WO2000030640A1 - Use of prucalopride for the manufacture of a medicament for the treatment of dyspepsia - Google Patents
Use of prucalopride for the manufacture of a medicament for the treatment of dyspepsia Download PDFInfo
- Publication number
- WO2000030640A1 WO2000030640A1 PCT/EP1999/009048 EP9909048W WO0030640A1 WO 2000030640 A1 WO2000030640 A1 WO 2000030640A1 EP 9909048 W EP9909048 W EP 9909048W WO 0030640 A1 WO0030640 A1 WO 0030640A1
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- prucalopride
- dyspeptic symptoms
- use according
- addition salt
- pharmaceutically acceptable
- Prior art date
Links
- ZPMNHBXQOOVQJL-UHFFFAOYSA-N Prucalopride Chemical compound data:image/svg+xml;base64,<?xml version='1.0' encoding='iso-8859-1'?>
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- 210000004080 Milk Anatomy 0.000 description 1
- YGSDEFSMJLZEOE-UHFFFAOYSA-N Salicylic acid Chemical compound 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- 230000009610 hypersensitivity Effects 0.000 description 1
- 230000001771 impaired Effects 0.000 description 1
- 239000004615 ingredient Substances 0.000 description 1
- 230000002401 inhibitory effect Effects 0.000 description 1
- 238000002347 injection Methods 0.000 description 1
- 239000007924 injection Substances 0.000 description 1
- 230000000968 intestinal Effects 0.000 description 1
- 235000015110 jellies Nutrition 0.000 description 1
- 239000008274 jelly Substances 0.000 description 1
- 210000002429 large intestine Anatomy 0.000 description 1
- 239000000314 lubricant Substances 0.000 description 1
- 235000012054 meals Nutrition 0.000 description 1
- 230000001404 mediated Effects 0.000 description 1
- 235000013336 milk Nutrition 0.000 description 1
- 239000008267 milk Substances 0.000 description 1
- 150000007522 mineralic acids Chemical class 0.000 description 1
- 230000002536 noncholinergic Effects 0.000 description 1
- 239000003921 oil Substances 0.000 description 1
- 239000006186 oral dosage form Substances 0.000 description 1
- 150000007524 organic acids Chemical class 0.000 description 1
- 235000005985 organic acids Nutrition 0.000 description 1
- 230000002572 peristaltic Effects 0.000 description 1
- 230000002980 postoperative Effects 0.000 description 1
- 230000003389 potentiating Effects 0.000 description 1
- 230000000644 propagated Effects 0.000 description 1
- 230000000069 prophylaxis Effects 0.000 description 1
- 230000004044 response Effects 0.000 description 1
- 230000033764 rhythmic process Effects 0.000 description 1
- 235000019698 starch Nutrition 0.000 description 1
- 239000008223 sterile water Substances 0.000 description 1
- 150000008163 sugars Chemical class 0.000 description 1
- 239000000375 suspending agent Substances 0.000 description 1
- 230000005062 synaptic transmission Effects 0.000 description 1
- 239000006188 syrup Substances 0.000 description 1
- 235000020357 syrup Nutrition 0.000 description 1
- 235000012431 wafers Nutrition 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4525—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with oxygen as a ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
Abstract
Description
Claims
Priority Applications (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP98203943 | 1998-11-23 | ||
EP98203943.0 | 1998-11-23 |
Applications Claiming Priority (6)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP99972536A EP1135130A1 (en) | 1998-11-23 | 1999-11-16 | Use of prucalopride for the manufacture of a medicament for the treatment of dyspepsia |
JP2000583523A JP2002530334A (en) | 1998-11-23 | 1999-11-16 | Use of prucalopride for the manufacture of a medicament for the treatment of indigestion |
CA002352278A CA2352278A1 (en) | 1998-11-23 | 1999-11-16 | Use of prucalopride for the manufacture of a medicament for the treatment of dyspepsia |
KR1020017004376A KR20010080025A (en) | 1998-11-23 | 1999-11-16 | Use of Prucalopride for the Manufacture of a Medicament for the Treatment of Dyspepsia |
AU13857/00A AU770580B2 (en) | 1998-11-23 | 1999-11-16 | Use of prucalopride for the manufacture of a medicament for the treatment of dyspepsia |
