WO1999043650A3 - Process(es) for the preparation of 6-trifluoromethyl-indoline derivatives - Google Patents
Process(es) for the preparation of 6-trifluoromethyl-indoline derivatives Download PDFInfo
- Publication number
- WO1999043650A3 WO1999043650A3 PCT/EP1999/001273 EP9901273W WO9943650A3 WO 1999043650 A3 WO1999043650 A3 WO 1999043650A3 EP 9901273 W EP9901273 W EP 9901273W WO 9943650 A3 WO9943650 A3 WO 9943650A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- trifluoromethyl
- indoline
- preparation
- benzyl
- nitro
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
Abstract
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
AU30308/99A AU3030899A (en) | 1998-02-25 | 1999-02-22 | Process(es) for the preparation of 6-trifluoromethyl-indoline derivatives |
Applications Claiming Priority (8)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB9803802.9 | 1998-02-25 | ||
GBGB9803802.9A GB9803802D0 (en) | 1998-02-25 | 1998-02-25 | Novel compounds |
GB9805195.6 | 1998-03-11 | ||
GBGB9805195.6A GB9805195D0 (en) | 1998-03-11 | 1998-03-11 | Process |
GB9805196.4 | 1998-03-11 | ||
GBGB9805196.4A GB9805196D0 (en) | 1998-03-11 | 1998-03-11 | Process |
GB9809046.7 | 1998-04-29 | ||
GBGB9809046.7A GB9809046D0 (en) | 1998-04-29 | 1998-04-29 | Process |
Publications (2)
Publication Number | Publication Date |
---|---|
WO1999043650A2 WO1999043650A2 (en) | 1999-09-02 |
WO1999043650A3 true WO1999043650A3 (en) | 1999-12-09 |
Family
ID=27451756
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/EP1999/001273 WO1999043650A2 (en) | 1998-02-25 | 1999-02-22 | Process(es) for the preparation of 6-trifluoromethyl-indoline derivatives |
Country Status (2)
Country | Link |
---|---|
AU (1) | AU3030899A (en) |
WO (1) | WO1999043650A2 (en) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE102006038113A1 (en) | 2006-08-14 | 2008-02-21 | Qiagen Gmbh | A method of synthesizing a cDNA in a sample in an enzymatic reaction and simultaneously providing a first enzyme having polyadenylation activity and a second enzyme having reverse transcriptase activity |
Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1996023783A1 (en) * | 1995-02-02 | 1996-08-08 | Smithkline Beecham Plc | Indole derivatives as 5-ht receptor antagonist |
WO1997048700A1 (en) * | 1996-06-20 | 1997-12-24 | Smithkline Beecham Plc | Indoline derivatives useful as 5-ht-2c receptor antagonists |
WO1997048699A1 (en) * | 1996-06-20 | 1997-12-24 | Smithkline Beecham Plc | Indoline derivatives useful as 5-ht-2c receptor antagonists |
-
1999
- 1999-02-22 AU AU30308/99A patent/AU3030899A/en not_active Abandoned
- 1999-02-22 WO PCT/EP1999/001273 patent/WO1999043650A2/en active Application Filing
Patent Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1996023783A1 (en) * | 1995-02-02 | 1996-08-08 | Smithkline Beecham Plc | Indole derivatives as 5-ht receptor antagonist |
WO1997048700A1 (en) * | 1996-06-20 | 1997-12-24 | Smithkline Beecham Plc | Indoline derivatives useful as 5-ht-2c receptor antagonists |
WO1997048699A1 (en) * | 1996-06-20 | 1997-12-24 | Smithkline Beecham Plc | Indoline derivatives useful as 5-ht-2c receptor antagonists |
Non-Patent Citations (1)
Title |
---|
BROMIDGE S.M. ET AL.: "Novel and selective 5-HT2C/2B receptor antagonists as potential anxiolytic agents: Synthesis, quantitative structure-activity relationships, and molecular modeling of substituted 1-(3-pyridylcarbamoyl)indolines", JOURNAL OF MEDICINAL CHEMISTRY, vol. 41, no. 10, 7 May 1998 (1998-05-07), pages 1598 - 1612, XP002110144 * |
Also Published As
Publication number | Publication date |
---|---|
AU3030899A (en) | 1999-09-15 |
WO1999043650A2 (en) | 1999-09-02 |
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