique Sa | Piperidine compounds and pharmaceutical compositions containing them |
WO2005110982A2 (fr) | 2004-04-07 | 2005-11-24 | Neurogen Corporation | Analogues substitues 1-benzyl-4-substitues piperazine |
PT2723732T (pt) | 2011-06-22 | 2017-02-17 | Purdue Pharma Lp | Antagonistas de trpv1 incluindo substituinte di-hidroxilo e suas utilizações |
WO2013164954A1 (fr) * | 2012-05-01 | 2013-11-07 | 住友化学株式会社 | Composé de pipéridine et son utilisation pour la lutte contre des organismes nuisibles |
AU2019405477A1 (en) | 2018-12-17 | 2021-06-24 | Vertex Pharmaceuticals Incorporated | Inhibitors of APOL1 and methods of using same |
TW202139996A (zh) | 2020-03-06 | 2021-11-01 | 美商維泰克斯製藥公司 | 治療apol-1依賴性局灶性節段性腎小球硬化之方法 |
BR112023003423A2 (pt) | 2020-08-26 | 2023-03-21 | Vertex Pharma | Inibidores de apol1 e métodos de uso destes |
US20230203000A1 (en) * | 2021-11-30 | 2023-06-29 | Vertex Pharmaceuticals Incorporated | Inhibitors of apol1 and methods of using same |
Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1994024124A1 (fr) * | 1993-04-08 | 1994-10-27 | Ciba-Geigy Ag | Nouvelles pyrrolidines et piperidines 2-nitromethylidene/2-cyanimino/2-nitro-imino, leurs intermediaires et leur utilisation comme pesticides |
US5780466A (en) * | 1995-01-30 | 1998-07-14 | Sanofi | Substituted heterocyclic compounds method of preparing them and pharmaceutical compositions in which they are present |
US5824690A (en) * | 1993-05-06 | 1998-10-20 | Hoechst Marion Roussel Inc. | Substituted pyrrolidin-3-yl-alkyl-piperidines |
-
2000
- 2000-09-05 WO PCT/EP2000/008660 patent/WO2001017965A2/fr active Application Filing
- 2000-09-05 AU AU75147/00A patent/AU7514700A/en not_active Abandoned
Patent Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1994024124A1 (fr) * | 1993-04-08 | 1994-10-27 | Ciba-Geigy Ag | Nouvelles pyrrolidines et piperidines 2-nitromethylidene/2-cyanimino/2-nitro-imino, leurs intermediaires et leur utilisation comme pesticides |
US5824690A (en) * | 1993-05-06 | 1998-10-20 | Hoechst Marion Roussel Inc. | Substituted pyrrolidin-3-yl-alkyl-piperidines |
US5780466A (en) * | 1995-01-30 | 1998-07-14 | Sanofi | Substituted heterocyclic compounds method of preparing them and pharmaceutical compositions in which they are present |
Non-Patent Citations (3)
Title |
---|
BUOLAMWINI, J. K. ET AL: "Synthesis and analgesic activity of 3-methyl derivatives of 4-(pyridyl) isosteres of ketobemidone", EUR. J. MED. CHEM. ( 1992 ), 27(1), 81-6, XP002158922 * |
BURKHOLDER T P ET AL: "Synthesis and structure-activity relationships for a series of substituted pyrrolidine NK1/NK2 receptor antagonists", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,GB,OXFORD, vol. 7, no. 19, 7 October 1997 (1997-10-07), pages 2531 - 2536, XP004136479, ISSN: 0960-894X * |
IORIO M A ET AL: "NITROGEN ANALOGUES OF PHENCYCLIDINE: 1-ALKYL-4-PHENYL-4-(1-PIPERIDINY L)PIPERIDINES", FARMACO, EDIZIONE SCIENTIFICA,IT,SOCIETA CHIMICA ITALIANA, PAVIA, vol. 39, no. 7, 1984, pages 599 - 611, XP000872767 * |
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8889690B2 (en) | 2007-04-27 | 2014-11-18 | Purdue Pharma L.P. | TRPV1 antagonists including dihydroxy substituent and uses thereof |
US9365563B2 (en) | 2007-04-27 | 2016-06-14 | Purdue Pharma L.P. | TRPV1 antagonists including dihydroxy substituent and uses thereof |
Also Published As
Publication number | Publication date |
---|---|
WO2001017965A2 (fr) | 2001-03-15 |