NZ511117A NZ511117A (en) | 1998-11-23 | 1999-11-16 | Use of prucalopride for the manufacture of a medicament for the treatment of dyspepsia |
Publications (1)
Publication Number | Publication Date |
---|---|
WO2000030640A1 true WO2000030640A1 (en) | 2000-06-02 |
Family
ID=8234369
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/EP1999/009048 WO2000030640A1 (en) | 1998-11-23 | 1999-11-16 | Use of prucalopride for the manufacture of a medicament for the treatment of dyspepsia |
Country Status (7)
Country | Link |
---|---|
EP (1) | EP1135130A1 (en) |
JP (1) | JP2002530334A (en) |
KR (1) | KR20010080025A (en) |
AU (1) | AU770580B2 (en) |
CA (1) | CA2352278A1 (en) |
NZ (1) | NZ511117A (en) |
WO (1) | WO2000030640A1 (en) |
Cited By (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2000066170A1 (en) * | 1999-04-29 | 2000-11-09 | Janssen Pharmaceutica N.V. | Prucalopride oral solution |
WO2003059906A1 (en) * | 2002-01-16 | 2003-07-24 | Janssen Pharmaceutica N.V. | Prucalopride-n-oxide |
EP1493441A1 (en) * | 2002-04-08 | 2005-01-05 | Zeria Pharmaceutical Co., Ltd. | Therapeutic agent for food competence disorder in stomach |
Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0389037A1 (en) * | 1989-03-22 | 1990-09-26 | Janssen Pharmaceutica N.V. | N-(3-hydroxy-4-piperidinyl)(dihydrobenzofuran, dihydro-2H-benzopyran or dihydrobenzodioxin)carboxamide derivatives |
EP0445862A2 (en) * | 1990-03-06 | 1991-09-11 | Janssen Pharmaceutica N.V. | N-(4-piperidinyl)(dihydrobenzofuran or dihydro-2H-benzopyran)carboxamide derivatives |
WO1996016060A1 (en) * | 1994-11-24 | 1996-05-30 | Janssen Pharmaceutica N.V. | Enterokinetic benzamide |
-
1999
- 1999-11-16 NZ NZ511117A patent/NZ511117A/en unknown
- 1999-11-16 EP EP99972536A patent/EP1135130A1/en not_active Withdrawn
- 1999-11-16 JP JP2000583523A patent/JP2002530334A/en not_active Withdrawn
- 1999-11-16 WO PCT/EP1999/009048 patent/WO2000030640A1/en not_active Application Discontinuation
- 1999-11-16 CA CA002352278A patent/CA2352278A1/en not_active Abandoned
- 1999-11-16 AU AU13857/00A patent/AU770580B2/en not_active Ceased
- 1999-11-16 KR KR1020017004376A patent/KR20010080025A/en not_active Application Discontinuation
Patent Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0389037A1 (en) * | 1989-03-22 | 1990-09-26 | Janssen Pharmaceutica N.V. | N-(3-hydroxy-4-piperidinyl)(dihydrobenzofuran, dihydro-2H-benzopyran or dihydrobenzodioxin)carboxamide derivatives |
EP0445862A2 (en) * | 1990-03-06 | 1991-09-11 | Janssen Pharmaceutica N.V. | N-(4-piperidinyl)(dihydrobenzofuran or dihydro-2H-benzopyran)carboxamide derivatives |
WO1996016060A1 (en) * | 1994-11-24 | 1996-05-30 | Janssen Pharmaceutica N.V. | Enterokinetic benzamide |
Cited By (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2000066170A1 (en) * | 1999-04-29 | 2000-11-09 | Janssen Pharmaceutica N.V. | Prucalopride oral solution |
US6413988B1 (en) | 1999-04-29 | 2002-07-02 | Janssen Pharmaceutica N.V. | Prucalopride oral solution |
JP2002543161A (en) * | 1999-04-29 | 2002-12-17 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | Prucalopride oral solution |
MY119880A (en) * | 1999-04-29 | 2005-07-29 | Janssen Pharmaceutica Nv | Prucalopride oral solution |
HRP20010764B1 (en) * | 1999-04-29 | 2011-01-31 | Janssen Pharmaceutica N.V. | Prucalopride oral solution |
JP4773619B2 (en) * | 1999-04-29 | 2011-09-14 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | Purcarapride oral solution |
WO2003059906A1 (en) * | 2002-01-16 | 2003-07-24 | Janssen Pharmaceutica N.V. | Prucalopride-n-oxide |
US8063069B2 (en) | 2002-01-16 | 2011-11-22 | Janssen Pharmaceutica N.V. | Prucalopride-N-oxide |
EP1493441A1 (en) * | 2002-04-08 | 2005-01-05 | Zeria Pharmaceutical Co., Ltd. | Therapeutic agent for food competence disorder in stomach |
EP1493441A4 (en) * | 2002-04-08 | 2007-10-17 | Zeria Pharm Co Ltd | Therapeutic agent for food competence disorder in stomach |
Also Published As
Publication number | Publication date |
---|---|
KR20010080025A (en) | 2001-08-22 |
NZ511117A (en) | 2002-11-26 |
AU1385700A (en) | 2000-06-13 |
JP2002530334A (en) | 2002-09-17 |
EP1135130A1 (en) | 2001-09-26 |
CA2352278A1 (en) | 2000-06-02 |
AU770580B2 (en) | 2004-02-26 |
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