WO2000049001A3 - Phenoxy-, phenylthio-, phenylamino-, benzyloxy-, benzylthio- or benzylaminopyrimidine insectidices and acaricides - Google Patents

Phenoxy-, phenylthio-, phenylamino-, benzyloxy-, benzylthio- or benzylaminopyrimidine insectidices and acaricides Download PDF

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Publication number
WO2000049001A3
WO2000049001A3 PCT/US2000/003180 US0003180W WO0049001A3 WO 2000049001 A3 WO2000049001 A3 WO 2000049001A3 US 0003180 W US0003180 W US 0003180W WO 0049001 A3 WO0049001 A3 WO 0049001A3
Authority
WO
WIPO (PCT)
Prior art keywords
ocr18r19
insectidices
benzylaminopyrimidine
benzylthio
acaricides
Prior art date
Application number
PCT/US2000/003180
Other languages
French (fr)
Other versions
WO2000049001A2 (en
Inventor
Thomas Martin Stevenson
Original Assignee
Du Pont
Thomas Martin Stevenson
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Du Pont, Thomas Martin Stevenson filed Critical Du Pont
Priority to AU33577/00A priority Critical patent/AU3357700A/en
Publication of WO2000049001A2 publication Critical patent/WO2000049001A2/en
Publication of WO2000049001A3 publication Critical patent/WO2000049001A3/en

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/34—One oxygen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/38—One sulfur atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52—Two oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/56—One oxygen atom and one sulfur atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

Compounds of Formula (I), and their N-oxides and agriculturally suitable salts, are disclosed which are useful as arthropodicides wherein Q1 is O, S, NR?17, OCR18R19, or NR17CR18R19¿; wherein when Q?1 is OCR18R19 or NR17CR18R19¿, then Q1 is attached to the pyrimidine through the O or N atom respectively; Q2 is S, CR?3R4, OCR18R19, SCR18R19 or NR17CR18R19¿; wherein when Q?2 is OCR18R19, SCR18R19 or NR17CR18R19 then Q2¿ is attached to the pyrimidine through the O, S or N atom respectively; R?1 and R2¿ are each independently H, C¿1?-C4 alkyl, halogen, NR?7R8, C¿1-C4 alkoxy, C1-C4 haloalkyl, C1-C4 alkylthio or nitro; each R5 is independently H, halogen, C¿1?-C4 alkyl, C1-C4 haloalkoxy, C1-C4 haloalkyl, C1-C4 alkoxy, SF5, S(O)nR?9¿, cyano or CO¿2R?11; each R6 and each R22 is independently H, halogen, cyano, C¿1?-C4 alkyl, C1-C4 haloalkyl, C1-C4 haloalkoxy, C1-C4 alkoxy, NR?17¿ or S(O)¿nR?9; p is 0-4; and J, R?3, R4R7, R8, R9, R11, R17, R18, R19¿ and n are as defined in the disclosure. Also disclosed are compositions containing the compounds of Formula (I) and a method for controlling arthropods which involves contacting the arthropods or their environment with an effective amount of a compound of Formula (I).
PCT/US2000/003180 1999-02-16 2000-02-08 Phenoxy-, phenylthio-, phenylamino-, benzyloxy-, benzylthio- or benzylaminopyrimidine insectidices and acaricides WO2000049001A2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU33577/00A AU3357700A (en) 1999-02-16 2000-02-08 Phenoxypyrimidine insecticides and acaricides

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US12013099P 1999-02-16 1999-02-16
US60/120,130 1999-02-16
US13930299P 1999-06-15 1999-06-15
US60/139,302 1999-06-15

Publications (2)

Publication Number Publication Date
WO2000049001A2 WO2000049001A2 (en) 2000-08-24
WO2000049001A3 true WO2000049001A3 (en) 2000-12-21

Family

ID=26818082

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/US2000/003180 WO2000049001A2 (en) 1999-02-16 2000-02-08 Phenoxy-, phenylthio-, phenylamino-, benzyloxy-, benzylthio- or benzylaminopyrimidine insectidices and acaricides

Country Status (2)