AU7514700A (en) | 2001-04-10 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
MY126559A (en) | Fungicidal 2-methoxybenzophenones | |
HUP0202573A3 (en) | Phenyl substituted hetercyclic compounds as herbicides, preparation and use thereof | |
HK1071510A1 (en) | Acetylene derivatives having mglur 5 antagonistic activity | |
AU2002304109A1 (en) | Substituted anilide derivatives, intermediates thereof, agricultural and horticultural chemicals, and their usage | |
AU1416695A (en) | 1-H-3-aryl-pyrrolidine-2,4-dione derivatives as pesticides | |
HUP0100817A3 (en) | 2-pyridylmethylamine derivatives useful as fungicides, their use, intermediates and preparation thereof | |
WO2001044215A3 (fr) | Combinaisons fongicides de substances actives | |
CA2318976A1 (fr) | Derives de 3-hydroxy-4-aryl-5-oxopyrazoline a activite herbicide | |
WO2001046165A3 (fr) | Composes organiques | |
PT1130963E (pt) | Combinacoes de substancias activas fungicidas | |
WO2001040223A3 (fr) | Composes organiques | |
AP9400655A0 (en) | New pesticides | |
WO2001055066A3 (fr) | Composes organiques | |
AU6116800A (en) | 1-aryl-3-thioalkyl pyrazoles, the synthesis thereof and the use thereof as insecticides | |
WO2001017965A3 (fr) | Cyanopiperidines | |
AU1657100A (en) | 4-trifluoromethyl-3-oxazolylpyridines, method for producing them, products containing the same, and their use as pesticides | |
AU2001297622A1 (en) | Substituted 4,5-dihydro-1,2,4-triazin-6-ones, 1,2,4-triazin-6-ones, and their use as fungicides and insecticides | |
AU1399297A (en) | Dihalopropene compounds, their use as insecticides/acaricides and intermediates for their production | |
GB0229081D0 (en) | Multifunctional cationic photoinitiators, their preparation and use | |
WO2000046210A3 (fr) | Nouveau procede de preparation d'intermediaires pesticides | |
WO2002048143A3 (fr) | Composes 2-pyridones antimicrobiens, compositions et utilisations de ces composes | |
AU2001286839A1 (en) | Compounds useful as insecticides, compounds useful as acaricides, and processes to use and make same | |
AU1651001A (en) | Difluoromethyltriazolone compounds, use of the same and intermediates for the production thereof | |
BR0207217A (pt) | Derivados de 2-heterociclil-3-4-dihidro-2h-pirrol e sua aplicação como composições praguicidas | |
WO2004057960A3 (fr) | Composes utilises en tant que pesticides |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
AK | Designated states |
Kind code of ref document: A2 Designated state(s): AE AG AL AM AT AU AZ BA BB BG BR BY BZ CA CH CN CR CU CZ DE DK DM DZ EE ES FI GB GD GE GH GM HR HU ID IL IN IS JP KE KG KP KR KZ LC LK LR LS LT LU LV MA MD MG MK MN MW MX MZ NO NZ PL PT RO RU SD SE SG SI SK SL TJ TM TR TT TZ UA UG US UZ VN YU ZA ZW |
|
AL | Designated countries for regional patents |
Kind code of ref document: A2 Designated state(s): GH GM KE LS MW MZ SD SL SZ TZ UG ZW AM AZ BY KG KZ MD RU TJ TM AT BE CH CY DE DK ES FI FR GB GR IE IT LU MC NL PT SE BF BJ CF CG CI CM GA GN GW ML MR NE SN TD TG |
|
121 | Ep: the epo has been informed by wipo that ep was designated in this application | ||
DFPE | Request for preliminary examination filed prior to expiration of 19th month from priority date (pct application filed before 20040101) | ||
REG | Reference to national code |
Ref country code: DE Ref legal event code: 8642 |
|
122 | Ep: pct application non-entry in european phase | ||
NENP | Non-entry into the national phase |
Ref country code: JP |