WO1997008190A3 - Compounds - Google Patents
Compounds Download PDFInfo
- Publication number
- WO1997008190A3 WO1997008190A3 PCT/EP1996/003731 EP9603731W WO9708190A3 WO 1997008190 A3 WO1997008190 A3 WO 1997008190A3 EP 9603731 W EP9603731 W EP 9603731W WO 9708190 A3 WO9708190 A3 WO 9708190A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- compounds
- combinatorial
- relates
- particular synthesis
- chemistry
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C40—COMBINATORIAL TECHNOLOGY
- C40B—COMBINATORIAL CHEMISTRY; LIBRARIES, e.g. CHEMICAL LIBRARIES
- C40B50/00—Methods of creating libraries, e.g. combinatorial synthesis
- C40B50/14—Solid phase synthesis, i.e. wherein one or more library building blocks are bound to a solid support during library creation; Particular methods of cleavage from the solid support
- C40B50/16—Solid phase synthesis, i.e. wherein one or more library building blocks are bound to a solid support during library creation; Particular methods of cleavage from the solid support involving encoding steps
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H21/00—Compounds containing two or more mononucleotide units having separate phosphate or polyphosphate groups linked by saccharide radicals of nucleoside groups, e.g. nucleic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/04—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers
- C07K1/047—Simultaneous synthesis of different peptide species; Peptide libraries
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J2219/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
- B01J2219/00274—Sequential or parallel reactions; Apparatus and devices for combinatorial chemistry or for making arrays; Chemical library technology
- B01J2219/00277—Apparatus
- B01J2219/00497—Features relating to the solid phase supports
- B01J2219/005—Beads
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J2219/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
- B01J2219/00274—Sequential or parallel reactions; Apparatus and devices for combinatorial chemistry or for making arrays; Chemical library technology
- B01J2219/00277—Apparatus
- B01J2219/0054—Means for coding or tagging the apparatus or the reagents
- B01J2219/00572—Chemical means
- B01J2219/00581—Mass
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J2219/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
- B01J2219/00274—Sequential or parallel reactions; Apparatus and devices for combinatorial chemistry or for making arrays; Chemical library technology
- B01J2219/00583—Features relative to the processes being carried out
- B01J2219/00592—Split-and-pool, mix-and-divide processes
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J2219/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
- B01J2219/00274—Sequential or parallel reactions; Apparatus and devices for combinatorial chemistry or for making arrays; Chemical library technology
- B01J2219/00583—Features relative to the processes being carried out
- B01J2219/00596—Solid-phase processes
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Biochemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Engineering & Computer Science (AREA)
- Genetics & Genomics (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Analytical Chemistry (AREA)
- Structural Engineering (AREA)
- Biophysics (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Biotechnology (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Other Investigation Or Analysis Of Materials By Electrical Means (AREA)
- Pyridine Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Priority Applications (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP96930092A EP0852583A2 (en) | 1995-08-30 | 1996-08-23 | Compounds |
JP9509838A JPH11513027A (en) | 1995-08-30 | 1996-08-23 | Compound |
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB9517661.6 | 1995-08-30 | ||
GBGB9517661.6A GB9517661D0 (en) | 1995-08-30 | 1995-08-30 | Novel compounds |
Publications (2)