Country Link
AU (1) AU3357700A (en)
WO (1) WO2000049001A2 (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2003034682A (en) * 2000-09-19 2003-02-07 Sumitomo Chem Co Ltd Pyrimidine compound and its use
EP1574502A1 (en) 2004-03-08 2005-09-14 Novartis AG Use of pyrimidine compounds in the preparation of parasiticides
KR101400632B1 (en) 2006-07-21 2014-05-27 노파르티스 아게 Pyrimidine derivatives and their use as pesticides
US7737149B2 (en) 2006-12-21 2010-06-15 Astrazeneca Ab N-[5-[2-(3,5-dimethoxyphenyl)ethyl]-2H-pyrazol-3-yl]-4-(3,5-dimethylpiperazin-1-yl)benzamide and salts thereof
NZ612075A (en) 2010-12-24 2015-04-24 Nihon Nohyaku Co Ltd Benzyloxypyrimidine derivative, agricultural/horticultural insecticide comprising derivative and method for using same
WO2012094451A1 (en) * 2011-01-06 2012-07-12 Beta Pharma Canada Inc. Novel ureas for the treatment and prevention of cancer
US20140179712A1 (en) 2012-12-21 2014-06-26 Astrazeneca Ab Pharmaceutical formulation of n-[5-[2-(3,5-dimethoxyphenyl)ethyl]-2h-pyrazol-3-yl]-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide
CN113264924B (en) * 2020-02-14 2022-11-08 山东省联合农药工业有限公司 Dioxane pyrimidine derivative and preparation method and application thereof

Citations (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1997014684A1 (en) * 1995-10-17 1997-04-24 Janssen Pharmaceutica N.V. Amino substituted pyrimidines and triazines
US5707995A (en) * 1992-07-17 1998-01-13 American Cyanamid Company Pesticidal pyrimidine compounds
WO1998012184A1 (en) * 1996-09-19 1998-03-26 Nippon Soda Co., Ltd. Pyrimidine compounds, process for the preparation thereof, and pest controlling agents
WO1998054154A1 (en) * 1997-05-28 1998-12-03 Nippon Soda Co., Ltd. Pyrimidine compounds, process for producing the same, and pesticides
EP0945442A1 (en) * 1998-03-27 1999-09-29 Janssen Pharmaceutica N.V. Trisubstituted pyrimidine derivatives
JPH11269154A (en) * 1998-03-17 1999-10-05 Nippon Soda Co Ltd Pyrimidine compound, its preparation and pest-controlling agent
WO1999050250A1 (en) * 1998-03-27 1999-10-07 Janssen Pharmaceutica N.V. Hiv inhibiting pyrimidine derivatives
EP0972770A1 (en) * 1998-07-14 2000-01-19 American Cyanamid Company Acaricidal and insecticidal substituted pyrimidines and a process for the preparation thereof

Patent Citations (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5707995A (en) * 1992-07-17 1998-01-13 American Cyanamid Company Pesticidal pyrimidine compounds
WO1997014684A1 (en) * 1995-10-17 1997-04-24 Janssen Pharmaceutica N.V. Amino substituted pyrimidines and triazines
WO1998012184A1 (en) * 1996-09-19 1998-03-26 Nippon Soda Co., Ltd. Pyrimidine compounds, process for the preparation thereof, and pest controlling agents
WO1998054154A1 (en) * 1997-05-28 1998-12-03 Nippon Soda Co., Ltd. Pyrimidine compounds, process for producing the same, and pesticides
JPH11269154A (en) * 1998-03-17 1999-10-05 Nippon Soda Co Ltd Pyrimidine compound, its preparation and pest-controlling agent
EP0945442A1 (en) * 1998-03-27 1999-09-29 Janssen Pharmaceutica N.V. Trisubstituted pyrimidine derivatives
WO1999050250A1 (en) * 1998-03-27 1999-10-07 Janssen Pharmaceutica N.V. Hiv inhibiting pyrimidine derivatives
EP0972770A1 (en) * 1998-07-14 2000-01-19 American Cyanamid Company Acaricidal and insecticidal substituted pyrimidines and a process for the preparation thereof

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Publication number Publication date
AU3357700A (en) 2000-09-04
WO2000049001A2 (en) 2000-08-24

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