UY32703A - Una nueva sal 4-metilbencenosulfonato y un proceso para preparar una composición farmacéutica que comprende la sal - Google Patents

Una nueva sal 4-metilbencenosulfonato y un proceso para preparar una composición farmacéutica que comprende la sal

Info

Publication number
UY32703A
UY32703A UY0001032703A UY32703A UY32703A UY 32703 A UY32703 A UY 32703A UY 0001032703 A UY0001032703 A UY 0001032703A UY 32703 A UY32703 A UY 32703A UY 32703 A UY32703 A UY 32703A
Authority
UY
Uruguay
Prior art keywords
salt
pharmaceutical composition
methylbenbenosulfonate
prepare
new
Prior art date
Application number
UY0001032703A
Other languages
English (en)
Inventor
Nilsson Karolina
Mete Antonio
nystrom Stefan
Trofast Eva
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of UY32703A publication Critical patent/UY32703A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/439Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/007Pulmonary tract; Aromatherapy
    • A61K9/0073Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/0075Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/145Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

La invención proporciona una sal 4-metilbencenosulfonato de un antagonista muscarínico y su uso en terapia, y un proceso para preparar una composición farmacéutica que comprende la sal y su uso en terapia.
UY0001032703A 2009-06-12 2010-06-11 Una nueva sal 4-metilbencenosulfonato y un proceso para preparar una composición farmacéutica que comprende la sal UY32703A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US18645909P 2009-06-12 2009-06-12
US24938309P 2009-10-07 2009-10-07
US28686509P 2009-12-16 2009-12-16

Publications (1)

Publication Number Publication Date
UY32703A true UY32703A (es) 2011-01-31

Family

ID=43309104

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001032703A UY32703A (es) 2009-06-12 2010-06-11 Una nueva sal 4-metilbencenosulfonato y un proceso para preparar una composición farmacéutica que comprende la sal

Country Status (4)

Country Link
AR (1) AR077081A1 (es)
TW (1) TW201100414A (es)
UY (1) UY32703A (es)
WO (1) WO2010144043A1 (es)

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0012261D0 (en) * 2000-05-19 2000-07-12 Astrazeneca Ab Novel process
CA2672446A1 (en) * 2006-12-19 2008-06-26 Astrazeneca Ab Quinuclidinol derivatives as muscarinic receptor antagonists
GB0811099D0 (en) * 2008-06-17 2008-07-23 Astrazeneca Ab New combination 376
GB0811100D0 (en) * 2008-06-17 2008-07-23 Astrazeneca Ab New combination
JP2011524897A (ja) * 2008-06-20 2011-09-08 アストラゼネカ・アクチエボラーグ β2−アドレナリン受容体活性の調節のための、4−ヒドロキシ−2−オキソ−2,3−ジヒドロ−1,3−ベンゾチアゾール−7−イル化合物を含む医薬組成物

Also Published As

Publication number Publication date
WO2010144043A1 (en) 2010-12-16
TW201100414A (en) 2011-01-01
AR077081A1 (es) 2011-07-27

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Legal Events

Date Code Title Description
DESI Application deemed to be withdrawn

Effective date: 20130124