Publication Number | Publication Date |
---|---|
WO1997008190A2 WO1997008190A2 (en) | 1997-03-06 |
WO1997008190A3 true WO1997008190A3 (en) | 1997-03-27 |
Family
ID=10779919
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/EP1996/003731 WO1997008190A2 (en) | 1995-08-30 | 1996-08-23 | Compounds |
Country Status (4)
Country | Link |
---|---|
EP (1) | EP0852583A2 (en) |
JP (1) | JPH11513027A (en) |
GB (1) | GB9517661D0 (en) |
WO (1) | WO1997008190A2 (en) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1997037953A1 (en) * | 1996-04-08 | 1997-10-16 | Glaxo Group Ltd. | Mass-based encoding and qualitative analysis of combinatorial libraries |
US6004823A (en) * | 1997-05-07 | 1999-12-21 | Smithkline Beecham Corporation | Compounds |
US5908960A (en) * | 1997-05-07 | 1999-06-01 | Smithkline Beecham Corporation | Compounds |
EP1728776A3 (en) * | 1998-01-05 | 2006-12-13 | Neogenesis, Inc. | Method for identifying a member of a mass-coded combinatorial library |
EP2241541A1 (en) * | 1998-01-05 | 2010-10-20 | Neogenesis, Inc. | Method for identifying a member of a mass-coded combinatorial library |
US6207861B1 (en) * | 1998-01-05 | 2001-03-27 | Neogenesis, Inc. | Method for producing and screening mass coded combinatorial libraries for drug discovery and target validation |
WO2000009527A1 (en) * | 1998-08-10 | 2000-02-24 | The Scripps Research Institute | Programmable one-pot oligosaccharide synthesis |
EP1254367A4 (en) | 2000-02-03 | 2006-07-05 | Nanoscale Combinatorial Synthe | Structure identification methods using mass measurements |
US6576472B1 (en) | 2000-07-26 | 2003-06-10 | Smithkline Beecham Corporation | Chemical constructs for solution phase chemistry |
US6584411B1 (en) | 2000-07-26 | 2003-06-24 | Smithkline Beecham Corporation | Methods to facilitate the calculation of yields of reaction products |
CA2354921A1 (en) * | 2001-05-24 | 2002-11-24 | Yasuo Konishi | Drug evolution: drug design at hot spots |
US20070048752A1 (en) | 2004-07-12 | 2007-03-01 | Applera Corporation | Mass tags for quantitative analyses |
Citations (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5288514A (en) * | 1992-09-14 | 1994-02-22 | The Regents Of The University Of California | Solid phase and combinatorial synthesis of benzodiazepine compounds on a solid support |
WO1994008051A1 (en) * | 1992-10-01 | 1994-04-14 | The Trustees Of Columbia University In The City Of New York | Complex combinatorial chemical libraries encoded with tags |
WO1995004160A1 (en) * | 1993-07-30 | 1995-02-09 | Isis Innovation Limited | Tag reagent and assay method |
WO1995019359A1 (en) * | 1994-01-12 | 1995-07-20 | Massachusetts Institute Of Technology | Process for making xanthene or cubane based compounds, and protease inhibitors |
-
1995
- 1995-08-30 GB GBGB9517661.6A patent/GB9517661D0/en active Pending
-
1996
- 1996-08-23 JP JP9509838A patent/JPH11513027A/en active Pending
- 1996-08-23 WO PCT/EP1996/003731 patent/WO1997008190A2/en not_active Application Discontinuation
- 1996-08-23 EP EP96930092A patent/EP0852583A2/en not_active Withdrawn
Patent Citations (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5288514A (en) * | 1992-09-14 | 1994-02-22 | The Regents Of The University Of California | Solid phase and combinatorial synthesis of benzodiazepine compounds on a solid support |
WO1994008051A1 (en) * | 1992-10-01 | 1994-04-14 | The Trustees Of Columbia University In The City Of New York | Complex combinatorial chemical libraries encoded with tags |
WO1995004160A1 (en) * | 1993-07-30 | 1995-02-09 | Isis Innovation Limited | Tag reagent and assay method |
WO1995019359A1 (en) * | 1994-01-12 | 1995-07-20 | Massachusetts Institute Of Technology | Process for making xanthene or cubane based compounds, and protease inhibitors |
Also Published As
Publication number | Publication date |
---|---|
WO1997008190A2 (en) | 1997-03-06 |
JPH11513027A (en) | 1999-11-09 |
GB9517661D0 (en) | 1995-11-01 |
EP0852583A2 (en) | 1998-07-15 |
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