UY34033A - ?nuevos inhibidores de quinasa?. - Google Patents
?nuevos inhibidores de quinasa?.Info
- Publication number
- UY34033A UY34033A UY34033A UY34033A UY34033A UY 34033 A UY34033 A UY 34033A UY 34033 A UY34033 A UY 34033A UY 34033 A UY34033 A UY 34033A UY 34033 A UY34033 A UY 34033A
- Authority
- UY
- Uruguay
- Prior art keywords
- new
- quinasa
- inhibitors
- quinasa inhibitors
- página
- Prior art date
Links
- 239000003112 inhibitor Substances 0.000 title 1
- 241000950314 Figura Species 0.000 abstract 1
- FWYUJENICVGSJH-UHFFFAOYSA-M sodium;2-[bis[2-[2-(2-methyl-5-nitroimidazol-1-yl)ethoxy]-2-oxoethyl]amino]acetate Chemical compound [Na+].CC1=NC=C([N+]([O-])=O)N1CCOC(=O)CN(CC([O-])=O)CC(=O)OCCN1C([N+]([O-])=O)=CN=C1C FWYUJENICVGSJH-UHFFFAOYSA-M 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/26—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
La presente invención se relaciona con nuevos compuestos de fórmula (I) capaces de inhibir una o más quinasas, especialmente SYK (tirosina quinasa esplénica), LRRK2 (quinasa con repeticiones ricas en leucina 2) y/o MYLK (quinasa de cadena ligera de miosina) o mutantes de estas. Los compuestos encuentran aplicación en el tratamiento de una variedad de enfermedades. Estas enfermedades incluyen enfermedades autoinmunes, enfermedades inflamatorias, enfermedades óseas, metabólicas, neurológicas y neurodegenerativas, cáncer, enfermedades cardiovasculares, alergias, asma, enfermedad de Alzheimer, enfermedad de Parkinson, trastornos de la piel, enfermedades del ojo, enfermedades infecciosas y enfermedades hormonales.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP11003372 | 2011-04-21 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UY34033A true UY34033A (es) | 2012-11-30 |
Family
ID=44236959
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UY34033A UY34033A (es) | 2011-04-21 | 2012-04-20 | ?nuevos inhibidores de quinasa?. |
Country Status (2)
| Country | Link |
|---|---|
| AR (1) | AR086195A1 (es) |
| UY (1) | UY34033A (es) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2017004133A1 (en) * | 2015-06-29 | 2017-01-05 | Nimbus Iris, Inc. | Irak inhibitors and uses thereof |
-
2012
- 2012-04-20 UY UY34033A patent/UY34033A/es active IP Right Grant
- 2012-04-20 AR ARP120101359 patent/AR086195A1/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| AR086195A1 (es) | 2013-11-27 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| UY34559A (es) | Inhibidores de bromodominios | |
| UY34374A (es) | Benzilindazoles sustituidos | |
| UY33925A (es) | Inhibidores tricíclicos de quinasas | |
| UY34515A (es) | Triazolopiridinas sustituidas | |
| UY34156A (es) | Compuestos inhibidores de metaloenzimas | |
| UY34034A (es) | Triazolopiridinas | |
| UY34765A (es) | Compuestos novedosos. | |
| UY34039A (es) | Compuestos fungicidas | |
| UY33978A (es) | Piridinonas bicíclicas nuevas. | |
| UY33943A (es) | Derivados espirocíclicos de isoxazolina como agentes antiparasitarios. | |
| UY34051A (es) | Derivados de pirrolotriazinona como inhibidores de pi3k | |
| UY4149Q (es) | Golosina para mascota | |
| UY34004A (es) | INHIBIDORES DE QUINASA RELACIONADOS CON PIRROLO[2,3-d]PIRIMIDINA TROPOMIOSINA | |
| UY34648A (es) | Amidas como inhibidores de pim | |
| UY34763A (es) | Inhibidores de la agregación plaquetaria | |
| UY34027A (es) | Inhibidores sustituidos de acetil-coa carboxilasa. | |
| UY34145A (es) | Compuestos inhibidores de metaloenzimas | |
| UY34146A (es) | Compuestos inhibidores de metaloenzimas | |
| UY34472A (es) | Derivados modificados de 4-fenil-piridina | |
| UY34817A (es) | Tienopirimidinas | |
| UY4153Q (es) | Batería | |
| UY34302A (es) | COMPUESTOS DE HEXAHIDROPIRANO[3,4-d][1,3]TIAZIN-2- AMINA | |
| UY34503A (es) | ?sal de bromhidrato de pridopidina? | |
| UY34550A (es) | Bencilpirazoles sustituidos | |
| UY34318A (es) | ?derivados de isotiazolina útiles como compuestos insecticidas? |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 110 | Patent granted |
Effective date: 20220308 |